,SMILES 0,C(=O)(C(C)(C)C(C)O)NCc1ccc(C(C)NC(Cc2cc(C)[nH]n2)=O)cc1 1,N1(C(c2cn(C3CCC3)nn2)=O)CCN(c2ncnc3[nH]ccc23)CC(O)C1.C 2,C1(NC(C2N(C(C)=O)CCCC2)=O)CN(C(C2CC2c2ccco2)=O)CC12CC2 3,C(=O)(C1=CS(=O)CCC1)N1CCC(CN(C)C(C2CC(O)(C(F)(F)F)C2)=O)C1 4,c1(C(=O)NC(CCCNC(C2(SC)CC2)=O)CO)ccc2ccn(C)c2c1 5,c1(CC(=O)NC2C(NC(c3cc(C)ns3)=O)C2)cc(Cl)sc1Cl 6,CC(C)CC(O)CC(=O)NC(Cn1ccnn1)C(N1CCC(N(C)C)CC1)=O 7,C1(C(=O)OC)CS(=O)(=O)CC1N1C2C=CC(C2)C1C(=O)OC 8,c1(CCC)ccc(C(=O)NC2CC2C(=O)NCc2ocnc2C(C)C)cc1 9,C(=O)(C1=Cc2ccccc2C1)NCC(C(C)(C)C)NC(C1N(C)CC(O)CC1)=O 10,N1(C(C2C(C#N)C2)=O)CCN(C(=O)CCc2n[nH]c3ccccc23)C2(CCC2)C1 11,N1(C(C(N2CCC(O)CC2)C)=O)CCC2(NC(=O)C=Cc3cscn3)CCCC12 12,C#Cc1ccc(C(=O)NCCN2CCC(C)(C)CC2)cc1 13,c1(C(N2C(CC)CN(C(=O)C(C)C(C)(C)C)CC2)=O)nn(C)c2ccccc12 14,C12(NC(C(CSC)(C)NC(C3CCCN3C(C)C)=O)=O)CCC(C1)OC2C 15,c1(C(N(CCSC)C)=O)cccnc1CNC(c1ccncc1N)=O 16,c1(C(=O)OCCCC)ccc(C(C)NC(=O)CC)cc1.N12CCCC(C1)C2 17,c1(NC2CC(C)n3c2ncc3)nc(N(C)CCc2cnccn2)nc2c1ncn2C 18,C1(C(=O)NCC(CNC(COC(CC)(C)C)=O)CO)CC2C(C1)C2(F)F 19,C(=O)(C(=O)N=c1cc(-c2cc(F)cc(F)c2)o[nH]1)N1CC(F)CC(OC)C1 20,N1(CCN(C(C(=O)NCCn2cc(C(=O)OC)nc2)=O)C)CCOCC1(C)C 21,Cc1cn(C)nc1C(N1CCC(C)C1CNC(=O)C(C)CN(C)C)=O 22,C1(C)(COC)CC(NC(=O)COc2cn[nH]c2)CN1C(C1(CN(C)C)CC1)=O 23,N1(C(CC=C)=O)CCN(C2CCN(C(=O)CC3CCOC(C(C)C)C3)C2)CC1 24,N1(C(C2N(C(=O)Nc3ccn(C)n3)CCC2)=O)CCC(C2(O)CC2)CC1 25,C1(CNC(CCCc2n(C)cnn2)=O)CC(C)(C)CN1C(=O)CC(F)(F)Cl 26,C1(CNC(C(=O)NC(CCC)C(=O)N(C)C)=O)CC2(C1)CC(C(F)(F)F)(OC)C2 27,C1(CNC(=O)OC(C)(C)C)(CNC(=O)CC(C)c2ccccc2)CCCCC1 28,c1(C(=O)NC2(C3N(C(COCC=C)=O)CCC3)CC2)ccc(F)c(NC(C)=O)c1 29,CS(=O)(=O)c1cc(Br)ccc1NC(=O)Nc1nccc(-c2ccccc2)n1 30,N1(C(C(C)OCCCC)=O)CC(CNC(c2ccc(CSC(F)F)o2)=O)(OC)C1 31,C1(NC(C2CCC(=C)CC2)=O)CCN(C(c2onc(Br)c2C)=O)CC(O)C1 32,C1(NC(CC=CC)=O)CCS(=O)(=O)C12CN(C(c1cc(F)cc(F)c1OC)=O)C2 33,O=C1CC(C(F)(F)F)C(C(N2CCC3(CC3)C2)=O)CN1 34,Cc1cc(N2CCC(N(C)CCN(C)C)C(O)C2)nc(NC2CCCO2)n1 35,C1(C)(C(N(c2cccc(O)c2)CC)=O)CCN(C(c2cnc(C)nc2)=O)C1 36,c1(C(=O)NC(CC=C)CNC(=O)C(CC)OC)cc2c(F)ccc(Br)c2[nH]1 37,C(=O)(C1CCOc2ccccc21)NC(CC=C)CNC(c1ccnn1CCF)=O 38,N1(C(C(C)CC2CC2)=O)CCCN(C(c2ccncc2)=O)CC1C 39,C=CC(C)(CCOC)C(=O)NCC1CC1NC(=O)CCc1cc(F)ccc1OC 40,c1(C(=O)NCCC2CCC(NC(C3CC=CCO3)=O)C2)c[nH]c(=O)cn1 41,c1(C(N(CC(C)NC(=O)CC2CC(=O)NC2=O)C)=O)cc(N)cc(O)c1 42,N1(C(C2C(C)(Br)C2)=O)CCCC(C2CN(C(=O)Cc3cccc(Cl)c3)C2)C1 43,O=C1Nc2ccc(S(=O)(=O)N(c3ccccn3)C3CCCC3)cc2C1(F)F 44,C1(OC)CC(NC(=O)CCOC2CCOCC2)CN(C(C2(C)CCC(=O)C2)=O)C1 45,CCC(C)(C)C(=O)NCCN(C(=O)COC(F)(F)F)CC1CC1 46,c1(CN(C(=O)NC(c2cnn(C)c2)c2ccccn2)CC)n[nH]c2c1CCCC2 47,c1(C(=O)NC2CN(C(C(CC#C)C3CC3)=O)CC2O)cnc2sccn12 48,C1(OCC)CC2CN(C(C3(CNC(=O)C(CO)N(C)C)CC(C)(C)C3)=O)CC12 49,C1(CCN(C)C)COCCN1C(=O)NCc1cccc(-c2ccncc2)c1 50,CCCC(C)C(C)(c1nnnn1CCC)Nc1cnn(CC2CC2)c1 51,c1(C(N2CC(CCNC(c3[nH]ccc(=N)n3)=O)OCC2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 52,c1(NC(C2CCCN2C(C2(F)CC2)=O)=O)cccc(I)c1 53,c1(CC(=O)NCC2(C(C)NC(C(CC)OCC)=O)CC2)sc2ccccc2c1C 54,N1(C(C(C(=O)OC)C)=O)CCC(NC(c2cc(-c3ccc(C)s3)[nH]n2)=O)C12CC2 55,C#Cc1cn(C)nc1C(=O)NC1CCN(C(=O)C(C)CF)C1c1ccccc1 56,C(=O)(C(CCO)N(C)C)NCC(c1ccccc1)NC(Cn1c(C)cnc1)=O 57,Cn1cc([N+](=O)[O-])cc1C(=O)NCC1CCN(C(=O)Cc2ccns2)C12CC2 58,C(C(F)(F)C(=O)NC1CCCC1NC(c1cn(C2CCOC2)nn1)=O)OC 59,CCC(CNC(=O)CC(O)Cc1ccccc1)(CC)NC(=O)CSCC(N)=O 60,c1(CNC(CN2CCC(C)C2)=O)cnn(C)c1C(=O)NCCC1CCOC1 61,C1(NC(C2CNC(=O)N2)=O)CC2(CCCN(c3ncns3)C2)C1 62,c1(C(=O)NCC=CCNC(CCOC)=O)cccc2[nH]c(=N)oc12 63,C1(CC(N2CCCC(N(C)C)C2)=O)C2CCCC2N1C(=O)C=CC1CCOC1 64,C1(C(N(C2CCCC(NC(C3(O)CC(C)(C)C3)=O)C2)C)=O)CCC(C)(F)CC1 65,C1(F)(CNC(c2cncc(OC)n2)=O)COCCN(C(c2cnsc2C)=O)C1 66,N1(C(CSCCC)=O)C(C(=O)NCC2CNC(=O)O2)CC2CC12 67,Cc1nc(NC(c2ccnc(CNC(C3CC3(F)F)=O)c2)=O)cnc1Cl 68,N1(C(Cn2c(C)cc(C)n2)=O)CCC(O)C(NC(=O)Cn2ccnn2)C1 69,N1(C(CC)C)CCN(C(c2ccc(SC3CC3)cc2)C(=O)NCC(C)C)CC1 70,C1(C2CC2)(C(N(C2CCCC(O)C2)C)=O)CN(C(C2CCN2C(C)(C)C)=O)C1 71,C(=O)(C1CCCc2c[nH]nc21)N(CC(CN(C(Cc1c(C)cc(C)s1)=O)C)O)C 72,N1(C(C2(CC=C)CCC2)=O)CCSCC1C(=O)NCC1CCN1CC 73,C(CCC(O)C(=O)N1CC(SCC)C1)NC(C(CC)OCC=C)=O 74,CC1(C)CN(c2nccnc2C#N)CC(CNC(c2ccc[nH]2)=O)O1 75,c1(CC)cncc(C(N2CC(OC)C(NC(=O)C(C)CCC)C2)=O)c1 76,c1(C(=O)NC(CC)CN(C)C(c2ncoc2-c2cnn(C)c2)=O)ncc[nH]c1=O 77,C=CCCC(CC(C)C)c1nc(-c2cncnc2)nn1C(c1ccc(Br)cc1)C 78,C(C(CC(C)C)NC(=O)Cc1cccs1)NC(c1cn(CC=C)nc1)=O 79,C1(C(=O)NC2CN(C(c3cc(CC)no3)=O)CC2C)(OC)CCCCCCC1 80,C12(NC(C3CCC(CC)CC3)=O)CN(C(=O)C(C)(C)F)CC1CS(=O)(=O)C2 81,C1(N(C(=O)CCc2cscn2)C)CN(C(=O)Cc2ccc(N(C)C)cc2)CC1O 82,c1(OCC)ccc(C(N2CCC(NC(=O)C(C)O)C(CO)C2)=O)c(F)c1F 83,N1(C(c2c(CC)onc2C)=O)CC2CCN(C(C3CN(CC)CCO3)=O)C(C2)C1 84,c1(C(N)=O)cccc(C(=O)NCC2CCCCC2NC(c2cccs2)=O)n1 85,CC(C)CCCC(=O)NCC(C)C(=O)N1CCC1C(C)O 86,C(CC(C(=O)NCc1cc(OC)ccn1)NC(c1ccc(C)cc1)=O)=CC 87,C1(CNC(Cn2ccc(C)n2)=O)CC2(CCC2)CN1C(C12CC=CC(C1)OC2)=O 88,c1(C(=O)NCC2N(C(C3CC(C(F)F)(OC)C3)=O)CC2)c(C)sc2ccccc12 89,O=C(C1=Cc2ccccc2OC1)NCC1CCCCN(C(C2CC2F)=O)C1 90,c1(C(N2CC(C3N(C(C(C)C)=O)CCC3)(O)C2)=O)ccc2oc(S)nc2c1 91,C1(NC(c2nn(C)c(C(F)F)c2)=O)CCCN(C(C2CC3(CCOC3)C2)=O)CC1 92,c1(C(=O)NC2C(O)CCN(C(CNC(CC(C)C)=O)=O)C2)ccc2c[nH]nc2c1 93,N1(Cc2cc(OC)c(C)cc2)CC2(CCC(C(=O)Nc3cc(O)ncc3C)O2)C1 94,C(CC(C)C(=O)NCCCC(C)(C)NC(=O)COCc1scnc1C)=CC 95,C#CCC(C)(CC)C(=O)N1CCCC(CNC(C2CCCSC2)=O)C1 96,c1(NC(C(CC)C)=O)ccc(NC(=O)NC2CCN2C)cc1 97,N1(C(C2C(C)=CCS2)=O)CCN(C(C2CCNC(=O)C2)=O)C(CC(F)F)C1 98,c1(CC(C(=O)NCC2CC23CC3)NC(c2cccc[n+]2[O-])=O)ccccc1Br 99,C1(C(=O)NCCC2(O)CCN(C(C=Cc3ncc(C)[nH]3)=O)C2)C2CC(F)(F)CC12 100,C(=O)(C1CCCc2n[nH]cc21)NC(CC)(C)CNC(C1CC2(CCC2)C1)=O 101,C1(C(=O)NCC2(C)CCN(C(=O)CC3(O)CCCCC3)C2)(OC)CCCCCC1 102,c1(CC(=O)NC(CCNC(C(CCCC)O)=O)(CC)CC)cc(F)c(F)cc1F 103,C1(N(C(C=CCOC)=O)CC(=O)N(C)CC2CCOC2)CC(C#N)C1 104,c1(C(N2CC(NC(c3c(-c4nc(C)sc4)c[nH]c3)=O)C(F)C2)=O)cccc(C#N)c1 105,c1(C2C(C(=O)NCC(C)(CO)Sc3ccc(C(=O)OC)o3)C2)ccc(F)c(F)c1 106,c1(C(C)Nc2cc(NC3CC(SC)C3)ncn2)c(C)cc(C)cc1C 107,C1(NC(c2c(CC)ncs2)=O)C2CCC(C2)C1C(=O)NC12CC(C1)C2 108,N1(C(c2ccc(NC(c3cc(F)nc(F)c3)=O)nc2)=O)Cc2ccccc2C1 109,C(=O)(C(C)CC(N)=O)NC1C(C)CN(C(=O)COc2cnc(Cl)cn2)C1 110,CON(CCC(=O)NCC1C2CCCC12)C(=O)C1(CO)CCCC1 111,N1(C(CC2(COC)CCCC2)=O)CC(NC(C2(Cl)CCC2)=O)CC(O)C1 112,C(C(F)(C(=O)N(C)CCN(C)CCO)C(C)C)NC(c1cn(CCC)nc1)=O 113,C(=O)(C1COc2ccc(Cl)cc21)NCCNC(C1N(C(C)=O)CCC1)=O 114,Cc1ccnc(C(=O)NC(Cc2ccccc2Br)C(N2CC(=O)NCC2C)=O)c1F 115,N1(C(C=C(C)c2cnn(C)c2)=O)CCCC2CN(C(=O)CNS(N)(=O)=O)CCC12 116,C1(C)(CNC(C(CC)OC)=O)CN(C(=O)Cc2cccc(C)c2C)CCO1 117,c1(C(N2CCCN(C(CCC3OCC(C)(C)C3)=O)CC2)=O)cc(F)c(O)c(F)c1 118,C#Cc1ccc(Br)c(C(N2CCN(C3CCN(C4CCOCC4)C3=O)CC2)=O)c1 119,N1(C(=O)NCc2cn(C3CCOCC3)nn2)CC2OCCC2(CO)C1 120,N1(Cc2c(Br)cn(C)n2)C2CCC(C2)C1C(=O)Nc1cc(C(=O)O)cc(CO)c1 121,C1(NC(N2C(c3nc(C)[nH]n3)CCCC2)=O)CCC(=O)N(C(C)C)C1 122,C1(NC(c2cn(C3CC3)nn2)=O)CCC2CC1CN2C(c1cc(F)cnc1O)=O 123,C(=O)(C(O)CC(F)(F)F)n1cc(-c2cnn(C)c2CN2CC(CO)C2(C)C)nn1 124,N1(C2CN(C(c3ccc(N4CCCCC4)cc3)=O)C2)CCN(c2ccncn2)CC1 125,c1(C(=O)NCCOCCN(C(=O)COCCOCCO)C)[nH]nc([N+](=O)[O-])c1Cl 126,c1(CCC)cc(C(=O)NC2CCCCC2NC(=O)C(C)(C)c2cnsc2)n(C)n1 127,N1(C(=O)OC(C)(C)C)CC(NC(C2CSC2)=O)C(C)(C)C1.C12(CCSC1)C(=O)N2 128,C12CCCN(C1)C2=O.c1(NC(CNC(COC)=O)=O)cccc(OC(F)(F)F)n1 129,c1(C(=O)NCCCC(CO)NC(C=C(COC)C)=O)cnc(CO)nc1C 130,C1(C(C(=O)NC2CC(CNC(C3(O)CC3)=O)C2)OC)CCCCCC1 131,c1(C(N2CC(c3ccncc3)C2)=O)c(-n2cccc2)sc2c1CCC2 132,C1(C(=O)NCC(=O)NC2CC2)CCN(C(c2ccc(OC(F)F)cc2)=O)CC1O 133,N1(C(C2(NC(C3CCC(=O)C3)=O)CC(O)C2)=O)Cc2ncsc2C1 134,C(c1cncs1)=CC(=O)NCCN(C(C1(NC(N)=O)CC1)=O)CC 135,Cn1cc(CNC(=O)NCC2(CCN)CC2)c2ccccc12 136,S(=O)(=O)(c1cccnc1N1CCCc2ccccc21)NCCCOCCN(C)C 137,Cc1ccc(C(=O)N(C(CNC(c2ncncc2Cl)=O)C2CC2)C)cc1F 138,C1(C(N2CC(CC=C)(NC(C(C)OCC#C)=O)C2)=O)COC(C)(C)CO1 139,C(c1c(Cl)nc2ccccn12)=CC(=O)NCC1(CN(C)C(C2CCCS2)=O)CC1 140,c1(C(=O)NCCC(C)(C)CNC(c2c(O)cccc2F)=O)ncnc2sccc12 141,c1(OC)ccc(COCC(=O)NC2CC(C)(NC(C3CSC3)=O)C2)cn1 142,c1(CCC)nsc(N)c1C(=O)N(CC(C)N(C(=O)CC1C=CCC1)C)C 143,C1(CNC(C2(CC#C)CCCC2)=O)COCCN(C(=O)CCn2cncn2)C1 144,C(=O)(CC(F)(F)C(C)(F)F)N(CCCCCC(=O)N1CCS(=O)(=O)CC1)C(C)=O 145,CC(C(F)C(=O)N1CCc2cnccc2C1)C(F)(F)F 146,C(=O)(C(CC(N)=O)NC(=O)C(C)c1cc[nH]n1)N(C(C(C)C)CO)C 147,Cc1nc[nH]c1CC(=O)NCCN(C(=O)CC(=O)OC(C)(C)C)C 148,C1(C)(C(N(CCNC(c2ccn(CC)c2C)=O)CC)=O)CCCN(C)C1 149,c1(CC(N2CCC(CC(=O)NCC3CCCCC3O)CC2)=O)cc(F)ccc1F 150,c1(C(N2C3(CN(C(C(CCCCC)O)=O)C3)CC2)=O)ccc2[nH]ccc(=O)c2c1 151,CC1CCN(C(=O)C(c2ccccn2)O)C1CNC(=O)CCc1cccnc1Cl 152,c1(C(C(=O)NC2CC(CN(C)C)C2)NC(C2CCCCC2)=O)cnn(C)c1 153,c1(C(=O)NC2CCC(NC(C3CCN(C)C3)=O)C2)ccc2ccccc2n1 154,Cc1conc1CC(=O)NC1CCC(CCNC(c2cc(C3CC3)on2)=O)C1 155,c1(C(=O)NCCCC(c2ccccc2)NC(C(C)=CC)=O)cnc2c(c1)COC2 156,c1(OC)cc(-n2nc(CC(C)C)nc2C(CC2CSC2)OC(C)=O)ccc1Cl 157,N(C1CCCn2nccc21)C(c1cc(Br)cn1C)c1n(CC)nnn1 158,Cc1cc(S(C)(=O)=O)cc(C(N2CC(NC(c3cnns3)=O)CC(O)C2)=O)c1C 159,c1(OC)ccc(CC(N2CCC(NC(C3CCC(C)(C)C3)=O)C(F)C2)=O)cc1O 160,C1(COC)(NC(=O)C(C)NC(=O)OC)CCCN(C(C2C=C2C)=O)C1 161,Cc1ccc(CC(=O)NC2CCC(CNC(C3(C)COCCO3)=O)C2)cc1 162,CN(C)S(C)(=O)=NS(=O)(=O)NC1CCN(C(C)(C)C(=O)N(C)C)C1 163,C1(CNC(CCNC(C)=O)=O)CC2(CCN(C(c3ccc(Cl)nc3O)=O)C2)CO1 164,c1(C(C(=O)NC(C)CCNC(C2OCCCO2)=O)C)ccc(F)c(F)c1 165,C1(C(=O)OCCC2CC2C2CC2)(CO)CCc2ccccc2O1 166,c1(N(C)CC)ccc(CNC(=O)C=CC(=O)NC2CCC(C)CC2)cc1 167,c1(C(c2nnnn2C)NCCCC(=O)NC)nccc(OCCN(C)C)n1 168,C1(C(=O)NCC2CC(SC)C2)CC12CC(NC(=O)C=C1CCCCC1)C2 169,C1(C(F)(F)F)COC2CN1C(=O)NC2.C1(OC(C)=O)COC1 170,N1(C(c2ccc(COC)s2)=O)CC2(CC(NC(c3cccn3C3CC3)=O)C2)C1 171,c1(C(N(CCCNC(c2ccc(C)s2)=O)Cc2ccccc2)=O)cnn(C)c1C 172,C1(C(N2CCN(c3n(C)cnn3)CC2)=O)CC2OC1C1CC21 173,CCCCC(O)C(C)C(=O)N1CCC(CCCNC(c2ccoc2)=O)CC1 174,c1(CCC(=O)NC2C(OC)CN(C(=O)COCC(C)(C)C)C2)c(F)cccc1Cl 175,n1(CC)nc(C(N2CCC(C)(CNC(=O)C(COC)COC)C2)=O)cc1C 176,N1(C(C2CCC(SCC)CC2)=O)CC2CC1CN2Cc1ccc(F)c(C(=O)O)c1 177,N1(C(=O)CSc2ccccn2)CCC2CC2(C(=O)NCc2cncnc2)CC1 178,C=C(F)C1(CC(=O)NCC2CN(C(c3c[nH]nc3C3CC3)=O)CC2C)CCC1 179,C12(CNC(c3nc(CC)oc3C)=O)CCCC(CN1C(=O)CSC(C)(C)C)C2 180,C12(NC(=O)CC3CCC4CC34)CCC(C(=O)NCCc3ocnc3CO)(CC1)C2 181,Cc1coc2cc(C(N3CCC(NCc4cc(F)cc(Cl)c4)C3)=O)ccc12 182,C1(NC(=O)COC2CCOC2)CC2(C1)CN(C(c1cccc(C3CC3(F)F)c1)=O)C2 183,C(C)(C)(CCNC(=O)C(C1CN(C(C)=O)C1)OC)OC 184,c1(C(CNC(=O)CCn2cnnn2)NC(=O)Cc2cncs2)ccc(F)cc1 185,C1(C(=O)NC2CC(CNC(CN=S(C)(C)=O)=O)C2)CC2C=CC1CCC2 186,C1(CCC(=O)NCc2ccc(C)s2)CCCCN(C(C2CC3CCC(C2)C3)=O)C1 187,c1(C(N2CCCC(N(C(C3(CC)CCCC3)=O)C)CC2)=O)ccc2nsnc2c1 188,CCCC(C)CC(=O)N1CC(O)CC1CNC(c1cn(CCC(C)(C)C)nn1)=O 189,C1(C(N2CC(C)OCC2)=O)CN(Cc2ccn(CCF)n2)CCC1(F)F 190,N1(C(C2C(=C)C2)=O)C(CC(=O)N(C(C)C(=O)OC)CC)C2CCCC12 191,C1(C(=O)NCC2CCCCC2)CCC(Nc2cc(N3CCCCC3)ncn2)CO1 192,C1(C(=O)NC2C(NC(c3c(C)nc(CO)nc3)=O)COC2)Cc2ccccc2O1 193,c1(C(C(NOCC)=O)SCCCCCNC(=O)C(F)(F)F)ccc(O)cc1 194,c1(Cc2cc(NCC(=O)OCC)nc(N(N(CC)CC)CC)n2)c(C)ccc(C)c1C 195,N1(C(c2cc(OC)n[nH]2)=O)CCCC(O)(CNC(c2c(C)nn(C)c2Cl)=O)C1 196,N1(C(c2cn(CC=C)nn2)=O)CCC2(CCCCN(C(=O)CC3CC3(C)C)C2)C1 197,C1(C(N(CC(C)CNC(c2nnc(O)nc2O)=O)C)=O)CC2OC(=O)OC2C1 198,N1(C(CC(CC)C)=O)CCC2(CC1)OCCC2NC(c1cccc(Cl)c1)=O 199,N1(C(C2(C=C)CCOCC2)=O)CC2CCC(C1)N2C(C1CC(C)(C)CO1)=O 200,N1(C(N(C)CCOCCN(C)C)=O)CCCC(C2OCCO2)C1 201,c1(NCC2(C)CC(F)(F)C2)nc(Br)cnc1N.n12cc(nn1)C2 202,c1(C(=O)NC2CN(C(Cc3cc(C)sc3)=O)CC23CC3)ccc2nnc(C)n2c1 203,N1(C(CCC(N)=O)=O)CCCC2CN(C(c3ccc(CCF)cc3)=O)CC12 204,Cn1cc(S(N)(=O)=O)c(C(N2CCC(C)(CNC(=O)CN3CCCCC3)C2)=O)n1 205,CC1=C(C(=O)NCC(C2CCC2)NC(=O)CCc2cccc(N(C)C)c2)CCC1 206,c1(OC)cc(C(=O)NC2CCCC(C(=O)Nc3sc(C)cc3C#N)C2)cc(C)c1 207,c1(C(=O)NC(C(C)C)(C)CNC(C2CCOC2)=O)cc2c(F)cc(F)cc2o1 208,c1(C(N(CC(N2CCCCC(O)C2)=O)C2CC2)=O)cccn2ccnc12 209,CCCC(CC(=O)NC1CCN(C)C1)NC(=O)CC1CC(OC)C1 210,n1(CC(N2CCC(C(C)NC(CC(C(=O)OC)C)=O)C2)=O)cc([N+](=O)[O-])nc1C 211,c1(C(=O)NC2CCCCN(C(c3c(CC)non3)=O)C2)nc2cc(F)ccc2s1 212,C1(C(N(C2CCN(C(=O)CC34CCC(CC3)CC4)C2)C)=O)CCCCC1(F)F 213,CC1CC(C(=O)NC(c2ccc(Br)cc2)CO)N(C(=O)CCc2ccco2)C1 214,N1(C(C2CCN(C(C)=O)C2)=O)CCC2CCC(NC(c3ccnn3C3CC3)=O)C12 215,C1(n2cc(COCC)nn2)CCOC(CC(=O)NC(CC)C(=O)NCC)C1 216,c1(C(=O)NCCC2CCCN(C(C(CCOC)C)=O)C2)nc(SC)ncc1Cl 217,C(C(C(=O)NCCn1cc(CC)cn1)NC(C1CC1C(F)(F)F)=O)OCC 218,C(=O)(CC1(NC(=O)NCCO)CC1)N(CCC)CC1CC1.OC 219,Cc1cc(CC(=O)NCCC2CN(C(=O)C(C)OCC(C)C)CC2C)ccc1F 220,CC1(C)CC(C)(C(N2CC(n3ccccc3=O)C2)=O)CN1C(C1CC(C)(O)C1)=O 221,N1(C(CC(C)O)=O)CC2(CNC(c3csc(-c4ncc[nH]4)n3)=O)CC1CO2 222,C1(CNC(=O)CCC2CC2(F)F)CCCCN1C(c1coc(C(F)F)n1)=O 223,C(=O)(C(CC(C)(C)C)NC(=O)CC(C)(F)F)N(CC(CN(C)C)O)C 224,N1(CC(=O)NCC(CN(C(CCN(CC)CC)=O)C)C)CCCC1=O 225,C(CC(C(=O)N1CCC(OCCC)CC1)NC(C1CCOC1(C)C)=O)=CC 226,c1(CC)ncoc1C(=O)NCCCCNC(C1CSCCS1)=O 227,C(=O)(C(C)(C)CCCN=[N+]=[N-])N1CCC(CCNC(C(C)C2CC2)=O)C1 228,C=CCCCC(C(=O)NCC1CC12CCOCC2)NC(c1ncc(C)s1)=O 229,c1(C(=O)NC2CC(NC(=O)CCSc3ccccc3)C2)csc2ccccc12 230,CCC(C)(F)C(=O)N1CC(NC(c2cc(-c3ccc(Cl)cc3)on2)=O)C(C)C1 231,C1(NC(C2C(C=C)OCC2)=O)CC12CCN(C(c1ncoc1CC)=O)CC2 232,C=CC(C)(C)C(=O)NC(CNC(c1ccncc1I)=O)CC 233,C(CCC(=O)N(CCN(C)C(=O)Oc1nc(C)no1)C(C)C)N(C(C)=O)C 234,CC(C)C(CC(=O)NC1(C)CCN(C(C2CC3CC3C2)=O)CC1)C(C)C 235,c1(NC(=O)NCCC2CCN(C(C)=O)CC2)ccc(I)nc1Cl 236,Cc1ccc2sc(N(CC(C)CNC(c3ccc4oc(O)nc4n3)=O)C)nc2c1 237,c1(OC)cc(CN(CC(F)(F)F)Cc2ccccc2)c(O)cc1F 238,C(C(C(=O)NC1CCC1)N(C)C(C1(S(C)(=O)=O)CC1)C)(C1CCOC1)OCC 239,c1(NC(CSCC#C)=O)cccc(NC(C2CC2C(=O)OC)=O)c1 240,c1(C(N2CC(C(=O)NC3CC3)CC(C)C2)C(=O)NC)cccn2ccnc12 241,N#CC1CN(C(=O)Nc2ccccn2)CC1NC(c1ccnc(Br)c1)=O 242,c1(CC)cnccc1C(=O)N(CC(O)CN(C)C(c1c[nH]nc1C1CCC1)=O)C 243,C(C(N=c1[nH]c(CC)nc(Cl)c1F)C1CCC1)NC(C=CCC)=O 244,Cc1nn(CC(F)(F)F)c(Cl)c1C(=O)NC1CCN(C(c2cnc[nH]2)=O)C(C)C1 245,n1(CC)ccc2cc(CN3CCC(CC(N4CCNCC4C#N)=O)C3)ccc12 246,CC(C)CCC(C)NC(C1(CNC(C2CCCOC2)=O)CC12CCC2)=O 247,N1(C(c2cn(CCC=C)nn2)=O)CCC(C)(NC(=O)CCC2OCCO2)C1 248,Cc1cc(NC(C2OCCN(C)C2=O)=O)ccc1NC(=O)CCC(C)(C)F 249,c1(CNC(C(=O)NCCOc2cncc(C3CC3)c2)=O)nc2cc(Br)ccc2o1 250,c1(C(N(C(C)C)CCNC(=O)Cn2cnc(C(F)(F)F)c2)=O)cn2ccnc2s1 251,c1(OC)cc(C(N2CCCCC2c2nc[nH]n2)=O)nc2ccccc12 252,CC1(O)CC(NC(C2CSCN2C(=O)CCC2CCCC2)=O)C1 253,N1(C(c2c(CCC)nco2)=O)CC2CCC1CN2C(=O)CSc1cnn(C)c1 254,N1(C(CC(C)(C)O)=O)CCC(C(=O)NCC2C3CC4C(C3)C24)C(C)(C)C1 255,Cc1cc(F)ccc1C(=O)NCCC(O)CNC(C12CCCC1(C(N)=O)C2)=O 256,c1(CC(=O)NCCNCC2(C)ON=C(C)C2)c[nH]c(=N)nc1O 257,c1(OC)cccc2[nH]c(C(=O)NC3CCN(C(C4C(C(F)F)C4(C)C)=O)C3)cc12 258,C1(CNC(CC=C=C)=O)CC2(CC2)CN1C(=O)C(C)C=Cc1ccccc1 259,CC(CN1CCOC1=O)CN=c1[nH]c(=N)[nH]c(=NCc2cnccc2Cl)[nH]1 260,C(=O)(C(C)(F)C(=O)N1CCN(C(=O)CCC2(C)CC2)C(c2ccncc2)C1)OC 261,Cc1ccc(Cl)c(C(=O)Nc2ccc(C(=O)Nc3ncnc(Cl)c3Br)nc2)c1 262,CC(CC(F)(F)F)C(=O)NC1CC(C)(C(=O)N(C2CCCC(C)C2C)C)C1 263,C1(NC(c2c(OCCOC)nccc2)=O)CCN(C(c2cnc[nH]2)=O)C1(C)C 264,CCC(CC)(C(=O)NC1CCC(CNC(c2cc(N)ccc2O)=O)CC1)OC 265,c1ccc(Cl)cc1.c1(NC(C)=O)ccc(OCCC(=O)OCCCl)cc1.C1C(=O)N1 266,C1(NC(c2cccc(OC)c2O)=O)C2CC3CN(C(=O)CCOC(C)C)C1C3C2 267,N1(C(CCC(C)SC)=O)CCC(C2(NC(=O)CC(C)n3ccnc3)CC2)C1 268,c1(OC)ccc(CNC(C2CCC(NCc3ccc(C)cc3C)CC2)=O)c(Cl)c1 269,N1(C(CCNC(=O)OC)=O)CC=CC1(C)C(=O)NCCc1ccc(O)cn1 270,C(CC(=O)N1CCN(C(C2CC23CC3)=O)CC1)(C(F)F)NC(=O)OC(C)(C)C 271,N1(C(=O)NC2(CCCC)CC2)CCC(N(CC(C2CCCO2)O)C)CC1 272,C(=O)(CCCCCF)NC(CCOCC)C(=O)NCC1CCN(C(=O)CC)C1 273,C1(CNC(C(c2ccco2)NC(CC=CCC)=O)=O)C(=O)NN=C1C 274,CN1CCC(C(=O)NCC2(CNC(=O)CC(=O)NC3CC3)CC2)C1=O 275,C1(C)(C(=O)NC(CC=C)CC=C)CCCN(C(C2CCN(C(C)=O)C2)=O)C1 276,c1(C(=O)NCC2C=CC(NC(C(C3CCCC3)OC)=O)C2)ccc(C(C)C)cc1 277,c1(C(N2C(CNC(CSC(C)C)=O)C=CC2)=O)cc([N+](=O)[O-])cc([N+](=O)[O-])c1 278,c1(OCCC(=O)NCCC2CCCN(C(C(C)C#N)=O)C2)ccc(F)c(F)c1 279,C=CC(CC)C(=O)NCC(c1ccccc1F)NC(=O)CN(C)C(C)=O 280,N1(C(c2cc(C)ncc2)=O)CCCC2CCN(C(=O)C=C3SCC(=O)N3C)CC12 281,c1(C(CNC(Cc2nc(CC)[nH]n2)=O)O)cc(Br)ccc1OC 282,S(=O)(=O)(c1ccc(Cl)c2ncccc12)N1C(CC)C(=O)N(CC)CC1 283,C(CN=C(NCc1cc(Br)ccc1O)NC1CCCCC1)OC(C)C 284,CCC(C(=O)NCC(C(=O)NC(C)Cc1ncn(C)n1)C(C)(C)C)C(C)(C)CC 285,N1(C(C2N(C(C)(C)C)CC2)=O)CC2CC(NC(=O)C(F)=C3CCCC3)CC(C2)C1 286,C(=O)(C1=CC2CCCCCC12)NC1(C)CCN(C(=O)CC2CC(=O)C2)C1 287,C(c1cccnc1)=C(C)C(N1CC(CF)(NC(c2cnn(CCF)c2)=O)C1)=O 288,c1(C(=O)NCC(CNC(c2c(C)onc2CO)=O)C)ccc([N+](=O)[O-])cc1F 289,CCCC(CCCNC(=O)C(C)OC1CCCC1)N=c1[nH]c(Cl)nc(C)c1F 290,c1(C(=O)NC(C2OCCN(C(CNC(=O)NC)=O)C2)C)ccc2c(c1)OCCN2 291,CCCC(C)(CCC)C(=O)NCC1CC2CC2N1C(=O)CN1CCCCC1 292,CCC(CC(=O)NCC1CCCN(C(=O)C#CC2CC2)C1)C(C)C 293,Cc1cc(C(=O)NC2CC3CC2N(C(C2(N4CCOC4=O)CC2)=O)C3)cc(F)c1 294,c1(C(N2CCC(CC=C)(NC(C3C=CCC3)=O)C2)=O)ccc(C#N)n1C 295,C12(C(=O)NCCN(C(=O)CC3CN4CCC3CC4)C)CCCCC1NC(=O)CC2 296,C1(CNC(CCC(C)SC)=O)CC2(CCC2)CN1C(c1sc(N(C)C)nc1C)=O 297,C1(C(=O)NC2(c3ccc(C)cc3)CCC2)CCCN(c2ccc(Cl)c(Cl)c2)C1=O 298,C(N=c1[nH]c2c(c(=NCc3cnn(CCO)c3)[nH]1)CCC2)c1c(C)cc(Br)cc1 299,Cc1ncsc1Cc1cn(Cc2nc(C(=O)O)co2)nn1.C1C(=O)N(C2CC2)O1 300,N1(C(c2cc(OC)no2)=O)CCC2(CC1)CC2NC(C1CCC(C)(C)OC1)=O 301,C#CC1(NC(=O)CC2CN(C(=O)CC(C)(C)C3CC3)CC2C=CC)CC2CCCC12 302,Cc1ccc(C(=O)NC2CN(C(=O)CCc3cn[nH]c3)CC2C)c(Cl)c1C 303,C#CCCC(O)C(=O)NCC1CCN1C(c1ccnc(C(C)(F)F)c1)=O 304,c1(C(c2n(CC)nnn2)NC23CC(F)(C2)C3)nc(Br)c2ccccn12 305,C1(C(N(CCOC)CCNC(=O)CCN(C)CCO)=O)CCC(O)CC1 306,c1(NC(N(C)Cc2c(C)occ2)=O)ccc(C2CC2(F)F)cc1 307,Cc1ccc(F)c(C(N2CC3CC2C3C(=O)NC2CCC(N(C)C)CC2)=O)c1F 308,CCCC(O)(CNC(c1ccc(NC(=O)CNC)cn1)=O)CCC 309,c1(C(=O)NC(C2CCCCC2)C#C)ccc(CNC(=O)C(C)c2ccco2)nc1 310,CC1(C(=O)NCCC2CCCN2C(=O)CCCN2CCOC2=O)CC2CCC1C2 311,N(S(=O)(=O)N(C)C)CC(=O)NCC(C1CC1)NC(C(C)N(c1cnccn1)C)=O 312,c1(CC(=O)NC(C2CCCCN2C(c2ncoc2C(C)C)=O)C)ccc(O)nc1 313,N1(CC#C)CCN(C(=O)CC(C)CNC(=O)C(C#N)C(C)C)CC1=O 314,S(=O)(=O)(c1ccc(NC(C23CC4CC(CC(C4)C2)C3)C)c(F)c1)NC1CC(C)C1 315,C=CCCCC(C1CC1)NC(=O)NCCc1nccn1-c1ccccc1 316,c1(C(N2CCN(C(=O)CC3CC34CC4)C(C3CCC3)C2)=O)cncc2c[nH]nc12 317,C1(C)(NC(C(C)SC(C)C)=O)CCCN(C(=O)Cc2coc(C(F)F)n2)C1 318,CC1(CNC(=O)CC2CCOCC2)CC(F)(F)CN1C(c1cnsn1)=O 319,c1(C(N2CCCCC(NC(C(CC=C)(F)F)=O)C2)=O)cccc2c1NCC2 320,C(=O)(C(=O)C(C)(C)C)N1CCC(NC(C2OCC(C)(C)C2)c2ccccn2)CC1 321,N1(C(C2C(C)(C)COCC2)=O)CCc2[nH]nc(CNC(C3CCCCS3)=O)c2C1 322,c1(OC)ccc(F)c(C(N2CC3CC2C3CNC(c2cscn2)=O)=O)n1 323,O=C(C#CC1CCCCC1)NC(CC(=O)NC(CCO)C(F)F)C1CC1 324,c1(C(N(CC(C)N(C)C(c2ccn(C3CCC3)n2)=O)C)=O)cc2cccnc2s1 325,N1(CC(N2C(C)CCCC2C)=O)CC2CC(NC(C3(C)CS(=O)(=O)C3)=O)CC1C2 326,Cc1nccc(C(=O)NC(CCF)C(=O)N(CC(F)(F)CO)C)n1 327,C1(CC)CC(C(N2CCCC2C2CCN(c3ccc(C(C)C)cn3)C2)=O)CCO1 328,C1(C(C)NC(C2(O)CCOCC2)=O)CN(C(C2CC(F)(F)C2)=O)CCO1 329,N1(C(C2N(C(c3c(C)nc(CC)o3)=O)CC2)=O)CCCC(C)C1CO 330,N1(C(c2cc(OC)n[nH]2)=O)CC2CC1(C(=O)NOC(C)(C)CO)C2 331,c1(C(N2CCC(C(C)NC(C(C(C)C)SC)=O)C2)=O)c(C)nn(CCO)c1C 332,c1(Cn2c(C(C)(CCSC)NCC(COC)(C)C)nnn2)nn(C)c(Cl)c1Br 333,FCCN=c1[nH]c(NC2CC2c2ccccc2Cl)nc2c1CCC2 334,c1(C(=O)NCC=CCNC(CCn2ccc(C)n2)=O)cc2c(s1)CCCNC2=O 335,N1(C(C=CCC)=O)CC2CCC1CN2C(=O)CSc1ccccc1C 336,c1(N(C)C)ccc(C=CC(N2CCC(NC(=O)C(F)C3CC3)C(O)C2)=O)cc1 337,CC(C(=O)OC(C)(C)C)C(=O)NC1CN(C(c2ccc[n+]([O-])c2)=O)CC1C 338,c1(NC(c2cc(Cl)no2)C)[nH]c(=NCC2CCN(C)C(=O)C2)nc2c1cnn2C 339,C=C(C)CCC(=O)N1CCC(CNC(=O)C(C)OCC(F)(F)F)C1 340,CC1(C)CC(C(=O)NCC=CCNC(c2cc[nH]c(=N)c2)=O)CC(C)(C)O1 341,c1(CNC(=O)COC(F)F)cnn2c1CN(C(C1Cc3ccccc3O1)=O)CC2 342,c1(SC)ccc([N+](=O)[O-])c(C(N2CC3CC(NC(=O)C(C)(C)C)CC3C2)=O)c1 343,c1(C(=O)NCC2C(C(=O)NC(CCCCC)C)C2)cc2cccnc2[nH]1 344,c1(C(N(CC(C)NC(C(CC=C)c2ccccc2)=O)C)=O)csc([N+](=O)[O-])c1 345,c1(C(c2n(CC(=C)C)nnn2)NC2C(C)C2C)cn(C)nc1-c1ccccc1 346,N1(C(c2cc(CC)on2)=O)CCN(C(=O)C(=O)NC2CC2)C(C(C)C)C1 347,N1(C(c2nnc(C(C)(C)C)s2)=O)CCCC(C2CC2NC(C2CCCSS2)=O)C1 348,C1(CN(C(COC2CCC(C)CC2)=O)C)CCCN(C(=O)CCNC(N)=O)CC1 349,c1(C(N2C3CC(NC(C(C=C)O)=O)CC2CC3)=O)csc2ccc(Br)cc12 350,Cc1ccc(C(=O)NC(CNC(c2ccc(C#N)s2)=O)CO)c(=O)n1C 351,C#Cc1ccccc1CNC(=O)C(C)(C)NC(c1ccn(C(F)F)n1)=O 352,N1(C(C(C)N(C(C)=O)C)=O)CCC2(C1)CN(C(=O)Cc1ccccc1C)CCO2 353,C12(CC(=O)NC(CCNC(c3cnc(C)n3C)=O)C)CC3CC(CC(C3)C1)C2 354,C1(CNC(CSCC(C)C)=O)CCCN1C(=O)Cc1cc(C2CC2)n[nH]1 355,N1(C(CC(CCC)O)=O)CCc2nc(CNC(C34CC(O)C3C4)=O)sc2C1 356,C1(C(=O)NCC2(C)CN(C(=O)CC3CCOCC3)C2)CCS(=O)(=O)C1 357,C(=O)(CCCC1CC1)NC(c1ccccc1)C(=O)N(CC(C)(C)OC)C 358,CCCC(C(=O)OCC(=O)Nc1ccc(-n2cncn2)cc1)S(N)(=O)=O 359,CCCC(C(=O)OC)C(=O)NC12CC(CNC(=O)Cc3coc(C)n3)(C1)C2 360,CC1(C(N2CC(C#N)C2)=O)CN(C(=O)CNC(=O)C(C)(C)C)C1 361,CC1(C(F)F)CN(C(c2cc(C(=O)O)nn2C2CCCC2)=O)CCO1 362,c1(OC)ccc(F)cc1CC(=O)N(CCCN(C(=O)C1=CCCC1)C)C 363,c1(OC)cncc(C(=O)N(C)CC2CCCN2C(c2ccnn2C(C)C)=O)c1C 364,C(=O)(C1=C(Cl)CCOC1)NCc1cn(CC(=O)NC(c2ccccc2)C)nn1 365,C(=O)(CC(C)CC(=O)OC)N1CC2C(CC(=O)NC3(CC=C)CCC3)C2C1 366,C(CN=c1[nH]c(=NCc2cnc[nH]2)[nH]c2cccc(F)c12)c1cnc(C)[nH]1 367,c1(C(N2CCC(NC(c3cn(C4CC4)cn3)=O)C(O)C2)=O)c[nH]c2cnccc12 368,C1(O)(Cc2nc(CC(=O)O)on2)CCN(C(C2CCCS(=O)(=O)C2)=O)CC1 369,C1(C(=O)NCC=C(C)C)C2CC(O)C(C2)N1C(C1CS(=O)(=O)C1)=O 370,CCCCCCCCCC(C)CCC(=O)N(C)CC.C(C(C)C)N(CCN)CC 371,C(=O)(C(CN(C)C)C(C)C)N1C(CNC(CC2(OC)CCC2)=O)CC1 372,N1(CC(N2CCCN(C(C3CC(=O)N(O)C3)=O)CC2)=O)CCCC(C2CC2)C1=O 373,N1(C(C(C2CCCC2)NC(C)=O)=O)CCC(C)C(CNC(=O)C=CC(N)=O)C1 374,O=C1NCC2CCCN(C(c3cncnc3)C(=O)NCCCF)C12 375,N1(C(C(CC(C)C)N(C)C(c2cccc(O)c2F)=O)=O)CCN2C(=O)OCC2C1 376,c1(NCC)cccc(C(=O)NCC2CC2NC(C2CCNC2=O)=O)c1 377,C(=O)(C1=NOC(C)C1)N(c1scc(CC(N2CCCC2)=O)n1)CC.NC=O 378,Cc1onc(Br)c1C(c1nnnn1CCN1CCOCC1)Nc1cn(C)cn1 379,c1(OC)cccc2c(C(N3CCN(C(=O)C(Cl)=CCl)CC3C(C)C)=O)cccc12 380,C(=O)(CCCCCF)NCc1c(C(N(C(C)C(C)(C)O)C)=O)nco1 381,C1(Nc2c[nH]nc2Cc2ccccc2)CCN(C(C2CC(OC)C2)=O)CC1C 382,N1(c2nnc(C(N)=O)s2)CCOCC(CNC(=O)C(C2CC2)C2CC2)C1 383,C(=O)(C1Cc2cccc(Br)c21)OC1CCC(C(=O)OC)C1 384,c1(C(N2CCN(C(C3CCCS3)=O)C3C2CCC3)=O)cc(=O)c2ccccc2o1 385,N1(C(c2c(C)nc(C3CC3)s2)=O)CCN(C(=O)CC2(O)CCC2)CC1C(C)C 386,C1(NC(C2N(C(C)=O)CCC2)=O)CCC(O)CN(C(c2ccc(C(N)=O)o2)=O)C1 387,N1(C(C(C)OCCCC)=O)CC(NC(=O)C(C)N(C)C)C2(CC2)C1 388,c1(C(=O)NC2CC(NC(C(C(C)C)c3cnc(C)s3)=O)C2)ccc(F)cc1C#N 389,c1(OCC(=O)NC2CC(C)(NC(Cn3ccc(C)n3)=O)C2)ccc(F)cc1Cl 390,n1(CC)cnc2c(NCCS(=O)(=O)CC)nc(N3CCC(CC#N)C(C)C3)nc12 391,C1(CC)CN(C(=NCc2cnccc2N(C)C)NCC(C)(C)C)CC(C)S1(=O)=O 392,CC(CN(C)C(C1(N(C)C)CCC1)=O)C(=O)NCCc1cscn1 393,N1(C(C)=O)CCC2(CCC(CNC(=O)CN3OC(C)(C)CC3=O)CC2)CC1 394,C1(C)(CNC(CCC2C(C)C2)=O)CC(NC(=O)C2CC2)C1 395,CCC(CC(=O)NCC1CC(NC(=O)CCOCC2CCC2)CCO1)C1CC1 396,n1(CC(=O)OCc2scc(C(=O)OCC)n2)c(S)nc2ccccc2c1=O 397,CC(CNC(=O)OC(C)(C)C)CC(=O)N1CCC1CNC(C1(CO)CC1)=O 398,C1(F)(CNC(c2noc(CC)c2C)=O)CCCN(C(C2CC2c2nc[nH]n2)=O)CC1 399,C=C(Cl)CC(C(=O)NC(c1cc[nH]n1)C)NC(c1cnc(O)cc1C)=O 400,c1(C(C(=O)NC2C(CNC(C3(C=C)CCC3)=O)CC2)O)cc(F)c(F)c(F)c1 401,C1(CC(=O)N(C2CCC(CC)CC2)C)CC(C)(C)CN1C(C1CCC(C)CC1)=O 402,CC(CCN(CCCN1CCNCC1)C)CC(C)(C)C 403,N1(C(c2ccc(C)cc2C)=O)CCC2CCN(C(C3C4COCC34)=O)C2C1 404,c1(CSc2c(C)nn(-c3cccc(Br)c3)c2Cl)cn(-c2ccccc2)c(=O)nc1O 405,C(=O)(C1CCCc2ncnn21)NCC1CCCN(C(CC2=CCN(C)CC2)=O)C1 406,n1(-c2ccn(CC)n2)nc(CCCc2ccccc2)nc1CCc1ccccn1 407,N1(C(c2c(N)ccc(F)c2)=O)CCN(C(c2cc(O)ncn2)=O)C2CCCCC12 408,C(=O)(C(C)(F)C(=O)OC)N1CCC(N(C(=O)CCc2cn[nH]c2)CC)C1 409,CCCCC(O)C(C)C(=O)NCC1(O)CCN(C(=O)C=Cc2ccncn2)CC1 410,CN1N=C(CC(=O)N2CCC(F)(F)C(CNC(C3(O)CCSCC3)=O)C2)CC1=O 411,c1(C(=O)NCCCN(C(CCC=C)=O)C2CC2)cccc2c1OC(C)(C)C2 412,C1(OC)CC(NC(=O)NC2C3CC4C(C3)C24)C(OC)C1 413,CCCCC(C(=O)NCCc1cccc(O)n1)NC(=O)CCC1CC1(F)F 414,N1(C(C2(CC#C)CN(C(=O)OC(C)(C)C)CCO2)=O)CCC(F)(F)CC(C)C1 415,c1(CCC)c(C(=O)NC2(CF)CCN(C(c3ccc(C)s3)=O)C2)nnn1C 416,CCCC(C(=O)NCC1CCCCN1CCOc1cccc(Cl)c1)OC 417,CC(C(=O)OC(C)(C)C)C(=O)N1CCC(CCNC(c2ccnn2C2CC2)=O)C1 418,Cn1cnc(CC(=O)NCC2C=CCN2C(=O)CCc2nnc(C(F)F)o2)c1 419,C1(C(=O)N)CC=CCC1C.c12cc(on1)CNC(=O)N(CC)C2.C(C)(C)(C)OC(C)=O 420,N(C1CCc2ccccc21)C(C(CNC(c1ncnc(C)c1C)=O)O)=O 421,C12(C(N3CCC(CNC(CC(C)N(C)C)=O)C3)=O)CCC(CC1)OC2 422,C(=O)(C1CCc2cccc(Cl)c21)N1C2CC(NC(C3(CC)COC3)=O)CC1CC2 423,C1(C(=O)NCCOC2CN(C(c3ccc(=N)[nH]c3)=O)C2)CC2(CCOCC2)CO1 424,CC1(C)CCCCC1=CC(N1CCC(F)(CNC(C2CC2C(C)(C)C)=O)C1)=O 425,c1(OC)cc(OCC(=O)NC2CC3CCC2CC3)ccc1[N+](=O)[O-] 426,S(=O)(=O)(c1cccnc1)NCC(=O)NC1CCCCN(C(=O)C2=COCC2)C1 427,c1(Sc2n(C)nnn2)cc(F)cc(F)c1Oc1cccc(F)c1 428,N1(C(CS(CC)=O)=O)CC2CCCC2(NC(C23CC(COC)(CO2)C3)=O)C1 429,C1(NC(c2c(C)cno2)=O)C=CCN(C(=O)Cn2cccc2)C1 430,O=C1NC(C(=O)NCC2CCN2C(=O)Cn2cnccc2=O)CCO1 431,C(Cn1cccn1)(C(=O)NOC1CC1)NC(C1CCCC(=O)C1)=O 432,c1(CCC(=O)N(CC(C)NC(=O)CC(C)n2cccc2)C)ccc(Cl)c(Cl)c1 433,c1(C(N2CCCC(NC(c3c(C)[nH]cc3)=O)C2)=O)cn(C)c(=O)cn1 434,C1(C(N2C(CCNC(C3N(C)CC(F)C3)=O)CCCC2)=O)CC(C)(C)OC1=O 435,C(N=C(NC1CCCC1)N1CC(O)C2(CC2)C1)C1C(C)(C)C2CCC1C2 436,N1(C(CCOCCC)=O)CCCC2CCN(C(c3cccn4cncc34)=O)CC12 437,N1(C(c2c(CCC)nco2)=O)CCC2(CC1)CC2C(=O)NC1(C)CCCC1(C)C 438,c1(C(N(CCNC(C(C)Cc2cnn(C)c2)=O)C)=O)cc2n(c1)CCOC2 439,C1(C(=O)NCCn2ncnn2)CN(C(=O)COCCOCF)CC(F)(F)C1 440,C1(NC(C(C)SCC)=O)CCCCC1CNC(c1ccn(C)c1CC)=O 441,N1(C(CCCC2(C)N=N2)=O)CC(NC(c2cc(C3CC3)on2)=O)C2CCCCC12 442,c1(OC)ccc2nc(CNC3CCCC(SC)C3)ccc2c1Br 443,c1(C(=O)NC2COCCN(C(C(CC)F)=O)C2)cccc2c[nH]nc12 444,c1(NC(c2nnnn2CCC)CCC)cc([N+](=O)[O-])ccc1C 445,CCCC(C(=O)N1CCCCC12CC(NC(=O)C(C)(CC)CC)C2)S(N)(=O)=O 446,C1(n2cc(-c3c(Cc4ccccc4)nc(C)cc3)nn2)CCOC2(CCSC2)C1 447,c1(CC)cccc2sc(NC(c3sc(COC)nc3C)=O)nc12 448,c1(NC(C23C(CN(C(C(C)OC4CC4)=O)C2)CC3)=O)ccc2c(c1)OCO2 449,c1(C(=O)NC2C(CNC(c3cc[nH]n3)=O)COC2)coc2ccc(Cl)cc12 450,CC(C)C(CO)C(=O)NC1CCCCC1CNC(c1cnc(C(=O)OC)cn1)=O 451,C(=O)(C(CO)C(C)(C)C)N1C(CN(C(Cc2nc(C(C)OC)sc2)=O)C)CCC1 452,CCC(CO)C(=O)N1CC(CN(C)C(c2c(OC)noc2C)=O)C1 453,C12(C(N(CC(N3CCCC(CO)C3)=O)CC)=O)CCC(CC1=O)C2 454,CCCC(C)(O)CC(=O)N(C)CCOCCN(c1nnccc1C#N)C 455,c1(C(=O)NCC2CCCC(NC(CCC(=C)C)=O)C2)ccc2c(=O)cc[nH]c2c1 456,C1(N(C(CCN(C(c2csc(C)c2C)=O)C)=O)C)CCCCCC1O 457,C(N1CCOC2(C1)CN(N1CC3CCCCCC3C1)C2)C1CC(=O)NC1=O 458,N1(C(C(C2CCOCC2)C)=O)CC(N(C)C(c2c[nH]nc2Br)=O)C(C)(C)C1 459,CC(C)C(C)C(CNC(=O)CC1(CS(C)(=O)=O)CC1)NC(C1CC(O)C1)=O 460,Cc1ccc([N+](=O)[O-])c(NNC(=O)NCC23CCCC(C2)C(=O)N3)n1 461,C1(C(=O)NC2CCN(C(c3nc(C(N)=O)sc3)=O)C2)CC2(CCC2)CCO1 462,c1(C(C(=O)OC(C(C(F)F)c2ccco2)=O)NC(=O)OC(C)(C)C)cccnc1 463,N1(C(CC(=O)OC)=O)CC(C2CN(C(c3cccc(-c4nnc(C)o4)c3)=O)C2)C1 464,c1(OCC(=O)NC2(Nc3ccc(-n4cncn4)cc3)COC2)cccc(F)c1 465,c1(C(=O)NCCC(C)CCNC(=O)C(F)CC2CC2)cccc2ccnn12 466,C(N=c1[nH]c(=NC2CC=CCC2C(F)(F)F)[nH]c2c1COC2)C1(N(C)C)CCC1 467,Cc1c(C(N2CCOC(CN(C)C)C2)=O)cnn1CCC(C)C 468,N1(C(C(CC)=CCCC)=O)CC(C)CN(C(c2ccc(C(F)F)cc2)=O)CC1C 469,C1(C(=O)NC(c2ccccc2F)C)CC(F)CN1C(=O)C(c1ccccc1)O 470,N1(C(CCCn2ncc(C)c2)=O)CCC(n2cc(CNC=O)nn2)CC1 471,N1(S(CC=C)(=O)=O)CCc2nc(C)sc2C1.N12CC(C)CC1C2=O 472,C=C(Cl)CCC(=O)NCC(C)(CNC(c1csc(C(C)=O)n1)=O)OC 473,c1(OC(CCCCN=[N+]=[N-])=O)cccc2ccccc12.C12(CC1)C(=O)NC2 474,C1(CC=C)(NC(CCN(C(=O)C(O)CN(C)C)CC#C)=O)CCCC1 475,c1(C(=O)NCCC2N(C(C3C(C)C3(F)F)=O)CCSC2)c2c(nn1C)CCCC2 476,C=CC1CN(C(c2ccc(F)c(C)c2)=O)CC1NC(C1CCCS1)=O 477,N1(C(C(C)CC(F)F)=O)CCC(CNC(c2ccc3n[nH]cc3n2)=O)C(F)(F)C1 478,c1(C(=O)NCC(C2CC2)NC(c2cnc(CC)s2)=O)c(F)cncc1Cl 479,c1(C(=O)OC)cc(F)c(OC(C2CC(=O)N(C(C)C)C2)=O)c(F)c1N 480,C1(NC(c2c(C)oc(-c3cnn(C)c3)n2)=O)CCCCN(C(=O)C2=CCCC2)C1 481,c1(OC)ccc(C2(CNc3cnc(I)cn3)CCC2)cn1 482,C1(C(=O)NC2C(C(C)(C)C)C2)CCN(C(C2CC3(CC(=O)C3)C2)=O)C1(C)C 483,C1(CNC(c2c(SCC)cncc2)=O)COCCN(C(C2(C)CCCN2C)=O)C1 484,C1(CNC(C(C)N2CCC2)=O)CC2CCC1N(C(=O)CC(C)c1cccnc1)C2 485,c1(OC)ccc(Cl)cc1C(=O)NCC1CN(C(=O)CCC2CC2)CC12CC2 486,Cc1c(NCC2COC(C)(C)C2)ncnc1NCc1ccc(C2CCC2)cc1 487,C(C)(CCCC(C)C)NC(C(CC=CC)NC(c1c[nH]c(C)c1)=O)=O 488,Cn1ccc2cccc(C(N3CC(F)CC3C(=O)Nc3cccc(N)c3)=O)c12 489,C(=O)(CCCCC(=O)NC1CC(CC(=O)NC2CC(F)C2)C1)OC 490,C(=O)(C(O)C(C)CC)NC(CC=C)CNC(c1ccc(C(N)=O)cc1)=O 491,c1(N2CCCC(NC(COCc3onc(CC)n3)=O)C2)nc2ncc(Cl)cc2s1 492,C1(CC(=O)NC2CCC(CNC(c3ccc(O)cc3)=O)CC2)CCS(=O)(=O)C1 493,C(=O)(C1CCc2ccccc21)NCC1N(C(CCCC#C)=O)CCCCC1 494,C1(NC(C=CCC)=O)CC2CCC1CN2C(=O)Cn1cc(C2CC2)cn1 495,C#Cc1cc(NC(=O)CN(C(=O)C(C(C)CC)N(C)C)CC(C)(C)C)cc(F)c1 496,N1(C(C2C=CC(NC(C#CC(C)(C)O)=O)C2)=O)CCOC2(CCCC2)C1 497,N#CC1CCCCN1C(C1CN(C(c2cccc(C(F)(F)F)c2)=O)C1)=O 498,C(c1cnn(C)c1C)=CC(=O)NCC(CC(C)C)NC(c1nccc(CC)c1)=O 499,C1(C(=O)NCC(CN(C(C(CC)O)=O)C)(C)C)CCN(c2ccc(Cl)nn2)CC1 500,c1(C(=O)NC2C(NC(Cc3c(CC)con3)=O)CC2)cn(C2CC2)c(C)cc1=O 501,N1(C(C(CC)C)=O)CCC(C(C)NC(C2CC23CCOC3)=O)CC1 502,c1(C(N2CC(NC(=O)CC3(CO)CC3)C(O)CC2)=O)cncc2c[nH]nc12 503,C(=O)(CCCC(N)=O)NCCC1C(C)CN(C(c2c[nH]nc2Br)=O)C1 504,CC(O)(CC(=O)N1CC=CC(NC(=O)CCCCc2cnc[nH]2)C1)C(F)(F)F 505,N1(C(C(N2CCOCC2)C)=O)CCC2(CCC(NC(c3cnc(O)o3)=O)C2)C1 506,CC(CNC(c1ccnnc1)=O)CC(=O)N(C1CCCC1)C 507,n1(CC)cc(Br)c(C2CCCN2C(=O)CNc2cnn(C)c2)n1 508,C1(c2ccc(Cl)cc2)(C(=O)NCCN(C(COC)=O)CC(C)O)CCN(C)C1 509,N1(C(CSCCC)=O)CCCCC(C2CN(C(=O)Cc3ccccc3C)C2)C1 510,c1(C(=O)NC(COC)CNC(C2CCC3CC23)=O)ccc(C2CC2)c(F)c1 511,Cn1ncc2c1CCC(C(N1C3CCCC1CN(C(=O)CC(F)(F)F)C3)=O)C2 512,c1(C(N2C(CNC(C3(F)C(C)C3)=O)CC2)=O)cc2cc(Cl)ccc2o1 513,C1(C(C#N)NC(C(C(C)C)c2cccnc2)=O)CCC(F)(F)CC1 514,CC1=CCC(C(=O)NC(C)CC(=O)NCC(C)(C)OCC2CC2)CC1 515,CC(C)(C(=O)NCC1CC1NC(=O)CCN1CCCC1=O)N1CCCCC1 516,CCN=c1[nH]cc(C(=O)NC(C)(CNC(C2CCCN2CC)=O)CO)s1 517,C(=O)(C(CC)C(=O)NC(c1cccnc1)C(=O)NCCOC1CCCC1)OCC 518,c1(C(=O)NCCCN(CCCNC(C(CC)N(C)C)=O)C)cnc2[nH]cnc2c1 519,c1(OC)ccc(CCC(=O)NCCNC(=O)CC2COCCOC2)cc1N 520,N1(C(C(C)C(C)(C)C)=O)CCCN(C(c2cncc(C3CC3)c2)=O)CC1C 521,CC1CCC(O)(C(=O)NCCOCCNC(=O)CCc2cccc(F)c2F)CC1 522,c1(C(=O)NCC2(CCNC(c3n(C)ncc3)=O)CC2)cc(N2CCCC2)ccn1 523,N1(C(=O)OC(C)(C)C)CC2CC1C2C(=O)OCc1nn(Cc2ccccc2)cc1I 524,C1(NC(C2CCCN(CC)C2)=O)CCN(C(C2CCCC2O)=O)C12CCC2 525,N1(C(c2c(=N)cc[nH]c2)=O)CCC2(CCCN(C(C34CCC(CC3)C4)=O)C2)CC1 526,c1(C(=O)NCCC2CCC(NC(C=CC(=O)OCC)=O)C2)n[nH]c2c1COCC2 527,c1(C(N2CC(C)C(NC(c3cc(F)c(F)cc3F)=O)C2)=O)c(F)cc(F)cc1F 528,n1(CC)ncc2c(NC(=O)CC3(O)CN(C(=O)NCC4CCCC4)C3)ncnc12 529,CC1CC2(CCC(CNC(=O)Nc3ccnn3C)O2)CO1 530,CC(C)C(C(C)NC(C1(N(C)C)CC1)=O)NC(c1ccsc1Cl)=O 531,CCC(C(C)(C)O)NC(=O)CC1CCCC(NC(=O)CC(C)=C(C)C)C1 532,C1(OC)CC(C)CN(C(C2C(O)CCN2C(=O)C(C)=NOCC#N)=O)C1 533,c1(C(N2CCSCCC2)=O)c2c(nc3ccc(Cl)cc13)CCC2 534,C=CC1(C(=O)NCCC2CCCN(C(C3(C)CCCNC3=O)=O)C2)CCCCC1 535,c1(CNC(=O)NCC2C(F)(F)C23CC3)[nH]nc2ncccc12 536,c1(C(=O)NC)ccc(C=CC(=O)N(C)CCN(C(=O)CCS(C)=O)C)cc1 537,C#CCCCCCCCNC(=O)C(CC1CCOCC1)NC(c1cnns1)=O 538,CC1c2c[nH]nc2CCC1C(=O)NC1C=CCN(C(c2csc(Cl)n2)=O)C1 539,c1(C(=O)NCCCN(C(C(C=CC)O)=O)CC)ccc2nc3n(c2c1)CCC3 540,C1(CNC(C2(C(=O)NC)CC2)=O)CC2(CO1)CN(C(=O)C(C)CC1CC1)C2 541,C1(OCC(=O)N(CCN(C(C(C)NC(=O)OC)=O)C)C)CCC(F)(F)CC1 542,C1(NC(=O)NCC(C)Oc2cccnc2)CCCCCC1CO 543,C1(CNC(C2C(C(C)NC(C(CSC)OC)=O)C2)=O)OCCCC1(C)C 544,Cc1cc(C#N)ccc1C(=O)NC(C)(C(=O)NCCOCC(C)(C)O)C1CCC1 545,C(=O)(C(CNC(c1cccc(O)c1F)=O)CC(C)C)NCC1C(OC)CCC1 546,c1(C(N(CCN(C(C2(C)CCC(C)C2)=O)CC)CC)=O)cc(F)ccc1O 547,C(=O)(C1=CCN(C)C1)N(CC(CNC(CCOCC)=O)(C)C)C 548,c1(NC(=O)CCC2CCCOC2)ccc(OC2COCC2CC2CCCC2)nc1 549,CCC(CC)CC(=O)N1CCC(C)C1CNC(C1(NC(C)=O)CCC1)=O 550,C(=O)(CCC(C)C)NCC(CN(C(=O)CN(C)C(C)=O)CC)(C)C 551,c1(NC(C2CCC(CC)O2)=O)c(C(C)(C)C)cccc1C(C)(C)C 552,C1(O)(CC)CC2CCC(C1)N2C(=O)CCc1nc(C2CCCC2)no1 553,N1(C(c2c(N)nccc2)=O)C2CCC1C(CNC(=O)CCCN1CCCCC1)C2 554,N1(C(C#CC2(C)CC2)=O)CCC2CN(C(c3c(Cl)cccc3Cl)=O)CCC2C1 555,C12(CC(N3C(CNC(C4CCC(C)C4)=O)C=CC3)=O)CC3CC(C1)CC(O)(C3)C2 556,C1(NC(c2n(CC)ncc2)=O)CCN(C(C23CCN(CC2)C3)=O)CCC1COC 557,c1(C(=O)NC2CCCN(C(c3cc(C)sc3)=O)C2)ccc2[nH]c(=O)cnc2c1 558,S(=O)(=O)(c1ccc2oc(O)nc2c1)N1CCC(Nc2cc(OC)nc(OC)c2)C1 559,c1(C(N2CC(CNC(C3C(C)(C(C)C)C3)=O)C2)=O)ncoc1C1CCCO1 560,Cc1cc(F)ccc1C(=O)NC1CN(C(c2ccncc2F)=O)CC1C 561,C(=O)(CC1=CCN(C)CC1)N1CC(C)C(NC(c2ccnc(Cl)c2O)=O)CC1 562,Cc1cc(NC(C2(NC(C3COCCO3)=O)CSC2)=O)c(C)s1 563,Cc1cnc(NC(C2CCN(C(c3ncc(F)cc3F)=O)C2)=O)c(Br)n1 564,c1(OC)ccc(S(=O)(=O)N2CCC(O)C(C)C2)c(C(F)(F)F)c1 565,c1(C(c2nnnn2Cc2cncc(F)c2)NC2(C(C)C)CC2)cccc(Br)c1Cl 566,N1(C(=O)Cc2ccnc(F)c2)CCC2(NC(C3(F)CCOC3)=O)CCCC12 567,c1(C(N2CCC(C(N3C(C)(COC)CCC3)=O)C2C)=O)ncc(N)cc1C 568,Cc1nn(C)c(Cl)c1CC(=O)N(C(C)CCNC(C1CCC(C)(C)CO1)=O)C 569,C#CCC(O)C(=O)NCC1CC1NC(c1cccnc1OCCCC)=O 570,c1(C(N2CCC3CN(C(C=C4CCC(C)C4)=O)C3C2)=O)ccc2c(c1)SCCN2 571,C(=O)(C1=CCCSC1)NCC(C)NC(c1ccccc1CSCC(F)(F)F)=O 572,Cc1ccc(C)c(C(N2CCC(C)N(C(c3cc(Cl)no3)=O)CC2)=O)c1N 573,C(=O)(C1=NN2CCCN=C2N1)NC(C)(CO)C1CCCO1 574,CC1CC(C(=O)NCc2ocnc2C(N2CCC(CO)C2)=O)CC(C)C1 575,C1(C(C)(C)CNC(C2C=CCC2)=O)CCN(C(=O)CC2CCCS2(=O)=O)CC1 576,C1(CNC(c2ncn(C)n2)=O)CC2(CO1)CN(C(=O)CC1(CO)CCCCC1)C2 577,N1(C(CCC=C)=O)CCC(CNC(C2CCC(F)CC2)=O)(COC)CC1 578,N1(C(c2ccc(C#C)cc2C)=O)CCC(NC(=O)C(C#N)C2CC2)C2(CCC2)C1 579,c1(OC)ccncc1CC(N1CC2CC1C2NC(=O)C(CO)NC(=O)C(C)C)=O 580,C1(C(N(C(C)CCNC(=O)Cc2ccc(O)nc2)C)=O)CCC(C)(O)CC1 581,c1(NCC2(NC(=O)C=CC3CCCO3)C(C)CCCC2)ncnn2cccc12 582,N1(C(CC2CCC(C)C2)=O)CC2(CCN2C(=O)CC(C)(F)F)C1 583,CCCCCS(=O)(=O)CC(=O)N1C2CCCC1CN(C(=O)CCc1cccs1)C2 584,c1(C(=O)NC(C)CN(C)C(c2ccc(OCF)cc2)=O)ccc(O)nc1Cl 585,C1(C(=O)NCC2CCN(C)C2)(CNC(=O)CC2COCCO2)CCCCC1 586,Cn1c(O)nc2cccc(C(N3CCCCC(NC(=O)CCS(C)(=O)=O)C3)=O)c12 587,c1(NCC(N2CC(CC)(NC(C3CCCN3S(C)(=O)=O)=O)C2)=O)ccc(F)nc1 588,CC(C)(C(=O)NCC1CC(F)CN1C(C1CC(=C2CCC2)C1)=O)C1=CCSCC1 589,C1(CNC(c2n(C)cnn2)=O)COCCN(C(=O)CCN2CCCC2)C1 590,N1(C(c2nc(CC)sc2N)=O)CC2(C)CN(C(C3CNC(=O)N3)=O)CC2(C)C1 591,CCCCC#CC(C)(C)NC(=O)CC(CC(C)C)NC(C1(C)C=CCCC1)=O 592,Cc1cc(C(=O)NCCCC2(NC(c3ccncc3Br)=O)CC2)[nH]c1C 593,N1(Cc2c(C)ccnc2)CCC(NC(c2cccc(F)n2)=O)C(F)C1 594,CC(=O)C(C)CC(C)C(=O)NCc1ccc(C(N2CCCC(CCF)C2)=O)nc1 595,C1(CCC)CN(C(c2ccc(OC)cc2OC)=O)CCN1C(=O)Cc1cnsc1 596,C(=O)(C(C)CC1CC1)NCC(C1CCCC1)NC(CSCC=C)=O 597,Cc1ccn(C)c(=O)c1NC(=O)CN(C(=O)C(F)CC1CCOC1)CC(C)C 598,Cc1cncc(C(N2CC(CCNC(c3cc(C(F)F)ccn3)=O)C2)=O)c1C 599,c1(C(=O)NCCN(C(c2ccsc2SC)=O)CC)c(Br)nnn1C 600,c1(NC(c2ccc(-n3cccn3)cc2)C)ccc(O)c(Br)c1 601,N1(C(CNC(=O)OC)=O)CCC(NC(c2c[nH]cc2-c2ccc(C)s2)=O)C(C)C1 602,N1(C(C(CN(C)C)O)=O)CC(NC(=O)CSCc2cccs2)C(C)(C)C1 603,C12(CNC(C(CC(C)C)SC)=O)CC(C(N)=O)(C1)C1(CN(C(=O)C(C)C)C1)O2 604,c1(CC(=O)NC2(COC)COC2)cc(F)ccc1F.C=C(C)CN1CC(=O)N1C 605,N1(C(c2cscc2F)=O)CCN(C(c2cccc(F)c2Cl)=O)C2COCC12 606,CC1(C(N2CCCC(NC(C3CCC3)=O)C2)=O)CS(=O)(=O)C1 607,C12CCCC(C1)CNC2=O.c1(CSC)ccc(OCC(N)=O)cc1.c1(=O)c(=O)[nH]1 608,c1(COC(=O)NC(C2CCN(C(=O)C(C)(C)C)C2)C(=O)OC)nc2ccccc2[nH]1 609,c1(C(N(CCNC(=O)C(F)CC2CCC2)CC)=O)ccc2c(C)nn(C)c2n1 610,C=C(C)CC(C)C(=O)NCC(=O)NOC(C)(C)CO 611,C1(NC(CCC(=O)NCCC)=O)CC2(NC(C3CC4CCC3CC4)=O)COC1C2 612,C#CC1CCCN(C(=O)COC(C)(C)CNC(=O)CC(C)C(F)F)CC1 613,Cc1cc(CNCC(C)(O)C2CC2)ccc1Br 614,C(c1ccc([N+](=O)[O-])cc1)=CC(=O)NC1CN(C(c2cc(Cl)cnn2)=O)C1 615,C(=O)(C(C(C)(C)O)NC(C12CCCC1C2)=O)NCCC(CC)(F)F 616,C1(F)(C(N(CCC(C)NC(C2CCCC23CC3)=O)C)=O)CCC(F)(F)CC1 617,C1(CNC(CC2(C(=C)F)CCC2)=O)CCCCCN1C(=O)C=Cc1cc[nH]c1 618,C1(CNC(CCOCCCNC(C(C)=C2CCC2)=O)=O)CC(O)C12CCC2 619,C(=O)(C1=CCS(=O)(=O)C1)N1CC(NC(=O)CCc2ccc(F)cc2Cl)C2(C1)CC2 620,C1(C2CC2)(NC(=O)C(F)n2ccnc2)CCN(C(c2ccc(Cl)o2)=O)C1 621,C1(C)(CC(=O)NC2CN(C(CCOCCOC)=O)C(C)C2)CCS(=O)(=O)N1 622,C=C(C(=O)N1CCN(c2ccc(OCC(F)(F)F)nc2)CC1)C1CCCC1 623,c1(C(N2C(C(=O)Nc3nnc(Br)s3)CC2)=O)ccc(C(F)(F)F)cn1 624,N1(C(CS(CC)=O)=O)CCN(C(=O)C(C)CSC(F)(F)F)C(C(C)C)C1 625,C1(CNC(COCC(N2CCCC2)C)=O)CCCN(C(C2CC(F)(F)CS2)=O)C1 626,C1(CCCCNC(Cc2cc(C)no2)=O)CCCN(C(c2ccnc(O)c2)=O)C1 627,N1(C(C2(c3ccccc3Cl)CCC2)=O)CCCc2c(-c3nn[nH]n3)cccc21 628,c1(CC)cccc(C(=O)NC2(C(=O)NCC(C)CC3CC3)CC2(C)C)n1 629,C1(C(=O)NCc2cccc(C(C)C)n2)Cc2cccnc2C1 630,c1(OC)oc(C)nc1C(=O)NCCC1CCN(C(C2CCOC2=O)=O)CC1 631,C1(NC(c2c(SC)cn(C)n2)=O)CC(F)CN(C(C2CC=CCC2)=O)C1 632,c1(CNC2(C(=O)NC(CC)(C)CNC(=O)Cn3cncn3)CC2)ccc(C)cc1 633,c1(CC(=O)NC(Cc2cn(C3(C(=O)OC)CCC3)nn2)C(=O)O)ccccc1Br 634,CS(=O)(=O)C1(CNC(C2(c3ccc(F)cc3)CC2)=O)CCC1 635,c1(C(=O)NCC2CC(NC(C(C)(C)c3cccnc3)=O)C2)[nH]c(=N)sc1C(F)F 636,C1(COC)CN(C(c2ccc(Cl)cn2)=O)CCN1C(c1ccc(F)c(CO)c1)=O 637,CCC(CC)C(=O)N1CC=CC1(C(=O)NC1C(C)C1(C)C)COC 638,c1(OC)ccc(OC)c(C(=O)CCC(=O)NC(C)CCNC(C2CC2F)=O)c1 639,N1(C(C2(CC)CCN(C(=O)CC(C)C(F)F)CC2)=O)CC2(COC(=O)C2)C1 640,C1(C)(CN(C(C)C(=O)NC2COCC2O)C)CCN(C(=O)OC(C)(C)C)CC1 641,C(=O)(C(C)C(C)(C)c1ccccc1)NC1CC(N(C(=O)CC(=O)OC(C)(C)C)C)C1 642,N1(C(C(CC#C)C)=O)CC(NC(=O)C(C2CC2)C2CC2)CCC(O)C1 643,Cc1nn(C)cc1C(C)NC(C1CCN(C(c2cc(C(N)=O)[nH]n2)=O)C1)=O 644,Cc1ccc(C(N2CCCC(NC(c3ccn(C)n3)=O)C2C)=O)c(F)c1Cl 645,c1(C(N2CCC(NC(C(CC#C)C3CC3)=O)C(O)C2)=O)ccc2c(C)[nH]nc2c1 646,C(=O)(CC(CC)C1CC1)NCC(CNC(C(C)(C)OCCC)=O)(C)F 647,C1(CNC(C2CC2(Cl)Cl)=O)CN(C(=O)COCC2CCC2)C2(CCC2)C1 648,C(=O)(C1=CC2CC(C1)CC2O)NCC1N(C(CCC(=O)NCCC)=O)CCC1 649,C1(CC)OCCCC1C(=O)NCc1ncoc1CCNC(C1CCN1C)=O 650,N1(C(C2(CC(C)C)COC2)=O)CC2OCCN(C(=O)C(F)CC(C)C)C2C1 651,C(=O)(C(C(=O)N1CCC(CNC(C2(CF)CC2)=O)C1(C)C)C(C)C)OCC 652,C1(NC(c2c(CC)nns2)=O)(CO)CCN(C(C2(OC)CC(CF)C2)=O)C1 653,Cc1cc(N(C)C(C2CSC(c3ccc(C(F)(F)F)cc3)C2)=O)cc(F)c1 654,CC(CCC(=O)NCCCC(O)CO)NC(=O)C(C1CCOCC1)=O 655,CON(CCC(=O)N1CC2CC2(CO)C1)C(=O)Cc1ccccn1 656,N1(C(c2c(CCC)n(CC)nn2)=O)CCC(NC(C2(CC(F)F)CC2)=O)C(C)C1 657,C1(NC(CC(C(C)C)O)=O)CCC2(CC1)CN(C(=O)C1=CCC(F)(F)CC1)C2 658,CCCC(C(=O)N1CCC(NC(c2cc(C)n(C)n2)=O)C1)NC(N)=O 659,c1(C(N2CCCCC(NC(C(C(CC)C)C)=O)C2)=O)cc(OC)cc(OC)c1N 660,CC(C(=O)N1CCC(CC2CC2)CC1)C(C)NC(c1ncccc1Cl)=O 661,c1(CCC)onc(C)c1C(=O)NCC(F)CNC(=O)C(F)(F)c1ccccn1 662,N#Cc1ccc2cc(C(=O)NCCCCNC(c3ccc(Br)o3)=O)ccc2c1 663,Cc1c(CN2CCCC(C(=O)N(CCC(C)(C)O)C)C2)cnn1C 664,C(C(C(=O)NC1CCC(C2CC2)C1)C(C)(C)C)NC(C(CCC)(F)F)=O 665,C(N=c1ncnc(N2CCCCC2)[nH]1)c1c(C(=O)OC)snn1 666,Cc1c(F)ccc(N)c1C(=O)NC1CC(CNC(C23CCC2C3)=O)C1 667,N1(C(c2cc(CC)no2)=O)CC(NC(=O)C(C)NC(=O)NC)CC2(CC2)C1 668,n1(CC)nc(C(=O)NC2(C)CN(C(=O)CC(F)(F)F)C2)c(Cl)c1Br 669,[N-]=[N+]=NC1(C(N2CCC(O)(C(N)=O)C2)=O)CCN(C(C2CCCS2)=O)C1 670,N1(C(C2CCN(C(C(C)CC(N)=O)=O)C23CC3)=O)CCCC(C)(C#N)C1 671,Cc1nc(C2CCN(C(c3ccoc3)=O)C2)n[nH]1 672,N1(C(C(C)O)=O)CCN(C(C2CS(=O)(=O)C2)=O)C(C2CCC2)C1 673,C12(NC(c3n(C)nc(O)c3)=O)CCCC1CN(C(C1CCCS1)=O)C2 674,c1(NC(CC2CCN(S(CC)(=O)=O)CC2)=O)ccc(C)nc1F 675,c1(OC)nc(C)ncc1C(=O)NC1CCN(C(c2cc(CN(C)C)on2)=O)C1C 676,c1(NC(C2C(CN)OCC2)=O)cccc(CC2CCNCC2)c1 677,c1(C(=O)NCCC(CNC(CC2(C)CCCC2)=O)O)ccc(F)cc1N 678,CCC1=NOC(C(N2CC3CC3(CNC(=O)C(F)=C3CCC3)C2)=O)C1 679,CCCC(C(=O)NC(c1ncccc1F)C)NC(c1csc(Cl)n1)=O 680,N1(CCCOC)CC2CC(NC(=O)Cc3csc(NS(C)(=O)=O)n3)C1C2 681,Cc1cc(=NC2CS(=O)(=O)CC2NC(=O)C=CCO)nc(-c2cccs2)[nH]1 682,c1(C(C)=O)cc(C(=O)N(CC(C)NC(c2cnc(O)s2)=O)C)cnc1C 683,C(c1ccccc1OC)=CC(=O)NCC(CNC(c1cc(CCC)nn1C)=O)F 684,N1(C(CCSCCC)=O)CCCC2C1CCN2C(=O)C(C)CC1CCCC1 685,c1(C(=O)NCCC2CCCN(C(C3CN(C(C)=O)C3)=O)C2)cn(C)c(C)cc1=O 686,C1(OC(=O)N(C)C(c2cn(C3CC(C(=O)OC)C3)nn2)=O)(OC)CCC1(C)C 687,CC(CS(C)(=O)=O)C(=O)NC1CN(C(c2cc(O)c(O)c(O)c2)=O)CC1C 688,CN1C(=O)CCCC1C(=O)NCC1CCCN1C(C1CC2CCC1C2)=O 689,CCCC(C(=O)N1CCC(CNC(=O)CCCOCCc2ccccc2)C1)OC 690,n1(CCN(C(c2csc(CO)n2)C(=O)NC2CCOCC2)C)cc(C2CC2)nn1 691,N1(C(CCCC(C)(C)C)=O)CCC2CCN(C(=O)CC3C=CS(=O)(=O)C3)CC12 692,O=C(CC1CN(C(c2csnn2)=O)CCO1)N=c1cc(Br)[nH][nH]1 693,c1(CC)cc(C)c(C(=O)NCc2ncccc2C(=O)NOCC2CCOCC2)o1 694,Cc1nc(N2CCCC(C)(CNC(C34CCC(C)(C3)OC4)=O)C2)cc(C#N)n1 695,c1(NC2CC(C(CSC)C)C2)nc(=N)nc(C(F)F)[nH]1 696,C=CCC(C(=O)N1CCC(C)(C(N2CC=CC(OC)C2)=O)C1)OC 697,N1(C(CSCCC(C)C)=O)CCOC(CC(=O)NC(C)CCCCO)C1 698,c1(NC(C2N(C(C(C)n3cccn3)=O)C3C(C2)C3)=O)ccc(F)c(Cl)c1 699,C(CCN=c1[nH]c(C)cc(=NC2CCC(C)(C)CC2C)[nH]1)N(S(CC)(=O)=O)C 700,CCCC(CC(=O)NCC1(O)CCCC1(C)C)NC(c1c[nH]nc1Cl)=O 701,c1(C(N2C(CNC(=O)Cc3cc(C(F)F)no3)CC2)=O)c(Cl)cccc1Cl 702,c1(CCC(=O)NC(CC2CN(C(CS(CC)=O)=O)C2)C)cc(F)ccc1F 703,CCC1=C(C(=O)NC2CCC2NC(=O)C(N2CCN(C)CC2)C)CCCO1 704,C1(CNC(C(C(=O)NC2C3(CN)CCC2C3)(C)C)=O)Cc2ccccc2CO1 705,C1(CNC(=O)CONC(=O)C2CCOC2)(COCCO)CCOC1 706,Cc1nc(NC2CN(C(C3CC(C)CO3)=O)CCC2C(F)(F)F)c(C)c(O)n1 707,C1(NC(C(C)NC(c2cccs2)=O)=O)CN(C(=O)CSC2CC2)CC1C 708,c1(C(C)C(=O)NC(C2CCCN2C(C2CCC2)=O)C)ccccc1F 709,c1(CSC)cc(C(=O)NC2CN(C(c3cc(C)c(Cl)cn3)=O)CC2F)ccc1F 710,CC1CC(NC(c2ccc(C(F)F)cc2)=O)CN1C(=O)C(F)=CC1CC1 711,c1(C(N2CCC(CCCNC(C3CCCC3)=O)CC2)=O)c(O)cc(F)cc1F 712,N1(C(C2CC(OC)C2)=O)CCC2(CCC2)C(NC(=O)C(n2nc(C)cc2C)C)C1 713,c1(OC)ccc(OCC(N2CCC(C(=O)NCCOc3ccccc3)C2)=O)cc1 714,c1(NC(C(C)NC(c2ccc(CO)nc2)=O)=O)cccc2ccoc12 715,C(=O)(C(O)C1=CCCCC1)NCCCCCCC(=O)NC1(C)CCC(C)CC1 716,N1(C(C(CCC)C)=O)CCC2(CNC(C3(C(N)=O)CC3)=O)CCCCC12 717,c1(C(=O)NC(C(C)NC(C2COCCO2)=O)(C)C)ccc2cn(C)nc2c1 718,c1(OCC)ncc(Cl)cc1C(=O)Nc1nc(-c2cccc(C(=O)O)c2C)cs1 719,N1(C(C(CCCC)O)=O)CC2CCCC(C1)N2C(c1[nH]cnc1CC)=O 720,C1(C(C)NC(=O)CCCn2cc(C(C)(C)C(=O)O)nn2)COCCO1 721,O=S(=O)(c1c[nH]c2ncccc12)NCCc1nc(-c2cccs2)n[nH]1 722,C1(NC(C(C)Sc2ccccn2)=O)CCCC12CN(C(=O)Cn1cnnc1)C2 723,N1(C(c2cc(C)c(C)o2)=O)CCC(C(=O)NCc2cc(Cl)no2)C(C)(C)C1 724,N1(C(C2=C(C)OCCS2)=O)CC(C)OC2(CCN(C(c3ccc(=N)[nH]n3)=O)C2)C1 725,O=C(C(O)CC(F)F)NCc1cc(Cl)cnc1Cl 726,N1(C(C(C)C(F)F)=O)CCC2CC2(C(N2CCC3C(O)CC23)=O)CC1 727,O=C(CC(C(F)F)n1cccn1)N1CCCC(Nc2ncns2)CC1 728,c1(NC(C)=O)ncc(S(=O)(=O)N2CCC(O)(CNC(C3C4COCC34)=O)CC2)s1 729,C=C(C)CC(C(=O)N1CC(C(N)=O)C2(CC2)C1)NC(c1sccc1C#N)=O 730,C1(CNC(c2cccs2)=O)CN(C(c2c[nH]nc2Br)=O)CCO1 731,c1(C(=O)NC2C3(CC(NC(C(C)CN4CCCCC4)=O)C3)C2)cccc(N)c1F 732,C1(CC(=O)N(C2C(C)COCC2)C)C2CCCC2N1C(C1C2CC3C(C2)C13)=O 733,C1(C(=O)NCC(C)NC(=O)CN2CC(C)(C)C2)COc2ccc(O)cc2O1 734,C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)N(C1CCN(C(CCCC)=O)CC1C)C 735,C1(CC(=O)N(CCNC(C2C(C)(CC)C2)=O)CCOC)CCC(=O)NC1 736,N1(C(C(=O)N(c2ccc(OCCOC)cc2)C)=O)CCn2cc(C)nc2C1 737,C1(c2n(CCC)nnn2)(Nc2ccc(CCO)c(O)c2)CC2CC(OC)C2C1 738,CC(C)CC(C(=O)NCCNC(c1cccnn1)=O)N(C)C.C1(C)CNC(=O)N1 739,C1(C(N2CC(C(=O)OC)C2)=O)CC=CCN1C(c1csc(CO)n1)=O 740,N1(C(c2cn(C(C)C)nc2)=O)CCN(C(=O)COc2ccc(F)cc2)C(C)C1C 741,C1(CNC(c2c(CC)nc[nH]2)=O)CN(C)CCN1C(=O)COc1ccsn1 742,C(=O)(CS(=O)c1ccc(Cl)cc1)N1CC2C(NC(c3c(C)coc3)=O)C2C1 743,S(=O)(=O)(c1cc(C(C)(C)C)ccc1C)Nc1ccc(OC)cc1.C1CC(=O)O1 744,CCC(C(=O)NCCCC(C)NC(c1ccc(C)nc1N)=O)C(C)C 745,C1(CNC(c2cnc(C(C)(C)C)[nH]2)=O)CC(NC(=O)Cc2nc(=N)[nH][nH]2)C1(C)C 746,N1(C(C2CC(C)CN2C(c2c(Cl)cnn2C)=O)=O)CCC(=O)N(C)CC1 747,C1(N(C(COCC)=O)CC)CN(c2cc(COCC)ncn2)CCO1 748,Cc1ccc(=N)[nH]c1C(N1CCN(C(=O)C(C)C2CCCC2)CC1C)=O 749,C1(C(C)NC(C(F)OC)=O)CCN(C(c2ccccc2OCF)=O)CC1 750,C1(C)(NC(CC2CCCN(C(C(C)NC(CC)=O)=O)CC2)=O)CCC2(CC1)CC2 751,N1(C(c2cc(CC)oc2C)=O)C2CCC(C2)C1C(=O)NC(c1cccc(C)n1)C 752,c1(C(=O)NC(c2nnc(CC)s2)C)ccc(NC(=O)COC)c(Cl)c1 753,c1(OCC)nc(N(CCCN(C(=O)C(CO)c2ccccc2)C)C)ncc1Cl 754,C1(C(=O)N(C2CCC(NC(=O)C(C)NC=O)CC2)C)(OC)CCCCC1 755,N1(C(c2c(C)nncc2)=O)CCC(CO)(CNC(C2CCSCC2)=O)CC1 756,N1(C(C(OC)OC)=O)CC(CO)C2(C1)CN(C(=O)C(CC(C)C)NC(C)=O)C2 757,Cc1cccc(CNC(C23CC2CN(C(C2CCC(=O)N2C)=O)C3)=O)c1O 758,c1(NC(CNC(C2(C)CCC(C)C2)=O)C2CC2)cc(=O)n2cc(Cl)ccc2n1 759,n1(CC)ccnc1C=CC(=O)NCC1C=CCN1C(=O)C(c1ccc(Cl)cc1)C 760,C1(C(=O)NCC(CC)N(C)C(c2cncc(OC)n2)=O)CCCCN1C 761,C1(C(=O)NCCCCNC(CN(CC)CC)=O)CCc2nnc(Br)n2C1 762,C#CCC(CC(=O)NCc1ccncn1)NC(c1ccc(C)cc1F)=O 763,c1(N2C(C(=O)NCc3cn(C(C)C)nc3)CC(F)C2)ncnc2c(Br)csc12 764,C1(C(=O)NCC2N(C(C34OCCC(C)(C3)C4)=O)CCOC2)CCc2ccnn2C1 765,C1(CCNC(C(=O)NCCc2nc(-c3ccc(C)o3)sc2)=O)COCC(C)O1 766,C(=O)(CCCCCC(C)(C)C)NCC1(OC)CCN(C(CC=C=C)=O)C1 767,N1(C(C=C(C)C)=O)CCCC2(CCN(C(c3c(Cl)ccc(Cl)c3O)=O)CC2)C1 768,C1(NC(CCC(C)N(C)C)=O)CC2(C1)CC(NC(C1CCC1C)=O)C2 769,Cc1cc(C(=O)NC2CCC2CNC(c2cn(CC(F)(F)F)nn2)=O)n[nH]1 770,c1(CC(=O)NCC(CN(C(C(C2CCCC2)OC)=O)C)O)cccc2occc12 771,C(=O)(C1=CCCCCC1)NC1C(N(C)C(C2CC23CCOCC3)=O)CCCC1 772,C1(C)(C(N(CCN(C(=O)CN(C2CCCC2)C)C(C)C)C)=O)CCOC(C)C1 773,C1(C2CCCN(C(C3(OC)CCC3)=O)C2)(NC(c2c(C)nn(CC)c2C)=O)CC1 774,c1(NC)c(C(=O)NC(C)(C)CNC(=O)CC2CC3CC3C2)cccc1[N+](=O)[O-] 775,Cc1cnn(C(C)C(=O)NCCCCNC(=O)C(C)OCCN(C)C)c1 776,C(=O)(CCS(=O)(=O)c1ccc(Cl)cc1)NC(C(C)NC(CC(C)OC)=O)C 777,N1(C(c2c(CC)nccn2)=O)CCC2(CC1)CCN2C(=O)CCC1CCOC1 778,C1(CC)CCN(C(c2coc(CO)c2)=O)C(C(=O)NC(COC)C(C)C)C1 779,c1(C(N2CCCC(CCNC(C3(NC(C)=O)CCC3)=O)C2)=O)cnc(O)c(C)c1 780,C1(C)(C(=O)NCCCN(C(=O)C(C)(CC)CO)CC)CC2(C1)CC(F)(F)C2 781,N1(C(c2c(C(C)C)sc(Cl)n2)=O)CC2(CCN(C(c3ccns3)=O)CC2)CC1C 782,C1(OC)CCC(N=CC(N2CC(O)(CNC(=O)COc3ccncc3)C2)=O)CC1 783,CCC(F)(F)C(C)(C)C(=O)NC1CCCCCC1NC(C1CCN(C)CC1)=O 784,Cc1cnc(CCCC(=O)NC(CNC(C2(Oc3ccccc3)CC2)=O)CO)o1 785,C1(CC(=O)NC2CC2C2CC2)CCN(C(C2CC2(Cl)Cl)=O)C1 786,C#CCCN=C(NCC(c1cc(C)oc1C)C)NC(C)C 787,Cc1cccc(C(F)C(=O)NC2CC(CNC(C3CC4CC4C3)=O)CC2O)c1 788,C1(NC(CCCc2cc(C)no2)=O)CC2CN(C(C3CCC3)=O)CC2C1 789,C=CCCCCC(=O)N1C2CCC1C(CNC(=O)CCC1CCCOC1)C2 790,Cc1cc(Br)oc1C(N1CCC(Cn2cc(CC(O)C3CC3)nn2)CC1)=O 791,S(=O)(=O)(c1ccc(=NCC2(n3cccn3)CC2)[nH]c1)N1C(CC=C)CCC1 792,C1(C(=O)NCC(C)(CC(C)C)NC(CCN(C)CC)=O)COc2ccccc2C1 793,c1(CCNC(=O)CCC2(NC(C3CCCCO3)=O)CCC2)ncccc1F 794,C12CCC(F)(CC1)CNC(=O)C(=O)NC2.N1(C(C)=O)CCC(C(=O)NC2CC2)C1 795,N1(C(CCCCC)=O)CC(C(=O)NCC(C)C(F)F)CC1(C)C 796,N1(C(C=C(C)C)=O)CCN(C(c2ccc(C(C)(C)C)cc2C)=O)C(C(F)(F)F)C1 797,CCCCC(C)CCC(=O)N(CCNC(c1cc2nnn(C)c2s1)=O)CCOC 798,C1(C(=O)NC2CCN(C(c3cc(C)nn3CC(F)F)=O)C2)CCC(=C(F)F)CC1 799,N1(C(C(CC)(C)CC)=O)CCCC2(C1)C(NC(=O)C(C)SC)CCN2C 800,C(c1ccc([N+](=O)[O-])s1)=CC(=O)NC1CCN(C(CSCC(=O)OC)=O)C(C)C1 801,c1(C(N2C(CCOC)CN(C(C3CC3(C)C)=O)CC2)=O)nc(C)n2ccccc12 802,c1(C(=O)NC23CCN(C(c4ccc(Br)o4)=O)CC2C3)ccc2occc2c1 803,CCN=C(NCCOCCOCCOC)NCC1(c2ccccc2F)CCCC1 804,c1(OC(C(=O)NC(CNC(CCC=CC)=O)C2CC2)CC)cccc(C)c1 805,c1(CC)ccccc1C(N1CCCC(CN(C(=O)COCCOC)CC)C1)=O 806,c1(C(N(C2CN(C(CSCC=C)=O)CC2F)C)=O)cc(Cl)c(F)cc1C 807,c1(C(=O)NCC(CN(C(c2c(C)nn(C)n2)=O)C)(C)C)nc2ncccn2n1 808,C1(F)(CNC(C2(OCC)CCOC2)=O)CCCN(C(=O)C=Cc2ccsc2)CC1 809,C1CC(C(C)(C)C)OC(=O)C(=O)N(C)C(C(F)F)CC(=O)O1.C(C)(C)(C)OOC 810,C1(CNC(Cn2nc(C3CC3)n(C)c2=O)=O)CNCCS(=O)(=O)C1 811,Cc1ncc(CC(N2CCC(N(C(=O)C=Cc3cn[nH]c3)CCO)C2)=O)[nH]1 812,Cc1cccc(C(N2CCC(C(=O)N(CC(O)C(C)(C)C)C)C23CC3)=O)c1C#N 813,CCC(CC(C)C)C(=O)N(C)CC1COCCN1C(c1nn[nH]c1Cl)=O 814,c1(N2CCN(Cc3cccc(-c4ccc(OC)cc4)n3)CC2)cnc(C)c(C)c1 815,N1(C(C2C(CC)CCN2C(c2ccc(N)cn2)=O)=O)CCC2(CCCO2)CC1 816,N1(C(CCC2(C)CCCN2C(c2cc(N)cc(F)c2)=O)=O)CC2(CCC(=O)N2)C1 817,N1(C(CCCCC)=O)CC2CC(NC(=O)C(O)Cc3cc(Cl)cc(Cl)c3)C1C2 818,N1(C(CSCCOC)=O)CCCC2C1CCN2C(c1ccc2ccn(C)c2c1)=O 819,c1(OC)cccnc1C(=O)NC1COCC1NC(c1ccc(=O)oc1)=O 820,c12ccc(cc1)C1(CC1)CNC(=O)C2C.N1(C(C)=O)CCCC1C(F)(F)F 821,C(=O)(C(F)(F)C(F)(F)F)NCC1(C)CN(C(c2cscc2C#N)=O)CCO1 822,C1(NC(c2ccc(Br)o2)=O)CC2CCC(C1)N2C(=O)CC1CCC(F)(F)CO1 823,C1(NCc2cccc(C(N)=O)c2)C=CCCCCC1 824,c1(C(c2n(CCCOC)nnn2)NCc2nnnn2C)ccncc1Br 825,CCC(C)(CO)C(=O)NCC1CC2CN(C(c3oc(C4CC4)nc3C)=O)CC12 826,C1(N(C(CN(CC)CC)=O)C)CCCC2CN(C(=O)CCc3cn(C)nn3)CC12 827,c1(C(N2CCC(N3C(CSC)CCC3)C2=O)=O)cccc2c1OCO2 828,C(C(=O)N=c1cc(C)o[nH]1)NC(C1(NC(C)=O)CCCC1)=O 829,c1(C(=O)NCC(C)(C)NC(c2c[nH]ccc2=N)=O)cccc2c1CCOC2 830,C(CS(=O)(=O)NCC1CCC(O)C1)OCCC(C)C 831,C(=O)(C(CCC(C)C)NC(c1ccncc1O)=O)N1C(COC)CCC1 832,c1(C(=O)NC2C(F)CCN(C(Cc3c(C)n(C)nc3)=O)C2)n[nH]c2c1CSCC2 833,Cc1nccc(NC(=O)NCC2CN(C(=O)Cc3ccccc3F)C2)n1 834,c1(C(=O)NC2C3CN(C(COCC)=O)C2CC3)cc2ccc(NC(C)C)cc2[nH]1 835,N1(C(C2CCN(CCCc3ccccc3)C2=O)=O)CCCC(O)(C(F)F)C1 836,c1(-c2ccc(C(N(C)CC3CC(=O)CCC(=O)N3)=O)cc2)cc2ccccc2[nH]1 837,c1(C(N2CC3C(CNC(CC4(NC(C)=O)CC4)=O)(C3)C2)=O)cc(C(C)C)n(C)n1 838,C(=O)(C(F)(F)CC(C)C)N1CCCC(CC)(NC(=O)Cn2ccc([N+](=O)[O-])n2)C1 839,c1(OC)ccnc(C2CCN(C(=O)CN3CCNC3=N)C2)c1 840,N1(C(c2cc(C)c(Cl)s2)=O)CC(N(C(=O)CCc2ccc(=N)[nH]c2)C)C(C)(C)C1 841,c1(CN2C(C(=O)Nc3c(C#N)ncc(C)n3)COCC2)ccc2nc(C)oc2c1 842,C1(NC(Cn2ncc(C)c2)=O)CCC(C)N(C(=O)Cc2cncn2C)C1 843,C12(CNC(C(C3CC3)OC)=O)CCCC1N(C(C1CCC(C)C(C)C1)=O)CCC2 844,c1(CNC2(c3n(CC(=C)C)nnn3)COC(C)(C)C2)ccc2[nH]nc(F)c2c1 845,CC1CCC(C)(C(N2CCN(C(=O)C=Cc3ccc(Cl)s3)C(CCO)C2)=O)CC1 846,N1(C(CCNC(C)=O)=O)CC2C(N(C(=O)CN(C)C(c3ccccc3)=O)C)C2C1 847,N1(C(c2n[nH]c(=N)s2)=O)CCCC2(NC(=O)Cc3cc(O)nnc3O)CCCC12 848,c1(C(N2CC(NC(C(C)(C)F)=O)C2)=O)cc(Cl)ncc1Br 849,Cc1[nH]c(C)c(C(=O)NCCCCC2CCN(C(C3OCCCO3)=O)CC2)c1C 850,c1(C(N2CCC(O)(CN(C(C(CC)O)=O)C)C2)=O)cnc2ccccn2c1=O 851,C#CC1CCCC1NC(=O)CC(CC1CC1)NC(=O)C=CC1CCCC1 852,Cc1cc(F)c(C(=O)N(C2CN(C(=O)C(C)(C)c3cccs3)C2)C)cc1F 853,c1(CC(=O)NCC(CC)NC(=O)C(C(C)C)NC(=O)OCC)ccc(C)cc1Cl 854,C(=O)(C(C)C(O)CC(C)C)NC(CC=CC)C(=O)N(C)CC1OCCC1(C)C 855,c1(C(=O)NCC(C)NC(c2c(SC)cccc2)=O)cnn2c(C)ccnc12 856,C(=O)(C1CCCc2n[nH]cc21)N1CC(CNC(C(C)(C)N(C)C)=O)C(C)(C)CC1 857,c1(C(=O)OC)ccc(NC(c2cccc(C3CC3(F)F)c2)=O)c(OC)c1Cl 858,c1(COC)nn(C)c(Cl)c1C(N1CCC(F)C(NC(=O)Cc2cc(C)no2)C1)=O 859,c1(C(=O)NCC(CN(C)C(C2COC(=O)N2)=O)(C)C)cccc[n+]1[O-] 860,c1(CN2CCC(OCC(=O)O)C2)cc2cncn2c(O)n1 861,c1(C(=O)NCC(CCC)C(=O)NCc2scnc2C)n[nH]c2ccccc12 862,CC1CCCC(C)N1C(N1CCN(C(c2ccc(SC#N)cc2)=O)CC1)=O 863,c1(C(=O)NC2(C)CN(C(C(CC)(C)C)=O)C2)cc(OC)c(OC)c(OC)c1N 864,c1(OCCC#C)ccc(C(=O)NCCNC(c2ccccc2CSCC)=O)cc1 865,c1(C(=O)NC2C(NC(=O)CCN3CCOC3=O)CC2)ccc(OC2CCC2)cn1 866,O=C(C1SCCc2sccc21)N1CC(c2cn(CC3CCOCC3)nn2)C1 867,N1(C(c2ccc(C)c(C)n2)=O)CC=C(C(=O)N2CCC(CC3CC3)C2)CC1 868,c1(C(=O)NC(CCN(C)C)C(=O)NC2CCN(CCF)C2)ccnc(O)c1F 869,c1(CCC(=O)NC2CC2NC(c2cc(C3CCOCC3)no2)=O)cccnc1F 870,C1(CNC(C2C(C)(C)C2)=O)CCC2(CCN(C(c3n[nH]cc3[N+](=O)[O-])=O)CC2)O1 871,c1(OC)cc(C(C)NC(=O)Nc2c(OC)ccc(F)c2OC)c(F)cc1F 872,C1(CN(C(=O)CC2CC2(C)C)C)CCCN(C(=O)Cc2cnco2)C1 873,c1(OC)ccc(-c2cccc(NC(C3(C(C)(F)F)CCC3)=O)n2)cc1 874,C1(OC)CC2CC(C(N3CC=C(CNC(=O)C(N)=O)CC3)=O)CC12 875,N1(C(c2on(C)c(=O)c2)=O)CCC(NC(=O)CCc2ccccn2)CC(C)(C)C1 876,N1(C(CCN(C(c2ccc(CC)cn2)=O)CCO)=O)CC(=O)NC2(CC2)C1 877,N1(C(c2cc(C)sc2)=O)CC(CNC(C2CCCC(C)O2)=O)CC1C 878,C(=O)(C1=Cc2cc(F)ccc2OC1)NC1C(NC(CSC(C)(C)C)=O)C1 879,c1(NC2C(C)CN(C(C=C(C)C(F)F)=O)CC2C)cc(C)ccc1[N+](=O)[O-] 880,C1(CNC(c2ccc(CC)o2)=O)CCCCN(C(=O)C=C(C)C2CC2)C1 881,N1(CC(N2CCOCC(NC(C(CC)O)=O)C2)=O)CCc2ccccc21 882,C12CN(CCC1(F)F)CCOC2.C1(C(=O)O)CC2CCC2C1 883,C(C1=CCCN(C(C2COCOC2)=O)C1)NC(Cc1c(C)nsc1)=O 884,N12CCC(C)(C1)CNCC1(CCCC1)CC2=O.C(=O)C(C)C.CO 885,N1(CCC(N2CCC(CNC(COCCC)=O)C(C)C2)=O)C(=O)NC(C)(C)C1=O 886,CC1(C)CCCCCC1NC(=O)C(CNC(C1OC2CCC1C2)=O)C(C)(C)C 887,C1(C(=O)NC2CCC(O)CC2)C2CC(CC2F)N1C(=O)CC1(O)CCC1 888,N#Cc1c(CN2CC3CC2CN3S(=O)(=O)Cc2ccc(Cl)cc2)cccc1Cl 889,N1(C(=O)OC)CCC(C(=O)NCC2CCN2C(c2ncsc2C(C)C)=O)CC1 890,N1(C(C2(CC)CCN(C(C3CC4C=CC3CC4)=O)C2)=O)CCC2(CCCCC2)C1 891,C1(CCC)(NC(=O)CC2CC(O)CN2C(c2cccnn2)=O)CCNC1=O 892,N1(C(C(=O)NC(C)C)=O)CC(NC(=O)CSCC2CCCCO2)C(C(F)F)C1 893,C1(CNC(C(=O)NC(C)C)=O)CC2(CCC2)CN1C(C1CCCC1C(C)C)=O 894,c1(C(N2CC(NC(CC3N(CC)CCC3)=O)C2)=O)ccc(C(C)=O)cc1C 895,c1(OC)cc(-c2cn(CCN(C(=O)CCn3ccnn3)C)nn2)ccc1F 896,C1(C(N(CC(F)F)C)=O)C(CNC(C2CCCS2)=O)C1(C)C 897,c1(C(N2CCC(OCCNC(C3(CC)CCOC3)=O)C2)=O)c([N+](=O)[O-])cnn1C 898,N1(C(CN(S(C)(=O)=O)C)=O)CCN(C(=O)CC2OCCCC2(C)C)C2COCC12 899,S(=O)(=O)(C1CCC2(CC1)CC2)N(C1C(C)CCC1)C 900,c1(COC(C2CC(C)N2C(c2ccc(CN)nc2)=O)=O)ccc2c(c1)N(C)CC2 901,N1(C(c2c(C)c(C3CC3)on2)=O)CC2CCCC1C2CNC(=O)Cn1cncn1 902,Cc1cc(C(=O)NC2CC3CC2N(C(=O)COCc2cc(C)no2)C3)nc(C)c1 903,c1(C(N2CCN(C(COCC(C)(C)C)=O)CC2C2CC2)=O)cc2c(s1)CCOC2 904,CC1=C(C(=O)N(CCCNC(C2CN(S(C)(=O)=O)C2)=O)C)CCO1 905,N1(C(C(C(CC)C)O)=O)CC2CCN(C(C3C4(CC4)C34CC4)=O)CC2C1 906,c1(C(N2CCC3CN(C(CCCOC)=O)CC32)=O)cc2cc(C)ccc2[nH]1 907,CCC(C)(F)C(=O)NC(C)CNC(C1(Sc2ccccc2)CC1)=O 908,O=C(CC1=CCCC1)NCc1ncccc1C(=O)NC1CCCCC12CC2 909,c1(N(CCCCN(C(=O)CC2COC(=O)C2)C)C)nnc(C2CC2)o1 910,CC1(C)CC2CC(C)(CN2C(c2cc3ccncc3[nH]2)=O)C1 911,C1(Nc2cccc(C(C)=O)n2)CCN2CCCCC12 912,c1(OC)cc(O)ncc1C(N1CC2C(CNC(c3n[nH]cc3[N+](=O)[O-])=O)C2C1)=O 913,CCC(CC)C(=O)N1CC(O)CC1CNC(C1CCCN(c2nccs2)C1)=O 914,C(=O)(C(CO)C(F)(F)F)NCCC1(C)CCN(C(C2CCC2(F)F)=O)C1 915,c1(C(N2CC(CCNC(C(CC(C)C)C)=O)OCC2)=O)cc2ccccc2cn1 916,c1(C(=O)NC2CCCCN(C(C3OCCN(C)C3)=O)C2)cncc2ncccc12 917,C#CC1(C(=O)NCC(C)C(C)C)CCN(C(=O)COCCC(C)C)C1 918,c1(CNc2cc(NC(c3nccs3)C)ncn2)cc([N+](=O)[O-])ccc1Cl 919,CCC(CCCC(=O)N=c1ccn(C)[nH]1)NC(=O)COCCF 920,N1(C(=O)CC23CC(C2)C3)CCC2C1CCCN2C(=O)CCc1cccnc1 921,N1(C(=O)NCCCC2CC2(F)F)CC2CCCCC12c1ccccc1 922,C(CCC(O)C(=O)NC1CCCCCC1F)NC(CC1(N(C)C)CCC1)=O 923,C1(CNC(CCN(C(=O)Cc2cn(C)nc2C)CC)=O)CC(F)(F)CO1 924,N1(C(c2c(CC)nc(C)o2)=O)CCC(NC(c2cc(Cl)cs2)=O)C(C)(C)C1 925,CC(C)C(C)(C)C(=O)NC1CN(C(C2CCCN(CC(F)F)C2)=O)CC1O 926,CC#CCCCC(=O)NC(CCSC)C(=O)NCCNC(=O)CC.OC 927,Cc1nc(NC(c2nnnn2C2(C)CC2)(C)COC(C)(C)C)sc1C 928,N1(C(c2c(N)c(F)cc(F)c2)=O)CCC2CN(C(c3ccnnc3)=O)CCC12 929,c1(C(N2C(CCNC(c3c(CC)scn3)=O)CSCC2)=O)cc(F)c(O)c(F)c1 930,c1(C(=O)NC2C(NC(CC(=O)NCC)=O)CCCC2)cc(Cl)c(OC)cc1C 931,N1(C(c2c(N)cc(C)cc2F)=O)CC(NC(c2cscn2)=O)CC12CCOCC2 932,Cc1nc(C(N2CCC(C)(NC(c3cc(C(C)(C)C)c[nH]3)=O)C2)=O)c(C)o1 933,CC(C)CC(CNC(C1CCCCC(=O)C1)=O)C(=O)NCc1nn(C)cc1CO 934,c1(C(N2C(CNC(C(C)(C)c3ccno3)=O)CCC2)=O)c[nH]c2ccncc12 935,c1(C(=O)NCC2(NC(c3ccc(C)c(C)c3)=O)CCC2)nnc2n1CCCCC2 936,c1(C(N2CC(F)(CNC(c3cncc(C#C)c3)=O)C2)=O)cc2cc(Cl)cnc2[nH]1 937,C(=O)(C1CCCc2n[nH]cc21)NCC1(CN(C(C(C(CC)(F)F)(C)C)=O)C)CC1 938,CC1(C)CC(c2nnnn2CC2CCOCC2)(NCCC2CCSC2)CS1 939,C(CCC(O)C(=O)N1CC=CC1C(=O)N(C)C)NC(CC(C)=C(C)C)=O 940,c1(N2C3CC(CN(C(c4ccc5ncnn5c4)=O)C3)C2)cccc(F)c1[N+](=O)[O-] 941,N1(C(CCc2ccc(C)o2)=O)C2CCC(C(=O)NCCCOCCO)C1CC2 942,c1(C(=O)NCC2N(C(c3n(C)cnc3)=O)C3CCC2C3)cc(F)c(F)c(C#N)c1 943,CC(C)C(C)CC(=O)NCCCOCCCNC(=O)C(c1cccc(F)c1)(C)C 944,N1(C(CC)=O)CC=CC(NC(=O)CC(c2ccccc2)NC(=O)OC(C)(C)C)C1 945,c1(C(=O)NC2CC(C)N(C(c3cc(Cl)on3)=O)CC2)cc(F)cc([N+](=O)[O-])c1 946,c1(CC)cc(F)ccc1C(=O)NC1CCN(C(C2CC(F)CN2C)=O)C1(C)C 947,C(=O)(C(C)CC(C)(C)C)N1CCC(NC(C(CCCC)O)=O)C1C 948,C1(NC(c2ccc(F)o2)=O)CN(C(C2CC2c2cccs2)=O)CCC12CCC2 949,c1(C(N(CC(CN(C(C(C)SC(F)(F)F)=O)C(F)F)(C)C)C)=O)nnn(C)c1C(F)F 950,c1(C(N2CC(C)N(C(c3cccc(C(F)F)c3)=O)CC2)=O)ncc(C#N)cc1Cl 951,c1(CC(N2CCN(C(C(CSC)O)=O)C(C)C2)=O)ccc(Cl)c2cccnc12 952,N1(C(COCCC)=O)CCC(N(C)C(c2ccc(C(C)(C)C)s2)=O)C(C)C1 953,c1(C(N(C)CC2CCCN(C(c3cnc(C(C)O)s3)=O)C2)=O)cc(Cl)nc(=N)[nH]1 954,C1(NC(=O)C(F)C2CC2)CN(C(c2ccc3sccc3c2)=O)CCC12CCC2 955,Cc1oc(C(C)C)nc1C(=O)N(C(C)CCNC(C1(S(C)(=O)=O)CC1)=O)C 956,C1(NC(c2nnc(O)cc2O)=O)CCN(C(=O)CNc2ncccn2)CC1F 957,CC(CC(=O)NC(CC1CCC1)C(=O)NCCCC1(O)CCC1)C1CC1 958,Cc1cc(N)c(C(N2CC(NC(c3ccc(CC4CC4)s3)=O)CC2C)=O)cc1C 959,Cc1cc(NCC2CCCCO2)ncc1S(=O)(=O)NC(C)(C)CCn1ccnc1 960,CC1(C)COC(C(N2CCN(C(c3cscn3)=O)CC2CC2CC2)=O)CO1 961,CCS(=O)(=O)CC(=O)NCC1CCCN(C(C2CC2c2ccccc2C#N)=O)C1 962,C1(CN(C(COCCOC)=O)C2CC2)CCCCN1C(=O)C(F)CC1CCC1 963,C1(C(N2CC(C(C)NC(CC(COC)C)=O)C2)=O)OCCN(C)C1=O 964,C1(CC(C)NC(C2(C(F)(F)F)CC(O)C2)=O)CCN(C(=O)Cc2cc[nH]n2)CC1 965,c1(-c2nn(CC(=C)C)c(C3CCCC(F)(F)C3)n2)cc(OC(F)(F)F)ccc1Cl 966,Cc1cc(Cl)c(C(N2CCCCC(NC(c3coc(Br)c3)=O)C2)=O)cn1 967,C1(NC(C(c2ccnn2C)C)=O)CN(C(=O)C(F)(F)c2cccnc2)CC1(C)C 968,N1(C(CN(C(=O)C=C(C)C(C)C)CC)=O)CC2(COCC(=O)N2)C1 969,CCS(=O)(=O)CC(C)N(C(c1ccc(F)cc1)C(=O)NCC(C)C)C 970,CC(CCCCNC(c1cnc(S)[nH]1)=O)NC(=O)CC(C)(O)C1CC1 971,C#Cc1ncc(N)nc1N1CCC(Cc2cccnc2)C1 972,c1(C(N2CC(C(C(=O)NC(CC#C)C(N)=O)O)C2)=O)c(C)ccnc1C 973,c1(C(=O)NCC23CC(CN2C(c2coc(Cl)c2)=O)C3)cc2cc(F)ccc2s1 974,c1(C(=O)NCC2C(NC(C3C(CC)C3)=O)C2)cnn(C)c1C(F)(F)F 975,C1(CNCCC2(C(NOC(C(=O)OCC)C)=O)CC2)COCCC1C 976,c1(C(=O)NC2CCC(NC(CCC(N)=O)=O)C2)cnn2cccc(Cl)c12 977,C(C1CCOCC1)=CC(N1CC(C(C(N2C(C(=O)NC)C=CC2)=O)O)C1)=O 978,C(C(C(=O)NCC1(CNC(=O)CSC)CCCC1)OC)OC 979,CCCCC(O)CC(=O)N1CCOCC(F)(CNC(c2cnc(SC)s2)=O)C1 980,c1(NCC(C)(C)C(F)F)ncnc2sc(Br)cc12 981,N1(C(C(C)C(F)(F)F)=O)CCC(C2(O)CN(C(=O)C=CS(C)=O)C2)CC1 982,CCC(C)C(CC(=O)NCC1CCCOCC1)NC(=O)COC(C)(C)C 983,c1(C(N(C)Cc2ncccc2F)=O)c(Br)ccc(F)c1F 984,C1(CC=C)COCC1NC(=O)CCN(C(=O)CCOC)CC 985,C1(Nc2ccc(C(=O)NC3CC3)cn2)CC2CCC(C1)N2C(=O)CC1OCCO1 986,c1(OCC)ccccc1C(N1CC(CO)(NC(c2cc(O)n(C)n2)=O)C1)=O 987,N1(C(C(CCN(C)C)NC(C(C(C)C)=O)=O)=O)CCC12CN(C)C2 988,C(=O)(CC(=O)NC1CC(F)(CNC(=O)C(c2ccc(Br)s2)C)C1)OC 989,C(CCCCC)(C(=O)NC1CN(C)C(=O)N1)NC(Cc1cn(COC)nc1)=O 990,N1(C(c2cc(CC)ncn2)=O)CC(C)N(C(=O)C(c2cccn2C)=O)CC1C 991,C1(CCC(C)(C)NC(C2CCC(C)(C)O2)=O)CCN(C(=O)CSC(F)F)CC1 992,C1(C(=O)NCC(NOCC)=O)CCCN(C(=O)CCC(=O)N(C)C(C)C)CC1 993,CC(C)C(C(=O)N(C(C)CNC(c1cncc(CO)c1)=O)C)N1CCCC1=O 994,C1(N(C(=O)C(C)(F)F)CC)CCCN(C(=O)C(O)c2ccsc2)C1 995,S(=O)(=O)(c1[nH]c(=NCc2cc(Br)no2)ccc1Br)NC(C)CCC1CCCCC1 996,C12(NC(c3c(C)nc(C)s3)=O)CCCC1N(C(=O)Cc1c(Cl)cccc1Cl)CC2 997,c1(NCCN(C)CC)nc(C)cc(=NCCCN2CCCCC2)[nH]1 998,C1(NC(Cc2n(C)ccn2)=O)CC2CCCC(C1)N2C(C12CC(C)(C1)C2)=O 999,CC(C(=O)N1CC(CS(C)=O)C1)N(C(=O)C(C)N(C)C)CCN(C)C 1000,c1(C(=O)NCC2(CNC(C3(C)CCC3)=O)CC2)ccncc1-c1ccccc1 1001,c1(C(C(=O)NC2CC2)N(C2CCCCC2)CC(C)(C)C)cccc(C(C)(C)C)n1 1002,C1(NC(c2ccc(OC)s2)=O)CCN(C(=O)Cn2ccnn2)CC1CO 1003,c1(C(C)C)ccc(N)c(C(=O)NC2CC(O)(CNC(=O)CC3CC3(Cl)Cl)C2)c1 1004,C1(OCC)(CNC(=O)C(C)CSc2ccccc2)CN(C(C2(O)CC2)=O)C1 1005,c1(CC)cc(N)c(C(=O)N(CCCCNC(c2sc(C)nc2C)=O)C)c(F)c1 1006,c1(OC)cccc(I)c1C(=O)NC1CC=CCC1C(F)(F)F.n12cc(nn1)C2 1007,CC(CC(=O)N1CC2CC2C1C(=O)Nc1ccc(Cl)cc1O)C(F)F 1008,N1(C(C(CCOC)C)=O)Cc2n[nH]cc2C1C(=O)NC(=O)C1=C(Cl)CC1 1009,C(C)(C1=CCN(C)CC1)NC(c1cc(CNC(C(C2CC2)OC)=O)ncc1)=O 1010,CC(C)CC(CC(C)C)C(=O)NC1(C2CN(C(C3(O)COC3)=O)C2)CC1 1011,C(=O)(CS(=O)(=O)CC(C)C)N1C2C(NC(CCC(=C)C)=O)(CCC2)CC1 1012,N1(C(CN2C(C)CC2)=O)CCCC2(C1)CN(C(c1ccc(F)c(Cl)c1)=O)C2 1013,N1(C(C2CCCC(NC(c3cc(C)sn3)=O)C2)=O)CC(F)(F)C(F)(F)C1 1014,C1(N(C)C(C23CC(C)(C2)C3)=O)CCCN(C(=O)CSCCC(F)(F)F)C1 1015,CCCCC(CNC(=O)COc1ccccc1Cl)NC(c1[nH]nnc1COC)=O 1016,c1(C(=O)NCC2C3CN(C(C4C5CCCC45)=O)CC23)cc(O)nc(O)n1 1017,c1(C(=O)NCC2(F)CC(NC(c3nccc(OC)c3)=O)C2)cc2sccc2cn1 1018,C1(NC(c2c(CC)ncnc2)=O)CC2CC(C1)CN(C(c1coc(SC)c1)=O)C2 1019,C(=O)(CCC(=O)NC(CNC(c1occ(C)c1C)=O)C1CC1)N(CCC)CCC 1020,c1(C(N(CCNC(C(CC)NC(N)=O)=O)CC2CC2)=O)ccc2c(cnn2C)c1 1021,c1(OC)ccnc(C(=O)NC(C)CNC(c2ncn(C(C)(C)C)n2)=O)c1O 1022,CCCC(C(=O)N(C1CCN(C(=O)C(C)NC(=O)NC(C)=O)C1)C)OC(C)(C)C 1023,c1(CC)nc(C(C)C)ccc1NC(c1ccc(C[SH](C(C)C)CC)cc1)=O 1024,N1(C(CCCOC)=O)CC(CNC(C23C4CC(CC24)C3(F)F)=O)OC2(CCC2)C1 1025,CCCCCCCC(O)CC(=O)NCc1ccc(-c2cccc(OC)c2C)cn1 1026,c1(C(=O)NC(C)CN(C)C(c2cc(Cl)ccc2N)=O)cnc2[nH]cncc1-2 1027,N(C1c2ccccc2C2CCC1C2)C(=O)NC(CC)CCOC 1028,C(=O)(C(C(C)(C)C)NC(N)=O)N1CCC(NC(C2OCCN(CC)C2)=O)C1 1029,C1(NC(c2ccn(CC(C)C)n2)=O)CC2(C1)CC(NC(c1c[nH]ccc1=O)=O)C2 1030,CCCCC(C(=O)N(C1CC2CCC1O2)C)NC(=O)C(CCC)OCC 1031,S(=O)(=O)(c1sc2ccc(C#N)cc2c1C)NC(C)CC1CCOC1 1032,C1(CCO)(CN(CCC)CC2COCCN2)CCOCC1 1033,C#CC1(O)CCN(C(=O)COC2(C)CN(C(=O)C(C)(C)n3cncn3)C2)C1 1034,CC1CCCN(C(=O)C(=O)NCC2CCN(C(C3CC3OC(C)(C)C)=O)C2)C1 1035,CC1(C)CC(C(N2CCCCC2CCO)=O)CCN1C(C1CC=CC1)=O 1036,c1(CC)ccc(F)cc1C(=O)NC1CCCCN(C(=O)C(C(C)CC)N(C)C)C1 1037,c1(OC)ccc2c(c1)CN(Cc1cc(F)ccc1C(F)(F)F)C2 1038,Cc1nc(C)c(CCC(=O)N(CC(C)CNC(C2OCCC2C)=O)C)c(O)n1 1039,C(=O)(C(C)CCC(C)(C)C)NC(CNC(Cc1c(C)nsc1)=O)C(C)C 1040,S(=O)(=O)(c1cc(Br)ccc1Cl)N1C2CC(C(=O)Nc3ccnc(F)c3)C1CC2 1041,c1(C(=O)NC2CCC(NC(=O)CCCCC3CC3)C2)cc2cccc(F)c2o1 1042,Cc1cc(O)ccc1CC(N1CCOC(CCNC(C2CCSC2)=O)C1)=O 1043,C1(C(=O)NCC(C(=O)N(CC(F)F)C(C)C)C)CCCC(C#N)C1 1044,C1(NC(CC)=O)CCCC12CCN(C(C1CCCC1C(F)F)=O)CC2 1045,C1(OCC)CN(C(=O)C(C2CCC2)OC)CC1CNC(=O)CCOC 1046,C1(CC)CN(C(C2C=CC=CC=C2)=O)CCC1NC(c1cncc(C)c1)=O 1047,CC(C)(C)C1CCNc2c(C(N3CCCCC3CC3CCCCC3)=O)cnn21 1048,c1(C(=O)NCCCCN(CC)CC)nn2c(c1-c1cc(F)nc(F)c1)CCCC2 1049,C(=O)(C(O)(C(F)(F)F)C1CC1)NCCC(C)N(C(CCC#C)=O)C 1050,c1(NC(C(c2cnc(CC)s2)N(CCC(C)(C)C)CCOC)=O)ccccc1Cl 1051,C(=O)(CCCCCN=[N+]=[N-])NC(CC=CC)C(=O)NCC1CCCC(CO)C1 1052,C1(NC(c2cc(C)sn2)=O)CCN(C(c2cccc(OC3CC3)c2)=O)CC1O 1053,c1(C(CC)C)ccc(C(N2CC(NC(C3CCC(=O)O3)=O)C(C)C2)=O)cc1 1054,C(=O)(CCCCCN(C(=O)CN(C)C)C)N(CCCSCCC)C 1055,c1(OC)ccc(C(=O)NCC2CC2CNC(c2ccco2)=O)cc1C 1056,C1(C)(C(=O)NCC2CC(NC(C3CCCC(OC)C3)=O)C2)CCN(C)C1=O 1057,C=CC(C(=O)NCCCNC(=O)Cc1cnc(C2CC2)[nH]1)c1ccccc1 1058,C1(CC)CN(C(=O)CN(C2CCS(=O)(=O)C2)C)CCN1C(=O)CCn1ccnn1 1059,CC1CCCc2cc(C(=O)NCC(O)CN(C(=O)C=CBr)C)nn21 1060,C(=O)(C(O)CCCCC)N(c1n[nH]c2c1CCCC2)CC(=C)C 1061,C1(CNC(Cc2nc(C)c(C)[nH]2)=O)COCCN(C(c2ccnc(CO)c2)=O)C1 1062,CON1CCC(CC(=O)NCC2(F)CCN(C(c3nccc(Cl)c3F)=O)C2)CC1 1063,C12CCCN(CC1)C2.c1(CC)ccccc1NCc1cn[nH]c1 1064,Cc1cc(C)n(C(C)C(=O)NC2(C)CCN(C(=O)CCc3cc[nH]n3)C2)n1 1065,c1(C(N(CCC(C)NC(c2cc(C(C)(C)C)on2)=O)C)=O)cnn(C)c1F 1066,C1(CNC(c2cccs2)=O)CCC2CN(C(c3ncn4ccccc34)=O)CC12 1067,Cc1ccc(=O)n(CC(=O)N(C2CCN(C(c3cc(O)ccc3C)=O)C2)C)n1 1068,c1(C(=O)NC(c2ccnn2C)C(=O)N(C)Cc2c(C)cco2)nn(C)cc1Cl 1069,c1(C(=O)NC2C(CNC(C3CCN(CCC#C)CC3)=O)CC2)cc(C)c(F)cn1 1070,C(=O)(C(C(C)C)NC(c1cccc(CNC(=O)Cc2cc(C)[nH]n2)n1)=O)OC 1071,Cc1ccn(CCC(=O)NC(C)(CNC(=O)CC2COCC2O)C2CCC2)n1 1072,c1(C(=O)NCC(CC)NC(c2cnc(O)c(Cl)c2)=O)c(C)[nH]c2ncccc12 1073,C#Cc1cccc(CNC2CC2C(=O)NC(CO)C(C)C)c1 1074,N1(C(c2cccc(C#C)n2)C(=O)Nc2ccccc2)CCOC2CS(=O)(=O)CC12 1075,Cc1ccnc(C(=O)NC(C)CN(C(=O)COCC2CCCOC2)C)n1 1076,CCC(C#N)C(=O)N(C(C(N1CC(O)(c2nn[nH]n2)C1)=O)C1CC1)C 1077,CN=C(NCCCNC(C1CCCO1)=O)NC(C1(CNS(C)(=O)=O)CC1)C 1078,N1(C(C2(C)CCOC2)=O)CCC2(CC1)Cc1ccccc1C2 1079,C1(O)(CNC(C(C)CC2CCCC2)=O)CCN(C(C2CC3CC23)=O)CC1 1080,c1(N2CC(=C(CNC(c3cnccn3)=O)F)C2)cc(-n2ccnc2)ncn1 1081,C1(NC(c2nn(CC)c(C3CC3)c2)=O)CCCN(C(c2nnc(S)n2C)=O)C1C 1082,c1(OCC)ccc(C)nc1C(N1CCCC(NC(C2CCCN2C(C)C)=O)C1)=O 1083,c1(CNC(c2ccco2)C)ccccc1CNCc1ccc(OC(F)F)cc1.COCO 1084,c1(CC)ccncc1NC(=O)C(c1cnn(C)c1)NC(=O)CC1CC(C)C1 1085,N1(C(C(C)OCCOC)=O)CCC(C)(NC(c2cc(Br)sn2)=O)C1 1086,c1(NC)ccc(C(=O)NCC(C2CC2)NC(c2ncc(F)cn2)=O)c(Cl)c1 1087,Cc1cc(C(=O)NC(C2CCN(C(=O)C(C)(C)OCC(F)(F)F)C2)C)cc(Cl)c1 1088,CCC(CC)(CCNC(C1(CCF)CC1)=O)NC(C1CCC(C(N)=O)C1)=O 1089,CCC(C)C(=O)N1CC(C(=O)NCCS(=O)(=O)NC(=O)OC(C)(C)C)(OC)C1 1090,C#CCCCCCCCC(=O)NC(CCN(C(=O)C(C)NC=O)C)C(C)(C)C 1091,c1(N(CCN(C)C(C2CCCN(C)C2=O)=O)C)cc(F)ccc1F 1092,c1(OCC)ccc2nnc(CCC(=O)NCc3cc(F)ccc3O)n2n1 1093,Cc1ccc(C)n1CCC(=O)NCC(C1CC1)N(C)C(C1CC(F)C1)=O 1094,CC1CC(=O)NC1C(N1CC(CNC(=O)CCc2cccc(Cl)c2)C1)=O 1095,C(C)(C(=O)N(CC(C)(C)NC(=O)CC(C)C1CC1)C)(C1CCCCC1)OC 1096,O(NC(=O)CCCNC(=O)C(c1cncn1C)O)C1CCCN(CC)C1 1097,c1(CCN2CCCC(CCNC(C3C=CCC3)=O)C2)c(F)cccc1Cl 1098,C1(O)(CCNC(C(C=C)O)=O)CCN(C(c2cc(C(F)(F)F)cc(F)c2)=O)CC1 1099,C1(C(=O)NCCCC2N(C(Cn3c(C)csc3=O)=O)CCC2)Cc2nccn2C1 1100,C1(c2n(CC=C)nnn2)(N(c2cccc(I)c2)CC)CCC(CCCC)CC1 1101,C(=O)(C(F)CC(C)(C)NC(C1CCCC2(CC2)C1)=O)N(CC#C)CC 1102,N1(CC(=O)NC2(C)CN(C(C(c3ccccc3Cl)C)=O)C2)CCc2ccccc21 1103,c1(C(C)C)cccc(C(=O)NCCCC2CCN(C(=O)C(C)C(C)O)CC2)c1F 1104,C1(NC(=O)CC2CCCCC23CC3)CN(C(=O)CN2CCCC2)CC2(CC2)C1 1105,c1(CC(=O)NCC2(C(=O)NCC3CCCNC3=O)CC(=C)C2)cccc(C)n1 1106,c1(OCC#C)cccc(-c2nnc(N3CCC(C)(C)C3)n2CC(C)C)c1 1107,CN1CCN(CC(=O)N(C2CC(NC(C3CC(C)(C)CO3)=O)C2)C)CC1 1108,N1(c2cc(C)nc(C)n2)CCC(F)(F)C(CNC(c2c[nH]nc2C2CCC2)=O)C1 1109,c1(C(C)CN(C)C)nc(-c2ccc(F)cc2)nn1C1CCS(=O)(=O)C1 1110,n1(CC)cnc2nc(N3Cc4cccnc4C3)nc(NCC(C)(C)C(C)C)c12 1111,c1(N(C2CCNC2)C(c2c(C)ccc(Br)c2C)=O)ncc2c(ccn2C)n1 1112,C1(CC)(NC(c2cnn(CCOC)c2C)=O)CCCN(C(c2cc(C)ns2)=O)C1 1113,N1(C(C=CSC)=O)CC2CCCCC2(CNC(c2cccc([N+](=O)[O-])c2N)=O)C1 1114,N1(C(C2CC(CC)C2)=O)CCCC(NC(=O)C(Cc2cccc(F)c2)NC=O)C1 1115,C(C1CCOCC1)=CC(=O)NCCC(C)NC(=O)C=Cc1ncc[nH]1 1116,C1(C(=O)NC2C(NC(c3ccnn3CCC(F)(F)F)=O)C2)CCCCCC1 1117,C(C)(CCC(=O)NCC1CCCN1C(=O)COc1ccc(C(C)=O)cc1)OC 1118,c1(C(=O)NCC2CCCN(C(C=CCOC)=O)C2)noc2c1CN(C(C)C)CC2 1119,c1(C(C(=O)NC2CCOC2)N(CCC)CCN(C)CC)cnc(Br)n1C 1120,c1(N(CCCCNC(C2C=CCCC2)=O)Cc2ccccc2)cc([N+](=O)[O-])n[nH]1 1121,c1(OC)cc(C(=O)NC2CN(C(=O)C(C)(O)c3ccccc3)CC2O)cc(F)n1 1122,C=CC1(C2(C(=O)NCCN(CCCC)C=O)CCC2)CCC1.C(=O)(CCC)NC 1123,CN1CCC(C(=O)NC(C(=O)N(C)CC2CCC2)c2cccs2)CC1=O 1124,c1(C(CC)=O)ccc(C(N2CCC2C(=O)N(c2cccs2)CC)=O)cc1 1125,C1(CNC(C(N2CCC(C)C2)=O)=O)CCCCN(C(c2cc(O)ccc2F)=O)C1 1126,c1(C(=O)NCC2CC(NC(CN(C3CC3)CC)=O)C2)cc(C)cnn1 1127,C1(Nc2cc(OCC)ncn2)CN(C(=O)CC2CCC(=O)N2)CCC1CO 1128,c1(C(c2nnnn2C2CCCC2)NC2CCC(CCCC)C2)cncc(CC)c1 1129,CC1CN(C(c2ccn(Cc3ccccc3)n2)=O)C(C)CN1C(=O)CCC(F)F 1130,c1(C(N(CCOC)CCNC(C2SCCC2C)=O)=O)ccc2oncc2c1 1131,c1(C(N2CC3CC(C2)N(C(=O)C2=CCCSC2)C3)=O)cc2nc[nH]c2cc1F 1132,N1(C(c2cn(C)nc2)=O)CCC(NC(c2cc3cccn3cn2)=O)C(F)(F)CC1 1133,CN1C(=O)OC2CN(C(c3csc(CNC(C4(C)C=CCCC4)=O)c3)=O)CC12 1134,CCC(CNC(c1ncn(C)n1)=O)(CC)C(=O)NC(c1ccccc1F)C 1135,C(=O)(CC1=CCCC1)N1CCC(C(C)NC(C#CC(C)C)=O)C1 1136,N1(C(C2C(C(=O)OC)CCO2)=O)CCN(C(=O)C=CCCC=C(C)C)C(CO)C1 1137,C1(CCNC(c2nc(OCC)oc2)=O)CCCN(C(=O)C(C)n2cccc2)C1 1138,C1(OC(N2CC(CCNC(CC)=O)C2)=O)CCCCC1CC 1139,c1(C(N2CC(CNC(=O)CC3CCCO3)C3(C2)CC3)=O)cc2ccc(F)cc2s1 1140,CCCCC(CC)C(=O)N1CCCC1C(C)(C)C(N1CCSC2(CCC2)C1)=O 1141,Cc1cnc(C(=O)NCC(CO)NC(c2cc(F)cc(F)c2)=O)c(C)c1 1142,N1(C(C2C(C)OC(=O)N2)=O)CCC(CNC(=O)CNS(N)(=O)=O)C(O)C1 1143,C12(CNC(C(CC)COC)=O)CCC(CN(C(=O)C(=Cc3cnn(C)c3)C)C1)C2 1144,c1(NC(CN(C)C)=O)ccc(C#N)c(C(F)(F)F)c1.C12CC(O)CN(C1)C2=O 1145,C1(C)(NC2CN(C3CN(C(C(=O)N(C)CC)=O)C3)C(=O)C2)CCCC(F)(F)C1 1146,Cc1ccc(CCCCC(=O)NC(CNC(c2cc(C)ncn2)=O)CO)cc1 1147,C1(CNC(C(COC)C)=O)COC(C)(C)CN1C(=O)CC1(N(C)C)CC1 1148,c1(OC)ccc(C)c(C(=O)NCCC2CC(NC(c3ccc([N+](=O)[O-])s3)=O)C2)n1 1149,CC1(CNC(C2C(F)(F)C23CCC3)=O)CCN(C(C2C3CCCC23)=O)CC1 1150,C12(C(=O)NCC3N(C(c4c(Cl)ccc(CC)c4)=O)CC3)CCCCC1NC(=O)C2 1151,c1(CSC)cc(C(=O)NC(CCNC(=O)Cc2cncn2C)C(C)C)ccc1F 1152,C1(C(=O)NC2(C)CCN(C(c3cc(C(C)(C)C)ncc3)=O)C2)CCOCC1(C)C 1153,C12(CNC(COCC(=O)NC)=O)CC1CN(C(=O)CNC(=O)CC(C)(C)C)C2 1154,Cc1cc(=NC(C)c2cccnc2O)[nH]c(=NCC2CCCc3scc(C)c32)[nH]1 1155,Cc1cnc(F)c(CNC(=O)CC(C(F)F)NC(C23CSCC2C3)=O)c1 1156,Cc1cc(OCC(=O)NCC(F)CNC(c2ccc(C3CC3)cn2)=O)cc(C)c1 1157,c1(C(=O)NCC2CCN(C(=O)C(O)CN3CCOCC3)C2)ccc(F)cc1F 1158,CC1CCC(NC(C2CC3CCC3C2)=O)CN1C(C1CCCCO1)=O 1159,c1(C(N2C(CNC(c3c(C)onc3Br)=O)CCC2)=O)ccc(C)n(C)c1=O 1160,C(=O)(C(F)(F)C(F)(F)F)NCC1N(C(C2CC(C)(C)C2C(F)(F)F)=O)CCC1 1161,CCCC(C(=O)N(CC(CC)NC(c1[nH]nnc1C)=O)CC)NC(C)=O 1162,Cc1nn(C)c(C)c1C(=O)OCC1(NCc2ccc(-c3nn[nH]n3)cc2)CC1 1163,C1(C(=O)NCc2cccc(NC(C(C)(C)F)=O)c2)CCn2cncc2C1 1164,O=C1NCCCC12CCCN(c1cc(NCCCCN3CCCCC3)ncn1)C2 1165,c1(CNC2CC(NC(c3nccnc3Cl)=O)C2)ccccc1N1CCOCC1 1166,N1(CC)CCC1C(=O)NC1CC(C(C)NC(=O)Cc2ccco2)C1 1167,c1(NC(C2(CNC(COC(CC)(C)C)=O)CC2)=O)c(SC)noc1C 1168,c1(C(N2CCN(C(CCC3CCC(C)O3)=O)CC2CO)=O)ccc2cncn2c1 1169,O=C(CCCCCCNC(c1c[nH]c2ccccc12)=O)NC1CC(O)C12CCC2 1170,C1(NC(C(C)C2CCOC2)=O)CCN(C(=O)COc2ccc(Cl)cc2)C12CCC2 1171,N1(C(CSCCOC)=O)CCCN(C(C2(NC(C)=O)CCCOC2)=O)C(C)C1 1172,c1(CCNC(CCN(c2ccncc2)C)=O)cn(CCc2ccccn2)nn1 1173,CC1CCOCC1C(=O)NCC1CCC(C(=O)NCCn2ccc(=O)cc2)O1 1174,C1(NC(C(C)NC(C)=O)=O)CC2CC1CN2C(c1cncc(Cl)c1)=O 1175,n1(CC)nc(C(=O)NC(C2CCN(C(=O)C(C)CCOC)C2)(C)C)c(C)n1 1176,C(CC(C(C)C)NC(c1ccn(C)c1C1CCC1)=O)N(C(C=C(C)C1CC1)=O)C 1177,c1(C(=O)NCC2(CNC(CC)=O)CC23CCC3)ccc2nc(O)n(C3CC3)c2c1 1178,c1(NC(c2cnc(-c3ccc(F)c(O)c3)cn2)=O)cc(Cl)cc(Cl)c1O 1179,C(=O)(C(Cn1ccnn1)NC(c1cc(Cl)no1)=O)NCC(C)N(CC)CC 1180,C1(C)(C(N(CC(CC)NC(=O)CCc2nnc(C)n2C)CC)=O)CCC(=O)N1 1181,C1(CC(=O)NCC2CN(C(c3c(C)nnn3C)=O)CC2O)CCC(C)(C)CC1 1182,c1(OC)cccc2[nH]c(C(=O)NCCN(C(C34CSC(C3)C4)=O)CC3CC3)cc12 1183,N1(C(C(c2scc(C)n2)C)=O)CCC(NC(=O)CC(C)(F)F)C12CC2 1184,C(N=c1nc2c(F)c[nH]c2c(N2CCCC(F)C2)[nH]1)C1(OC)CCOCC1 1185,c1(C(N2C(CC)CN(C(c3ns[nH]c3=O)=O)CC2)=O)cccc2cncn12 1186,c1(CC(N(Cc2cn(-c3ccc(N(C)C)cc3)nc2)O)=O)cc(F)c(F)cc1F 1187,CCCC(C(=O)N(C)CC1(O)CCN(C(=O)CCN2CCCC2)C1)OCC 1188,N1(C(C(C)SC)=O)CCN(C(C2CCS(=O)(=O)CC2)=O)C(CC(C)(C)C)C1 1189,c1(C(=O)NCC2(CNC(C(C3CC3)OC)=O)CCC2)cncc2nc(C)[nH]c12 1190,c1(OC)cccc2c(C(=O)NC3CN(C(c4cncc5sccc45)=O)C3)n[nH]c12 1191,c1(C(=O)NCC(CC=C)NC(=O)CNC=O)ccc(=O)n(C)c1 1192,CC1=C(C(=O)N2CCC(C(C)CNC(=O)C(O)(C3CC3)C3CC3)CC2)SCCO1 1193,c1(C(N2C(CNC(CCCC)=O)C(C)CC2)=O)cc(Br)c([N+](=O)[O-])[nH]1 1194,C(CCC(C)C(=O)NC(C)CC1CN(C(C2(C(=O)OC)CC2)=O)C1)OC 1195,Cc1nnccc1C(=O)N(CC(C)O)CCNC(=O)CC1(O)CCC1 1196,c1(CN(C)C(c2ccc(Cl)s2)=O)ccccc1CNC(C1CC2CC1C2)=O 1197,C1(CNC(c2ccn(CCF)n2)=O)CC(C(=O)N2CCC(CCCO)C2)=NO1 1198,C#Cc1ccccc1CC(=O)NCCCN(C(=O)CC(C)OC)C 1199,CN1C(CNC(=O)N(CC(c2cccs2)O)C2CC2)CCS1(=O)=O 1200,S(=O)(=O)(c1cccc(Br)c1F)N1CC2CCN(C(C(C)OC)=O)C2CC1 1201,C12(NC(C(C)OCOC)=O)CC(C(N3CCC3N3CCNC3=O)=O)(C1)C2 1202,Cc1ncc(Br)c(NC2CN(C(c3ccccc3I)=O)CCC2F)n1 1203,c1(C(C)(C)C)cc(NC(=O)C(=O)NC2CCC(Cc3ccccc3)C2)cc(O)c1 1204,C(=O)(CCCC(C)(C)NC(c1cc[nH]c1)=O)N(C)Cc1c(C)ncs1 1205,N1(c2cc(NCc3c(OC4CC4)ccc(F)c3)ncn2)CCSC2(CCOCC2)C1 1206,c1(C(=O)OCCCCCC2(C)OCCO2)c[nH]c2cnccc12 1207,CC(CC(F)(F)F)C(=O)N1CCN(C(=O)COc2cccc(Cl)c2)CC1CO 1208,C1(NC(c2cc(CC)ncn2)=O)CN(C(=O)Cc2csc(Cl)c2)C2(CCOC2)C1 1209,C(C(C)(O)CC(=O)NC(CCF)C(=O)N(C)Cc1ncnn1C)OC 1210,C1(NC(CCC2CCC(NC(C3=NOC(C)C3)=O)C2)=O)CC(C)CC(C)(C)C1 1211,N1(C(NNC(c2c(C)n(C)nc2)=O)=O)CC2CC3CC1C2O3 1212,C(=O)(CCCCC(=O)NC(CC)CC(=O)OC)NC(C)COC 1213,c1(CC(C)C)ccc(C(=O)NC(CNC(c2ccncc2N)=O)C(C)(C)C)cc1 1214,C12(NC(C=C(C)C)=O)CCCC1N(C(C1CN(C)CCN(C)C1)=O)CCC2 1215,CCC(CC)CC(F)C(=O)NC1(C)CCCCC1C(=O)N(CC1CC1)CC1CC1 1216,c1(C(=O)NCC(CC=C)NC(C2CC(=O)NC2(C)C)=O)ccc(P(C)(C)=O)o1 1217,N1(C(CCNC(C)=O)=O)CCC(C2CCCN(C(=O)C(F)=C3CCC3)C2)C1 1218,C1(F)(NCCC(=O)NC(C2CCCCC2)C)CC(C(=O)O)C1 1219,C1(NC(C(C)SC(C)C)=O)CN(C(c2cnc3sccn23)=O)CC12CCC2 1220,c1(NC(c2sccc2NC(C2CCCO2)=O)=O)ccc(OC(F)F)cn1 1221,c1(C(N2CC(C#C)(C(=O)NCCc3cocn3)C2)=O)cc2cccnc2[nH]1 1222,C(=O)(CC(C(F)(F)F)OC)NCC1N(C(C(=O)OCC)=O)CC1 1223,C1(NC(CSCC=C)=O)CC2(CCC(NC(c3c(F)ccc(F)c3O)=O)CC2)C1 1224,N(C(=NCCC(C)=O)NCc1cccc(C(F)(F)F)n1)C(CC)CO 1225,CC1CC2CN(C(c3ncn(C)n3)=O)CC2N1C(c1ccnc(C2CCC2)c1)=O 1226,c1(C(C)C)nnc2n1CC(CN1CCN(C)CC1c1ccccc1)CC2 1227,CC1CN(C(=O)CN(C(=O)C=CC(C)(C)C)C2CCC2)Cc2nncn21 1228,CCCCN=C(NCC1COC(=O)O1)NCC(c1ccc(F)c(F)c1)C 1229,C1(NC(=O)CC2CC2(Cl)Cl)CCN(C(C2(c3ccno3)CC2)=O)C1 1230,c1(-c2ccc(C)c(C)c2)ccc2sc(C(N3C(CO)CCC3C)=O)cc2c1 1231,C1(O)(C(C)NC(C(COC)OC)=O)CCN(C(=O)Cc2cc(C)cs2)CC1 1232,c1(OCC)ccc(CN2CC3CN(C(c4ncsc4Br)=O)CC23)cc1OCC 1233,c1(CC(=O)NC2CN(C(c3c(C)ccs3)=O)CC2C)c[nH]c2c(F)cccc12 1234,C1(N(C(c2ccc(Br)c(F)c2)CC)C=O)CC2CCC(C1)S2 1235,C1(NC(C=NOC)=O)CCCC(CNC(c2cc(Br)c(Cl)s2)=O)C1 1236,C1(C(N(CCCC#C)C)=O)(C(C)C)CCN(C(C2(COC)CC(=O)C2)=O)C1 1237,c1(C(N2C(CC(N3C(C)(CCC)CC3)=O)CCC2)=O)ccc(C#N)s1 1238,N1(C(C2CC(NC(Cc3n(C)ccc3)=O)C(O)C2)=O)CC2(C1)CC2(F)F 1239,N1(C(C(CCC)(C)CC)=O)CCC2(C=C(C(=O)NC(C)CCO)C2)C1 1240,c1(C(=O)NCC(C(=O)N2CCCC2C(C)O)OC)cc(C)n(C)c1C 1241,c1(C(=O)NCCC2N(C(C(CCC)C#N)=O)CCC2)[nH]c2ccccc2c1OC 1242,C(=O)(CCC(F)(F)C(=O)NCC1CCN1C(C12CC(CN1C1CC1)C2)=O)OCC 1243,C(=O)(CC(CC)C(C)C)NCc1ccc(CNC(c2cncc(C#C)c2)=O)cc1 1244,c1(C(=O)NC2C(CNC(C(C)C(F)(F)F)=O)CC2)ccc2nncn2c1 1245,c1(OC)ccc2c(N(C3CC(N)C3)Cc3ccc(O)cc3C)ncnc2c1 1246,C1(CC=C)(C(N2CCC(O)(CO)C2)=O)CCN(C(=O)C(C(C)OC)N(C)C)C1 1247,N1(C(=O)NC2(C3N(C(CC4C(=O)NC(=N)S4)=O)CCC3)CC2)CCC(=O)NC1=O 1248,c1(CC)ccnc(C(=O)NCC(CC(=O)N2CCC(O)C2)C2CCC2)c1 1249,c1(CC(=O)NC(CCCNC(c2c(CC)cco2)=O)C)cnc(O)nc1O 1250,C12(NC(COCC)=O)CCC(CC1)N(C(=O)CCc1nc(C)cs1)C2 1251,CC(C(=O)NNC(=O)Cn1cc(C(N)=O)nn1)NC(N1CCc2sccc2C1)=O 1252,CN(C(=NCCC(=O)N1CCCC1)NCc1cccs1)CC1(C(F)(F)F)CCC1 1253,c1(CCC(c2nnnn2C)NCC2(OC)CC2)ccccc1F 1254,c1(CN2CC(C(=O)Nc3ccc(C)cc3Cl)SCC2)ncc(Br)cc1[N+](=O)[O-] 1255,C1(C(c2n(C)nnn2)Nc2ccc(Cl)cc2)CCC2(CC1)OCCCO2 1256,C1(CNC(C(C(=C)C)(C)C)=O)CC2(CO1)CN(C(c1ncc(C)cc1F)=O)C2 1257,Cc1cc(Br)cc(C)c1C(=O)OCC(N1CCCC(C(C)(C)O)C1)=O 1258,CCC(CC(=O)N1CCN(C(C2CCCN2C)=O)C(CO)C1)C(=O)OC(C)(C)C 1259,N1(C(C(CC)C(C)O)=O)CC2CCC1C(CN=c1ncc(OC3CCC3)c[nH]1)C2 1260,c1(N2C(CCNC(C(C(COC)C)C)=O)CSCC2)ccc([N+](=O)[O-])cc1 1261,c1(N(C)CC2CCN(C)CC2)nc(N2CCOC(C)(C)C2)nc2c1COCC2 1262,Cc1cc(=O)oc(C)c1C(N1CCN(C(C23CCC(F)C2CC3)=O)C(CO)C1)=O 1263,C1(COCC)CCCN(C(C2(C(C)NC(c3[nH]cnc3C)=O)CC2)=O)C1 1264,C(=O)(C1=C(C)N2CCN=C2S1)N1CCC(O)(C=O)CC1.N(CCO)(CC)CC 1265,c1(C(=O)NC(C2CCN(C(C3CC=CC3)=O)C2)C)cc(F)c(F)cc1N 1266,c1(N(C2CN(C(C(C=C)c3ccccc3)=O)C2)C)nc(C)ncc1F 1267,c1(-c2ncn(C)n2)ccc(C(N2CC(O)CC2CNC(C2CC2CF)=O)=O)cc1 1268,N1(C(C=CCC)=O)CCC(C)C(CNC(c2cc(C(=O)OC)oc2C)=O)C1 1269,S(=O)(=O)(c1ccc(N(C2(N)CC2)C)o1)OC.C(=O)(CCC1CCC1)NCC1CC1C(O)COC 1270,c1(CCC)cc(C(=O)N(C2CCCC(NC(c3cnc(O)n3C)=O)C2)C)sc1C 1271,c1(CC(C)C)cc(C(N2CC(F)(CNC(=O)CC3CC(O)C3)C2)=O)n[nH]1 1272,C(=O)(CC1OCCc2ccsc21)NCCOCCN(C(=O)C(C#N)=CC1CC1)C 1273,c1(C(=O)NCC2N(C(C(n3c(C)ccn3)C)=O)CCC2)cnc(Cl)c(F)c1N 1274,Cc1cc(NC(=O)CC2CC(C)N(C(C3COCCC3C)=O)C2)cc(C)c1F 1275,N1(C(c2sc(NC)c(C)c2)=O)CCC2CCN(C(c3cc(=O)cc[nH]3)=O)C2C1 1276,C=C(C)CC(C(=O)NCc1cnn(CCO)c1)NC(C1CCCN1C=O)=O 1277,N1(C(c2cc(C(=O)OC)oc2C)=O)CC2CN(C(C3COCCN3C)=O)CC2C1 1278,N1(C(c2c(CSC)cccn2)=O)CC2CC(NC(=O)Cn3cc[n+](C)c3)CC2C1 1279,C1(NC(c2c(C)sc(O)n2)=O)CCN(C(=O)C(c2ccccc2Cl)O)CC1C 1280,Cc1ccc(C)c(C(=O)NCCCC(=O)NC2CCN(C(C)C)C2)c1 1281,C1(F)(C(=O)NC(c2c(C)ncs2)C)CCN(C(c2ccc(C#N)[nH]2)=O)C1 1282,c1(C(N2CCN(C(C=CCN(C)CC)=O)C(C)C2)=O)cn2c(C)cccc2n1 1283,c1(C(c2n(CCCC)nnn2)NCCc2ncnn2C)cccc(CC)c1F 1284,C1(CNC(C2N(CC#C)CCC2)=O)CC(F)(F)CN1C(C1CN(C)CCO1)=O 1285,N1(C(c2c(CNC(c3c(=N)[nH]cnc3)=O)c[nH]n2)=O)CCCNC(=O)C12CC2 1286,N1(CCC)CC(C(N2CCCC2CN(C)C(C2CCC(=O)N2)=O)=O)CC1=O 1287,CC#CCC(C(=O)NCCC(O)C1CCC1)NC(c1ccccc1OC)=O 1288,c1(C(=O)Nc2cccc(I)n2)cc2ncc(-c3ccc(F)c4ccoc34)cc2[nH]1 1289,C1(CC=C)(NC(c2sc(C3CC3)nc2C)=O)CCCN(C(=O)C(C)COC)C1 1290,N1(C(c2n(CCC)ncc2)=O)CCN(C)C(CNC(=O)Cc2csc(Cl)c2)C1 1291,c1(C(=O)Nc2cccc(CO)c2F)ncn2cc(-c3ccco3)sc12 1292,c1(OC)ncc(C)cc1NC(=O)C(CN(C)C)NC(=O)CCCC1CCCO1 1293,Cc1c(F)ccc(C(=O)NC2CC3CC(NC(=O)C(C)C(C)C)CC23)c1C#N 1294,C(=O)(C(CC(C)C)NC(=O)CC(C)(C)O)OCC#C 1295,N1(C(C=C(CC)C)=O)CCN(C(=O)Cc2cc(C)[nH]n2)CC1C1CCCC1 1296,CCC(CC(=O)N1CC(C(=O)N(CCCC(C)C)C)C(CC)C1)C1CCC1 1297,c1(C(=O)OCC)cnc(N2CC(NC(=O)CN=S(C)(C)=O)CC2C)nc1C 1298,C(=O)(CCC(F)(F)C(F)F)N(CC(C)O)CCNC(C1CC1c1nc[nH]n1)=O 1299,C1(C)(C(N(CCCNC(=O)CC(=O)Nc2nccs2)C)=O)CS(=O)(=O)C1 1300,Cc1ccc(C)c(C(N2CCN(C(C3CN(C)CCO3)=O)CC2C)=O)c1 1301,C1(NC(C(C)(C)OC(C)C)=O)CN(C(=O)CC2CCCC2)C2(CCOC2)C1 1302,N1(Cc2n(C)c(Cl)nc2)C2CCC1CN(C(C1CCC(O)CC1)=O)C2 1303,Cc1c(C(=O)NC2CN(C(C3CCC3(C)C)=O)CC2C)ccn1C(C)C 1304,C(CCSC)(C(=O)NC(C)(C)CCN(C(=O)CC12CCC(CC1)C2)C)OC 1305,N1(C(C(CC2CCCC2)NC(=O)CC(C2CC2)C2CC2)=O)CCC(CO)C(O)C1 1306,c1(C(N2CCC(N(C(=O)CCN(C)CCOC)CCC)C2)=O)cnc(O)n1C 1307,C1(C(N2C(C#C)CC2)=O)CN(C(c2occc2COC)=O)CC12CCC2 1308,c1(C(=O)NC23CCC(CNC(=O)C4=CCCC4)(OC2)C3)cccc2ccsc12 1309,N1(C(CCc2scc(C)n2)=O)CCN(C(C2CCCC3CC23)=O)C2(CCC2)C1 1310,C1(CC)CN(C(=O)Cn2cc(C)cn2)CCC1NC(=O)C(C(F)(F)F)OC(C)=O 1311,N1(C(C2ON=C(C)C2)=O)CC2CC(C)N(C(c3csc4c(F)cccc34)=O)C2C1 1312,N1(CCNC(C(C2CCCCC2)NC(c2[nH]cc(C(C)=O)c2)=O)=O)CCOCC1C 1313,CC(C)C(C)C(=O)N1CCN(CCOCCN(C(=O)CC2CCCCC2)C)CC1 1314,C(=O)(CC(F)(F)C(F)(F)F)N1CCC(C)(CNC(C(C(C)C)n2cccc2)=O)C1 1315,N1(C(c2cc(C(C)C)on2)=O)CC(NC(C2CC2(Cl)Cl)=O)C2(CCOCC2)C1 1316,N1(C(Cc2cc(C)sc2C)=O)CC2CC(NC(C3(C#N)CCCC3)=O)C(C2)C1 1317,CCC(CC)C(C(=O)N1CCN(CCNC(C23CC(C)(CCO2)C3)=O)CC1)OC 1318,c1(-n2ncc(NCC3(C(=O)OCC)CCNC3)c2)ccnc(F)c1 1319,C1(NC(C(CN(C)C)(C)C)=O)CC12CCN(C(c1sccc1I)=O)CC2 1320,N1(C(CC2(CC)CCC2)=O)CC(CC(=O)NCC2(CO)CC3CC3C2)CC1C 1321,C1(CNC(c2ccncn2)=O)CN(C(C2CC3(C2)CC(F)(F)C3)=O)CCC1(F)F 1322,N1(C(COCCN(C)C)=O)CCC(C)(NC(C2CCCN(CC(F)F)C2)=O)C1 1323,C=CCCC(C(=O)N1CC(CC(=O)OCC)C1)NC(=O)C(C(C)CC)N(C)C 1324,C1(CNC(CC2C(CNC(C(CC)OC)=O)C2)=O)CCC2(CC1)CC2 1325,c1(NC(C23CCCCC2C3)=O)ccc(OC(F)F)cc1F 1326,C(CCCCCN(C(=O)CCN1CCC1)C)NC(C(C)C1CCCO1)=O 1327,N1(C(C2(C#N)CC2)=O)CCC2(CCC2NC(C2CN(C(c3ccccc3)=O)C2)=O)CC1 1328,C1(NC(c2cccc(C#C)c2C)=O)CC2CCC(C1F)N2C(C1(CF)CC1)=O 1329,Cc1ccc2c(c1)CC(NC(=O)N(C)C(c1cccs1)C)CO2 1330,C1=C(c2cc(NCc3ccc(-c4cccnc4)cn3)n[nH]2)CCNC1 1331,C(=O)(C1=CC2C=CC1C2)NCC1CN(C(C(c2c(C)n[nH]c2C)C)=O)CC1(F)F 1332,C1(c2nnnn2C)(NC(C2CCOCC2)C)CCCC1NC(=O)OC(C)(C)C 1333,N1(C(C=CSC)=O)CCCC(CNC(=O)C(F)(F)C2CCOCC2)CC1 1334,N1(C(c2n[nH]c(C)c2Cl)=O)CCC2C(C(=O)NC3(C)CCCC3(C)C)C2C1 1335,C1(C(=O)NC2C3CN(C(C(C=C)(C)C)=O)C2C3)Cc2cc(C)ccc2O1 1336,Cc1nc2c(o1)CCN(C(=O)C(CCOCCO)NC(=O)CN(C)C)C2 1337,c1(C(=O)NCC2C(NC(c3c(C#C)ccc(F)c3)=O)C2)csc2c(F)cccc12 1338,N1(C(CCC2CC(OC)C2)=O)CCN(C(c2ccc(O)cc2Cl)=O)C(C(C)C)C1 1339,c1(CCC)ncoc1C(=O)NC1(CCNC(=O)CCn2ccc(C)n2)CCC1 1340,C1(NC(c2c(C)ncs2)=O)COC2(CCN(C(C3(C#N)CCCOC3)=O)CC2)C1 1341,c1(NC(C2C3CC2N(C(=O)C(Cl)(Cl)Cl)C3)=O)cnc(Br)nc1 1342,c1(SCC)ccccc1C(N1CCC(N(C)C(c2oc(COC)nc2C)=O)C1)=O 1343,C(CC)(C(=O)N(C)CC1CCN(C(C2(C3CCCO3)CCC2)=O)C1)=CC 1344,C1(C(N2C3(C(=O)Nc4c(OC)ncnc4)CC3CC2)=O)CCCCC(=O)N1 1345,C(=O)(C#CC1CCOCC1)NC(C1CCN(C(c2cc(Cl)cc(C)c2O)=O)C1)C 1346,C1(C(=O)NCC(C)NCCO)CCN(C(N2CCCC2)=O)C1 1347,c1(C(N2CC(CN(C(CC(C)SC)=O)C)C3(C2)CC3)=O)cc2cc(C)ccc2[nH]1 1348,c1(C(=O)NC2(C)CC(NC(c3cn(C)c(=O)cc3)=O)C2)coc2ccc(F)cc12 1349,c1(C(=O)NC(CC)(C)CNC(=O)COCc2nc(CC)no2)cc(Cl)ccc1N 1350,C(=O)(C(CC1CCC1)C1CCC1)NCCCCN(C(=O)C(c1cccnc1)O)C 1351,c1(NC(C2(CC)CCN(C(c3cc(O)cc(=O)o3)=O)C2)=O)ccc(O)c(Cl)c1 1352,C1(C(=O)NCC(C)CN(C)C(C2CC3CC3C2)=O)CCc2ccnn2C1 1353,C1(OC)CC(NC(c2ccsc2)=O)CN(C(c2cncc(OC(C)C)c2)=O)C1 1354,C1(C(N)=O)CN(C(C2(F)CN(C(C3(c4cccs4)CC3)=O)C2)=O)CCC1O 1355,O=C(N=c1cc2ccccn2[nH]1)N1CCOC(C2CCCCC2)C1 1356,CCCC(C(=O)NCC1CC2CN(C(c3ccc(Cl)cc3OC)=O)CC12)C(C)C 1357,CC#CCCCC(=O)NCc1ccc(C(=O)NC(C)CN(C)C)cc1 1358,C1(NC(C(CC)CC)=O)CC(F)(F)CC1NC(c1cc(Cl)c(Cl)s1)=O 1359,c1(NC(=O)CSCc2ncc[nH]2)ccccc1.CC1C(=O)NCC(CO)N1C 1360,C1(O)(C(N)=O)CCCN(C(C2CSCCN2C(c2cc(Cl)cs2)=O)=O)C1 1361,c1(CC(N2C(CNC(CC=CCC)=O)CC2)=O)cc2ccccc2nc1O 1362,N1(C(c2c(CCC)n[nH]c2)=O)CC(C(=O)NCC=C(C)C)C(C)C1 1363,C1(C(=O)OC)C2C=CC(CC2)C1C(N1CCC(NCC2CC2c2cnc[nH]2)C1)=O 1364,C1(N(C(C(C=C=C)C)=O)C)CN(C(=O)C(F)(F)Cc2ccccc2)CC12CC2 1365,C1(NC(C(C)OCCCC)=O)CCC(O)CN(C(C2(c3ccn(C)n3)CC2)=O)C1 1366,c1(CNC(C(=O)Nc2c(C(=O)OC)scc2)=O)cccc(NC(C)=O)c1 1367,C1(C(N(C2(CO)CC2)C)=O)CN(C(=O)CC2CCSC2)CCC1(C)C 1368,N1(C(C(CC)C#N)=O)CC2C3CCC(C2C1)N(C(C1CC1(C)C(F)(F)F)=O)C3 1369,CCC(C(=O)N1CCN(C)CC1C(=O)NCC1(OC)CCOC1)C(C)(C)CC 1370,C1(C(C)C)CCC(C(=O)N(C)CC2CCCN(C(C3(CO)CCCO3)=O)C2)CC1 1371,N1(CC(N2C(CN(C(C3COCCO3)=O)C3CC3)CCC2)=O)CCCCC1=O 1372,c1(C(N2C(CNC(CCC#C)=O)CC(O)C2)=O)cc(OC)cc(F)c1 1373,CO[Si](CCCNC(N1CCC2(CCCCO2)C1)=O)(OC)OC 1374,C12(NC(COCCCC)=O)CCC(CNC(=O)C=CC(C)C(C)C)(CC1)OC2 1375,CCCCC(C(=O)N1CCC(C)C1CNC(=O)C(C1CCOC1)OC)C(C)C 1376,N1(C(CCCOC)=O)CCCC2(NC(=O)CN(c3ccccc3)C)CC12 1377,N1(C(CCCC=C)=O)CCN(C(C23CC=CC(C2)OC3)=O)C(CC)C1 1378,c1(C(N2CC(NC(CSC(C)C)=O)C(C)(C)C2)=O)c(F)cccc1[N+](=O)[O-] 1379,c1(C(=O)NC2CC3(C2)CN(C(C2CCS(=O)(=O)N2)=O)C3)cc2cccnn2n1 1380,CCC#CCN=c1nc(N2CCC(c3ccccn3)CC2)c2c([nH]1)CCC2 1381,c1(C(=O)NCC(CO)NC(CCNC(N)=O)=O)coc2c1C(=O)NCC2 1382,c1(NC2(CNC(c3nc(NC(C(C)C)=O)sc3)=O)CCC2)ccccc1[N+](=O)[O-] 1383,CCC(CC(=O)NC(CC(F)F)C(=O)N1CCCC(C(C)C)CC1)CC(C)C 1384,CN1CC=C(CC(=O)NC2CCN(C(C3CC3C(=O)NCCO)=O)C23CCC3)CC1 1385,Cc1ccc2cc(C(N3CCCCC3CN(C)C(C3COC3)=O)=O)cnc2c1 1386,C1(C(=O)NC(C)(CNC(c2cc(C(F)(F)F)n[nH]2)=O)CO)COC2(CCC2)CO1 1387,c1(C(=O)NCC(CC)(CC)NC(C(C2CC2)OCC)=O)c[nH]c2c(F)cccc12 1388,C(C(O)CCNC(C1CN(C2CCOC2)C1)=O)NC(c1cccs1)=O 1389,C(=O)(C(CNC(c1ccc(C)nc1)=O)C(C)(C)C)NCCC(COC)O 1390,c1(CC(=O)NCC2(C(=O)NCC(F)CO)CCC2)cnoc1 1391,C12(NC(C(C(CC)C)OC)=O)CCCN(C(=O)Cc3ccnc(C)c3)CC1C2 1392,N1CCC2(CCC(O)CC2)C1.C1(OC)CC2(C(C(=O)C=CC(C)C)c3cccs3)CC12 1393,N1(C(c2ccc(C(C)(C)C)o2)C(=O)NCCCC)CCCC(COCCOC)C1 1394,C(=O)(N=c1ccn(CCF)[nH]1)NC(c1cc(Br)ccc1OC)CC 1395,c1(OC)ccccc1-c1c[nH]cc1C(=O)NC1CC1NC(=O)C=Cc1cscn1 1396,C(C1=NOC2OCCC12)NC(=O)Nc1cn(C2COC2)nn1 1397,Cc1ccc(N)cc1C(N1CC2(C1)CN(C(c1cccnc1SC(F)F)=O)C2)=O 1398,C1(NC(C2CCCN(C(=O)CCC3CCOC3)C2)=O)CCC([N+](=O)[O-])CC1 1399,C1(C(=O)NCc2n(CC)ncn2)CCN(C(C2CCOC2C)=O)C1C(C)C 1400,c1(C(=O)NCCC(C)NC(C2(c3c(OC)cccc3)CC2)=O)cccc(F)c1N 1401,N1(C(C2CCC(C)CC2)=O)CCOC2(CCN(C(=O)C=C3CCC3)C2)C1 1402,N1(C(c2n[nH]cc2Br)=O)CCC(C2CC2)C1CNC(C1(CCF)CCC1)=O 1403,c1(C(N(C2CCN(C(CCC(=C)C)=O)CC2)C)=O)c(Cl)cccc1[N+](=O)[O-] 1404,C(=O)(C(C)(c1ccccc1)OC(C)C)N(CC(C)NC(C=CCC)=O)C 1405,C12(C(=O)NC(C(=O)OC)C)COCC1CN(Cc1ccc(OCCN(C)C)nc1)C2 1406,C1(C(=O)NCC2(SC)CC2)CCCN1C(C)C.C1=CC(=O)NC1(C)C 1407,C(CC(C)(C)C)(C(=O)NCCCC1(O)CCC1)NC(C(CCC)C)=O 1408,c1(SC)ccc(C(N2CC3CC3(CNC(=O)CC(C)C)C2)=O)cc1Br 1409,c1(C(=O)NC2(CC(=O)NC3CC(CC)(CC)C3)CC2)cccc(F)c1O.O 1410,N1(C(CC2ON=C(C)C2)=O)CCCC(CN(C(=O)C(c2ccc(Cl)cc2)O)C)C1 1411,c1(C(=O)NC2C=CC(CNC(c3n(CC)ncc3)=O)C2)c(F)cccc1F 1412,C(c1cc(F)cc(F)c1)=CC(=O)NCC1C=CC(NC(Cc2c(C)cnn2C)=O)C1 1413,N1(C(c2c(C)c[nH]n2)=O)CC(C(=O)N(C2CCCC2C#N)C)CC(C)C1 1414,C1(NC(c2c(C)cn(C)n2)=O)CC2(C1)CC(NC(c1csc(C)c1N)=O)C2 1415,N1(C(CC2CN(C)C2)=O)CCC(NC(=O)CC(O)C2CC2)C2(CCC2)C1 1416,c1(C(C)NC(C2(C)CCCN(C(C=C(C)C(=O)O)=O)C2)=O)ccc(C#N)cc1F 1417,C(=O)(C1CCCc2n[nH]cc21)N(CC(C)NC(c1ccc(CC)cc1N)=O)C 1418,c1(C(=O)NCC(CNC(c2c(CC)nns2)=O)(C)F)ccc2ncncc2c1 1419,CON=C(C(=O)NCC1(C)CCN(C(=O)C2CC2)CC1)c1ccco1 1420,n1(C(C)(C)C)nc2c(c1C(=O)NCCCNC(c1cc(Cl)ccn1)=O)CCCC2 1421,Cn1c(=O)[nH]c(NCC2(CNC(C34CC=CCN3CCC4)=O)CC2)c(C#N)c1=O 1422,C1(CC#C)(C(=O)O)CCN(C(C2CCC(N)CC2)=O)CC1 1423,c1(C(N2CC3C(C(N4CC(C)NC(=O)C4)=O)(CC3)C2)=O)ccn2cncc2c1 1424,Cc1nc(C(=O)NCC2CC2CNC(c2ccc(Br)s2)=O)cn1C 1425,c1(NC(C2COCCN2C(=O)CCCc2ccccc2)=O)ccc(Br)cc1CO 1426,C1(C(=O)NCCN(C(COCC=C)=O)CCC)CC(C)CO1 1427,CC(C)(C)CC(=O)NC1CC2C(NC(=O)COC3CCCOC3)C2C1 1428,Cc1ccc(SC(C)C(=O)N=CCC2(CO)CN(C(C3C(C)CC3C)=O)C2)cc1 1429,c1(C(N(CC(N2CC(OC(N)=O)C2)=O)C2CCC2)=O)coc(CO)c1 1430,c1(C(=O)NCC(CC)NC(c2ccc(C)nc2NC)=O)nsc2c(Cl)cccc12 1431,n1(CCCC)nnnc1C(CCC1CC=CCC1)NCC=C(C)C 1432,CC1CCN(C(c2cnn(-c3ccc(F)cc3)n2)=O)CC1NC(c1cnns1)=O 1433,C(=O)(CC(O)CNCC(F)(F)F)N(CCCOCCNC(C1C(COC)C1)=O)C 1434,C1(C(=O)Nc2cn(CC)nc2)CC2C=CC1N(C(C1CC1c1ccccc1)=O)C2 1435,c1(CC)cccc(C(=O)NCC2(O)CCN(C(=O)Cc3cnn(C(F)F)c3)C2)c1 1436,C(N=c1cc(C)nc(Cl)[nH]1)C1CN(C(C2(COC)CCCCO2)=O)C(C)C1 1437,C=CC(C)(O)C(=O)NCC(C)(C(C)C)NC(c1cc(Cl)sc1Cl)=O 1438,C1(NC(=O)NCCc2n(C)ccc2)CCCCC(C)(C)C1 1439,CC1CCC(CC(N2CC(CC(F)C(=O)N3CCC3(C)C)C2)=O)C1 1440,N1(C(c2c(C)nsc2)=O)CC(N(C)C(c2cncs2)=O)C(F)C1 1441,CCC(CC)C(C(=O)NCCC(=O)NC(CO)C(C)C)OC 1442,C=CCC(CC(C)C)C(=O)N1CCCC(C)(C)C1CNC(C1(C(C)C)COC1)=O 1443,CCC(c1cccc(Cl)c1)=CC(=O)NCC1CCC1NC(=O)CC1CC1 1444,CC1CCCC1(C)NC(=O)CCOCCCNC(C1CCC(N(C)C)C1)=O 1445,CC1CCCC(O)(C(=O)Nc2ccc(F)c(NC3CCCCC3)c2)CC1 1446,Cc1nc(C(C)C)sc1C(=O)NC1CCC(CNC(c2n[nH]cc2Cl)=O)C1 1447,c1(NCc2ncc(CC)[nH]2)ncc(Br)c2cccnc12 1448,N1(C(C23CCC(C)(CC2)OC3)=O)CCCC2CN(C(c3ccsc3Cl)=O)CCC12 1449,C(=O)(NNc1c(Cl)cccc1Br)C1CC(=O)NC1 1450,c1(NC(=O)Nc2cc(CCCC)oc2C)c(Cl)ccnc1Br 1451,c1(C(=O)NC2C(C(N3C(CC)C(O)CC3)=O)CCCC2)ccc(C)c(C#N)c1 1452,C1(C#CC(=O)N2CCC(O)C2C(=O)NC2(COC(C)=O)CC2)(CC)COC1 1453,N1(C(CCC(C)(C)F)=O)CCC2(CCCN(C(=O)CC(C)(C)C3CC3)C2)C1 1454,n1(CC)cc(NC(C2CC(C)CN2Cc2cnc(N(C)C)cn2)=O)c(C)n1 1455,N1(C(=O)NC(C)(CO)C(F)F)CCC2(C1)CN(C(c1ccccc1)=O)CCO2 1456,C#CCC(C)(C(=O)NC(c1nc[nH]n1)CC)NC(=O)CC1CCC(=O)N1 1457,c1(C(=O)NCC2CC(OC)CN2C(c2cnnn2C)=O)cc(Br)cnc1N 1458,c1(C(N2CC(CN(C(c3cc(C)n(C)n3)=O)C)OCC2)=O)ccn2cnnc2c1 1459,c1(OC)ccc(C(=O)NCC2CC(F)(CNC(C3(F)CC3C)=O)C2)c(F)c1 1460,c1(C(=O)NCC2(F)CCC(NC(c3c(C)noc3)=O)C2)cnc2ccccn12 1461,n1(CC(N2CCCC(N(C(C(CCC)C)=O)C)C2)=O)ncc(C#N)c1Br 1462,C1(C(N(CCC(=O)NCC2(C3CC3)CCC2)CC#C)=O)CCCC(C#N)C1 1463,c1(C(N(CC(C)NC(=O)CCc2cn[nH]c2)CC)=O)ccc(SC(F)(F)F)o1 1464,C1(C(=O)NC2CC3N(C(CCOCC)=O)C(CC3)C2)Cc2cc(C)c(C)cc2O1 1465,CCCCCC(O)CC(=O)NC(CNC(=O)CCOc1cccnc1)CCC 1466,C(=O)(CC1=NNC(=O)C1)NCCC(CCNC(C(C)C1CC1)=O)C 1467,N1(C(c2c(C(C)C)c[nH]n2)=O)CCC2CN(C(c3csc(C(N)=O)n3)=O)CC2C1 1468,C(=O)(C1=C(C#N)CCC1)N1CCC(OC)(CNC(C2CN(C)C2)=O)CC1 1469,C(C(=O)N(C)CC1C2CN(C(=O)C=CC(F)(F)F)CC12)(C(C)C)n1ncc(C)c1 1470,N1(C(c2c[nH]c(=NC)s2)=O)CCN2CCN(C(=O)C(C)C3CC3)CC2C1 1471,C12(CNC(CC3CCN(C(C)=O)C3)=O)CC(NC(C3CCCSC3)=O)(CCO1)C2 1472,C1(C(=O)N(CC(O)CO)C)(CC)CCN(C(c2ccnn2CCF)=O)C1 1473,C1(C(N(C(CNC(N)=O)C)C)=O)CCC(NCc2cn(CCCC)nn2)CC1 1474,C(=O)(C1=CS(=O)CCC1)N1CCC(n2cc(CC(COC)O)nn2)CC1 1475,Cc1cc(=NC2CCC(N(C)C)C2)[nH]c(NCc2[nH]cnc2C)n1 1476,O=C(C=CCN(C(=O)CN1CCCCC1)C1CC1)NOCC1CCC1 1477,n1(CC)c(C)cc2c1CCCC2NC(=O)C(=O)NCC1OC(=O)CC1(C)C 1478,c1(OC)cc2[nH]ncc2cc1COC(C1CN2CCC1C2)=O 1479,N1(C(C(c2cnn(C)c2)NC(Cc2cc(C)n(C)n2)=O)=O)CCCCCC1C 1480,N1(C(C2C(COC)CC2)=O)CCc2ccccc2C1CO 1481,c1(C(=O)NC2C(CNC(COC(C)C)=O)C2)coc(Cl)n1 1482,C1(CNC(=O)C(O)CC2CCCCC2)COCCN(C(C2CC=CC2)=O)C1 1483,C1(NC(=O)C(F)C2CCOC2)CC2(C1)CC(N=c1[nH]ncs1)CCS2(=O)=O 1484,C1(NC(Cc2ccc(C)cc2)=O)CCN(C(c2ccc(C)n2C)=O)CC1C(N)=O 1485,c1(C(=O)NC(CN(C(c2cc(CC)on2)=O)C)(C)C)sc2nccnc2c1N 1486,O(NC(=O)C(F)C(C)CNC(C1(C)CC(=O)C1)=O)CCCC=C 1487,CC1CCN(C(=O)C(O)CC2CCCC2)CC1CNC(c1ccc(C2CC2)nc1)=O 1488,c1(OC)cc(CN2CCC(NC(c3cccc(F)c3I)=O)C(F)C2)ccc1C 1489,CN1C(=O)CN(CC(=O)NC2COCCN(C(C3(F)CCCOC3)=O)C2)C1=O 1490,C1(C2CCN(C(=O)C(C)P(C)(C)=O)CC2)(NC(CCCC(C)C)=O)CC1 1491,N1(C(CN(CCC#C)C)=O)CC2CC1(C(=O)NC1CCN(C(N)=O)C1)C2 1492,Cc1nccc(Cl)c1C(N1CC(N(C(=O)C(Cl)=CCl)C)C(C)(C)C1)=O 1493,N1(CC(=O)NCC2CC(F)(F)CN2C(=O)CCc2ccco2)CCCNS1(=O)=O 1494,c1(NC(C2(C)CCN(C(=O)Cn3cc([N+](=O)[O-])cn3)C2)=O)ccc2oncc2c1 1495,Cc1csc(C(=O)NC2(C(=O)N(C)CC3(O)CCOC3)CC(O)C2)c1 1496,N1(C(C2CCN(C(=O)OCC)CC2)=O)CCCC(NC(C2CC(C)(O)C2)=O)C1C 1497,C1(CNC(c2n[nH]c(C)c2Cl)=O)CC2CN(C(=O)C=Cc3ccc(Cl)cc3)CC12 1498,c1(OCCC)cccc(C(N2CC(O)CC2CNC(C2(C)CCNC2=O)=O)=O)c1 1499,C(C(C)C(F)C(=O)NCC1CCC(=O)NC1C)NC(CC=CC=C)=O 1500,C1(CNC(=O)CCCN2CCCC2)CCN(C(=O)CCCC2CC2)C12CCC2 1501,Cc1cc(C)n(CC(=O)NC2(Cn3cc(-c4cscn4)nn3)CC(F)(F)C2)n1 1502,C1(CNC(CCNC(=O)NC)=O)(NC(=O)C(CO)NC(N)=O)CCOC1.C(C)C 1503,C1(CC)CCCC1(C)C(=O)NCC1CCCC1NC(c1cc(C)[nH]n1)=O 1504,C#CCCN=C(NCC1CCCC(C)(C)C1)NC1CC(=O)N(CC(F)(F)F)C1 1505,N1(C(C)C)CCC(CNC(=O)C(O)CNC(=O)C(F)=CC2CC2)C1 1506,C1(NC(Cc2cn(C)nc2)=O)CC2(C1)CN(C(C1CNC(=O)C1)=O)C2 1507,CCCCN=C(NCCN1CCCCC1=O)NC1Cc2ccccc21 1508,Cc1ccccc1CC(N1CC2C(C(=O)NCc3cnon3)C2C1)C 1509,c1(C(c2n(C(C(=O)OC)C)nnn2)NC2C(C)C2(C)C)ccc(OC)nc1 1510,C1(NC(C(C2CCCCC2)N(C)C)=O)C2CCCN(C(=O)CNC=O)C2C1(C)C 1511,c1(C(N(C2CCCN(C(C3CCCCN3C)=O)C2)CC)=O)[nH]c(O)nc1C 1512,c1(C(=O)NC(c2ccccc2)C(C)NC(CSC)=O)ccc(O)c(Br)c1 1513,N1(C(C(CC)C(C)O)=O)CCC2CC(NC(c3cc(F)ccc3Cl)=O)CCC2C1 1514,N1(C(CC(=O)NCC#C)=O)CC2CC(NC(=O)CC3COCC3(C)C)C(C2)C1 1515,c1(C(N2CCN(C(c3c(CC)cncc3)=O)C(C)C2)=O)cc(F)cc(Cl)c1O 1516,C(=O)(C(C)CC(=C)C)NCC(CC=C)NC(c1cc[nH]c1C1CC1)=O 1517,C1(OCC)CN(C(=O)C=Cc2csnc2C)CC1CNC(=O)CSC1CCCO1 1518,c1(C(=O)NC(CC)CNC(=O)C(=O)NC(C)C)sc(C(C)C)nc1C 1519,CCCC(C)CCN=c1[nH]ccc(=NCCOc2ccc(Cl)cc2Cl)[nH]1 1520,CC(C(=O)NC1CCCCC1CNC(=O)CSCCC(F)(F)F)C(C)(F)F 1521,c1(CNC(c2cc(C)ncn2)c2n(CCCSC)nnn2)ccc2nsnc2c1 1522,Cc1[nH]c(C)c(C(=O)NCc2ccoc2C(=O)N(C)CC2CCN(C)CC2)c1C 1523,S(=O)(=O)(c1cccc(=NC2CCC(F)(F)C2)[nH]1)NCc1c(C)nc(C)c(C)n1 1524,C1(N(C)C)CC(N=c2[nH]c(N3CCc4nc(N(C)C)sc4C3)nc(=N)[nH]2)C1 1525,C(=O)(C(C(C)NC(=O)CCc1cnco1)C(C)C)NCCC(=O)OCC 1526,N1(C(CC2CC(C)(C)C2)=O)CCN(C(C2CCO2)=O)CC1c1cccc(Cl)c1 1527,CN1C(=O)NCC1C(=O)NC1CCN(C(=O)CCSc2ccc(F)cc2)C1 1528,C1(C)(CNC(C(C)C2CCOC2)=O)CCCN1C(=O)CS(=O)(=O)NC(C)(C)C 1529,N1(C(c2cc(C)c(Cl)cc2Cl)=O)CCC2(CC(NC(=O)CC3(C)CC3)CO2)C1 1530,C(=O)(C#CC1CCOCC1)NC1C(CNC(CC2(CC(=O)OC)CC2)=O)CCC1 1531,N1(C(C2C(=C)C2)=O)CCc2ccccc2C1CNC(c1cnn(C2CC2)c1Cl)=O 1532,C1(CN(C)C(C2CC23CC(NC(C24CCC(C2)C4)=O)C3)=O)CCCCC1(C)C 1533,C#CCC(C)(CC)C(=O)N1CCC1CNC(C1(O)CCSCC1)=O 1534,Cc1ccc2c(N(CCC(N)=O)C)nc(N(C)CC3CCCS3(=O)=O)nc2c1 1535,C(C)(C(CC(=O)NCCc1ccc(F)nc1)NC(=O)CCN1CCCCC1)OC 1536,C1(NC(CCc2ccc(SC)cc2)=O)CCN(C(=O)Cn2nccc2C)C(C)C1 1537,CC(C(C)NC(=O)NCc1ccnc(OCC(F)F)c1)S(C)(=O)=O 1538,C1(CNC(c2cn(CC(C)C)nc2C(F)F)=O)CCCCN(C(=O)C=C(C)Cl)C1 1539,c1(CCC(=O)NC(CCNC(C2C(C(=O)OC)CCC2)=O)C)ccccc1OC 1540,CCCCCC(=O)NC(c1ccccc1)C(C)NC(c1cccnc1S)=O 1541,Cc1cc(F)ccc1CC(=O)NCC1CC(NC(=O)C(C)(C)c2ccccn2)C1 1542,c1(SC)ccc(OCC(=O)NCCN(C(=O)C(C)SC(F)(F)F)C2CC2)cc1 1543,N1(C(CC(=O)OC)=O)CCCC(O)(CNC(=O)CNS(C)(=O)=O)C1 1544,C1(O)(CNC(C2CCCS2)=O)CCCN(C(=O)CN2CCCC2)CC1 1545,C(=O)(C(CO)c1ccccc1)NC(C1CCN(C(=O)CCc2cc[nH]n2)C1)(C)C 1546,n1(CC)ccc(CN(C(=O)COCCNC(=O)C(C)C2CCOC2)C)n1 1547,c1(C(=O)NCCCN(C(CC2CC(CC)C2)=O)CC)ccc(F)cc1C(F)(F)F 1548,N1(C(CC(C=C)CC)=O)CCC(C(=O)N(C)Cc2ccc(C)nc2)C(C)(C)C1 1549,C1(NC(C2C=CCN(C(c3ccccc3)=O)C2)=O)CC2(CCC2)C1O 1550,C1(C(N2CCN(C(CC(n3ccc(C)n3)C)=O)CC2C)=O)CC2CCCCN2C1 1551,C1(CC(=O)NC(CNC(C(C(C)C)OC)=O)(C)C)CCC(=O)NC1=O 1552,Cc1nc2ncc(C(=O)NC(CNC(=O)Cn3cncn3)CC(C)C)cc2o1 1553,C1(NC(C23CCC(C2)C3)=O)CCCC(NC(C2(Br)CC2)=O)C1 1554,C1(CC(=O)NCC2CCC(C)C2)CCN(C(=O)C2=NNC(=O)C2)C1(C)C 1555,C#Cc1ccc(C(=O)NCC(O)CCNC(c2c[nH]cc2C)=O)cc1 1556,C(C(N=c1[nH]c(Cl)nc2[nH]cnc12)C1CCC1)NC(C=CC)=O 1557,C1(NC(C(CCF)NC(COCCC)=O)=O)C2CCC(C2)C1C 1558,C(=O)(C#CC1CCCOC1)NC1C(C)(C)N(c2nc(C#N)ncc2Cl)CC1 1559,N1(C(C2=CCCN(C(CCCC(C)=O)=O)C2)=O)CCCC2COCC12 1560,c1(C(C)C)cccc2c(C(=O)NCC3CCOC3C(=O)O)ccnc12 1561,CC(CCC(=O)N1CCC(C)(CNC(=O)COCC(C)(C)C)C1)N(C)C 1562,C1(N(C(=O)CCc2ccccc2)CC)CCCN(C(C2(Cl)CC2(F)F)=O)C1 1563,c1(CC)nn(C)c(CC(N2CCCC(NC(c3cncn3C)=O)C2C)=O)c1Br 1564,N1(C(CCCSC)=O)CC(NC(=O)C=CC2CCCCCC2)CC(C)(C)C1 1565,c1(N(C2CC3(CNC3)C2)C(c2cc(OC)cc(C)c2)=O)ncnc2ncn(C)c12 1566,c1(OC)nc(C)sc1C(=O)NCC1CCC(NC(c2ccc(C(C)C)nc2)=O)C1 1567,C1(CC(C)NC(C(C)(C)SC)=O)CC2CCC(C1)N2C(=O)CCn1ccc(=N)[nH]1 1568,C(=O)(CCCS(C)(=O)=O)N1CC(NC(C(C=C)(C)C)=O)C2C(C1)C2 1569,C1(C(=O)OCC)CC2CCC1N(C(=O)C(=O)NCc1cccc3c[nH]nc13)C2 1570,C1(CC(=O)N(C)Cc2nccs2)CCCN(C(C2CC3C=CC2C3)=O)CC1 1571,N(C(=NCC(C)(C)C(N)=O)N1CCN2C(CCS2(=O)=O)C1)C(C)C1CC1 1572,S(=O)(=O)(c1cc(C(F)(F)F)ccc1NCCC(F)(F)Cl)NCC(C)CC(C)O 1573,C12(CCN(C(=O)CSCCN(C)C)C1)C(=O)N2.C1(CC)CC(CN(C)C)C1 1574,CCCC(CCCNC(c1coc(C(C)C)n1)=O)NC(c1cc(Br)n[nH]1)=O 1575,c1(CCC(N2CCC(C(C)NC(=O)CCc3cnn(C)c3)C2)=O)ncc(F)cn1 1576,CC1(C)CC(NC(C2CC2F)=O)CCN(C(=O)CCc2cc(Cl)cs2)C1 1577,C1(C(=O)OCC)(C(=O)NC2CCN(C(c3cn(CC)nc3C)=O)C2)CCOCC1 1578,N1(C(C(C)(F)F)=O)CCCC(C2CCN(C(C3(C#N)CC4CCC3CC4)=O)C2)C1 1579,CN=c1[nH]c(C(N2CCN(CC(C)(C)NC(C3CC34CC(O)C4)=O)CC2)=O)cs1 1580,C1(CNC(c2n(C(C)(C)C)ncc2)=O)CN(C(C2CC2(F)F)=O)CCC1(C)C 1581,C12=NC=CC(=NC3CCC4CN(CC34)C1=O)N2.CCCCCCC(C)C(=O)NCC 1582,N1(C(c2c(CC)oc(C)c2)=O)CC(CNC(C2(CC)CC2(F)F)=O)CC12CCC2 1583,c1(C(=O)NC2(C)CN(C(Cc3c(C)nc(C)s3)=O)C2)cc(S(N)(=O)=O)sc1C 1584,Cn1c(O)ncc(C(N2CCC3C(NC(C4CCS(=O)(=O)N4)=O)C23)=O)c1=O 1585,c1(N2CCC(NC(c3ccc(C)cc3)=O)C(C)C2)cc2nncn2c(C)n1 1586,C1(CC(=O)NCC2=CCN(C(C3COCCO3)=O)CC2)CN2CCC1CC2 1587,C(=O)(C(C)CCCC(C)C)NCCn1ncc(C(=O)NC2CN(CCC)C2)c1 1588,c1(N2CCCC(C)(OC)CC2)nc(N2CCn3ncc(Cl)c3C2)c2c(n1)CCC2 1589,N1(C(c2cccc(I)c2)=O)CC2CCN(C(c3nc4ccccc4[nH]3)=O)C2C1 1590,CCC(CC(=O)Nc1cccc(CNC(C23COC(CF)(C2)C3)=O)c1)C(C)C 1591,C(CC(C(=O)NCC12CC(F)(C1)C2)NC(c1cnc(Cl)n1C)=O)N(C)C 1592,C1(COC(=N)O)CCN(C(=O)C(Cn2ccnn2)NC(=O)CC2CCCCO2)CC1 1593,Cc1ccccc1C1CC1.C12(CCCC1)CC2.N12CCC1C(=O)OCC(=O)NC2 1594,N1(C(C23OC(C)C(C2)C3)=O)CCCN(C(=O)CSc2n[nH]c(O)n2)C(CO)C1 1595,C=C=C(C)CC(=O)NCCCN(C(c1cccnc1OC(F)(F)F)=O)C1CC1 1596,CC(CC(=O)N(C1CN(C(=O)COCc2ccccc2)C1)CO)C(F)(F)C(F)(F)F 1597,Cn1nc(C(N2CCOC(CNC(C3C4CCCCC34)=O)C2)=O)cc1F 1598,c1(OC)cc(CC(N2CC3CC2CN3C(=O)C(O)CC2CC2)=O)c(F)cc1O 1599,c1(CC(=O)N(CC(C)C#N)Cc2cccn(C)c2=O)cc(F)c(F)cc1F 1600,S(=O)(=O)(c1cccc(OC)c1)NCC(c1ccccc1)C.CCCC1CCCN1 1601,Cc1ncc(C(=O)NC(CNC(=O)CC(C)C(C)C)CC(C)C)cc1C#N 1602,Cc1ccc2oc(N3CC(C)(NC(c4cnc(F)c(Cl)c4)=O)C3)nc2c1 1603,N1(S(CCC)(=O)=O)CCCCC1C(=O)NCCCN(C(=O)CCC(C)O)C 1604,C1(C)(C(=O)NC(C(CC)C)CO)CCCN(C(=O)CCc2cc(C)n(C)n2)C1 1605,c1(C(=O)NCC2(CNC(C(CC=C)C)=O)CC2)cc(C)nc2ccc(OC)cc12 1606,Cc1cccc(C(=O)NCC2CC(C)N(C(=O)CC3CCCC(C)(C)O3)C2)c1F 1607,N1(C(CC(C)F)=O)C(C(=O)NC2(C)CCC(C)(C)C2)C2CC(O)C1C2 1608,N1(C(C2(CC=C)CC2)=O)CC(CNC(=O)C(COC)N(C)C)CC(C)(C)C1 1609,N1(C(CCC(=O)NCC)=O)CC2(CNC(=O)Cc3cnccc3Cl)CC1CO2 1610,CC1(NC(=O)Cc2ccco2)CCC(NC(c2ccnn2C2CCC2)=O)CC1 1611,N(C1CCc2c(C(=O)O)cc(F)cc21)C(CS(CC=C)(=O)=O)=O 1612,c1(C(=O)NCCC2CCCN(C(C3CC3(Cl)Cl)=O)C2)cc2cc(Cl)ccc2o1 1613,N1(C(c2c(C)ccc(C)n2)=O)CCC2(CCC(NC(C3CCOCC3)=O)C2)C1 1614,CCC(CC)(CO)C(=O)N1CCCC(O)(CNC(c2cc(C(N)=O)cs2)=O)CC1 1615,C12(O)CCCN(C1)C(=O)c1cnc(cn1)C(=O)N(C)C2.c1(CC)ccsc1OC 1616,c1(C(N2CC(F)(C(=O)NCc3cscn3)C2)=O)ccc(Cl)nc1 1617,C1(NC(CC2N(C(C3CCCC(C#N)C3)=O)CCCC2)=O)CCC2(CCCC2)C1 1618,C12(NC(C3C(OC)C3)=O)CC3CC(C1)CC(CNC(=O)C1=NNC(=O)C1)(C3)C2 1619,O=C(C1=CC2(CCOC2)C1)NC(C1CCN(C(c2cnccn2)=O)CC1)CO 1620,c1(C(=O)NCCCC(C)NC(CC(CC)(C)C)=O)cc2ncccc2o1 1621,CCC(C)CCCCC(=O)N(C)CCNc1ncnc2[nH]c(Cl)cc12 1622,C(=O)(CCS(=O)(=O)CC(C)C)N(CC(CN(C(c1nc(C)oc1)=O)C)O)C 1623,C1(CNC(C(n2cc(-c3nccs3)nn2)C)=O)CC(C2CC2)=NO1 1624,C12(CC(=O)NCCC(C)NC(CCCC)=O)CC3CC(CC(C3)C1)C2 1625,Nc1ccc(C(N2CC(NC(C3CC3C3CCC3)=O)C(F)C2)=O)cc1[N+](=O)[O-] 1626,c1(NC(C(CNC(=O)CN2CCOCC2=O)O)=O)ccc(=O)n(CCO)c1 1627,c1(C(=O)NC(COC)CC(=O)NCC=CCSC)cc(C)cc(O)n1 1628,c1(Oc2c(F)cc3c(c2)NC(=O)CC3)cn(C2CCc3c(F)cc(Cl)cc32)nn1 1629,C(=O)(C(C)CS(C)(=O)=O)N1C(C(N2CC(OC(C)C)C2)=O)C2CCC1C2 1630,C1(CC)CN(C(=O)CCc2cccs2)CCC1CNC(c1cnc(C)cc1Cl)=O 1631,C(=O)(CCC(F)(F)F)NC(C(C)C)CNC(c1cccnc1N(C)C)=O 1632,C#CC1(NC(C2CC2C(C)NC(=O)C(CC)n2ccnc2)=O)CCCCC1 1633,c1(OC)cc(F)c(C(=O)NCC2CCC(C)CN2C(=O)CCNC(N)=O)cc1N 1634,c1(CN(Cc2cn(CCCC)nn2)O)ccc2c(c1)CC(C)(C)O2 1635,C1(C(N2CC(C(C)NC(=O)C(C)C3=CCCC3)C2)=O)CCc2[nH]nc(O)c2C1 1636,c1(C(N2CC(CNC(c3ccc(C#C)o3)=O)C3(C2)CC3)=O)cc(C)c(F)cc1N 1637,CC1c2ccccc2CN1C(N1CCCCC(O)(CNC(=O)NC(C)(C)C)C1)=O 1638,Cc1nc2[nH]c(C(=O)NC(C)CCN(C(=O)C(C)C3CCC3)C)cc2s1 1639,Cc1c[nH]cc(C(=O)NC2(CCCNC(=O)COCC3CC3)CC2)c1=O 1640,c1(C(N(CCCNC(c2c[nH]c(=NCC)s2)=O)C)=O)cc2ccccc2n1C 1641,c1(C(N2C(C(N3CCN4CCC3CC4)=O)CC(=C)C2)=O)cc2nc(C)ccc2o1 1642,C1(CNC(Cn2c(C)cnc2)=O)CCCN(C(=O)Cc2cscn2)CC1 1643,N1(C(C(C)O)=O)CCOC2CCN(C(c3n[nH]cc3OC(F)F)=O)CC12 1644,C1(C(N(C2CN(C(C3(CCOC)CC3)=O)C2)C)=O)CCCCC12CC2(F)F 1645,c1(C(N(C(C(=O)N(C)CCOC2CC2)C2CC2)C)=O)ccc2n[nH]cc2c1 1646,Cc1cc(F)ccc1CC1(C(=O)NCC(CNC(C2CC2F)=O)CO)CC1 1647,C1(C(=O)NC(C2CN(C(=O)Cc3ccncc3Cl)C2)C)CC=CCC1C 1648,Cc1cc(-n2nc(-c3cccc(N)n3)nc2-c2csc(C(C)(C)C)n2)cc(C)n1 1649,c1(C(N(CC(C)(C)NC(=O)CNS(C)(=O)=O)C)=O)ccncc1F 1650,c1(C(=O)NC2CCC(N(C(=O)COc3cccnc3)C)C2)cnn2ccccc12 1651,C1(F)(C(N(CCC(=O)OCC)C)=O)CCCN(C(C2CCC3(CCC3)C2)=O)C1 1652,CC1CCCn2ncc(C(N3CCN(C(=O)C(C)C(F)(F)F)CC3)=O)c21 1653,C1(OCC)CN(C(=O)C(C)SC(F)(F)F)CC1CNC(=O)CSc1ccccc1C 1654,C#CC1(O)CCN(C(=NCCC(=O)N(C)C)NCC2(NS(=O)(=O)CC)CC2)C1 1655,c1(C(N(C)CCNC(=O)CC(F)(F)c2ccccc2)=O)cccc2oncc12 1656,c1(C(C)NC(C(C)N(CCOCC)C)=O)ccc(C)nc1 1657,c1(OC(C)C)cc(C(N2CCN(C(=O)CN(C)C(C)C)CC2C)=O)ccc1Br 1658,C1(C(=O)NC(c2ccno2)C)CC(F)CN(Cc2scnc2Cl)C1 1659,C12(C(=O)NC3C(CNC(c4ncc(C)cc4F)=O)C3)C3CCC(CC13)C2(F)F 1660,c1(C(N(C2CCCN(C(C(COC)C)=O)C2)CCF)=O)cccc(C)c1Cl 1661,C12(CNC(C(C)OCCC#C)=O)CC(CO1)N(C(=O)C(C)(C)n1cc(Cl)cn1)C2 1662,c1(CNC(C2COC(c3ccccc3)C2)=O)nc(C(F)(F)F)cs1 1663,O(N1CCC(CC(=O)NC2CC(C)(SC(c3[nH]cc(C(=O)N)c3)=O)C2)CC1)CC.OC 1664,C1(NC(C2CC2(F)F)=O)CCCN(Cc2cn(C3CCCNC3=O)nn2)C1 1665,Cn1cnc2ccc(C(=O)NCC3CCC(NC(C4CC(F)C4)=O)C3)nc12 1666,N1(C(c2c(CCC)n[nH]c2)=O)CC2CC2C1C(N1CCC1C1CCOCC1)=O 1667,C(=O)(C(=O)N=S(C)(C)=O)N1CC2(CN(C(CC3CC(N(C)C)C3)=O)C2)C1 1668,C12(CC(=O)NC3C(C(=O)Nc4c(Cl)cc(C)c(O)c4)C3)CC3CC(CC(C3)C1)C2 1669,C1(CC=C)(NC(=O)C(CC)OC)CC2CCC(C1)N2C(c1c(C)n[nH]c1C)=O 1670,c1(C(N2CCN(C(C=CC=CC)=O)CC2)=O)cc(S(=O)(=O)NCC(N)=O)c[nH]1 1671,C1(O)(CNC(c2c(C)nn(C(C)C)c2)=O)CCN(C(C2CC2F)=O)CC1 1672,C1(CC(=O)N(CC(O)CNC(c2conc2C(F)(F)F)=O)C)CCN(C)C1=O 1673,c1(CC)cc(=NC(=O)C2CC2CNC(C2CNC(=O)N2)=O)[nH]n1C 1674,C(=O)(C1COc2ccccc21)N1C2CCC(NC(=O)C(O)C3CCC3)(CC2)C1 1675,C1(C(=O)N(CCC(=O)N)CCO)(CNC(=O)CC(C)n2cccn2)CCCO1.CO 1676,N1(C(c2cn(CC=C)nn2)=O)CCOC(C)(CNC(=O)CC=CC=C)C1 1677,N1(C(C)=O)CCN(Cc2nc(CNC(CCF)C(=O)O)no2)CC1 1678,CC1(C)C2CN(C(C3C4CCC(C4)N3C(C3CCC(=O)NC3)=O)=O)CC12 1679,C(=O)(CC(C)C(=O)OC)NCCN(C(c1ccn(C2CCOCC2)n1)=O)CC 1680,C(=O)(CC(CN(C)C)C(F)(F)F)NCCCN(C(CC1(CC=C)CCCC1)=O)C 1681,C1(C(=O)NC(C2(O)CCN(C(C3CC(O)C3)=O)C2)C)CCc2nnnn2CC1 1682,C#CCCCCCC(=O)N1CC2(CC(CNC(=O)C(C)C3=CCCC3)C2)C1 1683,c1(C(=O)NCc2ccc(C(N3CCC(CN(C)CC)C3)=O)s2)n[nH]c(C)c1Cl 1684,c1(C(=O)NCC2CC(NC(CCC=C(C)C)=O)C2)cc(F)cc(Br)c1F 1685,c1(OCC)cncc(C(N2CC(CN(C)Cc3ccc(OC)nc3)C2)=O)c1 1686,N1(C(C(CCC2CC2)NC(C(=O)C2CCC2)=O)=O)CC2(CCC(O)CC2)C1 1687,C(=O)(C(C)S(=O)(=O)C(C)C)N(CCN(C(c1c(N)sc(C)c1C)=O)C)C(C)C 1688,c1(C(C)NC(c2ccc(OCC)cc2)CSC)c(F)cc(Cl)cc1F 1689,c1(C(N2C(CNC(c3sccc3Cl)=O)CCC2)=O)cc(O)nc(C2CC2)n1 1690,N1(C(C(CCC=C)NC(c2ccc(N)c(F)n2)=O)=O)CC2CCC(O)C2C1 1691,C(C(=O)N1CCN(C(=O)CC(C)(O)C2CC2)CC1CCO)(C(C)(C)C)NC(C)=O 1692,N1(C(CC(n2c(CC)ncc2)C)=O)CCC(O)(CCNC(c2ccon2)=O)C1 1693,C(C(CO)(CO)NC(c1ccn(C)n1)=O)N(C(C1C(C=C)C1)=O)C 1694,C1(C(=O)NC(c2cncnc2)C)(CC)CCN(C(=O)CC2CSCCO2)CC1 1695,C1(NC(c2ccc(C(N)=O)[nH]2)=O)COCCN(C(c2cc3occc3[nH]2)=O)C1 1696,CP(C)(=O)C(O)C(=O)N1CCC(O)(CNC(c2ccc(=O)oc2)=O)CC1 1697,c1(C(c2cn(C3CN(SC)CC3C)nn2)C2CC2)cc(N)c(=O)n2c1CCCC2 1698,c1(N2CC(C)(C)C(O)C2)ccc(S(=O)(=O)N2CCCC2c2cccnc2)cn1 1699,c1(C(=O)NCC2(C(=O)NC(C3(CO)CC3)C)CCC2)ccc(F)cc1C1CC1 1700,C1(C(=O)NCC2N(C(C(C(C)C)N(CC)CC)=O)CCOC2)CCCCCCC1 1701,S(=O)(=O)(c1cn(C)cn1)NCC(=O)N(C1CN(C(c2c(C)cc(C)s2)=O)C1)CCO 1702,CC1(C(=O)NC2C=CC(CC(=O)NCCc3noc(=O)n3C)C2)CC=CCC1 1703,N1(C(c2c(C)nn(CCF)c2)C(=O)NC(CC2CCCC2)CO)CCNC(=O)CC1(C)C 1704,N1(c2nc(C(C)C)nc(Cl)c2)CCS(=O)(=O)C(CCNC(=O)CC=C(C)C)C1 1705,N1(C(CC)=O)CCC(C)C(NC(=O)N(C2CCCCCCC2)CCOC)C1 1706,N1(C(c2cc(C)ns2)=O)CCC(NC(c2ccsc2C(F)(F)F)=O)C1C 1707,Cc1nc(O)ccc1C(N1CSCC1C(=O)NCC(C)(C)C#N)=O 1708,c1(C(N(C2CCN(Cc3ccccc3-n3ccnc3)C2)CC)=O)ccc(Br)cc1 1709,c1(C(N2C(CN(C(=O)CCC(N)=O)C)CCCC2)=O)ccc2[nH]cc(C#N)c2c1 1710,CCC(C)C(C(=O)N1CCOCC(CNC(c2ccsc2OC)=O)C1)OC 1711,CN1CC=C(CC(=O)NCC2COCCN2C(=O)Cc2c(O)ncnc2O)CC1 1712,C1(C)(C(=O)NC(C)CNC(=O)C(Cc2ccccc2)n2cnnn2)COCCO1 1713,c1(C(N2CCC(CCOC)(NC(CSCC=C)=O)CC2)=O)ccn2nncc2c1 1714,C1(NC(C=NOC)=O)(CO)CCCN(C(=O)C(c2ccnn2C)C)C1 1715,CC1(C)CCC(O)(C(N2CC(CNC(c3csc(C(F)F)n3)=O)C(O)C2)=O)CC1 1716,CC1CN(C(=O)Cc2cccnc2Cl)CC1NC(=O)C(O)C1CC1 1717,C1(N(C(=O)CC2CC2(Cl)Cl)CC)CCN(C(=O)Cc2cncnc2O)CC1 1718,CC(C)(C)C(O)C(=O)NC1CCCN(C(c2cc(F)ccc2Cl)=O)CC1 1719,c1(C(c2n(CCOC)nnn2)NCCCCO)ncc(C)cc1C 1720,N1(C(C(C)Oc2ccccc2)=O)CC2CCCN(C(c3cnsc3)=O)C2C1 1721,c1(NC(CC(C)O)=O)sc2c(c1C(N1CCNCC1C(C)C)=O)CCOC2 1722,c1(C(=O)NC2(CF)CCN(C(C3N(C(C)=O)CSC3)=O)C2)cncc2ccsc12 1723,n1(C2CCN(C(=O)Cn3nnnc3C(O)C3CC3)CC2)cc2ccccc2n1 1724,C12(C(N3CC(F)(CC)C3)=O)CC(CO1)N(C(C1C(C(C)=O)C1(C)C)=O)C2 1725,Cc1cc(C(N2CCC2C(N2CCC(O)C(C)C2)=O)=O)ccc1F 1726,N1(C(c2cc(C=C)cc(F)c2)=O)CCN(C(=O)C(C)(C)C)CC2CCCCC12 1727,N1(C(c2cc(C)[nH]n2)C(=O)NC(CC)C)CCCC(S(C)(=O)=O)CC1 1728,c1(C(=O)NCC(CN(C(C(c2cccc(C)c2)=O)=O)C)(C)C)cc2n(n1)CCC2 1729,c1(CC)cc(C(=O)N(CC(C)CNC(=O)C=CCN(CC)CC)C)sc1C 1730,CCC(O)C(C)C(=O)NCC1CN(C)CCN1C(C1C=CC=CC=C1)=O 1731,N1(C(C2CC(CC)C2)=O)CC(CNC(c2ccc(Cl)c(F)c2O)=O)CC12CCC2 1732,CC(C(=O)NC1C=CCN(C(c2ccc(-c3cn[nH]c3)cn2)=O)C1)C(F)(F)F 1733,n1(CC(=O)NC(CN(C(=O)CCN2CCCC2)C)(CO)CO)cnc([N+](=O)[O-])c1 1734,C(C)(CNC(c1ccn(C)n1)=O)(CC)NC(C=C(CCC)C)=O 1735,c1(C(N(C2CN(C(c3c(F)ccc(F)c3N)=O)C2)C)=O)cccn2c(O)nnc12 1736,c1(OC)nc(N(C2CCN(C(=O)Cn3ccnc3)C2)C)ncc1OC 1737,CCCC(CNC(=O)C(=O)NC(C)C)C(=O)NCC1COC(=O)N1 1738,N1(C(c2cnc(CNC(CC(CC)(C)C)=O)nc2)=O)CCC2C(CCN2C)C1 1739,c1(CC(=O)NC2C3(CC(NC(C4N(CCC)CCC4)=O)C3)C2)cccc(F)c1F 1740,N1(CCC(=O)NC2(C)CN(C(CC3CC(OC)C3)=O)C2)C(=O)NC(C)(C)C1=O 1741,C1(NC(c2cc(Cl)c(Cl)[nH]2)=O)CN(C(c2cnn(CCF)c2)=O)CC2(CCC2)C1 1742,C1(CCO)CC(N=c2[nH]c(=NC3CCC(C4CC4)CC3)[nH]c3c2COC3)C1 1743,C(CC(=O)N(C)Cc1ccc(SC)cc1)(C1=CCCC1)OCC 1744,C1(CNC(C(CC#C)O)=O)CCN(C(c2scnc2CC)=O)CC1(F)F 1745,c1(C(N2CC(O)(CN(C(C(C=C=C)C)=O)C)C2)=O)cc(C)nc2ccnn12 1746,CC(C)CC(CNC(C1CCCN1C=O)=O)NC(=O)C(C)(C)COCC(F)F 1747,c1(C(C(=O)NCCC)N(CCC#C)C)cc(C(F)(F)F)cc(C)c1 1748,CN1CC(C(=O)NCCC2CCN(C(c3c[nH]c(=O)cn3)=O)C2)CCC1=O 1749,c1(C(N(CC(C)N(C(C(C)OCCC=C)=O)C)C)=O)ccc(Cl)cc1O 1750,C1(C(=O)NC(c2cccnc2)C(=O)N(CCCC)C)CCN(CC)CC1 1751,c1(CN2C(CCNC(C3(C=C)CCCCC3)=O)CCCC2)ccc2c(c1)COC2 1752,C1(C(=O)NCC2(NC(c3cc(N)nc(Cl)c3)=O)CCC2)Cc2ccccc2O1 1753,[nH]1ccc2ccccc12.Cc1ccc(C(O)CNC(=O)CCn2cc(C)nn2)o1 1754,c1(C(N2C(CNC(CCC3N(C)CCC3)=O)CC2)=O)cccn2cncc12 1755,c1(OCCCC(=O)OCC2C3CCC23)ccc2ccccc2c1 1756,C1(C)(NC(C(C2CCCCCC2)C)=O)CCN(C(c2cscn2)=O)C1 1757,CCC(C)(C)C(=O)C(=O)N1CCC(C2CCCN2C(c2ccc(Cl)o2)=O)C1 1758,c1(C(N(C2CN(C(CN(C)C)=O)C2)C)=O)cc(=O)cc[nH]1 1759,C(=O)(C1=CC2(CCOC2)C1)N1CCC(C(N(CC(CC)CC)CC)=O)CC1 1760,c1(C(=O)NC2C(NC(c3scc(OC)c3OC)=O)CC2)ccc2occ(C)c2c1 1761,C1(C2CCCN(C(C3C(C)(C)C3(F)F)=O)C2)(NC(C=C(CCC)C)=O)CC1 1762,c1(OC)ccc([N+](=O)[O-])cc1C(N1CCN(C(=O)COc2nnc(C)s2)CC1)=O 1763,c1(C(=O)NC(C(=O)NC(CC#C)CCOC)CCC)cccc(C#N)c1C 1764,c1(Cc2cn(C3(C(=O)OC)CN(C(=O)CC(C)F)C3)nn2)c(F)cccc1F 1765,c1(CNC2C(C(=O)NC(c3cncs3)C)CCC2)c2c(nn1C)CCC2 1766,c1(N(C(C2N(C(C(CC)N)=O)CCC2)=O)C)cc(C)cnc1C(N)=O 1767,C1(O)(CC)CCCN(C(=O)C=CCN(C(=O)CCn2nc(C)nc2C)C)C1 1768,Cc1nc2cc(C(=O)NCC(O)CN(C(=O)CC3=NNC(=O)C3)C)cc(O)c2o1 1769,CC(C)CCC(F)C(=O)N1CCCC(C)(C)C1C(=O)N(C1COC(C)(C)C1)C 1770,C1(C)(NC(C(C)Cc2cnc[nH]2)=O)CCN(C(C2CCN(CC3CC3)CC2)=O)C1 1771,C(=O)(C(C)CCCOC)NCCCC(C)(C)NC(c1cc(CCCCC)[nH]n1)=O 1772,C#CCCCC(C)C(=O)NCC(CO)NC(c1cc(C(N)=O)[nH]n1)=O 1773,C(C(CC(=O)N1CCC(C)(N(C)C)C1)NC(C1CCCN1C1CC1)=O)OC 1774,C(=O)(C1CCOc2ccc(F)cc21)N1CC(CNC(C(Br)=C(C)C)=O)C1 1775,N1(C(C23C(C)(C)C(CC2)C3)=O)CCCCC(NC(C2CC(=C3CCC3)C2)=O)CC1 1776,Cc1[nH]c(C#N)cc1C(=O)NC1(CO)CCN(C(C2CC(C)(C)CN2C)=O)C1 1777,CP(C)(=O)CCC(=O)NC1CCN(C(=O)CCCc2csc(=N)[nH]2)C1 1778,Cn1ccc2c(C(=O)NCCC3CN(C(=O)Cn4ccnn4)CCO3)ccnc12 1779,c1(SCC(=O)NCC2(COC)CN(C(C3CCC3(C)C)=O)C2)ccccc1Br 1780,c1(CC(=O)NC(CNC(c2n(CC#C)ccc2)=O)C2CCC2)cnc(Cl)cc1C 1781,S(=O)(=O)(c1cccc(NC(=O)CNC(=O)NCCc2nc(=O)o[nH]2)c1)NC 1782,Cc1cnn(C)c1C(=O)NCC(c1ccccc1)NC(=O)CCS(C)=O 1783,n1(CC)ncc(C(=O)NCC=CCNC(=O)CC(C)(C)O)c1C(F)(F)F 1784,C12(NC(CC3CCC(C)CO3)=O)CC(CNC(c3cncc(N)c3)=O)(C1)OC2C 1785,C1(C(=O)NC(c2nc(=O)o[nH]2)C)CC12CCN(C(c1ccc(C3CC3)cc1)=O)C2 1786,CS(=O)CCC(O)C(=O)NC1(C)CN(C(=O)Cc2csc(-c3ncccn3)n2)C1 1787,C1(C(=O)NC2CCOC2=O)CCCC2CN(C(=O)C3Cc4ccccc43)CC12 1788,N1(C(C(N2CC3C(C)(C)C3C2)=O)=O)CC2CS(=O)(=O)CC2C1 1789,N1(C(C2(OC)CCSC2)=O)CCCC(N(C(=O)CNS(=O)(=O)N(C)C)C)C1 1790,c1(N(CCNC(C2CC23CCOC3)=O)CC)c(Cl)cncc1[N+](=O)[O-] 1791,Cc1noc(C)c1C=CC(=O)NC1CC2(C1)CC(NC(c1nonc1N)=O)C2 1792,c1(CC(=O)NC2CCN(C(C=CC(CC)C)=O)CC2CO)cn2ccccc2n1 1793,c1(OC)ccc(Cl)cc1C(=O)NC(C)CNC(c1cccc(F)c1O)=O 1794,CC(CC(F)(F)F)C(=O)NC(CC1CC1)C(=O)N1CC(N2CCC2)C1 1795,c1(OC)c(NC(C2CSCCN2Cc2ncc(C)s2)=O)ccc(Cl)c1Cl 1796,C1(CNC(CCOCCOCC)=O)(CC)CCCN1C(=O)C(C)(F)F 1797,c1(C(C(=O)NC2(CN(C(COC(CC)C)=O)C)CC2)C)cccc(N(C)C)c1 1798,C1(CC(=O)NCCC(CNC(=O)CC(=O)Nc2nccs2)O)CC2C=CC1CC2 1799,c1(CNC(=O)OC2CN(C(=O)C3CC3)C2)ccc(I)nc1 1800,N1(C(C(C(CC)C)O)=O)CC2N(C(=O)Cc3nnc(C)o3)CCC2(C)C1 1801,CCCCC(C(=O)N1CCN(C(C2CC3C(C2)C3(F)F)=O)CC1)NC(N)=O 1802,c1(NC(C23CC(NC(c4ccncc4Cl)=O)(C2)C3)=O)ccc2c(Cl)n[nH]c2c1 1803,C(=O)(C(=O)N=S(C)(C)=O)N1CCC(O)(CN(C(=O)CCC2(C)CC2)C)C1 1804,C(=O)(C1SCCc2sccc21)N1C(C(C)NC(c2cc(C)ncc2)=O)CCC1 1805,c1(CNC(C23CC(NC(C(C(C)C)OCC)=O)(C2)C3)=O)cc(OC)nc(C)c1 1806,N1(C(C2(O)CCCC2)=O)CCCCC1C(=O)Nc1nccc(C(F)(F)F)n1 1807,N1(C(COCC(C)C)=O)CC(CNC(c2csc(Cl)n2)=O)OC(C(F)(F)F)C1 1808,C(C1CN(C(c2cc(C(N)=O)co2)=O)CC1C(N1CCC(C(N)=O)C1)=O)=CC 1809,c1(CC(=O)NC2CN(C(=O)C(O)CC(F)F)CC2O)cnc2ccccc2c1 1810,CC(O)C(C)(C)C(=O)NCCOCCNC(=O)C(Cl)=CCl 1811,C=CCCC(c1nnnn1-c1ccccc1Cl)(C1CC1)NC(C)CCC(=C)C 1812,c1(CN2CC3C(C(=O)NCc4cscn4)C3C2)cccc2cccnc12 1813,c1(C(=O)NCC(CN(C(=O)CC2(O)CC2)C)O)n[nH]cc1-c1ccccc1 1814,c1(C(=O)NC2COCCN(Cc3cccc(OC)c3)C2)n[nH]c2cc(Br)ccc12 1815,N1(C(COCCCCC)=O)CCC(CNC(=O)C=CI)C(C)C1 1816,C1(NC(C(C)(C)c2ncco2)=O)CC2CC(NC(c3ccc(F)s3)=O)CC2C1 1817,C1(C(N2CC(C(=O)NC(C)C(C)(C)C#N)OCC2)=O)CC2CC(=O)C1O2 1818,c1(NCC2C(C)CN(C(C3CCCC3C)=O)C2)ncnc2c1nnn2CC1CC1 1819,C1(NC(COCCCC#C)=O)CC2(C1)CC2NC(=O)CCCOC1CCCCC1 1820,c1(CC)ccc(C=CC(N2CCCC2CN(C(=O)Cc2ncc(C)o2)C)=O)cc1 1821,N1(C(c2cc(OC)n[nH]2)=O)CCC(C)(CNC(C2CCC(=O)CC2C)=O)CC1 1822,C(=O)(C(C(C)CCC=C(C)C=CC#N)N1CCC(OC(=O)NC2(C)CC2)CC1)OC 1823,C1(OC)CC(NC(c2occc2CNC(=O)CNc2ncccn2)=O)CC1OC 1824,Cc1cc(N2CCC(NC(C3C(F)(F)C34CCC4)=O)C2C)n2nc(C)nc2n1 1825,C(=O)(CS(=O)(=O)C1CC1)NCC(CCNC(c1c(C(=O)OC)nn(C)c1)=O)(C)C 1826,C(=O)(C1=CCC2(COC2)OC1)N(C1CCC(NC(C2(CC)CCOCC2)=O)C1)C 1827,C1(CNC(c2cnc(OC)nc2)=O)COCCN(C(=O)C(C)SC(F)(F)F)C1 1828,c1(C(=O)NCC(C)(C)NC(Cc2c(C)noc2)=O)cnc2c(c1)nnn2C 1829,C1(CNC(C(CC)C)=O)COC(C)(C)CN1C(c1cnc(SC)nc1O)=O 1830,C12(NC(Cc3cc(C)no3)=O)CCCCCC1N(C(C1CC(=O)C1)=O)CC2 1831,c1(C(=O)NC2CC(NC(c3scc(OC)c3OC)=O)C2)c(C(C)C)cccc1C 1832,CC1CCCCN1C(=O)CCNC(=O)C(=O)Nc1nc(-c2ccc(F)cc2)cs1 1833,c1(C(=O)NCC2CC2CNC(C2CC(O)(c3ccccc3)C2)=O)ccc(O)cn1 1834,C(C(C)CC(=O)NC(CNC(=O)COC(C)(C)C(F)(F)F)C1CC1)SC 1835,C1(NC(CCc2nc(C)c(C)o2)=O)CC2CC(NC(C3OCCC3(C)C)=O)CC12 1836,C=CC(CCC)CC(=O)NC(COC)C(=O)N(CCCCC)C(C)C 1837,C(CC(O)CNC(=O)C(Cn1ccnn1)NC(=O)CC1(O)CCOC1)OC 1838,Cc1ccc(C(=O)NC2CCCC(N(C)C(c3nocc3Cl)=O)C2)c(F)c1 1839,CC(CC(=O)N(C1CCCN(C(=O)CCN2CCC2)C1)C)C(F)F 1840,c1(NC(C2CN(C(c3cnc(Cl)nc3)=O)CCC2O)=O)cc2c[nH]nc2cc1Br 1841,c1(C(C)=O)cn(CC(N2CC(C)(OCC(=O)NC3CCCCS3)C2)=O)nn1 1842,c1(OCC(=O)NC(CNC(C2(CC)CCCC2)=O)(C)C2CC2)ccc(F)cn1 1843,c1(C(N2CCC(CCNC(=O)C=CC3CCCC3)C2)=O)cccc([N+](=O)[O-])c1O 1844,N1(C(CCc2n(C)cnn2)=O)CC2CC2(NC(=O)CCC2CCCOC2)C1 1845,c1(CC(N2C(CNC(C(C)C3CC3)=O)CCC2)=O)cc(O)ccc1Br 1846,C1(OC)CN(C(C2(CSC)CC2)=O)CCC1NC(=O)C(O)CCSC 1847,c1(C2C(C(N(CC(C)(C)C)Cc3csnn3)=O)C2)ccccc1 1848,Cc1nc(C(N2CC3(NC(c4cnoc4C)=O)CC2C3)=O)ccc1C#N 1849,CC1CCCCCN1C(=O)Nc1ccccc1-c1ccc(Cl)c(F)c1 1850,C1(C(N2C3(CN(C(C(CCC)CC)=O)C3)CC2)=O)Cc2ccccc2C(C)(C)C1 1851,Cc1cc(C(N2CCC(C(=O)NCC3CCCC3O)(CF)C2)=O)ncc1N 1852,C1(NC(N(CCN(C(C(C2CCCC2)NC(C)=O)=O)C)C)=O)CCC2CC1CO2 1853,Cc1cc(C)c(CN2CC(F)CC2C(=O)Nc2cccc(F)c2CO)cc1C 1854,c1(C(N(C2CN(C(=O)Cn3cc(Cl)cn3)C2)C)=O)cc(C(F)F)cs1 1855,Cc1cc(S(=O)(=O)NC(C)CCCCCO)c(C)cc1-c1cccnc1Cl 1856,CC1(CNC(=O)CCc2ncccn2)CCN(C(C2CC(n3ccnc3)C2)=O)C1 1857,C(=O)(CC1C(=O)Nc2ccccc21)NC(C)C(CO)NC(=O)Cc1csc(Cl)n1 1858,C(=O)(CC(F)(F)CS(C)(=O)=O)NCC(CNC(C(CC#C)C1CC1)=O)C 1859,N1(C(C)=O)CCC(C2OCCC2NC(=O)C=C(C)C(C)C)CC1 1860,C12(C(=O)NCCCNC(C3(c4ccc(Cl)cc4)CCC3)=O)C=CC(CC1)C2 1861,C(C)(CC(=O)NCC(C1CC1)NC(=O)CC#N)(C(F)(F)F)N(C)C 1862,n1(C(C=C)C)nc(C2CCOC2)nc1-c1cncn1-c1ccccc1 1863,c1(CC)cc(C(N2CCCC2C(N2CC(CC(=O)OC)C2)=O)=O)ccn1 1864,c1(C(N(C2C(C)CN(C(C34CC(F)(C3)C4)=O)CC2)C)=O)ccnc2cc[nH]c12 1865,Cn1cc(CNC(C2CC=CCN2C(=O)C(O)CC2CCCC2)=O)ccc1=O 1866,Cc1cnsc1C(=O)N(CC(C)C(=O)NC1CC(CF)C1)C 1867,CCCCC(CNC(C1(C(=O)NC)CC1)=O)NC(=O)C(N1CCN(C)CC1)C 1868,c1(N(C2CSC2)CC)nnc(-c2cc(-c3ccc(N4CCCC4)cc3)[nH]n2)n1C 1869,CCCC(C)CC(=O)NC1CCCC(NC(c2c(C)nc(C)n2O)=O)C1 1870,CC1=NOC(C(=O)N(CCNC(=O)C(n2ccc(C)n2)C)CCOCCO)C1 1871,c1(C(N2CC(NC(C(C)(C(C)C)OC)=O)C2)=O)c(C)nc(C(C)(C)C)nc1O 1872,c1(C(N2CCC(C)(NC(COC)=O)CC2)=O)nccc2cnn(C)c12 1873,c1(C(=O)NC23C(CN(C(C4CC(=O)N(O)C4)=O)C2)CC3)sc2sccc2c1Cl 1874,C1(NC(c2ccc(CN(CCC)C)o2)=O)CCCN(C(=O)CCN(C)C(C)=O)C1 1875,c1(CC)ccc(C(=O)NC(COC)C(=O)NCC(=O)NCC(F)F)o1 1876,c1(C(N2Cc3[nH]nc(-c4cccc(OC(F)F)c4F)c3C2)=O)ccc2ncsc2c1 1877,Cc1ccc(=O)n(CC(=O)NCC2CC2NC(=O)COC2(C)CCCC2)n1 1878,C1(NC(c2c(OC)cccn2)=O)CCCC12CN(C(=O)CC(C)c1ccco1)C2 1879,O=C(C1=CCCN(C(C2CCC2(F)F)=O)C1)NC(C(F)(F)F)C1CC1 1880,C12(NC(C(C)NC(=O)CC3C=CCC3)=O)CC1CN(C(=O)C(C)(Cl)Cl)C2 1881,n1(CCC(=O)NC2CC(NC(CN3CC(C)(OC)C3)=O)C2)c(C)cc(O)cc1=O 1882,c1(OC)ccc(O)cc1C(N1CC=C(CNC(C2(OC)CC2)=O)CC1)=O 1883,CC1CCN(C(c2cc(C(C)(C)C)no2)=O)CCN1C(C1CC1C(F)F)=O 1884,CN1CC(C(=O)NC(C)(C)CC=CC(=O)NCCOC2CCCC2)NC1=O 1885,c1(C(=O)NC(C(=O)OC(C)(C)C)Cc2ccccc2)noc2c1CCCCC2 1886,N1(CC(=O)Nc2ccccc2)CC2(CCC(CNC(C34CCCCC3C4)=O)O2)C1 1887,C1(NC(c2c(C)n(C(C)C)cc2)=O)CCN(C(=O)CCC2CCOC2)CC1O 1888,N1(C(c2c(CC)nc[nH]2)=O)CCCC(O)(CCNC(c2cnc(C3CC3)[nH]2)=O)C1 1889,c1(C(C(C)C)NC(=O)NCC2CS(=O)(=O)C2)ccc(Cl)cc1 1890,N1(C(=O)CN2CCOCC2)CCC(C(=O)N(C2CC2)CC2CCCCO2)C(O)C1 1891,C(=O)(C(C)(C)C(C)C)NCC(C)N(C(C1N(C(CCC)=O)CCCC1)=O)C 1892,C1(C(=O)NC(=O)C2CC2)CCOC(=O)CC1.CC(C(=O)NCCN)NC(C1CCC1)=O 1893,CC1CCN(C(=O)Nc2cnn(C(C)(C)C)c2)C1C 1894,CCCC(CNC(c1ccn(CC)n1)=O)C(=O)NCC(F)(F)C(C)(C)O 1895,c1(C(=O)NCC2COC(CNC(c3cc(Cl)no3)=O)C2)cccc(CO)n1 1896,CC(C)(C)C(=O)NCC(=O)NCC1CCCN1C(=O)Cc1ncc(Cl)s1 1897,Cc1sc(-c2nc[nH]n2)nc1C(=O)NCC1CCCCN1C(=O)CNS(N)(=O)=O 1898,C1(C(N2CCC(CNC(c3c(CC)noc3)=O)CC2)=O)CC1C1CCCC1 1899,CC1CCC(NC(=O)OC(C)(C)C)CN1C(c1ccoc1I)=O 1900,c1(C(N2CCN(C(c3ccc(C)cc3)=O)C3C2C3)=O)ccnc2ccnn12 1901,c1(C(C)NC(C2CC=CC2)=O)ccc(CNC(C2(c3cccs3)CC2)=O)cc1 1902,c1(OC)ccc(C(N2CC(OC)C(NC(=O)CSC(C)C)C2)=O)c(N)c1Br 1903,C1(NC(c2cccc(OC)c2)=O)CCN(C(c2cn(C)nc2SC)=O)C1(C)C 1904,CCCC(O)CC(=O)N1CCC(C(C)(C)C)(CNC(=O)CCS(C)(=O)=O)C1 1905,CC(C)S(=O)(=O)CC(=O)N1CC(OCCC(=O)NC2CC3(C2)CC3F)C1 1906,CCC(C)(COC)CNC(C1CCN(C(=O)CCCCN(C)C)C1C)=O 1907,N1(C(C=Cc2ccc(C)o2)=O)CCCC(NC(C2(N(C)C)CCC2)=O)C1C 1908,N1(C(COCC(=C)C)=O)CCC(N(C)Cc2cncs2)CC1 1909,N1(C(c2cc(Cl)cc(Cl)c2O)=O)CCC2CCN(C(C34CCC(CC3)O4)=O)CC12 1910,C1(C)(C(N(CC(CNC(c2c(C)n(C3CC3)nc2)=O)(C)C)C)=O)COC(C)CO1 1911,CC1(C)CC(NC(=O)NCC(C)(F)C(C)(C)F)c2ccccc2O1 1912,C(C)(C(=O)N(CC(C)(C)CNC(=O)CC(C)C1CC1)C)(C(C)C)NC(C)=O 1913,C(=O)(CC(C)(O)COC)NC1CCN(C(c2c(N(CC)CC)nccc2)=O)C1C 1914,n1(CC)cnc2c(NC(C)CCCO)[nH]c(=NCCCCCN3CCCC3)nc12 1915,Cc1ccc(CC(=O)NC2CCC2NC(c2cccs2)=O)s1 1916,N1(C(COC)C)CCC(C)C(NC(C2CCCN(CC(C)(C)C)C2=O)=O)C1 1917,Cc1ccc(C)c(C(=O)NCC(CC(C)C)NC(c2cccnc2)=O)c1O 1918,C1(NC(CCOCC)=O)CCC2(CCN(C(c3ccsc3C#N)=O)CC2)C1 1919,c1(C(N2CCC(O)(CC(N3CCC(C#N)CC3)=O)CC2)=O)c(Cl)cc(Br)cc1Cl 1920,C(CN=c1nc(SC)cc[nH]1)C1CCN(C(c2cc(C)nc(O)c2)=O)CC1 1921,C1(C(N(CCCNC(C(C)Cc2ccco2)=O)C2CC2)=O)(C(F)F)CCCCC1 1922,N1(C(CC2CCN(C)CC2)=O)CC(NC(C2CC2c2ccncc2)=O)CC(O)C1 1923,c1(C(=O)NCCCN(C)C(C2CCCS2)=O)cc(S(=O)(=O)N2CCOCC2)c[nH]1 1924,C1(NC(c2c(C(N)=O)csc2)=O)CS(=O)(=O)C2CN(C(c3cnns3)=O)CC12 1925,c1(C(=O)NC2CC(CCNC(CC3(OC)CCC3)=O)C2)cncnc1C 1926,c1(CC)cnoc1C(=O)NC1CC(C)(NC(=O)C(C)C2CCCO2)C1 1927,N(C(=NCC(C)C)NC1CCCC1CNS(C)(=O)=O)Cc1cc(C)nc(C)n1 1928,CC(C)(CNC(c1sccc1F)c1nnnn1C1CCOC1)CC(F)F 1929,N1(C(CCSCCC)=O)CC(CO)C2(C1)CN(C(C1(C(F)F)CCCCC1)=O)C2 1930,C(CCC(C)(C)NC(C1CC1C(C)(C)O)=O)NC(COCCOCC)=O 1931,CC1OCCCC1C(=O)NC(C1CN(C(C2CCCN2C=O)=O)CCO1)C 1932,CCC(CC)(CO)C(=O)N(C)CC1(CNC(C2CCC3CCC23)=O)CC1 1933,Cc1cnc2c(C(N3CC4CCC4(NC(=O)Cc4cscn4)C3)=O)cccn12 1934,C1(C)(CNC(c2n(CCOCC)nnn2)c2cscc2Cl)CC2(C1)CC2(F)F 1935,N1(C(C2N(C(c3ccc(OC)nn3)=O)CC3C2C3(C)C)=O)CCC(O)C(F)(F)C1 1936,C1(C)(C(=O)Nc2cccc(NC(C3(C)CC(C)OCC3)=O)c2)CCCCC1(F)F 1937,c1(C(N(CC(C)NC(=O)CCC2CCCC2)C)=O)ccc(N)c(Cl)c1 1938,c1(NC(=O)Nc2ccc(C(=O)NCC(N3CCCC3)C)cc2)cc(Cl)nnc1O 1939,c1(OC)ccccc1C(C)C(=O)N(C1CN(C(c2c(Cl)nsc2Cl)=O)C1)C 1940,c1(C(=O)NCCOC2CN(C(c3c(C)oc(Cl)n3)=O)C2)ccc2c(c1)CC(=O)N2 1941,c1(CN(C(CC)C)C(C2CCCC23CC3)=O)ccc(F)cc1 1942,c1(OC)ccc(S(C)(=O)=O)cc1C(N1CC2CCC(C1)N2C(C1C(C)C1C)=O)=O 1943,c1(OC)nc(C)cc2ccc(C(=O)NC(C)CN(C)C(C3C=CCCC3)=O)cc12 1944,c1(C(=O)NC2CC(NC(C=CC3(C)COC3)=O)CC2O)cc2cnccc2o1 1945,C1(CN(C)C(c2ccc(C(C)(C)C)nc2)=O)CCN(C(=O)C(F)(F)CF)CC1 1946,C1(CNC(C(CSC)O)=O)CN(C(c2ccc3nccn3c2)=O)CCC12CCC2 1947,Cc1scc(C(=O)NCC(c2ccc(F)cc2)NC(c2nnsc2C)=O)c1C 1948,CC1CCC=C1C(=O)N1CCC(NC(=O)CN2CC(=O)N(C)C2=O)C12CC2 1949,Cc1cc(F)c(C(=O)NC2CCCCC2CNC(c2ncccn2)=O)c(Br)c1 1950,c1(C(=O)NC2CCN(C(C(CC=C)C)=O)CC2OC)c(F)ccc2occc12 1951,C12(NC(C(CC(C)C)OC)=O)CCCC1CN(C(c1c(C)ncn1OC)=O)C2 1952,C1(NC(=O)Nc2cccc(C3CC3)c2)C2Cc3cc(Br)ccc3C12 1953,c1(OC)ccnc(O)c1C(=O)NCC(C)N(C)C(c1cc(CO)[nH]n1)=O 1954,CC(C)(CCCCNC(=O)C(O)C1CC1)NC(c1cc(Cl)n[nH]1)=O 1955,C(=O)(C1CCCn2ccnc21)NCC.C(=O)(C(C)(C)OC)N(CCC)CCN 1956,c1(NCC(C(C)C)OC)ccc(S(=O)(=O)N(C)Cc2ccnc(SC)c2)c(Cl)c1 1957,C1(C(N2C(C(=O)OC)C=CC2)=O)N(C(=O)Cc2ccc[nH]2)CCCC1(C)C 1958,c1(C(N2C(C)(CNC(=O)C(F)CC3CC3)CCC2)=O)cccc2c1NCCC2 1959,N#Cc1sc(=NC2(C3CN(C(c4n[nH]c5ccccc45)=O)C3)CC2)[nH]c1Cl 1960,c1(C(N(CCCNC(C=C(C)C)=O)C(C)C)=O)nncn1C1CC1 1961,C1(OC)(CNC(C2CC(n3cnnc3)C2)=O)CCN(C(=O)C(C)(CO)OC)CC1 1962,C1(CCNC(=O)C(O)C2CC2)CCCCN1C(C1CCC(O)CC1)=O 1963,c1(C(N(C)Cc2cc(OC)no2)=O)cc2ccncc2c(O)n1 1964,S(=O)(=O)(c1ccc(NCc2ccn(C3CC3)n2)cc1Cl)NC(c1cnoc1)C 1965,C1(NC(C2C(CC)C2)=O)CCN(C(=O)C(Cc2ccccc2)N(C)C)CC1(C)C 1966,c1(OCC=C)ccc(CC(=O)NC2CC(C)(NC(C3CCCC3(F)F)=O)C2)cc1 1967,N1(C(C(CC)OC)=O)CCC(C2(NC(c3nc(O)nc(O)c3OC)=O)CC2)C1 1968,C1(C(N2CCC(CCc3cn(C(C)(C)C)nn3)CC2)=O)CCc2ccccc2C1 1969,C1(C(=O)NCC2CN(C(=O)CCc3ccsc3)CCO2)CCc2nncn2CC1 1970,C(=O)(C(C)(CC)CO)NCC(N1CCN(C(C=CC)=O)CC1)C(F)F 1971,C(CCN=c1nc2c(c[nH]1)CCCC2)OCCNC(=O)CN1CCCCC(O)C1=O 1972,N1(C(CC2(N(C)C)CCCC2)=O)CC2CCCC1C2CNC(C1CC=CC1)=O 1973,CC1(C)CN(C(c2cccnc2)=O)CC(CNC(=O)Cc2ccc(F)cc2Cl)O1 1974,Cc1cnc(NCCC2CCS(=O)(=O)C2)c(S(=O)(=O)NCCCCCF)c1 1975,C1(NC(C(COC)(C)C)=O)CCN(C(=O)C(C)OCC(C)C)C12CC2 1976,N1(C(C2(C(F)(F)F)CC=CCO2)=O)CCN(c2ccccc2OC(F)F)CC1 1977,c1(C(=O)NCC2CCN(C(C3CN(CCC)C(=O)C3)=O)CC2)cc(C#N)[nH]c1C 1978,C(CC(=O)N1CC2(CCCC2)C1)(C(F)F)NC(C1CC2(CCC2)C1)=O 1979,c1(NC(N2C(C)CN(Cc3ccc(Cl)c(Cl)c3)CC2)=O)cn2cccnc2n1 1980,C=C(C)CCCC(=O)NC(C)Cn1cc(CN(C(C)C)C(C)C)nn1 1981,N1(C(C=C2CCN(C)CC2)=O)CC2CN(C(=O)CC3CCCO3)CC2C1 1982,C1(NC(CC(C=C)C)=O)CC2CC1N(C(c1cnc(C(C)(C)C)o1)=O)C2 1983,CN1CCN(CCOCC=O)N1CCCCC(=O)OC(F)F 1984,C12(C(=O)NC3CCCN(C(c4[nH]cc(C)c4)=O)CC3)CCCC(CCC1)C2 1985,CCCCC(O)CC(=O)NC1CCCN(C(=O)C(C)(C)C(C)C)CC1 1986,C12(C(=O)NC(C(C)C(=O)N(CCC(O)CO)C)C)CCC(CC1F)C2 1987,N1(C(C2(C=C)CCCCC2)=O)CC2CCC1CN2C(C1CC1(C)C)=O 1988,N1(C(Cc2n(C)nnc2)=O)CCC(CNC(C2CNC(=O)C2)=O)C12CC2 1989,C1(C(=O)NC2C(CNC(c3sc(CCC)c(COC)c3)=O)C2)C(C2CC2)C1(F)F 1990,N1(C(CC(=C)C)=O)CC(C(=O)NC(c2nccc(=N)[nH]2)C)C(F)(F)C1 1991,C=CCCCCCCC(=O)NC1CCCCN(C(=O)C(C)C(O)CC)C1 1992,N1(C(Cc2n(C)nnc2)=O)CCCCC(Nc2nccc(C#N)n2)C1 1993,C1(C(N2CC(CN(C)C(C3SC4C=CC3CC4)=O)C2)=O)C2(CCC2)C12CCC2 1994,n1(C(C)C)cc(CC(=O)NC2CCCC2NC(=O)CCOC2CCCCC2)nn1 1995,c1(C(=O)NC(C2CCOC2)CNC(=O)Cn2ccnn2)ccc(O)c(Br)c1 1996,C1(NC(C(C#C)(C)C)=O)CC2CCC1CN(C(C1CCC(F)CC1)=O)C2 1997,c1(C(=O)NCCC2(C)CCN(C(C34OC(C)C(C3)C4)=O)C2)cccc2occc12 1998,C1(c2nnnn2CCCF)(NCCc2ccc(C(C)C)s2)CSC(C(C)(C)C)C1 1999,n1(CCC)ncc(C(N2CC(NC(=O)CCc3cnco3)C3CC23)=O)c1C 2000,c1(C(=O)NCC(C2CCC2)NC(c2csc(Cl)n2)=O)ccc([N+](=O)[O-])cn1 2001,C12(NC(C3CC3[N+](=O)[O-])=O)CCC(C1)N(C(=O)CNc1ccc(C(F)(F)F)cn1)C2 2002,C12(CNC(CC(=O)OCCC(C)C)=O)CN(C(=O)C(F)=CC3CC3)CC1CCO2 2003,N1(C(CC2N(C(CC(C)C(F)F)=O)C3C2CCC3)=O)CCC2(CCC(O)C2)C1 2004,C1(NC(C2CCC(CC)O2)=O)(CO)CCN(C(=O)CCN2CCC2)C1 2005,Cc1ncnc(C)c1CC(=O)NCCCNC(C1CC2(F)CC1C2)=O 2006,c1(C(N2C(C(=O)NC(CC=C)CO)CCC2)=O)ccc(Cl)nc1F 2007,Nc1cc(C(N2CCCC2C2(NC(=O)C3=COCCC3)CC2)=O)cc(Br)n1 2008,C1(CNC(CSC(C)C)=O)CCN(C(=O)CN2CCC(C)C2)C1 2009,C1(CC(=O)N(CCn2cc(-c3ccncc3)nn2)CC2(O)CC2)CC2COCC12 2010,N1(C(C2C3(CCN(C(C4(CCCC)CCC4)=O)C3)C2)=O)CCC(C2(C)CC2)CC1 2011,c1(C(N(C2COC3(CCNCC3)C2)c2cc(C)[nH]n2)=O)cc2c(Cl)cccc2s1 2012,N1(C(C2C(CC)CCN2C(c2cc(C3CC3)[nH]n2)=O)=O)CCc2oc(C)nc2C1 2013,C1(NC(C=CCOC)=O)CCCCC12CCN(C(=O)C(O)C(C)CC)C2 2014,c1(OCC(=O)N(CCC(C)(C)NC(c2ccsc2Cl)=O)C)ccccc1C(N)=O 2015,CCC(CCC(=O)N1CCOCC1C(N1CCC(OC)C1C(C)C)=O)OC 2016,C1(NC(C(c2ccnn2C)C)=O)CCOCC1C(=O)NCc1cccnc1O 2017,C(=O)(CCC(C)(C)c1ccccc1)N(C(c1ccc(F)cc1)(C)C(=O)O)C 2018,C(=O)(C(O)C1=CCCCC1)N(CC(=O)NC(CCC(C)C)C)C 2019,N1(C(c2c(OC(F)F)cc(C)s2)=O)CC(NC(c2ccnc(O)c2)=O)C(C#N)C1 2020,c1(-c2c(C)n[nH]c2)cccc2c1CN(C(=O)Nc1ccc(Cl)cc1)CC2 2021,c1(NC2C(NC(c3cccc4nc(O)[nH]c34)=O)CC2)ncc(Cl)cc1[N+](=O)[O-] 2022,CCCC(O)CC(=O)NC(CNC(c1cc(N2CCCC2)ncn1)=O)CCOC 2023,Cc1cccn2cc(C(=O)NCC3(NC(=O)C(O)P(C)(C)=O)CC3)cc12 2024,C(=O)(C(C)C(CC)CC)N1CC(CC(NCP(OCC)(C)=O)=O)C2(C1)CC2 2025,c1(C(N2CC(CC(C)NC(c3cccn3C)=O)C2)=O)ccc(CC2CC2)o1 2026,c1(NC(C2(NC(C3CC(Cl)(Cl)C3)=O)CCSC2)=O)cccc(F)c1 2027,C=C=C(C)CC(=O)NC(C(=O)NCCC1CC2C=CC1C2)c1cccs1 2028,CC(N=c1ccnc(Cl)[nH]1)C1CCN(C(=O)C(C)Cc2ccccc2)C1 2029,C1(C(N2CCC(NC(c3c(C)ocn3)=O)C(O)C2)=O)CCc2ccc(F)cc2C1 2030,c1(C(N2CCC(N(C(c3cc(C)cc(O)n3)=O)C)C2)=O)ccc2c(c1)N(C)CC2 2031,Cn1cc(C(N)=O)c(=NC(=O)C2CCC(NS(=O)(=O)c3ccccc3Br)CC2)[nH]1 2032,C1(OC)(CNC(=O)Cn2cc(Br)cn2)CCN(C(C23COCC2C3)=O)CC1 2033,C1(C(=O)NC(c2nccc(O)n2)C)C=CCN(C(=O)Cn2ccnc2)C1 2034,C=CCCC(F)(F)C(=O)NC1CN(C(c2cc3ccccc3s2)=O)C1 2035,Cc1nc2cc(C(=O)NC(C)CCNC(C3CC(C)CC(=O)N3)=O)[nH]c2s1 2036,C(C(C)C(=O)NCCCC1(NC(C2CCC(=O)C2)=O)CC1)OC 2037,C1(C(=O)NC(C)CNC(=O)Cn2cnnc2)CCCCC12CCC2 2038,N1(C(Cc2c(C)n[nH]c2C)=O)CCCC(C)(C(=O)NCC2COC(=O)N2)C1 2039,C1(CNC(c2n(C)c(S)nn2)=O)CCN(C(=O)Cn2cc([N+](=O)[O-])cn2)C12CC2 2040,c1(C(=O)NCCC(C)(C)NC(C(C)NC(COC)=O)=O)cnn(C)c1Cl 2041,C1(NC(C(C(COC)C)C)=O)CCCC12CCN(C(=O)Cn1nnc(=N)[nH]1)CC2 2042,C1(C(N(C)CC2COCCN2C(c2n[nH]cc2Br)=O)=O)CCC2(CCC2)O1 2043,c1(CC)ccc(NC(=O)CC2COC(CNC(=O)OC(C)(C)C)C2)cc1Br 2044,C1(NC(COCC)=O)CCN(C(C2C=CCCC2)=O)CC1OC 2045,C1(NC(C2CC(CNC(C3(CC)CCCC3)=O)C2)=O)CN2CCCC1C2 2046,c1(N2C(C)C(N(C)C)CC2)ccc(S(=O)(=O)NCCCc2cnoc2)cn1 2047,C1(C(N(CCC(=O)Nc2cnsc2)C2CC2)=O)C=CCCC1 2048,c1(OC)ccc(C(=O)NCCNC(C2CCCN(C(C3CC3[N+](=O)[O-])=O)C2)=O)cc1 2049,c1(OCC)c(Cl)cc(NC(c2ccc([N+](=O)[O-])o2)=O)cc1Cl 2050,O=C1COC(C(=O)NCc2cn(C3CN(C(c4ccco4)=O)C3)nn2)C1 2051,N1(C(C2CCN(C)CC2)=O)CCC(NC(=O)CO)C(F)(F)CC1 2052,N1(C(c2c(CC)nco2)=O)CC2CCC2(NC(=O)CC2CCC(=O)N2C)C1 2053,c1(C(=O)NC2CC3CN(C(CCCC(C)O)=O)CC32)ccc(Cl)c2occc12 2054,N1(C(CC(C)(C)O)=O)CCN(C(=O)C=Cc2ccccn2)CC1C1CCCC1 2055,C1(CNC(=O)COc2ccccc2)CCC(NC(C2CC2C2CC2)=O)CC1 2056,CCCC(C)CC(=O)N(C1CCCN(C(c2sc(CSC)nc2C)=O)C1)CCF 2057,C1(CNC(c2cc(C)sn2)=O)CCCCN(C(c2cc3[nH]ccc3s2)=O)C1 2058,c1(CC(=O)NCCNC(c2c(Cl)csc2Cl)=O)ccc2cccnc2c1 2059,c1(C(=O)NCCSCCC(F)(F)F)cnc2c(Br)cc(Br)cc2c1 2060,C1(C(NOCCCC#C)=O)CCCN(C(=O)CSc2cccc(C)c2)C1 2061,C(CC1=CCCCC1)NC(C(C(C)NC(c1c(C)oc(Cl)n1)=O)C)=O 2062,N1(C(CCCOCCC)=O)CCCC2CN(C(C3(F)CC34CCCCC4)=O)CC12 2063,c1(C(=O)NCCCCCNC(c2c[nH]c(=O)cn2)=O)cccc2cnccc12 2064,C=CCC(CNC(c1ccn(Cc2ccccc2)c1)c1nnnn1C)CC(C)C 2065,C(=O)(CS(=O)(=O)C1CC1)NCCOC1CN(C(Cc2c(OC)c(F)ccc2)=O)C1 2066,C1(CC)CCCN(C(c2ccc(OC)s2)=O)C1C(=O)NC(C12CCC(CO1)C2)C 2067,c1(CCC)c(C(N2CC(O)(C(C)NC(=O)CNS(=O)(=O)CC)C2)=O)nnn1CC 2068,c1(CC)nnsc1C(=O)NC1CN(C(=O)CCc2ncccn2)C1 2069,c1(C(=O)NC2C3CC(NC(C4C(=O)NCC4)=O)CC32)ccc2[nH]ccc2c1 2070,C12(NC(c3cnns3)=O)CCN(C(=O)CCc3cncc(Br)c3)CC1C2 2071,N1(C(c2nn(CC)c(C3CC3)c2)=O)CCN(C(=O)C=C(C)Cl)CC1CO 2072,c12c(Cl)ccc-1c2F.N1(C(c2cc(Br)c[nH]2)=O)CCN(c2ccnc(O)c2)CC1 2073,c1(CNc2ccc(OCC=C)cc2)cnc(OC)cc1C(N1CCOC2CC12)=O 2074,N1(C(C(CC)SC)=O)CCN(C(=O)CCCn2cncn2)CC1COC 2075,C=CCC(CC)C(=O)NCC1CN(C(c2nnn(C(C)C)c2C)=O)CCN1C 2076,c1(C(N2CCC(C(C)NC(C3CN4CCC3C4)=O)CC2)=O)cn2ccccc2n1 2077,C1(C(=O)NC(CN(C(C2(C)ON=C(C)C2)=O)C)(CO)CO)CC2CC1CC2O 2078,CS(=O)(=O)c1ccccc1C1=CCN(CC(C2CCCCC2)CBr)CC1 2079,C(C(=O)NCCCC1CC1)(c1ccns1)N(CCN(C)C)CC1CCC1 2080,C1(NC(c2cc(CC)sc2)=O)C=CCN(C(=O)COc2ccccc2)C1 2081,c1(CC)ccc(N)c(C(=O)NC2CN(C(=O)C(O)CC)CCC2C(F)(F)F)c1 2082,Cn1ncnc1C(=O)NCCNC(=O)CC1OCCO1 2083,O(C=CC(=O)N(C1CN(C(=O)CCc2ccc(Br)s2)C1)C)CC 2084,c1(CNC(=O)NC23COC(CCO2)C3)ccc(S(=O)(=O)C2CCCC2)cc1 2085,C=Cc1cnn(C)c1C(N1CCC(N(C(c2cc(OC)ccc2F)=O)CC)C1)=O 2086,C1(CNC(=O)NCCS(N)(=O)=O)(Cc2nccc(C(F)(F)F)n2)CC2(CCC2)C1 2087,N1(C(C2(OC)CCOC2)=O)CC2=C(C1)CN(C(=O)C(c1cncnc1)C)C2 2088,N1(C(c2cc(C)[nH]n2)=O)CCC(C(=O)N(C)CCn2ccnc2C)C(C)C1 2089,C1(NC(C2C(C)C2)=O)CCCCC1NC(=O)CCOc1cccnc1 2090,N(C1CCCOc2c(Br)cccc21)C1CCCN(C(=O)OC(C)(C)C)C1 2091,C12(CC(=O)NCC3(F)CN(C(C4C(C)C4)=O)C3)CCCN1CCC2 2092,C(C(C)(C)C)N(CCCC1CCC1)CCN(CCC)CCOC 2093,c1(C(CC(N2CCC(N(C(C3CN(C4COC4)C3)=O)CC)C2)=O)C)c(C)noc1C 2094,n1(CC(N2C3C(NC(COCC)=O)C(CC3)C2)=O)nc2ccccn2c1=O 2095,c1(C(=O)NCC(CN(C(=O)COc2ccsc2)CC)O)cc(C)n(C2CC2)c1C 2096,c1(C(=O)OC)nccc(NCC(N2CCCC2CNC(N)=O)=O)n1 2097,c1(COC)cccc(S(=O)(=O)NC(CCc2ccccc2)C(F)F)c1 2098,c1(C(N2C(CNC(CC(CC)C)=O)CCCC2)=O)cnc2sc(C)nc2c1 2099,CCCC(CC(=O)N1CCC(C(N)=O)(OC)C1)NC(C1(n2nccn2)CC1)=O 2100,Cc1cc(C(N2CC3CC(C(N4CC=CC4CF)=O)(C3)C2)=O)cc(O)c1 2101,Cc1nccnc1C(=O)NCC1(C(C)NC(C2CN(C(C)C)CCO2)=O)CC1 2102,c1(C(N2CCC(C#N)(NC(C3CCOCC3)=O)C2)=O)cc(O)c(O)c(O)c1 2103,CC1CC(C(=O)N(CCCO)CCCO)N(Cc2ccc(-c3cccs3)cc2)C1 2104,C1(NC(C(C=C)O)=O)CN(C(=O)CCc2cn(C)nc2C)C2(CCOCC2)C1 2105,C1(NC(C2N(C(=O)OCC)C(CO)CC2)=O)CCN(C)C(=O)C1 2106,CCCCC(O)C(C)C(=O)N(C(C)C(=O)NCCOC1(C)CCC1)C1CC1 2107,c12c(nc3ccccn13)n1cc2nn1.N1(c2ccnc(Br)n2)CCC(O)C(C)C1.CC 2108,c1(C(N2CCC3(NC(=O)Cc4cnns4)C(C2)C3)=O)ccc2sccc2c1 2109,CCCCC(C)C(=O)NCc1csc(C(=O)NC(c2ccc(O)cc2)C)c1 2110,c1(C(N2C(C3(NC(CC(C)F)=O)CC3)CCC2)=O)ccc(OCCF)cn1 2111,Cc1c(C(=O)NC2CC(NC(c3cc(Cl)cc(Cl)c3)=O)C2)c[nH]c2nccc1-2 2112,Cc1ccc(OC(C)C(=O)NCC2CC(F)CN2C(=O)CC=C(Cl)Cl)cc1 2113,c1(NC(=O)OCC)cn(CC(=O)NCC(C)OCCO)nn1 2114,c1(CC)ccc(C(=O)NC2(C)CCCN(C(c3cc(N)cc(O)c3)=O)C2)c(F)c1 2115,C(=O)(CC(C)CC(F)(F)F)NC(CC1CN(C(CC2(COC)CC2)=O)C1)C 2116,c1(CN)ccc(Br)cc1C(=O)NC1CCCC1CO.N12CCC(CC1)CC2=O 2117,C(=O)(C(F)C1=CCCCC1)NC1C2CN(c3nnc(C(N)=O)s3)CC21 2118,C12(COC)CCC(C(N3CCC(CNC(=O)CC(C)(F)F)C3)=O)(CO1)C2 2119,N1(C(CSc2n(C)c(S)nn2)=O)CCCC(S(=O)(=O)N(C)C)C1 2120,C1(C(N2CC(Cc3c(-c4cn(C)nn4)cccc3)C2)=O)CCC2C(C1)C2(F)F 2121,c1(C(=O)NC(C)(C)CNC(C2(C)CCC(=O)NC2)=O)ccc([N+](=O)[O-])cc1F 2122,C#Cc1ccc(NC(=O)C(C)(C)C2CCCN2C(=O)C(C)COCC)cn1 2123,N1(C(c2cncc(OC)c2)=O)CCN(C(c2cc(N)c(Cl)cn2)=O)CC(C)(F)C1 2124,N1(C(c2c(COC)ncs2)=O)CC(NC(c2cnn(C)c2C)=O)CC1C 2125,C12(CNC(C(C)C3CCC3)=O)CCCC1CN(C(c1cnc3[nH]ncc3c1)=O)C2 2126,c1(C(=O)NC(CC2CN(C(C3(CCOC)CC3)=O)C2)C)ccc(O)nc1 2127,Cc1cc(NC(C2CC2NC(c2cc(Cl)ccc2O)=O)=O)ncc1F 2128,C(=O)(C1=CCS(=O)(=O)C1)N1CC(CNC(C2(C(=O)NC)CC2)=O)C(F)(F)C1 2129,Cc1ccccc1OCCC(=O)NCC1CC(F)CN1C(=O)CC(F)(F)Cl 2130,N1(C(C2CN(CC)C(=O)N2)=O)CCN(C(c2cc(C)cs2)=O)C2COCC12 2131,C(CC(F)F)(C(=O)NCC1(O)CCN(C)C1)N(C(=O)Cn1cc(CO)nn1)C 2132,C1(CNC(C2(OC)CCOC2)=O)CN(C(=O)CC2(C)OCCO2)CCC1(C)C 2133,C(CCCCC(=O)NC1CCCC(CC)C1)=CCC 2134,C1(NC(C23COCC2C3(F)F)c2n(C3(C)CC3)nnn2)CCC=CCCC1 2135,c1(CNC(CCC(C)NC(=O)COC2CCOCC2)=O)c[nH]c2ncccc12 2136,c1(C(=O)NCC2(C)CCCN(C(C3(C)CNC(=O)C3)=O)C2)cccn2nnnc12 2137,c1(Cc2cccc(NC(N3CCC(=CC)C3)=O)c2)ccn(C)c(=O)c1 2138,N1(C(c2n(C)ncc2)=O)CCC2CCN(C(c3n[nH]c4c3CCC4)=O)CC12 2139,C12(C(=O)NCC3(OCC)CC3)CC(NC(C3CCSC3)=O)(C1)C2 2140,c1(C(=O)NC2CC3(C(C(N(C4CC(=C)C4)C)=O)C3)C2)ccc(C#N)cn1 2141,N1(C(C(C=CCCC)O)=O)CCCCC(NC(c2ccc(SCCC)cc2)=O)C1 2142,CCC(C)(COC)C(=O)NC(C(=O)N(C)CC1(COC)CCC1)C(C)C 2143,C(=O)(C1=CSCS1)NCCCCNC(=O)C=Cc1ncc[nH]1 2144,C1(NC(C2CCO2)=O)(CO)CCN(C(c2ccc(SC(F)(F)F)cc2)=O)C1 2145,c1(C(N2CCN(C(C#CC3(CC)CC3)=O)CC2)=O)cccc2cc(F)ccc12 2146,N1(C(c2cn(CC(N)=O)nn2)=O)CCCC(N(CCO)C(c2cnccn2)=O)C1 2147,Cc1nn(CC(=O)NC(C)CNC(=O)Cc2ncc(Cl)s2)c2ncccc12 2148,CC(F)CC(=O)N1CCC(NC(=O)Cc2cc[nH]n2)C1 2149,c1(OC(C)C(N2CCCCC2CNC(c2ccc(Cl)cn2)=O)=O)ccccc1F 2150,n1(CCSC)nnnc1C(c1csc(-c2ccsc2)n1)Nc1nccn1C 2151,c1(C(=O)NC2CCN(C(C3CCC(CC)CC3)=O)C2)nn(C)c2ccc(Br)cc12 2152,N1(C(C2CCC(CC)CC2)=O)CCC2(COCC(CNC(=O)C(F)(F)CC)O2)C1 2153,c1(OC)ncc(C(=O)NCCC2CCN(C(C3CC(F)C3)=O)C2)cn1 2154,c1(C(=O)NCC2C(CNC(c3c(C(C)C)cco3)=O)C2)ccc(N)c(N)n1 2155,c1(OC)c(N2CCOC(CNC(C3COCCN3C(C)=O)=O)C2)ncnc1C 2156,Cc1cc(CC(=O)NC2CN(C(c3cn[nH]c3C(C)C)=O)CC2(C)C)cc(F)c1 2157,CC(O)CCC(=O)NCC(C)N(C(=O)CCc1ccco1)C 2158,Cc1ncc(Cl)cc1CC(N1CCCCC1CNC(=O)CN(S(C)(=O)=O)C)=O 2159,CS(=O)(=O)c1cnn(CC(=O)NCC2OCCC2C(=O)O)c1 2160,C(=O)(CN1C(=O)C(NCC2CCCN2C)CCc2ccccc21)NC(C#C)C 2161,N1(C(c2c(C)cccc2Cl)=O)CCOCC12COCCN(C(C1CCOC1)=O)C2 2162,c1(C(N(CC(C)N(C(=O)CCc2ccon2)C)C)=O)ccc(S(N)(=O)=O)o1 2163,C1(CCC(=O)OC2(CNC(CC=C)C3CC3)CCCC2)CCN(C(C)=O)CC1 2164,c1(C(N2CC3C(N(C(c4c(OC)csc4)=O)C)C3C2)=O)cccc(C)c1O 2165,C(=O)(CC(C(F)(F)F)NC(C1(C2(C)CC2)CC1)=O)NCc1ccc(C)cc1 2166,N1(C(=O)CC2(C)CCCO2)CCC(CCN(CC(N2CCCC2C)=O)C)CC1.CS 2167,C1(OC)(OC)CCC1C(=O)N(CC(=O)NCc1ccoc1)C(C)C.C1CC1 2168,N1(C(c2cc(CCC)on2)=O)CCC(NC(C2CC(SC)C2)=O)CC(C)(C)C1 2169,c1(N2CCCC(N(C(COCc3cc(C)on3)=O)C)C2)ncc(Br)cc1C#N 2170,N1(C(C(C)NC(=O)OC)=O)CCCC(C)(C)C1C(=O)NCCCP(C)(C)=O 2171,c1(C(N(C(CC)C(=O)NCCC2(C)CC2(F)F)C)=O)ccc2n[nH]cc2c1 2172,N1(C(Cc2cc(C)no2)=O)CC2C(C(=O)N(n3cccc3)C)C2C1 2173,c1(NC2CN(C(C)=O)C2)ncccc1S(=O)(=O)N1CCC(=C(F)F)CC1 2174,C1(C(=O)NCC(CCOC)NC(c2nocc2Br)=O)CC1C1CCC1 2175,C1(C(=O)NCCC(CNC(c2c(C)ccs2)=O)O)Cc2c(F)cccc2O1 2176,N1(C(C2C(Cl)(C(=O)O)C2)=O)CCS(=O)(=O)CC1c1cccs1 2177,N1(C(Cn2c(CCC)ncc2)=O)CCOCC1CN(C)C(C1C=CCS1)=O 2178,c1(C(=O)NCC(CCC)NC(=O)CCc2nc(CC)no2)ccc(CCF)cc1 2179,c1(C(=O)OC)c(C)[nH]c(C(=O)NCCN(C)C(c2c[nH]nc2S(N)(=O)=O)=O)c1C 2180,N1(C(=O)Nc2ccc(C(=O)NC)c(Cl)c2)Cc2cccc(Cl)c2C1 2181,c1(CC)cc(Br)ccc1CN1CC(C(=O)NCc2ccnc(Cl)c2)CC(F)C1 2182,C1(NC(C2(NC(c3cccc(=O)n3C)=O)CCN(C)C2)=O)CN2CCC1(F)CC2 2183,C1(O)(CC(N2C(Cn3cc(C(C)(C)OC)nn3)CCC2)=O)CCN(C)CC1 2184,c1(CSC)cccc(C(=O)NCCOCCCNC(=O)C(C)=C2CCC2)c1 2185,C1(NC(C(=O)N(C2CCCC(C(=O)NC3CC3)C2)C)=O)CC(=O)NC(=O)C1 2186,C1(NC(C2C3CN(C(c4c(C)cnnc4)=O)CC32)=O)C=CC(C)(C)CC1 2187,c1(-n2c(CCCCCSC)nc(CCOC)n2)cc(C)ccc1C 2188,C1(NC(COCC)=O)(CO)CCCN(C(c2cnc(N)c(Br)c2)=O)C1 2189,C(=O)(C(C)(C)C(C)NC(=O)C=Cc1ccc[nH]1)NCC1CCN(CCC)C1 2190,C1(C(N(CC(O)CNC(C2(Br)CC2)=O)C)=O)CC12CCOCC2 2191,N1(C(C2N(C(CCCCCC#N)=O)CCC=C2)=O)CC2(CCC(=O)NC2)C1 2192,CCC(Cc1ccccc1C)C(=O)NCC(C)(O)CNC(C1(C(C)(F)F)CC1)=O 2193,C12(NC(C(CSC)OC)=O)CCCC1(F)CN(C(=O)CCCC(F)(F)F)C2 2194,N1(C(c2cnc(OC)s2)=O)CC(C)CN(C(c2ccc(F)cc2N)=O)C(C)C1 2195,N1(C(c2ccc(OC)cc2)=O)CCC(F)CC1C(=O)Nc1cc(C)cc(O)c1 2196,c1(OC)nccc(C)c1NC(C1CCCCN1C(=O)C(C)(C)OC)=O 2197,C(=O)(CC(C)C(C)(C)C)N1CC(C=CC)C(C(N2CCN(C(C)CC)CC2)=O)C1 2198,c1(C(N2C(C3CCN(C(CCC4(C)CC4)=O)C3)CCC2)=O)cncc(Cl)c1 2199,c1(OC)ccc(C)c(C(N2CCC(C(C)NC(=O)CCN(C)C(C)=O)C2)=O)c1N 2200,C1(C(=O)NC2CC(CF)C2)C2CC(O)C(C2)N1C(c1ccn2ccnc2c1)=O 2201,Cc1cc(C(N2CCOCC(NC(c3ccc(C(N)=O)o3)=O)C2)=O)nc(C)c1 2202,CCCCCC(C)CC(=O)NC1CN(C(C2CC(F)(CO)C2)=O)CC1C 2203,C1(C(=O)NOCCC)(CC#C)CCN(C(c2c[nH]c(=O)cn2)=O)C1 2204,CCC(C(=O)NCc1cn(CC(C)NC(=O)C(O)C2CC2)nn1)SC 2205,c1(C2(NC(c3n(C4(C)CC4)nnn3)CCOCCSC)CC2)ccccc1Cl 2206,c1(C(=O)NCC2(NC(C3CCCCC3F)=O)CC2)c(F)ccc(F)c1Cl 2207,C1(NC(C2CCCC2C(F)F)=O)CC2CC1N(C(c1ccncc1)=O)C2 2208,c1(CC)onc(C)c1CNC(=O)CCC1CCN(C(=O)CC2CCCC2)CC1 2209,Cc1c(C(=O)NCCCn2cc(Br)ccc2=O)cccc1Cl 2210,Cc1nc(C(N2CC(NC(c3cc(F)ncc3Br)=O)C(C)C2)=O)ccc1F 2211,C1(NC(C2(CS(C)=O)CC2)=O)CC(NC(c2nn(C)cc2Cl)=O)C12CCC2 2212,N1(C(CCSC)=O)CC(S(=O)(=O)N2CCN(C(=O)C=C(C)C(C)(C)C)CC2)C1 2213,c1(C(=O)NC2C(CNC(C(CC#C)O)=O)C2)ccc(COC)c(F)c1 2214,C1(C(=O)O)(NC2CN(C)CC23CC3)CCOc2ccccc21 2215,c1(CC)cnc(O)c(C(=O)NC2CN(C(=O)Cn3cc(CO)nn3)CC2C)c1 2216,c1(OC)cccc(C(=O)NC(C2(O)CN(C(=O)CC3CCC4CC34)C2)C)c1C 2217,C(=O)(CC(C)CC)NCC1(C(=O)NC(C(=O)N(C)CC)C)CC1 2218,c1(C2(C(=O)NC3C(NC(C4CCCC4)=O)C3)CC2)cccc(F)c1F 2219,c1(N(CCCS(C)(=O)=O)C)ccc(S(=O)(=O)N2CCSC3CCC23)cn1 2220,CC1CN(C(c2ccn(CC(F)F)n2)=O)CC1NC(C1CCC1(C)C)=O 2221,N1(Cc2ccc(OC)c(O)c2)CC2CCN(C(c3occc3C)=O)C2C1 2222,N1(C(C(C2CCC2)OC)=O)CC2(CC2)CC1CNC(=O)CCOCCN(C)C 2223,C1(CNC(c2c(OCC)scc2)=O)CCC(C)(C)CN1C(=O)C(C)CF 2224,c1(C(=O)NCC(C2CC2)NC(c2c[nH]cc2Br)=O)ccc(CO)c(F)c1 2225,N1(C(c2ncn(CC)c2)=O)CC(C(N2CC(NC(C)=O)C2)=O)C(C2CC2)C1 2226,C(C)(CCC(=O)N(C1(C(N2CCC(O)(C(N)=O)C2)=O)CC1)C)OCC 2227,N1(C(c2cncc(OC)c2)=O)CCOCC12COCCN(C(=O)C(C)C(C)C)C2 2228,N1(C(CC=CC(C)(C)C)=O)CC2CCN(C(=O)CS(=O)(=O)C(C)(C)C)CC2C1 2229,c1(NC(c2ccc(C)nc2)=O)ccc2nc(C3CC3)oc2c1.C12CC1CNC2=O 2230,N1(C(C=C(CCC)C)=O)CCN(C(=O)CC2COCC2O)CC1COC 2231,c1(C(=O)NCC(CC(=O)N(CCOC)CC2CC2)OC)ccc2[nH]ccc2n1 2232,C(C(C)(CC)C(N)=O)NC(C1(CCC=C)CN(C(C2CCC(=O)N2)=O)C1)=O 2233,N1(C(C(C(C)C)O)=O)CCC(C)(C)C1CC(=O)NCC1CCCSC1 2234,C1(CC)OCCC1C(=O)NCc1cc(C(=O)NCC2(CO)CCCO2)on1 2235,c1(C(=O)NCCCCCN(C(=O)CCCN=[N+]=[N-])C)cc2n(n1)CCCC2O 2236,c1(C(=O)NC2CCN(C(c3cn(CC)nn3)=O)C2C)cc2ccc(Cl)cc2[nH]1 2237,C(=O)(CC1=CCOCC1)NCC(c1cccc(Cl)c1)NC(C(CC#C)(C)C)=O 2238,C(CCN=C(NC(C)C)NC1CC1(C)C)N(CC)CC 2239,C=Cc1ccc(C(N2CC3CCC2C3NC(=O)Cc2ccn(C)n2)=O)cc1 2240,C(=O)(C(O)CC(F)F)N1C(CCN(C(CCC(C)C)=O)C)CCCC1 2241,C1(CNC(C(CC)CCOC)=O)CN(c2ncnc(=N)[nH]2)CC(C)(C)O1 2242,c1(-c2nc(CSC)nn2-c2nc3ccccc3[nH]2)cc(C)nc2c1nc(C)n2C 2243,CC(C)(CC#N)C(=O)N1CCC(NC(=O)C(c2ccccc2F)(F)F)C(O)C1 2244,Cc1cc(C(N2CC(c3ccccn3)(C(=O)O)C2)=O)cc(-n2cccc2)c1 2245,c1(C(=O)NCCCN(C(=O)C(O)Cc2ccccn2)C(C)C)cnn(C2CC2)c1 2246,c1(CC(=O)NCC2(C)CCC(NC(=O)C(N)=O)C2)ccc2c(c1)OC(F)(F)O2 2247,c1(NCCCC(=O)NCC2C(NC(C(C=C)O)=O)C2)ccc(C)cc1 2248,C(=O)(N=c1ccc(Cl)n[nH]1)C1C2(CN(Cc3c(OC)nccc3I)C2)C1 2249,c1(C(=O)NC(C(C(C)C)NC(c2ccccc2O)=O)C)cncn(C)c1=O 2250,N1(C(C2CCCN(C)C2)=O)CCC(F)(CNC(c2sccc2C#N)=O)CC1 2251,CC1CCN(C(c2cccc(C3CC3)c2)=O)CCN1C(=O)Cc1ncc(Cl)s1 2252,C(=O)(CCCCCCS(N)(=O)=O)NCCC(C)NC(Cn1ncc(CC)c1)=O 2253,c1(CC(N2CCOCC(NC(c3ccn(C)c3)=O)C2)=O)cnc2ncccn12 2254,c1(C(N2C(C)CC(NC(C=C(C)C)=O)C2)=O)[nH]c2c(c1C)CCCC2 2255,C1(CC)CCCCCCN1C(=O)CC(C)C(C)(C)NC(c1cccc(O)c1F)=O 2256,C(=O)(CC1=CCN(C(C2(N(C)C)CC2)=O)CC1)N1CC(CC)OCC1C 2257,CC(C)(CCC#N)C(=O)N1CCC2(CC(NC(C3(n4cnnn4)CC3)=O)C2)C1 2258,C=C=C(C)CC(=O)NCC(CNC(c1ccc(OC(C)C)nn1)=O)CO 2259,N1(Cc2nnc(C(C)C)o2)CCC(NC(c2c[nH]c(Br)c2)=O)C(C)C1 2260,C1(CO)C(=O)N1.CC(C)CCOC(C)C(=O)N(CC(C)(C)C)C1CC1 2261,c1(NC(C2N(C(c3cc(C)no3)=O)CC(F)C2)=O)cc2nccn2cn1 2262,Cc1nn(CC(C)C)c(C)c1CNC(C12CCC(CN1C(=O)OC(C)(C)C)C2)C 2263,CCC(C)C(C(=O)NCC[Si](C)(C)C)N(C)C(C1CC2CC1CC2O)=O 2264,CCC(CC)(CO)C(=O)NC(C)CNC(=O)C(CO)NC(N)=O 2265,c1(NC(c2ccc(CNC(CCC(C)OC)=O)cn2)=O)ccc2c(c1)OCC2 2266,N1(C(CS(CC)=O)=O)CCN(C(c2cn(C3CC3)nc2C)=O)C2(CC2)C1 2267,N1(C(C(C)N(C)C)=O)CCOC2(CCN(C(=O)CC(C)(O)C(F)(F)F)C2)C1 2268,c1(C(=O)NCC2C3CN(C(CCC(=C)Cl)=O)CC32)cc(C)c(=O)n(C)c1 2269,C(CCC(N)=O)(C(=O)NCC1CCN(C(c2cc(O)n(C)n2)=O)CC1)NC(C)=O 2270,C(=O)(C(C)(C)CC#N)NCCCC(C)(C)c1cn(CCC(CC)O)nn1 2271,c1(C(=O)Nc2ccc(OC(F)F)cn2)ccnc(CNC(C2CC2C2CC2)=O)c1 2272,N1(C(C(C(C)O)NC(C)=O)=O)CCc2ccccc2C(NC(=O)C(C)C(C)C)C1 2273,N1(C(c2c(C)nc(C)s2)=O)CCN(C(c2cccc(Cl)c2O)=O)C(C2CC2)C1 2274,Cc1ccc(C(N2CCN(C(=O)CS(=O)(=O)N3CCOCC3)CC2C)=O)c(C)n1 2275,C12(C(N3C(C#C)CCCC3)=O)CCC(CN(C(=O)C(C)OC3CCCC3)C1)C2 2276,O=C1CCC(CC(N2CCN(C3CN(C(=O)C(Cl)=CCl)C3)CC2)=O)CN1 2277,Cc1cc[nH]c(=N)c1C(=O)NCC(C)NC(c1cnn(-c2cccc(F)c2)c1)=O 2278,C(CC(C(=O)N1CSCC1C(N1CCC(CCCO)CC1)=O)OC)OC 2279,c1(CNC(Cn2cc(-c3c(Cl)ccc(C)c3)nn2)=O)cc(C)cc2c1CCC2 2280,N1(C(CCc2ccn(C)n2)=O)CC(CNC(C2(C#N)CC3CC3C2)=O)C(C)(C)C1 2281,C(=O)(C(CC(C)C)C(C)C)NC(C(C)NC(c1c(C)cc(C)nc1S)=O)C 2282,c1(C(=O)NCCN(C(=O)CC2CC2(C)C)C)cccnn1 2283,N1(C(c2cc(C)no2)=O)CCN(c2nccc(Br)n2)C(C#N)C1 2284,C(=O)(CC(CC)C(C)C)N1CCC(CC)C1C(=O)NCCCn1cncn1 2285,C1(NC(C2(C)CC(=C)C2)=O)CN(C(c2cnn(C(C)C)c2C)=O)CC1C(F)F 2286,c1(C(=O)NC2C(CNC(CCCc3onc(C)n3)=O)CCC2)cc(F)ccc1N 2287,c1(C(N(CCCCCNC(c2c(SC)snn2)=O)C)=O)[nH]cc2c1CCCC2 2288,N1(C(c2c(C)cc(C)[nH]2)=O)CCC2CCC(C1)N2C(C1CN=C2N=CNN2C1)=O 2289,C(C(C)CN=C(NCCC1CC1)NCC(C(C)C)OC)SC 2290,c1(C(=O)NC2CC(C(=O)NC(CCC)CCO)CC2O)cccc(O)c1C 2291,C=C=CC(C)C(=O)NC1CC(C)(NC(=O)CSc2ccc(C(C)(C)C)cc2)C1 2292,N1(C(=O)Cn2cnnc2)CCC2(CCN(C(c3c(F)ccc(F)c3F)=O)C2)C1 2293,c1(C(C(=O)NCCN2CCOCC2)N(CC(C)C#N)CC)cccc(F)c1Br 2294,C(=O)(CCC(=O)N1CCCC1(CC(C)C)C(=O)O)OCC 2295,n1(CCC)ncc(C(=O)NCC2CCCC(NC(=O)Cc3cnnn3C)C2)c1C 2296,FC1(F)C2(NCc3nccn3-c3ccc(F)cc3)CCCCC12 2297,C1(NC(c2cc(OCC)ncc2)=O)C2CC1CN(C(c1cscn1)=O)C2 2298,CC(CC(=O)N1C2CCC1(CNC(=O)CC1CC1(C)C)CC2)C(F)(F)F 2299,C1(CNC(C2(C(=O)NC)CCC2)=O)CCC(C(=O)NCc2ncc(C)o2)C1 2300,c1(CNC(C(C)OCCOC)=O)cccc(CN(C)C(c2sc(C)nc2C)=O)c1 2301,N1(C(C(CCC)OC)=O)CC2(CCCCN(C(=O)C(c3cncc(F)c3)C)C2)C1 2302,c1(CN(C)CC2CCCN(C(C3C(CC)CCCC3)=O)C2)ccc(O)c(O)c1 2303,C1(C(=O)NC(CCC)C)CN(C(=O)CCCF)CCC1(C)C 2304,c1(C(=O)NCCN(C(=O)C(n2ccc(Br)n2)C)CC)c(C)ncn1O 2305,c1(OC)cc(C)ccc1C(N1CCC(=CCNC(c2nc(C3CC3)cs2)=O)CC1)=O 2306,c1(C(=O)NCC2(CNC(c3cc(COC)no3)=O)CC2(F)F)cnc[nH]c1=N 2307,CCC(C)CCCC(=O)NC(C)(C)CCN(C)C(c1cc(C(C)=O)[nH]n1)=O 2308,c1(C(C(N2CCN(C(c3cc(C)nnc3)=O)CC2)=O)=O)c(C)nn(C)c1C 2309,C1(NC(=O)Cn2cnnn2)CN(C(c2cc(F)c[nH]2)=O)CC2(CCC2)C1 2310,c1(CC)[nH]ccc1C(=O)N(CCCCNC(c1ccsc1COC)=O)C 2311,c1(C(N2CC(N(C)C(C3CC4C=CC3O4)=O)C3(C2)CC3)=O)ccc(S(C)(=O)=O)[nH]1 2312,C(=O)(C(C)(C)CC(=O)N1CCC(C(C)NC(=O)C2=NOC(C)(C)C2)C1)OCC 2313,C(Cc1ccccc1)(CCNC(=O)CN(C1CCC1)C)NC(C(C)O)=O 2314,N1(C(c2csc(Cl)c2)=O)CCCN(C(=O)C(O)C2CCC2)C(CO)C1 2315,O=C(C1NCCc2ccccc21)NCC(C1CCCCC1)=O 2316,c1(C(=O)NC(C2OCCN(C(C(C)=CC3CC3)=O)C2)C)cncc([N+](=O)[O-])c1 2317,CCC(F)(CNC(=O)NC(C1CS(=O)(=O)C1)C)CC 2318,c1(N(CC(C)NC(=O)CSCCC(F)(F)F)C)nc(C2CC2)ns1 2319,c1(C(=O)NCC2CCCC(NC(C(C#C)(C)C)=O)C2)nccc(F)c1Cl 2320,c1(C(=O)NCC(CNC(C2(OC)CCOC2)=O)OC)cc(C2CC2)n(C)n1 2321,C1(CN(C)C(C2(NC(=O)CC3CS(=O)(=O)C3)CC2(C)C)=O)COC(=O)N1 2322,C1(NC(c2c(C)nn[nH]2)=O)CCN(C(=O)Cc2cc(F)cc(Cl)c2)C(C2CC2)C1 2323,C12(C(=O)NCCCC(C)NC(c3ccc(C4CC4)cn3)=O)CCC(CC1)CO2 2324,c1(CC)cc(F)ccc1C(N1CC(O)CC1CNC(C1(C#N)CC(C)C1)=O)=O 2325,n1(CCC(=O)NCC(CC=C)NC(=O)CC(CC)OC)ccc2cccnc12 2326,C1(CCCC(=O)NC(C(C)C)CNc2ccccc2)CCCC(=O)N1 2327,CC1CN(C)CC1C(=O)NC1CC(CNC(c2ccc(OCC(F)F)cc2)=O)C1 2328,C1(C(N(C(C2CCCCC2)C)C)=O)COC2(CNC2)C1 2329,c1(C(=O)NCC23CCC(CN(C(CNC(C)=O)=O)C2)C3)ccc2[nH]c(=N)[nH]c2c1 2330,Cc1sc2ncnc(N3CCCC(C)(c4ccccc4)C3)c2c1C 2331,C(C(O)CC(=O)NCc1ccc(C(=O)NCCOC(C)(C)C)nc1)N(C)C 2332,c1(N2C3CC(CN(C(C4C(CC)CCC4)=O)C3)C2)ncc([N+](=O)[O-])cc1C(N)=O 2333,CC1=CCC(C(=O)NCC23CC(NC(c4cnn(C(C)(C)C)c4N)=O)(C2)C3)CC1 2334,C1(CC(=O)NCC2(F)CN(C(c3ccc(C(F)(F)F)cc3)=O)C2)CCCC1(F)F 2335,N1(C(Cc2c(C)nc[nH]2)=O)CCC(NC(=O)CCc2cncn2C)C12CCC2 2336,CCC(CCC(=O)NCCOCC1CCCC1)NC(=O)CS(=O)CC 2337,c1(NC(=O)NNC(=O)c2ccccc2F)ccc2cc[nH]c2n1 2338,c1(NC(C2C(NC(CCCOC)=O)CC2)=O)ccc(SC)nc1 2339,C1(CC(C)C)CCN(CCCc2nnc(-c3cccs3)o2)CC1 2340,C1(C(=O)NC(CC#C)C(=O)NC(CO)C(C)(C)C)CC2C(C1)C2(F)F 2341,CC1(C)C(C(N2CC(NC(c3ccoc3Cl)=O)C2)=O)CC1(F)F 2342,N1(C(CSCCC)=O)CCC2(CC2)CC1C(N1CC2CC2(C(=O)OC)C1)=O 2343,Cc1noc(Cl)c1CC(N1CCCC(C2CCCCN2C(C2SCCS2)=O)C1)=O 2344,N1(C(CCC)=O)CC2CC1CN2C(=O)Cc1cc(Cl)ccc1Br 2345,c1(CC(CC)C)nc(-c2nn(C)nc2Br)n(-c2cnnn2C)n1 2346,Cc1ccc(C(N2CCC2C(N2CC(CC(N)=O)C2)=O)=O)[nH]1 2347,Cc1ccn(CC(=O)N(CCNC(=O)Cc2nc[nH]n2)C(C)C)n1 2348,C=CCC(C)C(=O)NC1CC(NC(=O)CCSc2nccn2C)C1 2349,c1(OC)cc(C(N2CC(CCCCNC(c3csc(Cl)n3)=O)C2)=O)cc(F)c1 2350,c1(C(=O)NCC2(F)CC(C(=O)OC)C2)cnn(CC2CCOCC2)c1Cl 2351,Cc1nn(C2CC2)cc1C(=O)NCCC1CCCN(C(C2CC2(Cl)Cl)=O)C1 2352,CC(C)(C(=O)NCC1CCCN(c2nnc(C3CCCC3)s2)CC1)C(N)=O 2353,C1(CNC(Cc2c(C)n(C)cn2)=O)CCCCCN1C(=O)C(c1cccn1C)=O 2354,C(=O)(CCC1=CCCCC1)NCC(CCOC)NC(=O)C(n1nccc1C)C 2355,N1(CC)CC(NC(=NCC2CCC(F)(F)C2)NC2CC2)CCC1=O 2356,S(=O)(=O)(c1cccc2scnc12)NC1CCN(C(c2ccn(CC)n2)=O)CC1F 2357,CON(CCC(=O)NC(C)C(F)F)C(=O)C1CC(C(C)C)C1 2358,c1(C(=O)Nc2cccc(C(=O)NCCC(O)CCO)c2)cc2ncccn2n1 2359,N1(C(c2cc(C)cc(C)c2)=O)CCN(C(c2nnsc2C)=O)C2CCCCC12 2360,CC1CC(NC(c2cc(Cl)c(Cl)s2)=O)CN(C(=O)Cc2cc(F)ccc2O)C1 2361,C12(C(=O)NCCCCNC(C(CC)OC)=O)CC(c3ccccc3)(C1)C2(F)F 2362,C1(Nc2cccc(SC(C)(C)C)c2)CC(=NOC2COC2)C(N)C1 2363,C1(CN(C(=O)CC(O)CN(C)C)C)CCCCN1C(=O)CC1(O)CCCOC1 2364,C=CC(C)(O)C(=O)NCC1CCN(C(=O)C(C)NC(=O)OC)CC1 2365,C1(CCC)CN(C(=O)CC(C)COCC)CCN1C(=O)C(C)Cc1cnc[nH]1 2366,c1(C(=O)NC2(CNC(c3ccnnc3S)=O)CCOC2)ccc(Cl)cc1Cl 2367,Cc1cc(P(C)(C)=O)oc1C(N1CCN(C(=O)Cn2cc([N+](=O)[O-])cn2)CC1)=O 2368,N1(C(COC2CC(NC(C34CCC(C)(OC3)C4)=O)C2)=O)Cc2cncnc2C1 2369,C(=O)(C(C)(CO)NC(c1cnnn1C)=O)N(C(CC(C)C)C)C 2370,c1(CNC(CCN(C)C(C2CCCN2C)=O)=O)ncc(Cl)cn1 2371,c1(C(=O)NC2C(C)N(C(c3csc(C(F)F)n3)=O)CC2)cccc2nn(C)cc12 2372,c1(N(C(C(C=C)F)=O)C(=O)CCc2ccc(C)cc2)ccccc1C(C)C 2373,C(C)(CO)(C(=O)N(C)CC1(CNC(=O)CCn2ccnc2C)CC1)NC(C)=O 2374,N1(C(C2C(COC)CC2)=O)CC2CN(C(=O)CN3CCCS3(=O)=O)CC2(C)C1 2375,CC1CCN(C(c2cccc3c2CCC3)=O)CCN1C(=O)CCc1ccncn1 2376,CC1=C(C(=O)N2CCCC2CCNC(c2cnc(O)c(Br)c2)=O)CCO1 2377,C1(CC(=O)NC2CC(NC(=O)Cc3nc(C4CC4)cs3)C2)CCC=CCC1 2378,Cc1ccccc1CN(C(=O)C(c1ccoc1)NC(=O)COC1CC1)C 2379,C=C(C)C1CN(CC2CC(=O)N(C(=O)C(C)C)C2c2cc(C)c(=O)n(C)c2)CCO1 2380,c1(C(N2C3(CNC(c4nn(C)c(Cl)c4)=O)CCC3CC2)=O)cc(S(C)(=O)=O)cs1 2381,N1(C(C(C)=CC)=O)CCC(NC(c2nccc(OC)c2OC)=O)C(CC)C1 2382,Cc1cccc(N)c1C(N1CC(CCNC(c2ccnn2C(C)C)=O)C(C)C1)=O 2383,CC1(N=c2[nH]nc(-c3ccccc3)s2)CCC(NC(=O)CCF)CC1 2384,CCC(C)C(C)C(=O)NC(C)Cn1cc(-c2cn(C)nc2C(=O)OC)nn1 2385,c1(CNC)ccc(NC(c2sc(C(C)C)nc2C)=O)cc1 2386,CC1CN(C(=O)Cc2ccn(C)n2)CC1(C)CNC(=O)Cn1ccccc1=O 2387,c1(C(=O)OC)cn(C)nc1C(=O)NC(C)CN(C(=O)CC12CCCC1C2)C 2388,Cc1cc(C)c(C(=O)NCC2C=CCN2C(=O)CN2CCCCCC2)s1 2389,Cc1cc(C(=O)N(CCCN(C)C(c2cc(=O)n(C)cn2)=O)C)nc(O)c1 2390,c1(N2CCC(C(C)C)C2)nc(N2CCC(C)(c3ccccc3)C2)c2ncsc2n1 2391,C=CCCCC(C(=O)NCCNC(c1csc(C)n1)=O)NC(c1ccoc1)=O 2392,CS(=O)(=O)c1sccc1C(=O)NCC1CC(CNC(=O)Cn2ncnn2)CO1 2393,CS(=O)(=O)C1(NC(C2CC3CN(C(=O)OC(C)(C)C)CC3C2)=O)CCCC1 2394,N1(C(C(Br)=C(C)C)=O)CCC(C2CC2)(CNC(c2ncnc3c2CCC3)=O)C1 2395,C1(C(N2CCSCC(C)C2)=O)COC2(C1)CN(C(c1c[nH]c(C#N)c1)=O)C2 2396,N1(C(c2cc(C)on2)=O)CCN(C(=O)Cc2nonc2C)C2CC12 2397,N1(C(C2C(C)OCC2)=O)CCC2OCCN(C(c3ns[nH]c3=O)=O)C2C1 2398,c1(C(N(C)CC2C3CN(C(C(CCC)C#N)=O)CC32)=O)cc(Cl)c(F)cc1OC 2399,c1(NC(C2CCCC2NC(C2CC23CCOC3)=O)=O)c[nH]ccc1=O 2400,C1(OCC)CC2CN(C(=O)C(CN(C)C)NC(c3c(C)ccnc3C)=O)CC12 2401,c1(N2CC(C=C)OCC2)cc(S(=O)(=O)NC2CC3(CC3)C2)ccc1C#N 2402,c1(C(N2C3CN(C(C(C)O)=O)C(C3)C2)=O)ccc2c(O)nnc(O)c2c1 2403,c1(C(=O)NC2CN(C(c3c(CC)n(C)cc3)=O)C3C2C3)ccc([N+](=O)[O-])cn1 2404,C1(CC(=O)NCC(CC)NC(c2n[nH]c(C)c2Cl)=O)OCCCC1(C)C 2405,Cc1cc(Cl)cc(C)c1C(=O)NC1CC(NC(=O)CC(C)(C(F)F)N(C)C)C1 2406,C12(COC)CN(C(=O)Cn3cncn3)C(CNC(C3CC(N(C)C)C3)=O)(C1)C2 2407,C1(O)(C(C)NC(=O)CC2NC(=O)NC2=O)CCN(C(C2(C)CC2(F)Cl)=O)CC1 2408,C1(C(N(CCOCCOC)C)=O)CN(C(=O)CCn2ccc(C)n2)C(C)(C)C1 2409,N1(C(CNC(CN(S(C)(=O)=O)C)=O)C(F)F)CCN(C(C2(C)CC(C)C2)=O)CC1 2410,C(C(C)C(F)C(=O)NCCCNC(C)=O)NC(C1(OC)CC1)=O 2411,C1(CN(C)C(C2CC(C)(NC(=O)C(C3CC3)C3CC3)C2)=O)CCCCO1 2412,C1(CC)C(NC(c2cnc(CC(C)(C)C)o2)=O)CCCN1C(c1cnco1)=O 2413,c1(C(N2C(CNC(C3N(N=O)CCCC3)=O)C=CC2)=O)ncnc2ccsc12 2414,N1(C(c2nc(CCC)sc2)=O)CCCCC1CCCNC(C1(C)COC1)=O 2415,CC(C)(C)CC(O)C(=O)N1CCN(C(=O)CNC(N)=O)CC(CO)C1 2416,Cn1ncc2ncnc(N3CCN(Cc4ccc(Cl)o4)CC3CC#N)c12 2417,N1(C(CCNS(CC)(=O)=O)=O)CCCC1CNC(=O)CCn1cccc1 2418,Cn1c(O)nc2c(C(=O)NC3CCN(C(c4cnc(O)s4)=O)CC3F)cccc12 2419,c1(SC)cc(C(=O)NCC=CCNC(=O)CCC2(C)CC2(F)F)oc1C 2420,c1(C(N(CC(C)CNC(=O)Cc2cccnc2Cl)C)=O)ccnc2c1CC(=O)N2 2421,n1(CC)nncc1C(=O)NCC(CNC(C1CC=CCC1)=O)CO 2422,N1(C(C(C(=C)C)(C)C)=O)CC(NC(=O)C(C)(C2CC2)OC)CC2(CCC2)C1 2423,c1(C(=O)NCCCCC(C)NC(Cc2c(C)nccc2)=O)ccc(S(C)(=O)=O)o1 2424,C(=O)(C#CC1(C)CC1)NC1CC(NC(C(C)Sc2ccccc2)=O)C1 2425,C1(N(C(=O)CSCCCl)C2CC2)CCCCC1.C1CCOCC1 2426,C1(C(N2CC(C(C)NC(C3CCC(=O)O3)=O)C2)=O)CCC2CC2CC1 2427,O=S(=O)(c1ccc(NCC(CO)C2CC2)c(F)c1)N1CC2CC3CC2C1C3 2428,C1(CN(C(c2cc(CNC(c3scc(C)c3)=O)oc2)=O)C2CC2)CCCC(C)C1 2429,N1(C(Cn2nc(C)n(C)c2=O)=O)CCC2CCN(C(C3(C)CC3(F)Cl)=O)CC2C1 2430,C1(CN(C)C(c2cnoc2)=O)CCCN1C(c1cc[nH]c1C1CCC1)=O 2431,CCC(C(=O)NCC(Cc1ccccc1)N(C)C(C12CC(CO1)C2)=O)N(C)C 2432,C(=O)(C(F)C1=CCCCC1)NC(CCNC(c1ncc(CC)s1)=O)C 2433,Cn1cnc(CCC(=O)NCCSCC(N2CC(OCC(N)=O)C2)=O)c1 2434,Cn1ncc(C(N2CCCCC2C2CCCN(C(=O)CCCF)C2)=O)c1F 2435,C1(C)(NC(COC(C)=O)=O)CCN(C(C2(c3cccnc3)CCCC2)=O)C1 2436,C(=O)(CC1=NNC(=O)C1)N1CCC(NC(C(C)N(CC)CC)=O)C(C)C1 2437,C1(NC(CN(C(C)C)C(C2CCC3CC2CO3)=O)=O)CN2CCC1CC2 2438,n1(CC(=O)NC2CCN(C(=O)C=CC3CCCCC3)C2)nc(Cl)ccc1=O 2439,CCC(C(=O)N1CCCC(c2cn(Cc3cnoc3)nn2)C1)C(C)(C)CC 2440,C(=O)(C1CNC(=O)c2ccccc21)N1CC2C(NC(CCOC)=O)C(C2)C1 2441,C1(C(C(N2CC(CC=CC)C2)=O)C)CCCN(C(=O)C(C)=C(C)CC)C1 2442,CC(CCCCNC(=O)C=CC1CCC1)NC(c1cscc1Cl)=O 2443,C1(CCCNC(C=C(C)C)=O)CCCCN1C(C12CC(C(C)C)(CO1)C2)=O 2444,C1(CC(N2CC(C(C)(C)O)C2)=O)COC2CC1C2.C12CC(C1)C(C)NC(=O)C2 2445,c1(C(C)=O)ccccc1C(=O)NC1CCN(C(C)=O)C1C(=O)O 2446,c1(C(N2C(C(=O)NC3(CC#C)CC3)CC2C)=O)ccc(C)c(F)c1 2447,C1(C(=O)NC(CC2CN(C(CC3C(C)CCC3)=O)C2)C)(CO)CCCCO1 2448,c1(NC(N2C(C(=O)Nc3ncn(CC)n3)CC2)=O)cc(OC)c(F)cc1F 2449,c1(C(=O)NCC2CC(CCO)C2)cccc2occc12.C1CCCNC1=O 2450,C1(C2CCN(C(=O)CC3(C#N)CCC3)C2)(NC(COC(C)(C)C(F)(F)F)=O)CC1 2451,N1(C(C2C(C)(C)C2(C)C)=O)CC2CCN(C(=O)C3Cc4ccccc43)C(C2)C1 2452,Cc1oc(C(C)C)cc1C(=O)NCCC(O)CNC(C1CC1c1ccccc1)=O 2453,C(CCC(=O)NCC=CCNC(c1c[nH]cc1C(C)C)=O)=C(C)C 2454,C12(NC(C3C(CNC(c4cc(OC)n(C)n4)=O)CCCC3)=O)CC1COC2(C)C 2455,C(=O)(CC(O)CC(C)(C)C)N1CC(NC(CCCOC)=O)C2(C1)CC2 2456,c1(NC)c(C(N2CCCC(NC(C3(C)CCC(F)(F)C3)=O)C2C)=O)cccc1N 2457,C12(C(=O)NCC3(OC)CCN(C(C4CCOC4C)=O)CC3)CCC(F)(CC1)CC2 2458,Cc1nscc1C(=O)NCCCC1CCCN1C(=O)COCC1CCCCO1 2459,N1(C(CCCC2C(C)C2)=O)CCOC(C(=O)NC(C(F)(F)F)C2CC2)CC1 2460,C1(CN(CC(=O)N(C2CCCCC2)CCC)C)CCN(C)C1 2461,N1(C(C2N(CC)CCCC2)=O)CCCC(C2CCN(C(=O)C(C)CCO)C2)C1 2462,c1(C(N2CCCC(C(=O)O)(COC)C2)=O)ccc2c(c1)CCC(C)(C)O2 2463,C1(C(N2CCC(O)(CN(C)C(C3C=CCC3)=O)CC2)=O)C2CCC1(C)C2(C)C 2464,N1(C(CCCOCCOC)=O)CCC(CC(=O)NCC(F)Cl)CC1 2465,c1(COC)ccccc1C(=O)N(CC(C)N(C(=O)CC1OCCC1(C)C)C)C 2466,S(=O)(=O)(c1ccc(F)cc1)NCCC(N1CCC(n2nnnc2C2CC2)CC1)=O 2467,c1(C(=O)NCC(CNC(c2coc(Cl)c2)=O)OC)ccc2ccn(C)c2c1 2468,C(CCC(=O)NCCC(=C)CNC(=O)C(C)NC(=O)CC1C=CCC1)=CCC=C 2469,C=C(Cl)CC(C(=O)N(C1CCCC1C)C)NC(C1CNC(=O)O1)=O 2470,c1(N(C(C)C)C)ncc(CN2CCSCC(C)C2)cc1F 2471,C1(N(C(C(CC)C)=O)C)CN(C(=O)Cn2nc(Cl)ccc2=O)CC1(C)C 2472,C(CN=C(NCc1cnn(C)c1)NCCN1CCOCC1)C1CC(C)OCC1 2473,C12(C(=O)NCC=CCNC(c3cccc(O)c3F)=O)CCC(CC1)CC2 2474,C1(C(N2C(CNC(c3cc(C)sn3)=O)CCCC2)=O)CN2CCN1CC2C 2475,CCC(CC(=O)NCC(C)(C)C#CC(=O)NCc1cccnc1CC)CC(C)C 2476,C1(C(=O)NCC(C)N(C(CSc2ccc(C)cc2)=O)C)CCc2cnn(C)c2C1 2477,C1(NC(NCC2(O)CCCC2)=NCCF)CC2(CCC2)C12CCC2 2478,c1(N(CC(=O)N(C)C)C)ccc(S(=O)(=O)N(C(CO)C2CCC2)CCO)c(Br)c1 2479,N1(C(CNC(C2(C#N)CC2)=O)=O)CCN(C(=O)CC2CC3(CC3)CO2)CC1 2480,c1(C(=O)NCCCCC(C)NC(=O)CN(CC(C)(C)C)C)cccc(C#N)c1Br 2481,C1(NC(c2c(C3C(C)C3)noc2)=O)CC(F)CN(C(=O)Cc2cn(C)nn2)C1 2482,c1(C(=O)NCCCCN(C(=O)Cn2cnnn2)C)sccc1Cl 2483,CC1CN(C(=O)CC2CCN(C(c3ccn4c3CCC4)=O)C2)CC(=O)N1C 2484,N1(C(CN(C)C)=O)CC(C(=O)O)C2(CC2)C1.C(=O)(COCCCOC(C)(C)C)NCC 2485,c1(CCC)c(C(N2CC(CNC(c3occc3C)=O)CC2C)=O)nnn1CC 2486,N1(C(CC(C)=C(C)C)=O)CCC(C)(CCNC(c2ccc(C3CC3)o2)=O)C1 2487,c1(C(N2CCOC(CCCNC(=O)C3CC3)C2)C(=O)NC)ccc(C2CC2)cc1 2488,c1(CNc2ccc(C(=O)NCC3CCC(F)C3)cn2)cc(Cl)ccc1[N+](=O)[O-] 2489,c1(CC)c(C(=O)NCCC(C)(C)NC(=O)CCc2ncc(F)cn2)csc1C 2490,N1(C(c2nc(CC)oc2C)=O)CCN(C(C2CC(O)C2)=O)CC2CCCCC12 2491,C(=O)(C1=CCC2CCC1N2C(=O)C(C(=O)OC)OC)N(CC)CC1CCOC1 2492,C1(COC)CN(C(C2(N(C)C(C3CCCS3)=O)CC2)=O)CC1C 2493,N1(C(C(c2ccc(Cl)s2)C)=O)CC=C(CNC(=O)C(F)C2CCC2)CC1 2494,N(C(=NCCN1CCC(C)C1)NC1CCN(C(=O)OC)CC1)CC(=C)C 2495,C(=O)(C1=NNC(=O)CC1)N1CCC(O)(C(=O)Nc2cc(OC)cc(Br)n2)C1 2496,c1(CN(C(c2ncc(C)o2)C(=O)NCC2CCOC2)C)ccccc1Br 2497,C1(NC(C2CCCC23CC3)=O)COCCN(C(c2ccc(F)cc2F)=O)C1 2498,c1(C(C2(CC)CC2)=O)cnn(C)c1C(F)F.C1(CC)(CC)CC(C(=O)NC)C1 2499,Cc1cnc(C(=O)NCCCN(C(=O)C(c2cccc(F)c2)(C)C)C2CC2)cn1 2500,c1(NCC(=O)NC(C2CS(=O)(=O)C2)C)cccc(Cl)c1Cl 2501,C1(C(=O)OC)CC(n2cc(C3(C(C)=O)CC3)nn2)CN1C(c1cccc(C)c1)=O 2502,c1(CSC)nn(C)c(C(F)(F)F)c1Cl.c1(CC)nc2nn1Cc1ccc-2cc1 2503,Cc1cccc2c1N(C(C1CCCC1NC(=O)CC1(O)CCOC1)=O)CC2 2504,c1(C(=O)NCC2CCN2C(C2(C(O)C(F)(F)F)CCC2)=O)cnc2[nH]cncc1-2 2505,c1(C(=O)NCC(CC)(C)NC(C2CCN(C)C2=O)=O)nccc2c1CNC2=O 2506,C1(C(=O)NC2C(=O)OCC2CO)(NC(C(C(C)C)F)=O)CCc2cc(Br)ccc2C1 2507,O=C1COc2ccc(C(=O)NC3CN(C(=O)C=CCF)CCC3F)cc2N1 2508,C(=O)(C(F)(F)Cc1ccccc1)N(C)CCNC(C12CC(CO1)C2)=O 2509,CCCCC(CCCC)NC(=O)CC(C)(C)N(C(=O)Cc1cccc(C#N)c1)C 2510,N1(S(CCC)(=O)=O)Cc2ccccc2CC1CC(=O)Nc1ccc(Cl)c(Br)c1 2511,C(=O)(C1=NNC(=O)CC1)NCC=CCNC(c1cnc(OCC)nc1)=O 2512,c1(C(=O)NC(CC)CNC(=O)C(C)=C(C)C)ccc2nnnn2c1 2513,c1(OC)ncc(C(=O)NCC2(C)CN(C(=O)C(C)N(C)C)CCO2)nc1C 2514,N1(C(CCC=C(C)C)=O)CC2CC1(C(=O)NC1(C)CS(=O)(=O)C1)C2 2515,CC1CN2CCN1C(C(N1CCCCC1CNC(C1(C)COC(=O)C1)=O)=O)C2 2516,C1(C(N(CCCCCCNC(CCCC)=O)C)=O)C2CCC(C2)S1(=O)=O 2517,C(CC(=O)NCC1(NC(C2CC2CC)=O)CC1)OCC#C 2518,Cc1coc(C2CC2)c1C(N1CCC(OCCNC(C2CC(O)C(F)C2)=O)CC1)=O 2519,c1(CNCC23C(CN(C(c4cc(CC)nn4C)=O)C2)C3)c(Cl)ccnc1Br 2520,CCC(CC(=O)N(C)CC1CN(C(c2n[nH]c(C3CC3)c2C)=O)CCO1)C(C)C 2521,N1(C2CN(C(=O)C(COC)NC(c3c[nH]nc3C(C)C)=O)C2)CC(CC)CC1=O 2522,C#CC1CN(C(=O)CCC2CCCN(C(=O)C(C)=C(C)CC)C2)CC1OC 2523,C#Cc1ccc(C(=O)NCCN(C(=O)Cc2conc2C)CC2CC2)cc1Cl 2524,N1(C(C2C(CNC(C3(CC#C)CCOC3)=O)OCC2)=O)CC2CSCC(C2)C1 2525,CC(CC(C)(C)C)C(=O)N(C1CCN(C(C2CCN(C)C(C)C2)=O)C1)CCO 2526,CCC(CCOC)C(=O)N1CC(NC(C2Cc3nccn3C2)=O)C1 2527,c1(NC(C2CC(NC(CCCNC(C)=O)=O)C2)=O)ccc(Br)nc1 2528,C(c1cc(C)no1)=CC(=O)NC(CNC(CNS(CC)(=O)=O)=O)(C)C1CC1 2529,N1(C(C2C(C)(C)N(C(c3n[nH]cc3Cl)=O)CC2)=O)CC2(CCOC2=O)C1 2530,C1(C(=O)NCC(C)CNC(C2(C)CC(C#N)C2)=O)CC(c2cccc(F)c2)=NO1 2531,c1(C(N2CC(N(C(C(C=C)O)=O)C)C(O)C2)=O)nn(C)cc1S(N)(=O)=O 2532,C(=O)(C(C(=O)NC1(CNC(C2CC2C)=O)CCCCC1)C1CC1)OCC 2533,C1(NC(C2C=CCC2)=O)(CF)CCN(C(c2cncc(C(F)(F)F)c2)=O)C1 2534,C1(CNC(C2(CC#C)CCC2)=O)CN(C(c2cnc(C(C)OC)[nH]2)=O)CC1(F)F 2535,CCCC(C)C(=O)N1CCC(C2OCCCC2NC(=O)CCc2cnco2)CC1 2536,C12(NC(C=COCC)=O)CCCC1N(C(c1cncs1)=O)CC2 2537,c1(CC)cnc(O)c(C(N2CC(NC(C3(CN(C)C)CC3)=O)C(C)C2)=O)c1 2538,N1(C(C(C)C2CC2)=O)CCN(C(C2CCC(OC(F)F)CC2)=O)CC1C 2539,N1(C(C)C)CCCC1CC(=O)N(C(C)CCNC(=O)CCCN(C)C)C 2540,C(CCN(C)C(C1(Cl)CC1(C)C)=O)(C(C)C)NC(c1cc(CCCCC)[nH]n1)=O 2541,N1(C(c2ccc(CC)s2)=O)CCC(C)C(NC(=O)CCC(F)F)C1C 2542,CC1(C2CCCN(C(=O)CC3CCCN(C(c4cn[nH]c4)=O)C3)C2)CC1 2543,N1(C(CNC(C2C=CS(=O)(=O)C2)C)=O)CCCC2(C1)NC(=O)N(C)C2=O 2544,C1(CNC(CCN(C)CC)=O)COCC2(CCN(C(=O)C(F)=C3CCCC3)C2)O1 2545,c1(C(N(C(=O)C(N2CCCC2CC2CCC(OC)C2)=O)CC)C)cccc(C)c1 2546,C1(NC(C(CC#CC)NC(c2cc(C(C)=O)[nH]n2)=O)=O)CCN(C)CC1C#N 2547,N1(C(C2(CC=C)CCOC2)=O)CC(C2CCCN(C(=O)CN(C)C)C2)C1 2548,C1(CC)CCC(C)CN1C(C1CN(C(c2cnn(C(C)C)c2)=O)CC1(C)C)=O 2549,C1(CNC(c2nnnn2-c2cccs2)C2(O)CSC2)CCCCN1C1CC1 2550,c1(CC(=O)N(CCCNC(c2cccn2C)=O)C(C)C)cccc2ccccc12 2551,C(=O)(CC(C(F)F)n1ccnc1)NC(CN(C)Cc1nc(C(C)C)sc1)C 2552,C(=O)(N=c1[nH][nH]c2c1CN(C(=O)C(C)=CC1CC1)C2(C)C)c1c(OCC)cccc1 2553,c1(C(=O)NC(C(C(=O)N(CC(=C)C)C)C)C)ccc(=NC)[nH]c1 2554,C(=O)(CC(F)(F)C(C)C)N1CC(CCNC(C2N(CC)CCCC2)=O)OCCC1 2555,c1(C(N2CCC(CN(C(C(CC)(C)OC)=O)C)CC2)=O)ncncc1C#N 2556,O=C(CCC(F)(F)F)NC1CCC(C(=O)N(CCO)CC2CSC2)CC1 2557,C=Cc1cncc(C(=O)NCC2CC3CC3N2C(c2cc(CO)[nH]n2)=O)c1 2558,CN1CCC(C(=O)NCC2N(C(c3cnn(C(C)C)n3)=O)CCC2(C)C)CC1=O 2559,c1(CN2CCC(NC(c3ccc(CN(C)C)cc3)=O)CC2)ccc(F)c(CO)c1 2560,C1(C(=O)NCCS)CCc2ccccc2O1.Cc1nc(CC(=O)NCCC)co1 2561,C(=O)(CC1OCc2ncccc21)NCCCN(C(C(CCSC)O)=O)C(C)C 2562,c1(C(=O)NCC2C(NC(c3ccc(CN(CCC)C)o3)=O)CC2)csc(C#N)c1 2563,N1(C(c2cnn(C)c2Cl)C(=O)NCCCSC)CCN2CCCCC1C2 2564,C(C(C)C(=O)NCCC(Cc1ccccc1)NC(c1nscc1N)=O)SC 2565,CC(C)C(C)C(CNC(C1CCCCC1)=O)NC(c1cn(C)nc1C(C)(F)F)=O 2566,N1(C(c2scc(C)c2)=O)CCCCC2(CCN(C(C)C(=O)NC3CCCC3)C2)C1 2567,CCC(C)CCCC(=O)N1CC2(CC2)CC1C(N1CCC2(CC1)N=N2)=O 2568,C(CCCC(C)NC(c1cnc(Cl)s1)=O)NC(C1(CC)CC1(F)F)=O 2569,C1(C(=O)NC(CSC)C)CC2CC1CN(C(c1ccc(O)cc1F)=O)C2 2570,C=C(C)C1OCCCC1C(N1CCC1CNC(c1cc(C)n(C)n1)=O)=O 2571,C(=O)(CC(O)C(Cl)(Cl)Cl)N1C(CNC(Cc2c(C)ccc(F)c2)=O)CCC1 2572,C1(CC#C)(C(N2CC(CC=C)(NC(=O)C(O)Cc3cnc[nH]3)C2)=O)CCCCO1 2573,N1(C(C2(CC)CC2)=O)CCOC(C)(C)CC1 2574,C1(C(N2CCC(C)(F)C2)=O)N(C(=O)Cc2nc(=N)[nH][nH]2)CC12CCCC2 2575,c1(CC)n[nH]c(CC)c1CC(=O)NCC12CC1CN(C(C1(C)CC(F)C1)=O)C2 2576,C(=O)(C(C)(C)CC#N)NC(C(C)C)CCN(C(=O)C(c1ccccc1)C1CC1)C 2577,C#Cc1cn(C)nc1C(=O)NC(C)CC(C)NC(=O)C(C)(C)C#C 2578,c1(NCC2N(C(c3c(C)ccc(F)c3)=O)CCCC2)ncnc2[nH]cc(C)c12 2579,C1(CNC(C2(C(CC)(F)F)CC2)=O)(NC(=O)Cc2ncccc2C)CCOCC1 2580,N1(C(C(CC)CO)=O)CCC(O)(C2(NC(=O)CSC(F)(F)F)CC2)CC1 2581,C1(CNC(C2(CC)CC2)=O)CN(C(=O)Cc2cn3ccccc3n2)CCC1(C)C 2582,c1(OC)c(C)n[nH]c1C.C(CCC(=O)N1CCC(C2CCCN2CC)C1)OCCO 2583,C(=O)(CC(C)C(C)C)NCC(CC(C)C)NC(c1scnc1C1CCCC1)=O 2584,C1(C(c2nnnn2CCC2CC2)NC(C)C(=O)NCc2cscn2)CC2CCC1CC2 2585,CN1CCN(C(=O)C=Cc2ccc[nH]2)C(C(=O)N(C2(C)CC2)C)C1 2586,CC1(C)OCC2CC12C(=O)NC1CC(NC(=O)C(c2ncccc2F)(F)F)C1 2587,C1(CNC(CCc2cccc(OC)n2)=O)CCCCN(C(=O)CCS(C)(=O)=O)C1 2588,C(CC=C)(CC(=O)N(CC(C1CCCC1)O)C)NC(C(C=C=C)C)=O 2589,C(C(=O)O)(C(C)OC)NC(CNC(C1CCN(CC)C1)=O)=O 2590,Cc1c(C(=O)NC2CCC23CN(C(C2COC(=O)C2)=O)C3)oc2ccc(F)cc12 2591,Cc1c(NC(=O)CN2CCN(C(c3ccccc3O)=O)CC2)cnn1C 2592,C1(CNC(=O)CCC2(C)CC3(CC3)C2)CCCC(c2ccccc2)CC1 2593,C1(C(=O)NC2(CC=C)CC2)CN(C(c2c(C)cccc2C)=O)CCC1(C)C 2594,c1(N(C(C)CCNC(c2ncn3ccccc23)=O)C)ncnc(Cl)c1C#N 2595,C=C(C)CCCC(=O)N1CC(CNC(c2c[nH]cc(Cl)c2=O)=O)C(C)C1 2596,CCC1=C(C(=O)NC(CNC(=O)Cn2nccn2)C2CCC2)CCCO1 2597,c1(C(N(CC(C)NC(C2(C)CCCCO2)=O)C)=O)ccnc(C2CC2)c1 2598,c1(C(=O)OC(Cc2ccc(OC)cc2)C)ccc2cc(OC)ccc2c1 2599,S(=O)(=O)(C1CN(C(=O)CCC(C)O)C1)N1CCN(C(C(COC)OC)=O)CC1 2600,N1(C(Cn2c(C)ccn2)=O)CCC2CCN(C(=O)CCC3CCCCO3)CC12 2601,c1(OCC)ccc(F)cc1CC(=O)NCC(C1CCC1)NC(c1ncsc1C)=O 2602,c1(N(CC(CN(C(C2CN(CCOC)C(=O)C2)=O)C)O)C)nc(C)nc(=N)[nH]1 2603,C1(C)(NC(c2cn(CCNC(CC=C)=O)nc2)=O)CN2CCC1CC2 2604,c1(NC(C2(C(=O)NCc3cc(C)nn3C)CC2)=O)cc(Br)cc(Cl)n1 2605,C=CCC(C(=O)N1CC(C(=O)NC2(CO)CCC(C)C2)OC(C)C1)C(C)C 2606,N1(C(CC(COC)C)=O)CCC(F)(CNC(C2(C)CCC(C)C2)=O)CC1 2607,C1(=CCC)CN(C(=O)C(C)NC(=O)C(C)SC)C1 2608,C1(NC(CCC(=O)OC)=O)CCN(C(C2CCCC2OC)=O)CC1C 2609,C1(CN(C)C(c2ncccc2O)=O)CN(C(=O)Cn2ccccc2=O)CC12CC2 2610,Cn1ccc2c(C(=O)NC3CC(O)CN(C(c4coc(Cl)n4)=O)C3)[nH]cc2c1=O 2611,C1(CNC(CCCC=C)=O)(OC)CCN(C(c2ccnn2CCF)=O)CC1 2612,C1(Cn2cc(C(C)O)nn2)CN(C(c2csc(-c3ccoc3)n2)=O)CCO1 2613,N1(C(c2nc(CNC(C(CC)C(C)C)=O)oc2)=O)CC(C)CC(C)(C)C1 2614,C12(CC1)C(=O)N2.C(CCN(C(=O)CN(C)CC)C(C)C)OCC 2615,N1(CC2CC(=O)N(Cc3ccco3)C2)CCC(O)(c2cccc(Cl)c2)CC1 2616,c1(NC(C(C)(C2CCC2)NC(c2cc(CCC)[nH]n2)=O)=O)sccc1C#N 2617,C1(C)(CC)C=C(C(=O)N2CC(CNC(=O)CCc3nccs3)C(O)C2)C1 2618,N1(C(c2nccc(C#C)c2)=O)CCC(C(=O)NCC(F)(F)CO)=C(F)C1 2619,C1(OCC)CCN(C(=O)C(C)(C)NC(C2CCC(F)C2)=O)CC1 2620,CC(=O)CCCCC(=O)NCC(C)(C)OCC(=O)NC(C1CC=CCC1)CO 2621,N1(C(c2ncn(C)n2)=O)CC(O)CC1CNC(c1cc(C2CC2)n(C)n1)=O 2622,C1(CNC(C2CC(C)=C(C)CC2)=O)COC(C)(C)CN1C(=O)COC1CCC1 2623,C1(CNC(CCC(=C)C)=O)CC2CCC1N2C(c1cccc(-n2cncn2)c1)=O 2624,c1(C(=O)NC2(C(N(CCC#C)CCOC)=O)CC2C)ncc(F)cc1F 2625,C1(OC(c2ccc(-n3cncn3)cc2Cl)=O)CCOC2(CCCC2)C1 2626,C12(NC(Cc3nc(C(C)(C)C)sc3)=O)CC1CN(C(C1CCC(C)(C)C1)=O)C2 2627,c1(C(N(C(CN(C(Cc2cn(CC)nc2)=O)C)C)C)=O)ncncc1C 2628,C(C)(CO)(C(=O)N1CC(CCNC(c2cnn(C)c2Cl)=O)(OC)C1)OC 2629,c1(C(=O)NCCCOC(CC)=O)cc(-c2ccncc2)ccn1 2630,c1(C(N(CC(CNC(CCOCCOCC)=O)C)C)=O)cnn(CSC)c1C 2631,c1(C(N(C(C)CNC(=O)C(F)OC(F)(F)F)C)=O)cccc2ccc(O)nc12 2632,C(=O)(CCN=c1cc[nH]cc1S(=O)(=O)NC1CC(n2cccn2)C1)NC(C)C 2633,c1(OC)ccc2c(n1)NC(C(N1CCC(NC(=O)CC(C)C)C(CO)C1)=O)C2 2634,c1(C(N(CCNC(CCN(C(C)=O)C)=O)C2CC2)=O)ncc(F)c2ccccc12 2635,N1(C(C(C=CC)O)=O)CC(F)(F)CC1CNC(=O)Cn1cc(C)cn1 2636,Cc1cc(C)c(C(=O)NC2COCCC2NC(c2conc2C)=O)c(O)n1 2637,C(C(=O)NC1CCN(C(=O)C=Cc2ccc(C)o2)CC1C)(C(F)(F)F)OC(C)=O 2638,CC(O)CCCCCC(=O)NC1CCN(C(=O)CC2CCCCCC2)C1 2639,CC1(C(=O)NCC2(NC(C3CCC4CC34)=O)CCOC2)CCn2ccnc21 2640,C(=O)(C1CCCCc2ccccc21)NCCN(C(=O)C(C)C#N)CC 2641,CC1(C)CN2CCN1N1CC3(CCC(O3)C2=O)C1.[SH](=O)(=O)C(F)(F)F.CCO 2642,c1(-c2cn(C(C)C)nc2CNC(C(C)CC(C)(C)C)C2CC2)cc2ccccc2[nH]1 2643,C(=O)(CC(C)C(=O)O)N(CCn1cc(-c2ccc(F)c(F)c2)nn1)CC 2644,C(=O)(CC1=CCCC1)NC1CC(C)(NC(C2(Cc3ccccc3)CCOC2)=O)C1 2645,c1(C(=O)Nc2scc(-c3c(CC)cc(F)cc3)n2)n[nH]c2c1CN(C)CC2 2646,C1(C(N2CCC(NC(CC3CC(=O)C3)=O)C2)=O)CC2(CCOCC2)C1 2647,N1(C(C2CCC(C)(C)OC2)=O)CC2CCCC2C1C(N1CC2CSCC(C2)C1)=O 2648,C1(CNC(CCNC(=O)OC(C)(C)C)=O)CCN(C(=O)Cc2ccoc2)C1 2649,C(CCC)(C(=O)NCCCN(C(C1CC1c1ccn(C)n1)=O)CC)=CCC 2650,C=C(C)C(C)(O)C(=O)N1CCCC(C)(NC(c2cccc(CC(F)(F)F)c2)=O)C1 2651,N1(C(C2(NC(C(CC(C)(C)C)OC)=O)CCN(C)C2)=O)CCC2(COC(=O)N2)C1 2652,C(C(=O)NC1(C(=O)OCCOC)CCC1)(C1=CCSC1)N(CCCC)C 2653,C12(CNC(c3cn(CCC)nn3)=O)CCC(CC1)N2C(c1conc1C1CC1)=O 2654,c1(C(=O)NC2COCC2CNC(C2CC2C2CCC2)=O)nccc2[nH]ccc12 2655,C12(CSC)CC(C(N3CCC(N(C(=O)CC4(O)CCCCC4)C)C3)=O)(CO1)C2 2656,C(=O)(C1CCCc2nncn21)NC1C(C=C)CN(C(C2(n3cnnn3)CC2)=O)C1 2657,C=CCC(CC)C(=O)NC1(CC=C)CCN(C(=O)C(C)(C)c2cscc2Cl)CC1 2658,Cc1cc(F)cc(C)c1C(N1CC2CCC1CN2CC1CCS(=O)(=O)CC1)=O 2659,c1(CC(N2C(CC)C(NC(=O)C(C)CSC)CC2)=O)ccc(C)cc1C 2660,N1(C(C(F)=CC)=O)CC(C)(NC(=O)CC(NC(=O)O)SC)C1.C(C)(C)(C)OC 2661,CC1=C(C(=O)NC2CC2NC(=O)CNC(=O)CC2CCCC2)CCS1(=O)=O 2662,CC1(NC(=O)CCCc2c(F)cccc2Cl)CCCN(C(=O)CNS(C)(=O)=O)C1 2663,C#CC1(O)CC(C(=O)NC(C)C=CC(=O)NCc2nncn2CC)C1 2664,C(=O)(C1=NNC(=O)C1)N1CC(CNC(=O)CCC=Cc2ccccc2)C1 2665,c1(NC)cnc(C(N2CCC(C)(CNC(c3ncccc3C3CC3)=O)C2)=O)nc1 2666,C1(C(=O)NCC2C(C(=O)NCCc3n(C)cnn3)C2)CC(=O)CCO1 2667,CC1(C)CCN(C(=O)CCC2CCOC2)C1C(N1CCOCC1C1CC1)=O 2668,C1(F)(C(=O)NCC2C=CC(NC(C3CCN(c4nncs4)C3)=O)C2)CCCCC1 2669,N1(C(c2cccc(C(=O)OC)n2)=O)CCC(NC(C2(C(C)(F)F)CC2)=O)C(O)C1 2670,c1(C(=O)NC2CCCN(C(C=C(C)C(C)(C)C)=O)CC2)c[nH]c2c(F)cccc12 2671,C1(C(=O)NC2CC3CN(C(c4ccc(C#N)cn4)=O)C2C3)CCCCC1C1CC1 2672,N1(c2cc(NCC3CSC3)nc(C)n2)CCC(C)C(C)(C)C1 2673,C1(C(N(CCC(C)(C)NC(=O)Cc2nc[nH]n2)C)=O)CC(S(C)(=O)=O)C1 2674,c1(-c2nc(SC3C(=C)COC3)on2)ccccc1F 2675,c1(C(=O)NCC2(C)CCN(C(CC(=C)C)=O)C2)cc(OC)cc(Cl)c1F 2676,C1(C(N(c2cnn(C)c2)C)=O)CCCCCCN1C(c1cnn(C)c1Cl)=O 2677,c1(CNC(C2ON=C(CC)C2)=O)n[nH]c2c1CN(C(=O)C(C)(C)SC)CC2 2678,c12ccc(cc1)CC(=O)N2CCOC.C(C(=O)OC(C)C)NC 2679,C1(NC(c2n(C(C)C)ncc2)=O)CCCC(NC(=O)C(C)(C)c2cnc[nH]2)C1 2680,C(=O)(CCC(=O)NC(c1ccccc1)CNC(=O)CSCC1CCCCO1)OC 2681,CCC(C)(O)C(=O)NCC1(C)CC(NC(=O)Cn2nccn2)C1 2682,C1(C(C)C)C(C(C)C)CN1C(=O)C(C1(O)CN(C(C2(F)CCC2)=O)C1)F 2683,c1(COC)ccsc1C(=O)N(C(C)CCNC(c1ncn(C(C)(C)C)n1)=O)C 2684,C1(NC(C2CCC(C)CN2C(c2c[nH]c(C(N)=O)c2)=O)=O)CCn2nnnc2C1 2685,CCCC(O)CC(=O)NCCN(C1CCCC1)C(=O)CN(CC(C)(C)C)C 2686,N1(C(C2(CNC(C(C)C3CCCC3)=O)CC23CCC3)=O)CCC2(CCCCC2)C1 2687,Cc1cc2[nH]c(C(=O)NCC3CC3NC(c3ccc(Br)c(N)n3)=O)cc2o1 2688,C1(NC(CCOCC#C)=O)CCCCC12CCCN(C(c1ccc(C)o1)=O)C2 2689,C(CC(C(C)(C)C)NC(c1c[nH]ccc1=O)=O)N(C(=O)CC1(C(F)(F)F)CC1)C 2690,C=C(C)CCC(C)OC(c1ccc(-c2ccncc2C)s1)=O 2691,c1(N(CC(=O)NCC)CC2CCCCC2)ncc(C(F)(F)F)n1C 2692,C(CN=c1nc2ncn(C)c2c(NCCC(COC)OC)[nH]1)N(CCO)CC 2693,C1(c2ccn(C)n2)CN(C(=O)CCCCN)C(C)(C)C1 2694,c1(C(=O)NCC2(NC(C(C=C=C)C)=O)CC(F)(F)C2)ccc2nonc2c1 2695,C1(CNC(=O)C=C2CCC2)CCCCC1NC(=O)C(=O)NC1CC1 2696,C12(C(=O)NCC3(CCNC(c4cnc(SC)[nH]4)=O)CC3)CCC(CC1O)C2 2697,C(C(O)CNC(C1CCSC1)=O)N(C(C=C(C)Cl)=O)C 2698,Cc1cc(S(=O)(=O)NCC(=O)OC(c2ccccc2)c2ccco2)cc(C)c1Cl 2699,C1(NC(N(C)CCC(C)(C)C)=O)CN(C(=O)OC(C)(C)C)C2(CCCC2)C1 2700,N1(C(C2C(=C)C2)=O)CCOCC(NC(c2cnc(C)c(CC(C)C)c2)=O)C1 2701,N1(C(C(C)CC2CCC2)=O)CCN(C(N2CCN(C(=O)C3=CCC3)CC2)=O)CC1 2702,C(C)(C(C(=O)N1CC(O)CC1CNC(=O)C(c1ccccc1)=O)N(C)C)OC 2703,C1(F)(CNC(c2ccc(CC)nc2)=O)CCC(CNC(=O)Cc2ccsn2)CC1 2704,C1(N(C)C(c2ccccc2C(N2C(C)C(C)(C)C2)=O)=O)(CO)CC2CCCC12 2705,c1(C(=O)NC2CCC(NC(C(COC)OC)=O)C2)nn(C)cc1C 2706,C(C(C)(CC)C(=O)NCC1CC1C(C)C)NC(CC(=C=C)C)=O 2707,Nc1cc(Cl)c(Cl)cc1C(N1CC2C(CNC(c3ccnnc3)=O)C2C1)=O 2708,O=C(C1=CCCOCC1)NCC1CC2CCCC2N1C(c1cc(C2CC2)on1)=O 2709,C12(CNC(c3c(CC)nc[nH]3)=O)CCCC(CN1C(=O)C1=NOC(C)C1)C2 2710,C1(NC(N2CCC(C(=O)NCCCC3CS(=O)(=O)C3)C2)=O)CCN(S(C)(=O)=O)C1 2711,C1(OC)CN(C(C2CCN2Cc2ccccc2)=O)CC1NC(c1c[nH]nc1C)=O 2712,Cc1oc(C(F)(F)F)c(C(=O)NC2CC(CNC(C3CCCSC3)=O)C2)c1C 2713,c1(OCC)cccc(C(N2CC(O)(CNC(C3CCC3C(F)(F)F)=O)C2)=O)c1N 2714,C(CC)(C(=O)N(CCCNC(c1nsnc1O)=O)CC1CCCC1)=C(C)C 2715,C1(CCCCNC(CCSCCC)=O)CCN(C(c2c(SC)cnn2C)=O)CC1 2716,C1(NC(c2c(CC)cccn2)=O)CN(C(=O)COc2ccsn2)CCC1CO 2717,c1(C(=O)NC(COC)CNC(c2coc(Cl)n2)=O)cc(O)cnc1Cl 2718,C1(NC(=O)Cc2nc[nH]n2)CC2(C(=O)NCC(Cl)Cl)COC1C2 2719,N1(C(C2CC(C)(C)O2)=O)CCCC(O)(CNC(=O)Cc2csc3nccn23)CC1 2720,CCCC(C)C(=O)NC1(COC)CN(C(=O)CC2(C)CCCC2)C1 2721,c1(C(N2CCC3(C(NC(C4C(=C)C4)=O)C3)CC2)=O)cc2cncn2c(O)n1 2722,N1(C(C(c2cccc(C)c2)C)=O)CC2CC(NC(c3c(C)n[nH]c3C)=O)C2C1 2723,C(=O)(CC(F)(F)C(F)(F)F)NCCC(C)NC(C1CC1(Cl)Cl)=O 2724,N1(C(C(C)NC(CC)=O)=O)CCN(C(c2ccc(C(C)(C)C)nc2)=O)C(CO)C1 2725,c1(C(N)C)cccc(N(C(C2CC3C=CC2C3)=O)C(C2(c3ncccn3)CC2)=O)c1 2726,CCCC(C(O)C(=O)N(C)CC1CC1(C)C)NC(c1ncc(C)cc1C)=O 2727,C1(CNC(CCC=CC)=O)COCCN(C(c2cnn(C)c2C)=O)C1 2728,CC(C(=O)NCC1(C)CCCN1C(c1n[nH]cc1Br)=O)P(C)(C)=O 2729,C1(C)(CNC(=O)NCC2(NC)CCCC2)COCC(C)(C)O1 2730,C1(C(N2CCC(O)(CN(C(C3(CC)CC(C)(C)C3)=O)C)C2)=O)CC2C=CC1CC2 2731,C1(NC(CC2(OC)CC2)=O)COCCN(C(C2CC3C(C2)C3(F)F)=O)C1 2732,CCCC(C)(O)C(=O)N1CCC(NC(c2cccc(CSC)c2)=O)C1 2733,C1(N(C(CN(c2ccccc2)C)=O)C)CCC(NC(=O)CCCC2CC2)C1 2734,Cc1nc(C)c(C(=O)NCC(O)CNC(c2ccsc2)=O)o1 2735,N1(C(COCCC=C)=O)CCCC(C)(NC(=O)C(C)Oc2ccccc2C#N)C1 2736,C1(C(=O)NCCCS(N)(=O)=O)CC12CCN(c1cc(C(F)(F)F)ncn1)CC2 2737,C1(CN(C(=O)Cc2cn(C3CC3)cn2)C)CCCN(C(c2cnc(Cl)n2C)=O)C1 2738,c1(C(=O)NCC(CNC(c2n(CC)ncc2)=O)O)cc(C(F)F)cc(C)c1 2739,Cc1c(C(=O)N(CCNC(C2CC23CCC3)=O)C2CC2)cncc1Br 2740,C(=O)(N1OC2C=CC1CC2)c1nc(CNC(CC2N(C)CCC2)=O)oc1 2741,Cc1ncnc(C)c1OCC(=O)NCCC(C)CCNC(c1ccc(O)nn1)=O 2742,c1(NC(C(c2cnc(CCOC)s2)N(C)CCN(C)C)=O)ccc(C)cn1 2743,C1(C(=O)NCC(C)(C)C(N)=O)CCCCCN1C(=O)CCC1CCC(=O)C1 2744,C(N=c1ccc2c([nH]1)CCCCC2=O)C1(C)CCN(C(C(CCC)C)=O)CC1 2745,N1(C(CC(C)(C)N(C)C)=O)CCC(C2CCCN(C(=O)Cc3c[nH]nc3O)C2)C1 2746,C1(NC(CSCC(C)C)=O)CN(C(C2(C#N)CCCC2)=O)CC(C)(C)C1 2747,S(=O)(=O)(c1ccc(F)cc1C)N(c1cc(SC)nc(C)n1)C1CCNCC1O 2748,C(=O)(N(OC)C1CCC1)c1c(CC(=O)NC)c(CC(CC(=O)OC)=O)c(C)[nH]1 2749,N1(C(CC2CC(OC)C2)=O)CCCOC(C2CCC2)C1.C1(C)(C)CC(=O)N1 2750,N1(C(C(C)OCCC=C)=O)CCCCC1CNC(=O)CC(O)C1CCCC1 2751,c1(COC)nc(C(=O)NC(C)(CNC(C2CC2F)=O)Cn2cccn2)co1 2752,C(=O)(CC(C)C(C)C(C)C)NCC(CC)(CC)NC(c1n[nH]c2ccccc12)=O 2753,C1(OC)CC(C(=O)NCc2ncon2)N(C(c2ccc(Br)cn2)=O)C1 2754,N1(C(c2c(CC)cns2)=O)CCCCC1CN(C(=O)CN1CCC(C)C1)C 2755,c1(C(=O)NCC2CC2NC(C2(F)CCC2)=O)c(Br)ccc2ccccc12 2756,CC1CCc2c(C(=O)NCC(C)(O)CNC(=O)Cn3ncn(C)c3=O)csc2C1 2757,C(=O)(C1=CCCCC1C)N(CC(CO)(CO)NC(CC(C=C)(C)C)=O)C 2758,S(=O)(=O)(c1cnc(C(C)(F)F)s1)NCC(C(=O)OC)Cc1ccncc1 2759,C1(CC(=O)NCC2CC(OC)CN2C(=O)C=CC(C)C)CC2(CCCC2)CO1 2760,c1(C(C)NC(C2CSCCN2C(c2nccn2C)=O)=O)cc(Cl)ccc1O 2761,c1(C(N2CC(OCCNC(CN3CCC(C)CC3)=O)C2)=O)ccc(F)nc1F 2762,c1(OCOC)cc(-c2ncsc2C(=O)NCCc2ccccn2)c(F)cn1 2763,Cc1nc(C(=O)N(CCCN(C(=O)C(O)C2CC2)C)C)c(Br)s1 2764,C(=O)(C(C)C(C)NC(=O)CCn1cccn1)NC(c1nc(C)on1)(C)C 2765,C#CCCCCCCC(=O)N1CCC(C(C)C(N2CC=CC2CF)=O)CC1 2766,C1(N(C)C)(C=O)CCCC1.C(=O)(CCNC(c1ccsc1)=O)NC(CC)C1CC1 2767,c1(N2CC(O)(C(C)NC(CC(C(C)C)O)=O)C2)ccc(S(=O)(=O)N(C)C)cn1 2768,N1(C(c2c(C)cc(CO)o2)=O)CCN(C(=O)C=Cc2cc[nH]c2)C2CCCCC12 2769,Cc1cc(Cl)ccc1OCC(=O)NCCC(C)N(C)C(C1COC(=O)N1C)=O 2770,Cc1ccc2c(N(C)CCOCCO)nc(N3CCC(CN(C)C)C3)nc2c1 2771,Cc1c(C(=O)NC(C)(C)CNC(=O)C(F)CC2CCCC2)cccc1N 2772,c1(OC)ccc(S(=O)(=O)N2CCC3CN(Cc4cccc(Cl)c4Br)CC23)cc1 2773,C#CCC(C)C(=O)NC(CNC(c1cncc(SCC)n1)=O)CCCC 2774,Cc1coc(C)c1C(=O)Nc1ccccc1.N12CC3C(C3C1)c1cn(nn1)CC2 2775,N#Cc1ncc(C(N2CC=CC(NC(=O)Cc3csc(C(N)=O)n3)C2)=O)s1 2776,Cc1nn(C(C)(C)C)cc1C(=O)NC1CCN(c2cccnc2)C1 2777,CCC(CC)C(=O)N1CCC1C(=O)Nc1cnn(CCO)c1 2778,Cc1c(O)ccc(NC(=O)CC2CC(NC(c3cccc(O)c3O)=O)C2)c1C 2779,C(C1COc2ccccc21)NS(=O)(=O)Cc1nnsc1C(F)(F)F 2780,c1(C(=O)NCCCN(C)C(C2CCCNC2=O)=O)scc(Cl)c1Cl 2781,Cc1ccc(C=CCC(N2CCC(CNC(=O)CC(C)O)C2(C)C)=O)cc1 2782,C(CC)(CCCC(=O)N1CCOCC1C(C)O)NC(CCCCCC)=O 2783,C12(C(=O)OC)CC(C(=O)N(CCCN(C(=O)CSc3n[nH]c(O)n3)C)C)(C1)C2 2784,N1(C(COCC)=O)C(CNC(c2nocc2C(C)(C)C)=O)CC2CCCCC12 2785,c1(C(=O)NC(c2cn(-c3ccccc3Br)nn2)CCC)sc(C)cc1Br 2786,c1(C(N2CC3(CCN(C(C(CCC)OC)=O)C3)C2)=O)ccc(Br)c2cn[nH]c12 2787,C(=O)(C1=CN=C2N=CNN2C1)NC1(C)CCCN(C(C2(F)CC3(CCC3)C2)=O)C1 2788,c1(OC2CCN(C(=O)CSn3cc(C(=O)O)nn3)C2)ccc(Br)cc1 2789,C1(NC(c2cc(C)no2)=O)C2CCC(C2)C1C(=O)Nc1cc(C(N)=O)cc(Cl)c1 2790,c1(CC(=O)N(CCN(C(=O)C=CC2CCCN2C)C)C)ccc(C(F)(F)F)cc1 2791,c1(O)c(C)ncnc1C.C1(SC)CC(NC(=O)NCC(=O)NC2CCCC2)C1 2792,C1(CC(=O)NC(=O)CN2CCCC2C(C2CC2)CC2CC2)CCCC12CC2 2793,N1(CC(N2CCC(C(C)(C)NC(C(CC=CC)C)=O)C2)=O)OC(C)(C)CC1=O 2794,C1(CCCNC(CCCC)=O)CCN(C(=O)C(C)(C)Oc2ccc(Cl)cc2)CC1 2795,c1(C(=O)NC)cc(NC(=O)C(C)n2ccnc2)cc(Cl)c1 2796,c1(CC)nc(NC(=O)NC2CN(C)CC2C)cc(Nc2ccccc2)n1 2797,c1(C(N(CC(C)NC(=O)CN2CC=CC2)C)=O)cn2c(n1)CCC2 2798,c1(C(N(C)CCNC(c2cccn2C)=O)=O)cc(F)cc(F)c1 2799,C1(C(=O)NC(C2CCN(C(C3(CC=C)CCOC3)=O)C2)C)CN=C2N=CNN2C1 2800,C1(C(=O)NCC2N(C(CS(CC)(=O)=O)=O)CCN(C)C2)CC2(C1)CS(=O)(=O)C2 2801,C#CC1(C(=O)NCCC2CC(C)(C)C2)CCN(C(=O)CCC2CCCO2)CC1 2802,C12(NC(C3N(CC)CCOC3)=O)CCOC(CNC(=O)C(C3CC3)SC)(C1)C2 2803,CC(CNC(=O)C=CC(=O)NC1CC1)(CO)NC(=O)CO.C1(S)CCOC1 2804,C1(C(=O)NC2C(C)CCN(C(C3CCS3(=O)=O)=O)C2)CCC2(CC1)CNC(=O)C2 2805,N1(C(=O)CSc2nncs2)CC(C2CN(C(c3ncc(Cl)cc3F)=O)C2)C1 2806,Cn1cnc(C(C(=O)NCC2CCOC2)N(CCCCO)C)n1 2807,C(C)(C(O)C(=O)N(CC(C)(C)CNC(C1CCC=CCC1)=O)C)OC 2808,C1(CC)CN(C(c2coc(CNC(=O)C(C3(O)CCCC3)F)c2)=O)CCS1 2809,c1(OCC(=O)NCC2(F)CCC(NC(c3ccc(CO)o3)=O)C2)cccc(F)c1 2810,N1(C(c2nc(CCCC)sc2)=O)CCC2CN(C(c3cnc(C)cc3Cl)=O)CC12 2811,c1(OC)cnccc1C(N1CCC1(C)CC(N1CC(O)C1)=O)=O 2812,N1(C(c2cc(OC)n(C)n2)=O)CCC(C(N2CC(O)(CO)C2)=O)C12CC2 2813,c1(OC(CC)C)ccc(C(N2CCCC(CCNC(=O)CC(F)(F)F)C2)=O)cc1 2814,N1(C(=O)CN2CCOC2=O)CCOC2CN(C(c3ncc(Cl)cn3)=O)CC12 2815,CCCCC(C)C(=O)NC1CC(CNC(C2(C(F)(F)F)CC=CC2)=O)C1 2816,C12(CNC(c3c(C)nn(C)c3)=O)CC(CCO1)N(C(=O)COC(C)(C)C)C2 2817,C1(F)(C(=O)NCC2N(C(CC(=O)NC)=O)CCC2C)C(C)(C)C1(C)C 2818,C(CCC(C)(C)NC(C1CCCN1S(C)(=O)=O)=O)NC(CN(CC(C)(C)C)C)=O 2819,CC1(NC(C23CC(CN2C(C2CN4CCC2C4)=O)C3)=O)CC2CCC1C2 2820,c1(C(N2CC3(CCN(C(C4CC(=O)NC4)=O)C3)C2)=O)ccc2c(c1)COCCN2 2821,C(=O)(C(F)CC(C)(C)NC(=O)C1=NOC(C)C1C)N1CCC(COCC)C1 2822,CC(C)(CNC(c1cncs1)=O)CC(=O)NC1(CO)CC(F)C1 2823,CCC(C(=O)NC)NC(C1CC(O)(CNC(C2(C(=O)OC)CC2)=O)C1)=O 2824,N1(CC)C(=S)NC(c2cc(C(C)C)no2)C=C1CCN(C)C 2825,C(=O)(C(C)(C)CS(N)(=O)=O)NC1CCN(C(C2(Oc3cn(C)nc3)CC2)=O)C1 2826,CC1NC(=O)CCC1CNC(=O)CC1CCN(C(C2CC(=C3CCC3)C2)=O)C1 2827,N1(C(c2c(OC)cc(Cl)cc2)=O)CCn2nnc(C(=O)NC3CCOC3)c2C1 2828,CC#CCCCC(=O)N1CCC(O)C(NC(=O)CC2CCCC(C)(C)C2)C1 2829,CC(C)C(CO)C(=O)N(C(CNC(c1cnn(C2CC2)c1)=O)C1CC1)C 2830,C1(C(=O)NCC2(SC)CCC2)CN(C(=O)CCc2ccoc2)CCO1 2831,c1(CN2CC(CC(=O)NCc3nc(C)[nH]n3)OCC2)cccc([N+](=O)[O-])c1 2832,C1(O)(CCNC(c2ccccc2Cn2cnnn2)=O)CCCN(C(=O)C2CC2)C1 2833,c1(CNC2CCC(NC(c3c(Cl)ncc(C)c3)=O)C2)ccc2nc(O)[nH]c2c1 2834,C1(CN(C)C(C2CC3(CC3)C2)=O)CCCN(C(c2snnc2C2CCC2)=O)C1 2835,N1(C(C2C(=C)CC2)=O)C2CCCC1CC(CNC(c1c(Cl)ccc(F)c1N)=O)C2 2836,Cc1cccc(CC(c2ncc[nH]2)NC(=O)N(C)Cc2ccccc2C)c1 2837,C1(C(C(=O)OC(C(COC(C)(C)C)N(C)C)=O)CCF)CN(CC)CC12CC2 2838,Cc1nn(CC(N2CC(NC(C34CCCC3(C(N)=O)C4)=O)CC2CO)=O)c(=O)o1 2839,c1(NC(CN(C(CC2ON=C(C)C2)=O)CC2CC2)=O)ccc(C)nc1O 2840,CC(C(=O)N1OC2C=CC1CC2)C1CCN(C(C2CC(C)(C)CO2)=O)C1 2841,c1(-c2cc(Cl)cc(Cl)c2)nc(-c2ccccn2)nn1C1CCCc2ccccc21 2842,c1(CC)c(C(N2CCC(CF)(NC(c3oncc3C)=O)C2)=O)cccc1C 2843,c1(SCC(N2CCOC(Cc3ccc(Cl)cc3)C2)=O)ccccc1F 2844,C1(CNC(c2c(CNC(CCC3(C)CC3)=O)ccs2)=O)C(C)(C)C1(C)C 2845,CCCCC(C(=O)N1CCN(C(=O)CCOC)C(C2CC2)C1)COC 2846,N1(C(C(CC)COC)=O)CCOC2CN(C(=O)C(C)Cn3ccnc3)CC12 2847,N1(C(C2CCCCC2CO)C(=O)NCC(C)C)Cc2cccc(N(C)C)c2C1 2848,c1(C(=O)NC(C(CO)NC(c2csc(C)c2C)=O)C)ncc(F)c2ccccc12 2849,N1(C(CNC(C)=O)=O)CCCC2C1CCN2C(c1snc(O)c1Cl)=O 2850,C1(C(=O)NC(CCNC(C(N2CC(C)C2)C)=O)(C)C)CCC(F)(F)C1 2851,CCCC(CCC)=CC(N1CCN(CC(=O)NC2CCOC(C)C2)CC1)=O 2852,FC1(F)CCC2C(CNC(c3nnnn3C3CCCC3)c3ncco3)C12 2853,N1(C(C(C)(C)OC)=O)CCCC(C)(C(=O)Nc2ccc(-n3ccnn3)cc2)C1 2854,CCC(CC(=O)N(C(C)C(C)C(=O)NCCOCCC(C)C)C)CC(C)C 2855,c1(SC)ncc(Br)c(N2CC(NC(=O)C(C)(CO)CO)C(F)C2)n1 2856,N1(C(=O)OC(C)(C)C)CC(CN2CC(C(=O)O)CC2C(=O)O)C2(CC2)C1 2857,N1(C(C(c2cnccn2)C)=O)CCC(O)(C(C)NC(=O)C(F)=CC2CC2)C1 2858,C(c1cccnc1)=CC(=O)NC(CNC(C1CCN1C1CCCC1)=O)CO 2859,Cc1ccc(CCC(=O)N(CC(C)NC(c2c(C)ccn2C)=O)C)c(Br)c1 2860,C1(CCOC)CCCCN1C(=O)COCCn1cc(-c2cnccc2C)nn1 2861,N1(C(CCS(N)(=O)=O)=O)CCOCC2(COCCN2C(c2cccnc2Cl)=O)C1 2862,c1(C(=O)NCC2(NC(C3C(C)=C3)=O)CCCCCC2)cc(C)c(F)cc1N 2863,N1(C(C(=O)OCC)COC)CCC(c2noc(Cc3ccccc3)n2)CC1 2864,c1(NC(NCC(F)F)=N)ccc(Cl)c(N2CCCC2)c1 2865,c1(C(N2C(C(C)NC(C3(C)CC(=C)C3)=O)CCC2)=O)nc(OC(C)C)ccc1Cl 2866,c1(C(=O)NCC2CCC(NC(CC3(C=C)CCOCC3)=O)C2)c(C)ccc(F)c1N 2867,c1(-n2c(C)cc(C)n2)cnc2c(c1)N(C(=O)CC(C)(C(=O)O)N(C)C)CCO2 2868,C1(COC)(CNC(=O)CCCCCN(C)C)CCN(C(=O)CCCCSC)CC1 2869,C1(C(=O)OCC)CN(C(=O)CC2(N(C)C)CC2)C2(CCC2)C1 2870,C1(C(N(C2CCCN(C(C3CCC(=O)N3C)=O)C2)CC)=O)CCC(=C(F)F)CC1 2871,CCCC(CCCNC(c1scc(C)c1Cl)=O)NC(c1ccn(C2CCC2)n1)=O 2872,c1(C(=O)NC(COCCCNC(C(CC#C)O)=O)(C)C)cc(C)n(C)c1C 2873,N(C1CCCn2nccc21)C(C(C)(C)CCCNC(=O)CCN1CCCC1=O)=O 2874,c1(C(=O)NC(CNC(CCCc2ncc(C)o2)=O)(C)C2CC2)ccc(F)c(C)c1 2875,C1(CNC(C=Cc2n(CC)ncc2)=O)C2CCCC1N(C(=O)CCSC)C2 2876,N1(C(Cc2cc(C)nn2C)=O)CCC2CCCC12CNC(c1cnc(C)nn1)=O 2877,C1(C(=O)NCC#CCC)CC2(CCC2)CN1C(c1cc(F)ccc1C)=O 2878,C1(C#N)(C(N(CCCNC(=O)CCCN2CCCC2)C)=O)CCS(=O)(=O)CC1 2879,C(C(CNC(c1cnn(-c2ccc(Cl)cc2)n1)=O)C(F)(F)F)NC(C1C(C)C1)=O 2880,C12(C(=O)NCCCN(C(=O)CCN3CCC(O)CC3)C3CC3)CCCC1C2(F)F 2881,C1(C(=O)NC2CCCC(F)(F)C2)Cc2cc(O)ccc2CN1S(=O)(=O)CCCl 2882,c1(C(=O)NC(C)CCN(C)C(C2CC2C2CCC2)=O)ccc2c(c1)C=CS2(=O)=O 2883,Cc1cc(=NCCC2(N(C)C)CCC2)[nH]c(=NCC2(N3CC(C)CC(C)C3)CC2)[nH]1 2884,C(N=c1cc(C(C)=O)c([N+](=O)[O-])c[nH]1)C1C(C)CCN(C(C(CC)(F)F)=O)C1 2885,C1(C)(C(N(C)CC2CCN(C(CCC(=C)Br)=O)CC2)=O)CC(OC)CN1C 2886,C(=O)(C1c2c[nH]nc2CN1C(c1cc2ccccn2c1)=O)NCCOCCC#C 2887,CCCCC(CC)C(=O)NCCCN(C)C(C1CC1C(C)(C)O)=O 2888,C1(C(N2C(C)CC(CNC(=O)CSCc3csc(=N)[nH]3)C2)=O)CC2C(C1)C2(F)F 2889,C1(C#N)(C(N2CC(COC)(CNC(=O)CCCc3ccncc3)C2)=O)CC1(C)C 2890,C#CC1CN(C(=O)CCN(C(=O)CN(C)CCOC)CC)CC1O 2891,c1(C(=O)NC2C3CN(C(C=C(C)C(F)F)=O)C2C3)ccc(F)cc1C(F)(F)F 2892,c1(C(=O)NC2(COC)CN(C(C3CC(O)C3)=O)C2)cc(C2CC2)nc(O)c1 2893,C(=O)(CC1=NNC(=O)C1)NCC1(O)CCN(C(CCc2cc(C)on2)=O)C1 2894,C1(C)(C(N(CCN(C(C)C)C(C2CCC(F)(F)C2)=O)C)=O)CCCN1C 2895,CC(C)CC(C)CC(C)C(=O)Nc1nnc(SCCCC(C)CO)s1 2896,CC(CCCCCO)NC(=O)C=CC(C)(C)NC(C1CC(=O)OC1(C)C)=O 2897,N1(C(C2CC(C(=O)OC)C2)=O)CCC2C(C1)CN2C(=O)CCCCSC 2898,C12(C(N3CCC(CNC(C(C)(C)OCC)=O)CC3)=O)CCC(OC)(CC1)C2 2899,c1(C(N2CC(C)C(NC(C3CC3C)=O)CC2)=O)ccc2c(c1)CCN2C 2900,C1(NC2CC(C(=O)NC)N(N(C)C)CC2)CN(C(=O)OC(C)(C)C)CCN1C 2901,C(=O)(CC(CC)CC)NC(C(=O)NC(CCCCC)C)COC 2902,Cn1c(=O)c2ccc(NC(=O)NCC3(CCCO)CC3)cc2n(C)c1=O 2903,N1(C(Cc2c(CC)con2)=O)CCC(NC(C2(C)CC(C)=NO2)=O)C(O)C1 2904,N1(C(c2cc(C)oc2)=O)CC2COCCC2(NC(c2cccc3[nH]ncc23)=O)C1 2905,C1(N)COCCN(C(C2(C(=O)N(C)C)CC2)=O)C1.c1(C(=O)OCC)c[nH]n(CC)c1=N 2906,CC1CC(CNC(C2CN(C3COC3)C2)=O)CN1C(=O)CCCCN(C)C 2907,C1(CC=C)(NC(C2(C)CC2(F)Cl)=O)CCN(C(=O)C(C#N)=COCC)CC1 2908,C(=O)(CC(C)(C)CNC(=O)C(c1ccc(C)o1)C)N1C(COC)CCC1 2909,CC1=C(C(=O)NC2CN(C(C3(C(F)F)CCCC3)=O)CC3CC23)CCO1 2910,c1(C(=O)NC2CC(NC(CN(CC)CC)=O)C2)cnn(-c2cccc(F)c2)c1C 2911,c1(C(=O)OC)[nH]c(C)c(C(=O)NC2CN(C(=O)CCC(F)F)CC2(C)C)c1C 2912,C1(C(N2C(C(C(=O)NCCC(C=C)C)(C)C)CCC2)=O)CC12CCOCC2 2913,CCC(C)CCCC(=O)NCC1(NC(=O)COCC(=O)OC)CCCCC1 2914,C1(C(N2C(C(C)NC(c3n(C=C)ncc3)=O)CCC2)=O)CCc2cnnn2C1 2915,N1(C(c2cn(CC)nc2)=O)CC(NC(c2coc(C(C)OC)n2)=O)C2(CCC2)C1 2916,c1(C(N(CCCCNC(C(C2CCCOC2)OC)=O)C)=O)c(C)nnn1C 2917,c1(C(=O)NC)ccc(OCC(=O)NC2CCC2NC(=O)CCc2nncs2)cc1 2918,C1(C(N2CCC(COC)(NC(=O)C=CCOC)CC2)=O)Cc2cccnc2C1 2919,c1(C(=O)NCCN(C(=O)C(C)NC(=O)NC)CC)ccc(N(C)C)c(F)c1 2920,N1(C(C=CCN(C)C(C2CCCC(C)C2)=O)=O)CC2CCCC(C1)N2C 2921,c1(C(=O)NCC2C(CC(=O)N(C(CCO)C(F)F)C)C2)nccnc1N 2922,c1(C(=O)NCC(=C)CCNC(=O)C(F)=CC)cncc(P(C)(C)=O)c1 2923,C(C)(C)(CCC(=O)N1CC(NC(C2CCCCCN2C)=O)CC1CO)OC 2924,n1(C(C)C)ccnc1C(=O)NCC1CC(CC(=O)NC(C2(CO)CC2)C)C1 2925,N1(C(C2(C#N)CC=CC2)=O)CC(C2CCCN(C(=O)CCCN=[N+]=[N-])C2)C1 2926,N1(C(CCn2ncc(C)c2)=O)CCC(NC(C2(c3ccnn3C)CC2)=O)C(O)C1 2927,C1(CC(=O)NCC2C(C(=O)OC)CC2)CCCN(C(=O)CC2CCSCC2)C1 2928,Cc1ncsc1C=CC(=O)NCCC1(O)CCN(C(=O)Cc2ccccc2)C1 2929,C(=O)(C1CCCCn2ccnc21)N1CCC(C(=O)O)(CO)C1 2930,C1(NC(=O)CN(C(=O)Cc2ccsn2)CC2CC2)CCN2CCC1C2 2931,c1(C(=O)NC2C(CNC(CCCNS(C)(=O)=O)=O)C2)c[nH]c2cc(F)ccc12 2932,c1(NC(c2cc(OC)c(-c3cccnc3O)cn2)=O)nccc2occc12 2933,C1(Sc2c(C)non2)CC(F)CN1C(=O)OC(C)(C)C 2934,C1(CC=C)(NC(=O)CCOCCOC)CCN(C(=O)CCc2cscn2)CC1 2935,c1(CC)nc(C)c(C(=O)NCC2(C(N)=O)CN(C(=O)C(Cl)=CCl)C2)s1 2936,C1(C(=O)NCCNC(c2cc3sccc3[nH]2)=O)Cc2ccccc2C(=O)O1 2937,c1(OC)nc(C(=O)NCCCCCN(C(C2CCCC(C)C2)=O)C(C)C)cc(O)n1 2938,c1(C(N2CC(NC(c3cc(C(C)C)[nH]n3)=O)C2)=O)cc(N(C)C)ccc1N 2939,C1(NC(CC2N(CC)C(=O)CC2)=O)CC12CCN(C(=O)CCc1ncco1)CC2 2940,n1(CC(=O)NC2CCCC(NC(c3oc(CC)c(C)c3)=O)C2)nc(O)ccc1=O 2941,C1(NC(CCC=C(C)C)=O)CCOC(C(=O)NCCc2c[nH]nc2O)C1 2942,CCC(CCC(=O)NCC(N1CCN(C(=O)C(c2cccnc2)O)CC1)=O)OC 2943,N1(C(CCC#CC)=O)CCC(NC(c2ncccc2OC)=O)C(C)C1 2944,N1(C(C2(NC(C3CC(CC)C3)=O)CCSC2)=O)CCC2C(=O)NCC2C1 2945,c1(NC(COC2CN(C(C3CC(=C)C3)=O)C2)=O)cccc2c1CCCC2 2946,C(C(C)(O)CC(=O)NC1CCCCN(C(=O)CC2CCSCC2)C1)OC 2947,c1(C(N2CCC(N(C(c3c(CC)c[nH]c3)=O)C)C(C)C2)=O)cc2ccccn2c1 2948,C(=O)(C#CC(=O)NC(CNC(=O)C(=O)N(C)C)C(C)(C)C)NC(C)C 2949,c1(C(=O)OC)ccc(C2CCN2C(=O)CS)o1.n1(CC)ccnc1-c1ccccc1 2950,C(C(=O)N1CCC(C(C)NC(=O)NC)O1)(C1CCCCO1)OCC 2951,C12CCCN1C(=O)NCC(=O)NC2C.C1(C(=O)NCC2CCCC2)CC(C)(F)C1 2952,C(=O)(CN1C(=O)COc2ccccc21)N(C)Cc1cn(Cc2ncon2)nn1 2953,c1(C(=O)NCC2CN(C(=O)CCN3CCCC3=O)C2)cccc(Cl)c1 2954,C1(CNC(C2C=CCN2C(c2cc(C3CC3)no2)=O)=O)CCCCCCC1 2955,C1(C(N(CC(CC)NC(c2cccc(C)c2O)=O)C)=O)CC12CCCCC2 2956,Cc1cc(OCC(=O)N(CCNC(=O)CCc2nc(O)n[nH]2)C(C)C)ccc1F 2957,C#Cc1cc(C(=O)NCC(C)NC(=O)CCC2CC2)ccc1C 2958,C1(NC(c2cn[nH]c2)=O)CC2(C1)CC(C(=O)NC1(CO)CC(F)C1)C2 2959,CC(C)C(O)C(F)(F)C(=O)N(C)CC1COCCN1C(c1ccc2c(c1)CC2)=O 2960,N1(c2nc(C)nc(O)c2)CC2(CN(C(=O)C=Cc3ccco3)CC2CO)C1 2961,CCC(CC(=O)NCCCC1(NC(c2coc(C#N)c2)=O)CC1)SC 2962,c12noc(n1)C1CC21.C(C)(CC#C)N(CCC#C)COC 2963,C1(OC)CCN(C(=O)CN(C(=O)CCCN2CCCC2)C2CCC2)CC1 2964,C1(NC(C(F)=C(C)C)=O)CC2CC(C1)CN(C(C1CCCN1CC(F)(F)F)=O)C2 2965,c1(C(=O)NC(CC(C)NC(=O)Cc2ccon2)C)sc2sccc2c1Cl 2966,c1(C(=O)NCCN(C(c2cc(C(N)=O)c[nH]2)=O)CC)csc2c1CCC(C)C2 2967,c1(CC(=O)NCC2CCN(CC(=O)Nc3cccc(Cl)c3)C2)ccc([N+](=O)[O-])cc1 2968,C12CN(CCN1C(=O)OC(C)(C)C)C2=O.c1(CCC(=O)NC)cnc(C2CC2)o1 2969,c1(CC(N2CCC(C)(CNC(c3ncc[nH]3)=O)C2)=O)cc(O)nc(O)n1 2970,CC1(NC(=O)CN2CCCC2)CCN(C(c2sccc2C(F)F)=O)CC1 2971,c1(C(CNCCC)NC)ccc(NC(c2ncnn2CC2CC2)=O)cc1 2972,C(=O)(C(C(C)(C)C)NS(C)(=O)=O)NCCCN(C(c1cscc1Cl)=O)CC 2973,C(C1CC1)(C1CC1)=CCC1CCN(C(C(N2CCNC(=O)C2)C)=O)C1 2974,C1(=O)CCC(=O)N2CC3C(C3C2)N1.N1(CCC)CCOC(C)C1 2975,c1(C(=O)OC)c(C)[nH]c(C(N2CC(C)(NC(=O)CNS(N)(=O)=O)C2)=O)c1C 2976,C(=O)(C(C)(C)C(F)c1ccccc1)Nc1[nH]nc(N(C)C)n1 2977,C(CCCCC(=O)N1CC(CONC(C)=O)C1)n1cc(COC)nn1 2978,C(CCC(=O)NC(C)CC(C)NC(c1occc1-c1cnn(C)c1)=O)OCCC 2979,c1(NC(=O)NC2(c3ccccc3)C(C)C2)ccc2nc(O)oc2c1 2980,C12(C(N(C(CCNC(C3(CC=C)CCCCC3)=O)C)C)=O)CCOC(C)(C1)C2 2981,N1(C(C2C(CCC)C2)=O)CC(OC)CC(NC(c2cnc(C(C)(C)C)nc2)=O)C1 2982,C12(CO)CN(C1)C(=O)CCCC1(CCC1)N2.c1(C(=O)OC)sccc1CO 2983,c1(NC(N2CCC(C(N)=O)CC2)=O)cc(C(F)(F)F)cnc1O 2984,N1(C(=O)C=CCF)CC2CCCC(C1)N(C(=O)Cc1ccsn1)C2 2985,c1(OC)nc(C)cc(=NC2CC23CC(NC(=O)C(C)CC(N)=O)C3)[nH]1 2986,C1(C(=O)OCCCC2CCCC2)CC2(COC2)C1 2987,c1(OC)cc(C(N2CCCC(NC(=O)CC3SC(=N)NC3=O)CC2)=O)cc(C)n1 2988,C#Cc1cncc(NC(=O)CC23CCC2CN(C(=O)C(C(C)C)NC(C)=O)C3)c1 2989,CN1CC(C)(C(N2CC3(CCN3C(=O)CC3CSCCS3)C2)=O)CCC1=O 2990,N1(C(c2ccc(C)s2)=O)CCN(C(=O)CCCc2ncco2)C(CF)C1 2991,N1(C(CP(C)(C)=O)=O)CC2C3CCC(C2C1)N(C(=O)C=C1CN2CCC1CC2)C3 2992,C(=O)(C1CCCc2nn[nH]c21)NCC1(NC(c2ccc(Cl)c(O)c2)=O)CCOC1 2993,Cc1ccc(C(N2CCCC(C3(NC(c4cncs4)=O)CC3)C2)=O)c2c1CCC2 2994,N1(C(CCCC#CC)=O)CCC2(CCC2NC(=O)CC2OCCC2(C)C)CC1 2995,c1(C(=O)O)cc2oc(CN3CCC4C(C(=O)O)C4CC3)cc2[nH]1 2996,N1(C(C2C(C)(C)COC2)=O)CCN(C(=O)Cc2cnsc2)CC(O)C1 2997,CC1CCCC(C(=O)NCc2cc(C(=O)N(C3CCOC(C)C3)C)n[nH]2)CC1 2998,N1(C(C(CC=C)C(C)C)=O)CCC(C2CN(C(c3ccc(O)nn3)=O)C2)C1 2999,C1(C(=O)NCCN(C(=O)OC)C)C2CC3C(C2NC(=O)C(CC(C)C)OC)C13 3000,Fc1ccc(C(c2nnnn2CC2CC2)NCc2nncn2C2CC2)c(F)c1Br 3001,Cc1nc(CSCCC(=O)NC2CCCC2NC(c2cnc(C)s2)=O)cs1 3002,CC1CCC(C)C1NC(c1c(CNC(=O)CN=[N+]=[N-])nnn1C)=O 3003,c1(CC(=O)OCCC2C(C)(C)CCO2)cccc2nsnc12 3004,Cc1cc(C(=O)NCC(C)(CO)NC(C2CCOC2)=O)nn1-c1ccc(F)cc1 3005,Cc1nn(C)c(NNC(=O)Nc2nccc(C(F)(F)F)n2)c1C#N 3006,c1(C(N2CC(C(=O)OC)CC(O)C2)C(=O)NCCC)ccc(F)c2ccccc12 3007,Cc1ccc(C(=O)NCCCN(CCCNC(=O)C(C)n2ccnn2)C)cc1 3008,c1(C(c2n(CC)nnn2)NCc2ccn(C(C)(C)C)c2)ccc(C(F)F)cn1 3009,C(CCC[Si](C)(C)C)N(c1cc(C)c(-c2cccc(C(C)C)c2)s1)CC 3010,n1(C(C)C)ccc(C(=O)N(C(C)CNC(C2CC2(C)C(F)F)=O)C)n1 3011,C#CCCCCC(=O)NCC12CCC(C1)N(C(c1ccc(C3CCC3)nc1)=O)C2 3012,c1(-c2ccnc(NCC(c3ccccc3C(F)F)(C)C)n2)cccc([N+](=O)[O-])c1 3013,c1(C(N(CCCNC(C=CC)=O)C)=O)cc2cccc(O)c2[nH]1 3014,c1(CC)cc(F)ccc1C(=O)NCC1CN(C(C2CC3C(C2)C3(F)F)=O)CC1O 3015,N1(C(C2(C)CCC2)=O)CCC2(CCOC2)C(CNC(=O)CCCCNC(N)=O)C1 3016,C1(NC(C#CC(C)(C)O)=O)CC2CC1CN(C(=O)CCC(C)(C)N1CCCC1)C2 3017,Cc1ncnc(N2CCC(C)(CNC(=O)Cn3nnnc3C3CC3)CC2)c1Br 3018,C(C1CCCN1C(c1csc(Cl)c1)=O)=CC(=O)N(CCSC)C 3019,C1(NC(c2c(CC)ccs2)=O)CC2CN(C(c3c(C)noc3CC)=O)CC2C1 3020,C1(C(=O)NC(C(C)O)CO)CCCCCC1NC(C1(C)CCOC1)=O 3021,c1(C(N(C2(C(=O)NC(C3CCCC3)C#C)CC2)C)=O)ccc(N)cc1C 3022,n1(CC#C)cc(CNC(=O)C(C)N(C(=O)C=CCN2CCC2)CC)cn1 3023,C(=O)(C(F)(F)C(O)C1CC1)NC1CC2C(NC(C3(C(N(C)C)=O)CC3)=O)C2C1 3024,N1(C(c2cc(Cl)ncc2Br)C(=O)NCC=C)CC=C(c2cccc(Cl)c2C)CC1 3025,C(=O)(CCCC(=O)N1CC2CC2(NC(C2CCC3CCC2O3)=O)C1)NC(C)C 3026,CN=c1ncc(-c2c[nH]nc2C(=O)Nc2cncs2)c[nH]1 3027,C1(CO)CCCN(C(C2(C)CC(C(=O)O)C2)=O)C1.C1(N(CC(=O)NC)C)CCCCC1 3028,Cc1c[nH]cc1C(=O)NCCC(O)CNC(=O)Cc1cnn(Cc2ccccc2)c1 3029,c1(CC)[nH]nc(C(N2CC(OCCNC(=O)CN(C3CCC3)C)C2)=O)c1Cl 3030,Cc1nc2c(cc1C(=O)NCCC1COCCN1C(=O)C=C1CC1)c(C)nn2C 3031,C1(C(N(CCN(C(Cc2cc(CC)no2)=O)C)C)=O)CC12CCC(=O)CC2 3032,Cc1ccc(C(=O)NCc2cc(C#N)ccc2C(F)(F)F)c(N)c1F 3033,C(C(=O)NC1(C2CCCN2C(c2nccnc2N)=O)CC1)(C(C)C)SCC 3034,C(=O)(C(O)CC(C)(C)C)N(CC(CNC(CC(C)(C)OC)=O)C)C 3035,CCCCC(O)C(=O)N1CCC1CNC(=O)CC12COCC(C1)C2 3036,c1(OC)c(F)cc(C(=O)NCC2CN(C(C3CN(C)CCO3)=O)CC2C)cc1Cl 3037,N1(C(c2cc(OC)cc(C)c2)C(=O)NCCCC)CC(C)(C)C12CCOCC2 3038,C#CCCC(O)C(=O)NC(C)CCNC(c1snnc1CC)=O 3039,C1(C(N2CCCC(NC(CCc3ncc(C)[nH]3)=O)C2C)=O)CS(=O)(=O)CC(=O)N1 3040,C(=O)(CCCCC#N)NC1CN(C(CCCC)=O)CC1C 3041,N1(C(CC)C(=O)NC(C)(C)C)CC2COCC2(C(=O)N(c2cnn(C)c2)C)C1 3042,CCC(C)C(=O)C(=O)NOC(CC(C)C)C(N1CCCC(C)C1C)=O 3043,N1(C(C(C(CC)C)N(C(=O)CN2CCCCC2)C)=O)CCN2CC(O)CC2C1 3044,N1(C(c2c(OC(CC)C)cccc2)=O)CC2CN(C(=O)C(C)(C)F)CC2(C)C1 3045,C1(C(N(CC(C)NC(=O)CCc2ccncc2Br)C)=O)OC2CCC1CC2 3046,CC1C(C)C(C)CN1C(=O)C(=O)Nc1ccc(OCC(=O)N(C)C)cc1 3047,CCC(CCC(=O)NCCc1cc(C)n(C)n1)NC(c1cc(Cl)cn1CC)=O 3048,Cc1cc(=NC(=O)C(=O)Nc2ccc(C3OCC3(F)F)cc2)[nH]n1-c1ccccn1 3049,c1(C(=O)NCC(C)N(C(C2CCCC2C(C)C)=O)CC)ncc(C)cn1 3050,CC(C)CC(F)C(=O)NC1CCCN(C(=O)CCN(C)C(=O)OC(C)(C)C)C1 3051,C(CC(C)C)(C(=O)NCC1(N(C)C)CCC1)ONC(COC(CC)CC)=O 3052,c1(CCNC(C)=O)ccc(C(=O)NCC2C(NC(=O)CCCF)C2(C)C)cc1 3053,c1(C(=O)NCCN(C(CCCn2c(C)ncc2)=O)CC(C)O)c[nH]c(=S)cn1 3054,CCCC(C)CC(=O)N(CCCC(=O)NCCOC1CCOC1)C 3055,c1(C(C=CC(=O)N(C2CCC(C)C2)C)=O)ccc(C(F)F)cc1 3056,C(=O)(CC1OCc2ccccc21)N(CCNC(C(=O)NCC)=O)C(C)C 3057,Cc1nnc2n1CCN(C(=O)C(C1CCCN(C(=O)CC#N)C1)C)C2 3058,c1(C(N2C3CCC(CNC(C4C(=C)CC4)=O)(C3)C2)=O)cccc2ccn(C)c12 3059,CC1CN(C(=O)Cc2cc(Cl)ccc2O)CCC1N(C(=O)Cn1ccnn1)C 3060,N1(C(c2cnn(C)c2C)C(=O)NCCCSCC)CC(C)CCCC1C 3061,C1(C(=O)NCC(CC)NC(c2cc(C)on2)=O)(CN2CCCC2)CCCC1 3062,C(C(CC(C)C)C(=O)NC(c1snnc1C)C)NC(c1c(C)noc1)=O 3063,c1(C(N2C3C(N(C(CS(CC)=O)=O)C)CC(C3)C2)=O)cn2cccc(C)c2n1 3064,C12(NC(c3cncc(-n4cnnn4)c3)=O)CC1CN(C(C1CCC13CCC3)=O)C2 3065,N1(C(C2CC(OC)C2)=O)CC2(CNC(=O)COC3CCOC3)CC(F)(C1)C2 3066,CN1C(=O)CC(C(N2CC(C(N)=O)(CNC(=O)CNC=O)C2)=O)C1c1ccnn1C 3067,S(=O)(=O)(c1ccc(C(C)NC(=O)NCC2CCCC23CCC3)cc1)NC 3068,C(=O)(CC(C(F)(F)F)n1cccn1)NCCNC(c1c(Cl)cc(C)s1)=O 3069,N1(C(C=C(COC)C)=O)CCC(N(C(=O)COC2CC2(F)F)CCO)C1 3070,c1(OC)ccccc1C=CC(=O)N(C)CCNC(=O)CC(c1c(C)noc1C)C 3071,C1(NC(C=CCC(C)(C)NC(=O)CC2(O)CCOCC2)=O)CC2(CNC(=O)O2)C1 3072,Cc1cc(CNC(C2(O)CCN(C(C3CCCN(C)C3)=O)C2)=O)cc(O)n1 3073,C1(CNC(C(C=CCCC)O)=O)CN(C(=O)C(C)(C)CF)CCO1 3074,C(C(O)CN=c1[nH]c(C2CCCC2)nc(=N)[nH]1)NC(c1c(S(C)=O)cccc1)=O 3075,C(N=c1[nH]nc(-c2cccnc2)s1)C1CCC(NC(c2cc(C)ncc2)=O)C1 3076,c1(C(=O)NC(C(C(C)C)NC(=O)CC(C)(C)C)C)nc2ccccn2c1F 3077,Cc1nn(CC(=O)NCC2CCC2NC(=O)CC=CC(C)(C)C)c(C)c1C=NO 3078,N1(C(Cn2c(C(=O)OC)cc(C)n2)=O)CCC(F)C(NC(c2sccc2Cl)=O)C1 3079,CC1CCN(C(c2cncnc2)=O)CC1N(C)C(C1CCCCCC1)=O 3080,N1(C(CCCCCOCC)=O)CCC2CCN(C(=O)C(C(C)C)C(C)C)CC12 3081,C(=O)(C(C)(C)CNC(C1C(C)CCN1C(c1cc[nH]c1)=O)=O)NCC 3082,c1(N2C(CO)CN(Cc3ccncc3Br)CC2)ncnc2ccc(F)cc12 3083,c1(C(=O)NCC(CNC(=O)C=CCO)O)cc(Cl)cc2c1CCC2 3084,Cc1cccc(OCC(N2CCC(N(C(=O)CCS(C)=O)CCO)C2)=O)c1C 3085,c1(NC2C(C(N(CC)Cc3cccc(Br)c3)=O)C2)ncnc2[nH]c(C)cc12 3086,C1(CNC(c2cc(O)ncn2)=O)CN(C(C2C(F)(F)C23CC3)=O)CCCO1 3087,CC1CC(C(=O)NC2CC3CCC(C2)N3C(=O)C(F)(F)F)Cc2nn[nH]c21 3088,C(C(CC(C)C)C(=O)NCC1(C)COCCO1)NC(c1cc(C)no1)=O 3089,C1(CC(C)NC(C2C(C)C2C)=O)CCN(C(=O)Cn2ccc(C(F)F)n2)CC1 3090,c1(C(=O)NC2CC(N(C(C=CSC)=O)C)C2)ccc(NC(=O)N(C)C)cc1 3091,N1(C(C2C(CC(C)C)C2)=O)CCCC1CN(C)C(C1(CCC(C)C)CCCC1)=O 3092,C1(C(N2CC(O)(CNC(C3C(C(C)(C)C)C3)=O)C2)=O)CCCC12CCC2 3093,N1(CC(=O)NCCNC(C2C(C)OC(=O)N2)=O)CCC(=O)NC1=O 3094,C1(c2nc(C)[nH]n2)CN(CC(=O)NC2CCC(C(F)(F)F)CC2)CCO1 3095,CC1CC(C)(C(N2CCCC(NC(=O)C(c3ccccn3)O)CC2)=O)CC(C)O1 3096,c1(CNC(N(C2(C#N)CCNC2)Cc2ccc(OC)cc2)=O)c(C)cc(C)cc1C 3097,c1(C(N(C2CCN(C(C3CCCC4CC34)=O)C2)CC)=O)ccc(Cl)c(Cl)c1 3098,c1(OC)nc(C)cnc1C(=O)NCc1cccnc1CNC(=O)CC(C)F 3099,c1(C(=O)NCC(c2c(CC)cccc2)NC(=O)C(C)(C)F)cc(N)c(F)cn1 3100,N1(C(c2cccc(CC)n2)=O)CC(NC(=O)Cc2csc(NC=O)n2)CCC1C 3101,c1(OCC)cccnc1C(=O)NC1CCOCC1NC(=O)CCC1CCCCC1 3102,N1(c2cc(C(C)(C)C)ncn2)CCOCC(NC(c2cscc2Cl)=O)C1 3103,c1(C(=O)NCC2CN(C(c3c(C)n[nH]c3)=O)C2)ccnc2c1ccn2C 3104,C(=O)(C(C(C)CC)N(C)C(c1cscc1Cl)=O)NC(CCC)(C)CC 3105,c12cnc(nc1)NC(C)C1CCN(CC1)C2=O.c1(CC=O)csnc1C.CCO 3106,Cc1ccnc(O)c1C(=O)NCC(C)NC(c1cn(C)c(-c2ccccn2)n1)=O 3107,c1(C(N2CCC(NC(C3CC(C)(O)C3)=O)C2C)=O)ccc(COC(C)C)cc1 3108,C1(CC(N2C(CC(=O)N(C)Cc3ncn(C)n3)CC2)=O)CCCC2CC12 3109,N1(C(c2ccc(CC)s2)=O)CCC2CC2(NC(=O)CCS(N)(=O)=O)CC1 3110,C1(NC(C(C2CCCC2)OC)=O)CCNC1(C)C 3111,c1(N2C(CNC(C3N(C(C)C)CCC3)=O)C(C)CC2)nc(Cl)ncc1C(F)(F)F 3112,N1(C(C(C)(O)C2CCC2)=O)CC2CC(C1)C2NC(c1sc(Cl)cc1Cl)=O 3113,C1(CNC(CCCC)=O)C(C)CCCN1C(c1ccc(CC(C)C)nc1)=O 3114,c1(C(=O)NC2CCCC(CNC(c3cnsc3)=O)C2)ccc2c(c1)CCCS2 3115,N1(C(C=CCN(C)CC)=O)C(C(=O)NCn2cc(CO)nn2)CCC1C1CC1 3116,C1(CC2CCC2)CCC(C)(C)OC1.c12ccccc1-n1cc(nn1)C1CN(C1)C2=O.CO 3117,c1(C(=O)NC23C(CN(C(CCCC(=C)C)=O)C2)C3)ccc2cncn2c1 3118,n1(C2CCC(C#C)CC2)c(-c2ccc(Br)s2)csc1=Nc1cccc(C)c1 3119,C1(NC(Cc2scc(C)c2)=O)CCN(C(=O)Cc2cnn(C)c2C)CCC1CO 3120,N#Cc1cc(C(N2CC(NC(c3cccs3)=O)C(C=C(F)F)C2)=O)cc(F)c1F 3121,C12(CNC(c3c(Cl)ccc(N)c3)=O)CCCCC1CN(C(=O)Cc1ccoc1)C2 3122,CN1CC(NC(C2CN(C(=O)CN3CCNC3=O)CC23CC3)=O)CCC1=O 3123,C1(NC(C(c2ccc(Cl)cc2)C)=O)CN(C(c2cccnc2)=O)CC12CC2 3124,CCC(C)(C)C(C)CC(=O)NCC1CC(NC(c2ncc3[nH]ncc3n2)=O)C1 3125,CCCC(C)C(=O)N1CCCC1Cn1cc(CNC(=O)CSC(F)(F)F)nn1 3126,c1(OCC)cc(Cn2cc(-c3ccccc3C#N)nn2)ccc1Cl 3127,C1(C(N2CCCCC(CNC(C3(CC)CC3)=O)C2)=O)CC2CCC(C1)C2O 3128,c1(C(=O)NC(CC(C)NC(c2cc[nH]c2)=O)C)ccc(-c2cnc[nH]2)cc1 3129,N1(C(C2CC2(F)F)=O)CC2COCC2(C(N2CCCC2c2cc(C3CC3)on2)=O)C1 3130,C1(NC(C(C)C2(O)CCC2)=O)COCCC1C(=O)NOCC1CCOCC1 3131,C1(C(N(CC(CCC)O)C)=O)CC(OC)CN1C(=O)CC1CC2(CCC2)C1 3132,C1(NC(C2C(=C)C2C(=O)OC)=O)CCCN(C(=O)C(C)(C)C(F)F)CC1 3133,C1(C(=O)NC2(C)CC(=C)C2)CCN(C(C2CCCCCN2C)=O)C(C)(C)C1 3134,C(=O)(C(=O)CC(C)CC)NCCCC(N1CCCC(CC=CC)C1)=O 3135,C(=O)(C(C)CC(C)CC(C)C)NCC1(F)CC(NC(c2nnn(CC)c2C)=O)C1 3136,c1(C(N2CC3C(CNC(CN4CC(CC)C4)=O)(C3)C2)=O)ccc2c(c1)nnn2C 3137,C1(C(N2CCC(CNC(C3(C(=O)NC)CC3)=O)C2)=O)CCCC(CNC(C)=O)C1 3138,C12CN(C(C3CC3c3ccccc3)=O)CC1C2=O.c1(CCN)ccccc1.C(C(C)C)S 3139,C1(C(N2CC(C)C2C(=O)NCCc2cn(C)nn2)=O)CC12CCCCC2 3140,N1(C(C2CC23CCOC3)=O)CCC(OC)CC1.c12nnc(o1)SC1CN(C1)C2=O.CC 3141,Cc1ncc(NC(=O)C(CC2CC2)NC(=O)C(C2(O)CCCC2)F)c(C)c1C 3142,c1(C(=O)NC2CCN(C(C3(N(C)C)CCC3)=O)CC2)ccc(S(C)(=O)=O)cc1N 3143,c1(CC)cc(C(=O)NC(C)C(C)NC(=O)C(C)n2ccnc2)ccc1O 3144,C(=O)(C(F)C(C)CNC(C1CCS(=O)CC1)=O)NCc1c(OC)nn(C)c1 3145,C12(C(=O)NCc3cnc(C)o3)CC1CN(C(C1CCO1)=O)C2 3146,c1(C(=O)OC)cn(C)nc1C(=O)NC(C)CNC(=O)Cc1cnns1 3147,Cc1nc2cc(NC(C3C(O)CCN3C(C3CCCC(C)C3)=O)=O)cnc2[nH]1 3148,C(CNC(=O)C(F)(F)C(F)F)(CC(F)(F)F)NC(C(C)Cc1cnc[nH]1)=O 3149,C1(NCc2cc(C(=O)OC)c(C)cc2)CCN2CCCC2C1 3150,N1(C(=O)OC(C)(C)C)CCc2ccccc2C1CC(=O)OCC(F)F 3151,C1(C(=O)NC(C(N2CC(C)=C(C)C2)=O)CCN(C)C)CC2(CC(=O)C2)C1 3152,C1(CNC(Cc2scc(C)c2)=O)CCCN(C(c2cccc(OC(F)F)c2)=O)C1 3153,C1(c2nc(CCCCCC)nn2C(C)C(C)(C)C)CCn2c(C)cnc2C1 3154,C(=O)(CCCCCc1cn(Cc2ccoc2C(=O)O)nn1)Nc1cc(C)nn1C 3155,Cc1ccc(C(=O)NCC2CCN2C(=O)Cn2c(C)c(C)sc2=O)cc1[N+](=O)[O-] 3156,N1(C(CN(C)C2CC2)=O)CC(NC(C2C=CC=CC=C2)=O)C(c2cnn(C)c2)C1 3157,C1(C#N)(NC(C(C)C)=O)CCN(C(=O)CN2C(=O)CSC2=S)C1 3158,CCCC(C(=O)N1CC(C)(NC(c2nccn3ccnc23)=O)C1)C(C)C 3159,CC1(NC(c2cnc(Br)s2)=O)CCN(C(C2(O)CCC2)=O)C1 3160,CC(C)(C#N)CCCC(=O)NC1CCCC(NC(C2CC23CCSCC3)=O)C1 3161,c1(CC)cc(C(N2CC(F)CC2CN(C(=O)C2=CCCS2)C)=O)sc1C 3162,c1(OC)ccc(Br)cc1CNC(c1ccnn1C(C)(C)C)c1nnnn1C(C)C 3163,c1(C(=O)OC(C)(C)C)ccccc1NS(C)(=O)=O 3164,C1(CC(=O)NCC2CCN2C(=O)C=C2CCCCC2)CC2(CCC2)C1 3165,c1(OC)cc(NC(=O)C(C(C)OC)NC(=O)C=CC2CCCN2C)cc(O)c1 3166,c1(C(N2CCCCC2c2n[nH]c(C(C)C)n2)C(=O)NCC(C)C)nc(Br)nn1C 3167,C1(CCC)CN(C(=O)Cn2nc(C)nc2C)CCN1C(=O)C1=C(Cl)CCC1 3168,N1(C(C2N(C(C3CC3c3ccc(Br)cc3)=O)CCC2)=O)CCN2CC(O)CC2C1 3169,C1(NC(C2CN(CC(C)C)C2)=O)CCC(CNC(=O)C=Cc2ncc[nH]2)C1 3170,C(=O)(C(C)(C)C(C)C)N(C)CC1CCN(C(CCOCCCOC)=O)C1 3171,C1(NC(CC(C)N(C)C)=O)CC(C(=O)NCC2=CCCC2)C1(C)C 3172,c1(OC)ccc(Br)c(CCN(CCO)C(=O)NCc2cnc(C3CC3)o2)c1 3173,C(=O)(C1=NN(C)C(=O)CC1)Nc1ccc(-c2c(F)ccc(-c3ccc(OC)s3)c2)s1 3174,C(=O)(CCCCCF)NCCN(CCOC)C(C1CC1C1CCCC1)=O 3175,CCCC(C)(O)CC(=O)NC1(C)CCCCC1C(N1CC=CC1CF)=O 3176,CC(CNC(c1cscc1Cl)=O)C(F)C(=O)NC1(CO)CC1 3177,N1(C(c2cnc(OC)s2)=O)CC2(CCC2NC(=O)C(O)Cc2cn(C)cn2)C1 3178,CCC(CC)(CCNC(C1CC1(Cl)Cl)=O)NC(=O)C(N)=O 3179,c1(OC)ccc2ncc(C(N3CCC(NC(=O)CNC=O)C3(C)C)=O)n2n1 3180,C1(CNC(C)=O)CCCN1C(=O)CCOC1CN(C(=O)CC(C)F)C1 3181,N1(C(C(C)OC)=O)CCN(C(=O)C(C)CSC)C(C2CC2)C1 3182,N1(C(C(C)OC2CCCC2)=O)CC(C(=O)NC(C2CCCOC2)(C)C)C(F)(F)C1 3183,N1(C(c2c(OC)cc(C)s2)=O)CCC2(CCCC2NC(c2cncc(N)c2)=O)C1 3184,C1(C(C)NC(c2c(C(C)C)c[nH]n2)=O)CN(C(=O)CCCC2CC2)CCO1 3185,C1(C(=O)NC(C(C)C)CNC(=O)CC2CSC2)CCn2cncc2C1 3186,N1(C(C2CCCN(CC(C)C)C2)=O)CCCN(C(c2ncccn2)=O)C(CO)C1 3187,CC(C)C(O)C(F)(F)C(=O)NCCc1ocnc1CNC(C1Cc2nncn2C1)=O 3188,c1(CC)ncc(NC(=O)C(Cc2cn[nH]c2)NC(=O)Cn2ccc(C)n2)cn1 3189,c1(-c2c(C(=O)O)cc(Cl)cn2)cccc2c1NCC2 3190,c1(CC)ncsc1C(=O)NCC1(CNC(=O)CC2CCCC2C)CC1 3191,Cc1cccc2[nH]cc(C(N3CCC=C(CNC(C4COC(C)C4)=O)C3)=O)c12 3192,c1(-n2ccc(C)n2)cccc(C(N2CC(NC(C3CC4(CC4)C3)=O)C(C)C2)=O)c1 3193,C(c1cn(C)nn1)=CC(=O)N(CC)CC1CCCN1C(c1cc(C(F)F)[nH]n1)=O 3194,C(=O)(N=S(C)(=O)c1cccc2cccnc12)c1c(N(CCN(C)C)C)nccc1 3195,C1(CCOC)CN(C(C2CCCCC2O)=O)CCN1C(=O)Cn1cc(C)cn1 3196,N1(C(C2C3CCCC(=O)C32)=O)CC2CCCN(C(C34CC(F)(C3)C4)=O)C2C1 3197,c1(NC(COc2cn(C)nc2)=O)ccc(NC(C2(C)CC2C(F)(F)F)=O)cc1 3198,c1(C(N2C(C(C)(C)NC(c3cncnc3)=O)CCC2)=O)nccc2ccncc12 3199,N1(C(C(CC)N2CCCC2=O)=O)CCCC(CNC(C2(OC)CC2)=O)CC1 3200,Cc1cc(C(N2CC(O)CC2C(N2CCC(C)(O)CC2)=O)=O)cc(Br)c1 3201,N1(C(C(c2ccc(Cl)cc2)=O)=O)CCN(C(c2nocc2Br)=O)CC1CF 3202,C1(C)(CNC(CN2C(C)CC2)=O)CCN(C(=O)C(C(C)(C)C)c2cc[nH]n2)CC1 3203,C#Cc1cncc(C(=O)NC(CN(C)C(C2CCS(=O)(=O)N2)=O)CC)c1 3204,n1(CC)nncc1C(=O)NCC1CC(NC(=O)C(F)(F)c2ncccn2)C1 3205,c1(CN2CC3C(C(N4CCCC(C(C)(C)O)C4)=O)C3C2)ccnc(F)c1Cl 3206,c1(NC2C(C)C2)cc(S(=O)(=O)NCc2ccc(F)cc2)ccc1C#N 3207,C1(C(N(CC(C)(C)O)CCC)=O)CSCN1C(c1cc(OCC)no1)=O 3208,CCC(CCC(=O)NC1CCN(CC2CC2)C1)NC(c1ccnnc1C)=O 3209,c1(C(=O)NC2CC(NC(Cn3ncn(C)c3=O)=O)C2)ccc2ncc(=O)[nH]c2c1 3210,c1(OC)cccc2c1CC(C(=O)N(C)CCN(C)C(C1CC(C#N)C1)=O)CO2 3211,C1(C(=O)NC(C)C(C)(C)NC(=O)C=C(C2CC2)C2CC2)CC2CCC(C1)S2 3212,N1(C(C=Cc2cc(OC)ns2)=O)CC2CCC(C1)N(C(=O)CSCCN(C)C)C2 3213,CCCCCCCCC(=O)N(CC(C)N(C(=O)CC(C)(C)C1CC1)C)C 3214,C(=O)(C(C)(C)C(=O)OC)NC.N1(CCCC)CCN(C(=O)COCCNC(C)=O)CC1 3215,N1(C(c2cscn2)=O)CCC2(CCCCN(C(C34CC(C3)C4)=O)C2)C1 3216,N1(C(C(C=C)(F)F)=O)CCCC(CCNC(C2CC3(CSC3)C2)=O)CC1 3217,C1(OC)CN(C(=O)C=C(C)Cl)C(C)(CNC(c2ccc(C(F)F)nc2)=O)C1 3218,Cc1cc(C(=O)NC(C)CC2CN(C(=O)C(C)OCC(C)C)C2)c(C)s1 3219,Cc1nc2ccc(C(N3CC(N(C)C(C4(C)CC4)=O)C3)=O)cc2s1 3220,C1(C(=O)NCCCCCN(C(COCC(C)C)=O)C)CC(S(C)(=O)=O)C1 3221,c1(C(=O)NC(C2CCCN2C(C2CCC2C(F)F)=O)C)cncc(F)c1 3222,C1(C(C)C)(NC(CC(C)NC(C(C2CC2)SC)=O)=O)CCOCC1 3223,Cc1cc(C(=O)NCC2CCN(C(c3ncc(Cl)cc3Cl)=O)CC2)ccc1F 3224,c1(C(=O)NCC2CC(F)(F)CN2C(C2CC23CC(O)C3)=O)cn2cnnc2cn1 3225,C(=O)(C(C)CN(C)C)NCC1(CNC(CNC(C(C)NC(C)=O)=O)=O)CC1 3226,C1(C)(C(=O)NC(C#C)CC)CCN(C(c2cccc(CNC)n2)=O)C1 3227,C1(NC(CN2CC(C)C2)=O)CCC2CN(C(c3ccc(N)c(N)c3)=O)CC2C1 3228,C1(C(=O)NCC2(C3(O)CN(C(C4CC(=C)C4)=O)C3)CC2)CC2(C1)CC1(CCC1)C2 3229,c1(OC)c(C)ccc(C(=O)NC(C)CCCNC(=O)CCn2cc(C)cn2)c1F 3230,c1(OC)ncc(C=CC(N2CCC(NC(=O)C#CC3CC3)C(CO)C2)=O)cn1 3231,C(=O)(NNC(=O)CCc1cccc(Cl)c1)c1ccc(C)cc1 3232,c1(CC)cc(C(N2CCC(c3cn(CCOC)nn3)C2)=O)nn1-c1ccccc1 3233,C1(CNC(Cc2c(CC)n[nH]c2CC)=O)C2CCC(C2)N1C(=O)Cn1ncnn1 3234,c1(NCC(=O)Nc2ccc(-c3cccc(C)c3)cc2)c(Cl)ccc(O)c1Cl 3235,CCCCCCN(C(=O)CC1CCCO1)CCN(C(=O)CCN1CCC1)CC 3236,N1(C(CC=C)=O)CCCC(C)(CNC(=O)CN(C)CCC)C1 3237,N1(C(CSCCC)=O)CCOC2CCN(C(=O)C(C)n3ccnc3)CC12 3238,N#Cc1ccc(CN(C(N2CCOCC2)=O)Cc2ccc(-c3nn[nH]n3)cc2)s1 3239,c1(C(N(CC(CNC(CCC(=C)Br)=O)O)C)=O)c(C)cccc1Cl 3240,N1(C(c2ccc(Br)cc2Br)=O)CC2CCN(C(c3cccc(F)c3O)=O)C2C1 3241,C=CCC(C)C(=O)NC1CN(C(c2cn(-c3cccc(CO)c3)nn2)=O)C1 3242,Cc1oc(S(N)(=O)=O)cc1C(=O)NC(C1CCCN(C(C2(C)CSC2)=O)C1)C 3243,CCC(C(=O)NC1CN(C(=O)CCC(=O)c2ccc(C)s2)CC1C)C(C)(F)F 3244,CCCC(C(=O)NCCN(C(c1ccc(=O)n(C2CC2)c1)=O)C(C)C)C(C)C 3245,C(C)(CCCNC(=O)C(N1CCC(C)C1)=O)NC(CCN(C)CC)=O 3246,c1(C(N2CCC(C)(C(N)=O)C2)C(=O)NCCC2(C)CC2)ccc(F)c(Cl)c1Cl 3247,c1(C(=O)NC(C(C)NC(C(C)OC)=O)C)ccccc1Oc1ccncc1 3248,C1(CNC(Cc2n(C)cnc2)=O)CCCN(C(=O)CCNC(C2CCC2)=O)CC1 3249,CCCCCC(F)C(=O)NCC1CC1NC(c1onc2c1CCCC2)=O 3250,C1(CNC(C(C)=C2CCCC2)=O)CN(C)CCN1C(=O)CNC(=O)C(F)(F)F 3251,C1(CC)(NC(=O)CN2CC(C)(C)C2)CCCN(C(=O)C(C)OCC2CC2)C1 3252,C1(C(N(CC(C)O)CC)=O)CCCN1C(=O)C(n1ccc(C)n1)C 3253,CCC(C)(C)C(=O)C(=O)N1CCOCC(CNC(=O)CCc2ccc(F)cc2)C1 3254,N1(C(C(C(=O)OCC)F)=O)CCC(CCNC(=O)Cc2nonc2C)C(F)(F)C1 3255,C1(C(=O)NC(C)CNC(c2csc(C(C)OC)n2)=O)(COC)CCCC1 3256,N1(C(CCCC#C)=O)CCC2CCN(C(c3cn(C)c(C)n3)=O)CC12 3257,N1(C(C2C(C(C)C)C2)=O)CCC(C2CCN(C(c3cc4sccc4[nH]3)=O)C2)CC1 3258,c12cc(OC)cc(c1)NC(=O)Nc1ccc-2cn1.c1(OC)ncccc1OC 3259,c1(C2C(C(N3CC(OCCNC(c4cncn4C4CC4)=O)C3)=O)C2)cccnc1 3260,N1(C(C(C)COCCc2ccccc2)=O)CC2CN(C(=O)CSC3CC3)CC2C1 3261,c1(SC(C)C(=O)N(C2CN(C(=O)CC3CCC34CCC4)C2)C)ccccc1Cl 3262,CC(C(C)C(=O)NC1(C(C)(F)F)CCC1)NC(=O)CSC(F)(F)F 3263,N1(C(C2(C(C)C)CCC2)=O)CC2CCN(S(=O)(=O)c3ccccn3)C2C1 3264,CN1C(=O)CCCC1C(N1CC2(CO)CC1(C(=O)NCc1nnnn1C)C2)=O 3265,CC(C)(C)C(O)CC(=O)N1CCCC(O)(CNC(c2cc(F)cnc2O)=O)C1 3266,c1(C(N2CCN(C(C3CCCN(C)C3)=O)CC2CC#N)=O)ccc(C#N)c(Cl)c1 3267,O=C(CC1CC(=O)c2ccccc21)Nc1ccc(Cl)c(S(=O)(=O)N2CCCC2)c1 3268,C(CO)(CCCCNC(c1ncccc1C)=O)NC(C(CC)CC1CCCC1)=O 3269,c1(C(N2CCC(CN(C)C(C3CCCC(=O)N3)=O)C2)=O)cccc(C(C)(F)F)n1 3270,N1(C(C(C)OCCC(C)C)=O)CC2CCC(C1)N2C(=O)CC(F)(F)F 3271,c1(CNC(=O)NCc2c(CC(N)=O)cccc2)ccc(Cl)cc1[N+](=O)[O-] 3272,C1(C2CN(C(=O)CSc3ccccc3Cl)C2)(CNC(C(C)CN(C)C)=O)CC1 3273,C=C=CCCC(=O)N(CC)CC1CCCCN1C(=O)CC1(OCC)CCC1 3274,N#CC1(CC(N2CC3CC2CN3C(=O)C=CBr)=O)CCOCC1 3275,c1(OC(=O)C(F)(F)F)cc(NCc2cnn(-c3cccc(F)n3)c2)ncn1 3276,C(=O)(C(CCOC)NC(C1(C)CC(C#N)C1)=O)NCCCOCCOC 3277,C(=O)(C(CCCC)NC(C1CC(C)CCO1)=O)N1CCC(O)(CC=C)C1 3278,c12ncc(cn1)CCO2.C1(OC(C)(C)C)CC(NCCNC(C#N)C2CC2)C1 3279,N1(C(C2(CCC=C)CC2)=O)CCN(C(=O)CCn2nc(C)cc2C)CC(C)C1 3280,C1(C)(C(=O)NCC2(NC(C(N3CCC(O)CC3)C)=O)CCCC2)COCCO1 3281,c1(C(N(c2ncnc(OC)c2C)C2CNCC2F)=O)cc(Cl)c(Br)cc1Cl 3282,CC1(C)CCc2cc(C(N3CCN(C(c4cnsc4)=O)CC(O)C3)=O)ccc2O1 3283,c1(OC)ccc(CN2CCCCC2C(=O)NC2CC(CO)C(O)C2O)cc1O 3284,c1(CCC(N2CCN(CCNC(C3(C)CC3)=O)CC2)=O)c(F)cccc1Cl 3285,C1(C(N(CCC(=O)NC2C=CCCC2)CC#C)=O)CCCC(=O)CC1 3286,C(=O)(C1=NOC2(CCN(Cc3csc4c3CCCC4)C2)C1)NC(C(C)C)CO 3287,c1(C(N2CCC(CC(=O)NC(CC3CC3)C3CC3)CC2)=O)cn2c(n1)CCC2 3288,CC1Cc2cc(C(N3CCN(C(=O)CC(C)(C)C(F)(F)F)C(C)C3)=O)ccc2O1 3289,N1(C(C(CC)C(F)(F)F)=O)CCC2CN(C(c3cnc4[nH]ccnc3-4)=O)C(C)C12 3290,CC1COC(NC(=O)NC(c2cccc(-c3nn[nH]n3)c2)C(C)(C)C)CO1 3291,c1(C(N)=O)c[nH]c(C(=O)NCCOCCNC(c2nncs2)=O)c1 3292,C1(OC)COCCC1CC(=O)NCCCN(CCO)C(c1ccc(C(C)=O)o1)=O 3293,c1(N(CCNC(CCCOCC)=O)CC)c(C#N)cnc2c(Cl)cccc12 3294,C1(NC(C2(C)CCCNS2(=O)=O)=O)Cc2ccccc2C1NC(=O)C=CBr 3295,Cc1[nH]c2ccc(C(=O)NCC(C(C)C)NC(=O)C(=O)C3CCCC3)cc2c1C 3296,N1(C(C2=CC(C)(C)C2)=O)CCC2CN(C(c3ccc4c(c3)CCOC4)=O)CC2C1 3297,C1(NC(c2c(C)cccc2C)=O)CC2CCC1C(NC(C1CC1(F)F)=O)C2 3298,N1(C(C2(C)CCCCCC2)=O)CC2(CC(NC(C3CCCS(=O)(=O)N3)=O)CO2)C1 3299,C1(C(=O)NCC[Si](C)(C)C)(CC)CN(C(=O)C(C)c2cccs2)C1 3300,Cc1cc(C(=O)NC(c2nccs2)C)c(C)n1N 3301,C1(CC(=O)NCC2C(C(=O)NCCc3onc(C)n3)C2)C(C)(C)C1(C)C 3302,c1(C(=O)NCC2CC(NC(C(c3n(C)ncc3)O)=O)C2)cc2cc(F)ccc2o1 3303,CN=c1[nH]cc(C(N2CCCC2C2(O)CN(C(c3cscc3C)=O)C2)=O)o1 3304,c1(OC(C)C)ccc(Cn2nc(-c3ccsc3)nc2CN2CCOCC2=O)cc1 3305,c1(C(=O)NC(c2cnn(C)c2)C(=O)NC(CC)CC)cn(C)cn1 3306,C(=O)(N=S(C)(=O)c1cccc(F)c1)c1cn(C)nc1C1CC2CCC1C2 3307,Cc1cncc(CC(=O)NCC(C)(C)CN(C)C(C2NC(=O)OC2C)=O)c1 3308,C=CC(C)(CC)C(=O)NCC(C(C)C)NC(c1cncc(-c2ccccc2)c1)=O 3309,C(=O)(CC(C)CCC=C(C)C)NC1(COC)CN(C(C2CCCC(C)O2)=O)C1 3310,CN1CCOCC(NC(C2(NC(=O)C(O)CC(N)=O)CSC2)=O)C1 3311,c1(C(=O)NCC)nc(N(C(C)CNC(c2cc(Cl)on2)=O)OCC)cc(Cl)n1 3312,CC#CCC(C(=O)N1CCC(C(C)C#N)CC1)NC(=O)C(n1cc(C)cn1)C 3313,N1(C(C2(SCC)CC2)=O)CCC(C)(CNC(=O)COc2ccsn2)CC1 3314,N1(C(C2CCC(C#C)CC2)=O)CCCN(C(c2cncc3sccc23)=O)C(C)C1 3315,c1(C(N(CC(CC)NC(=O)C(c2cccc(C)c2)C)C)=O)cncc(F)c1C 3316,C(=O)(CCCC(F)(F)F)NC1CC(C)(C)N(C(=O)CN2CCOCC2)C1 3317,C12(NC(CNC(=O)C=C(Cl)Cl)=O)CCCC1N(c1ncc3ncnc-3[nH]1)CCC2 3318,C#Cc1ccnc(C(=O)NCC(C2CC2)NC(=O)C(N2CCNC2=O)C)c1 3319,c1(CC)cc(C(=O)NC2CCC(N(C)C(c3ccnnc3)=O)C2)cc(F)c1 3320,C1(CC)CC(CC(=O)N(CC(O)CNC(=O)CC(C)c2cnn(C)c2)C)CCO1 3321,c1(SC)cccc(CC(=O)NCCOC2CN(C(=O)CC(C)C3CC3)C2)c1 3322,c1(NCC(CCCC)NC(C2(CO)CCCO2)=O)cc(=O)n2cc(Cl)ccc2n1 3323,C1(c2nnnn2C)(CNCCC(C(F)(F)F)OCC)CC2CCC1CC2 3324,Cc1ccc(NC(=O)C(c2ccoc2)NC(=O)Cn2ccnn2)cc1CO 3325,N1(C(CCC#C)=O)CC(NC(c2cccc(NC(=O)NC)c2)=O)CC12CCOC2 3326,c1(OC)csc(C(=O)NCCN(C(=O)C(n2ccnc2C)C)CC2CC2)c1 3327,n1(C(CC)C)ncc(C(=O)NC2(CCCl)CC2)c1C 3328,N1(C(c2c(OC)c(Cl)ccc2)=O)CCC2(CCN(C(=O)CN(S(C)(=O)=O)C)C2)C1 3329,C(=O)(C(C)P(C)(C)=O)NCc1c(CNC(CCNC(CC(C)C)=O)=O)ocn1 3330,N1(C(c2c(C)nsc2)=O)CC(NC(=O)CC2CC23CC3)C(c2cncn2C)C1 3331,N1(C(CCCNC(c2ccsc2)=O)=O)CC2CC1CN2C(C1(O)CCC1)=O 3332,N1(C(COCCCC)C)CCC2(CC1)CC(C(=O)OC)C2 3333,C1(C(=O)OC)C(C(N2CCC(NC(=O)Cc3cscn3)C2)=O)C1(F)F 3334,C(CCN=C(NCC1CN2CCN1CC2)NC(c1ccc(F)cc1F)C)OC 3335,C12(C(=O)NC(C)C(C)n3cccn3)CC1CN(C(=O)C(C)(C)C1CCOC1)C2 3336,c1(-c2n(C(C=C)C)nc(C(C)O)n2)cnc2cc[nH]c2c1 3337,C(=O)(C(C)(C)C(C)(C)C)N1CC(NC(c2c(C(C)C)con2)=O)C(F)C1 3338,C(=O)(C(C)S(=O)Cc1cccs1)OC(c1ccccc1)Cc1ccc(OC)cc1 3339,C12(C(=O)NC3C(C)CN(C(c4coc(Br)n4)=O)C3)CC(C)(C1)OC21CCC1 3340,c1(OCC(N2CC(C(C)(C)NC(CC=C)=O)C(C)C2)=O)cccc(C)c1F 3341,c1(C(=O)NCC2C=CC(NC(=O)C=C3CCCC3)C2)cc(F)c(F)cc1Cl 3342,CC1CCN(C(=O)CCc2ccccn2)C1C(=O)N(C)Cc1nc(=O)o[nH]1 3343,C1(O)(C(C)NC(=O)CCC2CCC(O)CC2)CCN(C(c2ccon2)=O)CC1 3344,C1(C)(NC(C(CC)N(C)C)=O)CCN(C(c2cnc(O)cc2OC)=O)CC1 3345,n1(CCC)ccc(C(N2CC(n3cc(CNC(c4n[nH]cc4C)=O)nn3)C2)=O)n1 3346,c1(C(=O)NC(c2nc(COC)sc2)=O)c(-c2ccccc2)noc1C(C)C 3347,c1(-c2cccc(CNC(c3cnccc3Cl)=O)c2)cc(F)c(C(F)(F)F)cc1F 3348,N1(C(C2CCN(C)C2=O)=O)CCC2(CC1)CC2NC(C1(O)CC(C)(C)C1)=O 3349,C1(N(C(=O)COCCOCCO)CCO)CCCN(C(=O)CC2(O)CCCC2)C1 3350,c1(C(C(=O)N(C)CCF)NC(CC(=O)OC)=O)c(C)cccc1Br 3351,N#Cc1cc(Cl)c(Cl)cc1NC(C1CCCC12CCN(C(C1CC13CC3)=O)C2)=O 3352,C1(c2ccccc2)(CNC(C23CCC2C3)=O)CCCO1.C12(O)CN(C1)OC(=O)C2 3353,N1(C(C2(CC(C)C)CCC2)=O)CCC2C(C1)CN2C(=O)C=C1CCN(C)C1 3354,Cc1cccc(C(N2CCC(C)C2CNC(c2cc(=O)cc[nH]2)=O)=O)c1 3355,C1(NC(c2c(C)cns2)=O)CN(C(C2CC2c2cncn2C)=O)C2(CCC2)C1 3356,C1(NCc2nnn(C)n2)CCN(C(c2cccc(Cl)c2)=O)CC1(C)C 3357,C1(CC)CCC(NC(=O)CCCn2cncn2)CC1 3358,c1(C(N2CCN(C(C=C(C)C)=O)CC2c2ccncc2)=O)ccc2c(c1)CCC2 3359,c1(C(=O)NCC2(F)CCC(NC(C3(C(F)F)CC(=C)C3)=O)C2)ccc(N)c(Cl)n1 3360,C1(CCCC)CN(C(C2(Br)CC2)=O)CCN1C(c1ccsc1SC)=O 3361,c1(C(N2C(C(C)O)CC2)=O)cc(CCNC(=O)C=CC(F)F)on1 3362,Cc1oc2ccccc2c1C(=O)NCC1CCCC1NC(c1cc(O)nn1C)=O 3363,N1(C(c2c(N)ccc(C(=O)OC)c2)=O)C2CCC1CN(C(=O)CN1CCC1C)C2 3364,c1(C(N2CCC(C)(CNC(C3C(C)C3(F)F)=O)C2)=O)n[nH]c2cccnc12 3365,N1(C(C2(CC)COC2)=O)CCC(NC(=O)CCOc2cccc(C)c2C)C(O)C1 3366,C(=O)(C(CNC(=O)Cc1nccn1C)C(C)(C)C)N(C)Cc1ccccn1 3367,CC(N=c1[nH]c(N(C)Cc2ccn(C3CC3)n2)nc2c1CCC2)c1csc(Br)c1 3368,c1(C(N(CCCCNC(=O)CN2CC3CC3C2)C)=O)ccc(F)c(N)c1 3369,c1(OC)cc(O)ncc1C(=O)NCCC1(O)CN(C(c2ccc(N)c(N)n2)=O)C1 3370,c1(NC(c2oc(CC)c(C)c2)=O)cc(CN(C)C)cc(F)c1 3371,N1(C(C(C)SC(C)C)=O)CC2(NC(C3CCCC3)=O)CC1C2 3372,c1(C(=O)NCC(=O)NCC(=O)NC(C2(C)CC2)CO)ccccn1 3373,C1(C(=O)NCC(CNC(C2C(C(=O)OC)CCO2)=O)CO)CCC(F)(F)CC1 3374,c1(C(=O)NCC23C(CN(C(c4ncnc(C)c4C)=O)C2)C3)cc2scc(C)c2[nH]1 3375,N1(C(c2c(C)coc2)=O)CCCC(C)(C)C1C(N1CCOCC1CO)=O 3376,c1(C(=O)NC2(CNC(C3C(C(N)=O)COC3)=O)CC2)ccnc(N2CCCC2)c1 3377,C=C1CC2(C1)CC(C(=O)NCC1CCCCN(C(C3(COC)CCC3)=O)C1)C2 3378,C1(CNC(c2cc(C)c(C)nc2)=O)CC2COCC2N1c1ncc(F)cn1 3379,CC1CCCc2ncc(C(=O)NCCOCCNC(C3CC34CCSCC4)=O)n21 3380,C1(O)(CNC(C2CC23CC3)=O)CC2CCC(C1)N2C(c1cccc2cnsc12)=O 3381,CC1CC(CCNC(c2csc(CO)n2)=O)CCN1C(=O)Cc1cncs1 3382,N1(C(C(C)CN2CCCC2)=O)CCC(C)(C)C(C(=O)NCC2CCC3(CC3)C2)C1 3383,C1(C(=O)NCCC2CC(NC(c3noc(CC)c3C)=O)C2)CCc2n[nH]cc2C1 3384,N#Cc1c[nH]c(C(N2CC3CC3(NC(c3cc(-c4ccccc4)cs3)=O)C2)=O)c1 3385,CC(C(=O)NC1(CC(=O)NCCc2ncon2)CC1)C1CCCO1 3386,C12(CNC(CCc3ccc(OC)nc3)=O)CCC(NC(=O)C(C)SC)(CO1)C2 3387,c1(C(N2CCC(N(C(=O)C(CCSC)OC)CC)C2)=O)cccc(C#N)n1 3388,N1(C(C(CC(C)C)=O)=O)CC2C=CC1C(C(=O)N(C1(C)CC1)C)C2 3389,C=CC(C)(CCOC)C(=O)N(C1CCCC1)CCNC(=O)CC(F)(F)C(F)F 3390,C12(CNC(c3ncn(C(C)C)n3)=O)CCC(CC1)N2C(C1(Br)CC1(F)F)=O 3391,N1(C(c2nc(C)[nH]n2)=O)CC(NC(c2ccc(C(C)(C)C)nc2)=O)C(C)(C)C1 3392,N1(C(CCNS(C)(=O)=O)=O)CCC(Cn2cc(CON3CCCC3CO)nn2)CC1 3393,CN1CC=C(C(=O)NC2COCCN(C(=O)Cc3ccoc3)C2)C1 3394,c1(CN2CC(C(CF)(F)F)(C(=O)O)C2)cnn2c1OCC2 3395,C(CCC)(C(=O)NCC1CC(NC(=O)C(F)=CC2CC2)CCO1)=CCC 3396,CCCCC(CC)(c1nnnn1CCSC)NCCS(=O)CCSC 3397,C1(NC(c2ncccc2Br)=O)CCN(C(c2cnsc2)=O)CC1CO 3398,N1(C(C(N2CCNC2=O)C)=O)CCC(C(=O)NCCCn2cnnc2)CC1 3399,N1(C(CCc2ccnc(C)n2)=O)CCN(C)C(CNC(c2csnn2)=O)C1 3400,c1(N2CC(C)C(NC(=O)Cc3ccc4c(c3)CC4)CC2)ccc([N+](=O)[O-])cn1 3401,c1(C(N2C(CNCc3c(C)n[nH]c3)CCCC2)=O)cnc2c(c1)CCCC2 3402,CC1CC2(C(N3CC(F)(CNC(C4(Nc5ccccc5)CC4)=O)C3)=O)CC12 3403,CC1CCCN(C(C2CCS(=O)CC2)=O)C1CNC(=O)C=Cc1cncn1C 3404,c1(C(=O)NCC2(C)C(C)CN(C(C(CCSC)O)=O)C2)cc(Cl)c(Cl)cc1N 3405,C1(CNC(CCSCCC)=O)C(C)CCCN1C(c1cc(C2(C)CC2)on1)=O 3406,C(=O)(C1=CC2CCCCCCC12)NC(C(C)C)(C)CNc1cncc(C#N)n1 3407,c1(C(N2CC(OCC)(CNC(=O)CCc3cc(C)no3)C2)=O)cn(C)nc1CC 3408,N1(C(C2(C)CC(=C)C2)=O)CCC(c2cn(-c3ccsc3NC(C)=O)nn2)C(O)C1 3409,C=CCCC(C)(C)C(=O)NC1CCCC(C(=O)NCCC(C)(C)N(C)C)C1 3410,N1(C(C(C)N(C(=O)CCN2CCCCC2)CC)=O)CCc2ccncc2C1 3411,CC1CCCc2ccc(NC(=O)NCC3CC4CCC3O4)nc21 3412,C=C(C)C(CC(=O)N1CCCC1CN(C(=O)C=Cc1ccccn1)CC)OCC 3413,C1(NC(C2(CC=C)CC=CC2)=O)COCCC1NC(=O)CCN1CCOCC1 3414,c1(NC(C(c2ncc(C)o2)N(C)Cc2ccccc2F)=O)c(C)cc(C)cc1C 3415,c1(N(C)C(C2CCC(Cc3ccccc3)O2)=O)cc(Cl)ccn1 3416,C(=O)(C1=CC2CCCC12)N(C1CCN(C(c2ccc3nncn3c2)=O)C1)CC 3417,C(=O)(CCCCC(=O)OC)N1CCN(C(COCCC=C)=O)CC1C(C)(C)C 3418,CCC(F)(F)C(=O)NCC1CCCC1NC(=O)Cc1cn(C2CC2)cn1 3419,CC1(CCC(=O)Nc2cnsc2)CCCN1C(=O)Cc1ccc(Cl)s1 3420,C1(N(C(=O)Cc2csc(Cl)n2)C)CN(C(=O)C#CC2CC2)CC12CC2 3421,C1(CNC(c2n(C=C)nnc2)=O)CN(C(=O)C(C2CC2)N(C)C)CC12CC2 3422,c1(C(=O)NC2C(NC(CCCC=C)=O)C2)cc(F)cc(C=C)c1 3423,N1(C(C(C)C(F)F)=O)CC(CC(=O)NC2CCN(C(N)=O)CC2)C2(CC2)C1 3424,N1(CC(=O)NC2C3CN(C(c4n(C)ncc4Cl)=O)CC2C3)C(=O)NC(C)(C)C1=O 3425,C1(C(N2C(C(=O)NC3(CCC)CC3)CCCC2)=O)C2CCCC(=O)C12 3426,Cc1ncc(C(=O)NC2CCC(NC(C3CCN(C)C3C)=O)CC2)n1C 3427,CCCC(CNC(c1cccn1C)=O)C(=O)N(CC)CC1CCCO1 3428,c1(C(C)Cc2cnn(C)c2)nnc(-c2cnsn2)n1C 3429,C1(CC(=O)NCCn2ncc(CC)c2)CCN(C(c2cnc(NC)cn2)=O)CC1 3430,N1(C(C(C)n2cnnn2)=O)CCCC12CCN(C(=O)CCCC#N)C2 3431,Cc1cc(=O)ccn1CC(=O)NCCCN(C)C(c1coc(C(F)(F)F)n1)=O 3432,C12(C(=O)NCC3(CC(=O)OCC)CC3)CC(CN(C(C3CC(C)=NO3)=O)C1)C2 3433,c1(OCCC)nc(C)ccc1C(N1CC2(C1)CN(C(c1ncc(CC)[nH]1)=O)C2)=O 3434,Cc1cc(S(=O)(=O)CCNCC(O)COC(C)(C)C)c(C)cc1-c1cn[nH]c1 3435,C=CCC(CC)C(=O)N1CCCC(O)(CNC(c2csc(Cl)n2)=O)C1 3436,C1(NC(CCc2cc(OC)no2)=O)C2CN(C(C3CC(C)OC3C)=O)CC12 3437,N1(C(C2C(C(C)C)C2)=O)CCC(OCCCNC(C2(CC#N)COC2)=O)CC1 3438,c1(C(=O)NC(CC)CNC(=O)COC2CCCOC2)c(Cl)n[nH]c1C1CC1 3439,OC1(CNC(=NCC2CCCSC2)NC2CCOCC2)CCCCC1 3440,c1(OC)ccc(O)cc1C(N1CC2CC1C2C(=O)NCCc1ncc[nH]1)=O 3441,N1(C(c2c(C)nc(CC)o2)=O)CCN(C(=O)COCC2CCOC2)C(C(F)F)C1 3442,C(=O)(C1=CCC(C)(C)CC1)N(C1CCN(C(=O)C(O)C(C)SC)CC1)CC 3443,Cc1ncc(NC(C2CC(O)CN2C(C2C3(CC3)C23CC3)=O)=O)cc1C#N 3444,Cc1cc(F)ccc1C(N1CCC(N(CCO)C(C2OCC2(C)C)=O)C1)=O 3445,N1(C(c2cc(C)n(C)c2)=O)CC2(C=C(C(=O)N(C3CCCCC3(C)C)C)CO2)C1 3446,C(CC(C)C)(C(=O)NC1CCN(C(=O)C(F)C(C)C)C1(C)C)OC 3447,Cc1c(F)cc(CNc2cccc(C(=O)Nc3c(F)cc(Cl)cc3Br)c2)cc1Br 3448,c1(NC(C(=O)NCC2C(C(=O)OC)C3C2CC3)=O)ccc2c(c1)OCC2 3449,C(CO)(C(=O)NCC=CBr)NC(c1cscn1)=O 3450,CCCCCCCC(=O)N1CCCC(C(C)NC(c2cccc(Cl)c2F)=O)C1 3451,C1(C(=O)NCCCN(C(=O)CCn2cnccc2=O)C)CN2CCN1CC2 3452,C1(C(=O)NCC=CC(=O)N(CC(COCC)O)C)CCC(C)O1 3453,C1(NC(CC2(COC)CCCC2)=O)(CO)CCN(C(=O)CC2CC(C)(C)CO2)C1 3454,c1(CN(C(C)(C)C(=O)NO)C(=O)COCC(=O)O)ccc2cc[nH]c2c1 3455,c1(C(N2CCC(NC(CC3=NNC(=O)C3)=O)C(F)C2)=O)cc(=O)n2nccc2[nH]1 3456,c1(C(=O)NC(C(C)(C)NC(C=CC)=O)C)cc2[nH]nc(C)c2cn1 3457,N1(C(CC=CC)=O)CCN(C(C2CCCN(C)C2)=O)C(c2cn[nH]c2)C1 3458,CCCC(C(=O)NCCC1CN(C(c2cccnc2-n2ccnc2)=O)C1)OC 3459,C1(NC(C2C(NC(C(C)S(N)(=O)=O)=O)CC2)=O)CCC2(CCC2)CC1 3460,c1(SCC)ccc(C(N2CCC(COC)(NC(=O)C(C)c3cc[nH]n3)C2)=O)cc1 3461,C1(NC(CC2CC(SC)C2)=O)C2CN(C(c3coc(CN(C)C)n3)=O)CC12 3462,CC1(CNC(C2C3(CC3)C23CC3)=O)CCN(C(=O)C=Cc2cnc[nH]2)CC1 3463,C=C(C)C(C)(O)C(=O)NCCOC1CCN(C(c2cccc(SC)c2[N+](=O)[O-])=O)C1 3464,Cc1nn(C)c2c(N(C)C(C)C)nc(=NC(C)CC3CCCCC3)[nH]c12 3465,C(CNC(C1CCN(CC(C)C)CC1)=O)(C(C)C(C)C)NC(c1cc(C)ns1)=O 3466,C1(NC(C(CC#C)O)=O)CN(C(=O)C=C2CCC2)CCC1(C)C 3467,C1(CC)CN(C(C2C(C)(C)C2(C)C)=O)CCN1C(c1cc(OC)ccn1)=O 3468,c1(OCC(=O)NC2(CCNC(Cc3n(C)ccn3)=O)CCC2)cccc(F)c1F 3469,N1(C(C(C)O)=O)CC(C)OC2(CCN(C(c3nccc4ncccc34)=O)CC2)C1 3470,N1(C(C(C(=O)NC)(C)C)=O)CCC2(CCN(C(=O)COC3(C)CCC3)C2)C1 3471,C1(C(N2CC(O)(CNC(C(C)CC(F)F)=O)C2)=O)CCCC(F)(F)CC1 3472,c1(NCC2CCCN(C(CCC(C)OC)=O)C2)c(C(C)=O)cc([N+](=O)[O-])cc1Cl 3473,Cc1nc(C)c(C(=O)NCC2(CNC(=O)CCC(=O)N(C)C)CCOCC2)[nH]1 3474,CN1CCCCCC1C(=O)NC1CC(O)CN(C(=O)C2=C(Cl)CC2)C1 3475,C1(CS(=O)(=O)Nc2cccc(-c3ccnc(C)n3)c2)COC2(CCC2)CO1 3476,[nH]1c(N2CCOCC2)nnc1-c1cnn(-c2ccccc2)c1.c1(C=O)ccoc1 3477,c1(OC)cccc(COCC(=O)NC2CC(CNC(=O)COC(F)F)CC2O)c1 3478,c1(C(C(N2CCN(c3ccc(OC)cc3)CC2)=O)(F)F)cnc(O)nc1O 3479,N1(C(=O)N(C)C)Cc2ccc(NC(CC(=O)OCC)c3ccccc3)nc2C1 3480,CC1CN(C(N2CCC(N3CCCC3)C2)=O)CC1CS(N)(=O)=O 3481,CC1CN(C(=O)CCc2ccc(O)nn2)CCCN1C(c1ccc(F)cc1Cl)=O 3482,N1(C(=O)Cc2ccco2)CCOC(CC(N2CCCOCC2)=O)C1 3483,c1(C(=O)NC(CCOC)CNC(=O)C(C)CSC(F)(F)F)cnc(C#N)s1 3484,N1(C(CCCc2onc(C)n2)=O)CC2(CCN(C(=O)CN(C)C)CC2)C1 3485,C1(C(N2CCCC2CNC(c2ns[nH]c2=O)=O)=O)(OC)CCSC1 3486,S(=O)(=O)(c1cc(C(N2CCC3(CC2)CC(CNC(=O)C2CC2)C3)=O)n(C)c1)NC 3487,Cc1nn(C)c(C(=O)NCc2cc(O)nc(CNC(=O)C(O)CF)n2)c1Cl 3488,C(=O)(C(C)(C)CC(C)C)N.C1(C(=O)OC2C(OC)CNC2)CC1C1CCCC1 3489,C1(C(=O)NCc2cc(CO)on2)(COC)CN(C(=O)CCc2cnc[nH]2)C1 3490,C1(NC(C2(C)C=CCC2)=O)CCC2(CC1)CC2NC(c1cncc(O)c1)=O 3491,c1(C(=O)NCCN(C(=O)CCn2ncn(C)c2=O)C)cncc([N+](=O)[O-])c1 3492,C1(C#CC(=O)NC2CCC(CNC(c3csc(C(C)=O)n3)=O)C2)(CC)CC1 3493,c1(COC)noc(CCNC(=O)NCCF)n1 3494,CN1CC=C(C(=O)NC2CCC(NC(=O)C(CCO)N(C)C)CC2)C1 3495,N1(C(CCC(=O)NCCC)=O)CCN(C(C2CCC(F)C2)=O)CC12CCC2 3496,C(C(CCC)C(=O)N1C(C(=O)OC)CC1C)NC(COC1(C#C)COC1)=O 3497,N1(C(C2C(NC(C3CN4CCC3C4)=O)CCOC2)=O)C2C=CCC1CCC2 3498,C(=O)(CS(C)(=O)=O)N1C(C(=O)NC(C=C)(C)CC)CC1 3499,Cc1cc(C(N2CCCC2CCCNC(=O)CCc2cnc[nH]2)=O)cc(C)c1F 3500,c1(C(CNC(c2ccc(F)cc2)=O)NC(=O)CN2CCOCC2)cc(F)cc(Cl)c1 3501,C1(C(N2C(CN(C(=O)C=C3CCC3)C3CC3)CCC2)=O)CC2C=CC1C21CC1 3502,c1(OC(CC)C)cc(NCC2CN(C(C3(O)CCCCC3)=O)CC2C)nc(C)n1 3503,c1(C(N2CC(NC(CSCC)=O)C(CO)CC2)=O)cc2c(C)sc(C)c2s1 3504,Cc1cnc(C(=O)N(C2CCN(C(c3ccc(C)s3)=O)C2)CCO)nc1 3505,CC1OC(=O)NC1C(=O)NCC#CC(=O)NCC#CCCO 3506,Cc1ccc(-c2nnc(S)n2CC(=O)OCc2noc(N(C)C)n2)cc1 3507,c1(-c2n(C3CC(OC)C(CO)C3)ccn2)ccc(-c2cccc(SC)c2)cc1F 3508,N1(C(c2cc(C)c(O)cc2)=O)CC(C)(CNC(C2CCC(=O)NC2)=O)CC1(C)C 3509,CC(C)CC(Cn1cc(C2(C)CC2)nn1)NC(=O)CSc1ccccc1 3510,N(C1CCc2ccccc21)(CC(=O)OC)C(=O)CO 3511,C1(CC)C(NC(c2cc(Cl)ccn2)=O)CCN1C(C1CC1c1ccccc1)=O 3512,CC1CN(C(=O)CSCCC#N)CCC1CNC(=O)Cn1ccccc1=O 3513,N1(C(C2CC(OC)C2)=O)CCC2(CC(NC(=O)Cc3ccnc(Cl)c3F)CO2)C1 3514,N1(C(c2ccc(C)c(Cl)c2)C(=O)NC(C)(C)C)CCOCC2(COCCN2C)C1 3515,c1(C(N2CC(O)CC(NC(C=CSC)=O)C2)=O)cc2cc(Br)ccc2o1 3516,c1(C(=O)NC2(C(=O)NCC(C)(C)C#N)CC2(C)C)ccc(C#N)cc1 3517,N1(C(C2N(C(c3cc(C)[nH]c3C)=O)CCC(F)C2)=O)CC2(CC(CO)CO2)C1 3518,c1(CC)ccc(C(N2CC(CNc3ncc(Br)c(C)n3)CC2C)=O)cc1F 3519,C(CC1=CCN(Cc2ncsc2Br)CC1)NC(C1CCCC(F)C1)=O 3520,c1(OC)ncnc(OC)c1CNC1CN(c2nccc(C(F)F)n2)CC1C#N 3521,c1(C(=O)NCC2C(C)CN(C(C34CC5CC3C4C5)=O)CC2)ccn2ccnc2c1 3522,N1(C(CSc2ccc(OCC)cc2)=O)CC(C(=O)O)c2ccccc21 3523,N1(C(C(CCC)=CCC)=O)CCCCC(NC(=O)C(C)N2CC(C)C2)C1 3524,C(CCCCCCC(=O)N(CCCOC)C)NC(C(CCC)OC)=O 3525,N1(C(C2C(C3CN(C(=O)C=CC(F)F)C3)C2)=O)CC(CO)C2(CCC2)C1 3526,c1(CC(=O)N(CC(C)CNC(=O)C(C)OCC2CC2)C)cc(Cl)ccc1Cl 3527,C#Cc1cccc(C(=O)NCC2CCCCC2NC(C2CCSCC2)=O)c1C 3528,c1(C(=O)NC2CC(C)CN(C(C3(O)CCOC3)=O)C2)ccc(S(N)(=O)=O)c(F)c1 3529,Cc1cc(C(N2CC3CC(C2)N3C(C2(F)CCC(C)CC2)=O)=O)cc(O)n1 3530,c1(COC)nc(Cl)cc(=NCC2(C)CCC(NC(C3C=CC=CC=C3)=O)CC2)[nH]1 3531,C1(C(=O)NCc2nn[nH]n2)(COC)C=CCN1C(c1cc(C)sn1)=O 3532,N1(C(C(C)(C)CF)=O)CCC(CNC(=O)C(c2ccc(F)cn2)(F)F)C(F)(F)C1 3533,C1(C(=O)NCCC2(O)CN(C(c3nccc(C)c3)=O)C2)CCCS(=O)(=O)C1 3534,Cc1nc2n(c(=O)c1COCCn1c(=O)ccn3c4ccccc4nc13)CCCC2 3535,N12CCN(C)C(C1)C=CC2=O.C(C)(C(=O)N(C1CCC1)C)SC 3536,C(=O)(C(CCCC(C)(F)F)N(CCc1ccccc1)CC)NCC=C 3537,c1(C(N2CC(SC)C(NC(C3C(C)C3C)=O)C2)=O)cc(C#N)ccc1Cl 3538,c1(C(=O)NCC2(C)CC(NC(C(CCC)CC)=O)C2)c(C)nc(C)nc1C 3539,CCC(CC)C(C(=O)NCC(CC(F)(F)F)NC(=O)CS(N)(=O)=O)OC 3540,c1(C(N(C(C)C(N2C(C)CC2(C)C)=O)C2CC2)=O)cc(C#N)n(C)n1 3541,C1(NC(C(c2ccc(OC)cc2C)C)=O)CN(C(=O)C(N)=O)C2(CCCC2)C1 3542,N(C(=NCCc1cc(Cl)ccc1Cl)NC1CC1C1CC1)CCC(C)C 3543,c1(C(C)NCC=C(Cl)Cl)ccc(C(C)(C)C)cc1 3544,C1(CN(C(=O)NC)CC)CCCS1(=O)=O.c12cccc(c1)C1(CCC1)N2 3545,C(=O)(C1=CCCOCC1)NCC(C(N1CC[Si](C)(C)C1)=O)CC1CC1 3546,Cc1cc(C(=O)NC2CC(CNC(c3[nH]cnc3C)=O)CC2O)nnc1O 3547,C1(C(=O)Nc2cnn(C3CCNC3=O)c2)CNCC2(CCC2)O1 3548,C1(N(C(C)C)C(=O)NCC(C2CCCO2)O)CCN(C)CC1 3549,C#CCC(C(=O)N1CCC(CC(=O)Nc2ccccc2OCC)C1)C1CC1 3550,Cc1cc(C(=O)NC2CCN(C(c3cn(C)nn3)=O)CC2C)ccc1Cl 3551,C(C(=O)N1CC(CCNC(C2CCCO2)=O)C1)(C(C)O)NC(C)=O 3552,S(=O)(=O)(c1cccc(Oc2ccccc2)n1)N(C(CCC)C(=O)O)C 3553,c1(C(=O)OC)cc(NC(=O)NC(c2cccc(OC(F)F)c2)C)ccc1F 3554,N1(CC(=O)NC2(C)CN(C(c3ncn(C(C)C)c3)=O)C2)CCn2nccc21 3555,C(C(N)=O)(C(C)CC)NC(C(C1CCN(C(CC2ON=C(CC)C2)=O)C1)F)=O 3556,N1(C(C(C=C)O)=O)CCC2(CCC(NC(c3cc(C)c4[nH]nnc4c3)=O)CC2)C1 3557,n1(CC#C)cccc1C(=O)NC1(C(=O)NCC2CN(C(C)C)C2)CCSC1 3558,N1(C(c2ccc(Cl)c(C(F)F)c2)=O)CCc2ccc(Br)cc2CC1 3559,c1(C(N2CC(CN(C(Cc3c(C)nccc3)=O)C)C2)=O)cc(F)c(F)c(Cl)c1 3560,c1(C(N2C(CCC(=O)NC(CC=C)C3CC3)CCC2)=O)ccc([N+](=O)[O-])[nH]1 3561,C(=O)(C1=NN2CCCN=C2N1)NC(CNC(=O)C=CC=C(Cl)Cl)C1CCC1 3562,C1(CN(C(Cc2cn(CC)nc2)=O)C)C2CN(C(C3CCCC3O)=O)CC12 3563,c1(OC)ccc2c(C)c(C(=O)NC3CCC4(CC3)CC4)[nH]c2c1 3564,c1(C(N(CC(CN(C(=O)Cc2cnoc2)C)O)C)=O)ccn(CCF)n1 3565,C1(F)(CNC(c2nc(CC)oc2C)=O)CCCN(C(c2ccon2)=O)C1 3566,N1(C(=O)Cn2ccc(C(F)(F)F)n2)CCCC2CCN(C(=O)C3=COCC3)CC12 3567,C=Cn1nncc1C(=O)NC1(CN2CCN(C(=O)C(C)O)CC2)CC1 3568,c1(CCCSC)cn(CCN(C)C(C2CC2(C)C)=O)nn1 3569,S(=O)(=O)(c1c[nH]ccc1=NC(CF)CF)NCc1cc(C)no1 3570,Cc1ccsc1CCCC(=O)NCCOCCNC(=O)C(C)C1(O)CCC1 3571,c1(C(=O)NC(CC)CNC(c2cc(C)no2)=O)c(Cl)ccc(Cl)c1OC 3572,C1(CNC(CCCCC=C)=O)CN(C(=O)C(F)(F)C(O)CC)CCC1(C)C 3573,C(=O)(C(C)(CC)CCC)N1CC(C(C(N2CCCC(OCCC)C2)=O)O)C1 3574,CCS(=O)(=O)CC(=O)NC(C)C(C)NC(c1ccoc1CC(N)=O)=O 3575,C(=O)(C(CSC)c1ccccc1)NCCN(C(C1CC=CCO1)=O)CC 3576,C1(C(N(CC(=O)NC(C)C)C)=O)(CO)CCN(C(c2cnn(C)c2N)=O)C1 3577,C1(CC(C)C)COCCN1C(=O)NCCNC(c1ccc(-n2nccn2)cc1)=O 3578,c1(C(=O)NC2C(CNC(C3(C#C)CC3)=O)C2)ccc2c(c1)CCN2S(C)(=O)=O 3579,N1(C(CC(C)(F)F)=O)CC2(CCC(NC(=O)CC3NC(=O)NC3=O)CC2)C1 3580,C1(C)(C(=O)NCCC2(O)CN(C(c3cc(COC)[nH]n3)=O)C2)CCCC(F)(F)C1 3581,C1(C(=O)NCCCNC(C(C(C)(C)C)O)=O)CC(O)c2ccccc2O1 3582,C(=O)(C1CCc2nccn21)NCC(=O)NCc1c(C)nsc1 3583,CC1=C(C(=O)NC2CCCCCC2NC(=O)Cn2nc(C)nc2C)CCS1(=O)=O 3584,N1(C(C(C)C)=O)CCn2ncc(CN(C)C(C3CC4CCC3C4)=O)c2C1 3585,c1(C(N2CCN(C(Cc3scc(C)c3)=O)CC2C)=O)nn(C)c2c1CCC2 3586,c1(CC)nc(O)c(C(N2CC(CNC(c3occ(C)c3C)=O)C2)=O)cc1C 3587,C(CC(C)N=c1[nH]c(=NCC2CC2c2ccc(Cl)cc2Cl)c2ccccc2[nH]1)OC 3588,C12CCN(C1)C2.C1(CC(=O)N(CC(F)(F)F)CC)(Nc2cn(C)nn2)CCCC1 3589,CCC(CN(C)C)CC(=O)NC(C)CC1CN(C(C2CC2C(C)O)=O)C1 3590,C(=O)(CC(C)(C)SC)OC1(CC=C)COC1 3591,C1(CC(=O)NCCc2ncc(C)o2)CCCN(C(c2sc(C)nc2C)=O)CC1 3592,Cc1cnc(NCC2CC(NC(C34CCCC3C4(F)F)=O)C2)nc1S(C)(=O)=O 3593,C#CCCCCC(=O)NCC(C)(O)CNC(c1ccc(C(=O)C2CC2)cc1)=O 3594,C1(NC(c2ccc(CNC(CC(C)O)=O)cn2)=O)CCCN(C)C1C 3595,c1(C(=O)NC2C(NC(c3c(N)nc(Cl)cc3)=O)COC2)cnn2c(=O)cc[nH]c12 3596,C(=O)(CC(C)CC(C)(C)C)NC1CCN(C(C(c2c(C)noc2C)C)=O)C(C)C1 3597,C(CCC)(C(O)C(=O)N1CC=CC1CF)NC(C(C)OCC#C)=O 3598,N1(C(c2c(OC)csc2)=O)CCCN(C(c2ccnn2CC(C)C)=O)C(CO)C1 3599,c1(C(=O)NCCC(CNC(=O)C=Cc2ccccc2)O)cccc2ccnn12 3600,C(CC(=O)NC1CC1C(N1CCC1C)=O)OC 3601,c1(C(CO)NC(=O)NCc2nc(C(=O)OCC)nn2C)ccc(C)c(C)c1 3602,C(=O)(CCS(=O)(=O)Cc1ccncc1)N1CC(N(C(=O)C2=CCSC2)C)C2(C1)CC2 3603,N1(C(CCN(C(=O)CC2CCOC2=O)CC#C)=O)CCC2(CC1)CC2C#N 3604,C1(CNC(c2ccc(OC)cn2)=O)CC2CN(C(c3cc(C)nc(C)c3)=O)CC12 3605,C(=O)(C1=C2CCN=C2NC=C1)N1CCC(N(C(=O)CS(C)(=O)=O)C)CC1 3606,C(N=c1nc(N2CCC3(CCCN(C)C3)C2)c2sccc2[nH]1)C1C(C)C1(F)F 3607,c1(CNC(C2CC(C(C)(C)C)C2)=O)ccc(Cl)nc1.C12(CC1)C(=O)NC2 3608,CC1CC(c2nn[nH]n2)CC(C)N1CC(C)(C)CO 3609,Cc1ccc(C(=O)NC2CCC(C)N(C(C3CC4(C3)CC(F)C4)=O)C2)cc1CO 3610,c1(CC)cccc(C(=O)NC2CC2NC(=O)COc2ccc(C)cc2)c1C 3611,N1(C(CC2C(OC)COCC2)=O)CCC2(CCNC2)C1 3612,C1(CC(=O)N(CCC(N)=O)C)CN(C(c2cc(O)cc(=O)o2)=O)C(C)(C)C1 3613,N1(C(COCCC)=O)CCC(C(=O)NCc2cn(C3CC3)nn2)C1C 3614,c1(C(N2CC(O)(CN(C)C(c3cc(C(N)=O)cn3C)=O)C2)=O)cnc(O)n1C 3615,c1(C(=O)NC(C)C(C)(C)NC(C2CCC(F)(F)C2)=O)cccc[n+]1[O-] 3616,c1(N(C)C)ccc(C(=O)NC2(CNC(c3ccc(C#N)[nH]3)=O)CCCCC2)cn1 3617,CN1CCC(C(=O)NCC23CC(CNC(=O)CC(F)(F)F)(CO2)C3)CC1=O 3618,c1(SC)ccc(C)c(C(N2CCOCC2CNC(c2ccc(C)c(C)c2)=O)=O)c1 3619,C(C(C)(O)CC(=O)N(C1CN(C(c2c[nH]nc2C)=O)CC1(C)C)C)OC 3620,c1(OC)ccc(OC(=O)CN(C(C(CNC(=O)C(=O)NC2CC2C)C)=O)C)cc1 3621,C1(C)(C(N(C(CNC(=O)CCC2CCCOC2)C2CC2)C)=O)CCCO1 3622,C(=O)(C(C)(C)C(C)(C)O)N1C(CNC(c2cccc(COC)c2)=O)CCC1 3623,c1(N2CC3CC4C(O)C2C3C4)nc(C2CC2)nc2ccccc12 3624,c1(C(N(C2CCCCC2)CCNC(C(c2ccccc2)C)=O)=O)nsnc1O 3625,Cc1nc(C(N2CCC(F)(C(N3CC(O)CC3C(N)=O)=O)C2)=O)ccc1Br 3626,C(CC(CC)C(=O)NC1C=CCC(C(=O)N(CCN2CCOCC2)CC)C1)=CC 3627,C1(CNC(c2n(C(C)C)ccc2)=O)CCC2CN(C(C3CN(C)C(=O)N3)=O)CC12 3628,C(=O)(C(CNC(c1cc(C2CC2)no1)=O)C(C)(C)C)NC(c1nncn1C)C 3629,N1(C(C2C(=O)CC2)=O)CC2(CCC(CNC(=O)Cc3ccc4c(c3)CCC4)O2)C1 3630,C(=O)(C1CNC(=O)c2ccccc21)NC1C2CN(C(C=COCC)=O)C1C(O)C2 3631,C=CC(O)(C(=O)NCCC(C)N(C(=O)C=CC(F)(F)F)C)C(F)(F)F 3632,c1(OC)cc(C)c(C(=O)NCCOc2ccc(NS(C)(=O)=O)cc2)o1 3633,C1(C(=O)NC(C)C)CC(NC(C2CC(C)(C)CO2)=O)C(O)C1 3634,C1(CCCNC(C(F)=CCC)=O)CN(C(c2ccnc(OC)n2)=O)CCO1 3635,n1(CC(=O)N(CCCCCNC(C2CC2Cl)=O)C)ccc([N+](=O)[O-])n1 3636,CCC(CNC(C1CN(C(=O)CCC(C)(C)C)CCN1C)=O)CC(C)C 3637,C(CC(=O)NCCC(O)C1CC1)(C(F)(F)F)NC(C1(COC)CCCC1)=O 3638,N1(C(=O)CC(F)(F)CCc2ccccc2)CCC2(CC1)CC(F)CO2 3639,C1(NC(C2N(C)CCCC2)=O)CCN(C(=O)CNc2cnn(C)c2)CCC1CO 3640,C=CCC(CC(C)C)C(=O)N(C(C)CCNC(=O)Cc1nsc2ccccc12)C 3641,N1(C(C(C)SC(F)(F)F)=O)CC2CCN(C(c3nnn4c3CSCC4)=O)CC2C1 3642,c1(C(N2C(CCCNC(C(C)OCC#C)=O)CCC2)=O)cccc(Cl)c1N 3643,C1(NC(c2cc(CCC)[nH]n2)=O)CC(O)CN(C(=O)Cn2cc(F)ccc2=O)C1 3644,C(CC(O)C(F)(F)F)NC(C(CC=CC)NC(=O)CC1CCOC1=O)=O 3645,C(=O)(C1=COCCC1)NCC(CC(C)C)NC(c1cncc(CO)c1)=O 3646,N1(C(C2CCCC(OC)C2)=O)CCC2(CC1)CCN(C(C1CC1C)=O)CC2 3647,CCC(C)C(C(=O)NCCCCC(=O)NCCN(C)CCOC)N(C)C 3648,N1(c2ncc(C(=O)OC)c(C)c2)CC2CC(NC(=O)CCC(C)(C)O)CC1C2 3649,c1(C(=O)NC(CNC(C(C(C)C)n2cccc2)=O)CO)cn2cnnc2cn1 3650,c1(CC(C)C(=O)NCCCNC(C)=O)ccc(F)cc1.c1(CSCC#N)ccc(C)o1 3651,N1(C(C2(CC#C)CCCOC2)=O)CCC2(CC1)CC2CNC(=O)CCOC 3652,C(=O)(CCN(OC)C(=O)c1ccc(C#N)[nH]1)N1C(C)CC1 3653,N1(C(Cc2ccc(C)cc2)=O)CCCC(C)C1CNC(=O)C=CC1CCOCC1 3654,C1(F)(CNC(C2C(C(N)=O)COC2)=O)CCN(C(=O)CC2CCCNC2=O)C1 3655,C1(C(N(C)Cc2cn(CC)nn2)=O)CCC(C)(C)N(C(c2ccc(OC)s2)=O)C1 3656,CC1CC2(CCO1)CC2C(N1CC(OCCNC(c2conc2C2CC2)=O)C1)=O 3657,c1(C(=O)NCC2(OC)CN(C(c3ccnc(OC)n3)=O)C2)c(C)cnnc1O 3658,N1(C(CCCC(N)=O)=O)CCC2CN(C(=O)C=CCN3CCOCC3)CC12 3659,N1(Cc2c(OC)nccc2)CC(NC(c2ccc(C)[nH]2)=O)C(C)(C)C1 3660,N1(CC)CC2CN(C(=O)C(CC)NC(c3ccc(F)cn3)=O)CC2C1 3661,Cc1c[nH]c(C(N2CCOCC2CCNC(C2(C(F)(F)F)CCC2)=O)=O)cc1=O 3662,C(c1cscn1)=CC(=O)N(C1CCN(C(c2sccc2CC#N)=O)C1)CCC 3663,c1(NC2(N(C(=O)OC(C)(C)C)NC(C=C(COC)C)=O)CC2)ccnc(C)n1 3664,c1(NCCNC(C2(N(C)C)CCCC2)=O)ncnc2ccccc12 3665,c1(C(=O)NCC(CNC(=O)C2=CCCS2)O)coc2c(Cl)cccc12 3666,Cc1nc2cccc(C(=O)NC3CC(NC(c4cc5sc(C)c(C)c5[nH]4)=O)C3)n2n1 3667,CCC(C)C(O)C(C)C(=O)NCC(C)(C)C(N1CCCC(F)(F)C1)=O 3668,N1(C(C2(SCC)CC2)=O)CCCC(CC)(NC(c2cc(C(C)=O)oc2C)=O)C1 3669,c1(C(N(CC(C)(C)CNC(=O)Cc2nncn2C)C)=O)cnc2c(c1)ncn2C 3670,N1(C(c2scnc2C2CC2)=O)CCN(C(C2(C(=O)NC3CC3)CC2)=O)C2CC12 3671,C1(C(N(C(CNC(c2cnc(CC)s2)=O)C)C)=O)(OC)CCC(F)(F)CC1 3672,Cc1cc(C)c(C(N2CC(NC(c3cncc4ccsc34)=O)CC2C)=O)cc1C 3673,C1(NC(c2n(CC)ccc2)=O)CN(C(=O)C=CC2CCCO2)CC2(CCC2)C1 3674,N1(C(C)C)CCCC1C(=O)NCCC(C)(C)NC(=O)C(C)CC1CCCCC1 3675,c1(OCCC(=O)NC2CCC2NC(=O)C(=O)NC2CC2)ccc(Br)cc1 3676,N1(C(C(CC)C(C)C)=O)CC2CCCC(NC(C3CCCS(=O)(=O)C3)=O)C2C1 3677,c1(C(=O)NCC(COC)NC(c2c[nH]nc2C)=O)ccc2n[nH]cc2c1Cl 3678,n1(CC(=O)NCC2OCCN(C(C)=O)CC2)ncc2ncccc12 3679,c1(C(=O)NCC2CC(OC)CN2C(=O)C(C)C2CCCC2)c(Cl)c(C)nn1C 3680,N12CCC(CC1)CC(=O)O2.c1(C(CC(C)(C)C)O)ccc(O)cc1 3681,C(=O)(C(O)CCS(C)=O)NC1CC(CCNC(CCCCOC)=O)C1 3682,N1(C(CN(C)C(c2ccco2)=O)=O)CCN(C(C2CCCS2)=O)CC1 3683,c1(C(=O)Nc2cccc(NC(c3cc(C)oc3C)=O)c2)cnc2n1CCCC2 3684,N1(C(C(CSC)OC)=O)CCN(C(c2cnnc(O)c2)=O)C(C)C1 3685,Cc1nn(C2CC2)cc1C(=O)NC(CNC(=O)CC(O)c1ccccc1)CO 3686,C(=O)(C(CNC(c1cccc(F)c1F)=O)C(C)(C)C)N1C(C=C)COCC1 3687,N1(C(C2(CC)CC=CC2)C(=O)NCC2CCCO2)CCC(C)(CCO)C1 3688,Cc1ncccc1C(=O)NC1CC1C(N1CCC(Cc2ccc(Br)cc2)C1)=O 3689,C(=O)(C#CC1(C)CCCO1)NC(C1CC1C(=O)NC1(C)CCCC1(F)F)C 3690,CC1(C)CCCN(C(C2OCCO2)=O)C1CNC(c1c(F)cc(F)cc1F)=O 3691,N1(C(CCCC)=O)CCC(C)(CC(=O)NCC(C)CC2CCC2)C1 3692,C1(NC(C(CC)(C)O)=O)CN(C(=O)CCn2ccnc2C)CC(C)(C)C1 3693,N1(C(C(CC)OC)=O)CC2(CNC(c3ccc(C(N)=O)[nH]3)=O)CC1CO2 3694,n1(CCNC(CC(C(C)C)c2ccc(F)c(F)c2)=O)cnc2c1CCCC2 3695,C(=O)(C(C(=O)N(C1CCN(C(=O)C(c2cccc(C)c2)(C)C)C1)C)OC)OCC 3696,N1(C(c2ccc(SCC)nc2)=O)CCN(C(c2ncc(C)cc2F)=O)CC1CO 3697,C(=O)(CC1CCc2ccccc21)N1C(CNC(=O)C#CC2CCOCC2)CC1 3698,c1(C(N2C(CNC(c3cn(CC)nc3)=O)C=CC2)=O)cc2cc(Cl)cnc2o1 3699,CC1CCCN(C(C2(n3cccc3)CC2)=O)C1CNC(=O)CC(C1CC1)C1CC1 3700,N(C1CN(C(=O)C(O)C2CC2)Cc2ccccc21)C(Cn1c(=O)ccc(C)c1)=O 3701,Cc1cc(F)cnc1C(c1nnnn1C1CCCCCC1)NC1CC(F)(F)C1 3702,C1(NC(CCC=C)=O)CC2C(NC(=O)C(C)(C)n3cnnn3)C2C1 3703,c1(N2CCC(NC(c3n(C(C)C)ncc3)=O)C(C)C2)nc2ccc(Br)cc2o1 3704,c1(COCC(=O)NCC(C)(CC)NC(c2cnc(OC)s2)=O)nnc(S)n1C 3705,C1(C(=O)N(CC(F)F)C)(CNC(c2c(CC)cns2)=O)CC(C)(C)C1 3706,Cn1ncc(C(=O)NCC(C)(C)OCC(=O)NCC2C(C)(C)C2(F)F)c1Cl 3707,n1(NC(=O)NCC2(O)C(SCC)CC2)ccc(Br)cc1=O 3708,CC(C)(C(=O)NCC1CC1CNC(=O)COCP(C)(C)=O)n1cccn1 3709,N1(C(C2(C#C)CC(=O)C2)=O)CCCC(CC(=O)NCC(C)C(=O)OC)CC1 3710,C=CC(C)CC(=O)NC(CCOC)C(=O)N(C)Cc1cncnc1 3711,N1(C(C2(C)N(C(c3c(C)oc(C#N)c3)=O)CC=C2)=O)CCC(O)C(F)(F)C1 3712,C1(NC(=O)OC)CCN(C(=O)C(F)C2CC(NC(=O)CC3(CSC)CC3)C2)C1 3713,C(=O)(CCS(=O)(=O)N(C)C)N1CCCC(CN(C(=O)C(Cl)=CCl)C)C1 3714,O(NC(=O)C(C(C)NC(c1cn2ccccc2n1)=O)C(C)C)CCOC 3715,CC(C)(C)C(C(=O)NC1CCN(C(C2CCCCNC2=O)=O)CC1)NC(N)=O 3716,N1(C(C=CC(C)NC(C=Cc2cc(C)no2)=O)=O)CC(CC2CC2)CC(C)(C)C1 3717,C(CCC(C)C)(C(=O)N1CCC(O)(C(=O)O)CC1)N1CC2C(C(=O)OCC)(C2)C1 3718,N1(C(C2CCN(C)C2)=O)CC2(CCC(CNC(=O)C(C)(C)C(C)(F)F)O2)C1 3719,c1(CN(C2(C)CCN2Cc2ccccc2)Cc2cc(SC)n[nH]2)ccc(O)nn1 3720,c1(C(=O)NCC2N(C(c3c(C)ncs3)=O)CCC2)cc(O)c2ccoc2c1 3721,c1(C(N2CC(COC)(CNC(=O)CNS(C)(=O)=O)C2)=O)cc(F)cc(F)c1O 3722,N#Cc1cc(CN2CC3C(C2)N3C(c2ccncc2O)=O)ccc1Cl 3723,N1(C(C23CCC(OC)C2C3)=O)CC2CCCC(C1)N2C(C1(C(C)(F)F)CCC1)=O 3724,c1(OC)ccc(C)cc1NC(C1CCN(C(=O)C2=COCC2)C1(C)C)=O 3725,C=CCC(CNC(C1CC(C)(C)CN1C(=O)CCCCOC)=O)CC(C)C 3726,CC(CC(=O)N1CCCCC1C(N)=O)C(C)(C)NC(=O)Cn1cnnc1O 3727,C(=O)(CC(C)(CN(C)C)C(F)(F)F)N1CCC2CN(C(CCC(=O)NC)=O)C2C1 3728,N1(CC(=O)N(C(C)CCO)C)CCN(C(=O)C(c2cnn(C)c2)O)CC1 3729,c1(C(=O)NC2CC(NC(c3cc(C)nc(C)n3)=O)C2)cc2ccccc2[nH]1 3730,c1(NC(CNC(C(=O)OC)Cc2ccc(I)cc2)=O)ccc(OC)nc1C 3731,c1(C(=O)NC(C(=O)N(CCC(=O)OCC)C)C2CCCC2)cc(CC)c[nH]1 3732,C=CCCN=C(NCc1cc(Cl)cn1C)NC1CCOC(c2ccccc2)C1 3733,C1(C(CC2N(CC#C[Si](C)(C)C)CCOC2)=O)CCOC2(CCC2)C1 3734,C=CC1CCN(C(C2(NC(C3CC4CC4C3)=O)CC(O)C2)=O)C1 3735,c1(OC)ccc(CNC(=O)NCC2CCCC(F)C2)nc1 3736,N1(CCNS(CC)(=O)=O)CCCC(C(C)NC2CC(=O)N(C)C2)C1 3737,Cc1nsc(N2CCN(C(=O)C(=O)N(CC(C3CCOC3)OC)C)CC2)c1C#N 3738,N1(C(CCC(=C)C)=O)CCC(F)(CNC(C2CCC(=O)N2C2CC2)=O)CC1 3739,C1(CCNC(C(C)NC(C=CCOC)=O)=O)CCN(C)C1 3740,CC1CN(C)CC(C(=O)N(C(C)C(N2CC(O)(CC(C)C)C2)=O)C)O1 3741,CCC(CC)C(=O)NC1CCC(NC(=O)CNC(=O)CCC2CC2C)C1 3742,C12(Sc3ncoc3C)COC(CN(c3ccc(C(=O)OC)cn3)C(C)=O)(C1)C2 3743,c1(CC)ccc(C)c(C(N2CC3(C2)CN(C(=O)C(c2ccc(Cl)s2)C)C3)=O)c1 3744,N1(C(c2c(OC)n(C)nc2C)=O)C2CCC1CN(C(C1CCC(OC)CC1)=O)C2 3745,c1(C(N2C(C)(CNC(c3cnsn3)=O)CCC2)=O)ccc2ocnc2n1 3746,C12(CNC(C(CCSC)SC)=O)CC1CN(Cc1ccccc1)C2 3747,c1(C(N2C(CNC(C3(CC=C)COC3)=O)CC2)=O)cc(Br)cnc1O 3748,c1(CC)cnccc1C(=O)NCCC1(O)CN(C(=O)CN(S(=O)(=O)CC)C)C1 3749,c1(C(=O)NCCCC2(NC(C3C(C)CCS3)=O)CC2)ccc(OC(F)(F)F)cc1 3750,c1(OC)cccc(OC)c1C(=O)NCCC1CCCN(C(=O)C(C(C)C)OC)C1 3751,c1(OC)ccc2nc(N3CCC4(CCC(CNC(=O)OC(C)(C)C)C4)C3)sc2c1 3752,CN1CCN(C(=O)C(=O)Cc2ccc(Cl)cc2)C(CNC(C2C3COCC23)=O)C1 3753,c1(C(=O)NCC2CCC(C(N(CC=C)Cc3ccco3)=O)O2)c(C)noc1C 3754,c1(-n2cc(CCN(C(=O)C(C)O)CCOC)nn2)ccc(C(F)(F)F)cc1 3755,c1(C(N2CC(NC(=O)C3=COCC3)C(C(F)F)C2)=O)cc2n(n1)CCNS2(=O)=O 3756,CCC(C)(C)CC(=O)NC1(CO)CCN(C(c2csc3cncn23)=O)C1 3757,C1(CC(=O)NCCC2CCCO2)COCCN1C(c1nocc1Cl)=O 3758,c1(C(N(C2CCN(C(=O)CCC3CCCC3)C2)CC)=O)ccc2nc(O)[nH]c2c1 3759,C1(C(=O)NC2(CC)COC2)C2C(CN1Cc1cccc3nsnc13)C2(C)C 3760,c1(C(=O)NCC2(CNC(CCC(=O)OCC)=O)CC2)ccc(C)cc1OC 3761,C(=O)(C1CCc2c[nH]nc21)NCCC1(C)CCN(C(C(CCCC)O)=O)CC1 3762,C1(NC(C2(C)CN(C(C(C=CC)O)=O)C2)=O)CNC(=O)OC1 3763,c1(C(N2CC(C)CCC2C)C(=O)NCCC)ccc(F)c(C)c1F 3764,N1(C(C2CC(C)N(C)C2)=O)C2CCC(C(=O)NCC3CCC3(F)F)C1CC2 3765,C1(F)(NCc2cnc(NC(CN(C)C)=O)s2)CCN(C(=O)OC(C)(C)C)C1 3766,c1(C(CC)C)ccc(NC(=O)Nc2cccc(C(=O)NC3CC3)c2)cc1 3767,c1(C(N(CCNC(=O)C(C)S(N)(=O)=O)CC)=O)c(OC)ccc(F)c1N 3768,C(C(CC(C)C)C(=O)NC1CN(C(=O)Cc2coc3ccccc23)CC1O)OC 3769,c1(OCC)cc(OC)cc(S(=O)(=O)NCC(c2ccncc2)OC)c1 3770,C#CCC(CC(=O)N(C(C)C#C)CCOC)NC(=O)CC(=O)OC(C)(C)C 3771,Cc1nn(C)c2nc(C(=O)NCC3(CNC(=O)Cn4cnnc4O)CC3)ccc12 3772,C1(C(=O)NCCC(CC)(F)F)CC2(CCN(C(=O)C(O)CC(C)(C)C)C2)C1 3773,CCCC(CC1CCCCC1)C(=O)NC1CCCC1NC(c1coc(C)c1)=O 3774,C1(NC(c2cn(CCNC(C(C(C)(F)F)F)=O)nc2)=O)CCn2nnnc2C1 3775,c1(C(N(CC(C)NC(=O)CC(C)C(=O)OC)CC)=O)ccc2ccnc(Cl)c2n1 3776,Cc1cc(C(=O)NC2CCC2NC(=O)C(C)N(C)C)ccc1O 3777,CC1(C)COC(CC(=O)NCC2CC(NC(C3(CO)CCCC3)=O)C2)CO1 3778,C1(COC)(NC(c2sccc2C#N)=O)CCCN(C(=O)CCn2cc(C)cn2)C1 3779,c1(CC)cc(C(=O)NCC(C)NC(c2ccnnc2O)=O)c2c(c1)CCO2 3780,c1(OCC)cc(NC2CC3CCCC(C2)N3C(=O)CSC)ccc1[N+](=O)[O-] 3781,C1(C(N(CCOC)C2CC2)=O)CN(C(=O)C(C)C(F)F)CCO1 3782,Cc1ccc(C(=O)N(C2(O)CCCCCC2)C2CC3(CNC3)C2)cc1C#N 3783,C(c1cccc(F)c1)=C(C(=O)NC(C)CNC(=O)CC1(CN(C)C)CCCC1)F 3784,c1(C(=O)NCCC)ccc(C(=O)NCC(C)(C2CC2)NC(=O)CCC(C)C)cc1 3785,C(C1CSc2ccc(Br)cc21)N1C(C(=O)NCC)CCC1 3786,CC1CC2(CCN(C(C3(c4ccncc4)CC3)=O)CC2)CN1C(=O)CCC(N)=O 3787,C1(C(=O)NC(C)Cc2ccccn2)C2CC1N(C(=O)Cc1ccns1)C2 3788,C(CCCCC1CC1)(c1n(C(CC)C)nnn1)Nc1cnn(C(F)F)c1 3789,N1(C(=O)Cc2ccco2)CC2CCCC(C1)N(Cc1ccc3nonc3c1)C2 3790,c1(C(=O)NCCN(C)C(C2(CO)CCOCC2)=O)sc2cccnc2c1Cl 3791,N1(CC#C)C2CCC1CC(CN1CC3(COCCO3)C1)C2 3792,c1(C(=O)NCC2N(C(C(C)C(F)F)=O)CCCCC2)ccc2ncn(C)c2n1 3793,c1(CC(=O)OCC(=O)NCC(C(=O)OCC)C2CCOC2)ccc(OC)cc1Br 3794,N1(C(c2ccn(C(C)(C)C)c2)C(=O)NC2(C)CC2)CCC2C(C(N)=O)C2C1 3795,C1(NC(CCCOC(C)=O)=O)C2CC3C1C3C2C(=O)NC1(C)CCCC1C 3796,C1(NC(C2CCN(C(C)=O)C2)=O)CCN(C)C(c2ccccc2Br)C1 3797,C1(CC(=O)NC(c2c(C)nccc2)C)CN(C(C2(N(C)C)CC2)=O)CC12CC2 3798,C=CCC(C(=O)NCC1CCC(C(=O)N(c2cccc(OC)c2)C)O1)OC 3799,CC(C)C(O)C(F)(F)C(=O)NC(C1CC(NC(c2ccncc2)=O)C1)C 3800,n1(C(C)C)ccc(C(=O)N(CC(O)CN(C(=O)CN(S(C)(=O)=O)C)C)C)n1 3801,C(N=c1[nH]c(N(C)Cc2ccc(Br)nc2)nc2c1CSC2)C1(OC)CCOCC1 3802,N1(C(C2N(C(N)=O)CCC2)=O)CCCCC1CCCNC(=O)CC1(CO)CC1 3803,CC1CN(CC(O)CNC(=O)C(=O)NC2CCCCNCC2)CC(C)O1 3804,C1(C(=O)NCC2N(Cc3ccccc3)CCN(C)OC2)CCC(C2CCCO2)O1 3805,C(=O)(C(C)CC(=O)N1CC2CC1C2NC(=O)Cc1ccc(Cl)c(Cl)c1)OC 3806,c1(C(=O)NC(CN2CCN(C(C(COC)O)=O)CC2)C)cccc(=S)n1O 3807,C1(CNC(C2C3CCCC23)=O)CCCN(C(=O)CCc2cnc(C3CCC3)s2)C1 3808,N1(C(C(C(C)C)NC(CC(C)C)=O)=O)CCC2(CCN(C(=O)C(=O)N(C)C)C2)C1 3809,c1(C(=O)NC2C(OC)CN(C(=O)CCc3csc(=N)[nH]3)C2)cc(C)nc(C)n1 3810,CC(C)(C)C(CCC1CCCC1)NCC(c1ccc(F)cn1)(F)F 3811,Cc1ccc(CCC(=O)NC(C)CCNC(C2C(C)C2C)=O)c(C)c1 3812,C(C)(C1=CCN(C)CC1)NC(C(c1ccccc1)NC(c1[nH]cc(C)c1)=O)=O 3813,c1(C(=O)NCC(C)CNC(c2n[nH]c3c2CCC3)=O)cc(O)nc(Br)c1 3814,C1(C(N(CC(C)NC(=O)Cc2cc[nH]c2)C)=O)CC(=O)N(c2ccccc2F)C1 3815,CCC1=NOC(C(=O)N(C2CCCCCC2)CCNC(=O)CCCC2CC2)C1 3816,c1(C(=O)NCC2(F)CCN(C(c3c(CC)cno3)=O)C2)cnc(C)cc1C 3817,c1(C(=O)NCC2CCC(NC(C3CC(C)N(C)C3)=O)C2)cc(Cl)ccc1[N+](=O)[O-] 3818,c1(C(=O)NC(CNC(C2N(C)CCC2)=O)(C)C)ccc2c(=N)[nH]cnc2c1 3819,CC(=O)CCCC(=O)NCC12CC1CN(C(=O)COc1ccc(F)nc1)C2 3820,n1(CC)cc(C(N2CCOC(CCCNC(=O)C=C(C)C(C)(C)C)C2)=O)c(C)n1 3821,c1(NC(=O)Nc2c(SCC)cc(Br)cc2)ccc([N+](=O)[O-])cc1Cl 3822,c1(SC(C)C(=O)NCCC2CCN(C(=O)C=CCn3cncn3)C2)ccccn1 3823,c1(C(C)NC2(c3cn(-c4ccsc4C(=O)O)nn3)CC2)cc(C2CCC2)nn1C 3824,CCC(C)(C)CCCC(=O)NC(CNC(c1cc[nH]c(=NC)c1)=O)(CC)CC 3825,c1(CC(=O)N(CC(=O)N(CCCO)CCO)CC#C)cncnc1 3826,c1(NC(=O)NC2C(OC)C2)ccc(SC2(C)CCC2)c([N+](=O)[O-])c1 3827,C1(C(=O)NC(CC(=O)NCC(CCC)C)COC)CC2CC1CC2=O 3828,C(=O)(C1=CCCN(C(=O)CCc2ccccc2Br)C1)NCc1cc(C#N)ncc1 3829,CC1CN(C(=O)CSCC(N)=O)CCC1CNC(c1ccnn1CC(F)F)=O 3830,c1(OC)cccc(C(=O)NCCC2CC(NC(=O)C(C)CS(C)=O)C2)c1C 3831,C#Cc1ccc(F)c(C(N2CCCC(CNC(C3CCCN3C)=O)C2)=O)c1 3832,N1(C(CCOC(C)=O)=O)CCC(O)(C2CCN(C(=O)C(C)=C(C)C)CC2)C1 3833,CN1CC=CCC1CCC(N1CCC(CC(=O)NC(c2ccon2)(C)C)C1)=O 3834,N1(C(c2cncc(F)c2)=O)CCCC(C2CCCN(C(c3c[nH]nc3F)=O)C2)C1 3835,N1(C(C(C)N(C(C)=O)C)=O)CC(O)(C(C)NC(=O)Cc2cnsc2)C1 3836,CC1CN(C(=O)CC2C=CCC2)C1C(=O)NCC(C)(C)CC1CC1 3837,C#Cc1ccc(C(=O)NC2CCN(C(C3NC(=O)CC3C)=O)CC2)cn1 3838,c1(NC(CNC(CNC(=O)CN2CCSCC2CO)=O)=O)ccc2ccoc2c1 3839,c1(C(N2C3CCC(NC(=O)C#CC4CCC4)C(C3)C2)=O)cnc2n1CCCCC2 3840,N1(C(C(=O)OCC)c2cccs2)CCOC(C2CC2)CC1.C(COC)S 3841,c1(C(C)(C)C)cc(C(N2CCC(C)(NC(=O)Cc3ccoc3)C2)=O)ccc1O 3842,c1(OC)c(C(=O)NCCCN(C(=O)COC)C)ncnc1C 3843,C(=O)(C(C)COC)NC(C(=O)N(CCC)CC1CC1)c1cccs1 3844,c1(OC)ccc(F)cc1CC1CCCCC1C(N1CCCC(Cn2cccn2)C1)=O 3845,C1(N(C(=O)C(O)CC)CCC)CCN(C(c2csc(C)c2Br)=O)CC1 3846,C12(CNC(C34CC(C)C3C4)=O)CC1CN(C(C1(CO)CC(C)(C)C1)=O)C2 3847,c1(C(N2CCC(F)(CNC(CCOCC#C)=O)C2)=O)cc2ccncc2s1 3848,N1(C(=O)NC(C2(N3CCOCC3)CC2)=O)CCCC(NC(C23CCCC2C3)=O)C1 3849,N1(C(C(=O)NCC)=O)CCC2(CCCN2C(=O)C(O)CC(C)(C)C)C1 3850,n1(CCC(N2CCC(O)(CNC(C3C(C)C3C)=O)CC2)=O)ccc2cccnc12 3851,CC(C)CC(F)C(=O)NC1(C2CN(C(=O)Cc3cc(-c4ccco4)on3)C2)CC1 3852,C1(NC(=O)CCc2cccnc2)CC2CC(NC(c3ccc(Cl)s3)=O)C2C1 3853,C=CCCC(C(=O)N1CCC(O)C(C)C1)NC(=O)CC1CC(C)(C)CO1 3854,C1(CNC(C(COC)O)=O)C2CCCC1N(C(c1ccc(O)c(Cl)n1)=O)C2 3855,CC1(C)OCC2CC12C(N1CCN(CC(C)(C)NC(=O)CC2=CCCC2)CC1)=O 3856,Cc1nc(CNC(C2CCOC2C(C)C)=O)sc1CNC(=O)COCC1CCC1 3857,c1(C(=O)NC(C(C(C)C)NC(c2n[nH]c(C)c2C)=O)C)ccc(Br)c(C)c1F 3858,C(=O)(CS(=O)C(F)(F)F)NC(CNC(c1c(CC)ocn1)=O)C1CC1 3859,CC#CCC(C(=O)Nc1ccc(CC)nc1)NC(=O)CCn1cncn1 3860,CCCCCC(O)C(=O)N1CCC2CC12C(=O)NCc1ncnn1CCC 3861,N1(C(C(C=CC)O)=O)CC(CNC(C2C(Cc3ccccc3)CSC2)=O)CC1(C)C 3862,C(=O)(C(C(=O)NC(C)(C)C(C)NC(c1occc1CN(C)C)=O)OC)OCC 3863,c1(C(=O)NCCC2CCC(NC(COCCOC)=O)C2)cc([N+](=O)[O-])ccc1N 3864,C1(COCC(=O)NC2CCCOC2)CCCNC12CC2 3865,C1(CC=C)(NC(C2CCS(=O)(=O)C2)=O)CCN(C(C2CCCNS2(=O)=O)=O)CC1 3866,Cc1cc(C)c(C(=O)NCc2ccccc2C)c(Cl)n1.N12CCC(C1)NC2=O 3867,CC1(C)OC(=O)NC1C(=O)NCC1CC(F)CN1C(=O)CC1(C)CC1(Cl)Cl 3868,c1(C(C(=O)OC)NC(=O)C(F)CC(C)C)cccc(Br)c1OC 3869,Cc1onc(CO)c1C(=O)NCCCN(C(=O)C=C(Cl)Cl)CCO 3870,N1(c2cc(COC)ncn2)CCC(C)C(NC(c2ccc3c(c2)CC3)=O)C1 3871,CC(C)C(C(=O)NCC1(NC(C2OCCO2)=O)CCOC1)c1ccn(C)n1 3872,C1(C(C)C(=O)NCC(=O)N(CCCO)C2CC2)CCC(=O)N1 3873,N1(C(CC2CN(C(c3c(CC)ccs3)=O)C2)=O)CCCCC1C1(COC)CC1 3874,CC(C)C(CCS(C)(=O)=O)NCC(=C1CCNCC1)F 3875,c1(OCC(=O)NCCCN(C(CC(=C=C)C)=O)C)ccc(C)cc1CC 3876,C1(C(N2C(C)CC2NC(c2cc(O)n(C)n2)=O)=O)CCc2ccccc2C1 3877,C12(CNC(c3ccc(C(C)C)o3)=O)CC(CN1C(C1CCCCO1)=O)C2 3878,C1(CNC(COCCC)=O)CC2(CC2)CN1C(c1cn(C2CCOC2)cn1)=O 3879,Cc1ccccc1N(c1nc(-c2cnn(C)c2)cs1)C1(CC2CC2(Br)Br)CC1(C)C 3880,c1(C(=O)NC(C2OCCN(C(c3scc(C)c3Cl)=O)C2)C)cc(O)nc(Cl)c1 3881,C=CC(C)(CC)C(=O)OCC.c12ccc(nc1O)C(=O)N1CCC(C1)NC2=O 3882,c1(NC(C2CC(F)CN2C(c2ccc(C3CC3)cc2)=O)=O)ccnc(C2CC2)c1 3883,C12(CNC(c3cc(CC)no3)=O)CCC1CCN2C(C1CCC(C)CC1)=O 3884,C(=O)(CCCCN=[N+]=[N-])N1C(C(=O)NC(CC=C)C(=O)OC)CC1C 3885,C1(CCC)(C(=O)NCC(c2cccc(Cl)c2)NC(c2ccco2)=O)CCNC1=O 3886,Nc1cccnc1C(=O)NCC1CCCCC1C(=O)NCc1ncc(CO)[nH]1 3887,C(=O)(CC(C)C(F)F)NC1C(C(NOC(CC)CC)=O)CC1 3888,C=CCC(CNC(C1(CO)CCCC1)=O)NC(C1(c2ccno2)CCC1)=O 3889,C1(NC=O)CN(C(C2CCCN2C=O)=O)CCC1Cc1nn(C)nc1Br 3890,C(CC(C(=O)NCCN(C(c1coc(C)c1)=O)Cc1ccccc1)OC)OC 3891,c1(C(=O)NCC2(C#N)CCC2)c(NC(C2CC(O)C2)=O)sc2c1CCCC2 3892,C=CCC(C)(CO)CN=c1ccnc(N2CCC(CN(C)CC3CC3)C2)[nH]1 3893,c1(CC)cccc(C(=O)N(CCNC(=O)CCc2ccn(C)n2)C2CC2)c1 3894,C#CC1CCCN(C(=O)C(=O)NCC2COC3(CCCC3)C2)CC1 3895,N1(C(C(COCC)C)=O)CCSCC1CCNC(=O)Cc1ccnn1C1CCC1 3896,C1(NC(C2(OC)CC2)=O)CC(O)CN(C(c2cnc(C3CCC3)s2)=O)C1 3897,C1(CN(C(=O)CNC(=O)NC2CC2)C)CCCCN1C(C1CNC(=O)N1C)=O 3898,Cc1nsc(NC(C2CCN(C(=O)CCC3CC3(C)C)CC2)C)c1C#N 3899,N1(C(C2CN(C)CC2C(F)(F)F)=O)CCCC(NC(C2(CO)CCC2)=O)CC1 3900,N1(CC(C)NC(=O)CS(=O)(=O)N(C)C)CCN(C(C2C=CCS2)=O)CC1 3901,C1(N(C(C=C(CC)C)=O)C)CCCCN(C(c2cn(C)c(O)n2)=O)C1 3902,Cc1c(F)cc(CN2CCN(C(c3ccc(F)cn3)=O)C(C)C2)cc1F 3903,N1(C(COC(C)C)=O)CCC2CCCN(C(c3c[nH]c4ccc(Cl)cc34)=O)C2C1 3904,C1(CN(C)C(C2CCCN(C(N)=O)C2)=O)COCCN1C(=O)CC1CSC1 3905,c1(OC)cc(CN(CCO)C(=O)NCC23CC(CN2)C3)ccc1O 3906,c1(C(N(CCN(C(C(C)OCC)=O)C)C)=O)cc(Cl)cnn1 3907,CC1=CCC(C(=O)NCCCCN(C(=O)CCSc2nccn2C)C)CC1 3908,C1(COCC)CCCN(C(=O)NC2CC2c2nc(OC)no2)CC1 3909,c1(N2CC(CC(=O)Nc3ccsc3Cl)C2)ncnc2cc(Br)sc12 3910,N1(C(C=CC(C)C)=O)CCC(N(C(=O)CSC(F)F)C2CC2)C(O)C1 3911,C(C(C)(C(=O)NOC1CCCC1)NC(=O)CCc1cc(C)[nH]n1)SC 3912,S(=O)(=O)(c1ccccc1C(=O)N(C)CCNC(=O)CC1(O)CCC1)NCC=C 3913,C(=O)(CCCS(C)(=O)=O)NC(C)C(C)(C)NC(c1nccc2cc[nH]c12)=O 3914,C1(C(=O)NCC(C)CN(C(=O)COCC2CCCO2)C)CCS(=O)(=O)C1(C)C 3915,C#CC1CN(C(=O)C(CCOC)NC(c2cnns2)=O)CCO1 3916,N1(C(C2(CC#C)CCOC2)=O)CCC2(CC(NC(=O)C(C)(C)CF)C2)C1 3917,c1(OC)cc(F)c(NC(=O)C(=O)NCC2CNCC2C)c(F)c1 3918,c1(COC)ccccc1C(=O)NC1CCCC1n1cc(CN2CCNC2=O)nn1 3919,C1(C(N2C(CNC(CC(CC)OC)=O)CC2)=O)CNc2ccnn2C1 3920,C#CCC(CC#C)C(=O)NCC1CCCC(NC(=O)Cc2cc(C3CC3)on2)C1 3921,C1(C(=O)NC(CNC(C(C)c2ccsc2)=O)C2CC2)Cc2nccn2C1 3922,C1(CNC(C2(c3cc(C)no3)CC2)=O)CCCN(C(=O)CP(C)(C)=O)CC1 3923,Cc1nnc2ccc(C(N3CCCCC(NC(=O)C(=O)N(C)C)C3)=O)cn12 3924,Cc1c(F)ccc(C(=O)NCC2CC2CNC(C2CCS2(=O)=O)=O)c1Cl 3925,c1(OC(CNCC(C)CO)(C)C)cccc([N+](=O)[O-])c1 3926,CCC(O)C(C)C(=O)N1CC(CNC(C2CCS(=O)CC2)=O)C(C)(C)C1 3927,C1(CC(C)C)C(=O)NCCN1C(=O)NCCc1ccc(F)cc1Br 3928,C1(CNC(C#CC(C)C)=O)CC2(CCOCC2)CN1C(=O)CC1CC(=O)NC1=O 3929,N1(C(C(C)OCCOC)=O)CCN(C(c2ccc(=N)[nH]n2)=O)CCC1C 3930,c1(C(=O)NC2CC(NC(c3ccc(C)n3C)=O)C2)cccn(C2CC2)c1=O 3931,O=C(CCCNC(C1CCCCC1)=O)NCC=CCNC(C1C=CCS1)=O 3932,C1(C(=O)NCC(c2ccccn2)CO)CCCN(Cc2ccccc2)C1=O 3933,C(C)(CC(C)(C)C)NC(C(=O)Nc1c(C)csc1)=O 3934,CC(C)(CC#N)C(=O)N1CCCC(NC(c2ccc(F)c(CO)c2)=O)C1 3935,c1(CNC(C2C(NC(c3ccc(C#C)o3)=O)CCOC2)=O)cc(O)ccc1C 3936,CCC(CC(=O)NCCNC(C1CCCN(C(c2cnc(S)n2C)=O)C1)=O)OC 3937,C1(NC(c2c(C)nc(CO)s2)=O)CN(C(=O)C2=CCCOC2)CCC1C(F)(F)F 3938,Cn1ncc2c1CCC(C(N1CCN(Cc3nc(-c4cccs4)no3)CC1)=O)C2 3939,N1(C(C(c2ccncc2)C)=O)CCC(O)(CCNC(=O)Cc2n[nH]c(=N)s2)CC1 3940,CC(N=c1[nH]nc(C(F)F)o1)c1ccn(-c2ccccc2F)n1 3941,O=C(CN=c1cc(F)nc[nH]1)NC1CCN2CCCC12 3942,C1(NC(C(C)(C)SC)=O)CCCCCN(C(c2c[nH]nc2C2CCOCC2)=O)C1 3943,C=Cc1cc(C(N2CCC(NC(COCCCCC3CC3C)=O)C2)=O)cc(F)c1 3944,c1(C(N2CC(CCC)N(C(c3ns[nH]c3=O)=O)CC2)=O)c(F)ccc(F)c1F 3945,c1(OC)ccc(F)c(CC(=O)N(C2CN(C(c3ncccn3)=O)CC2(C)C)C)c1 3946,N1(C(C(C)(C)CF)=O)CCCN(C(=O)CC23CCC(CC2)OC3)C(CO)C1 3947,C1(NC(=O)CC(c2ccc(F)cc2)C2CC2)CCN(C(=O)CSC(F)F)CC1O 3948,C=CCCC(O)CNC(=O)CC(O)CNC(c1csc(C)c1C)=O 3949,C1(NC(C(Cn2cncn2)NC(COCCCCC)=O)=O)CCCC2(CCC2)C1 3950,c1(C2(C(N3CCC(NC(c4cnc(C5CC5)o4)=O)C3)=O)CC2)ccc(F)cc1 3951,C1(NC(C2(C)CNC(=O)N2)=O)CCN2CCCC2C1 3952,N1(C(C(C)CC2CCC2)=O)CCC(CCCNC(c2ncc[nH]c2=O)=O)CC1 3953,C1(C)(C(=O)NCC2(CN(C(C(C)CC3CCCC3)=O)C)CC2)CC=CCC1 3954,N1(C(c2ccc(N(C)C)nn2)=O)CC=C(CNC(c2cnn(C3CC3)c2)=O)CC1 3955,CC1(C)CC(NC(c2csc3cncn23)=O)CN1C(c1ccncc1Cl)=O 3956,c1(NC(CC(C2CC2)NC(CC(C=C)C)=O)=O)cc(O)c(C)cc1C 3957,CC1C(O)CCCN1C(c1ccc(CNC(=O)CCN2CCCCC2)s1)=O 3958,Cc1[nH]nc(C(F)F)c1C(=O)NC1CCC(CNC(C2CCC(F)C2)=O)CC1 3959,C(=O)(CC(C)(C)CNC(C1CC1(C)C)=O)NC1(C(=O)OC)CC1 3960,c1(OC)cc(C(N2CCC(O)(CNC(=O)Cc3cccc(Cl)c3)C2)=O)ccn1 3961,N1(C(C(=O)NC(C(=O)OC)CC(C)C)C2CC2(Br)Br)CCC2C(O)CCCC2C1 3962,CC(CN(C)C)CCC(=O)NC1(C(=O)NC2(CO)CC3CCC2C3)CCOCC1 3963,CCC(CCC(=O)NC1CCCN(C)C1)NC(=O)C(C)(O)CCN(C)C 3964,N1(Cc2scc(CC)n2)C(=O)CN(CCN2CCC2CC)C1=O 3965,C12(C(N3CC4C(NC(C5C(OC)C5)=O)(C4)C3)=O)C3C4C1C1C2C3C41CO 3966,c1(C2CC(C(C)=NO)C2N(CCOc2ccccc2)C)nc2cc(F)cc(F)c2o1 3967,N1(C(C=CC(=O)NC2CC2)=O)CCCC(C2CCN(C(=O)C(O)c3ccsc3)C2)C1 3968,C(=O)(C(CC)(CC)C(=O)OC(C)(C)C)NC(CN(C(CCC(=C)Br)=O)CC)C 3969,c1(C(=O)NC2C3CC(NC(c4c(NC)snc4C)=O)CC32)ccc(O)nc1Cl 3970,c1(CC)noc2ncc(C(=O)NC(C)CNC(c3ccccc3CC#N)=O)cc12 3971,C(N=c1[nH]cnc2cc(F)c(F)cc12)C1N(C(C2(C)CCOCC2)=O)CCCC1 3972,Cc1nccn1CCC(=O)NCC1CCC1NC1(C2CCCCO2)CC1.C1=CC=C1 3973,c1(C(=O)NC2CCC(NC(C3C(C4C(C)C4)C3)=O)CC2)ccc2c(c1)CCN2C 3974,C#CCCN(C)N1CCCC(Cc2ccc(Cl)c(Cl)c2)C1 3975,CCCCCCCCC(=O)NC(C)CCCNC(=O)C1=COCCO1 3976,Cc1ccc(SCCC(=O)NCC(C)(C2CCC2)NC(c2cn(C)cn2)=O)cc1 3977,N1(C(CC(CC)C2CCC2)=O)CCOCC(F)(CNC(=O)Cn2ccnn2)C1 3978,C12(CC)CN(C(=O)Cc3nnc(C)s3)C(CNC(C3(C)CC3(F)F)=O)(C1)C2 3979,n1(CC(=O)OCC)nccc1C(=O)N(CC(C)NC(=O)C(O)C1CC1)CC 3980,c1(SC)ccccc1C(=O)NC1CCN(C(=O)C(C)C(F)F)C1C 3981,Cc1cnc2n1CCCC2C(=O)Nc1cc(-c2ccccc2)nn1C(C)(C)C 3982,N1(Cc2c(C)cc(Cl)nc2)CCCN(C(=O)C=Cc2cccc(O)c2)C(C)C1 3983,C#Cc1ccc(C)c(CNC(=O)NCCN(CCC)C(=O)OC(C)(C)C)c1 3984,C(C)(N=c1[nH]c(N2CCC(C(C)C)C2)nc2ccccc12)c1cc(C)cc(Br)c1 3985,C(CCCCCN=C(NCCS(=O)C(C)(C)C)N(C)Cc1ccc(F)c(Cl)c1)SC 3986,c1(C(=O)NC(CCOC)CNC(C2(SC)CC(CO)C2)=O)ncc(C)cc1OC 3987,N1(C(c2c(O)ccc(C)c2)=O)C2CCC(C(N3CCC(O)(CO)C3)=O)C1CC2 3988,N(C1CCCc2sccc21)C(N1CC(CC2CCOC2)C1)=O 3989,C(=O)(C(CC(F)F)NC(C1CC(=O)C1)=O)NC1(C(=O)OCC)CC1 3990,c1(C(=O)NCCCCCCNC(c2sc(C)c(O)n2)=O)cc(Cl)ccc1F 3991,N1(CC)Cc2cc(CNC(c3cc4cccc(F)c4[nH]3)C)ccc2C1=O 3992,C1(CNC(CC(C(CC)C)O)=O)CC2(CCN(C(=O)Cc3cnc[nH]3)CC2)C1 3993,C(=O)(C(CCSC)NC(=O)C(Cl)Cl)NCC(=O)OC 3994,N1(C(CN(C(=O)OC(C)(C)C)CC)=O)CCC(CC(C)NC(=O)C(F)CC)CC1 3995,CCCC(C(=O)N1CC(NC(=O)COCC(F)(F)F)C1)OC.C12CCN(C1)C2 3996,C1(C)(C(C(CC=C)Oc2nn(C)cc2-c2cn(C3CCCCC3N)nn2)=O)CC(O)CN1C 3997,CCC(CC1CCCC1)C(=O)NC(C)CC1CN(C(c2sc(CO)nc2C)=O)C1 3998,c1(C(=O)NC2C(NC(c3cn(C)nc3)=O)CCCC2)cnc2[nH]cnc2c1 3999,C1(NC(=O)CCc2cnccn2)CCCCN(C(C2CCC(F)(F)CO2)=O)C1 4000,C1(NC(c2ccccc2)=O)CN(C(=O)CC2CNCC3(CCC3)O2)C2(CCC2)C1 4001,CCCC(C(=O)N(C1CCN(C(c2ccc3nn[nH]c3n2)=O)C1)CC)S(N)(=O)=O 4002,CC(F)(F)C(C)(C)C(=O)N1CC(CCCCNC(c2ccc(C(N)=O)o2)=O)C1 4003,c1(C(=O)NC2C(C)CN(C(c3ncccc3O)=O)CC2)nnn2c1CCCC2 4004,C1(C(=O)NCc2ncc(C)s2)CC12CCN(C(c1n[nH]c(C)c1Br)=O)CC2 4005,O=C1CCC(C(=O)NCCC2CCCCN2C(c2ccsc2C(F)F)=O)CN1 4006,c1(C(N(CCNC(C2C(CC)CCO2)=O)CC)=O)[nH]c2ccc(F)cc2c1C 4007,CCCC(C(=O)NC1CCCCC1NC(c1cc(F)c(CO)c(F)c1)=O)C(C)C 4008,c1(C(N2C(CNC(c3ccns3)=O)CC(OC)C2)=O)cc(Cl)c(F)cc1O 4009,Cc1ccc(OCCC(N2CC(NC(=O)CCC(C)C#N)C3(CC3)C2)=O)cc1C 4010,CCCC(C(=O)NC1CN(S(=O)(=O)CC)C1)c1ccc(Cl)cc1 4011,c1(OC)cncc(Br)c1C(=O)NC1CC1CNC(=O)CC1CCCCC1 4012,CC(C)(C)CC(O)CC(=O)NC1CCCC1C(=O)NC(CCO)C(F)(F)F 4013,CCCC(C(=O)NCC1CCN1C(=O)CCC12CCC(CC1)C2)OC 4014,c1(C(C)OC)nc(C(=O)NC(CNC(c2cn(CCF)nn2)=O)CO)co1 4015,c1(C(N(C2CCCN(C(C(CC)O)=O)C2)C)=O)cc(O)cc(N)c1Cl 4016,N1(C(C2C(OC)CC2)=O)CCN(C(=O)COCCC(C)C)CC1C 4017,c1(CC(=O)NC2C(NC(c3cc(C)on3)=O)CCC2)c(C)[nH]c2ccnn2c1=O 4018,CCCCC(CC)CC(=O)N1CC=CCC1C(N1CC(C2=NOCC2)C1)=O 4019,C1(C(N2C(C3(NC(C4(CCCC)CC4)=O)CC3)CCC2)=O)CC(O)CN1C(C)=O 4020,Cc1nnc(O)c(C(=O)NCCC2CSCCN2c2ncc(Br)cn2)c1C 4021,c1(C(=O)NCC2(N3CCOCC3)CCCOC2)nc2ccc(F)cc2s1 4022,c1(CC(N2CC(F)(CNC(C3CC4(CCCO4)C3)=O)C2)=O)n[nH]c2c1CCCC2 4023,c1(CNC(C2CCCN(C(=O)COC3CCCCC3)C2)=O)cc(Br)ncc1F 4024,c1(C(N(C2C3CN(C(C(C4CCOCC4)OC)=O)CC32)C)=O)ccc(Cl)c(F)c1 4025,N1(C(c2ccc(F)c(Cl)c2)=O)CC2CCC1CN2C(C1SC2C=CC1CC2)=O 4026,N1(C(C2C(C(=O)OCC)C2)=O)CSCC1C(=O)NCC=Cc1ccco1 4027,C1(C(=O)NCCCC(C)NC(C(C)NS(C)(=O)=O)=O)CC2(C1)CC2F 4028,Cc1ccc2ccccc2c1CNC(c1sc(CC2CC2)nc1C)C1CC1 4029,c1(N2CCC(N(CC#C)C(c3cscc3C)=O)CC2)ncnc2cc(Br)sc12 4030,C1(OCC)COCCC1NC(=O)CC(C)NC(=O)C(C(C)C)NC=O 4031,C1(CC(=O)NCC(C2CC2)NC(C2CC2C2CCCC2)=O)CCCCC1(F)F 4032,C1(N(C(c2ccoc2C2CC2)=O)CCO)C=CCN(C(=O)COCC(F)(F)F)C1 4033,C(=O)(C(O)CC(N)=O)NC(C)CCC(=O)N(C)Cc1cccc(O)c1 4034,CC1CCC2(CC1)CCC(CNC(=O)NC(c1cccc(S(N)(=O)=O)c1)CO)O2 4035,c1(C(=O)NCC2CCC(NC(C(CC)(C)CO)=O)C2)n[nH]c2cccc(OC)c12 4036,C1(C(=O)NC(CNC(C(CC)=CC)=O)(C)C2CC2)CCc2cn(C)nc2C1 4037,C1(NC(Cn2ccc(C)n2)=O)CCN(C(C2CC(n3cnnc3)C2)=O)CC1F 4038,C(=O)(CCC(=O)N(C)C)N(C(C)C)C1CC1.C12COC(C1)CNC2=O 4039,C1(C(F)(F)F)(NC(C(C)NC(=O)NC2CC2)=O)CN(C(C2(C#N)CC2CO)=O)C1 4040,c1(NC(c2cn(CCNC(CNC(=O)OC)=O)nn2)=O)onc2ccccc12 4041,C(CCC(C(=O)Nc1ccccc1)N(C1CCN(C)CC1C)C)=C(C)C 4042,C12(NC(c3csnn3)=O)CCCC1CN(C(=O)C=Cc1ccc[nH]1)C2 4043,C(=O)(CC(F)(F)C(F)F)N1CCCN(C(C(c2ccc(OC)cc2)C)=O)CC1 4044,N1(C(CCC=C)=O)CCC(CO)(CNC(=O)CCN(C)C(C)=O)CC1 4045,c1(OC)noc(C)c1C(N1CCC(C(C)C(=O)NCC2(C)CCCCC2)C1)=O 4046,N1(C(C(C2CN(C(C(C=CC)O)=O)C2)O)=O)CC2(C1)CC2(F)F 4047,C(=O)(C(CC(C)C)NC(c1cnc(Cl)n1C)=O)NCC1CC(CC)C1 4048,N1(C(C(CC=C)CC)=O)CCC(C2(NC(=O)COC3CC(F)(F)C3)CC2)CC1 4049,c1(C(N(C(C)CCNC(C2CCOC(C)C2)=O)C)=O)cc2c(cc1F)NCCC2 4050,c1(C(=O)NCC2C=CCN2C(C2CCCC2(F)F)=O)ccc2c(n1)OCCO2 4051,C1(O)(CN(C(c2n(CC)ccc2)=O)C)CCCN(C(=O)C=CC2CCCO2)C1 4052,C1(NC(C(C)OCc2ccccc2)=O)CN(C(=O)C(=O)Nc2ncc[nH]2)CC1O 4053,c1(C(N(CCCCN(C(c2nccc(CC)c2)=O)C)C)=O)nc[nH]c2ncnc1-2 4054,c1(OC)ccc(Cl)c(C(=O)NCC23CC2CN(C(=O)CC(C)(C)OC)C3)c1 4055,N1(CC#CCOC)CCC2(CCN(C(c3csnc3OC)=O)CC2)C1 4056,c1(C(N2CCCC(N(CCO)C(C3C=CCCC3)=O)C2)=O)cnccc1Cl 4057,C1(CNC(c2n(CC)ccn2)=O)CCN(C(C2CSC(C)=N2)=O)C12CCC2 4058,N12CCN(C(=O)CSCC(N)=O)C(C1)C2=O.C1(CC#C)(OC)CCCOC1 4059,C(C(CC(F)(F)F)NC(=O)Cc1cc(F)cc(F)c1)NC(C(CC)NC(C)=O)=O 4060,C1(NC(CCCC=C)=O)CCCC(NC(C2CC(=O)C2C(C)(C)C)=O)CC1 4061,C(CCC(C)C)(C(=O)NCCc1nccnc1C)NC(c1c(CC)c[nH]n1)=O 4062,C(=O)(C(C)(O)C(F)(F)F)NC(CC#C)C(=O)Nc1ccc(C)c(Cl)c1 4063,c1(C(N2CCC(N(C)C)C2)C(=O)NCc2nnn(C)n2)nc2ccc(F)cc2s1 4064,Cc1ccc(C)c(CN2CCC(C)(C(=O)NC3CCN(S(C)(=O)=O)C3)C2)c1 4065,C1(C(N(C)CCN(C(=O)C(C2CCCO2)C2CC2)C)=O)CCCC2C1C2(F)F 4066,N1(Cc2onc(C(C)OC)n2)CCCC(CO)(NC(c2cn(C)nn2)=O)C1 4067,C(=O)(C(CCC1CCC1)NC(=O)CC(F)(F)F)N(C1CCCC1O)C 4068,C(N=c1ncc(C(C)(C)O)c[nH]1)C1CCC(NC(C2(N(C)C)CCCC2)=O)C1 4069,N1(C(c2c(N)cc(F)cn2)=O)CC=C(CC(=O)NC2CC2O)CC1 4070,C1(C(=O)NC2CN(C(c3c(CCC)occ3)=O)C(CO)C2)CC2(CC(OC)C2)C1 4071,C(CCC(C)(C)CO)NC(C#CCNC(C1C(C)CC(=O)N1)=O)=O 4072,C1(NC(c2c(CC)cno2)=O)CS(=O)(=O)CC1NC(c1cnc(C(C)C)nc1)=O 4073,C(C(C)(CO)CO)NC(C=CC(C)(C)NC(C1COC(=O)C1)=O)=O 4074,C1(C(N(C(C)C)CCF)=O)CN(C(=O)Cn2cnnn2)CC1(F)F 4075,c1(NC2CC(C(=O)Nc3nc(C)c(C#N)nc3)C2)ncnc2sc(Br)cc12 4076,c1cc(F)cc(Cl)c1.CC(C)(C)CC(=O)NCC(=O)NCCNC(=O)CN1CCCC1 4077,N1(C(C(CCCOC)C)=O)CC2CCC(NC(=O)CC(O)C3CC3)CC2C1 4078,c1(CCNC(=O)NCC2CCN(C)C(=O)C2)cccc2ncccc12 4079,N1(C(C(N2CCCC(C)C2)=O)=O)CCOCC(F)(CNC(c2ccsc2)=O)C1 4080,c1(C(C(=O)N(CC(CC)NC(=O)CCc2ccc(C)s2)CC)C)ccccc1C 4081,C1(F)(C(=O)NCCCCNC(=O)CCC2NC(=O)NC2=O)CCS(=O)(=O)C1 4082,C1(C(=O)NC(C)CNC(C2CCCC2)=O)CCCSC1 4083,N1(C(C=CC)=O)CC2CC(NC(=O)C(C3CCC3)OC)CC1C2 4084,N1(C(c2nc(CNC(C(C(C)C)OC)=O)oc2C)=O)CC(CO)CC12CCC2 4085,c1(C(C)C)cc(C(=O)N(C)CC2(NC(c3cc(Cl)no3)=O)CC2)ccc1F 4086,ClC1=CCCC12CCCN(CCOc1ccccc1Cl)C2 4087,N1(C(CN2C(C)CCC2C)=O)CC2(CCC(CNC(=O)C(C)N3CCCC3)O2)C1 4088,C1(C(N2CC(C)(NC(C(C)=CC)=O)C2)=O)CCCOC1c1cn(C)nn1 4089,C12(NC(=O)Cc3ccoc3)CCCC1N(c1cc(Cl)nc(C(F)(F)F)n1)CC2 4090,O(N1CCC(N=c2cccc(S(=O)(=O)N3CC(C)OC(C)C3)[nH]2)CC1)CC 4091,c1(CC(C)C(N2CCCCC(NC(C3(O)CCC3)=O)C2)=O)ccc(Cl)cc1Cl 4092,C1(NCC2CCCC(CNC(C(n3cc(CO)nn3)C)=O)C2)CCC(O)CN1C 4093,C12(COC)CC(NC(N3CCCC(C(C)(C)C(=O)O)C3)=O)(CO1)C2 4094,C1(C(N(CCCOCCNC(CC2CC(C)C2)=O)C)=O)OCCC1(C)C 4095,c1(C(N2CC3(C(=O)OC)CC(COC)(C2)C3)=O)cnc2c(C)nccn12 4096,Cc1cc(CNc2cc(F)cnn2)cc(C(F)F)c1 4097,C1(CCNC(C2N(C(CC)=O)CSC2)=O)COCCN1C(=O)COC1CC1 4098,N1(C(C2CCC(CNC(C3CCN(CC)C3)=O)C2)=O)C2CSCC1C2 4099,Cc1cc2c(Br)cccc2c(NCC2CCCCC2N2CCOCC2)n1 4100,c1(OC)ncc(NC(=O)CC(CNC(=O)C(N2CCNC2=O)C)OC)cn1 4101,Cc1cc(Br)cnc1C(=O)NC(CNC(=O)COC(F)(F)F)C(C)(C)C 4102,c1(C(=O)NC2CC(CNC(c3cc(CCOC)on3)=O)C2)nc(Cl)c(Cl)s1 4103,CC1=C(C)CC(C)(C(=O)N(CCNC(=O)CC#N)C(C)C)CC1 4104,c1(C(N(CCN(C(=O)CC(=O)NC2CC2)CC)CC)=O)ncsc1C 4105,c1(NCC(=C)C2CCOCC2)ccc(S(=O)(=O)NC2COC3(CCCC3)C2)cn1 4106,Cc1nc(N2CCC3(NC(=O)C4=NNC(=O)CC4)CCCC23)c2ccsc2n1 4107,C1(C)(C(=O)NC(C2OCCN(C(CCCOC)=O)C2)C)CC(C(C)(C)C)=NO1 4108,C1(C(N(C2CCCC(NC(C(C)OCCC=C)=O)C2)C)=O)C2CC3C(C2=O)C13 4109,N1(C(c2nc(C(C)NC(CSCC#C)=O)oc2)=O)CCC2(CCCN2C)C1 4110,c1(CNC(CSCC)=O)ccccc1CNC(c1ccsc1CC)=O 4111,Cn1cnc(C(=O)NC2(C(=O)NC3CN4CCC3CC4)CC2)cc1=O 4112,c1(C(=O)NCC2CCCC(NC(C(CC)(C)CO)=O)C2)ccc2cnoc2c1 4113,Cc1ncc(N)cc1C(=O)N(CC(C)NC(=O)C(C)NC(c1ccco1)=O)CC 4114,Cc1cnc(CNC(=O)CCCC2CN(C(=O)OC(C)(C)C)C2)o1 4115,Cc1nc(N2CC(F)(C(=O)Nc3ncc(F)c(Cl)n3)C2)c2ccccc2n1 4116,n1(CC)nccc1C=CC(=O)NC1C2CC(NC(=O)CCCc3ncco3)CC12 4117,c1(OC2CCN(C(C3CC3C(F)(F)F)=O)C2)cccc(F)c1 4118,c1(C(=O)NC2C(C(=O)Nc3ccc(OC)cc3C)CCC2)cn2ncccc2n1 4119,C1(C(=O)OC)CCOC1C(=O)NCCCNC(=O)CC1(C)CCC1 4120,[N-]=[N+]=NC1CN(C(C2(F)CCN(C(c3n[nH]c(O)n3)=O)CC2)=O)CC1O 4121,Cc1ccc(C(N2C3CCC2C(NC(C2CC4CCC2C4)=O)C3)=O)cc1C 4122,C1(CCC(=O)N(CC=C)CCC)CCCN(C(=O)C(C)NC(C)=O)C1 4123,C(=O)(C1CC=Cc2ccccc21)N1C2CN(C(C#CC3(C)COC3)=O)C(C2)CC1 4124,Cc1nc(CNC(=O)CCc2cccn2C)oc1C(=O)NC(C)Cn1cnnc1 4125,N1(C(C2CC(C(C)C)OCC2)=O)CCC(F)(CNC(C2C(C)C2C)=O)CC1 4126,c1(OC)cc(OC)cc(C(N2CC(NC(c3cc(C#N)oc3C)=O)C(C)C2)=O)c1 4127,C1(NC(C23CC(C)C2C3)C)CCN(CC2CCCO2)CC1 4128,Cc1ccc2c(C(=O)NCC3CC(NC(=O)C(=O)N(C)C)C3(C)C)csc2c1 4129,C(=O)(C#CC1(C)CCCO1)N1C(C(=O)NC2(CC=C)CCC2)(COC)C=CC1 4130,C=CCCC(C(=O)N1CCCC(O)(CC)C1)NC(=O)CSCCOC 4131,C1(F)(C(=O)NCC(C2CCOC2)NC(c2ccns2)=O)C2CCCC12 4132,C1(C(C(=O)OCC)CC)CCN(c2nnnn2CC2CC2C2CC2)CC1 4133,Cc1cocc1C(=O)NC1CCCC1CC(=O)NCCC1(C)CC1(F)F 4134,CCCS(=O)(=O)CC(=O)N1CCN(C(c2ccc(N(C)C)cc2)=O)C(C)CC1 4135,Cc1nc(C(N2CC(OCC(N3CC(C)CC3C)=O)C2)=O)c(C)o1 4136,CC1CC(C(N2CC(NC(c3c(Cl)noc3C)=O)C2)=O)CC(C)C1 4137,N1(C(c2c(C)cc[nH]2)=O)CCC2(CC1)CC2NC(c1cc(I)ccc1C)=O 4138,N1(C(c2ccc(F)nc2)=O)CC2(CCN(Cc3ccc(-n4cccc4)cc3)C2)C1 4139,c1(CC)c(C(N2CCCC(NC(=O)C(C)c3ccsn3)C2)=O)cnn1C(C)(C)C 4140,C(=O)(C(CO)C(C)C)NC(C1CCN(C(CCC(=O)NCCC)=O)C1)(C)C 4141,N1(C(C2ON=C(CC)C2)=O)CC2CC1CC2NC(=O)Cn1ccnc1 4142,c1(C(N(C)CC2(NC(C3N(C(C)C)CCC3)=O)CC2)=O)nc2ccccc2s1 4143,C12(C(=O)NC3C(C(C)C)C3)CCCC1CCN2C(=O)CCCN(C)C 4144,c12ccc3c(n[nH]c3c1)NC2=O.C1(NC(NCC)=S)COCC1O 4145,C1(CNC(Cc2c(C)scc2)=O)CC2CCC1N2C(C1(C(N)=O)CC1)=O 4146,c1(NC(C2CC23CCN(C(=O)Nc2cccc(F)c2)C3)=O)ccnc2c1CCO2 4147,C1(CN(C(=O)CN2CC(C)(C)C2)CC)CCN(C(=O)C(C)CC#N)CC1 4148,C=C=CCCC(=O)NCC1CN(C(=O)C=C(CCC)CCC)C1 4149,Cc1ncc(Br)c(C(N2CCC(NC(=O)C3=CCCCO3)C(O)C2)=O)n1 4150,C1(S(C)(=O)=O)(C(=O)OC)CC(NCC2CC2Cl)C1 4151,C1(C(=O)NC2CC3CC4C(C3)C24)(CC)CCCN(C(=O)COC2CCC2)C1 4152,C1(NC(CCC#CC)=O)CCC2(CC1)CC2NC(C1CC(=O)N(C)C(=O)N1)=O 4153,c1(C(N2CC=CC(NC(=O)CC3CCC(F)(F)CC3)C2)=O)ccc2n[nH]cc2c1 4154,CC1CCC(NC(=O)Cc2cc(O)cc(Br)c2)CN1C(c1cccnc1O)=O 4155,S(=O)(=O)(c1cccc(=NCCc2cnccn2)[nH]1)N(C(C)CC#N)C 4156,C(CCCCCN=[N+]=[N-])NC(CCc1cccc(OC)c1)=O 4157,CC1(C)CN(C(=O)CN2CCOC2=O)CCC1C(N1CCCN(CCO)CC1)=O 4158,N1(C(C(C)CN(C)C(C2CCCCC2O)=O)=O)CCOC2(CCC2)CC1 4159,C1(NC(c2c(C)sc(-c3ccco3)n2)=O)CN(C(C2CCC2C)=O)CC12CCC2 4160,c1(C(=O)NCCCNC(c2nnn(C)c2C(F)(F)F)=O)ccc(C2CC2)nc1O 4161,Cc1cc(C(=O)NC2(CO)CCN(C(C3OCCN(C)C3=O)=O)C2)nnc1C 4162,C1(NC(C2(C)CC(C)C2)=O)CN(C(=O)CCc2ccc(F)cc2F)CCC1CO 4163,N1(C(CC2CCN(C)C2)=O)CC2CCC(CNC(c3cnc[nH]3)=O)C2C1 4164,O=C(C1CCCn2ccnc21)N1CCCC1c1ccccc1 4165,Cc1c(CN2CCCC(C(=O)Nc3ncc(Br)nn3)C2)cccc1Cl 4166,c1(C(C)=O)[nH]ccc1C(=O)NCC1(NC(=O)CN2CCC(C)C2)CCC1 4167,C(=O)(C1=CC2(CCOCC2)C1)N1C(CCCNC(=O)CC2CCC2)CCC1 4168,c1(CC)ccc(O)c(NC(C2(CNC(=O)C(C)OCCC(C)C)CCC2)=O)c1 4169,C1(C(N2CCN(C(CC3CC(=O)C3)=O)C(CO)C2)=O)CC2C=CCC(C1)C2 4170,N1(C(c2ccc(C(C)O)cc2)=O)CCCCC(NC(C2(n3cnnn3)CC2)=O)C1 4171,C1(CC(=O)NCC2(NC(CC3(NC(C)=O)CC3)=O)CCOC2)C(=O)NN=C1C 4172,c1(CCC)nc(C(=O)N(C2CCN(C(C3(C)CCCO3)=O)C2)CC)cs1 4173,c1(OC)cccc(OCCC(=O)NCCC2COCCN2C(=O)C(F)C(C)C)c1 4174,C1(O)(CCNC(c2cn(C3CCOCC3)nn2)=O)CN(C(C2CCC2(F)F)=O)C1 4175,C(=O)(C1=CS(=O)CCC1)Nc1ccccc1C(F)(F)F.NC(=O)CCC1CN1 4176,c1(NC(C2(F)CCN(C(c3ccc(F)c(F)c3)=O)C2)=O)nc2ccc(Cl)cc2[nH]1 4177,n1(CCNC(C=C(CCC)C)=O)cc(CNC(=O)CN(c2cnccn2)C)nn1 4178,c1(CNC(Cc2onc(CC)c2CC)=O)cc2ccccc2nc1NC 4179,c1(SC)ncc(Br)c(C(=O)NCC2CC(F)CN2C(=O)CCc2scnc2C)n1 4180,c1(CNC(C2C(C(=O)OC)C2)=O)ocnc1C(=O)NCC1CCOC1 4181,C1(CCCNC(c2c(C)c[nH]n2)=O)CCN(C(c2cccnc2C2CC2)=O)CC1 4182,C1(C(N2CC(CNC(c3cc(C(=O)OC)nn3C)=O)C2)=O)(COC)CCOCC1 4183,C(C(=O)N=S1(=O)CCC2(C1)NC(=O)NC2=O)c1ccc(Oc2c(C)ncnc2)cc1 4184,N1(C(c2c(CC)ncs2)=O)CCC2CCCC12C(=O)N(CC(F)(F)Cl)C 4185,Cn1nccc1C(CNC(=O)Cc1ncco1)NC(=O)C(F)C1CCCC1 4186,c1(C(=O)NCC(CN(C(COC(C)C)=O)C)(C)C)ccc2[nH]cc(C#N)c2c1 4187,c1(OC)ccncc1NC(=O)CN(C1CCC1)C(c1ccncc1Cl)=O 4188,C1(CCCNC(COCC(=C)C)=O)CCCN1C(=O)C(F)n1ccnc1 4189,N1(C(c2nncc(C)c2)=O)CCC(F)(F)C(CNC(C2CC=CCC2)=O)C1 4190,O=C(N=c1[nH]nc(Cl)cc1Br)C1CC2CC2N1C(c1cn2cc(F)ccc2n1)=O 4191,C(=O)(CCC(C)OC)N1C(CNC(CCCOCC)=O)CCC1 4192,CCC(CC)CCCC(=O)NC(COCC)C(=O)N(CC(C)C(C)C)C 4193,c1(C(C(=O)NCCCN(C(CCCOC(C)=O)=O)C)C)ccc(C)cc1 4194,c1(C(C)NC(C)(C)C)ccccc1Br.c12cc(on1)C(C)(C)C1CCCN1C2 4195,C1(C(=O)NCCCOCC)CCCN(C(c2nc(C)sc2C)=O)CC1 4196,C1(CC)CCN(C(c2cc(F)c[nH]2)=O)C1CNC(=O)CCc1nncs1 4197,Cc1ccc(OCC(=O)NCC2(CO)CC2)c(C)c1.C(=O)CCC=CC(C)C 4198,C=CC(CC)CC(=O)NC1CN(C(c2cn(C)nc2-c2cccs2)=O)CCC1O 4199,C(=O)(C(O)CCCNC(c1cccnc1)=O)N1CCC(OC)C1C1CC1 4200,c1(C(N2C3C(C(=O)NCCCN(CC(C)C)C)C(C3)C2)=O)c[nH]c2ccccc12 4201,CCCC(CCC)C(=O)NC1(C(=O)NC2CCCC(OC)C2)CC(F)(F)C1 4202,C1(NC(c2c(CC)nc[nH]2)=O)COCCC1NC(C1(C2CCC2)CC1)=O 4203,c1(C2(C(=O)NC3CCC(CCNC(c4n(C)nnc4)=O)C3)CC2)ccc(Cl)cc1 4204,c1(C(=O)NC(C)C(C)NC(c2csc(O)n2)=O)ccc(-c2cnnn2C)cc1 4205,C(C(=O)NCC(F)C1CCC1)(C(C)(C)C)NC(c1cn(-c2ccn(C)n2)nn1)=O 4206,C=CC1OCCC1N(C(=O)COCC)CCC1CCCC1.N12CCCCC1C2=O 4207,C1(NC(CNC(CNC(C)=O)=O)=O)CCCN(C(=O)CC2CN(C)CC2O)C1 4208,N1(C(C(=O)NC(C)C)=O)CCC2CCC(NC(=O)CCCC(F)(F)F)C12 4209,C1(C(=O)NCC(c2ccccc2)NC(=O)CC2CCC2)CC2(COC(=O)N2)C1 4210,c1(-c2ccc(CNC(CCOC)=O)nc2)cccc2nn(C)c(C)c12 4211,C1(NC(COCCCC)=O)CCCC1(C)CN(C(=O)CC1CC1C(F)(F)F)C 4212,C1(NC(CC2C(C)CC2)=O)C2CCN(C(=O)C(C)(O)C3CCCCC3)CC12 4213,C1(CNC(CC(c2cccc(C(F)(F)F)c2)C)=O)CC(F)(F)CO1 4214,c1(C(N2CC(CO)C(CO)C2)C(=O)NC(CC)(C)C)nc2ccc(OC)cc2s1 4215,Cc1cc(NC(=O)Cc2csc(NC(c3ccc(Br)cc3F)=O)n2)cc(O)c1 4216,CC1CCn2cc(C(=O)NCC(C)(C)NC(C34CC(C)C3C4)=O)nc2C1 4217,c1(NC(=O)N(C2CCOC2C(F)(F)F)Cc2cccc(F)c2)cccc(Br)c1 4218,Cc1ccc(C2(C(N3CCC(CCNC(=O)CC(C)O)C3)=O)CC2)cc1Cl 4219,N1(C(C(C)OC)=O)CCC(F)(C(=O)NCCc2cnn(C)c2C)C1 4220,S(=O)(=O)(c1cnccc1N1CCC(F)CC1)NCC1(OCC)CCSC1 4221,c1(OC(C)C)cncc(C(=O)NCC23CC2CN(C(C2C=CC=CC=C2)=O)C3)c1 4222,C(Cc1ccco1)(C(=O)NOCCC(F)(F)F)NC(c1cc(C#N)[nH]c1)=O 4223,c1(C(=O)NCC(C)(C)OCCNC(C(C(CC)O)C)=O)c([N+](=O)[O-])c(C)nn1C 4224,C1(Cc2nnc(N3CCN(C(C)=O)CC3)n2CC2CCOC2)CCC(F)(F)CC1 4225,CC1(C)CCN(C(=O)C(c2ccc(F)cc2)(C)F)C(C(=O)O)C1 4226,c1(C(=O)NCCCOCCNC(=O)Cn2cncn2)coc2c1C(O)CCC2 4227,c1(CCC)cc(C(=O)N(C2CCC(NC(C3CC4CC3C4)=O)C2)C)cc(O)n1 4228,N1(C(Cc2c(C)nccc2)=O)C(C(=O)NCC2(C)CSC2)C2CC(O)C1C2 4229,N1(C(C(CC2CC2)OC)=O)CCC(C2CCN(C(=O)C(C)(C)CF)C2)CC1 4230,CCC(C(=O)NC(C)CCCNC(=O)C(=O)N(C)C)C(C)(C)CC 4231,c1(C(=O)NC2COCC2NC(C2CC2F)=O)cc2occc2[nH]1 4232,c1(-c2ccc(CN(C(C)(C)C)CC)cc2)ccc(F)c(C)c1 4233,S(=O)(=O)(c1ccc(Br)cc1NCC(C(F)F)c1ccccc1)N(C)CCOCCO 4234,Cc1ccc(C=C(C#N)C(=O)N2CC(NC(=O)C(C)OCC(C)C)C2)cc1.CC#N 4235,C(CC(C(=O)N1OC2CCC1CC2)NC(c1cncnc1C)=O)=CC 4236,Cc1nc2cc(C(N3CC4CC3C4NC(C3COCCN3C)=O)=O)cnc2[nH]1 4237,c1(C(C)(C)C)ccc(C(N2CCCC2(C)NC(=O)COc2ccccc2)=O)cc1 4238,N1(C(C(C)Cc2ccccn2)=O)CCN(C(c2cc(Cl)ccc2N)=O)C(C)C1 4239,C1(C(=O)NC(C(=O)OC)C)CCC(C)(C)N(C(=O)C=C2CCC2)C1 4240,CC(CC(F)F)C(=O)N1C(C(=O)NCC(=O)NCC2CC2)CCC1C 4241,N1(C(C=Cc2c(C)ccs2)=O)CCC(C)(C)C(CNC(=O)C(C)C(C)C)C1 4242,c1(C(=O)NCC2CCN(C(C3CSCC(=O)N3)=O)C23CC3)cn2ccccc2n1 4243,N1(C(C2CCC(C)C2)C(=O)NCCCSCC)CCC2(CC(C(=O)OC)=NO2)C1 4244,c1(C(=O)NCC(CNC(CN(C(=O)OC)C)=O)C(F)(F)F)cc(C)c(F)c(C)c1 4245,C1(C(N2CC(OC(=O)C3CC3)C2)=O)C2CCC(C2)C1NC(c1cnco1)=O 4246,c1(CCNC(C(=O)Nc2c(C(C)(C)C)cccc2)=O)nc2ccccc2s1 4247,C(C(CC(=O)N1CCC(NC(C2(C)CCCCCCC2)=O)C1C)C(F)F)N(C)C 4248,c1(C(C(=O)OC(C(C)=O)C(C)=O)=O)c[nH]c2ccc(F)cc12 4249,S(=O)(=O)(c1cc(F)ccc1C#N)NC1CCC(C)(C)CC1CN=c1[nH]ncs1 4250,C1(NC(C2N(CC)CCCC2)=O)CC=C(C(=O)NCC2CCOC2=O)C1 4251,c1(CNC=O)ccc(CO)o1.CCC(CNC(=O)OC(C)(C)C)OC1CC1(F)F 4252,c1(-c2cn(C(C)C(N3CCC(OCCO)C3)=O)nn2)c(Cl)cncc1Cl 4253,c1(C(=O)NC2CN(C(C3CC(=O)N(C4CC4)C3)=O)C2)cc2c(s1)CCOC2 4254,C(C)(C)(CC(F)C(=O)NC1CC(CO)C2CC12)NC(C(n1c(C)ccn1)C)=O 4255,c1(C(=O)NCC2(C)CC(NC(c3c(C)nc(O)cc3)=O)C2)ncnc2sccc12 4256,S(=O)(=O)(c1ccc(NCC2(C)CSC(C)=N2)c2cnccc12)N1C(CC)CC1 4257,N1(C(C(C)OCC2CC2)=O)CCCC(C(C)NC(=O)CCc2ccncc2)C1 4258,Cc1ccc(C#N)c(NC(=O)CC2CN(Cc3ccc4c[nH]nc4c3)CCO2)c1 4259,CCC(CC(F)(F)F)C(=O)NC1(C)CC(NC(c2cc(Br)cn2C)=O)C1 4260,N(C(=NCCCCl)NC1CC2(CC2)C1)C(c1c(C)nns1)C 4261,C(C)(C(=O)NC1CCC(n2cc(-c3ccc(C)nc3)nn2)CC1)(C(C)C)OC 4262,c1(C(N2CC(C(C)NC(CSCCC(C)C)=O)C2)=O)csc(N=S(C)(C)=O)n1 4263,C1(C(=O)NC(c2occ(C(N(C3CCOC3)CC)=O)n2)C)CC(C)N(C)C1 4264,C1(CNC(CNC(c2ccc(SC)s2)=O)=O)CCCN(C)C1=O 4265,c1(COCC(N2CC(O)(C(C)NC(CC=CC=C)=O)C2)=O)ccccc1Cl 4266,c1(OC)cccc(NC(c2cc(C)cs2)c2nnnn2-c2ccccc2C)c1 4267,C(=O)(CCCCCS(N)(=O)=O)N1CCC(C)C(NC(=O)CCCC(=O)C2CC2)C1 4268,C(=O)(CC1=NN(C)C(=O)C1)N1C(C(N2CCN(C)C3(C2)CC3)=O)CC(O)C1 4269,Cc1cccc(F)c1C(N1CCN(C(=O)C(c2ccc(Cl)cc2O)=O)CC1C)=O 4270,N1(C(C(COC)C)=O)CCCC12CCN(C(C1CCC(CN(C)C)O1)=O)CC2 4271,c1(CC(C(=O)NC2(CC)CCOC2)C)ccc(OC)c(OC)c1 4272,c1(C(=O)NCC2CN(C(CCCOCC)=O)CC2O)cnn2c1CC(C)CC2 4273,[N-]=[N+]=NC1CCC2(C(=O)NC3CC(F)C3)CC12 4274,N1(C(C2C(C=C)C2)=O)CCC(C2(NC(=O)Cc3cc(C(F)(F)F)n[nH]3)CC2)CC1 4275,c1(CN2CC(F)(C(N)=O)C2)nc(Br)ccc1N 4276,C1(NC(c2ccc(CC)o2)=O)CCN(C(=O)C(O)Cn2cncn2)C1(C)C 4277,c1(C(=O)NCC(C23CCC(CC2)C3)NC(CC(=C)C)=O)ccc2ncncc2c1 4278,N1(C(CC)=O)CC2CC2(CNC(=O)C(N2CCNC2=O)C)C1 4279,N1(c2cc(C)nc(Cl)n2)CC2CC1CCC2NC(=O)CC(C)n1ccnc1 4280,CC1CC(C(=O)NC(C)CNC(=O)CC2CCC(C(F)(F)F)O2)CC(C)C1 4281,C1(C(=O)NC(CC=C)CNC(c2csc(NC=O)n2)=O)CCc2ccccc2O1 4282,C12(C(=O)NCCC(C(C)C)NC(=O)C(C)(C)c3cc[nH]n3)COCC(C1)OC2 4283,c1(NC(c2scc(-c3ccc(N(C)C)nc3)c2)=O)ccc(Cl)nc1Br 4284,C1(C(N2CC(n3ncc(NC(C=C(C)C)=O)c3)C2)=O)COCCN1C 4285,N1(C(C=COCC)=O)CCSC(C(N2CCC(c3cncc(C)c3)CC2)=O)C1 4286,n1(C(C)C)nnc2c(N3CCC3CNC(C3CCC(C(N)=O)O3)=O)ncnc12 4287,N1(C(C=CC(=O)OC(C)(C)C)=O)CCC(C)(C)C1CC(=O)N1CCC1CO 4288,c1(C(N2CCC(C(C)NC(C3(CO)CCCO3)=O)C2)=O)cc2c(cn1)OCCC2 4289,c1(C(=O)NCC(C)(C2CC2)NC(C(C)OCC#C)=O)cncc(F)c1C(F)(F)F 4290,CC1CN(C(C2CCC3(CCC3)O2)=O)CCN(C(=O)CCc2cn[nH]c2)C1 4291,C(=O)(C(CC(C)(C)C)NC(=O)C1=C(C)OCCC1)N1CC(CCC)C(OC)C1 4292,c1(C(C(=O)N(CC(C)(C)NC(Cc2c(C)con2)=O)C)O)cc(F)cc(F)c1 4293,S(=O)(=O)(c1ccc(Cl)cc1)N1C(C(=O)NC(C(C)C)CCO)C2CCC1C2 4294,c1(C(N2C(CNC(CSCCCC)=O)C(CC)CC2)=O)cc(F)cnc1O 4295,C1(OCOCCOC)CCCCN1C(=O)C(C)OC(=O)CCCc1csc(C)n1 4296,CC1(C)C(NC(c2cc(Cl)ccc2Cl)=O)CC1N=c1ccnc(Cl)[nH]1 4297,C1(CNC(C(C)NC(c2ccco2)=O)=O)CC12CCN(C(=O)C=C1CCC1)CC2 4298,CCCC(O)C(=O)N(CC)CC1CCCN(C(=O)C(C)CC2CCCCC2)C1 4299,CC(C)CCN=C(NCC1(C)CCCO1)NC1CCCN(c2ccccc2Cl)C1 4300,N1(C(c2cc(OCC)n[nH]2)=O)CCC2(C1)CN(C(=O)C(C)(C)CCF)CCO2 4301,C1(NC(C(C)(C2CCC2)NC(C=CCC)=O)=O)CCCCNC1=O 4302,C(=O)(CCP(C)(C)=O)NCC(c1cccc(C)c1)NC(c1cnc(CC)[nH]1)=O 4303,N1(C(c2c(C)[nH]nc2Br)=O)CCN(C(=O)CC2CCCOC2)C(C(F)F)C1 4304,c1(C(N2CC(NC(CCC#CC)=O)C2)=O)cc(F)ncc1OC 4305,CC1(CCNC(=O)CC2(O)CCCC2)CCN(C(C23CC(F)C2C3)=O)C1 4306,N1(C(C(=O)NCC(CC)NC(=O)CCOC(C)C)C)CCCCC1 4307,c1(C(N(CCc2ccc(OC)nc2)C)=O)c(C)nn(-c2ccccc2)c1C(F)F 4308,N1(C(C2(CC)CC2)=O)CC2CCC1C1CN(c3c([N+](=O)[O-])c(C)nn3CC)CC21 4309,c1(OC)cc(C)ccc1C(N1CC2CC1C2NC(c1ccnnc1)=O)=O 4310,c1(C(N(CCNC(c2ccc(O)c(O)c2)=O)CC)=O)cc2cc(C)ccc2s1 4311,CC1COCC(C(=O)NCC#CCNC(c2cnn(C)c2Cl)=O)O1 4312,C1(C(=O)NCCCC(C)NC(CC2(C(=C)F)CCC2)=O)CCC2(CC1)CC(=O)C2 4313,c1(OC)cc(C(N2CCCCC2CN(C(=O)C(O)COC)C)=O)ccc1F 4314,c1(C(N2C(CNC(=O)CN(C)C3CC3)CC(OC)C2)=O)ccc2c(c1)N(C)CC2 4315,C(CCCCCS(=O)(=O)CCO)NC(=O)NC1CCC=CO1 4316,c1(C(N2CCN(C(C(C)CC3CC3)=O)CC2)=O)cccc2c1OC(C)C2 4317,n1(CCC(=O)NCC2CN(C(c3cnccc3Cl)=O)CCO2)cnc([N+](=O)[O-])c1 4318,c1(CN(C)C(C2CCN2C(C2CCCC2O)=O)=O)nccn1C 4319,c1(C(N(C)CC2CN(C(c3cn(CC)nn3)=O)C2)=O)ccncc1OC 4320,Cc1ccc(C(=O)NC2CC(CCNC(c3cccnc3N)=O)C2)c(Cl)c1 4321,c1(C(=O)NCCCOCCN(C(CSCC#C)=O)C)cnn(-c2ccncc2)c1 4322,Cc1n[nH]cc1NC(c1c[nH]nc1CCNC(c1c[nH]nc1C1CC1)=O)=O 4323,Cc1nc(NCc2ccccc2CO)cc(=NCC2C3CCCC23)[nH]1 4324,C(CCCCC1CC1)NC(C1CC(n2cc(-c3csc(C(F)(F)F)c3)nn2)C1)=O 4325,N1(C(C=CC=CC)=O)CC2CCCCC2(CNC(c2cc(F)ccc2F)=O)C1 4326,N1(C(c2nc(CC)oc2C)=O)CC2CC1CN(C(C1(C(N)=O)CCC1)=O)C2 4327,C(=O)(CC(c1ccccc1)C1CC1)NCCC(C)N(C(CCNC(C)=O)=O)C 4328,N1(C(CCN2CCC(C)CC2)=O)CCC(NC(c2ccc(Cl)s2)=O)C(CO)C1 4329,N1(C(C2CCC(N(C)C)CC2)=O)CCCC2(NC(=O)C3=CCOCC3)CC2C1 4330,c1(CNC2CC(C(N3CCC(F)C3)=O)C2)cnn(-c2ccccc2)c1 4331,c1(C(=O)NCCC(C)NC(=O)CCCCO)ccc(O)cc1 4332,CCC(C)CCC(O)CC(=O)NC1(CNC(C2CCCN2CC(C)C)=O)CCC1 4333,C#Cc1cc(C(C(=O)NCC2CCOC2)N(CCC#N)CC2CC2)cc(Br)c1 4334,N1(C(c2c(CC)[nH]nc2Cl)=O)CCC(NC(=O)Cn2cc(N)cn2)C(C)(C)C1 4335,C(C(CC1CC1)C(=O)N1CCCC1CCCO)NC(CC1CC(=C)C1)=O 4336,c1(CCN(C)C)ccc(C(=O)NCC(CO)NC(c2occc2C2CC2)=O)cc1 4337,c1(OC)cccc(F)c1C(=O)NNC(=O)NCc1csc([N+](=O)[O-])c1 4338,c1(C(N2CCC(N(C(C3CCC4CCC3O4)=O)CCO)C2)=O)c[nH]cc(F)c1=O 4339,CCCCCC=CCC(=O)NCCOCCN(C)C(c1cc(C)no1)=O 4340,N1(C(C(C)(CO)OC)=O)CCC2(CC1)COC(CNC(c1coc(C)c1)=O)C2 4341,Cc1ccc(C(N2CCC(CC(=O)NCCn3ccnc3C)C2(C)C)=O)cc1C#N 4342,C1(NC(=O)C=Cc2ccc(C3CC3C)o2)CN(C(=O)C(Cl)=CCl)CC2(CCC2)C1 4343,C(CC(C)(C)C(=O)NC1CCCCC1C)NC(C1C(C)CCOC1)=O 4344,Cc1ccc(F)c(NC(C2CCCCCN2C(C2CC23CCCCC3)=O)=O)c1 4345,CC1CCC(C(=O)NCc2cscn2)N(C(C2CC2C(=O)OC)=O)C1 4346,CCCC(CCC)C(=O)N1CC(CC(F)C(=O)N(C)CC2(C#N)CCC2)C1 4347,Cc1nn(C)cc1CC(=O)NCC1COCCN1C(C1CC(CC(F)(F)F)C1)=O 4348,C(=O)(C(C)(C)CC1CCC1)N1CCC(c2cn(CCC(C)(C)F)nn2)C1 4349,C1(NC(C(C)CF)=O)CC(CO)N(C(c2cncc(-n3cnnn3)c2)=O)C1 4350,C1(C(=O)NC2CCN(C)C(=O)C2)CC12CCN(C(=O)CC1C=CCC1)CC2 4351,c1(C(COCCNC(COCCOCC)=O)C)ccc(N(CC)CC)cn1.CC 4352,C(=O)(CCCN(C)C(c1cc[nH]n1)=O)N(CCC)C1CC1 4353,N1(C(C2CC(=C)C2)=O)CCC2(CC1)CN(C(c1n[nH]c(C)c1[N+](=O)[O-])=O)CCO2 4354,C(=O)(C(C)(C)S(C)(=O)=O)N(C(C1CCCO1)C)C(c1cc2c(s1)CCC2=O)=O 4355,C#CC1(O)CCN(C(c2ccnc(CNC(=O)CSC(F)F)c2)=O)CC1 4356,c1(C(=O)NCC(F)CNC(c2coc(Cl)n2)=O)cccc(N2CCOC2=O)c1 4357,c1(C(=O)NCCN2CCN(C(C3(C#N)CC(C)C3)=O)CC2)n[nH]c2ccccc12 4358,c1(NC(=O)CC2CCCN2Cc2cccnc2)cc(Cl)c(Cl)cc1F 4359,c1(CCC(=O)NCC2C(NC(c3c(CC)scc3)=O)CC2)c(C)n[nH]c1C 4360,c1(CN(C)C)ccc(C(=O)NCC=CCNC(C2CC2c2cccs2)=O)cc1 4361,Cc1c(C(=O)NC2CN(C(=O)CCc3nc(=N)[nH][nH]3)C3CC23)c(C(F)F)nn1C 4362,c1(N(CCCN(C(C2C(COC)CCCC2)=O)C)C)ccc(C#N)nc1 4363,C1(N(C)C(c2cc(F)ccc2F)=O)CN(C(=O)CN2CCS(=O)CC2)CC1(C)C 4364,CC1(C)CC=CCN(C(C23COCC2CN(C(C24CSCC2C4)=O)C3)=O)C1 4365,c1(NC)snc(C)c1C(=O)NC(CO)C(C)NC(c1csc(-c2cnc[nH]2)n1)=O 4366,CC1CCC(C2CCC2)CN1c1nnc(-c2ncc(Cl)cc2Cl)n1CC1CC1 4367,C1(NC(C=C(C)C2CC2)=O)CCN(C(=O)CC2CCCCO2)C12CCCC2 4368,C(CC(C(F)F)c1ccccc1)NC(c1nnnn1-c1ccccc1)CCC 4369,c1(SC)nc(Cl)cc(=NCC(C2CC2)NC(=O)CSCC(F)(F)F)[nH]1 4370,C(CCC(C)C(=O)NC12COC(C1)C(NC(=O)CN1CC(C)(C)C1)C2)OC 4371,C1(C(=O)NC2CC2C(=O)NCc2cccc(CO)n2)(CC)CCCCC1 4372,c1(C(=O)NCC2C3CN(C(Cn4nnc(C)n4)=O)CC32)ccc(F)c(Cl)c1N 4373,c12ccc(cc1C)NC1CC3(C(C3)C(=O)NC3CC3CNC(=O)C2C)C1.CCOC 4374,c1(CC(=O)NC2CC(C(=O)Nc3c(C(=O)OCC)ccs3)C2)ccnc(Br)c1 4375,C(=O)(CCC(F)(F)C(F)(F)F)NC(CSC)C(C)(C)C 4376,c1(C(C(=O)NC2C(NC(c3c(C)occ3)=O)C2)O)ccccc1F 4377,C(CN=c1ccnc(NCc2cccc(N3CCC(SC)CC3)c2)[nH]1)OC 4378,c1(NC(=O)NCC2C(OC)C2)cn(C(Cc2ccccc2)C(=O)O)nn1 4379,c1(CC(N2CC(O)CC(NC(c3cnc(Cl)[nH]3)=O)C2)=O)c(Cl)ccc(O)c1Cl 4380,C1(CC(=O)N(C)C(c2ccccc2)c2cccnc2)CC2OCCC2O1 4381,N1(C(CNC(CCC)=O)=O)CCCOC(CCNC(=O)C(C)(C)C(=O)NC)C1 4382,Cc1cccn2c(C(=O)NC(C3CCN(C(c4coc(O)n4)=O)C3)C)cnc12 4383,c1(NC(C2C(C)(C)C(F)(F)C2)=O)ccc([N+](=O)[O-])cc1-c1nn[nH]n1 4384,C(=O)(CCCCCCCC1CC1)N1CC2(CNC(CC(C)SC)=O)C(C1)CCO2 4385,CC1(C)COCCC1Cn1cc(-c2cccc(C(F)(F)F)c2)nn1 4386,c1(C(N2CC(OC)(CNC(c3cc(C)co3)=O)C2)=O)ncccc1C 4387,Cc1cc(=O)oc2cc(NC(C3CCN3C(c3cccc(F)c3F)=O)=O)ccc12 4388,n1(CC#C)cccc1C(c1nnnn1C1CCOC1)NCCC1(CSC)CCC1 4389,CCC(CC)C(C(=O)NCCCN(C(=O)CCC1NC(=O)NC1=O)C1CC1)OC 4390,C1(NC(c2ccc(C)c(O)n2)=O)CC2CCC1N(C(c1coc(Br)n1)=O)C2 4391,C=CCC(C(=O)NOCc1ccc(O)cc1)NC(=O)C(C)CC1CCC1 4392,C1(C)(C(=O)NCC(C=C)O)C=CCN1C(=O)C(CCOC)OC 4393,C1(C(=O)NCC(CN(C(COCCCOC)=O)C)C)CC1C1CCCC1 4394,CCC(C)CC(C)C(=O)N(CC(CO)(CO)NC(c1ccnc(OC)c1F)=O)C 4395,c1(CC(=O)N)cccc(OCC=CC2CC2)c1.C(=O)(CC1CC1)N(C)CCNC=O 4396,C12(C(=O)NCC(CC(C)C)(C)NC(=O)CSC3CC3)CCCN1S(=O)(=O)CC2 4397,C1(COC)(CNC(C2CCC2C#N)=O)CN(C(=O)Cn2cc(C)cn2)C1 4398,CC(CC(=O)N(CC(=O)NCc1nc(C(N)=O)co1)C1CC1)n1cccn1 4399,CCCC(CCC)C(=O)NCC1CCN(C(=O)CNC(c2ccco2)=O)CC1C 4400,N1(CC(=O)NCCN(CCC)C(C2CCCOC2C(C)C)=O)CCC(=O)NC1=O 4401,Cc1c(NC2CSC(C)C2)ncnc1N1CCCN(CCCO)CC1 4402,N1(C(C(CC)CC(C)C)=O)CC2(CCN(C(C3(COC)CC3(F)F)=O)CC2)C1 4403,c1(C(N2CC(CNC(=O)CCCOc3ccccc3F)C2)=O)cccnc1OCF 4404,N1(C(CCCN(C)C)=O)CC2CCC(C1)N2C(c1cc(=O)n(C)o1)=O 4405,c1(OC(C)C(=O)NC2CC(C)(NC(c3cc(Cl)cs3)=O)C2)cccc(Cl)c1 4406,N1(C(C(COC)(C)C)=O)CCC2CCC(C1)N2C(=O)CC(C(C)C)c1ccon1 4407,N1(C(CC=CCCCCC)=O)CCC2CC(NC(=O)CSCCOC)CCC2C1 4408,C(CC(O)C(=O)N1CCCCC1CN(C)C(c1cccc(C2CC2)n1)=O)SC 4409,N1(C(CNS(NC)(=O)=O)=O)CC2COCC(C1)C2NC(=O)C(C)n1cccn1 4410,C1(CNC(=O)CC2(O)CCC2)CC2COCC2N1C(C1CC2CCCC(C1)C2)=O 4411,CC1=CCSC1C(=O)NC1(C)CC(C(=O)NC(C)CCn2cncn2)C1 4412,C(=O)(CCS(C)(=O)=O)N(C1CCCCC1N(C(=O)CC1CCC2(CCC2)O1)C)C 4413,C(C1CCCCC1)=CC(=O)NC(C(=O)N(C(C)CC(N)=O)C)c1ccco1 4414,N1(C(c2ncn(CC)c2)=O)CC(F)(F)CC1CCNC(c1cc(F)ccc1F)=O 4415,c1(C(N2CCC(NC(C3N(C(C)=O)CSC3)=O)C(O)C2)=O)c[nH]c2ccncc12 4416,C1(CNC(CC(C)CF)=O)(NC(C2Cc3nccn3C2)=O)CCC(C)(C)CC1 4417,Cc1ccc(CN(C(C(N2CCOC(CN(CCC(N)=O)C)C2)=O)C)C)cc1 4418,c1(C(=O)NCC(CNC(CC2(C)CCCCC2)=O)F)nccc2c1CNC2=O 4419,C(=O)(NNC(=O)C(C)(C)CCCCNC(=O)C(F)(F)CC1CC1)C1CC(C)C1O 4420,c1(N2C(C)CC(NC(C3(C4CCC4)CC3)=O)C2)ncnc2[nH]ccc12 4421,C12CN(CCC1F)C(=O)c1c(nccn1)C(=O)N2.c1(SC(C)C)nncn1C 4422,C1(C(=O)NC(C(C)(C)C)CNC(=O)CNC(=O)C2CC2)CCC2C(CC1)C2(F)F 4423,Cc1ccc2ncc(C(=O)NC(C3CCCCC3)CNC(c3cnc[nH]3)=O)n2c1 4424,CN=c1nc(N2CCC(OCCO)C2)[nH]c(N(C)CC2(F)CCC2)n1 4425,c1(OCC)ccc(CN2CCC(N(C)C(c3cc(Cl)ccc3I)=O)C2)cc1OC 4426,N1(C(C(C)(C)OC(C)=O)=O)CCC(NCCOCC(F)(F)C(F)F)C(C)C1 4427,N1(C(C2CC(=O)OC2)=O)CCN(C(C2(CO)CC(F)(F)C2)=O)CC1C(F)F 4428,CCCC(CC)CCC(=O)NC1C=CCN(C(=O)C(C)(C)OC(C)=O)C1 4429,C1(C(=O)NCCCc2n(CC)ncc2)C2CCC1N(CC)C2 4430,c1(C(=O)NCC2C(NC(C)=O)CC2)cc(C)c2n[nH]cc2c1 4431,Cn1ccc2[nH]c(C(=O)NC3CN(C(C4COCCO4)=O)CC3CC3CC3)cc12 4432,c1(C(C)C)nn(C)cc1C(=O)NCC1CN(C(c2csc(C3CC3)n2)=O)CCO1 4433,C(=O)(C(O)CC(C)(C)C)N(C)CC1CCCN1C(=O)CCc1c(F)cccc1Cl 4434,C(=O)(C(C)(C)CC(=O)NC1CN(C(C2CCCN2C(=O)OC)=O)C1)NCC 4435,c1(CC(N2CCC(NC(=O)CC3CC4CC4C3)C2)=O)cccc(Br)c1Cl 4436,N1(C(c2c(C)cccc2)=O)CC(NC(=O)CC2NC(=O)NC2=O)CC2(CCC2)C1 4437,c1(C(=O)NCC2C(CNC(C3(C(C)(C)O)CC3)=O)C2)ccnc2[nH]c(O)nc12 4438,n1(CC(=O)NCC(CNC(c2c(CC)nc[nH]2)=O)CO)cc(Cl)c(C)n1 4439,N1(CC(=O)NCC2CC(NC(C3CCC(CCCCC)O3)=O)C2)CCNC(=O)C1 4440,C1(NC(C2CC3CC3C2)=O)CCC2CN(C(C3CC4(CC4)C3)=O)CCC2C1 4441,c1(C2(C(N3CC(CCNC(CC(C)OC)=O)C3)=O)CC2)ccc(Cl)c(F)c1 4442,N1(C(CC(CC)C)=O)CC2CN(C(=O)Cc3ccc(OC)c(O)c3)CC2C1 4443,c1(C(=O)NC)ncccc1NC(c1cn(CC(C)N)nn1)=O 4444,c1(C(C)NC(c2scc(COC)c2)c2nnnn2CCC2CC2)ncccc1F.OC 4445,N1(C(CN2C(C)CC2)=O)CCC2(C1)CN(C(c1ccc3nccn3c1)=O)CCO2 4446,N1(C(C(C)OC)=O)CCC(C(C)(C)NC(C2CC2C)=O)CC1 4447,C1(NC(C(CC)N(CC)CC)=O)CCN(C(c2cc(=O)c(OC)c[nH]2)=O)CC1C 4448,C12(C(=O)NC(CCOC)CNC(C3CCOC3)=O)CCC(CC1)CO2 4449,C(=O)(CCC(C)=O)NC1(CC)CN(C(=O)Cc2cnn(C)c2)C1 4450,CC1(C#N)CC(c2nnnn2CC2CCOC2)(NCc2cscn2)C1 4451,c1(C(=O)NC2C(NC(C3ON=C(C)C3)=O)CCC2)ccc(=O)n(C)c1 4452,CC1(C)CCC(NC2CCN(c3nc[nH]n3)CC2)c2ccccc21 4453,N1(C(C(n2cc(-c3cccc(N)c3)nn2)C)=O)CCN(C(=O)CO)C(C2CC2)C1 4454,Cc1cc(N(C)CCn2cncn2)nc(N(C)CC2CCCO2)n1 4455,c1(C(=O)NCC(CC)NC(C(CC=C)C)=O)ccc(Br)c(C(=O)OC)c1 4456,N1(CCS(=O)(=O)N2CCCCC2)CCOC(c2cccc(Br)c2)C1 4457,C(=O)(C(CC)C(=O)OC)NCCCC(=O)NC1C(CC=C)CCCC1 4458,N1(C(c2cc(CC)[nH]n2)=O)CCN(C(=O)C(O)CC(C)C)CC1C1CC1 4459,Brc1cccc2c1C(NC(c1nnnn1C1CCC1)C1CCC1)CC2 4460,C1(NC(c2cnc(Cl)[nH]2)=O)CCN(C(c2nccnc2C(F)F)=O)CC1F 4461,c1(NC(=O)NCc2ccc(N3CCS(=O)(=O)CC3)nc2)cc(I)c(O)c(I)c1 4462,C1(C(=O)NC(CCC=C)C)CCC(NC(=O)C(O)CN2CCCC2)CC1 4463,N1(C(CN(C(c2nn(C)cc2Cl)=O)CC)=O)CCC(CO)C(O)C1 4464,n1(CC(=O)N(C)CC2CCCN(C(c3cc[nH]c(=N)c3)=O)C2)nc(Cl)ccc1=O 4465,N1(C(CC=CC=C)=O)CC2CCCC1CN(C(c1cc(C)ccc1Cl)=O)C2 4466,C(CCN=c1ccnc(N2CCCC(C)(F)C2)[nH]1)N(CCC)CCN(C)C 4467,N1(C(Cc2cccc(NC(=O)OC(C)(C)C)c2)=O)CCC2CCOCC2C1 4468,CCS(=O)(=O)CC(=O)N1CC(C)CCC1C(=O)NCCC1CCCC1O 4469,C1(CC)CCCCC1NC(c1conc1CNC(=O)CC(C1CC1)C1CC1)=O 4470,c1(CC(N2CCC(N(C(c3[nH]cc(C)c3C)=O)CC)C2)=O)ccc(F)cc1F 4471,N1(C(C2(COC)CC=CC2)=O)CCC(C)(CNC(C2COC2)=O)C1 4472,C1(C(N2CCC(OC)(CNC(c3cncc(CO)c3)=O)C2)=O)CC(=O)NC(=O)N1 4473,CC1(C)CCC(C(=O)NC(C)(C)COCCCNC(=O)C=C2CCCCC2)OC1 4474,Cc1cc(N2CCN(S(C)(=O)=O)CC2)nc(=NCCC(C)OCC(F)(F)F)[nH]1 4475,N(C)(S(=O)(=O)NOC(C1(OCC)CC=CCC1)=O)CC#C 4476,CCC(CNC(=O)Cc1cnoc1)(CC)C(=O)N(C)Cc1cccc(O)n1 4477,N1(C(C2CCCSC2)=O)CCCC(C(N2CC(n3cccn3)C2)=O)C1 4478,C(CCCC(C)(C)C(=O)NNC(=O)C1SCCC1C)NC(c1[nH]cc(CC)n1)=O 4479,c1(NCc2c(C)nn(C)c2Cl)[nH]c(=NC(C)CC2CCOC2)nc2c1ncn2C 4480,C(=O)(C(C(C)C)C1CCC1)NCC1(OC)CN(C(c2cnc(O)o2)=O)C1 4481,Cn1ncc(C(=O)NCc2ccc(Br)cc2Cl)c1C#N 4482,c1(C(=O)NC(C)C(N2CCN(C(c3cncnc3)=O)CC2)=O)ccc(F)cc1F 4483,C1(OC)(CNC(C2(F)CCN(C(=O)Cn3cnnc3)C2)=O)CCCCC1 4484,C1(O)(CNC(C(N2CCNC2=O)C)=O)CCCN(C(=O)CCc2cnn[nH]2)CC1 4485,C1(C(=O)NC2CC(F)(CNC(C(C)OCC)=O)C2)CC(C)(C)CC(C)(C)C1 4486,c1(C(=O)NCC(C)NC(CCC(C)c2ccccc2)=O)cc2ccccc2n1C 4487,C(=O)(C(C(=O)NCC(C)(C)CCNC(C1(C)CCNC1=O)=O)OC)OC 4488,c1(C(=O)NCC2CC(F)(CNC(C3(CCCC)CC3)=O)C2)cnn(CC)c1C 4489,C1(C2CCN(C(=O)COCc3ccccc3Cl)C2)(NC(=O)CCC2CC2)CC1 4490,C1(NC(CCCC)Cc2ccccc2)CCc2cc(C#N)ccc2C1 4491,CC(C)C(CCN(C(=O)CC1C(C)C1(F)F)C)NC(c1cnc(S)n1C)=O 4492,c1(OC)cncc(-n2cccn2)n1.C123CC1CN(C2)C(=O)C1CC(C1)OC3=O 4493,C(N=c1nc2c(Br)csc2c[nH]1)C1(O)CCCN(C(Cc2c(C)cccc2)=O)C1 4494,N1(C(C2OCCN(C)C2)=O)CCC2(CC1)CN(C(c1ncccc1N)=O)CCO2 4495,c1(NC(C)C)ccc(C(=O)NCC2CC2CNC(c2cc(Cl)no2)=O)cn1 4496,O=C(C1CCCc2cccnc21)N1CCC2(CC1)CCN2C(C1C2C=CSC12)=O 4497,N1(C(CN(CC(C)C)C(C2CC(=C)C2)=O)=O)CCOC(C(N)=O)C1 4498,c1(CC(=O)NC2CN(C(CC(C)(C)C#N)=O)CC2(C)C)csc2c(F)cccc12 4499,CC1CCN(C(=O)CN2CC3CCC2C3)CC1CNC(c1cc(Cl)on1)=O 4500,c1(NCC2C(=O)NCCC2)[nH]c(=NCCc2cccc(Cl)c2)nc2scnc12 4501,C1(C(=O)OC)CN(C(C2CN(Cc3nc(Br)cs3)CCS2)=O)CCC1O 4502,N1(C(CC2C(=O)NCCC2)=O)CCCC(Cl)(O)CC1 4503,N#Cc1ccc(C(=O)NC2(C(N3CCC3CO)=O)CCSC2)s1 4504,CN1C2(CCN(C(c3cnnc(O)c3)=O)CC2)C(NC(=O)CCCF)CS1(=O)=O 4505,C1(CNC(Cc2cc(C)sc2)=O)COCCN1C(=O)CCCn1cncn1 4506,C(=O)(C(CCC(C)C)NC(=O)C=Cc1cocn1)N1C(CCCC)CCC1 4507,N1(C(C(Cc2cc[nH]n2)NC(=O)Cc2cnco2)=O)CCC12CCCC2 4508,n1(C(C(N2CCC(OCCOCC(=O)Nc3onc(C)n3)C2)=O)C)nc(C)cc1C 4509,CCC(CN=C(NCCn1cnnn1)NC1CCC1)c1nccs1 4510,c1(CN(C(C(=O)OC)C2CC2)C)ncc(C(C)(C)C)o1 4511,N1(C(=O)OC(C)(C)C)CCC=CC1C(=O)NCC12CC3CC1C2C3 4512,Cn1nc(C(N2CC3CCC(C2)N(S(=O)(=O)CC#N)C3)=O)c2cc(Br)ccc12 4513,c1(CC(=O)NCC23C(CN(C(C(CC#C)O)=O)C2)CC3)ccc(F)cc1[N+](=O)[O-] 4514,C1(C2CCN(C(C(=O)C)=O)C2)(NC(N(CC=C)CCC)=O)CC1.C(C)(C)(C)O 4515,C1(CCC(=O)NCC(CO)NC(=O)CSc2nncn2C2CC2)CCC(O)CC1 4516,C1(CNC(C2C(=C)C2)=O)(COC)CCN(C(c2cc(C)ccc2N)=O)CC1 4517,N1(C(C(C(C)C)O)=O)CCC2(CCN(Cc3cc(-c4ccc(F)cc4)n[nH]3)C2)C1 4518,Cc1cnc(C(=O)N(C2CN(C(c3cnnc(O)c3)=O)CC2F)C)c(Br)c1 4519,N1(C(c2oc(C)c(CO)c2)=O)CCC2(C1)CN(C(C1CC13CCOCC3)=O)C2 4520,N1(C(c2c(SC)cn(C)n2)=O)CC(NC(C2(C(=O)OC)CC2)=O)CC(C)C1 4521,C(=O)(CCCC(=O)C(C)OC(=O)C(Cc1cccc(Br)c1)CC)OC 4522,c1(C(=O)NC2CC(CCNC(C(C)P(C)(C)=O)=O)C2)cnc2ncnc(O)c2c1 4523,c1(C(=O)NCCCCCCNC(C(C)c2ccco2)=O)cc2n(n1)CCO2 4524,N1(C(c2c(C)cn(C)c2)=O)CCCN(C(c2cccc(O)c2Cl)=O)CC1C 4525,CCCC(CCCNC(C1CC1CC)=O)NC(c1ncccc1C(C)=O)=O 4526,C1(C2CCN(C(=O)C(F)CC3CCOC3)CC2)(NC(C(CC)C)=O)CC1 4527,C1(CNC(CCNC(=O)NC)=O)CC2COCC2N1C(c1oc(C)nc1C)=O 4528,C1(N=[N+]=[N-])(C(N(C(C#C)(C)C)CC)=O)CCN(C(=O)CN2CCSCC2)C1 4529,c1(OC)cc(NC(C2CCN2C(=O)C(C)(C)n2ccnn2)=O)ccc1Cl 4530,c1(-c2cc(C(=O)NC3CN(C(c4cnn(CC(F)F)n4)=O)C3)n[nH]2)ccccc1O 4531,C(=O)(CCCC(C)NC(=O)CN1CCCCC1)NCC(C)C#N 4532,N1(C(C(C)CCN(C)C)=O)CCN(C(=O)CC2(C)OCCO2)CC(C)(F)C1 4533,Cc1cc(CC(=O)NCc2nc(C(=O)N(CC(C)O)C)co2)no1 4534,C(=O)(C1=CCCC1P(C)(C)=O)NCC1CCN(C(c2c(CC)con2)=O)C1 4535,C1(NC(CCCOCC)=O)CCCN(C(=O)CCC(C)(C)F)CC1F 4536,CC(N=c1[nH]c(NC2C3COCC23)nc2c1SCC2)C1CCC1 4537,CC(C)C(C(=O)NC(C)Cc1ccncc1)C(C)NC(C1CC(=O)C1)=O 4538,C(=O)(CCN(CC(=O)OC)N1CCCC(CC#N)C1)OCC 4539,N1(C(CC#N)=O)CCC2(NC(c3ccc(-c4ccon4)cc3)=O)CCCC12 4540,CC1(C)OC(=O)CC1C(=O)NC1CC=CCC1C(=O)NCCc1cccs1 4541,Cc1ccsc1CC(=O)NCc1cc[nH]c1C(=O)NCC12CCCC1C2 4542,c1(-c2c(SC)scc2)ccc2ccnc(NC(=O)C(F)(F)Cl)c2c1 4543,c1(C(=O)NCC(C2CCOC2)NC(c2c(C#N)nc[nH]2)=O)cc2ccccc2o1 4544,n1(CC)c(C(=O)NCCC(CNC(=O)CCC2CCCCC2)OC)cnc1O 4545,C(=O)(CCCCCNC(c1cn(C2CC2)nn1)=O)NCC(CCCC)O 4546,C1(NC(c2ccc([N+](=O)[O-])[nH]2)=O)C2CC1CN(C(c1cncn1C1CC1)=O)C2 4547,N1(C(CC(C)C)=O)CCC(CNC(=O)C(O)CN2CCOCC2)C1(C)C 4548,c1(OC)nc(C(=O)NC2CCCCC2n2cc(C3(C)CCOC3)nn2)ncc1F 4549,N1(C(C(C)(O)CCc2ccccc2)=O)Cc2ccc(O)cc2C1 4550,C=CCC(C)C(=O)NC1CCCC(CNC(C2CCN(C(N)=O)CC2)=O)C1 4551,C(N=C(NCC1(C)CCCS1)NC1CCCC1)C1CCN(C(C(C)(C)C)=O)C1 4552,c1(Cn2cc(CC3CCCN(C(CC4(C)CC4)=O)C3)nn2)cc(Cl)ncc1Cl 4553,C1(C)(NC(c2nc(C)sc2)=O)CCCCC1C(=O)NCCc1cscn1 4554,CCC(O)CC(=O)NC(c1cccc(Cl)c1)CNC(c1cnn(CC)c1)=O 4555,C(CC(=O)N1CCC(C(=O)NC(CO)C(C)O)O1)OC(C)=O 4556,N1(C(c2cnn(CCC)c2C)=O)CCOCC(CNC(=O)C(O)C(C)CC)C1 4557,N1(CC(=O)NCCCC(C)NC(C(c2ccc(C)s2)C)=O)CCC(CO)CC1 4558,C12(C(=O)NCCC3CC(C(=O)NC(C(=O)OC)(C)C)C3)CCCC1C2(F)F 4559,C1(C(=O)O)CC12CN(CC(c1cccc(Cl)c1)O)C2 4560,N1(C(C=Cc2cnc(C)s2)=O)CC2CC(NC(c3cc(C#N)c[nH]3)=O)C1C2 4561,Cn1ncc2cccc(C(=O)N(C3CCC(NC(=O)C4=NOCC4)CC3)C)c12 4562,c1(NC(C2CC(CO)CO2)=O)cc(F)cc(I)c1 4563,n1(CC)nncc1C(=O)N(C)CC=CC(=O)NCCCc1cnn[nH]1 4564,C1(NC(=O)CCc2ncc(F)cn2)CCCC12CCN(C(c1ccc(Cl)cc1)=O)C2 4565,C(=O)(C1=C(C)OCCS1)N1CC(CCNC(C(CC=C)CC)=O)OCC1 4566,N1(C(C(CC)OC)=O)CCC2(C1)CN(C(=O)CC1CN3CCN1CC3)C2 4567,N1(C(CC(CC)OC)=O)CCN(C(=O)CCc2ccc(F)cc2F)C(C(C)C)C1 4568,N1(C(Cc2cn(C)nc2Cl)=O)CCCC(NC(=O)C(C)(C)n2cnnn2)CC1 4569,c1(NC(C2(C)CN(C(C3CC34CCC4)=O)C2)=O)ccc(O)c(N(C)C)c1 4570,Cc1sc(Cl)c(C(=O)NCC2(O)CC(CNC(=O)CCCC#N)C2)c1C 4571,N1(C(c2cc[nH]n2)=O)CC23CCCCC2(C1)CN(C(c1ccc(Br)o1)=O)C3 4572,Cc1ccc(C(=O)COC(c2cc(F)sc2NC(=O)OC(C)(C)C)=O)cc1 4573,C(=O)(C1=NOC2(CCC2)C1)N1CCN(C(C(C)N(CC)CC)=O)C2(C1)CC2 4574,C1(NC(c2nocc2Cl)=O)CCCC1CNC(C1(C(F)F)CCC1)=O 4575,C(=O)(CS(C)(=O)=O)NCCC(CNC(c1c(COC)noc1)=O)O 4576,C(=O)(C1CCc2ccccc21)N(C(CCNC(CC(CC)C)=O)C)C 4577,c1(C2(C)C(C(=O)NCC3(C)CCCS3)C2)cccc(Br)c1 4578,C1(NC(c2c(C)noc2)=O)C=CCCC1C(=O)NCC(F)(F)CO 4579,C1(COC(Cc2c(C(=O)OC)csc2)=O)CCC(OC2CCCCC2)CC1 4580,CC1(C)CCN(C(=O)CC2CCC(C(N)=O)O2)CC1CNC(C1CCSCC1)=O 4581,c1(C(=O)NCCC(CNC(C(C(CC)O)C)=O)OC)cc2cnccc2[nH]1 4582,N12CCN(CC1C)C(=O)C1(CCC1)C2=O.C1(CCC)(SC)CCNC1=O 4583,c1(NC(C2(C)CCN2C(C2CC2F)=O)=O)cncc(F)c1I 4584,C12CN(CCC1F)C2=O.CC1(C#N)CN(C(C2C3CCCCC23)=O)C1 4585,c1(OC)ccc(Cl)c(C)c1C(=O)NC1CC(C)N(C(c2ccc(F)o2)=O)C1 4586,c1(OC)cc(C(=O)NCC2CC(C)N(C(=O)CCC(C)N(C)C)C2)cc(F)c1F 4587,N1(C(N=c2[nH]nc(CN(C)C)s2)=O)Cc2cccc(Br)c2C1 4588,N1(C(c2cn[nH]c2)=O)CC2(C1)CN(C(=O)CC1CCCC1)CC2CO.CC(=O)O 4589,C1(NC(c2cc(Cl)ncn2)=O)C2CN(C(=O)CCOc3ccccc3Cl)CC12 4590,C(=O)(CCSCC(N)=O)NCC(N(CC(=O)NCC(F)(F)F)C)C1CC1 4591,Cc1cccc(Br)c1C(=O)NC(C)CNC(=O)Cc1ccc(Cl)nc1 4592,c1(OCC)ccc(Cl)cc1C(=O)NCC(C)NC(=O)CC12CCC(CC1)CC2 4593,c1(CN(C)CC2CCN(C(C3CCCC(CC(F)(F)F)C3)=O)C2)cccc(F)c1 4594,C(=O)(C(C)(CC)CCC(C)C)N(CC(CC)NC(c1cnc(OC)nc1)=O)C 4595,c1(C(N(CC(CN(C(=O)Cc2ccc(O)nc2)C)O)C)=O)ccc2oncc2c1 4596,Cc1sncc1C(N1CCCC1C1CCN(C(c2csc(C(N)=O)n2)=O)C1)=O 4597,N1(C(C2CC3CN(C(CCN(CC)CC)=O)CC2C3)=O)CCc2ccccc2C1 4598,N1(C(CC2(C(=C)F)CCC2)=O)CCCCCC1CNC(=O)C(O)C(C)CC 4599,c1(C(=O)NC2CN(C(C3C(C(C)C)CCC3)=O)CC2(C)C)cnc2ccoc2c1 4600,N1(C(C(C)C#N)=O)CCC(C(F)(F)F)CC1CNC(c1ccnc(S)c1)=O 4601,C1(CC(=O)NC2CN(C(Cc3c(C)cco3)=O)C(C)C2)CC(O)C12CCC2 4602,CCC(C)CCCCC(=O)NC(C1(O)CN(C(c2cc(F)cc(Cl)c2N)=O)C1)C 4603,c1(Cc2ccc(NC(c3n(CC=C)nnn3)(C)CCI)cc2)cccc(CO)n1 4604,CCC(F)(F)C(C)(C)C(=O)NCC1CCN(C(c2nn(C)cc2[N+](=O)[O-])=O)CC1 4605,C1(C(N2C(C)CC(CCNC(C3CCC3)=O)CC2)=O)CCc2nn[nH]c2C1 4606,N1(C(C2CC(=C)C2)=O)CCOCC1CCNC(C1(C(N)=O)CCC1)=O 4607,c1(C(=O)NC2CN(C(C)=O)CC(O)C2)nc2ccc(Br)cn2c1Cl 4608,N#Cc1cccc(NC(=O)CC2CCCC2NC(c2ccc(Cl)s2)=O)c1F 4609,C(CCCC(C(=O)NCCSC)N1CCC(OC(c2ccccc2)=O)C1)OC 4610,C1(CC)CN(C(C2OCCCC2(C)C)=O)CCN1C(=O)CSS(C)(=O)=O 4611,c1(CC(N2CCC(CNC(c3c(C)scn3)=O)CC2)=O)ccc2n[nH]cc2c1 4612,C1(C(=O)NCc2c(C)cco2)CCC(NC(C2CCN(C)C2=O)=O)CC1 4613,c1(C(=O)NC2CC(CNC(CN3C(=O)CC(C)(C)O3)=O)C2)ccc2cnnn2c1 4614,c1(NC(CCC(C)NC(=O)NCC(CC)N2CCCC2)=O)sc(F)cc1C 4615,Cc1nc([N+](=O)[O-])cn1CC(=O)NCC1CN(C(=O)C(Cl)=CCl)CC12CCC2 4616,C(=O)(C(O)C(C)(C)C)N1CC(C)C(n2cc(C3CCCCC3O)nn2)C1 4617,C1(NC(c2c(C)nsc2C)=O)CN(C(=O)CC(C)O)C2(CCCC2)C1 4618,C1(NC(CCc2n(C)ccc2)=O)CCCC12CN(C(c1cc(C(N)=O)[nH]n1)=O)C2 4619,C(CC(C)C)(C(=O)NCCCNC(N)=O)NC(C1N(CC)CC1)=O 4620,C1(C(=O)NCC(c2ccccc2Cl)N(C)C)CCC(N)C(F)(F)CC1 4621,C(CC(C(=O)NCCC(C)(O)CC)NC(=O)C(C)=CCC)=CC 4622,C(=O)(C(C)(C)C(F)F)N1CCC(C2N(C(C3C(C)C3)=O)CCCC2)C1 4623,C(C(=O)N1CCCO1)NC(C(CC=CC)NC(=O)C(C)NC(=O)C1CC1)=O 4624,C1(C(=O)NCCNC(=O)C(O)Cn2cncn2)(CC)CCCCO1 4625,CCCC(C(=O)OC)N(C)N1CC(C)CCC1C(=O)OC 4626,N1(C(CC2(CN(C)C)CCC2)=O)CCC(CNC(c2cncc(N)n2)=O)C(C)C1 4627,c1(C(N(CCCNC(CN(C)C2CC2)=O)CC2CCOC2)=O)nonc1N 4628,c1(-c2cnc(CNc3cc(C)nc(C)n3)nc2)ccc2c(c1)OCO2 4629,C(CCC1CCC1)(C(=O)NCc1ccc(F)cc1)N1C(C(C)(C)CO)CCC1 4630,c1(C(=O)NC2CC(C)(NC(C3CC(C(F)(F)F)C3)=O)C2)ccc(F)c(F)c1 4631,c1(C(=O)OC(C)(C)C)ccc(-c2nc(C(=O)NCCc3c(C)n[nH]c3)cs2)cc1 4632,C=C(CNC(c1ccnnc1)=O)CCNC(c1cscc1F)=O 4633,c1(C(N2CCC(CC)C2C(=O)N(C(C)CCC(C)C)C)=O)n[nH]c2ccccc12 4634,N1(C(CC2CC(C(=O)OC)C2)=O)CC(OCC(=O)Nc2cc(C)on2)C(O)C1 4635,c1(SCC)cc(C(N2CCCC(NC(=O)Cc3[nH]cnc3C)C2)=O)ccn1 4636,C1(CC)CN(C(C2CCOC2)=O)CC1CC(=O)NCC(c1ccccc1)N(C)C 4637,N1(C(C2CC(SC)C2)=O)CC2CC1CC2NC(c1csc([N+](=O)[O-])c1)=O 4638,c1(C(=O)NC2CCN(CCNC(C(CC)(C)O)=O)CC2)cc(C)cc(O)c1 4639,C(=O)(C1=CCCC1)NC(C1CN(C(C23CCCCC2C3)=O)C1)C 4640,c1(C(=O)NCC(CCC)C(=O)N2CCC2CN=[N+]=[N-])cc2cccnn2c1 4641,C1(=CC(=O)NCC(CN(C(C(C)(C)OC(C)C)=O)C)O)C2CC3CC(C2)CC1C3 4642,N1(Cc2cccc(C(=O)OC)c2)CCCN(C(C2CCCS2)=O)CC1 4643,C1(CC)(CC)CN(C(c2ccc(OC)nn2)C(=O)NCCOC)CCS1=O 4644,C12(NC(c3cc4sccc4[nH]3)=O)CCN(C(=O)C3=CCCSC3)CC1C2 4645,C1(C(=O)NC(C2CC(NC(=O)C(N3C(=O)CCC3=O)C)C2)C)CC(=O)C1(C)C 4646,N1(C(COCCOCCOC)=O)CC=C(CCNC(c2c[nH]nc2C)=O)CC1 4647,CCS(=O)(=O)CCCNC(=O)NC(C)CN1CCCCC1 4648,C1(OC)CC(NCc2nc(-c3ccccc3Cl)cs2)C12CCC2 4649,c1(C(N2CC3N(C(COCC)=O)CC(C3)C2)=O)cn2cc(Cl)cc(Br)c2n1 4650,CC1CCCN(C(=O)CCC(F)F)C1CNC(C1CCN(CC2CC2)CC1)=O 4651,C1(NC(CN2CCN(C)CC2)=O)CN(C(c2ccc(CF)cc2)=O)CC1C1CC1 4652,Cc1cc(=O)n(CCC(=O)NC2(CNC(=O)CN3CC(C)C3)CCOC2)cn1 4653,c1(CC)c(N2CCC(CNC(C3(OC)CCCC3)=O)C2)nc(C)nc1Cl 4654,N1(CC)CCCC2C1CCCN2C(=O)Nc1ccc(CC2CC2)cc1 4655,N1(C(CCC#CC)=O)CCCC(N(C(=O)COc2ccccc2)C)CC1 4656,c1(C(N2CCC(N(C(C(N3CCC(O)CC3)C)=O)C)C2)=O)ccnc2c1CCO2 4657,CCCCCC(F)C(=O)C12CC(C)(C1)CNC(=O)C(C)(CO)NCC2 4658,C1(NC(C=CC=CCC)=O)CN(C(c2cn(C)nc2Cl)=O)C2(CCOC2)C1 4659,Cc1cc(C(=O)NCC(C2CC2)N(C(=O)CC(O)C(C)C)C)cnc1C(F)(F)F 4660,c1(C(N2C(C)CC(NC(COCCC=C)=O)C2)=O)nccc2ncncc12 4661,C1(CNC(c2c(N)cc(Br)cn2)=O)CCC2(CCC2)C1NC(c1cnco1)=O 4662,C#CC1CC2(CC(C(N3CC(NC(c4cc(C)ccc4OC)=O)C3)=O)C2)C1 4663,C1(C(N2C(C(=O)NC(C3CCOCC3)CC)CC2)=O)CCC(=O)N(C)C1 4664,Cc1cccc(C(CCO)NCc2cn(CC(C)(C)[N+](=O)[O-])nn2)c1 4665,CC(C)CC(O)C(=O)NC1CN(C(=O)C=Cc2ccc(SC(F)F)cc2)CC1C 4666,C(=O)C1=CCNC1.C1(C(NOC(c2ccccc2)C)=O)C2CCCCC12 4667,C(=O)(C(F)(CNC(c1n[nH]cc1Cl)=O)C(C)C)N1CCCC(C(C)C)C1 4668,N(C1CCOc2ccc(Cl)cc21)CCC(C)SC.c1(S)nnco1 4669,N1(Cc2c(C)cc(Br)cc2)CCN(C(c2ccc(Cl)s2)=O)C(C#N)C1 4670,c1(C(N2CC(CC)N(C(=O)C(C)OCCOC)CC2)=O)cc(C)c(OC)c(Cl)c1 4671,Cc1ccc(N(C(=O)CC2(C)CCN2C(=O)CNC(=O)C(C)(C)C)C)cc1C 4672,C1(NC(C2CCCCS2)=O)CCN(C(c2ccc(CO)c(Cl)c2)=O)C12CCC2 4673,C1(C)(NC(CN(C2CC(C#N)C2)C(CCc2cnc(C)o2)=O)=O)CCCC1(C)C 4674,c1(C(N2CC(NC(C(CC(C)C)OC)=O)C(C)C2)=O)cc(Cl)c2n[nH]cc2c1 4675,CC1(C)CN(C(C2(CCNC(C3CCC(N=[N+]=[N-])C3)=O)CCCC2)=O)CCCO1 4676,c1(C(N2CCCC3(NC(c4c(N)c(Cl)ccc4)=O)C2C3)=O)cc2cnccc2[nH]1 4677,C=CC1(C(=O)NCC(C)C(F)C(=O)NCCCC(F)(F)F)CCCCC1 4678,N1(C(C2C(c3n(C)ncc3)C2)=O)CC(CNC(=O)COCC(F)(F)F)C(C)(C)C1 4679,N1(C(C2OCCC(C)(C)C2)=O)CCC2(CC1)CC2C(=O)NC1(C)CS(=O)(=O)C1 4680,c1(OCC(=O)N(C)CC2N(C(C(COC)O)=O)CCC2)nc(O)nc(O)n1 4681,c1(CC)nc(C)[nH]c1C(=O)NC(c1ccccc1)CNC(=O)CC1CSCCO1 4682,C(=O)(C1=C(C)C(C)(C)OC1=O)N1C2CC(CNC(C(COC)(F)F)=O)(OC2)C1 4683,C1(C(N(CCCC=C)C)=O)(NC(c2snnc2CC)=O)CCCC1C 4684,c1(C(=O)NC2CN(C(c3cc(C(C)=O)oc3)=O)C(C)C2)ccc(N)cc1Cl 4685,C1(F)(C(N(CCNC(C(C)C(=O)N(C)C)=O)CCOC(C)(C)C)=O)CCS(=O)(=O)C1 4686,C(=O)(CC(C)C(=O)NCC1CC(O)CN1C(=O)Cc1ccnc(C(F)(F)F)c1)OC 4687,N1(CC(N2CCN(Cc3ccc(C)cc3)CC2)=O)CCCC2(CCCCO2)CC1 4688,CC1CCC(C(=O)NOCC2CCCC2)CN1C(c1csc(CO)n1)=O 4689,c1(C(N)=O)cccnc1CNC(C1CCN(c2ccccc2F)C1=O)=O 4690,CC(C)P(=O)(CC(=O)NC1CC2CCC1(NC(=O)CCn1ccnc1)C2)C(C)C 4691,n1(C(CC(N2CCC(N(C(CC)=O)CC)C2)=O)C)nc(C)cc1C 4692,c1(C(N(C(CC)C(=O)OC)CC)=O)cc2sc(C)cc2[nH]1 4693,Cc1cc(C(=O)NCCC2CCCN2C(C2CCCCS2)=O)ccc1C(F)F 4694,Cc1ccc(C(=O)O)c(-n2cc(CNC(C3(CO)CCCO3)=O)nn2)c1 4695,CN1CCCC(C(N2CCCCC2C(=O)NCC(O)CCO)=O)C1 4696,C(C(Cl)C(C)(F)F)NC(CC1(N(C(Cc2cn(CC)nc2)=O)C)CC1)=O 4697,N1(C(Cc2scc(CC)n2)=O)CCOC(C(=O)NC(C)CCSC)C1 4698,N1(C(C2CCN(C)C(=O)C2)=O)CCN(C(=O)CC2CS(=O)(=O)C2)CC12CCC2 4699,C(=O)(C(C)(C)C(C)(F)F)N1CCN(C)C(CNC(C2CC23CCC3)=O)C1 4700,Cc1cc(CC(=O)NC2(CCNC(C3CCN(C(N)=O)CC3)=O)CCC2)n(C)n1 4701,N1(C(c2c(-c3cn(CCCN(C)C)nn3)cnn2C)=O)CCc2ncccc2C1 4702,n1(CC(=O)NCCCCCCNC(C2CC2CF)=O)nnc2ccccc2c1=O 4703,C(C1=CCN(C(=O)CC(O)CNC(=O)CC2CCOC2C)CC1)OC 4704,N1(C(CC=C)=O)CCC(O)CC1C(=O)Nc1cscc1C 4705,c1(C(=O)NC(CC#C)C(=O)NC2CCCN(C)C2C)ccc2[nH]ccc2n1 4706,C1(CC(=O)NCC2COCCN2C(c2cc(CF)on2)=O)CN2CCN1CC2 4707,c1(C(=O)NCCCOCCC(=O)NC(CCCCCC)C)cc2cccn2cn1 4708,CCC(C(=O)NCCNC(=O)CC1CCC(C)(C)CC1)C(F)(F)F 4709,c1(C(N2C(C)(C)C(O)CC2)=O)nc(=O)c2ccccc2s1 4710,c1(C(=O)NCCCCNC(c2cncs2)=O)cc(O)nc2ncccc12 4711,C1(CNC(CSCC(=O)OC)=O)CCCC(CNC(C2(C)CCC(=O)N2)=O)C1 4712,N1(C(CN(C(c2csc(Cl)c2)=O)CC)=O)CCCC(O)C1C 4713,C1(NC(COc2cccc(C)c2)=O)CCN(C(c2nccs2)=O)C12CCCC2 4714,C1(C(=O)OC)CS(=O)(=O)C2CN(C(=O)NCC3C(C)(C)CCCC3(C)C)CC12 4715,C1(Cn2cc(CC(C)O)nn2)CN(C(=O)Cn2ncnn2)CCO1 4716,CC1CCN(C(=O)CCCCNC(N)=O)CC1NC(C1CCC(=O)N1C)=O 4717,C(N=c1[nH]c2c(c(=NCC3CCCO3)[nH]1)CC(C)CC2)c1c(OC)cccc1 4718,c1(CC)cc(C(N2CC(C)(C(N3CCC(C(CC)CC)C3)=O)C2)=O)no1 4719,C1(NC(C2C(C)(C(F)F)C2)=O)CC2CCC(C1F)N2C(=O)CC1(C#N)CC1 4720,N1(C(c2cnc(C)c(N)c2)=O)CCCC2CN(C(=O)C3=CCN(C)C3)CC12 4721,C(=O)(CC(C)(C)C(=O)OC)N1CCCC(C(=O)NC2CCN(CCC)C2)CC1 4722,C(=O)(C(C)(C)C(C)C)N1CCC(N(C(=O)CN2C(C)CCC2C)CCC)C1 4723,N1(C(C2C(C(=O)OC)C2)=O)CCC2C(NC(c3cnn(CCF)c3)=O)C12 4724,c1(C(=O)NC(CCCNC(c2c(C)ccnc2O)=O)C)cnn2cc[nH]c(=O)c12 4725,C(=O)(C(CC)C(C)(C)CC)NC1CCN(C(c2cc(CC)cc(C)c2)=O)CC1O 4726,N1(C(C2OCCN(CC)C2)=O)CCCC2(C1)C(NC(=O)CC(C)(F)F)CCN2C 4727,c1(C(N2C(CN(C(=O)CC(C)CN(C)C)CC)CCC2)=O)cc(N)nc(Cl)c1 4728,N1(C(CCS(=O)(=O)NC)=O)CC2OCCN(C(=O)Cn3ccc(C)n3)C2C1 4729,c1(CN2CCC(N3C(=O)CCC3=O)CC2)nc2cc(Br)ccc2o1 4730,c1(CCC(=O)NCC(C2CC2)NC(C2CC(N(C)C)C2)=O)cc(F)cc(F)c1 4731,c1(OCC)nccc(C(=O)NCCCCCCNC(c2cnncc2O)=O)c1F 4732,CC(C)CC(CNC(=O)COCCF)C(=O)N1CCC(CC2CC2)C1 4733,N1(C(CCNC(=O)OCC)=O)CC(NC(C2C(C)(C)C2(F)F)=O)CC(C)(C)C1 4734,C1(C(N2CCC(CN(C(=O)Cc3ccc(Cl)nc3)C)C2)=O)CCC2CC1C2(C)C 4735,C(C)(C(C(=O)NCC1CCN(C(C)C)C1)C(C)C)NC(c1cn(CCC)nc1)=O 4736,CC1CCN(C(=O)C(C)C2CCOC2)CC1NC(=O)C=CSc1ccccc1 4737,C12(CNC(CCCCCN(C)C)=O)CCCC1CN(C(=O)COCP(C)(C)=O)C2 4738,N1(C(CCC(C)(C)N(C)C)=O)CC2(CCC2)CC1C(=O)NC1CCOC1(C)C 4739,Cc1ccnc2sc(C(N3C4CCC3CN(C(=O)COC(C)C)C4)=O)c(C)c12 4740,O=C(CN=c1nc(N2CCC(CO)C(F)(F)C2)c2c([nH]1)COC2)NC1CCCC1 4741,C1(NC(C2CC(S(C)(=O)=O)C2)=O)COC2CN(C(C3CC4C(C3)C4(F)F)=O)CC12 4742,c1(NC(c2nc(C)cs2)CC)nc(C)cc(=NCc2cccc(O)n2)[nH]1 4743,c1(CNC(C2N(C(c3cncc(CC)c3)=O)CCC2CC)=O)cccc(C)c1O 4744,Cc1cc(C)nc(N(C2CCCNC2)C(C2CCC(=O)NC2)=O)n1 4745,N(C1CCOc2c(F)cc(F)cc21)C(C(C)Oc1ccccc1CC(=O)O)=O 4746,c1(C(N(C2CCCCN(C(C(C)S(N)(=O)=O)=O)C2)C)=O)csc(=NC2CC2)[nH]1 4747,N1(C(c2c(Br)ncn2C)C(=O)NCC)CCCC2(C1)CC2(F)F 4748,C1(C(N(CC(=O)NC)C)=O)(OC)CCN(C(C2C(C)C2C)=O)C1 4749,S(=O)(=O)(c1cccc(Cl)n1)SCCC(N1CC(c2ccccc2)(O)C1)=O 4750,C1(C(=O)NCCC2CN(C(C3(S(N)(=O)=O)CC3)=O)C2)CC2CCC1C21CC1 4751,n1(CC)ncc(C(=O)NC2(CNC(=O)C(C)C#N)CCOC2)c1C 4752,CC(C(=O)NC1CCCC1)NC=O.C1(c2nc[nH]n2)(NC(C=CC)=O)CCC1 4753,Cc1cc(C(N2CCOC(C(N(CCCc3ccccc3)C)=O)C2)=O)nn1C 4754,C(=O)(C1=CSCCO1)NC(CCN(C(c1c(C)nns1)=O)C)C 4755,C1(C)(CC)CC(NC(=O)Cc2cc(C)[nH]n2)CN1C(C1(NC(N)=O)CC1)=O 4756,n1(CC=C)c(N(CC(C)CC)C)nnc1C1COc2ccccc21 4757,CC1CC(C(=O)N2CC(O)(C(C)(C)CNC(C3CCCC34CC4)=O)C2)=NO1 4758,C1(NC(c2c(CC)cccc2)=O)C2CC1N(C(=O)C(=O)NC1CC1)C2C 4759,C(CN=c1cc(F)nc[nH]1)(c1ccccc1F)NC(C(C(C)C)C)=O 4760,N1(C(c2ccccc2Br)C(=O)Nc2ccc(Cl)cn2)CCC2(C1)OCCO2 4761,C1(C(CC)C)CN(C(=O)C(=O)NC2CC(C(C)OC)C2)C1 4762,c1(C(N2C3CN(C(C(CC)C(C)O)=O)C(C3)C2)=O)onc2ccccc12 4763,C12(NC(C(C)n3ccnn3)=O)CCC(F)(F)CC1CN(C(=O)C(C)(C)CF)C2 4764,C1(C(=O)NCCN(C(C=CC(CC)OC(C)=O)=O)C)CCC(NC(C)(C)C)CC1 4765,c1(NC)ccc(C(N2CC3CCCC23)=O)cc1[N+](=O)[O-] 4766,C(=O)(C1CCc2cc(F)ccc21)NC1(C)CCN(c2cc(CC)nc(Cl)n2)C1 4767,c1(CC(N2CC(NC(c3n[nH]cc3Br)=O)C3C2C3)=O)cccc(F)c1O 4768,c1(COC(C(c2cc(F)cc(F)c2)C)=O)ccc2c(c1)C(=O)NCC2 4769,C1(CC(=O)NC(C#C)C(C)C)N(C(=O)CC2CCC(C)CO2)CCC1(C)C 4770,N1(C(C(=O)NCC(F)F)=O)CC(O)CC1CNC(C1CC2(CSC2)C1)=O 4771,CC(C)(C)CCCC(=O)NC1CCC(NC(=O)CCc2c[nH]c3ccccc23)C1 4772,C1(C(N2CCC(OCC)C2)=O)CC2(CC2)CN1C(=O)C(=O)C(C)CC 4773,CC1(C(=O)NCC2(NC(c3ccsc3Br)=O)CCC2)CCCC1 4774,N1(C(c2n[nH]c(C)c2C)=O)CC(NC(=O)C(CC2CC2)CC2CC2)CCC1C 4775,Cc1cc(C(N2CCC(N(CCO)C(C3(C)CCC(=O)NC3)=O)C2)=O)ccc1F 4776,N1(C(C(SC)SC)=O)CCCCC(N(C)C(c2ccc(F)c(F)c2)=O)C1 4777,c1(OC)cc(C(=O)NCCNC(c2c(C3CC3)cnn2C)=O)cc2cn(C)nc12 4778,C(CCCCC(=O)N(C)C)c1cn(CC(=O)NC2CSC2)nn1 4779,N1(C(C2C(C)(C)C2CNC(C2CC2C(F)F)=O)=O)CCC2(CC1)CSC2 4780,C1(CNC(=O)NCCC2CCCS2)CCCN(c2ccccn2)C1 4781,c1(OC)ccc(CNCCCCC2CC2C)cc1C#N 4782,C=C(C)C1OCCC1C(N1CCC(C(=O)NC2CCN(C)C2(C)C)(C(C)C)C1)=O 4783,C1(C(=O)OC2CC(C(=O)O)OC2)C2CCC1(c1ccc(OC(F)(F)F)cc1)C2 4784,c1(OC)cccc2[nH]cc(CC(=O)N(C)CC3(O)CCC(F)(F)CC3)c12 4785,C(=O)(C(F)(F)C(F)(F)F)N1CCC(N(C)C(c2cc(C(F)(F)F)ccc2O)=O)C1 4786,C=CCC(C)(C)CNC(=O)C(C1CC1)NC(=O)CC1CCCCN1C 4787,CC1C(NC(=O)Cc2cnsc2)CC2CCC1N2C(=O)C(F)(F)c1cnccn1 4788,N1(C(c2c(C)n[nH]c2)=O)CCN(C(=O)C=CC=CCO)CC1c1ccnn1C 4789,N1(C(CC(CN(C)C)(C)C)=O)CC2CCCCC2(NC(C2OCCC2(C)C)=O)C1 4790,c1(C(N2CCC23CC(C(C)(C)C)C3)C(=O)NCCC)cc(OCC)cc(CC)c1 4791,c1(N2CCC(CC(C)CO)CC2)c[nH]c(=N)nc1C(F)(F)F 4792,C(c1cc(Cl)ccc1Cl)=CC(N1CCN(C(C(C)(C)OC)=O)CC1)=O 4793,C1(C(N(C2CCN(c3nc(C)nc(O)c3C)C2)C)=O)CCC2(CC1)CC2(F)F 4794,c1(CNC(C(CO)NC(C2C(C)CC2)=O)=O)ccc2c(c1)CC2 4795,C(C(C(=O)NC1CCCC1)N(C1CCC1)CC1CC1)(C1CCC1)OC 4796,CCC(C)CC(=O)C(=O)NC(C1CC1C(=O)NCc1ccc(C2CC2)o1)C 4797,C1(CNC(C(C(C)(C)C)SC)=O)CC12CCN(C(c1cscc1C(N)=O)=O)CC2 4798,c1(N(C(C)=O)C)ccccc1C(=O)N(CC(C)CNC(C1CC(N=[N+]=[N-])C1)=O)C 4799,CCCCC(C)CCC(=O)NC1COCC1NC(c1cc(Br)cs1)=O 4800,CC1CN(C(=O)Nc2c(Br)cc(F)cc2Br)CCC1(O)C(F)(F)F 4801,C(c1ccc(Cl)c([N+](=O)[O-])c1)=CC(=O)NC1CC2CC1CN2 4802,C(CCCCCNC(=O)COc1ccsc1)NC(c1c(C)snn1)=O 4803,c1(C(N(C(C)C(=O)N(CC(F)Cl)C)CCC)=O)cc(C#N)cs1 4804,C(c1cncn1C)=CC(=O)N(CCC(=O)N(CC(O)C1CCC1)C)CC 4805,N1(C(C(COC)NC(C)=O)=O)CCC2CC1CN2C(c1cccc(C)n1)=O 4806,c1(SC)ccc(C=CC(=O)NCC2CC(NC(=O)CCNC(C)=O)C23CCC3)s1 4807,C1(C(=O)NCC2(C)COCCO2)CCC2(CCNC2)CC1 4808,CC(C)C(CC(=O)NCC(F)CNC(c1cocn1)=O)c1ccccc1 4809,CCC(CC)CC(F)C(=O)NC1CC2CC1N(C(c1cscc1C(N)=O)=O)C2 4810,Cc1cccc(NC(=O)NCC(c2ccc(C3CC3)cc2)(C)C)c1F 4811,C1(CNC(COCC)=O)CN(C(C2(CC(C)=O)CC2)=O)CCC1(C)C 4812,C1(CC(=O)NCC(C)(C)OC)CN(C(C2CC(C)=NO2)=O)CC12CC2 4813,c1(CNC(CC2(CC)CCC2)=O)cc(C(=O)N(C2CC2(C)C)C)on1 4814,CCCCC(C(=O)NCc1ocnc1CC)NC(c1cc(C)c(C)[nH]1)=O 4815,c1(CCNC(C=CC(C)(C)NC(c2cc(O)cs2)=O)=O)ccncc1F 4816,C1(NC(C(CCC)C)=O)CCC(C)N(c2nccc(C)c2C(=O)OCC)C1 4817,CCC(C)CC(CO)NC(=O)CC(CC)N(C(=O)CC1CC(=O)NC1=O)C 4818,Cc1nc2ccc(NC(C3CC(F)CN3c3ncnc4sc(Br)cc34)=O)cc2o1 4819,C(=O)(C(F)CCC(C)C)NCC1N(C(CC2CCC(OC)CC2)=O)CC1 4820,Cc1n[nH]c(=NC2CCCC(NC(c3cnn(C4CCCC4)c3C)=O)C2)s1 4821,c1(C(=O)NCCCC2N(C(c3c(CC)c[nH]n3)=O)CCCC2)c[nH]cc(C)c1=O 4822,N1(C(C(=O)OC)c2nc[nH]n2)CCCCC1c1ncc[nH]1.CCCCCCN 4823,C1(NC(CCCC(C)C)=O)CCN(C(c2cc(O)cc(=O)o2)=O)C12CCCC2 4824,C1(CNC(C=CCN(C)CC)=O)CC12CCN(C(C13CCC(CO1)C3)=O)CC2 4825,c1(C(N2CCOC(C3CCOCC3)C2)=O)[nH]cc2c1CCC2 4826,c1(C(=O)NCC2C3CN(C(CCCCCC)=O)CC32)cc2n(n1)C(C)CCC2 4827,c1(OC)c(C(=O)NC(CNC(=O)CC2(N(C)C)CCC2)C(C)(C)C)cnn1C 4828,c12cc(ccc1Br)OC2=O.c1(CNC(=O)OCC)cn(CCCO)nn1 4829,N1(C(C(C)SC)=O)CCC(F)(F)C(CNC(C2(C)CC(C)(C)C2)=O)C1 4830,C1(NC(C2CC3CCC2C3)=O)CC2CCC1N(C(=O)CN1CCCS1(=O)=O)C2 4831,C1(CNC(C(CC)N(C)C)=O)CC2COCC2N1C(c1cc2cccnc2s1)=O 4832,C12(CNC(c3ccc(O)nc3)=O)CCC(CN(C(=O)C=Cc3cscn3)C1)C2 4833,N1(C(C(CCCC)O)=O)CC(NC(c2ccncc2)=O)C2CCCC12 4834,c1(C(N2C3CN(C(c4c(CC)scc4)=O)C(CC3)C2)=O)ccnc2c1CC(=O)N2 4835,c1(C(N2CCOCC(NC(CC3(CSC)CC3)=O)C2)=O)cc(O)cc(C#N)c1 4836,C=CCC(C(=O)N(C(C)CCNC(C1(n2cccn2)CCCC1)=O)C)C(C)C 4837,C(CC(C)C(=O)NCC1CCN1C(=O)CN1CCCCC1)OC 4838,C1(CC(=O)NCc2cn(CC(F)(F)F)nn2)OCCCO1.C12CC(C1)CS2 4839,CC1CN(C(c2c(F)cccc2Cl)=O)CCN1C(c1ccc(C2CC2)cc1)=O 4840,N1(C(C2(C)CC2)=O)CCOCC12COCCN(C(C1C3CCCCCCC13)=O)C2 4841,N1(C(C=Cc2ccc(C)nc2)=O)CC2(CCN(C(=O)CC3CCOC3C)C2)C1 4842,C(CCCCC(=O)NC1CCC(CCC(=O)N(CC(C)C(=O)OC)C)C1)SC 4843,c1(C(=O)NCC(C)=CC(=O)NCCN(CC(C)(C)C)C)cnc(C)c(C)c1 4844,CC(C(F)(F)C(F)(F)F)NC(=O)Nc1ccc(Br)c(Cl)c1 4845,S(=O)(=O)(c1ccc(SCCNC(c2ccc(CC(=O)O)cc2)=O)cc1)NC(C)C 4846,c1(OC)ncc(C(=O)NCC2(C(=O)NC3CCCCC3)CCC2)cc1Cl 4847,CC(C)CCCCCC(=O)NCC12CCCCC1N(C(=O)C1=COCCO1)CC2 4848,n1(CC(=O)NC(c2cnn(C)c2)C(=O)NCCC2C(C)C2)[nH]cnc1=N 4849,C(=O)(CCCC(N)=O)N(C(C)CCNC(=O)CC1CN(C)C1)C 4850,CCCCCC(O)C(=O)N(CC(N1CC(c2cc[nH]n2)C1)=O)CC1CC1 4851,c1(OCC)cc(NCc2ccc(CNC(c3cscc3Cl)=O)cc2)ncn1 4852,c1(N(C)Cc2nc(C)[nH]n2)nc(NCN2CCNC2=O)c2ncn(C(C)C)c2n1 4853,C(=O)(C(O)C(F)(F)F)NCC(C)(C)NC(c1cn(C)c(O)n1)=O 4854,c1(N2CCC(C=C)CC2)nc2c(c(=NCC3CCC=CCCC3)[nH]1)CCC2 4855,c1(C(N2CCCC(C(c3c(C)nc(C)s3)=O)C2)=O)c(C#N)c(C(F)(F)F)nn1C 4856,C1(C(CC)NC(CCC=C)c2nnnn2CC2CC2)CCC(F)(F)CC1 4857,c1(CC(N2CCC(F)(COC)C2)=O)cccc2ccccc12 4858,C(=O)(CC1OCc2ccccc21)NCC(C)NC(c1n(CC)nnc1)=O 4859,C1(C(=O)OC)CC2CC(NC(=O)Cc3cnc(C)nc3O)C2C1 4860,C(CC(=O)NC1CCC(CNC(=O)C(C)CC2CCC2)C1)(OCC)OCC 4861,N1(C(C2C(C)(C)CO2)=O)CC2CC(NC(=O)CCCC3CCCCC3)CC2C1 4862,c1(C(=O)NCCN(C(c2[nH]nnc2C(F)F)=O)CC)cnc(O)n1CC 4863,N1(C(CCOCCCOC)=O)CCC(C(F)F)(CNC(c2sccc2Cl)=O)C1 4864,Cc1noc(N)c1C(N1CCC(NC(c2csc(C(F)(F)F)c2)=O)C1)=O 4865,c1(C(=O)NCC(C)NC(c2ccc(Oc3ccccc3)cn2)=O)nnc(S)n1C 4866,N1(C(CC(CC)C2CC2)=O)CC(NC(C2CCN(OC)CC2)=O)C2(CC2)C1 4867,CC1CC(c2cn(-c3ccncc3)nn2)CCN1CC(N1CCC(O)CC1)=O 4868,C1(C(=O)NC2CN(C(Cc3cccc(C#N)c3)=O)CC2O)CCc2ncnn2C1 4869,S(=O)(=O)(c1cccc(C(=O)NCCc2ccc3ccccc3c2)c1)N(C(C)C)C 4870,C12(OC)CN(C(=O)Cc3ccnc(C(=O)OC(C)(C)C)c3)CC(C(=O)O)(C1)C2 4871,N1(C(C(CC)(C)OC)=O)CCCC(CC)(NC(=O)CCc2ccccc2F)C1 4872,CC(C)S(=O)c1ccc(C(=O)NC2CN(C(c3c[nH]c(=N)o3)=O)CC2O)cc1 4873,N1(C(c2c(N)sc(C)c2C)=O)CCC(C2CC2)C1CNC(=O)C(O)C1CC1 4874,n1(CCC(=O)NCC2COCCN2C(C2CCC2)=O)cc([N+](=O)[O-])cn1 4875,c1(C(=O)OC)ccc(S(=O)(=O)NC2CCCN(C(c3cncs3)=O)C2)cc1 4876,C1(CC=C)(NC(=O)CC(O)CCSC)CCCN(C(c2ccc(CSC)o2)=O)C1 4877,N1(C(C=CC=CCC)=O)CC2OCC(NC(=O)CCCCCCC)C2C1 4878,c1(C(N2CCC(C(N(CCOC)C(C)C3CC3)=O)CC2)=O)nccc2ccccc12 4879,CC1CN(C(=O)C(CC(N)=O)NC(c2cnc(O)o2)=O)C(C)CO1 4880,c1(NC(C2(CC)CN(C(=O)CC3CCCCO3)C2)=O)cccc2cccnc12 4881,c1(C(N2CC(C(C)NC(c3cnn(C4CC4)c3)=O)OCC2)=O)cc2cscc2s1 4882,c1(C(N2CCCCC(NC(C(CC)(F)F)=O)C2)=O)cc2c(cn1)NC(=O)CO2 4883,C(CC)(CCCC(=O)NCC(C)(C)CCOC)NC(c1cnc(CC)o1)=O 4884,c1(C(N2CCCN(S(=O)(=O)c3cccs3)CC2)=O)noc2c1CCCC2 4885,C(CC(C(=O)NCCc1ccncc1)NC(=O)C1=NOCC1)OCC 4886,Cn1cc(C(=O)NC2CCCN(C(=O)CCC3CCCCC3)C2)c(O)nc1=O 4887,c1(OCC(=O)NC2(CNC(CSC)C)CCOC2)cc(C)ccc1Cl 4888,CC1CCC(C)(C(N2CCCCC2CNC(=O)Cc2cccnc2F)=O)CC1 4889,c1(NC(C)=O)ccc(C(=O)NC2CCN(C(=O)C(F)(Cl)c3ccccc3)C2)cc1 4890,c1(NC)ccccc1C(=O)N(C(C)(C(=O)NCc1cncc(OC)n1)C1CC1)C 4891,C1(C(N(C2CCN(C(C(CC)(C)O)=O)CC2)C)=O)CC(C(C)C)=NO1 4892,c1(-c2n(CC(CC)CC)nc(CS(C)(=O)=O)n2)ccc(C)c(Br)c1 4893,Cc1c(Cl)cc(C(N2CCC(N3CCC(C(=O)OC(C)(C)C)C3)CC2)=O)cc1Br 4894,CCS(=O)(=O)c1ccc(C(N2CCC(C(F)F)C2)=O)cc1 4895,C12(C(N(C)Cc3ccnn3C)=O)CC1CCN2C(=O)Cn1cnnn1 4896,N1(C(c2ccc(CCC)[nH]2)=O)CCC12CN(C(=O)CSC)C2 4897,c1(NC2(CNC(C3N(C(C)C)C(=O)CC3)=O)CC2)ncc2ccccc2n1 4898,c12ccc(cc1)C(CCC)(C)NN2CC.C1(C)CC1(Br)Br.CC 4899,CCCCC(CC(=O)N(C(C)CC(C)CC)C)NC(=O)CC1(C)CC1 4900,N1(C(C2(C)CC(OC)(OC)C2)=O)CC2(CCC(CNC(=O)C(O)C(C)C)O2)C1 4901,c1(C(N(C(Cc2ccc(O)cc2)C(=O)O)C)=O)cc(C(F)(F)F)cnn1 4902,C1(NC(C=CC(C)C)=O)CCCCN(C(=O)CC2CCCC(C)(C)O2)C1 4903,c1(OCC)ccc(C)nc1C(=O)NCC(F)CNC(C1CC1C(F)(F)F)=O 4904,c1(C(N2CCCC(CN(C)C)C2)C(=O)NCCCF)cc(Br)ccc1F 4905,c1(OCC(N2C(C3(NC(c4c(C)con4)=O)CC3)CCC2)=O)c(C)cccc1Cl 4906,C1(CC(=O)N(CCCNC(=O)CCn2ccnc2)CCO)CCCCCC1 4907,C1(F)(CNC(C(c2cccc(C)c2)F)=O)CCCN(C(c2snnc2C)=O)CC1 4908,N1(C(=O)NC)CCC(C(N2CCCC(CNC(=O)CSC(C)C)C2)=O)CC1 4909,CN1CCN(C)C(C(=O)NC2CCC2CNC(=O)CC#N)C1 4910,c1(C(=O)NC(C(C)NC(C2CCS(=O)(=O)C2)=O)(C)C)ccnn(C)c1=O 4911,CC1(C(N2CCCC(NC(c3coc(CC4CC4)n3)=O)C2)=O)CC2(CCC2)C1 4912,N1(C(C2(C)ON=C(C)C2)=O)CCN(C(c2cnc(O)n2C)=O)C(CC2CC2)C1 4913,N1(C(C(C=C=C)C)=O)CC2CCN(C(c3cc(CC)oc3C)=O)CC2C1.[SH](C)(=O)=O 4914,c1(C(N2CC3C(NC(c4n(C(C)C)cnc4)=O)C3C2)=O)c[nH]c2cccnc12 4915,N1(C(c2cnc(C)o2)=O)CC2CCC(NC(c3cccc(F)c3Cl)=O)CC2C1 4916,Cn1c(C(N2CC(F)(F)CC2CCNC(C2CC3(CC3)C2)=O)=O)cccc1=O 4917,c1(NC(C2CC(F)CCN2C(C2C3CCC(C3)C2C)=O)=O)ccc(CO)cc1O 4918,C(=O)(C(O)CC[S+](C)C)N1CCC(NC(c2c(C)oc(C(C)(C)C)c2)=O)C(O)C1 4919,C#CCC(C(=O)N1CCC(N(C(=O)CN2CCC(C)(O)C2)CC#C)CC1)C1CC1 4920,C1(CC(=O)NC2C(CNC(CN3C(=O)CSC3)=O)CCC2)CC(O)C12CCC2 4921,C1(C(=O)NCC=CCNC(C(N2CCC(O)CC2)C)=O)CCCC(CF)C1 4922,Cc1cc(C(=O)NC2(c3ccccc3)CN(C(=O)C=C3CCOCC3)C2)n[nH]1 4923,C1(C(=O)NCC2(C(=O)NC(c3ccncc3)C)CC(C)(C)C2)CCC(C#N)CC1 4924,C1(C(N2C(CN(C(=O)CC3CCC34CCC4)C)CCC2)=O)CCC2(CC1)CC2 4925,N1(C(CS(=O)(=O)NC)=O)CCCC(N(C(=O)Cc2cnc(C)s2)CC)CC1 4926,C(=O)(CCCCCN=[N+]=[N-])NCCC1(OC)CN(C(C2CCN(C(C)C)C2)=O)C1 4927,Cc1nn(C)c(C)c1CC(C)C(=O)NC(C)CN(C(=O)CN1CCCCCC1)C 4928,c1(C(C)C)conc1C(=O)NC1(CNC(=O)CC2(C#N)CC2)CC1 4929,n1(CC)cc(C(=O)NC(C)C(C)NC(c2cc(C(F)(F)F)ns2)=O)nn1 4930,c1(C(=O)NC2(C)CC(NC(c3noc(CC)c3C)=O)C2)cc2n(c1)CCC2 4931,c1(C(=O)NCCN(C(C2CC(CN(C)C)C2)=O)CC)ccc2nc[nH]c2n1 4932,N1(C(C2CN(C(C3CCN(CC)C3)=O)CC23CCC3)=O)CCCC(N=[N+]=[N-])CC1 4933,CCCCC(O)C(=O)NCCN(C(c1ccc(OC)cc1F)=O)C(C)C 4934,N1(C(CCc2n(C)ncc2)=O)CCOC(CCNC(C2CC2(C)C(F)F)=O)C1 4935,c1(CC)ccc(NC(=O)C(c2cccnc2F)(C)C)cc1Cl 4936,Cc1cc(C)c(C(=O)NC(C)C(C)NC(c2coc(N(C)C)n2)=O)cc1N 4937,CC(O)CC(C)(C)CNC(C1CCN(C(C2CC2Cl)=O)CC1)=O 4938,C12(NC(CC3(C)CC3)=O)CC3CC(C1)CC(NC(C1CCCC(O)C1)=O)(C3)C2 4939,Cc1cc(O)cc(C)c1CC(=O)NCC1(CNC(=O)Cc2ccccn2)CCC1 4940,c1(C(=O)NCC=C)cccc(S(=O)(=O)NC(C)CNc2cccnc2)c1 4941,CC1CCCCC1(CNC(=O)CCn1ncn(C)c1=O)NC(C1CC(=O)N1)=O 4942,c1(NCC(=O)NCC2CC2)cccnc1.C1(C(N(C)C(=O)C2CC2)=O)CCCS1 4943,N1(CC(=O)N(C)CC2CC2)CC(=O)NCC1CCCCN=[N+]=[N-] 4944,N1(C(C(CC=C)C)=O)CCCCC(NC(c2ccc(N3CC=CC3)cc2)=O)CC1 4945,C1(NC(CCC2N(C)CCC2)=O)CN(C(=O)CCc2ccc(=N)[nH]c2)CC12CCC2 4946,N1(C(c2cncc(C#C)c2)=O)CCC2CCN(C(c3nc(C)ccc3F)=O)C2C1 4947,c1(C(=O)NCC(CC)(C)NC(=O)C(C)NC(=O)COC)cc2cncn2c(O)n1 4948,CCCCS(=O)(=O)NC(C)C(N1CC(N(C)C(c2[nH]ccc2C)=O)C(O)C1)=O 4949,N1(C(CNC(CCCCC)=O)=O)CCN(C(=O)C(C)CO)CC1C(F)F 4950,C(=O)(CC(C)(C)C(F)F)N1CC(C2CN(C(CN(C(C(C)C)=O)CC)=O)C2)OCC1 4951,C1(NC(C(C)C2CCC2)=O)CCOC(C(=O)NCC2(CN(C)C)CC2)C1 4952,C1(C(=O)NCc2nc(C)sc2)C=CCN(C(=O)C(F)CC2CCOC2)C1 4953,N1(CCNC(C)C(=O)N(C(=O)CN2CCCC2C)C)CCCOCC1 4954,N1(C(C2(CCC=C)CN(C(=O)CC=CC)C2)=O)CC2CCC1C(O)C2O 4955,c1(C(N2CCC(CCNC(c3c(C)ccs3)=O)C2)=O)nc2c(s1)COCC2 4956,C(=O)(C1CCC(NCCCN2CCOCC2)c2ccccc21)OC 4957,Cc1ccc(O)cc1C(N1CC2CC(C1)N2C(c1nc(Cl)ccc1F)=O)=O 4958,N1(C(C(C#C)(C)C)=O)CCC2C(C1)CN2C(C1CC2(CCOCC2)C1)=O 4959,N1(C(=O)NC(C2CCOC2)C#C)CCCC2(CCCO2)C1 4960,CCCCC(C)C(=O)NCC12COC(CNC(=O)CC3COC(C)(C)CO3)(C1)C2 4961,C1(CC)(NC(=O)C=CSCc2ccco2)CN(C(=O)CNC(c2ccoc2)=O)C1 4962,c1(CN(C(c2cccc(O)c2)C)C(=O)C2CC2)ccc(Br)c2nsnc12 4963,c1(C(N2C3(C(=O)NC4C(OC)C(O)C4)CC3CC2)=O)cccc(F)c1F 4964,c1(COC)cc(O)nc(CNC(C2(CNC(=O)CC3CCCC3)CC2C)=O)n1 4965,c1(OC(C)C)ccc(C(=O)NCCCN(CCO)C(c2cn(C)nc2Cl)=O)cc1 4966,N1(C(C=CC)=O)CCCC(O)(CNC(=O)C(F)(F)CC2CCCO2)C1 4967,c1(C(=O)NCCSCC)n[nH]c2c1CN(C(c1ncc(C)cc1F)=O)C2 4968,CC1CC2(CCN(C(=O)C(C)n3cncn3)CC2)CN1C(=O)Cc1ccncc1 4969,c1(C(=O)NC2C(NC(c3c(Cl)nc(OC)s3)=O)COC2)ccc(=O)n2c1CCC2 4970,C1(=O)C2=C(C)N(C(=S)NC2c2cc(I)ccc2Br)C12CCOCC2.C(=O)OC 4971,C1(C(=O)NCCC(CCC)C2CC2)CC2(CCC2)CN1C(=O)CC1CCCSC1 4972,C(C)(CCN=c1c(Cl)c[nH]cc1[N+](=O)[O-])NC(CCCc1cc(C)no1)=O 4973,c1(NC)ncccc1C(=O)NCC(C)(C1CC1)NC(c1ncc(OC)cn1)=O 4974,c1(C(=O)NCC2(C)CCN(C(C(C=C)(C)O)=O)C2)cc(C)nc2c1cnn2CC 4975,C(=O)(C1CCCn2nccc21)NC1C(C)C2CCC(C1)N2C(C1CC1(C)Br)=O 4976,N1(C(=O)OCC)CCCCCC1CNCc1ccc(C)nc1OCCO 4977,C(C)(CCC(C)C)N(C)CCN(C)CC.CC(=CCSC)OC 4978,N1(C(CC(C)CNC(C2(C)CC(C#N)C2)=O)=O)CC2CN(C)CC2C1 4979,c1(CNC(C2OCCN(C(CCCN(C)C)=O)C2)=O)ccc(F)c(O)c1 4980,c1(NC(C)CCC(F)(F)F)[nH]c(=NC2CSc3ccccc32)nc2sccc12 4981,CC(CN(C)C)CC(=O)N1CCC(NC(c2cccc(C(=O)NC3CC3)c2)=O)C1 4982,C1(C2CCN(C(=O)C=Cc3ccc([N+](=O)[O-])s3)C2)(NC(CCSC)=O)CC1 4983,CC(=O)CCCC(=O)N1CC(N(C)C(C2CCCN2C(=O)OC(C)C)=O)C1 4984,C1(NC(=O)NC2CCC3(C(=O)OC)C2C3)CCC2OCCC2C1 4985,C12(NC(c3cncc(Cl)c3)=O)CCCCC1CN(C(C1CC(O)C1)=O)C2 4986,CN1CCOC2CN(C(C3(CNC(=O)C(=O)NC4CC4)CC=CC3)=O)CC12 4987,C1(C(=O)NCCC2CN(C(=O)CC3CCC4(CCC4)O3)C2)CC2C=CCC(C1)C2 4988,c1(C(=O)NCC2CN(C(CCC(C)C)=O)CC2C)cn2c(n1)C(C)CCC2 4989,C1(C)(NC(c2cc(NC(CC3(OC)CCC3)=O)no2)=O)CCCC1C 4990,C1(C2CCC2)(NC(C2C=CCCN2C(=O)CCCc2cnn[nH]2)=O)CC1 4991,Cc1cc(C(=O)NC2CN(C(c3ccc(Br)cc3)=O)C2)nnc1C 4992,C1(CC=C)(NC(=O)C(F)=CC)CCCN(C(=O)Cc2cc(Br)cs2)C1 4993,Cc1cncc(C(N2CCCCC2CC(=O)N(C2CC2)Cc2cc[nH]n2)=O)n1 4994,c1(C(N(C)CC2CCN(C(=O)CC3CC(=O)NC3=O)C2)=O)ccnc2c1CCO2 4995,C1(C(N2CCC(CC)CC2)=O)COCCN(C(=O)Cc2cccc(OC)c2Cl)C1 4996,c1(OC)cc(C)ccc1CNc1cnc(F)cc1C(=O)N(C)CCO 4997,C1(O)(CCNC(C2(CCCC)CCC2)=O)CCN(C(c2cc(C)no2)=O)C1 4998,C1(CNC(C(CC)n2cncn2)=O)CCN(C(c2c(C)noc2C)=O)C12CCC2 4999,Cc1cnoc1Cn1cc(CCCNC(c2[nH]nnc2-c2ccccc2)=O)nn1 5000,C(=O)(CC(C)(C)n1cc(-c2ccc(Cl)cn2)nn1)NC(C)COC1CCCC1 5001,C12(NC(C(N3CCNC3=O)C)=O)COC(CNC(c3cc(N(C)C)ccn3)=O)(C1)C2 5002,N(S(=O)(=O)N1CCC(C)(C)CC1)Cc1cccc(CN2CC(C)OC(C)C2)c1 5003,C1(CNC(c2cn(CCNC(c3cc(SC)oc3)=O)nc2)=O)CC(O)C(O)C1 5004,C(=O)(CC(C(F)(F)F)c1ccon1)N(C1CCN(C(CN(C)CCO)=O)C1)CCO 5005,c1(C(=O)NCC(C(=O)NCCSCCO)N(C)C)cccc(F)c1N 5006,C(=O)(CC(O)c1cnc(Cl)s1)N(CCNC(C1(CCC=C)CC1)=O)C 5007,C(C(C(=O)NOC(CO)C(C)C)NC(C1CC2(CCO1)CC2)=O)OC 5008,CC1(CNC(=O)NCCC2CCCCO2)Cc2ccccc2C1 5009,C1(NC(N(CC(C2CCCC2)O)C)=O)CCC2(CCCNC2)C1 5010,c1(OC)ccc2[nH]nc(CNS(=O)(=O)Cc3cccc(Cl)c3OC)c2c1 5011,c1(CNC(=O)NC(C2CCS(=O)(=O)C2)C)cccc(C(C)(C)C)c1 5012,C1(CNC(c2cccc(C3(C)CC3)c2)=O)CC2(C1)CN(C(=O)C#CC1CCC1)C2 5013,N1(C(=O)NC(c2scc(CC#C)n2)C2CC2)CCn2c(-c3ccccc3)nnc2C1 5014,C1(NC(CCCc2onc(CC)n2)=O)CCC(C)(CNC(=O)Cc2ccco2)C1 5015,c1(C(=O)NC2CC(N(C(=O)Cn3cccn3)C)C2)cc(Cl)cc2ccccc12 5016,N1(C(C(C)CC2CC2)=O)CCC(CNC(=O)CC2CCCOC2)C(C2CC2)C1 5017,C(=O)(C(C)C(F)F)NCC(N(C(Cc1cc(C)no1)=O)C)C1CC1 5018,C(=O)(C(O)CC(F)(F)F)NCCc1c(C(N(C(C(=O)OC)C)C2CC2)=O)c[nH]n1 5019,c1(C(N2CC(CNC(CC(=O)OC)=O)C3(C2)CC3)=O)ccccc1N=S(C)(C)=O 5020,c1(C(C)C)ccccc1C(=O)NC(C)(C)CN(C(=O)CC1CCN(C)C1)C 5021,c1(C(C)=O)ncoc1CNCC(C1CCOC1)NC(=O)COc1ccsc1Cl 5022,c1(C(=O)NC(CC=CC)C(=O)N2CCC(C)(CC)C2)ccc(C)cc1C 5023,C1(COC)(CNC(=O)C(C)(C)c2ccc(Cl)s2)CN(C(c2cnc(C)s2)=O)C1 5024,c1(OC(C)C(N2CCC(NC(=O)CC3(CO)CC3)C2)=O)ccc(O)cc1 5025,N1(C(CC2CCC(=O)NC2=O)=O)CCC(C2(NC(=O)CN3CCSCC3)CC2)C1 5026,C(=O)(C1CCc2c[nH]nc21)N1C(C(C)NC(c2cccc3nccn23)=O)CCC1 5027,C1(N(C)C(=O)Nc2ncsc2Nc2ccccc2)CCCCCC1(C)C 5028,c1(C(N2CC(CC(C)NC(C(CC)C(C)C)=O)C2)=O)cc([N+](=O)[O-])cnc1N 5029,C12(OC)CCC(C(=O)NC3CC(O)(CNC(C4(C)CCOC4)=O)C3)(CC1)CC2 5030,C1(NC(C(C)OCCCC)=O)CN(C(=O)C(c2ccccc2)C)CC(C)(C)C1 5031,CC(C)CC(C)(O)CNC(=O)CNC(=O)Cc1ccc(C#N)cc1 5032,N1(c2nnc(SC)s2)CCCC(C)(C)C1CNC(=O)CSc1ccncc1 5033,CCCCCCC(=O)NC1CC2(C1)CN(C(=O)C(C)C(C)c1ccc(F)cc1)C2 5034,c1(N(CC)CC)ccc(C(=O)NC2CC(NC(c3ccoc3Br)=O)C2)cc1 5035,C(=O)(C1c2ccccc2CN1C(=O)CCc1cccs1)NC1(C)CCCC1(F)F 5036,C1(CNC(c2c(OC)csc2)=O)CCCCN(c2cc(C)nc(CO)n2)C1 5037,C(N=c1[nH]c(C)cc(=NCC(C)N2CCC(C)CC2)[nH]1)C1CC(OC)C1 5038,c1(CC)cc(N)c(C(=O)NCC(C)CNC(c2ncc(C)cc2F)=O)c(F)c1 5039,C(=O)(CC(C)COC)N(C(C(N1C(CCC)CCC1)=O)C1CC1)C 5040,CCC(C(=O)NC(C)CN(C(=O)Cn1ccc(Br)n1)C)N(C)C 5041,c1(C(N(CC(C)CNC(C2CCS(=O)CC2)=O)C)=O)cccc(F)c1O 5042,Cc1cc(O)nc(N2CC(NC(c3cc(C4(CN)CC4)on3)=O)C2)n1 5043,C1(C(=O)NC2C=CC(CNC(c3ccc(CO)s3)=O)C2)CCC12CCC2 5044,Cc1cc(CN2CCCC(NC3CCN(C)C3)C2)cc(C)c1 5045,C1(NC(c2nc(CCC)sc2)=O)CN(C(C23CCC2C3)=O)CC1(C)C 5046,N1(C(c2cn(C)nn2)=O)CCN(C(c2ncc(Br)cc2Cl)=O)C2CC12 5047,n1(CC(=O)NCC2C(C(=O)NC3(CC#C)CC3)CCC2)nc(C)cc1C 5048,C(CC(=C)Cl)(C(=O)NCCC1CCOCC1)NC(C(CC=C)NC(C)=O)=O 5049,C(=O)(C1=NN(CCO)C(=O)CC1)NCC1CC(NC(C(CCCCC)O)=O)C1 5050,CCCCC1CN1.c12ccc(cc1)C(=O)NCCO2.C(=O)(C(C)C)NCC 5051,C(=O)(CC(C)(F)F)NC1(CN(C)C(C2CCN(Cc3ccc(F)cc3)C2)=O)CC1 5052,CCCC(CCC)CC(=O)NC1CCN(C(=O)CCC2CC(C)(C)CO2)C1C 5053,CCCCC(C)CCC(=O)NC(C)CN(C(C1CCC1)=O)CC 5054,c1(NC(C(C)(CO)NC(C(C)C2CCCC2)=O)=O)ccc2c(c1)OCO2 5055,CCCC(CNC(=O)C(C)(C)c1ccno1)C(=O)N(C)CC1CC1(C)C 5056,c1(C(N(CC(C)NC(=O)Cc2cn(CC)nn2)CC)=O)cc2c(C)cccc2o1 5057,C1(NC(C=NOC)=O)(CO)CCN(C(c2c[nH]nc2-c2cnn(C)c2)=O)CC1 5058,C(CCC)(C(=O)N(C1CCCC(NC(=O)CCC2CC(OC)C2)C1)C)=CCC 5059,C1(NC(CC2C(CC)C2)=O)CCCCC1CNC(=O)CC1CC2CCC1C2 5060,C(=O)(C1=C(F)CN(C(=O)CC2(O)CCC2)CC1)NCC1(SC)CCC1 5061,N1(C(COCc2cccc(C)c2)=O)CCCC12CCN(C(c1ncoc1C)=O)C2 5062,C1(NC(=O)C(c2ccccc2)F)CCN(C(=O)CC(O)c2cnc(Cl)s2)CC1 5063,O=C1NC2(C(N3CCC(Cc4ccccc4)C34CC4)=O)CC3CC1C2C3 5064,C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CC(NC(COCC)=O)C(F)CC1 5065,CCC(C)C(C(=O)NC(C)(C)C=CC(=O)NC1CC1(C)C)OC 5066,Cc1n[nH]c(C)c1C(=O)NCC1CN(C(=O)C(C)Oc2ccccc2F)CCO1 5067,C1(C#CC(=O)N2CCN(CCNC(=O)CCCF)CC2)(CC)CC1 5068,C1(N(C)C)CCC(C(=O)NCC2(O)CCN(C(c3cccnc3)=O)C2)CC1 5069,c1(C(=O)NC2C(CCC)CN(C(=O)C(CC)SC)C2)cc([N+](=O)[O-])ccc1CC 5070,c1(CC(=O)NCC(C2CCCC2)NC(C2C(OCC)C2)=O)cc(F)cc(F)c1 5071,c1(CCOC)nc(=NC(C)C2CN(C(C3(C)CC=CCC3)=O)CCO2)s[nH]1 5072,c1(CC)ccc(C(=O)NC2CN(C(=O)C(CC)SC)CC2(C)C)cc1C#N 5073,Cc1nc2c(N3CCCC(C)(C(N4Cc5cccc(Cl)c5C4)=O)C3)ncnc2[nH]1 5074,C1(NC(Cc2c(C)n[nH]c2)=O)CC2(CCN(C(=O)C(C)C3(O)CCC3)CC2)C1 5075,C1(CNC(C(C)N(C)C)=O)CCCCN(C(=O)CN2CCCCCCC2=O)CC1 5076,CCCCC(O)C(=O)NC(CNC(c1ccc(F)cc1CC)=O)CC 5077,C1(CNC(C(C2CC(NC(c3cc(C)c(C)s3)=O)C2)F)=O)CC2(CC2)C(=O)O1 5078,Cn1ncc2ncnc(N3CC4CN(C(c5cc(I)ccc5Br)=O)CC34)c12 5079,CC1CCCN(C(c2ccn(C(F)F)n2)=O)C1CNC(=O)C(c1ccc(Cl)s1)=O 5080,C1(CNC(C2CC(C(F)(F)F)CCN2)=O)CC2(CC2)C(=O)O1 5081,C=C1CC(C(=O)Nc2ccnc(-c3ccccc3)n2)N(C(C2C3COCC23)=O)C1 5082,C(=O)(C1CCCc2ccccc21)NCC1(CNC(c2coc(CF)n2)=O)CC1 5083,CN1CCCCC1CCC(=O)NC1CC2(C1)CC2NC(c1cc(O)cs1)=O 5084,Cc1cccc2c1CCOC2C(=O)NCCN(C(C1CCCSC1)=O)CC1CC1 5085,C(Cc1cn[nH]c1)(C(=O)NCC1COC(=O)N1)NC(CC=CCC)=O 5086,n1(CCC(N2CC(c3cccc(C)c3)OCC2)=O)ccc2ccccc12 5087,C1(O)(CN(C(=O)C(C2CCOCC2)F)C)CN(C(c2scnc2C(F)F)=O)C1 5088,c1(C(=O)NC(CNC(c2ccc(C#C)o2)=O)(C)C)cc2cc(C)cc(C)c2[nH]1 5089,CCCC(CCC)C(=O)N1CC2CC2(NC(=O)COc2ccc(C#N)cc2)C1 5090,CC1CN(C)CCCN1C(C1(C)CCCN(C(=O)CC2=CCCC2)C1)=O 5091,C1(C#N)(OC)CC(C(N2CC(F)CC2CNC(=O)C=CCCC(C)C)=O)C1 5092,c1(C(=O)NCCN2CCN(C(c3cc(C)sc3C)=O)CC2)cc(C)c(F)c(C)c1 5093,C1(Nc2nc(C)nc(N3CCCN(C(C)=O)CC3)c2)CC2(COC(C)C2)C1 5094,C(=O)(C(CC(C)(C)C)NC(=O)C(F)OC(F)(F)F)NCc1c(O)ncc(C)c1 5095,C1(CC=C)(NC(c2c(-c3ccsc3)noc2C)=O)CCN(C(C2CCCO2)=O)C1 5096,Cc1nn2cc[nH]c(=O)c2c1C(=O)NC1CCCN(C(=O)C(C)(C)C)CC1 5097,N1(C(C(CC)CN(C)C)=O)CC(C(N2CCCCC2CN(C)C)=O)C2(CCC2)C1 5098,Cc1nc(NC2CCCC(NC(=O)Cc3ccc(C)nc3)C2)c2scc(C)c2n1 5099,N1(C(CS(CC)=O)=O)CCOC2(C1)CN(C(=O)C(C)COC1CCOCC1)C2 5100,c1(C(=O)NCC(CNC(c2ccc(C3C(C)C3)o2)=O)F)cc([N+](=O)[O-])cnc1O 5101,c1(NC(C2CCCOC2)CC)nc[nH]c(=NCc2cc(C)ncn2)c1C 5102,C=CCC(CC(F)F)NC(=O)C(F)C(C)CNC(c1ncoc1C1CC1)=O 5103,c1(C(N2CC(C)N(C(C3COC(=O)O3)=O)CC2)=O)nn(C)c2ccccc2c1=O 5104,C1(C)(CNC(C2(CC#C)CCCO2)=O)CCCN(C(=O)C=C(C)C(C)C)C1 5105,Cc1ccccc1C(N1CCOC(CN(C(=O)Cc2csc(NC=O)n2)C)C1)=O 5106,N1(C(C(CNC(C)=O)(C)C)=O)CCN(C(c2cc(C)cc(C)c2)=O)C2CCCC12 5107,C(C)(C)(CCCCC(=O)NCCC1CCCN1C(=O)C(=O)NC(C)C)OC 5108,c1(C(N(CCNC(C2CC(CS(C)(=O)=O)C2)=O)CC)=O)cccc2ccnn12 5109,C1(C(N(CCCOCCNC(CC=CC)=O)C)=O)CCC(NC)CC1.C(C)(=O)O 5110,CCCCC(CC)CC(=O)N1CC(F)(F)CC1CNC(=O)CCOC1CCC1 5111,CCC(C)(C)CC(=O)NC(C)CC(=O)N1CC(CC(F)(F)F)C1 5112,C(CC(=O)NCCC1CC(F)C1)N(C(C1(C(=O)NC)CC1)=O)C1CC1 5113,c1(C(N2CC(C)C(NC(c3cc(Cl)cs3)=O)C2)=O)cc(N)c(F)c(F)c1Cl 5114,C1(Cl)(C(=O)NC(C)CNC(c2cnnn2C)=O)CC12CCC2 5115,c1(OC)ccccc1CNCc1cc(C(=O)Nc2cc(O)ccn2)ccn1 5116,Cc1ccc(Oc2ccc(SC(C3CC=CCC3)=O)cc2)cc1C 5117,c1(C(c2nnnn2-c2ccccc2)NCC(=O)NCC=C)cc(Cl)no1 5118,C12(C(N3C(CO)CC(NC(c4cc(C(C)C)n(C)n4)=O)C3)=O)CC(C)(C1)OC2C 5119,C1(C)(CNC(CN2CCN(C)CC2)=O)CN(C(C2CC(F)C2)=O)C(C)(C)C1 5120,C1(NC(C(=O)NCC2(CNC(C=CCC)=O)CCCC2)C)CCCCC1CC 5121,C1(C(N2CC(OCCNC(C#CC(C)C)=O)C2)=O)Cc2ccccc2N(C)C1=O 5122,CC(C)(C(=O)NC1(C(=O)NC2CC2)CC1)C1CCCN1C(=O)C(=O)N(C)C 5123,O(NC(=O)C(O)CNC(=O)C(F)(F)CCC)CC#C 5124,C(=O)(C1CCCn2ccnc21)N1CCC2(C(NC(C(C)=CC)=O)C2)CC1 5125,C12(C(N3CC4C(C)(C)C4C3)=O)CCC(CC1)N(C(=O)C1=CCCCO1)C2 5126,N1(c2cc(NCC3CC4(CC4)CO3)nc(COC)n2)CCN2C(=O)NCC2C1 5127,C1(CC(=O)NC(COC)C(=O)NCCCC2CCCC2)COCC(C)O1 5128,N1(CC(=C)Cl)CC2CCC(NC(c3ncn(CC)n3)=O)CC2C1 5129,c1(C(=O)NC2C(CNC(c3ccc(C(C)=O)cc3)=O)CC2)cc2n(n1)CCC2 5130,C=CCC(C(=O)NC(CO)C(C)NC(=O)CCC(N)=O)c1ccccc1 5131,c1(CCCC=C)ccc(C(=O)NCC(C2CC2)NC(C2(N3CCCC3)CC2)=O)cc1 5132,C(CC(C(=O)NCCC1CCN(C)C1)NC(=O)Cn1ccc(C)c1)OC 5133,C1(C(=O)NC2CC(C)(NC(C(c3ccc(C)o3)C)=O)C2)CN(C)CCO1 5134,N1(C(C(COC)COC)=O)CC(C)CN(C(c2c(N)sc(C)c2C)=O)CC1C 5135,c1(C(=O)NC2CC(NC(c3scc(OC)c3)=O)C2)cc2c(nc1O)CCCC2=O 5136,c1(C(=O)NCC2(F)CN(C(CCC)=O)C2)ccc(F)cc1OC(C)C 5137,Cc1cc(C)c(C(=O)NCC(F)CNC(=O)Cn2cnc(=N)[nH]2)cc1Br 5138,n1(CCNC(C=C(C)C)=O)ccc(C(N2CCC(CC(N)=O)C2)=O)c1 5139,CCC(C)(C)C(O)C(=O)N1CCCCC1CNC(=O)C(O)CC(C)C 5140,N1(C(c2nccc(Cl)c2F)C(=O)NCC)CC(C(=O)OC)OC(C)(C)C1 5141,N1(C(c2cc(C(=O)NC)nn2C)=O)CC(OC)CC(NC(=O)CCNC(=O)OC)C1 5142,C12(CNC(=O)CC3CC=CC3)CCC1CCN2C(=O)C1=NOCC1 5143,C1(NC(CC(C=C)CC)=O)(CNC(c2nn(CC)nc2C)=O)CC2CCC1CC2 5144,N1(C(c2ccc(C(F)(F)F)cn2)=O)CC2CN(S(=O)(=O)Cc3cccc(F)c3)CC12 5145,C1(SCC)CC2CCC1N2CC1=C(C)CCCC1 5146,c1(C(=O)NCC(CNC(CC2CCN(C(C)C)CC2)=O)O)nsc2ccccc12 5147,C=Cc1ccc(C(N2CC(C)C2C(=O)NCc2nc(C(N)=O)co2)=O)cc1 5148,N1(C(C(C2CC(F)(F)C2)OCC)=O)CCC(CN(C)C(C2CN(CC)C2)=O)CC1 5149,Cc1cc(C)nc(SCC(=O)NCC2(NC(c3csc(C#N)c3)=O)CCC2)n1 5150,c1(C(N)=O)c[nH]c(C(N2CCC(CCNC(=O)C=C3CCCC3)C2)=O)c1 5151,c1(C(N2CCC(CNC(c3cnc(Cl)[nH]3)=O)C2)=O)ccncc1N1CCCC1 5152,c1(OC)ccc(CNCc2cnc(C)c(C)c2)c(N)c1Cl 5153,C1(CNC(COC)=O)(CO)CC12CCN(C(=O)CC(F)(F)C(F)(F)F)CC2 5154,N1(C(C(C)N(C(C)=O)C)=O)CCN(C(=O)CCCCCN(C)C)CC1CO 5155,N1(CCC)CCCC1C(=O)NC1CC(C)(NC(=O)C(c2ccc(C)s2)C)C1 5156,C1(C(=O)NCCN(CCOC)C(c2cnn(C3CC3(F)F)c2)=O)CCNC(=O)C1 5157,C1(NC(CC2C(C)CCO2)=O)CC2(CCN(C(c3ccoc3C3CC3)=O)CC2)C1 5158,C1(CNC(C(C2CCCC2)OC)=O)CCCN1C(C1CCS1(=O)=O)=O 5159,Cc1nn(C)c(Cl)c1C(N1CCN(C(c2coc(Cl)n2)=O)C(c2cn[nH]c2)C1)=O 5160,CC1OC(C)CC1C(=O)NCC1(NC(c2sc(N(C)C)nc2Cl)=O)CC1 5161,Cc1ccc(Cl)c(F)c1C(=O)NCC=CCNC(=O)CCSc1ccccn1 5162,c1(C(=O)NCC2N(C(Cc3ccc(C)s3)=O)CCC2C)ccc(=O)n(C)n1 5163,C1(Cl)(C(=O)NCC2(CNC(C(C)OCC(C)C)=O)CCC2)CC1(C)C 5164,c1(NCCOCCNC(c2ccc(NC(C)=O)c(C)c2)=O)c(C)ccc(C)c1O 5165,c1(C(=O)Nc2ccc(C)nc2Cl)ccc2c(C(N3CCC(C#N)C3)=O)n[nH]c2c1 5166,c1(OCC)ccc(Br)c(NC(C)CSc2ccccc2)c1 5167,C1(C(=O)NC(CC=C)CO)CCN(C(=O)C(C)COC)C12CC2 5168,C(C)(CCCCNC(c1cnc(OC)s1)=O)NC(c1cnc(CCCC)s1)=O 5169,Cc1ccc(-c2cccc(NC(C3CC4CCC3O4)=O)c2)cc1 5170,N1(CC(=O)N(CCC(C)NC(=O)COC(F)F)C)CCCC(N(C)C)C1 5171,S(=O)(=O)(c1cccc(N2CCCC2)n1)N(C)Cc1cc(Br)cs1.C12COCC1N2 5172,C(=O)(C1CCc2cc(F)ccc21)N1CCC(C2CC2)(NC(CC=C(C)C)=O)C1 5173,N1(C(C(C)N=[N+]=[N-])=O)CC(C)(C)CC1CC(=O)NCCC(=O)NC(C)(C)C 5174,C(=O)(C1Cc2ccc(F)cc21)N1CC(OCCNC(=O)Cc2sc(O)nc2O)C1 5175,C1(C(=O)NCc2nc(C)oc2C)CCN(C(=O)CC(=O)OC(C)(C)C)CC1C 5176,CC(C)(CCCNC(C1CC12CC2)=O)C(=O)N1CCCC(CC2CC2)C1 5177,C(=O)(C(=O)CC(C)C)N1CC(CC=C)(NC(=O)Cc2cnsc2)C1 5178,CC(C)C(C)(CNC(=O)CN(C)C(c1cscc1C1CC1)=O)C(C)C 5179,C1(C(=O)NCCC(C(=O)N(CCCCN=[N+]=[N-])C)OC)CC2(CCCO2)C1 5180,C1(C(=O)NCC(C)(C)O)(CC)CCCN(C(c2csc(CO)n2)=O)C1 5181,c1(C(N(CCCN(C(c2nc(OCC)sn2)=O)C)C)=O)ccc(C#N)cc1F 5182,C1(NC(C2C(C)CCC2)=O)CCOC12CCN(C(=O)C(C)(C)CCCO)CC2 5183,c1(C(N2CC3C(NC(C(C)NC(C)=O)=O)(C3)C2)=O)ccc(F)c2[nH]ccc12 5184,c1(C(=O)NC2C(CNC(C(COC)(F)F)=O)C2)c(Br)nc2n1CCCC2 5185,C1(OCC)CCC(CC(=O)NCCNc2cnn(-c3ccc(Cl)cc3)c2C)CC1 5186,Cc1ccc(C(=O)NC(CNC(c2cccnc2)=O)CO)c(N)c1Br 5187,c1(N2CC(C)OC(CO)C2)ncc(S(=O)(=O)N(C)Cc2ccns2)cc1Cl 5188,Cc1cnn(C)c1CNC(=O)CCC(C)NC(=O)Cc1cn(C2CC2)cn1 5189,c1(C(=O)NC2(C)CCN(C(c3c(C)cccc3O)=O)C2)ccc2cnccc2c1 5190,C(=O)(C1CCCn2c(C)nnc21)NC(C(C)(C)NC(Cn1c(C)cc(C)n1)=O)C 5191,C1(C(=O)NCC(C(C)(C)C)NC(C=Cc2c(C)ccs2)=O)CCc2nc[nH]c2C1 5192,C(CC(C)(C)CC(=O)NCC1CCCCN(C(=O)CC2CC(=O)C2)C1)OC 5193,CC1CCC(CN(C(C2(O)CCC2)=O)C2CC2)CN1C(=O)Cn1cncn1 5194,N1(C(c2cccnc2S)=O)CC2CN(C(c3c(Cl)cncc3Cl)=O)C2C1 5195,N1(C(CCSCC)=O)CCC(C2CC2)C1CNC(=O)C(F)=CC1CC1 5196,Cc1c(C(N2CC(C)(NC(=O)CCn3cnnn3)C2)=O)oc2c(Cl)cccc12 5197,c1(C(=O)NCC(N(C)C(c2cn(C)cn2)=O)C2CC2)ccc2c(c1)NC(=O)C2 5198,CCCC(C)(O)C(=O)NCCn1ccc(C(=O)NC(C2CC(F)(F)C2)C)c1 5199,c1(OC)ccc(C=CC(=O)NCc2ccc(I)cc2C)cc1F 5200,C12(C(=O)NCC3(OC)CCOC3)COCC1CN(C(C1CCC1C#N)=O)C2 5201,c1(C(N2CCN(C(CN(C)C)=O)C3C2C3)=O)cc(Cl)cc(Cl)c1Br 5202,c1(C(C(N2CCCC(CNC(CCS(C)=O)=O)C2)=O)(F)F)ccc([N+](=O)[O-])cc1 5203,CON1CC(C(N2CCC(NC(C3CC=CCO3)=O)CC2)=O)CC1=O 5204,C=CCCCC(C(=O)NCCc1ccncn1)NC(C1C2CCCCCC12)=O 5205,N#Cc1cccc(C2(CNCC3CN(c4ccccc4)C(=O)O3)CCOCC2)c1 5206,N1(C(c2n(C=C)ncc2)=O)CCC(C)CC1CNC(=O)CC 5207,Cc1cccn2cc(C(N3CC(CNC(=O)NC(C)(C)C)C(F)C3)=O)cc12 5208,Cc1sncc1C(=O)NC1(CC(=O)N(CCS(C)(=O)=O)C)CCC1 5209,c1(C(C(=O)NCc2nnn(C)n2)N(CC(C)S(C)(=O)=O)C)cccc(Br)c1OC 5210,C(=O)(CC(C)C(C)(C)C)N1CCC(F)(CNC(c2c(C)con2)=O)CC1 5211,CC1(NC(=O)CC2CC=CCC2)CCN(C(C2CCC3CCC2O3)=O)CC1 5212,C(CC1CC1)(C(=O)NCC(CO)C1CCC1)NC(=O)Cc1cc[nH]n1 5213,N1(C(c2ccc(SC)o2)=O)CC(C)CCC1CNC(=O)COc1cnn(C)c1 5214,c1(C(=O)NCC2(C)CCC(NC(c3cnc(COC)s3)=O)C2)cc(C)ccc1O 5215,c1(CC(=O)NCCCCCNC(C(CCC)F)=O)ccc(F)cc1C 5216,Cc1cnccc1C(N1CCCC1CN(C)C(c1cnn(CC(F)F)c1C)=O)=O 5217,C1(C(=O)OC)C(F)(F)C12CC(C(N1CCN(C(c3cnnn3C)=O)C(C)C1)=O)C2 5218,C(CC(C)C)(C(=O)N(CCCCCNC(C1CC12CC(C)(C)C2)=O)C)NC(C)=O 5219,C(=O)(C1=CC2CCCCCCC12)NC1CN(C(C2N(C=O)CCC2)=O)C1 5220,C1(C(=O)NCC=CCNC(C2CCCCC2F)=O)CCC(=C(F)F)CC1 5221,c1(C(c2nnnn2C(C)CC)NCCn2c(CC)ncc2)cc(C)c(C)cc1C 5222,CC1OC2(C(=O)NCCCN(C(=O)CC#N)Cc3ccccc3)CC1C2 5223,CC(C)(C)CC(=O)C(=O)NCC(CCNC(=O)C=CCO)O.C(C)(C)(C)O 5224,CCCC(CC)C(c1nnnn1Cc1ccco1)NCc1nnnn1C1CCC1 5225,CC1c2ccccc2OC1C(N1CC(NC(=O)COCCF)C(C)C1)=O 5226,N(C(=NCc1cccc(F)c1)NCC12CC(C1)C(C)O2)C(C)C1CC1 5227,CC(C)C#CC(=O)N(C)CC1CCCN(C(=O)CCCc2ccccn2)C1 5228,N1(C(C2C(OC)C2)=O)CCC2CN(C(c3cnn(C)c(=O)c3)=O)CCC12 5229,c1(C2(C(=O)NCC3(F)CC(NC(C4ON=C(C)C4)=O)C3)CCC2)cccc(F)c1 5230,CN1CCC(C(=O)NC2CCN(C(c3oc(C(F)(F)F)nc3C(F)F)=O)C2)CC1 5231,C1(C(=O)NCC(C(C)O)O)CCC2(CC2)N1C(c1cccc(CO)n1)=O 5232,c1(C(=O)NCC2CCN(C(=O)CC3CCSC3)CC2)ccnc2ccnn12 5233,C(=O)(N=c1[nH]n(C)c2cc(Br)ccc12)C1N(C(Cc2cc(C)no2)=O)C2C(C1)C2 5234,C1(CNC(CC(C)(C)SC)=O)CCC(C)N(C(c2ccc(F)o2)=O)C1 5235,C(=O)(CC(C)CC(C)(C)C)NCC(CC)(CC)NC(c1cc(C)c(O)c(C)c1)=O 5236,CCC(C)(C)C(O)C(=O)NC1CN(C(c2cc(Cl)cc(C)c2O)=O)CC1OC 5237,C1(C(N(C(CO)C2CC2)C)=O)CC=CCN1C(c1cccc(CC#N)c1)=O 5238,c1(C(N2CCC(O)(CNC(Cc3c(C)n[nH]c3)=O)C2)=O)ncc(C2CC2)cc1F 5239,N1(C(C(CC)OCC)=O)CC2(CCN(C(=O)C(CC)C(C)(F)F)CC2)C1 5240,CC1SCCN(C(C23CC(CN2C(=O)C(C)(C)CN(C)C)C3)=O)C1C 5241,c1(NC(C(CNC(C(c2cn(C)nc2)O)=O)O)=O)ccccc1F 5242,N1(C(C(C(=C)Cl)(C)C)=O)CCC2CN(C(c3ccn4nncc4c3)=O)CCC2C1 5243,N1(C(C(CC)C)=O)CC2CCOC2(CNC(c2cc(CC3CC3)cc(C)c2)=O)C1 5244,N1(C(C(C(=C)C)(C)O)=O)CCC2(CC1)CC(CNC(=O)CCC(C)C)C2 5245,c1(C(=O)Nc2scc(C(=O)NCCNC(C)=O)n2)c(O)ccc(F)c1F 5246,C(=O)(C(CC(C)C)N(C)C)NCCN(C(=O)Cc1c(C)cnn1C)CCC 5247,Nc1ccccc1OCCCC1(O)CCNC1.C1C(=O)O1 5248,S(=O)(=O)(c1cc([N+](=O)[O-])c(N)cc1Cl)N1CCC(N2C(C)(COC)COCC2)CC1 5249,C1(NC(CSCC)=O)CN(C(=O)C(c2ccn(C)c2)C)C(C)(C)C1 5250,C1(NC(COCCC)=O)COCCN(C(=O)C(c2cccc(C#N)c2)(C)C)C1 5251,Cc1c(C(=O)NC2CCCC2CNC(C2(CN(C)C)CC2)=O)c[nH]c1C#N 5252,N1(C(=O)CC2CCCCN2C(=O)C(O)C2CCCC2)CC2(CCOCC2)C1 5253,CC1CC(C(=O)NCCC2CCCCC2O)N(C(c2ncncc2Cl)=O)C1 5254,C(C(CC)(CC)NC(=O)Cc1ncc(C)s1)NC(C(CC)F)=O 5255,C1(CC=C)(NC(c2sccc2Cl)=O)CC2CCC(C1)N2C(C1C=C1C)=O 5256,C(=O)(CC(C)CC(=O)NCC(CNC(c1cnc(C)cc1C)=O)S(C)(=O)=O)OC 5257,C1(NC(Cc2nc(COC)sc2)=O)CC(NC(c2cc(C)cs2)=O)C(O)C1 5258,C1(CC=C)(NC(C2CSC2)=O)CC2CCC(C1)N2C(=O)C(C1CCOCC1)O 5259,C(=O)(CS(=O)(=O)CC(C)C)NC1CCC(CNC(C(CC(C)=O)(C)C)=O)C1 5260,CC1CCN(C(=O)CCn2ccnn2)C(CNC(C2CCCS(=O)(=O)N2)=O)C1 5261,c1(OCC)nc(Cl)cc(=NC(=O)c2cc(-c3ccc(C4CC4)nc3)ccn2)[nH]1 5262,N1(C(c2ccc(CSC)cc2)=O)CCC2(CNC(C3CC3(C)C)=O)CCCC12 5263,C1(CNC(Cc2ccc(OC)cn2)=O)CC12CCN(C(=O)C(C)(O)C(C)C)CC2 5264,C(CCCC(=O)N(C)CC1CCC(=O)N1)N(C(=O)Cn1cnc(C#N)n1)C 5265,CCC(C)(C)C(C)(O)c1nc(Cc2ccsc2)no1 5266,c1(NC(N2CCN(CC(=O)Nc3ncc(C)s3)CC2)=O)ccc(CCCl)c(F)c1 5267,C(=O)(C(C)CC(=O)c1ccc(Cl)cc1)N(C(CCNC(c1c(C)cco1)=O)C)C 5268,C1(NC(COCCCCC)=O)C(C)(C)CN(C(=O)C(C)CC(C)CC)CC1(C)C 5269,N(C1c2ccccc2CCC1n1ccnc1)C(=O)NCCC#CC#CCO 5270,N1(C(CC(C=C)C)=O)CCC(C(=O)NC(c2nc(=O)o[nH]2)C)C1(C)C 5271,N1(C(=O)Cc2ccccc2F)CC2CC(C1)N2C(c1cc(F)ccc1I)=O 5272,c1(C(=O)NCC2CC(F)(CNC(C3CCC(C)O3)=O)C2)cnc(O)c2ccsc12 5273,c1(C(N(C2CCCN(C(C3CCS3(=O)=O)=O)C2)CC)=O)ccnc2c1nnn2C 5274,c1(CS(=O)(=O)NCc2c(N3CCN(C)CC3)nccc2)ccc2c(n1)OCCO2 5275,C1(C2CC2)(CNC(CCC(C)(F)F)=O)CCN(C(c2cncc3ccsc23)=O)C1 5276,c1(CC)cnn(CC(=O)NCCCN2CCC(NC(C3CCC4CC34)=O)C2)c1 5277,C(=O)(C(C(C)CC)NC(=O)C(C#N)C(C)C)NCC=CC 5278,Cc1nn(C)c(Cl)c1CN1CCCC1CNC(c1cc(C(C)C)nn1C)=O 5279,CCC1=C(C(=O)NCC2CC(CNC(c3cc4cscc4s3)=O)CO2)CCCO1 5280,N1(C(CCC=C(C)C)=O)CC(CN(C(=O)C(O)C(C)(C)C)C)C2(CC2)C1 5281,CCC(CCOC)C(=O)N1CC(OC)CC1CNC(C1(CF)CCOCC1)=O 5282,c1(CC)ccc(C)nc1NC(C1(F)CCCN(C(C2(C)CCCN2)=O)C1)=O 5283,CC1CC(N(C(=O)CC2(CNC(=O)COCCCF)CC2)C)CC(C)C1 5284,CC1CC(C)CN(c2nnc(-c3cc(F)ccc3Cl)n2Cc2n[nH]cc2Br)C1 5285,N1(C(COCCC(C)C)=O)CC2CC(C1)C2NC(c1ncoc1C1CCC1)=O 5286,c1(C(=O)NCC(C(C)(C)C)NC(c2ccc(C)n2C)=O)cc2n(c1)CCOC2 5287,c1(OC)ccnc(C(=O)NC2CC(CNC(=O)CC3CC(C)=NO3)C2)c1 5288,C1(C(N)=O)CCN(CC2CCC(C(=O)O)N2C(=O)CC2CSCCO2)CC1 5289,c1(C(c2n(CCCSC)nnn2)NCc2cccc(Cl)c2)c(F)ccc(Br)c1Cl 5290,C1(C(C)(C)CO)CCCN1C(=O)C(O)CNC(=O)C(C1CC(F)(F)C1)(CCl)c1ccccc1 5291,C1(CNC(C2C(C=C(C)C)C2C)=O)(NC(c2nncn2C)=O)CCCCC1 5292,c1(C(N2CCC(C)(NC(C3CN(CC)C(=O)C3)=O)C2)=O)ncnc2cc[nH]c12 5293,c1(SC)cccc(NC(N2CCCC2C2CCCN(C(C3CCCC3)=O)C2)=O)c1 5294,c1(C(c2ccccc2)OCC(C)NC(=O)NC2(C(F)F)CCOC2)ccccc1 5295,c1(C(=O)NCCCCNC(C2(CC#C)CCOC2)=O)cc(-n2ccnc2)ccn1 5296,O=C(C1=CCCC1)NCC1CN(C(=O)CCC(=O)c2ccc[nH]2)C2CC12 5297,CC1CN(C)CC(C(=O)N(C(CNC(=O)COc2cccc(O)c2)C2CC2)C)O1 5298,c1(CC(=O)NCCN(C(C2CC(O)C2)=O)C2CC2)cccc2[nH]ncc12 5299,c1(C(N2CC3C(NC(C(CCC)(C)C)=O)(C3)C2)=O)c(Br)ccc(F)c1OC 5300,Cc1ccc(Br)c(C(N2CC(O)(CNC(C3CC34CCCC4)=O)C2)=O)c1 5301,N(C(=NCc1cc(CN2CCCC2)on1)N1CCC(COC)C1)C(C=C)C 5302,C1(C)(C(=O)NCCN(C)C(C2(C)COCCO2)=O)CCC(C)(C)CC1 5303,N1(C(C(C)CN(C)C)=O)CC(CC(=O)NCCCC2CCOCC2)C(C)C1 5304,CC1CN(S(=O)(=O)N2CCCC(c3ccccc3)CC2C)CCN1C 5305,N1(C(C(c2ccc(OC)nc2)OC)=O)CC2(C1)CN(C(C1CCCC(=O)N1)=O)C2 5306,c1(C(c2ccncc2)N(C(=O)C(C2CC3CCC2C3)N)C)ccc(Cl)cc1 5307,c1(CC)cccc(C)c1C(N1CCN(C)C(CNC(C2CC(OC)C2)=O)C1)=O 5308,c1(C(N2CCCN(C(=O)C(C3CC3)C3CC3)CC2)=O)cc2c(nc1O)CCOC2 5309,Cc1cnc(C#N)nc1N(C)CCN(C)C(C1COCCO1)=O 5310,CC(C)(C)C(CNC(C1CCC(F)(F)C1)=O)NC(c1ncccc1Br)=O 5311,c1(C(=O)NC2C(C(N(CCO)CC)=O)C2)ccc(Br)c(C#N)c1 5312,C(=O)(CC(F)(F)Br)N(C1CCN(C(C2CCN(C)C2C)=O)C1)CC 5313,C(=O)(C1=CCC(C)(C)CC1)N1C(CNC(c2c(C)oc(C)c2C)=O)CC(F)(F)C1 5314,C1(C(=O)NC2CCN(C(=O)C(O)C3CCC3)CC2)CCCc2ccccc2C1 5315,Cc1cnc(NCc2nc(=N)n(C)[nH]2)c(S(=O)(=O)N2CCC(C3CCC3)C2)c1 5316,CC1(C)COCCC1C(N1CCC2C(NC(=O)CCc3ccc(Cl)cc3)C12)=O 5317,C(C#Cc1cccnc1)NC(C(CCOCC)NC(C1CN(C)CCN1C)=O)=O 5318,N1(C(C2CC(C)(F)C2)=O)CCCC12CCCN(C(c1cccc3c1CCN3)=O)C2 5319,N1(C(CNS(CC)(=O)=O)=O)CCN(C(c2ccnn2CC#N)=O)C(C(F)F)C1 5320,C1(C(=O)NC(CC2CN(C(CC=CCOC)=O)C2)C)Cc2cccc(F)c2O1 5321,c1(C(N2CCC(C)(CNC(=O)Cc3ccoc3)CC2)=O)ccc2nc[nH]c2n1 5322,c1(C(N(C2CCN(C(=O)CC3(OC)CC3)C2)CCC)=O)ccnc(C(C)(F)F)c1 5323,c1(C(N(CCN(C(=O)CN2C(=O)CCC2=O)CC)CC)=O)cccc(C2CC2)c1 5324,C1(C(N(C2CN(c3ccnc(C(=O)OC)c3)C2)CCC)=O)CC12CCCOC2 5325,CCC(CC(C)C)C(=O)NCCC(C)N(C)C(c1ccsc1C#N)=O 5326,Cc1nc2n(c1CC(N1CC(NC(=O)CC3CCC(C(N)=O)C3)C1)=O)CCCC2 5327,n1(CC=C)cc(C(=O)NCC(C)N(C)C(C2CCN(c3nccn3C)C2)=O)cn1 5328,C1(NC(=O)C(N2CCC(C(F)F)C2)=O)CCC2CN(CC3CC3)CC2C1 5329,c1(CN2CC3N(S(C4(CC=C)CC4)(=O)=O)C(C3)C2)cc(OC)c(O)c(I)c1 5330,N1(C(CN(C2CCCC2)C)=O)CCC1CNC(C1CC(n2ccnc2)C1)=O 5331,c1(C(N2CCCC(Cc3nc(C)on3)C2)=O)noc2c1CC(C)CC2 5332,CCC(C)C(CN(C)C)NC(=O)CCN(C(c1cccc(Cl)c1)=O)C(C)C 5333,C(=O)(C(C)C(O)CC(C)C)N1CC(F)(C(=O)NC(CCC=C)(C)C)C1 5334,CCCCCCC(F)C(=O)NC(CNC(c1cnccc1Cl)=O)C(C)C 5335,c1(OC)ccc(Cl)cc1C(F)(F)C(N1CCN(C(C2(CO)CC2)=O)CC1C)=O 5336,C=CCC(CNC(C1CC(CC)(CC)C1)=O)C(=O)NCC1CC12CCC2 5337,c1(C(C)=O)csc(C(=O)NCC(C)(C)CN(C(=O)C(F)(F)c2ccnn2C)C)c1 5338,N1(C(CCCC#C)=O)CC(C)N(C(c2ccc(C3(C)CC3)cc2)=O)CC1C 5339,N1(C(C)=O)CCC(c2nc(CC(C)C(C)(C)C)n(C3CCS(=O)(=O)C3)n2)CC1 5340,C#CCC(CC(=O)OC)NC(C1CCCCC1NC(=O)C(CCC)NC(C)=O)=O 5341,C1(C(N2CC(n3ccnc3)C2)=O)(CC)CCN(C(c2n[nH]c(C)c2Cl)=O)C1 5342,Cc1cnc(C(N2CCC(CNC(C3CC3(Cl)Cl)=O)CC2)=O)cc1C#N 5343,C1(C(N(CCC#C)CCO)=O)CN(C(c2ccc(F)c(C)c2)=O)C(C)(C)C1 5344,Cc1cc(C(C)NC2CCN(C(=O)OC)C2)cc(C)c1F 5345,c1(C(N2CC3CC(CNC(c4n(C)c(S)nn4)=O)C3C2)=O)cc2cccnc2[nH]1 5346,c1(CC(=O)N(C)CCNC(c2ccoc2)=O)csc2nccn12 5347,c1(C(=O)NCC2(C(C)NC(C3CC3CF)=O)CC2)cnc2ccccn12 5348,Cc1nn(CCO)cc1C(=O)NCC(O)CNC(C1(C(C)C)CNC(=O)C1)=O 5349,c1(N2CC(CNC(C(C)C3CC3)=O)OCC2)c(Br)cncc1[N+](=O)[O-] 5350,c1(C(N(C2CC2)CC2N(C(C3(CC)CCOC3)=O)CCC2)=O)ncccc1Br 5351,c1(C(=O)NC2(CNC(c3ncncc3Cl)=O)CCOC2)cn2ccccc2n1 5352,CC(CNC(=O)C(N)=O)C(F)C(=O)N(C)Cc1nncs1 5353,c1(OC)cc(C)ccc1C(N1CCNC(=O)C1c1cccc(Br)c1)=O 5354,C1(C(N2C(C(N3CCC(OC(C)C)CC3)=O)CC(=O)C2)=O)CC2(CCO1)CC2 5355,C(=O)(C(O)CC(=O)OC(c1cc(Cl)no1)C)NC(C)(C)C.C12CCCN(C1)C2=O 5356,C1(F)(CNC(C(C)(C)F)=O)CCN(C(C2(c3cccnc3)CCC2)=O)C1 5357,c1(N2CC3(CCN(C(c4c(CC)nco4)=O)C3)C2)nccc2c1C(=O)OC2(C)C 5358,c1(C(=O)NC2CC(CNC(Cc3ccc(C)nc3)=O)C2)cc2cc(F)ccc2o1 5359,C1(C(C(=O)NC(COC)C2CC2)N2CCC2C2CCCC2)CCCOC1 5360,C(=O)(C1c2ccccc2C2CC1C2)N1C(c2c(OC)cccc2)CNCC1 5361,N1(C(c2c(C(C)=O)cco2)=O)CCC2(CCN(C(c3c(Cl)nn(C)c3C)=O)C2)C1 5362,CCCCCC(CC)C(=O)N(C)CC1CCCN(C(c2cc(N)cc(F)c2)=O)C1 5363,c1(C(N(C2CCCN(C(C34CC(F)C3C4)=O)C2)CC)=O)noc2c1CCCCC2 5364,CC1CC(C(N2CCC(O)C2C(C)(C)C)=O)N(C(c2sccc2C#N)=O)C1 5365,C1(C(N2CCCC(CNC(c3ccc(C)cn3)=O)CC2)=O)Cc2cccnc2C1 5366,C1(C(=O)NC(CC(=O)NC)C)(COC)CCN(C(=O)C=Cc2cocn2)C1 5367,C(C1=CCCCC1)(c1nnnn1CCCF)NC(=O)OCc1ccccc1 5368,C1(F)(CNC(c2cnco2)=O)CC2CCC(C1)N2C(c1noc2ncccc12)=O 5369,C(=O)(C(F)C(C)C)N(C1(CC(=O)N(CC)CC2CC2)CC1)C 5370,CC(C(C(=O)NCCC1CC1)N1CCC(Oc2cccc(F)c2)C1)C1CC1 5371,C1(N(C2CCCC2)C(c2ccc(OC)cc2)=O)CCNCC12CC2 5372,C(CCCCO)N(C)C(c1cc(CNC(=O)C(c2cccn2C)=O)cs1)=O 5373,C1(NC(C(C)C2CCCO2)=O)CN(C(C2CCCCC2O)=O)CC2(CC2)C1 5374,C1(CNC(c2c(CC)ncnc2)=O)CCCCN(C(C2COC(=O)N2C)=O)C1 5375,N1(C(C2C(OCC)C2)=O)CCN(C(=O)C(C)(C)CNC(C)=O)CC(C)(F)C1 5376,c1(COC)ccccc1CN(C)C(c1cc[nH]c1NC(=O)C(C)N(C(C)C(=O)O)C)=O 5377,N1(C(C(C)(C)C2CCN(C(C3CC34CCC4)=O)C2)=O)CC2CC2(CO)C1 5378,CC1CCC(NC(C2(C)CCC2)=O)CN1C(c1cnn(C(C)(C)C)c1N)=O 5379,N1(CC(c2cc(C(=O)OCC)n(C)c2)=O)CCS(=O)(=O)C2(CCCC2)C1 5380,n1(CCC)cc(C(N2CC=CC2CNC(=O)CSCC)=O)nn1.C1C(=O)N1CC 5381,CC(F)(C(=O)NCC1CCN(C(=O)CCCc2cnccn2)CC1)C(F)(F)F 5382,N1(C(C(C)N(C)C)=O)CC(O)CC1CNC(C1CCC(CC(=O)N(C)C)CC1)=O 5383,Cc1cnc2n1CCC(C(=O)NC1CCC(NC(=O)Cc3cnn(C)c3)CC1)C2 5384,c12ccc(cc1Cl)[nH]c2=O.Cn1cc(Br)c(C(=O)OCC=CCN2CCCC2)n1 5385,c1(CC)cc(C(=O)NCC2CCN2C(c2c(NC(C)=O)c[nH]c2C)=O)cc(O)n1 5386,CCCCC(C(=O)NCCCN(C(c1cnn(C)c1C1CC1)=O)C1CC1)N(C)C 5387,c1(CN(C(=O)CC2(CNC(C3CC3Cl)=O)CC2)C)cncnc1 5388,N1(C(c2cc3cnn(C)c3nn2)=O)CCN(C(c2cncs2)=O)C2CCCCC12 5389,C1(CCC)CCCN(C(c2ccc(CNC(c3ccoc3)=O)o2)=O)CC1 5390,N1(CCC(=O)NC2CCC(NC(C3(F)CC3)=O)CC2)CCNC(=O)C1 5391,Cc1cccc(CC(=O)NCC(C2CCC2)NC(c2cc(O)ncn2)=O)c1 5392,CC1(C)CCC2(CCCN2C(c2ccc(S(=O)C(F)(F)F)cc2)=O)CC1 5393,C1(NC(CC(=O)OC)=O)CN(C(=O)CSc2c(C)n[nH]c2C)CC1O 5394,c1(NC(=O)NC2C3CC4C2C4(C(=O)O)C3)c[nH]c2ncccc12 5395,n1(CC)ncn(NC(=O)CN(C(=O)C(CC(C)C)NC(N)=O)C2CC2)c1=O 5396,N1(C(C2CC(=C)C2)=O)CC(OC)CC1CNC(=O)C(C)CC1CCCCC1 5397,CCC(C)C(C)C(=O)NCC1(C)CCN(C(=O)Cc2ncc(C)s2)C1 5398,N1(C(C2N(C(C3CC(F)(CF)C3)=O)CCC(=C)C2)=O)CCN2CCCCC2C1 5399,CCCCC(C(=O)N1CC2CC(NC(c3nnc4n3CCCC4)=O)C2C1)C(C)C 5400,CN=c1cc(C(=O)NCC23CC(NC(C4CCOC4C)=O)(CO2)C3)cc[nH]1 5401,c1(OCC=C)cccnc1C(=O)NCCN(C(=O)COCC(F)F)C(C)C 5402,c1(C(=O)NCC2OCCN(C(c3c(C)ccs3)=O)C2)ccc(N)c(F)n1 5403,Nc1c(C(N2CC=CC2CNC(=O)C(c2ccc(F)cc2)O)=O)nc(O)nc1O 5404,C1(O)(C(N2CCCC(CCNC(CCC=C)=O)C2)=O)CCCC(C)(C)C1 5405,C(=O)(C1CCc2c[nH]nc21)NCC1(C)CC(NC(C2CC3(CCC3=O)C2)=O)C1 5406,C1(NC(Cn2cc(-c3cc(N)cc(F)c3)nn2)=O)CCc2nncn2C1 5407,Cc1nc2ccc(-c3nc(C4CCCCC4)nn3C3(C)CCS(=O)(=O)C3)cc2o1 5408,C1(NC(C2C(C=C)C2)=O)COC2(C1)CN(C(=O)CCc1cncc(O)c1)C2 5409,c1(C(N2CC(NC(C3(COC)CC3)=O)C(OC)C2)=O)ccc(O)c(C(C)C)c1 5410,Cc1ccc(C=CC(=O)NCC(N2CC(C)C(C)C2C)=O)cc1 5411,CCCCC(C)CCC(=O)NC1(CO)CCCN(C(=O)Cc2c(C)n[nH]c2C)C1 5412,c1(CC(N2C(C(C)(C)OC)CCC2)=O)ccc(N)cc1F 5413,CCC(C)CC(C)C(=O)N1CCCC(NC(=O)CN2Cc3ccccc3C2)C1C 5414,C1(N(C(=O)CCc2ncc[nH]2)C)CCCCN(C(c2c[nH]c(Br)c2)=O)C1 5415,c1(C(=O)NC2C(NC(CN(C(COC)=O)C)=O)C2)cc(C2CC2)cs1 5416,C=CCN=C(NCCC1CC1(Cl)Cl)N1CCC(n2cccc2)CC1 5417,N1(C(c2n(C)c(O)nc2)=O)CCC(NC(=O)C(N2CCOCC2)C2CC2)C(F)C1 5418,N1(C(=O)Cc2cnccn2)CC(C(N2CCCC2CC2CC2)=O)C(F)(F)C1 5419,C1(CN(C)C(C2(C)CC=CCO2)=O)CN(C(=O)C2=CCCOC2)CC12CC2 5420,S(=O)(=O)(c1ccc2c(c1)OCC(=O)N2)NCCc1ccc(OC)c(OC)c1 5421,c1(OC)ccccc1S(=O)(=O)N1CCC2(CC2C(=O)Nc2ncc(Br)s2)C1 5422,N(C1CCc2ccc(Br)cc21)C(C(N1CCCC(CCC(C)O)C1)=O)=O 5423,N1(C(CC(COC)C)=O)CC2CCCC(CNC(C3(O)CCCC3)=O)(C2)C1 5424,C(=O)(CC(C)(O)C(F)(F)F)NCC1(CNC(C=C(C)c2cccs2)=O)CC1 5425,c1(NC(C2CCC(NC(c3cncc(C)c3)=O)C2)=O)ccc(Br)c(Cl)c1F 5426,c1(C(=O)NC(C)C(C)NC(c2cncc(C(N)=O)c2)=O)cnc(N(C)C)c(Cl)c1 5427,c12ccc(c(F)c1)C(=O)N1C(C)CC1C(=O)N2.C1(C)(CO)CCN(C)CC1 5428,C1(C(N2CC(c3ccco3)C2)=O)CC2CCC1N2C(=O)C(O)CC1CCCC1 5429,CCCCC(C(=O)NC1CCC(NC(c2ccc(F)cn2)=O)C1)C(C)C 5430,C1(CCNC(CCOCC#C)=O)CC(F)(F)CN1C(=O)C(CC)NC(N)=O 5431,CCC(C)CC(C(=O)NCc1cncc(F)c1)NC(C1CC(=O)C1)=O 5432,C(=O)(CC(C)(C)CNC(=O)C(N1CCNC1=O)C)N(C1C(C)CCC1)C 5433,N1(C(c2ccc(OC)o2)=O)CC(NC(c2ncoc2-c2cc(C)no2)=O)C(C)C1 5434,C1(F)(CNC(C(C)OCC)=O)CCCN(C(C2(CO)CC(C)(C)C2)=O)CC1 5435,C1(NC(=O)CCCNC(C2CCC3(CC3)C2)=O)CC(O)CN(C(=O)C2CC2)C1 5436,C1(C(=O)NCC(CCNC(=O)C(O)c2ccco2)OC)CCc2nn[nH]c2C1 5437,CC12CC(C(=O)NC3CN(C(C4(O)CCSCC4)=O)CC34CCC4)(C1)C(C)(C)O2 5438,N1(C(C(CC=C)(C)C)=O)CC2(CCN(C(C3C=CCS3)=O)C2)C1 5439,C1(NC(C2C(CCC)C2)=O)CC2(C1)CC2NC(=O)COCc1nc[nH]n1 5440,N1(C(=O)NCc2snc(C)n2)CCC(=Cc2cccnc2)CC1 5441,CC1CCN(C(=O)C(C)Sc2ccc(Cl)cc2Cl)CCN1C(C1CC1C)=O 5442,CC(C)C(C)C(=O)NC1CC(CCNC(=O)C(N2CCSCC2)C)C1 5443,C(=O)(C(C)(C)C(C)(F)F)N1C2CC(CNC(CNC(C)=O)=O)C(C2)C1 5444,CCC(CC)C(C)C(=O)NCC1CC(COC)CN1C(=O)Cc1cncn1C 5445,CC12CCC(C(=O)NC3CC(O)CN(C(c4cc[nH]n4)=O)C3)(CC1)CO2 5446,C(=O)(CCCN=[N+]=[N-])N(C1CN(C(C(C)CN2CCOCC2)=O)C1)C 5447,N12CC3CCN(C3C1)C(=O)CC2=O.c1(C(N2CCCCC2)=O)ncccc1O 5448,c1(C(N2C(CN(C(CCOC)=O)C)COCC2)=O)cccc(Cl)c1SC 5449,C1(NC(CC2N(C)CCCC2)=O)CCC2CN(C(C3CC3(C)C(F)F)=O)CC2C1 5450,c1(COC(C2N(c3nnc(C)s3)CCCC2)=O)ccc2c(c1)C(=O)NC2=O 5451,CC1(C)C(NC(c2ccncn2)=O)C2CCCN(Cc3csc(Br)c3)C12 5452,c1(COC)nc2ccccn2c1C(=O)NCC(C)NC(C1(C#N)CCOC1)=O 5453,c1(C(N2CC(C)C(CNC(=O)CCS(N)(=O)=O)C2)=O)cc2c(cnn2C)nc1O 5454,C1(C(=O)OC)CC(S(C)(=O)=O)CN1C(C1CC(C)N1C(C1CC=CCC1)=O)=O 5455,C1(C(CNC(C=CSC)=O)(C)O)CCCN(C(c2ncsc2C)=O)C1 5456,CCCS(=O)(=O)c1ccccc1S(=O)(=O)CCNC(=O)NC1(C(=O)OC)CC1C 5457,c1(C(=O)OC)cn(C)nc1C(=O)N(C(C)CNC(=O)C(C(C)C)OCC(C)C)C 5458,C#Cc1ccc(CNC(=O)Nc2c(C)nn(C)c2CC)nc1 5459,C1(C(N2CCC(O)(CNC(CCS(C)(=O)=O)=O)C2)=O)CS(=O)(=O)CC12CC2 5460,CCN=C(NCC12CC(CO1)C2)NC1CCCC(c2ccccc2)C1 5461,c1(C)ccc(S(C)(=O)=O)c(OCC(=O)NC(C2CCCO2)CC)c1.C(C)(C)(C)O 5462,N1(C(CO)=O)CC(=O)NC1=O.C1(CNC(COCCCN(C)C)=O)CCN1C(=O)C 5463,N1(C(c2nc3c(s2)CCCC3)=O)CC2(CCN(C3C(C)(C)CO3)CC2)C1 5464,C1(C(C)C)C(NC(C2(CO)CC2(F)F)=O)CCN1C(=O)CCN1CCCCCC1 5465,C1(CNC(C)=O)CCCCC1C(=O)NC(C)C(C(=O)C(C)CC1CCCC1)=O.OC 5466,Cc1c(C(N2CCCC(NC(C3(C)CNC(=O)C3)=O)CC2)=O)cccc1C1CC1 5467,CC(CCCC(=O)N1CCOC(CCF)C1)NC(=O)COCCN(C)C 5468,c1(C(=O)NCCCOCCN(C(c2c(C)cco2)=O)C)cc2cc(O)ccc2[nH]1 5469,C1(C(N(CCCNC(C(C)OC)=O)CCO)=O)CC(=O)NC(=O)N1 5470,C1(NC(c2ncn(CC)c2)=O)C(C)CN(C(C2(N(C)C)CCOCC2)=O)CC1C 5471,N1(C(c2cncc(CC)c2)=O)CCC2(CC1)CC(C)N(C(=O)C(F)C1CCC1)C2 5472,N1(C(c2ccc(CC)nc2C)=O)CCN(C(c2ns[nH]c2=O)=O)CC12CCC2 5473,c1(CCC(=O)NCC2(F)CCN(C(C(C)C(F)F)=O)C2)ccc2cccnc2c1 5474,C(C1CN(C(=O)CN2CCSCC2)Cc2ccccc21)NC(C1(C)CC1(F)F)=O 5475,N1(C(c2c(C)ncc(C)c2)=O)CC2CCN(C(c3ccc(C)c(Cl)c3N)=O)CC12 5476,c1(N(CC(=C)C)C)nc2cc(OC)ccc2c(=NCC2(CC#N)CCC2)[nH]1 5477,c1(C(=O)NCCOC2CN(C(C3CC(O)C(F)C3)=O)C2)cc2c(cn1)OCCC2 5478,CCC(C)(CNC(=O)CC(C)N(C)C)C(=O)NCC1(CO)CC12CCC2 5479,C(=O)(C(C)(C)C1CCCN1C(C1CC(C)(O)C1)=O)N(CCOCC#C)C 5480,C1(C(N2C(CNC(c3cc(CC)[nH]n3)=O)CC(O)C2)=O)CCC(F)(F)CO1 5481,C1(C(=O)NC(C(C)C)CCN(C)C(c2cc[n+]([O-])cc2)=O)CC(=O)N(C)C(=O)N1 5482,S(=O)(=O)(c1ccc(C#N)cc1)N1CCCC(CNC(C(CCC)(C)C)=O)C1 5483,c1(CC(=O)NCC2C(CNC(C3C(C#N)C3)=O)C2)ccc2c(c1)OCCO2 5484,N1(C(CN2CC(CC)C2)=O)CCCC(O)(CNC(C2CC3C=CC2O3)=O)C1 5485,CC1CCCc2c(C(n3cc(C4NC(=O)CCC4N4CCCC4)nn3)=O)cnn21 5486,N1(C(c2ccc(SC)o2)=O)C2CCC1C(C)C(NC(c1c(C)coc1C)=O)C2 5487,C(=O)(CCCS(N)(=O)=O)NCC1(CNC(CCC2N(C)CCC2)=O)CC12CCC2 5488,C(=O)(C(O)CNC(=O)CC1CC1)N(CCC)CC1CC1 5489,Cc1ccccc1CC(=O)N(CC(C)CNC(c1ccc(SC(F)(F)F)s1)=O)C 5490,C1(N(C(CCCOC)=O)C)CC2CCC(C1)N2C(=O)Cc1cccc(Cl)c1F 5491,c1(C(N2CCC(C)C(NC(c3sccc3F)=O)C2C)=O)cc([N+](=O)[O-])cnc1N 5492,c1(C(=O)NCc2nc(C)c(C(N3CC=CCC3)=O)o2)cc2cccnc2[nH]1 5493,Cc1nn(C)c2sc(C(=O)NCC3CC3NC(C3CNC(=O)CC3(C)C)=O)cc12 5494,c1(C(=O)NCC(CNC(c2c(C)con2)=O)CO)cc2c(C3CC3)cccc2[nH]1 5495,C(N=C(NCC1CCCN1S(C)(=O)=O)N1CCC(O)CC1)c1n(C)ncc1 5496,Cc1nnc2n1CCCC2C(=O)NC1C=CC(CNC(=O)CC2=CCCC2)C1 5497,N1(C(CCc2c(C)ncnc2O)=O)CC(C)CN(C(=O)C2=CSCCO2)CC1C 5498,C(=O)(CC(C)(C)C(=O)OC)NC1(C(=O)NCc2cnc(CC)[nH]2)CC(CO)C1 5499,c1(C(C)C)cc(=NCCCCNC(=O)Cc2ccc3c(c2)CCO3)[nH]cn1 5500,C(=O)(CCCCCNC(=O)C(c1cc(C)sc1C)N(CC(=O)NC1CC1)C)OC 5501,CN1CCN(CC(N2CC3CC2C3NC(c2ccc(Cl)o2)=O)=O)CC1 5502,Cc1cc(F)cnc1C(=O)NC(C(=O)NC1C(C)CCC1C)C1CCCC1 5503,N1(C(C2C(C)(C)C(=O)C2)=O)CC23CCCC2(C1)CN(C(=O)C1=C(Cl)CC1)C3 5504,N1(C(C(=O)NCCOC)=O)CCCN(C(c2ccnc(OC)c2)=O)CC1CO 5505,C12(C(=O)NC3C(C(=O)NC(C)C(F)(F)F)OCC3)CCCCC1C2 5506,C(C(C(=O)NCCCCOC)NC(c1cccn1C)=O)CSCC 5507,N1(C(C(CCCNC(CC(CC)O)=O)O)=O)CCC(C2CCC2)CC1 5508,N1(C(COCC)=O)CCC(CCNC(=O)CNC(=O)OCC)C(F)(F)C1 5509,C(=O)(C(F)(F)c1nc(C)cs1)N(CC(CNC(CSCC=C)=O)O)C 5510,c1(OCC)ccc(S(=O)(=O)N2CCN(C(=O)NCCC(C)CC)CC2)cc1 5511,C(=O)(C(Cl)=CCl)N(CCCNC(=O)C=CI)C1CC1 5512,C1(CNC(CC(=C)C)=O)(CO)CC12CCN(C(=O)COCP(C)(C)=O)CC2 5513,c1(C(N2CC(OCCNC(CNC(CC(C)(C)C)=O)=O)C2)=O)ccc(F)cc1Br 5514,c1(N2CCCC(CNC(C(C3CCCCCC3)C)=O)C2)ncccc1C#N 5515,N1(C(CN2CCC(N(C(C(C)CC3CC3)=O)C)CC2)=O)CCc2ccccc21 5516,N(C(=NCC1CCOC1)N1CCC2(C1)CC(F)(F)C2)CCC12NC(=O)C(CC1)C2 5517,c1(CN(C(CC(C)(C)n2cc(CCC(C)O)nn2)=O)C)c(C(=O)NO)cnn1C 5518,c1(NC(C2C(C(N(c3ccn4ccnc4c3)C)=O)C2)=O)cc2ccccc2n1C 5519,c1(C(=O)NCC(CC(=O)NCC2CN(C)CCO2)OC)cc([N+](=O)[O-])c[nH]1 5520,C1(COC)CCCCC1C(=O)NCCCCN(C)C(C)C.C1(C)(C)C(=O)N1 5521,c1(C(=O)NC2CC(CCNC(=O)CSc3ccccc3)C2)cncc2nc[nH]c12 5522,N1(C(CC(=O)NCCC(C)C)=O)CC(C(F)(F)F)OC(C)C1 5523,N1(C(c2cscc2F)=O)CC2CCC1CN2C(C12CC3CC1C2C3O)=O 5524,C(=O)(C1=NOC(C)(C)C1)N(CC(CNC(c1cc(COC)[nH]n1)=O)(C)C)C 5525,CCC(C)C(O)CC(=O)N(CCC(=O)NCCC1CC(=O)N(C)C1=O)C1CC1 5526,N1(C(C=C(C)C(F)F)=O)CC2CCC1C(NC(=O)CC1CC3CCC(C1)N3C)C2 5527,C=CC(C)(C)CCCNC(c1cccc(Br)c1Cl)C 5528,CC1CCN(C(=O)COCC(c2ccccc2)C)CCN1C(c1cc[nH]n1)=O 5529,C1(C(C)C)CCC(C)CC1C(N1CC(O)(CCCNC(=O)CN=S(C)(C)=O)C1)=O 5530,C1(CNC(=O)C=Cc2ncc[nH]2)CN(C(C2(C3CCC3)CC2)=O)CCC12CCC2 5531,c1(-c2nc(C(c3c(C)ccc(C)c3)C)on2)cc(Cl)c(Cl)cc1Cl 5532,N(C1CCS(=O)(=O)c2ccc(Cl)cc21)C(=O)NC(CCCCC)C 5533,CC1CCCC(N2CCN(C(=O)C(=O)NCCNC(=O)OC(C)(C)C)CC2)C1C 5534,C1(NC(Cc2c(CC)noc2CC)=O)CN(C(c2cnnc(Cl)c2)=O)CCC1C 5535,C(CN=C(NCc1cccs1)N(C)CC1CCOC1)c1c(C)n(C)nc1 5536,N1(C(CC2CCCC(NC(CN(CCOC)C)=O)C2)=O)Cc2cccc(O)c2C1 5537,c1(C(=O)NCCCN(C(=O)Cc2cc(C)ccc2F)CC)ccc(N)cc1F 5538,Cc1cc(C(=O)OCC(=O)Nc2ccc(Cl)cc2Cl)c(C)n1-c1ccccn1 5539,N1(C(CCC)C(=O)NCc2ccc(Br)cc2)CC2CC3CC2C1C3O 5540,N1(C(CC=CC)=O)CCC2(CCOC2)C(CNC(c2[nH]cnc2CC)=O)C1 5541,Cc1cc(C2CC2)ncc1C(=O)NC1CC(CCNC(C2(C)CCCN2C)=O)C1 5542,N1(C(c2nc(C)oc2)=O)CC2CCC1C(CNC(=O)CCCCF)C2 5543,c1(C(N2CC(CC(CNC(CC3ON=C(C)C3)=O)(C)C)C2)=O)cc(C)nc(O)n1 5544,c1(C(=O)NC(CNC(C(C)OCCCC)=O)C)cccn1C1CC1 5545,C(=O)(C(C)(C)C(F)(F)CC)NCC12CC(NC(CN(CC)CC)=O)(C1)C(C)(C)O2 5546,C1(CC(C)NC(COCCCOC)=O)CC2CCC(C1)N2C(=O)C(F)(F)C(C)O 5547,C1(N(C(CN(c2ccncc2)C(C(C)O)=O)=O)C)CN(C(=O)C(N)=O)CC12CC2 5548,CC1CN(C(c2csc(Cl)n2)=O)CCC1NC(=O)C(c1ccccc1)C1CC1 5549,N1(CC)CCN(CC(N2CC3(NC(C4CCS(=O)(=O)N4)=O)CC2C3)=O)CC1 5550,C1(NC(N2CCC(CCC)C2)=O)Cc2ccncc2C1.c12nc(cc(C)n1)N2C 5551,c1(NC(C2C(=C)CC2)=O)ccoc1CC(=O)NCCOCCOCCN(C)C 5552,C=C1CC(CC(N2CC(C)(OCC)C2)=O)(C(=O)NC(COC)CO)C1 5553,C1(NC(c2cc(OCC)n[nH]2)=O)C2CC1N(C(C1(C(F)(F)F)CC(F)C1)=O)C2 5554,C1(NC(c2c(OC)cc(O)nc2)=O)C(C)(C)C(NC(=O)C=CC(=O)N(C)C)C1(C)C 5555,c1(C(=O)NCC(CCNC(CCSCC)=O)O)ccc2cnc(C)n2c1 5556,CCC(C)(O)C(=O)N1CC(CNC(=O)C(O)Cc2cnc[nH]2)C(O)C1 5557,c1(OCC)ccc(Cl)nc1C(=O)NCC1CCCC1NC(=O)C(C)c1ccco1 5558,c1(CC(N2CC(=CC(C)(C)C)C2)=O)cncc(O)c1.N1(C(C(C)S)=O)CC(C)(C)C1 5559,C(=O)(C1CCc2cccnc21)NC(c1ccc(OC)cc1)C(=O)O 5560,c1(C(=O)NC(CC(C)NC(c2ncoc2C2CC2)=O)C)ccnc(NC(N)=O)c1 5561,c1(C(=O)NCC(C2CC2)NC(CN2CC(C)(C)C2)=O)oc2ccccc2c1Cl 5562,C1(NC(CCCCCC)=O)CCN(C(=O)N(C2CCCC2)CCCC)CC1(F)F 5563,c1(C(N(C(CCNC(Cc2ccn(C(C)C)n2)=O)C)C)=O)cnc2[nH]ncc2c1 5564,N1(C(C(CC)N(C)C)=O)CC2CCCC(CNC(=O)CCCN(C)C(C)C)(C2)C1 5565,C=CCCC(F)(F)C(=O)NCC1CN(C(=O)CN2CCCCC2C)CCC1C 5566,C1(NC(=O)CCC2CCCC(O)C2)CC2CC1N(C(C1CC3C=CC1CC3)=O)C2 5567,N1(C(Cn2ncc(C#C)c2)=O)CCC2CN(C(=O)CCC3CC(F)(F)C3)CCC12 5568,c1(C(=O)NCC2N(C(CCC#C)=O)CCC(C)C2)cc(OC)c2c(c1)CC(C)O2 5569,c1(CC)ccoc1C(=O)NCC(C1CC1)NC(c1ccnn1C(C)C)=O 5570,Cc1ccc(C(=O)NCC2C3CN(C(C4CC(n5cccn5)C4)=O)CC23)cc1 5571,N1(C(c2c(C)cns2)=O)CCN(C(=O)C#CC(C)(C)C)CC(O)C1 5572,N1(CC(=O)NCc2c(OC)cc(F)cc2)Cc2ccc(Sc3ncccn3)cc2C1 5573,C1(C(F)(F)F)(NC(=O)C2CC2)CCN(C(C23CCCC2CC3)=O)CC1 5574,CC1CCC(F)(F)CN1C(=O)C(=O)NC(c1ccccc1F)c1nnc(CO)s1 5575,C(=O)(CC(CN(C)C)C(F)(F)F)N1CC(O)(CCNC(C=C(C)C2CC2)=O)C1 5576,C(C(CC(C)C)C(=O)NC(CC(F)F)C(=O)N1C2CCC1COC2)OC 5577,N1(C(c2cccnc2O)=O)CC2CC(C1)N2C(=O)CC(O)c1ccccc1 5578,c1(C(N2CC(C)C(NC(c3coc(O)n3)=O)C2)=O)cccc2cnsc12 5579,C(CC(F)F)(C(=O)NC(C)C(O)C(F)F)NC(c1c(C)non1)=O 5580,c1(C(N(CC)Cc2occc2C)=O)cc2c(Br)cncc2s1 5581,Cc1cccc(C(N2CC=CC2CNC(=O)CC2CC(c3ccccc3)C2)=O)n1 5582,n1(CCOC)ncc(C(=O)NCC2CN(C(c3sc(C)nc3C)=O)C3CC23)c1C 5583,c1(C(C(N2CC(C)C(CNC(=O)CN(C)C)CC2)=O)(C)C)c[nH]c2ccccc12 5584,N1(C(C2N(C(=O)Cn3cc(CO)nn3)CCN(C)C2)=O)CCC12CC(C)(CO)C2 5585,N1(C(COCCOCC)=O)CCCC2CN(C(=O)CCS(=O)(=O)N(C)C)CCC12 5586,CC(C(=O)N1CCOCC1)C(=O)N1CC(C)(NC(=O)CC(=O)NC2CC2)C1 5587,N1(C(CC(CC)O)=O)CCCCC(C2CN(C(c3cc(C)ccc3F)=O)C2)C1 5588,N1(C(CC(C)n2ccnc2)=O)CCC2(COC(CNC(c3cnns3)=O)C2)C1 5589,c1(OC)nc(NC2CS(=O)(=O)CC2NC(c2c[nH]nc2C(C)C)=O)nc(C)c1F 5590,N1(C(c2cc(COC)[nH]n2)=O)CC(C)CN(C(=O)Cc2c(C)noc2C)C(C)C1 5591,Cc1cc(NC(C2CC2Cl)=O)ccc1NC(=O)NC1C=CC=CC=C1 5592,C1(CNC(CCCC(=C)C)=O)CN(C(=O)C=C(C)C(F)F)CCC12CCOC2 5593,N1(C(c2c(OC)cncn2)=O)CC(O)CCC1C(=O)NOCC(=O)N(C)C 5594,C(=O)(CCNC(=O)OC)NCC1C(CNC(CN(CCC)C)=O)C1 5595,C12(C(=O)NC3(C=C)CCC3)CCC(CN(C(C3C4COCC34)=O)C1)C2 5596,c12ccc(C(=O)C3CC3)c(c1)NC(=O)N2.C1(CC(=O)OC)OCCCO1 5597,c1(C(N2CC3(CCC3)C2c2ccncc2)=O)nn2c(c1Br)OCCC2 5598,C1(c2nnnn2C)(NCCC(C)S(C)(=O)=O)CCC(C2CCC2)CC1 5599,C(N=c1[nH]c(N2CC(=O)NC(=O)C2)nc2c1CCC2)C1C(C)(C)OCC1 5600,C(=O)(C1CCCc2nccn21)NC(CCCC)CNC(c1cc(C)oc1C)=O 5601,c1(C(=O)NC(CNC(COCC(=C)C)=O)C)c(C)c(Br)n(C)c1C 5602,C(=O)(C(C)CN(C)C(=O)C1CC1)N(C(CSC)C)C 5603,CC1CC2(CCO1)CC2C(=O)NCC1CCN(C(c2c[nH]ccc2=O)=O)CC1C 5604,N1(CCNC(=O)NC2C3CC4C(C3)C24)CCC(F)(C2CCN(c3ccccc3)C2)C1 5605,O=C1CCCC(c2ccccc2)(CNCCCF)N1 5606,N1(C(=O)CCC=CBr)CC2(CCN(C(C3CCC4CCC(=O)N34)=O)CC2)C1 5607,C(C(O)C(=O)NCC(N1CC(C)(CNS(N)(=O)=O)C1)=O)N(C)C 5608,C12(CNC(=O)CC3CCC34CCC4)CCCC1N(C(=O)C=C1CCCCC1)CC2 5609,c1(C(=O)NC2CC(N(C(=O)CN3CCCNS3(=O)=O)C)C2)ccc(Cl)c(N)c1Cl 5610,C1(C(=O)NCC2(F)CN(C(C=CC(C)(C)C)=O)C2)CC2C=CC1C2 5611,C1(NC(C(CC)NC(=O)C(C2CCOCC2)F)=O)CC2OC(=O)CC12 5612,C(=O)(C(=O)CC(C)C)NCC1(CC(=O)NCc2cn(CC)nc2)CC1 5613,c1(C(N2CC(NC(C(CC=C)C)=O)C(C)C2)=O)cncc(Cl)c1C 5614,C1(N(C(C=C(C)C)=O)C)CCCC(NC(=O)CCn2ccnc2)C1 5615,c1(C(N2CC(=CC)C2)=O)ccnc(CNC(=O)CC(C)(C)O)c1 5616,c1(C(=O)NC2(CC(=O)OCC)CCC2)ccc2c(C3=CCNCC3)n[nH]c2c1 5617,Cc1nc2nc(=S)[nH]n2c(C)c1CC(=O)NC(C)C(C)NC(=O)C(F)F 5618,C12(NC(C(C)CN(C)C)=O)CCC(CNC(=O)CCc3csc(=N)[nH]3)(C1)OC2 5619,N1(C(Cc2cc(C)no2)=O)CCC(NC(C2CCCOC2)=O)C(O)C1 5620,c1(C(=O)OC2CCCC2C(=O)NOCCF)ccc(OC2CC2)nc1 5621,c1(CNC(C(C2CCCN(C(CCSC)=O)C2)(C)C)=O)cnc(F)cc1C 5622,C(=O)(C1=C(Cl)CCC1)NC1CC(F)(CNC(c2c(NC)nccc2)=O)C1 5623,Cn1nnnc1SCCC(=O)NC1CC(F)(CNC(c2cc(CCO)on2)=O)C1 5624,CC(CC(N)=O)C(=O)N1CC(CNC(=O)C2CC2)C2(CC2)C1 5625,N1(C(c2ccc(OCC)cc2)=O)CC2(CCC2NC(c2ccc(CO)s2)=O)C1 5626,C1(NC(CC=CCC)=O)CC(C)CN(C(c2ccc(=O)n(CC(F)(F)F)c2)=O)C1 5627,N1(C(C(C)C2CCC2)=O)CCOCC(NC(c2occc2-c2cnn(C)c2)=O)C1 5628,N1(C(CC(C)C)=O)CCC(NC(C2(S(N)(=O)=O)CC2)=O)C(F)C1 5629,C1(F)(CNC(COCc2n(C)ncc2)=O)CCC(CNC(C2CCCO2)=O)CC1 5630,C(C(=O)N(C)CC1CCCC1NC(=O)COC1(C)CCCC1)(C(C)(C)C)OC 5631,C1(NC(c2c(C)oc(C(C)C)n2)=O)CCN(C(c2ccc(N)c(Cl)n2)=O)CC1F 5632,Cc1c(C(=O)NC(C(N2CC[Si](C)(C)C2)=O)C2CCCC2)ccn1C 5633,N1(C(CC(C)F)=O)CC2(CCN(C(=O)CC3COC(C)(C)CO3)C2)C1 5634,C(=O)(C1=CC2(CCN(C(c3ncc4ccccn34)=O)C2)C1)NCC(C)CCO 5635,N1(C(C2C(C)(C)CC2)=O)CC(NC(c2cc(O)cc(Cl)c2)=O)CC(O)C1 5636,CC1(C)CC(O)(CC(=O)NCC(C)(C2CC2)NC(C23CC(C)(CO2)C3)=O)CO1 5637,CNS(=O)(=O)N1CCC(C(=O)N(CCCN(C(=O)CCNC(=O)CO)C)C)CC1 5638,C1(C)(CC)CC(NC(=O)Cc2ccc(C)s2)CN1C(=O)CCCCOC 5639,c1(N(CCOCCN(C(C2C(CCC)CCC2)=O)C)C)ncnn2c(Br)ccc12 5640,c1(CNC(C(C)(C)C)c2nnnn2-c2ccccc2)ccc(C(F)(F)F)cn1 5641,c1(NC(=O)NC(CCc2cccc(OC)c2)C)ccc(S(C)(=O)=O)nc1 5642,c1(C(N2CC(C(=O)NCC3OCCN(C)C3)OCC2)=O)cccc2ccoc12 5643,n1(CC(=O)NC(C(C)NC(c2cnc(C)[nH]2)=O)C(C)C)ccc(=O)cc1C 5644,CC(C)CC(C)CC(=O)N(C1CCN(C(=O)C2=CS(=O)CCC2)CC1)C 5645,c1(CCC(=O)NC23CC(NC(C4NC(=O)OCC4)=O)(C2)C3)cc2ccccc2[nH]1 5646,C(=O)(C#CC(C)(C)CNC(=O)C=C(C1CC1)C1CC1)NCC1C(C)C1 5647,c1(CC#N)ccccc1C(N1CCOC(C(=O)NCC2CCO2)C1)=O 5648,C1(C(N2C(CNC(c3c(C)cnnc3O)=O)CC2)=O)Cn2c(C)nnc2CN1C 5649,C1(C(=O)NCCCOCCCC)CCN(C(=O)C(C2CCOCC2)O)C(C)C1 5650,c1(C(=O)OC(C)(C)C)cnc(NC(=O)NCC(=O)NCc2ccc(Br)s2)[nH]1 5651,Cc1ccc(NC(C2CCCC(NC(=O)Cc3ccc(Br)cc3I)C2)=O)c(I)n1 5652,c1(C(=O)NCCCN(C(=O)CCCCC#N)C(C)C)nccc2[nH]ccc12 5653,N1(C(c2ncc(C)s2)=O)CCc2c(Br)ccc(NC(c3ccnnc3)=O)c2C1 5654,C12(NC(=O)Cc3ccns3)CCC1CN(C(C1CCCOC1)=O)C2 5655,CC#CCCCC(=O)NC1CC(CNC(C2CCCCO2)=O)C1 5656,C(N=c1[nH]c(N2CCC(C(C)C)C2)nc2c1CCCCC2)C1(OC)CC1 5657,C(c1ccc(F)c(F)c1)=C(C)C(=O)NC1(C)CCN(C(C2CCOCC2)=O)C1 5658,C1(NC(c2nc(C)[nH]c3nccc2-3)=O)CC2CCC1(N=c1[nH]ccnc1F)C2 5659,c1(OC)cc(C(N2CCC(N(C(=O)Cc3coc(C)n3)C)C(C)C2)=O)ccc1Cl 5660,c1(C(=O)NCC(CC)NC(C2CCC2c2nc[nH]n2)=O)nc2cccnc2s1 5661,c1(NC(C)C(C2CCC2)NC(=O)OC(C)(C)C)cnccc1Cl 5662,N1(CCC(=O)NCCC(O)CNC(c2cnc(C(F)F)s2)=O)CCOC1=O 5663,c1(C(N2CCC(O)(C(F)F)CC2)C(=O)NCCCSC)cc2cc(Cl)cnc2o1 5664,N1(CC(c2ccc(C)o2)C)CCCc2cc(OC(C)C)ccc21 5665,CCN=c1[nH]c(C(N2CCCC2CCNC(=O)CN(C2CC2)CC)=O)cs1 5666,c1(C(N2CCC(NC(C(C3CCC3)OCC)=O)C2)=O)ccc(OC)cc1OC 5667,C(=O)(C(C)CC(C)C)NC(c1cnn(C)c1)C(=O)NCC(C(=O)OC)(F)F 5668,c1(C(=O)NC(CCNC(c2cccc(C)c2F)=O)C)cc2c(o1)CCCC2 5669,C(=O)(C(Cc1cnc[nH]1)NC(C)=O)NC(CC)C1CC1 5670,C1(C(=O)NC2CCN(Cc3nc(-c4ccccc4)no3)C2)CC2CCC1O2 5671,C(=O)(C(C#N)C(C)C)NCC(CN(C(=O)CCC1CC1(C)C)CC)(C)C 5672,c1(SCC)cncc(C(=O)NCCCN(C(=O)COCC(C)(C)C)C)n1 5673,c1(C(C(=O)NCCOCC)N(C)CC2CCC(C)CC2)ncc2ccccn12 5674,C(=O)(C(C)(CC)CCCCCC)NC1CC(Nc2ncc(C#C)cn2)C1 5675,c1(C(=O)NCC(CO)NC(c2cc(OCC)c(F)cc2)=O)cccc2sccc12 5676,c1(OC(C(=O)N2CC(n3cc(SNC(C)C)nn3)C2)(C)C)ccc(Cl)cc1 5677,C1(NC(CC2C(=O)NC(=N)S2)=O)CC2CC(C1)N(C(=O)CCC1CCCCO1)C2 5678,N1(CC=CC(=O)NCC2CCCN2C(=O)CSCc2ccccc2)CCOCC1 5679,N1(C(C2(CC=C)CCCN2C(c2ccc(CO)nc2)=O)=O)CC(=O)N(C)CC1C 5680,C(CCN=C(NCCc1cccc(C)c1)NC1CC1C1CCOCC1)OCC 5681,N1(C(CC(C)c2cnn(C)c2)=O)C2CCC1C(CNC(c1ccon1)=O)C2 5682,N1(C(C(C2CC2)SC)=O)CC=C(C(=O)NC2COCCC2O)C1 5683,c1(C(=O)NCC23C(CN(C(C(CC)SC)=O)C2)CC3)ccc2c(n1)CCC2 5684,N1(CC(=O)NC(C)(C)C=CC(=O)NC2(C(O)CO)CCC2)CCNC1=O 5685,n1(CC)ncn(NC(=O)C(C2CC=CCC2)NC(=O)CCC(C)=O)c1=O 5686,N1(C(CCc2ncn(C)c2)=O)C2CCC1C(NC(=O)CCN1CCOC1=O)C2 5687,C1(CNC(=O)Nc2cncc(SC)c2)CC2(C1)OCCO2 5688,C1(O)(C(C)NC(CCn2ncc(C)c2)=O)CCN(C(c2sc(F)cc2C)=O)CC1 5689,C1(O)(CC(=O)NCCN(C)C)CCN(C(c2ccc(C#N)cc2)=O)CC1 5690,c1(CC)sc(C(N2CCC(F)(C(N)=O)C2)=O)cc1CC 5691,c1(C(N2CC3C(CN(C(CC(CC)OCC)=O)C)C3C2)=O)cc(F)ccc1Cl 5692,C(=O)(C(C)(O)C(F)(F)F)N(CCCNC(c1c(F)ccc(CC)c1)=O)CC 5693,C(=O)(CC(O)C(C)C)N1CC2C(NC(C3(COC)CCCO3)=O)C2C1 5694,CC1(C(=O)NCC2(CNC(=O)CCF)CCC2)COC(=O)OC1 5695,c1(C2CN(CC(=O)N(C(CCC#C)=O)C)C2)ccc([N+](=O)[O-])cc1Cl 5696,C(CC)(c1ccccc1)=CC(N1CCN(C(C=C(CC)C)=O)CC1COC)=O 5697,c1(C(N2C(C(N(CC(C3CCC3)OC)C)=O)CC(=O)C2)=O)cc2cccnn2c1 5698,Cc1nccc(=NCC2CCN(C(=O)CC3(C)CCS(=O)(=O)N3)C2)[nH]1 5699,C1(CNC(C)=O)(CSC2(c3ccc(F)cc3)CC3(CC3)C2)CCCCC1 5700,Cc1cc(CNC(c2nccn2C)c2nnnn2C2CCCCC2)c(C)nn1 5701,N1(C(c2c(COC)noc2)=O)CC2CC(C1)CN(C(=O)C(C)(C)C1CCC1)C2 5702,c1(C(=O)NC(c2cnc(C)s2)C)cc(S(=O)(=O)CC2CC2)ccc1F 5703,c1(OC)ccc(CN2CCN(Cc3cc(Br)cs3)C3CC23)c(C)c1C 5704,CC(C)(C)CC(C(F)(F)F)NC(C1(c2ccccc2OC(F)(F)F)CC1)=O 5705,c1(OCC(=O)NC2CCCC2CNC(c2ccnc(O)c2)=O)ccc(Cl)cc1F 5706,Cn1cc(S(=O)(=O)NCC(=O)NC2CC(NC(=O)CC3CCCCC3O)C2)cn1 5707,C#Cc1ccc(C(=O)NC(CCC=C)C(=O)NC(C)CCC=C(C)C)nc1 5708,c1(CNc2cc(C(=O)OC)c(F)cc2Cl)c(Br)cc(F)c(C(=O)O)c1F 5709,C(=O)(CCCCC(C)CC)NCCC(=C)CNC(c1csc(Cl)c1)=O 5710,CCCC(C)(CC)C(=O)NC1CCCC(NC(=O)Cc2ccc(O)c(C)c2)C1 5711,N1(C(c2cnc(CCC)s2)=O)CCN(C(c2ccn(CC)c(=O)c2)=O)CC1CO 5712,N1(C(c2cc(C)c(Cl)c(N)c2)=O)CCC2(CC1)CN(C(=O)CC1CC3CC3C1)C2 5713,C1(NC(=O)CCc2ccncc2)CCCCC1NC(=O)Cn1cc(Br)cn1 5714,C(=O)(C1CCc2ccccc21)N1C(CN(C)C(C2CCCN2N=O)=O)CCCC1 5715,CC(C)CC(CCc1ccccc1)C(=O)NCC1CCCC1(C)C 5716,CC(C(=O)NC1CC(NC(=O)COCc2nnc(S)n2C)CC1O)C(F)F 5717,CCC(CCO)NC(=O)CCC1(NC(=O)C=Cc2cc[nH]c2)CCC1 5718,C12(C(=O)NCC3N(CC)CCC3)CCC(CC1)CN2C(c1ccnc(C)n1)=O 5719,CCCCC(CN=c1nc(-n2ccnc2)cc(C)[nH]1)NC(c1n[nH]cc1Cl)=O 5720,N1(C(c2c(SC)cc(C)cc2)=O)CC(NC(=O)C(F)CC2CCC2)C2(CCC2)C1 5721,c1(C(=O)NCC(C)NC(CN(C(=O)OC)C)=O)cc2c(nc1O)CCCC2O 5722,C1(C(=O)NCCN(C(CSCCCC)=O)CC2CC2)CNC(=O)N1C 5723,c1(OC)cccc(Br)c1C(N1CCC(NC(=O)CSC)C(C)C1)=O 5724,Cc1cc2ncc(C(=O)NCC3CC(C)CCN3C(C3CC3(Cl)Cl)=O)c(C)n2n1 5725,N1(C(C2(SC)CC2)=O)CCN(C(=O)C(N2CCNC2=O)C)C2CCCCC2C1 5726,C(C1=NOC2CN(C(=O)CC3(CC)CCOCC3)CC12)NC(c1n(CC)ncc1)=O 5727,Cc1nc(C(C)C)ccc1C(=O)N(CCNC(c1cc[nH]c1)=O)CC1CC1 5728,C(c1cc(F)c(F)c(F)c1)=CC(N1CCCN(C(C2(OC)CC2)=O)CC1C)=O 5729,CCC(C(=O)N(C)CC1(O)CN(C(C2CC(=O)N2)=O)C1)C1CCOCC1 5730,c1(NS(Cc2cn(C)nc2)(=O)=O)ccc(S(=O)(=O)NC2CC2)cc1 5731,c1(OC)ccc(C(N2CC3(CC(NC(C45CC(OC)C4C5)=O)C3)C2)=O)cc1OC 5732,c1(OC)ccc(F)cc1-c1nc(CC2CCCC2)nn1C1CCCC1O 5733,c1(CNC(c2ccc(Cl)c(F)c2)C(=O)O)cc2cc(F)ccc2nc1Cl 5734,c1(C(=O)NCC2(C)CCN(C(c3ccc(O)nn3)=O)C2)ccc(C#N)c(Cl)c1 5735,N1(C(c2c(C(C)C)scn2)=O)CCC(C)(C)C(NC(=O)CC2C=CCCC2)C1 5736,CC1(C)Oc2ccc(C(N3CCC4C(CCN4C(=O)C(O)C(F)F)C3)=O)cc2O1 5737,N1(C(c2c(C)oc(Br)c2)=O)CC(NC(c2ccnn2C)=O)CC(C)C1 5738,N1(C(CC(=O)OC)=O)CCN(C(=O)Cc2cc(F)cc(F)c2)CC1CF 5739,c1(SCC(=O)NCC2CCCC2C(=O)Nc2cccc(CO)c2)cncc(O)c1 5740,C(CC(CC)C(=O)N1CC2CC2(CNC(c2ccncn2)=O)C1)=CC 5741,C1(NC(C2CN(C(C)=O)C2)=O)CN(C(C2(c3ccccc3)CCC2)=O)CC1C 5742,C(CNC(=O)CCCNS(C)(=O)=O)(C(C)C(C)C)NC(c1c(C)oc(CO)c1)=O 5743,c1(C(=O)NC2C(NC(C3CCN(C(C)=O)CC3)=O)CCC2)cccn2nccc12 5744,c1(C(=O)Nc2cccc(C(=O)OC)c2N)cn2c(n1)CCCC2C 5745,c1(C(N(C2CCN(C(=O)C=CBr)C2)CC)=O)cc(Cl)nnc1Cl 5746,c1(CNC(c2c(CC)n[nH]c2)=O)cccc(CNC(=O)CC2COCC(C)O2)c1 5747,C(=O)(CC(C)C(=O)N1CCC(C)C(N(C)C(C2CCCCS2)=O)C1)OC 5748,Cn1cc(C(N2CCC(NC(c3cc(CO)[nH]n3)=O)C(F)C2)=O)c2cccnc12 5749,C(CCC(CC)CC)NC(C(C(C)NC(COCCC)=O)C)=O 5750,C(=O)(C(C)(C)CC(C)C)NC1CN(C(CCSCC)=O)CC1C(F)(F)F 5751,C1(NC(C2CCOC2)=O)CN(C(c2ccc(C(F)(F)F)cn2)=O)C2(CCC2)C1 5752,N1(C(Cc2c(COC)cccc2)=O)CC(NC(C2CCOCC2)=O)CC12CCC2 5753,C1(O)(C(N(CCCCNC(CCNC(C)=O)=O)C)=O)CC1(C)C 5754,N1(C(C2CCC(CC)O2)=O)CC2(C)CN(C(C3CNC(=O)N3)=O)CC2(C)C1 5755,c1(C(N2C(C#N)CN(C(C3CCCS3)=O)CC2)=O)cc([N+](=O)[O-])c(F)c(F)c1F 5756,c1(C(N2CCN(C(=O)CCc3cncs3)C3CCCC23)=O)n[nH]c2ccccc12 5757,N1(C(CCCC#CC)=O)CC2CC(F)(F)CCC2(NC(=O)COCC)C1 5758,S(=O)(=O)(c1cnn(C)c1)NC(C(=O)NC(C)CCNC(=O)C(C)NC1CC1)=O 5759,c1(C(=O)NCC2N(C(CSCC(=O)OC)=O)CC2)ncoc1CC1CCSC1 5760,C=CCC(C(=O)N(CCCNC(=O)CCCc1ncco1)C1CC1)OC 5761,C(c1ccn(C)c1)=CC(=O)NCCCC(C)NC(C1CN(C(C)=O)C1)=O 5762,N1(C(COC2CC(NC(C3C(C)CCOC3)=O)C2)=O)CC(F)CC(F)C1 5763,C(=O)(CCCCc1ccc(C)cc1)N1C(Cn2cc(COC)nn2)CCC1 5764,c1(C(=O)NC2(CN(C(CSCCCC)=O)C)CC2)cccc(OC)c1 5765,C(C(=O)NC1CCCCC1CNC(C1CCCN1CC(F)(F)F)=O)(C(C)C)OC 5766,C1(C(=O)O)CCCCCCN1C(c1cc(C(F)(F)F)ncc1Br)=O 5767,c1(OC)ccc(Cl)cc1NC(N1CC(c2ocnc2CNC(=O)C(C)(C)C)C1)=O 5768,C1(O)(C(C(=O)NC(C)CCN(C)C(c2ccns2)=O)(F)F)CCCCC1 5769,N1(C(c2nc(CCCC)sc2)=O)CCCN(C(c2cc(C)ncn2)=O)CCC1 5770,c1(C(=O)NC2CCC(Cn3cc(C4(C)CCCC4)nn3)C2)cnn2c1CCCC2 5771,N1(C(COC(C)=O)=O)CCN(C(=O)C(F)C2CCC2)C(C2CC2)C1 5772,CCC(C(=O)N1CCN(CC(O)COc2ccccc2)CC1)C(=O)O 5773,Cc1ccc(C(C)(C)C(=O)NC(C)CCN(C)C)c(C)c1 5774,c1(CC)noc2ncc(C(=O)N(CCN(c3nnc(C)s3)C)C(C)C)cc12 5775,c1(C(=O)NCC(C(C)C)NC(=O)C2=CC3CCCC23)c[nH]c2cc(Cl)ccc12 5776,N1(C(=O)NCCc2nc(CC)sc2)CCCN2CCCC12 5777,CC(C(C)(C)NC(=O)C=C1CCCC1)NC(=O)Cc1csc(Cl)n1 5778,C(C(COC)CC(=O)N1CC(CCNC(C2(Br)CC2(C)C)=O)C1)OC 5779,C(=O)(CC(CCC)NC(=O)C=Cc1ccncn1)NCC(=C)Br 5780,N1(C(C=C(CC)C)=O)CC2CN(C(c3ccc(OCC(N)=O)cc3)=O)CCC12 5781,C#Cc1ccc(NC(C2COCCN(C(C3(CC(C)=O)CC3)=O)C2)=O)c(C)c1 5782,C1(NC(C(F)=C(C)C)=O)CC2CC1CN(C(=O)C(c1c(C)noc1C)(C)C)C2 5783,c1(N2CC3CN(C(c4ccc(Cl)cc4F)=O)CC32)ncnc2[nH]ccc12 5784,Cc1cc([N+](=O)[O-])cc(C(=O)NC2CN(C(c3c(C)cnn3C)=O)C(C)(C)C2)n1 5785,c1(NC(=O)C(=O)NC2CC(CCc3ccco3)C2)ccccc1 5786,N1(C(CCc2cc(OC)c(F)cc2)=O)CC2CCC(C1)N2C(=O)C(C)CC(N)=O 5787,C1(C2CCCCC2)(C(=O)NC2CC(NC(C3(C#N)CCOC3)=O)C2)CC1 5788,C1(NC(C=CCOC)=O)CCN(C(C2CCC(=O)N2C(C)C)=O)CC1O 5789,N1(C(CCN(CC#C)C(C2CCCC2)=O)=O)CCOC(CN(C)C)C1 5790,c1(OCC)ccc(CCC(=O)N2CCC2C(=O)NCc2cc(C3CC3)on2)cc1 5791,c1(C(=O)NC2C(C(N(C3CCCC3)CC(C)C)=O)CC2)ccc2occc2c1 5792,C(=O)(C(CC)CC(C)C)N1CC(C2CC2)(C(=O)NC2C(CC=C)COC2)C1 5793,c1(C(=O)NC2CC3CN(C(C(C=C=C)C)=O)C(C2)C3)n[nH]c2c(C)cccc12 5794,N1(C(c2c(C)scn2)=O)CC2OCC(NC(C3CC4(C3)CC(C)C4)=O)C2C1 5795,c1(NC)cnc(C(=O)NCC2CCCN2C(C2CCN(C)C2)=O)cn1 5796,N1(C(CC2N(C(CC#N)=O)CC2)=O)CCOCC(F)(F)C1 5797,CCCCCCC(C)C(=O)NCC12CCC(C1)N(C(=O)CN1CC(=O)NC1=O)C2 5798,C1(C(N(C2CCN(C(=O)C(C)(C)C3CCC3)CC2)CCOC)=O)C2CC2C2CC12 5799,N1(C(C2CCC(C)(C)N(C(=O)COCCCF)C2)=O)CCC12CCC(C)CC2 5800,C(CC(=O)NCC1(CC2CC2)CC1)(CC(C)C)NC(C=Cc1cccc(C)c1)=O 5801,C(=O)(C(C)(C)CC(C)C)N(C(CC(=O)NC(C(=O)OC)C)(C)C)C 5802,C12(NC(c3n(CC#C)ccc3)=O)CCCN(C(c3cc4n(n3)CCO4)=O)CC1C2 5803,N1(c2ncnc(N(CC(CC)C)C)c2C)CCc2c[nH]nc2C1 5804,c1(C(=O)NCC2(O)CCN(C(COC(CC)(C)C)=O)C2)ccc2c(c1)CC2 5805,c1(OCC)nn(C)cc1NC(C1CC(C)N1C(C1C=CC=CC=C1)=O)=O 5806,CCCC(C)(C)C(=O)NC1CC(CCNC(=O)COCCOCC)C1 5807,CCC(C)(F)C(=O)N(C)CCN(C)C(C1(N2CCSCC2)CCCCC1)=O 5808,C1(NC(c2n[nH]c(C)c2O)=O)CCC2CN(C(C3CC(OC(F)(F)F)C3)=O)CC2C1 5809,c1(C(=O)NCC(c2ccc(Br)cc2)(C)C)ccc2c(c1)NC(=O)C2 5810,S(=O)(=O)(c1ccc(NC(c2cc(C)ccc2F)CO)nc1)N1CCC=C(C)C1 5811,C12(NC(c3c(C)ocn3)=O)CC1CN(C(=O)Cn1nc(C(F)F)cc1C(F)F)C2 5812,c1(C(=O)NCc2scc(CNC(CCC=C=C)=O)n2)cccc(F)c1C 5813,N1(C(c2cccs2)C(=O)NCCC(=O)OCC)CC(S(C)(=O)=O)CCC1C 5814,Cc1cc(C(=O)NC(CNC(c2cnsn2)=O)CC(C)C)cnc1C(F)(F)F 5815,c1(C(=O)NC2C(OC)CN(C(=O)C(O)C(C)(C)C)C2)cc(S(N)(=O)=O)c[nH]1 5816,N1(C(C2N(C(C)=O)CSC2)=O)CC2CN(Cc3ccc(Cl)cc3C(F)(F)F)C2C1 5817,c1(C(N(CC(CNC(C(COC)NC(C)=O)=O)O)C)=O)sc(C(C)(C)C)nc1C 5818,CC(C)CS(=O)(=O)CC(=O)NC1CC2CC(NC(c3coc(C(F)F)c3)=O)C2C1 5819,C(CS(=O)(=O)C1=NOC(C)(C)C1)NC(c1ccc(C(F)(F)F)cc1)C(=O)OC 5820,OCCC(N=c1[nH]c(=NCC2CCOC2)[nH]c2c1CCCC2)c1ccc(F)cc1 5821,c1(OC)ccc(C(N2CCOC(CNC(=O)CCOC3CC3)C2)=O)cc1Cl 5822,C1(CC(=O)NC(C)C(C2CCCCC2)NC(=O)OC(C)(C)C)CCCC2CC12 5823,C(=O)(CC1=NNC(=O)C1)NC1CCC(NC(CN(CC)CC)=O)C1 5824,c1(C(N(CCN(C(C=CC)=O)C(C)C)C)=O)cccc(C2CCCOC2)c1 5825,N1(C(c2ccc(C)n2C)=O)CC2CCC1CN2C(=O)Cc1ccco1 5826,C1(CN(C(=O)CC23CCCC2C3)C)CN(C(c2cc(CN(C)C)[nH]n2)=O)CCO1 5827,C12(C(=O)NCC3(OCC)COC3)CC(CO1)N(C(c1cscn1)=O)C2 5828,Cc1cccc(OCC(N2CC(OCCCS(N)(=O)=O)C2)=O)c1 5829,c1(C(=O)OC)n[nH]c2c1CCN(CC1CCC(C(F)(F)F)O1)C2 5830,S(=O)(=O)(c1cccc(=NCc2cc[nH]c(=N)c2)[nH]1)N(CC(C)OC)CC 5831,Cc1cc(S(=O)(=O)N(C(=O)C(CN)CC(C)(C)C)C(C)C)sc1C 5832,C1(C(=O)NCCC2CN(C)C(=O)C2)CCC2(CC2)N1C(=O)CCc1ccco1 5833,C1(NC(CC2(C)CC2F)=O)CCC2(CC1)CN(C(=O)CCCCC#N)C2 5834,C1(S(N)(=O)=O)(C(N(C2CCC(NC(C=C(C)Cl)=O)CC2)C)=O)CCC1 5835,c1(C(=O)NCCN(CCC)C(C2CCCOC2C)=O)ccc2nc(S)[nH]c2c1 5836,CC(C)(F)C(C)(F)CNC(c1cccnc1CNC(=O)CCC1CCCOC1)=O 5837,C1(n2cc(CCCC)nn2)CCC(NC(C2(O)CC2)=O)CC1 5838,c1(NCC2C(C)(C)CCO2)[nH]c(=NC2CCS(=O)(=O)C2)nc2scnc12 5839,c1(C(=O)OC)ccc(C(N2CCC(NC(=O)CC(C)c3ccccc3)C2)=O)nc1 5840,O=S(=O)(c1ccc(F)cc1F)NCC1CN(Cc2cnc(Br)c(F)c2)C1 5841,C1(NC(CN(C2CC2)CC)=O)CCCC(NC(c2ccnc(C3CCC3)c2)=O)C1 5842,C(=O)(C(C#N)C(C)C)N1C2C(C(=O)NCC(CSC)(C)O)C(C2)C1 5843,C1(CNC(COc2cc(C)on2)=O)COCCN(C(c2cnn(C)c2Cl)=O)C1 5844,C(=O)(C1=COCCO1)NCC1(CNC(C(C(C)C)C)=O)CC1 5845,CC1CCN(C(c2cc(Cl)ncc2F)=O)CC1NC(=O)Cc1cnn(C)n1 5846,C1(NC(c2cc(C3CC3)cs2)=O)CC12CCN(C(=O)CC1CC1(Cl)Cl)C2 5847,c1(C(=O)NCC(CC)NC(c2cc(C)nn2C)=O)ccc2c(C)cc(O)nc2c1 5848,c1(C(N2C(C)CN(C(C3CN(S(=O)(=O)C(F)F)C3)=O)CC2)=O)ccn2cccc2c1 5849,N1(C(C2CC=C(C)CC2)=O)CCC2CN(C(C3CCC(=O)N3)=O)C2C1 5850,n1(CC(=O)N(C)CC2CCCN(C(c3cccn3C)=O)C2)cc(Cl)c(O)nc1=O 5851,C1(C(=O)NC2C=CCCCC2)CN(C(=O)C(F)(F)CO)CC12CC2 5852,c1(C(=O)NCC(C)(C)NC(c2ccc(N)cn2)=O)ncc2cc(Br)ccc2n1 5853,CCC(C)C(O)C(=O)NCC1CC(C)(C)CN1C(C1CC1(F)F)=O 5854,C(=O)(CC(CCCC)NC(=O)Cn1cc(C)cn1)N1C(C#C)COCC1 5855,c1(C(=O)NC(CN(C(=O)C=C(C)C(C)C)CC)C)ccc(O)c(C(C)(C)C)c1 5856,Cc1ccc(NC(=O)CCN(C)C(C2CCCC2(C)C)=O)c(CO)c1 5857,c1(CC(C(=O)O)NC(c2ccc(-c3ccncc3)cc2)=O)coc2ccccc12 5858,C12(NC(CC(C=C)CCC)=O)CCOCC1CN(C(=O)C(F)=CCC)C2 5859,c1(SCCC(=O)NCCC2(CNC(=O)Cn3cnnn3)CC2)ccccc1Cl 5860,C1(C(N2CCC(CNC(C3C(=C)C3)=O)CC2)=O)OC2CCC1CC2 5861,C1(C(N2CCC(COC)(CNC(=O)C(=O)NCC(F)F)C2)=O)OCCCC1(C)C 5862,c1(C(n2ccnc2NCC2CCCOC2)C)cccc(OC(C)(C)C)c1 5863,CC1CN(C(c2occc2Cl)=O)CC1CNC(=O)CCOCC1CCC1 5864,n1(CC(=O)NCC2CCCC2C(=O)Nc2cc(O)cc(F)c2)cc([N+](=O)[O-])cn1 5865,CC(C)CCCCC(=O)NCC1CCC1C(N1CCC(n2cncn2)C1)=O 5866,C12(OC)CCC(C(=O)NC3(CNC(C4CCC(N=[N+]=[N-])C4)=O)CC3)(CC1)C2 5867,C=CC(C)CCN=c1[nH]c(=NCC2(CCO)CC2)c2cc(Cl)ccc2[nH]1 5868,N1(C(C(COC)C)=O)CCC(CC(C)NC(=O)CN2CCNC(=O)C2)CC1 5869,CCCCC(CNC(=O)CC=CC(C)(C)C)NC(=O)CCC(=O)N(C)C(C)=O 5870,C(C(C)C(C)C(=O)NCC(C)CN(C(=O)CC=Cc1ccc(F)cc1)C)OC 5871,C1(O)(CNC(c2ccnc(OC)c2F)=O)CCCN(C(=O)CN2CC=CC2)CC1 5872,N1(C(COCCC=C)=O)CC(O)CC1CNC(c1c[nH]nc1CCC)=O 5873,Clc1cccc2cc(C(c3nnnn3C(C)(C)C)NC3(c4ccsc4)CC3)oc12 5874,N1(C(CC=C=C)=O)CCN(C2CCCN(C(=O)C(C(C)C)OCC)C2)C(=O)C1 5875,C1(C(=O)Oc2cccc3c2OCCO3)COc2c(cc(Cl)cc2[N+](=O)[O-])C1 5876,C1(C(=O)NCC#CC#CCO)CC(O)CCN1C(c1ccc(Cl)cc1)=O 5877,CCCC(O)CC(=O)NC(C)(C)CCCNC(c1cc(-c2ccc(C)s2)[nH]n1)=O 5878,N1(C(c2c(C)n(C(C)C)nc2)=O)CC2CC1CN(C(=O)CC1CC3(COC3)C1)C2 5879,c1(C(C(=O)NCC=CCNC(C2CCC(F)C2)=O)(F)F)c(F)cccc1F 5880,N1(CC(=O)N(C(CN(C(C(C)CC2CCCC2)=O)C)C)C)CCCNC1=O 5881,c1(NC(C(Br)=C(C)C)=O)nccc(C(F)(F)F)n1.C12CCCC1CNC2=O 5882,C1(C(=O)NC(C)CNC(=O)C=Cc2cnc(C)s2)(CC)CCC(O)CC1 5883,C1=CCCC(Nc2ncc(-c3ccccn3)s2)CCC1 5884,C(CC(C)(C)CC(=O)N1CCCN(C(=O)Cc2c[nH]c(=N)nc2O)CC1)OC 5885,N1(C(CNC(C2(CC)COC2)=O)=O)CCN(C(c2cscc2F)=O)CC1 5886,C1(CC)(NC(=O)COc2ccccn2)CCN(C(c2coc(CC3CC3)n2)=O)C1 5887,C1(C(=O)NCc2ccccc2)CC2CN(C(C3(OCC4CC=CC4)CC3)=O)CC12 5888,N1(C(c2ncc(C)c(C)c2)=O)CCC(C)(C)C(C(=O)NC(c2cccnc2)C)C1 5889,c1(CN2C(C(C(=O)Nc3nc(C)c(C)[nH]3)(C)C)CCC2)cc(Cl)ccc1F 5890,C1(C(C)N(C(=O)C(N2CCCC(N3CCN(C)C3=O)C2)=O)CC)CN(C)CCN1C 5891,CCCCCC(O)C(=O)N1CCN(C(c2cnc3occc3c2)=O)C(C(C)C)C1 5892,c1(N2CCC(O)(C(=O)NCC(C)(C)O)C2)ncnn2cccc12 5893,c1(C(N2CC(NC(CCSCC(C)C)=O)C(C)C2)=O)cc2c(Cl)nccc2o1 5894,c1(C(=O)NC2C3CN(C(C4(SCC)CC4)=O)C2C(O)C3)sc2cccnc2c1Cl 5895,C1(CNC(c2cnsc2)=O)CCN(C(c2cn3ccccc3n2)=O)CC1(F)F 5896,Cc1ccc(C(N2CC(C(F)Cn3cc(C4CCCC4O)nn3)C2)=O)o1 5897,CC1(C)C(NC(=O)CCSc2ccccc2)CCN1C(c1cnns1)=O 5898,N1(S(CC)(=O)=O)C2CCC1CN(C(c1ccc(OC)c(I)c1)=O)C2 5899,N1(C(=O)C=CC(F)(F)F)CCC2CN(C(c3cnn(C(F)F)c3)=O)CCC2C1 5900,C1(C(N2CCC(NC(c3cc(COC)sc3)=O)CC2)=O)CCC(C)NC1=O 5901,C=Cc1cc(C(=O)NCC2CCC(C)CN2C(c2nnc(S)n2C)=O)cc(F)c1 5902,N1(C(C2C(CNC(c3cnn4c3CCC4)=O)OCC2)=O)CCC12CCCOCC2 5903,CCCCC(C(=O)NCC1(CCNC(=O)C(CC)C(C)C)CC1)NC(N)=O 5904,c1(N2CCN(Cc3nc(NC(CCC)=O)sc3)CC2)cccc(C(C)OC)c1C 5905,N1(C(c2ccc(Cl)c(N)c2Cl)=O)CCN(C(=O)C2=NOCC2)C2CCCCC12 5906,c1(CCCN2CCCCC2)nc(=NC2CCc3ccccc3C2)[nH]c2c1CSC2 5907,N(C(=NCCc1ncc(C)s1)N1CCCC(CNC(N)=O)C1)C(COC)C 5908,c1(CN(C(c2c(CC)ccs2)=O)C)cnn2c1CN(C(c1c[nH]c(=N)s1)=O)CC2 5909,C(=O)(CCCCC(F)(F)F)NCC(CNC(c1c(C)nn(CCC)c1C)=O)OC 5910,N1(C(CC=CCCCCC)=O)CCCCC1CC(=O)NCC1CCCN1C(C)=O 5911,c1(OC)nscc1C(=O)NC1COCC1NC(C1CC1(C)C)=O 5912,C(=O)(C(CC)CCOC)NC(CNC(C(CC=C)OC)=O)(C)CC 5913,c1(C(N(CC(C)NC(c2cnc(CC)o2)=O)CC)=O)ccc(C(F)F)cn1 5914,N1(C(C(=O)NCC)=O)CCN(C(c2sc(C)cc2OC)=O)C(C2CCC2)C1 5915,CC(=O)CCCC(=O)NC(C(=O)NCCCOC1CCCC1)C(C)C 5916,C(=O)(C(O)CC(C)C)Nc1ccccc1.CCC(C)(C)OCC(=O)NCC1CC1 5917,N1(C(c2ncnc(C)c2C)=O)CCC(N=[N+]=[N-])(C(=O)NCCCS(C)=O)C1 5918,CCC(CC)C(C(=O)NC(C)C(=O)NC(C)(C)CC(C)(C)C)OC 5919,O=[N+]([O-])c1ccc(NCc2cnn(-c3ccccc3)c2)cc1I 5920,N1(C(C2(C)CC(=C)C2)=O)CC2CC2(NC(=O)C=CCCC(C)C)C1 5921,C1(CC)CCCN(C(=O)C(=O)NCC2C(NC(C3(CC=C)CCCC3)=O)CC2)C1 5922,Cc1ccc(O)c(C(=O)NC2CCCC2NC(C2CCN(C)S2(=O)=O)=O)n1 5923,N1(C(=O)Cc2cn[nH]c2)CC(C2CN(C(=O)CCSc3ccc(F)c(F)c3)C2)C1 5924,C1(C(=O)NC(C)Cn2cc(CN3CC4CC4C3)nn2)CCC(=O)C(C)C1(C)C 5925,C1(CNC(Cc2n(C)ncc2Cl)=O)CCN(C(=O)Cn2cnccc2=O)C1(C)C 5926,N1(C(CC(=O)OC)=O)CCCC(O)(CN(C)C(c2cc(Cl)ncc2OC)=O)C1 5927,C1(CC(=O)N(CCCN)C(C(=O)Cn2nccn2)=O)CCCCC1(F)F.C1CC1 5928,N1(C(C(C(C)C)C)=O)CCC(C)N(C(=O)CCCCOCCO)CC1 5929,S(=O)(=O)(c1ccc(OCC(=O)O)c([N+](=O)[O-])c1)NC1C(C)(CC)CCO1 5930,C12(CNC(=O)Cc3csnn3)CCCC1CCN2C(c1ncccn1)=O 5931,n1(COC)ccc(C(N2CCC(CC(=O)N(C)CCN3CCOCC3)C2)=O)n1 5932,C(=O)(CC(C)C(=O)N1CCC(C(=O)NOC2CCC2)C1C(C)C)OC 5933,c12nc(cs1)C(=O)N2C(c1cc(O)cs1)=O.N1(C(C)=O)CCCC1 5934,CC(C#N)CN=C(NCC(c1cccc(Cl)c1)N(C)C)NCC1CCCCC1 5935,Cc1c(C(=O)NCC2(NC(c3csc(C(F)(F)F)c3)=O)CCC2)cnn1C 5936,C(CC(C(=O)NC(C)C(C)OC)NC(=O)CC1CC1)OC 5937,CC12CCN(CC1)CC2C(=O)NCC1CC(NC(c2cc3ncccc3s2)=O)C1 5938,N(C1c2ccccc2CC1C)C(C1CN(c2c(OC)cccc2)C(=O)C1)=O 5939,c1(C(=O)NCC2COCCN2C(=O)CCCF)cc2n(c1)CCCNC2=O 5940,C(N=c1[nH]c(N2CCc3ccncc3C2)nc(=N)[nH]1)C1(c2ccc(OC)cc2)CC1 5941,S(=O)(=O)(c1cnccc1N1CCCC(C(F)F)C1)N(C)CCC(C)(C)C 5942,c1(C(=O)NCC2CCN(C(C)=O)C2)cc2ncncc2s1 5943,N1(C(C2(N(C(c3c(C(C)C)onc3)=O)C)CC2)=O)CC(C#N)C2(CCC2)C1 5944,C(=O)(C(Cc1cn[nH]c1)NC(c1cnc(O)o1)=O)N(CCOC)CC 5945,C1(C2CCN(C(=O)CCC(F)(F)F)CC2)(NC(C2CC(C)(C)OC2)=O)CC1 5946,C1(NC(C2CCC(C)N2C(c2ccnc(O)c2)=O)=O)CCCOC12CCC2 5947,c1(CC)ccc(Br)cc1C(=O)N(C(C)CCNC(C1C(C)(C)C1(F)F)=O)C 5948,CN1CC(NC(=O)NCC23CC(C2)C(C(F)(F)F)O3)Cc2ccccc21 5949,c1(C(=O)NC2CN(S(=O)(=O)CC3CCC3)C2)nc2ccccc2o1 5950,C1(C)(NC(CN(CC(C)C)C(c2ccn(CCC)n2)=O)=O)CCC(C)(C)C1 5951,c1(-n2c(CC3SC(=N)NC3=O)nc(COC(C)C)n2)ccc(Cl)c(F)c1 5952,C1(NC(C(C)CO)=O)CN(C(c2cc3n(n2)CCCO3)=O)CC12CCC2 5953,N#Cc1cncc(CN2CC(NC(=O)Cc3cccc(F)c3)C(C#N)C2)c1 5954,c1(CC(C(=O)NC(C)CCCNC(C2CC2(C)C(C)C)=O)=O)ccc(F)cc1 5955,Cc1ncc(Cl)cc1C(N1CC(N(C(=O)CC2CCCCC2(C)C)C)C1)=O 5956,N1(C(CCc2n(C)ncc2)=O)CCC(C(N2CC(O)(C(F)F)C2)=O)C12CC2 5957,S(=O)(=O)(c1cccc(=NCCCOC(=O)N(C)C)[nH]1)NC1(CC=C)CCCC1 5958,c1(CC)cnoc1C(=O)NCCN(CCC(=O)NC1CC1)C 5959,c1(CC(N2CCC(NC(C3(CCC)CC3)=O)C2C(C)C)=O)ccc(S(N)(=O)=O)s1 5960,c1(C(N2CCC(C(C)(C)NC(CCOC(C)=O)=O)C2)=O)cn(C(C)C)nc1C 5961,c1(OC)cc(C(N2CCC(C(=O)Nc3cccnc3C(F)(F)F)C2)=O)cc(Br)c1 5962,c1(C(=O)NCC2CCCN(C(C3C(C#C)C3)=O)C2)cc2sc(Cl)cc2s1 5963,N1(C(CCC)=O)CCC(OC2CN(C(C3CCCN3C(C)=O)=O)C2)C1 5964,CC(C(C)C(=O)NCc1ccc(CNC(=O)CCS(C)(=O)=O)cc1)C(C)(C)C 5965,c1(CSC)cccc(C(=O)NCCCC(C)NC(=O)CCC2CC2(C)C)c1 5966,c1(OC)ncnc(N2CCN(C(c3ccc(C)nc3O)=O)C(C(F)(F)F)C2)c1C 5967,O(NC(=O)C(CNC(C1CCCSC1C)=O)N(C)C)CCCOCC 5968,C1(n2ccc(C)n2)CCN(C(=NCc2ccco2)NCC2C(C)C2C)CC1 5969,c1(-n2c(C3C(C)C3C)nc(CSC)n2)ccc(F)c(Cl)c1 5970,CC1CCN(C(=O)CC(C2CCC2)C2CCC2)C1CNC(=O)CC1OCCCO1 5971,C1(C)(C(N2CCC(O)(CN(C(=O)C3=CCOC3)C)CC2)=O)CC(C(C)(C)C)=NO1 5972,C12(C(N(C)CC3(CC(C)C)CC3)=O)CC(CNC(c3nnc(S)n3C)=O)(CO1)C2 5973,c1(C(=O)NC2CC(NC(=O)CCc3nccs3)C2)ccc(CO)nc1 5974,c1(NC(C)=O)ccc(CC(O)C)cc1.C(CNC)(CCOC)NC(COCC=C)=O 5975,c1(CC)ccc(C(C)C(=O)NC(C)CC2CN(C(C3CCCOC3C)=O)C2)cc1 5976,c1(C(=O)NC2CC(NC(=O)Cn3ncccc3=O)C2)cccc2c1C(=O)NC2 5977,C1(N(C(CCC#C)=O)C)CN(C(=O)C(CC)CC)CCC1C 5978,S(=O)(=O)(c1cnn(C)c1)NCC(N1CC(N(C)C(C2CCC(=O)N2)=O)C1)=O 5979,CC1CC(C(=O)NC2CCC2C(=O)NC2CCCCCC2C)=NO1 5980,c1(C(=O)NC2(C3CN(C(CSC(C)(C)C)=O)C3)CC2)nn(C)c2c1COCC2 5981,CC#CCCCC(=O)NC1CN(C(C2CCCN2C(=O)NC)=O)CC1C 5982,c1(C(C(N2CCC(c3cn(CCCOC)nn3)C2)=O)C)ccccc1F 5983,C1(C(=O)NC2C=CCN(C(c3nnc(C)s3)=O)C2)Cc2ccccc2C1 5984,C(=O)(C(F)(F)CCn1ccnn1)NCC1(NC(C2C(C)(C(F)F)C2)=O)CCC1 5985,c1(-n2cc(CN(C(CC)=O)C)nn2)c(C)cccc1[N+](=O)[O-] 5986,C(=O)(C(CC(F)F)N(C)C(c1ccc(C)nc1)=O)NC1CCCC(OC)C1 5987,C1(OCC(=O)NC2CN(C(C3(C(F)(F)F)CCOCC3)=O)C2)(CO)CCOCC1 5988,c1(OCC)ccc(OCC)c(NC(=O)NC2CCNC2C)c1 5989,CC(C(=O)NCCOCCCNC(C1CC(=O)NC(=O)N1)=O)C(C)S(C)(=O)=O 5990,n1(CC)cccc1C(=O)NCC(CCNC(c1ccc(CO)o1)=O)OC 5991,C(=O)(C1=CS(=O)CCC1)N(CCCNC(C(CC=C)C)=O)Cc1cccnc1 5992,c1(C(N2CC(NC(CC(CC)CC)=O)C(C)C2)=O)ccc2c(c1)N(C)CC2 5993,C(C(=O)N1Cc2ccccc2CO1)C1(C=C)CN(C(=O)C(=O)NC(C)C)C1 5994,Cc1ccc(N(C(=O)CC2CCCN2C(C2CC3CC3C2)=O)C)c(C)c1 5995,c1(CN2CC(C#N)C(NC(c3ccc(S)cc3)=O)C2)cc(Br)cc(F)c1F 5996,c1(C(=O)NC2(CC)CN(C(=O)CN3CCCCC3=O)C2)ncncc1C 5997,N1(C(C(C(=O)OC(C)(C)C)OC)=O)CCC(C(=O)NCC2CCC2)CC1(C)C 5998,N1(C(C(C)NC(=O)OC)=O)CCOCC1C(N1CC(F)(F)C1C1CC1)=O 5999,c1(C(=O)Nc2cccc(OC)n2)c[nH]c2ccc(-c3cc(C)c(F)cc3F)cc12 6000,C(=O)(C1=NN(C2CC2)C(=O)CC1)C(CCCC(=O)NC(CC)CN)=O.OC 6001,C(=O)(C1CCCn2nccc21)N1CC2N(C(c3cc(C)cc(Cl)c3)=O)C(CC2)C1 6002,C(N=c1[nH]c(N(C)CCC2CCC2)nc2ccc(Cl)cc12)c1n(CC)cnc1 6003,Cc1cc(CNC(C2CC(C)N2C(=O)CCC2(C)CC2)=O)ccc1F 6004,CC(C)CC(C(=O)O)NC(C1CCCN(C(c2ccnn2C)=O)C1)=O 6005,c1(CC)nc(CNC(C2CC(NC(=O)C(C)OCC(C)C)C2)=O)cc(O)n1 6006,c1(C(=O)NCc2scc(CC(=O)O)c2)cc2c(nc1O)CCC2 6007,c1(C(=O)NCC(=C2CN(C(C(C)OCCC=C)=O)C2)F)ccc(C(C)C)cc1F 6008,N1(C(C(COC)OC)=O)C2CCC1CC(NC(c1ccccc1SC(C)C)=O)C2 6009,C1(NC(C(CSC)C)=O)COCCN(C(=O)C(c2ccc(F)c(F)c2)(C)C)C1 6010,CCC(CC)CC(=O)NCC1CC1NC(=O)COc1ccc(C(C)C)cc1 6011,c1(C(N2CCCOCC2)C(=O)NCCCC(=O)OCC)nc(C)c(Br)s1 6012,C1(CC(=O)NCc2cn[nH]c2)CCN(C(C2CCO2)=O)CC1 6013,N1(C(CCSCCC)=O)CC(NC(c2c(C)csc2Cl)=O)CC1(C)CC 6014,C(=O)(CCCC(=O)N1C(C(N2CCC3CCCC23)=O)CC1C)OC 6015,C1(C(=O)NCCCCNC(=O)C=Cc2cccnc2)CCC(=O)N2CCCC12 6016,N1(C(C2CC23CCC3)=O)CC2CCC(C1)N2C(=O)C(O)CC1CCCCC1 6017,CCC(C)(O)CNC(=O)CCCC1(NC(=O)COCCF)CCC1 6018,Cc1nc(C(N2CC3CC2CN3C(C2CCN2S(C)(=O)=O)=O)=O)c2ccccn12 6019,C1(C)(C(=O)NC2C(NC(C(c3ccccc3)OCC)=O)CCC2)CC=C(C)CC1 6020,c1(N(CCOC)C)cccc(S(=O)(=O)N2CCSC(C)C2C)n1 6021,CCCCC(CN=c1[nH]c(Cl)nc(CC)c1Cl)NC(=O)CSc1ccccn1 6022,C(CCCCC(=O)NCC1(O)CCCN(C(=O)CC2CC(F)C2)C1)OCC 6023,C1(N(C(c2cncc(C)n2)=O)C)CCCN(C(c2cc(Br)nn2C)=O)CC1 6024,c1(C(=O)NC(C(=O)NC(C=C)CO)c2ccco2)cnccn1 6025,S(=O)(=O)(c1c(F)cc(F)cc1F)Nc1scc(CC(=O)Nc2cccc(Br)n2)n1 6026,CCCCC(C(=O)NCc1cc(C2CC2)no1)NC(C1OCCC1(C)C)=O 6027,n1(CC(=O)Nc2cccc(C(N(CC)CC)=O)c2Cl)c(C)cc(C)nc1=O 6028,c1(C(=O)NC2CN(C(C3C(C)CCC3)=O)CC2F)cn2ccc(Br)cc2n1 6029,C1(O)(CN(C(CCSCCC)=O)C)CCN(C(c2n[nH]c(C3CC3)c2Cl)=O)C1 6030,C=CCC(CC)C(=O)N1CCN(C(=O)CN(CC)CC)CC1CC(F)(F)F 6031,C1(C(=O)NC(C)Cc2nc(-c3ccccc3)no2)CC(O)C(O)C1 6032,N1(CC(C)C)CCC(C(N2CCCC(CN(C)C(C3(CO)CC3)=O)C2)=O)CC1 6033,Cc1cc(C(=O)NC2CC(NC(C3CNC(=O)N3)=O)C2)c2sc(=N)[nH]c2n1 6034,N1(C(C2CCN2C(=O)Cc2ccc(Br)cc2)=O)Cc2cccc(F)c2C1 6035,Cc1nc(C(=O)NCCC2CCCN2C(=O)CO)ccc1Br 6036,c1(N2CCC(CNC(=O)CCOCC3CCCO3)C2)ncc2ccccc2n1 6037,c1(C(=O)NC2CCN(C(C(C3CCC3)OC)=O)C2C(C)C)coc(S(C)(=O)=O)c1 6038,C1(C(=O)NCC2=CCN(C(CCC3CCC(=O)N3)=O)CC2)CCn2ncnc2C1 6039,N1(C(CC2(C=C)CC2)=O)CCCC2(NC(C3CCC(C(N)=O)CC3)=O)CC2C1 6040,c1(C(=O)NC2CN(C(c3cocn3)=O)C3CC23)cc2scc(Cl)c2[nH]1 6041,C1(C(=O)NC2CC(NC(=O)CCC3CCCCC3)C2)CCCN(C(=O)C2CC2)C1 6042,c1(CC)nn(C)cc1C(=O)NCC1(C)CCN(C(c2cnc(C)o2)=O)C1 6043,CCCCC(CNC(=O)CCCC1CCCC1)NC(=O)CC(C)C1CC1 6044,C(N=c1nc(N2CC3(C2)CC3(F)Br)c2[nH]ccc2[nH]1)c1ncn(C)n1 6045,c1(C(=O)NCC2CC(CNC(c3cnc(C)s3)=O)OC2)c(C)cccc1Cl 6046,N1(C(C(CC)F)=O)CCCC2(CCCCC2NC(=O)C(N2C(C)CCC2C)C)C1 6047,Nc1c(F)c(F)cc(C(N2CC3CC2C3NC(=O)Cc2cccc(F)c2)=O)c1Cl 6048,CC(CCC(=O)Nc1cn(C)nc1C(N)=O)NC(C1(CO)COC1)=O 6049,c1(OCC)ccc(C)nc1C(=O)NC(C)CCNC(c1cc([N+](=O)[O-])c[nH]1)=O 6050,c1(C(=O)NCC(CNC(C=NOC)=O)F)cc2ccc(F)cc2s1 6051,Cc1cc(F)c(C(=O)NC2CC(CCNC(C3CCOC3C)=O)C2)cc1F 6052,C1(C2CC2)(C(=O)NCCCCNC(=O)C=CCN2CCOCC2)CCC1 6053,C(=O)(C1SCCc2sccc21)N1CCC2(CC(NC(=O)CC=C(Cl)Cl)C2)C1 6054,c1(C(=O)NC2C(NC(=O)OC(C)(C)C)CCC2)ncc(Br)cc1O 6055,C1(C(N2CC(O)(CCNC(c3cn(CC)nc3)=O)C2)=O)CCc2nnn(C)c2C1 6056,O=C(C(F)C1=CCCCC1)NCC1CC2CCC1N2C(=O)CCC1CCCOC1 6057,c1(C(=O)NCCC2CCN(C(CCC(=C)Br)=O)C2)ncc(N)cc1Cl 6058,c1(OCC)nccc(C(=O)NCC(C)(CO)NC(=O)C=C(CC)CC)c1F 6059,Cc1nc(CO)ncc1C(N1CCC(NC(C2C(C)OC(C)C2C)=O)C1(C)C)=O 6060,c1(C(N2CCC(C#N)(NC(C(C(C)C)=O)=O)C2)=O)cnc2ccccn12 6061,C(=O)(C1=CC2(CCOCC2)C1)NC1CC(C)N(C(=O)C=C2CCCC2)CC1 6062,S(=O)(=O)(c1cccnc1NC1CCCC1CO)N(C1(C)CCCC1)CC 6063,C1(C)(CNC(C(C2CC=CCC2)NC(c2cnc(C)o2)=O)=O)CCN(C)C1 6064,C1(C(=O)NCC2C(NC(c3nc(C(C)=O)sc3)=O)COC2)CCN(CC)C(=O)C1 6065,C=CCCCCCCCC(=O)N1CC2CC1CC2NC(=O)C1CC1 6066,N1(C(C(C)CC2CCCO2)=O)C2CCC1CN(C(=O)CN1CC(C)(N(C)C)C1)C2 6067,c1(C(=O)NC(C(C)NC(Cc2c(C)n[nH]c2C)=O)(C)C)cnn2c1OCC(C)C2 6068,c1(CC2(C(=O)NC3CC(O)(CNC(C4CCCO4)=O)C3)CC2)cccc(F)c1 6069,N1(C(C(c2cn(C)nc2)=O)=O)CCC(C(=O)NC2CC=CC2)C1C(C)(C)C 6070,C(=O)(C(CNC(=O)C1=C(C)OCC1)C(C)C)NCc1cnc(CC)s1 6071,C1(CNC(c2n(C)ncc2)=O)CC2CC1CN2C(c1ccc(C(F)(F)F)cn1)=O 6072,Cc1nn(CC(N2CC(NC(c3ncc(F)cn3)=O)C(C)C2)=O)cc1Br 6073,C1(NC(C(n2ncc(C)c2)C)=O)CCCCC1NC(=O)C=Cc1ccoc1 6074,C(=O)(C(F)(CNC(c1cccc(=O)o1)=O)C(C)C)NC1(C(=O)OCC)CC1 6075,N1(C(C=C(CC)C)=O)CCN(C(=O)COC2CC(F)(F)C2)CC1CC 6076,N1(c2cc(N(C)CC3CCN(C)C3)ncn2)CCOC(C)(c2ccccc2)C1 6077,C(=O)(C(C)(C)C(=O)Nc1ccc(F)c(F)c1)NC1CC(C)N(C(C2CSC2)=O)C1 6078,c1(C(CC)C)ccc(C(=O)NCC(C(C)C)NC(C2(O)CC2)=O)c(O)n1 6079,c1(C(=O)NC(C)(C)C=CC(N2CC(N(C)C3CC3)C2)=O)n[nH]c(=N)[nH]1 6080,C1(C2CC2)(C(=O)NCC(CC=C)NC(=O)C(CC)C(C)C)CCOCC1 6081,c1(NC(c2ccc(OC=C(F)F)cc2)=O)cccc(-c2nc(O)n[nH]2)c1 6082,c1(COC)cc(N(CC(C)CNC(C2CCCOCC2)=O)C)nc(SC)n1 6083,CCCCC(CN1CCCC(C(N2CCCC(CO)C2)=O)CC1)CC 6084,CP(C)(=O)C1CCCN(C(=O)N(C2CC2)Cc2ccncc2)C1 6085,N1(C(C(CC2CC2)NC(C2CCCN2C2CC2)=O)=O)CC2(CCC2)C1 6086,N1(C(C(C2CC2)OCC)=O)CCC2(CCCN2C(c2cc(N)c(Cl)cn2)=O)CC1 6087,C1(NC(CCC(C)OC)=O)CC2CCC(C1C)N2C(=O)C1=CCCCO1 6088,C1(CNC(c2[nH]nnc2C2CC2)=O)CN(C(=O)CCc2ccccc2O)CCO1 6089,CC1=CCSC1C(=O)NC(C1CCN(C(=O)CC2CCCC2O)C1)(C)C 6090,C1(CC=C)(NC(C2(CN(C)C)CC2)=O)CCN(C(c2nc(Cl)c(CC)[nH]2)=O)CC1 6091,C1(N(C(c2cn(C3CC3)nn2)C(=O)NCC(=C)C)C)CS(=O)(=O)C12CCOCC2 6092,N(C1c2ccccc2CC1NC(c1ccnnc1)=O)C(C(C)(C)N1CCCC1)=O 6093,CCCC(CC)C(=O)NC1CN(C(=O)C2=NNC(=O)C2)CC1SC 6094,C1(NC(C(CC)CO)=O)CC2CN(C(=O)C(c3ccccc3F)(F)F)CC2C1 6095,N1(C(C(C)N(CCC)C(C2CC(NC(C)=O)C2)=O)=O)CCOC2C(O)CC12 6096,C1(NC(C(CC=C)C)=O)CC(OC)CN(C(c2cc(C)n(CC)n2)=O)C1 6097,C=CCCC(C(=O)N1CCCC1COC)NC(=O)C(CN(C)C)N(C)C 6098,C1(NC(c2c(OC)csc2)=O)CC2CN(C(c3ccc(CO)s3)=O)CC2C1 6099,N1(C(COCC=C)=O)CCC(CNC(c2cccc(C)c2)=O)C12CCC2 6100,CC1(C)C2CC1CN(C(=O)CC(=O)NCC(F)(F)F)C2 6101,C1(CNC(c2c(C)nsc2)=O)(CNC(c2cc(C)n(CCO)n2)=O)CC12CCC2 6102,S(=O)(=O)(CC(=O)NC(C)C(c1ccccc1SC)N(C)C)N(CCON)NCC 6103,C1(C(=O)Nc2cnn(CC(C)C)c2C(C)C)C2Cc3c(Br)cccc3C12 6104,C1(CNC(C(C)NS(C)(=O)=O)=O)CCC2(CN(C(=O)Cc3cnccn3)C2)O1 6105,N1(C(CC=CC)=O)CC=CC(NC(c2ccc(C3CCC3)nc2)=O)C1 6106,Cc1ccnc(C(N2CCC(N(C(=O)C(N3CCCCCC3)C)CCO)C2)=O)c1N 6107,Cc1cncc(C)c1-c1noc(-c2ccc(OCC(F)(F)F)cn2)n1 6108,C(CCCCCN(C(=O)CCn1ncn(C)c1=O)C)NC(C1(CC)CC1(F)F)=O 6109,C(=O)(CCN1C(=O)C(C)Oc2ccccc21)NC(CC)C(=O)NC 6110,n1(CC(=O)N(C2(N3CCOCC3)CCCOC2)CC)c(C)nc2ccccc12 6111,N1(C(C2CCSCC2)=O)CCOC2CN(Cc3nccc4ccccc34)CC12 6112,N1(C(C(C)n2cccc2)=O)CCC2(CC2)CC1C(=O)NCCN1CC=CC1 6113,O(NC(=O)C(O)C1CN(C(c2ccc(=N)[nH]n2)=O)C1)CCCOC 6114,C(=O)(N=c1[nH]n(-c2ncccn2)cc1I)c1ccc(-c2n(C)cnc2)cc1 6115,C#Cc1ccc(CNC(=O)C(C)C(C)NC(=O)CCN2CCOCC2)cc1 6116,n1(CC(=O)NC(C(C)NC(CC(C)F)=O)(C)C)c(=O)cnc2ccccc12 6117,N1(C(C(CC)NC(=O)C(=O)NCC2CC2)=O)CCOC(C)(C)C1C 6118,Cc1sc(-c2nc[nH]n2)nc1C(N1CC(O)(C(C)NC(C2CC2C)=O)C1)=O 6119,N1(C(C2C(C)(C)CC2)=O)CC2CN(C(c3ccnc(S)c3)=O)CC2(C)C1 6120,c1(OC)ncc(Cl)cc1C(=O)NC1CN(C(C2CC(=C3CC3)C2)=O)CCC1C 6121,C=CC(C)(CCOC)C(=O)NCC1COCCN(C(c2ccc(NC)cc2)=O)C1 6122,c1(CNC(c2c(C)noc2C)c2nnnn2C2CC2)ccc2c(c1)OC(C)(C)O2 6123,C1(C)(C(N(C)CC2CCN(C(C3(C)CCCC3)=O)C2)=O)CCCNC1=O 6124,n1(CC)ncc2c(C(=O)OC(C3CCCCC3)C(=O)OC)cc(C)nc12 6125,c1(C(=O)NCCN(C(C(C)Oc2ccc(C(C)=O)cc2)=O)C)cnc(C)c(Cl)c1 6126,C=CC(C)(C)CC(=O)NC1CC(C)N(C(=O)C(O)Cc2cnc[nH]2)C1 6127,Cc1cc(C(=O)NCc2ncc3n2CCC3)n2ncc(-c3nn[nH]n3)c2n1 6128,Cc1cc(NC(=O)NC2CCCC23CC3)cc(Br)n1 6129,c1(C(=O)NC(CN(C(c2cc(OCC)ncc2)=O)C)C)cc(F)c(N)cc1F 6130,Cc1nccc(NCC2CCCN(C(=O)CCc3ccc(C(C)(C)C)cc3)C2)n1 6131,C12(C(=O)NCCC3(C)CCCO3)C(NC(c3ccoc3)=O)C3CC1C2C3 6132,C1(NC(c2cn(C3CCOC3)nn2)=O)CC2CC1CN(C(=O)C(F)(F)C1CC1)C2 6133,c1(N2CCN(C(=O)CC3CCCS3(=O)=O)CC2)ncnc2ccc(O)cc12 6134,C(CC(C(=O)N1CCC1C1CCCC1)NC(=O)CCc1ccsc1)=CC 6135,CC1CCCC=C1C(=O)N1CCCC(F)(C(=O)NC(c2cncn2C)CO)C1 6136,CCCCCS(=O)(=O)CC(=O)NCC1(C)CCCN(C(=O)CC(=O)N(C)C)C1 6137,C1(C)(C(N2CCC(OCC#C)CC2)=O)CN(C(c2ccn(C)c(=O)c2)=O)CC1C 6138,c1(OC(C)C(=O)NC2CC2CNC(=O)Cc2ccc(O)nc2)ccc(Cl)c(Cl)c1 6139,N1(C(C2C(C(C)C)CN(C(=O)CS(C)(=O)=O)C2)=O)CC2CC(CO)C(C2)C1 6140,C1(C)(C(=O)NCCCNC(C(C)=C2CCC2)=O)CC2CCC(C1)S2 6141,N1(C(C2(C)CC(=O)C2)=O)CC2(CO)CC1(C(N1CCCC(F)(CO)C1)=O)C2 6142,C1(CNC(C(=O)NCC)=O)CN(C(C23CCC(F)(CC2)CC3)=O)C2CCN1C2 6143,CC1(C(=O)Nc2ccccc2)CC12CCN(C(C1(COC(C)(C)C)CC1)=O)CC2 6144,C1(CC(=O)NCCC(F)(F)CO)CCCC(NC(c2cscc2Cl)=O)C1 6145,C1(NC(COCc2ncc(C)o2)=O)CCCC(NC(=O)CC(C)F)C1 6146,C1(CNC(C(C)(C)F)=O)CN(C(c2cnc(-c3ccccc3)s2)=O)CCC1(F)F 6147,N1(C(=O)CCOc2ccccc2Br)CCCC2(CCN2)C1 6148,N1(C(COC(C)(C)C)=O)CCN(CCCNC(C2CC2(Cl)Cl)=O)CC1 6149,CN1CC=C(CC(=O)NC2CCC2NC(c2cc(Cl)c(Br)[nH]2)=O)CC1 6150,C1(OC)CN(C(=O)C=C(C)C(C)C)CCC1NC(=O)C(C)(C)c1csc(C)c1 6151,CC(C)(C(=O)NC(CNC(=O)CCCC1CC1)CC(F)(F)F)C1=CCSCC1 6152,N1(C(C(CC(C)C)C)=O)CC2CCCC(N(C(=O)COCCCF)C)C2C1 6153,CCC(O)C(C)(C)C(=O)NC1CCCC1NC(c1cccc(OC)c1O)=O 6154,C1(C(=O)NC(C=C)(C)CC)CCN(C(c2cccc(OC)c2O)=O)CC1(C)C 6155,CC(C(=O)NCc1noc(C(F)F)n1)(C1CCC1)NC(=O)Cc1ccc[nH]1 6156,C#Cc1cncc(C(N2CC(C)CC2C(N2CCCC(OC)CC2)=O)=O)c1 6157,CN1C(=O)CCCC1c1nc(-c2cccnc2O)nn1C1CCCC1 6158,Cc1cc(C(N2CC(NC(=O)CC3CC3)C3CC3C2)=O)c(C)n1-c1cnccn1 6159,C1(COC2(C#C)COC2)COCCN(C(=O)CC(CC)NC(C2(OCC)CC2)=O)C1 6160,C(C1C(C(=O)NC2CC(CNC(=O)CCc3cc(C)sc3C)C2)C1(C)C)=C(C)C 6161,C1(NC(c2c(CCC)n[nH]c2)=O)CN(C(=O)CC#N)CCC12CCC2 6162,n1(CC(=O)NC2CC(C)(NC(CC=C=C)=O)C2)nc(C)c([N+](=O)[O-])c1C 6163,Cc1cnc(F)c(NC(=O)C(=O)NC23CC(c4ccccc4)(C2)C3(C)C)c1 6164,C(CCCCCC(=O)NCc1ccnc(F)c1)NC(C1(CC#C)CCC1)=O 6165,Cc1ccc(C(=O)NCC(O)CNC(=O)C2=C(Cl)CCOC2)c2cccnc12 6166,c1(CNC(CC(C)NC(c2nc(OCC)oc2)=O)=O)ccc(F)cn1 6167,C(=O)(CC(CC)C(C)(C)C)NC(CCC)C(=O)NCCS(=O)(=O)NC 6168,N1(C(COCCC(C)C)=O)CC2CCN(C(c3cn(C)c(O)n3)=O)C(C2)C1 6169,c1(C(=O)NCC(C)NC(=O)C(C)CC2CCC2)c[nH]ccc1=Nc1cnn(C)c1 6170,C#Cc1cc(C(=O)NC(C2CCCN2C(c2cc(CC)nn2C)=O)C)cc(F)c1 6171,CCCCCCOCC(=O)NC1CC(CCNC(=O)C=CC(C)CC)C1 6172,CCCCC(O)C(C)C(=O)N(CC(C)NC(=O)C=CC(F)F)C 6173,c1(NC(C2CCN(C(CC=CCC)=O)CC2O)=O)ccc2c(c1)CCO2 6174,C(=O)(CC(F)(F)C(F)(F)F)NCC1(NS(CCCOC)(=O)=O)CCN(C(C)=O)C1 6175,c1(NC(=O)NCCCNC2CNC(CO)C2)ccccn1 6176,c1(CCC(=O)N(C)CC2CCN(C(CC(=O)OC)=O)C2)cc(C)cc(C)c1 6177,C(=O)(C(O)CCC(C)C)N1C2CCC(NC(C=Cc3ccc(SC)s3)=O)(C2)C1 6178,N1(C(COCc2cc(C)on2)=O)CCC(C)CC1CNC(c1ccc(C#N)s1)=O 6179,c1(OC)c(C)csc1C(N1CCC(CCNC(=O)CC(C)n2cccc2)C1)=O 6180,C(C(C)(O)CC(=O)NC1CCC(NC(=O)Cn2nnc(C3CC3)n2)CC1)OC 6181,C12(NC(c3c(SC)n(C)nc3)=O)CCCN(C(c3cccc(Cl)c3C)=O)CC1C2 6182,n1(C(C)C)ccc(C(N2CCCC2CN(C(=O)CCOCC2CCC2)C)=O)n1 6183,N1(C(c2ccc(CNC(C3CN(C4CCC4)C3)=O)nc2)=O)CCC2CCCCC2C1 6184,C1(C(=O)NCC(C)(C)CCO)CCOCCN1C(C1CC(C)(C)CO1)=O 6185,Cc1c(C(=O)N(C2CC2)CC2CCOC2)sc2cc(F)ccc12 6186,N1(C(CC=C)=O)Cc2n[nH]cc2C1C(=O)NCC(F)Cl 6187,Cc1cc(C)n(C2CCCN(C(c3nnc(C(C)C)s3)C(=O)NCC(C)C)C2)n1 6188,CCCCCCC(=O)NC(c1nc(C(=O)NC(CC)CC(F)(F)F)co1)C 6189,Cn1ccnc1CC(=O)NCC(C)(C)n1ccnc1.C12(CC1)CC(=O)NC2 6190,c1(NC(CN(C(Cc2ccc(C)nc2)=O)C)C)ncc([N+](=O)[O-])cc1C#N 6191,c1(C(N2CC(C(=O)NC(C#CC)(C)C)N(C)CC2)=O)coc2ccccc12 6192,C1(C(N2CC3(CCC3NC(C3CC=CCC3)=O)C2)=O)(CC)CCC(F)(F)CC1 6193,Cc1noc(C)c1C(N1CC2(NC(C3CCC3C)=O)CC1C2)=O 6194,N1(CC(N2CCC(CCNC(c3cc(C)on3)=O)C2)=O)CCC(F)(F)C1 6195,Cc1ccc(C(=O)N(CCN(C)C(c2coc(Cl)n2)=O)C(C)C)nc1 6196,Cc1cccc(F)c1CC(=O)NC1CC(N(C)C(c2c(C)ncn2C)=O)C1 6197,Cc1noc2ncnc(NC(C)CCNC(C3CCC(O)CC3)=O)c12 6198,C1(C(=O)NC(C)CNC(=O)CCC(N)=O)CC2(CC(NC(=O)OC(C)(C)C)C2)C1 6199,c1(NC(=O)OC)cc(C(=O)NC(C)(C)CCCNC(=O)C=CCO)ccc1F 6200,C1(C)(CNC(c2c(C)ncs2)=O)CCCN(C(=O)Cc2csc(NC=O)n2)C1 6201,Cc1cncc2cc(C(N3CCCOC(CNC(=O)Cc4csnn4)C3)=O)sc12 6202,N1(C(c2snc(C)c2N)=O)CCCN(CCNC(C2CN(C)C2)=O)CC1 6203,O=C1CCC(C(=O)N2CCC(NC(c3cc(C(F)(F)F)cc(Cl)c3)=O)C2)=NN1 6204,N1(C(C(F)=C(C)C)=O)CCC2CN(C(c3cc(Br)n(C)n3)=O)CC2C1 6205,C1(NC(C2CC3CC2C3)=O)CCCCN(C(c2cc3occc3[nH]2)=O)C1 6206,N1(C(c2c(N)cccn2)=O)CCC2(CCOC2)C(CNC(c2csc(Cl)n2)=O)C1 6207,C12(CNC(C(COC)O)=O)CCCCC1N(C(c1cc(OC)nn1C)=O)CC2 6208,C1(C(N2CC(CNC(C(C)C)=O)C2)=O)(N(C)C)CCCCC1 6209,C(=O)(C(CC(C)(C)C)NC(=O)C(C1(O)CCCC1)F)N1CC(SCC)C1 6210,C(CCCCNC(=O)COCC(C)(C)C)N(C(CCC1CC(C)C1)=O)C 6211,c1(C(=O)NCCN(C(=O)C(n2ccc(C3CC3)n2)C)CC)ccc(C)c(C)c1N 6212,c1(-c2c(C(=O)NCC(CNC(c3c(CC)noc3)=O)O)c[nH]c2)ccccc1F 6213,C1(COC)CC(O)CN1C(=O)C(CC1CCCC1)NC(=O)Cn1ncccc1=O 6214,N1(C(CCn2ccc(C)n2)=O)CCC(C(F)F)(CNC(=O)Cc2cc[nH]n2)C1 6215,C=CCCC(=O)NC(CNC(C1CN(C2CCOC2)C1)=O)C1CCC1 6216,CCCCCCC(C)C(=O)N(C1CN(C(c2cc(C#N)cn2C)=O)CC1(C)C)C 6217,C(=O)(C#CC1CCCO1)NCC1(C(C)NC(c2c(C)nn(C(C)C)c2C)=O)CC1 6218,c1(CCNC(N2CC(CC)C(c3cnn(C)c3)C2)=O)cc(C)ccc1Br 6219,C1(C(N(C2CN(C)CC2O)C)=O)CCCC(NC(=O)C=CCN2CCCC2)CC1 6220,c1(C(=O)NC(C(C)C)C(=O)N(C2CCCCC2)CC)cc2c(O)cc(Cl)cc2[nH]1 6221,C(=O)(C(CO)C(C)C)NC(CNC(CCn1c(C)cc(C)n1)=O)(C)C1CC1 6222,C(CC(C(C)C)NC(c1cscc1C(=O)OC)=O)N(C(C=C(CCC)C)=O)C 6223,N1(c2nnc(CSc3cccc(NC)c3)n2CCN(C)C)CCCC2(CCC2)C1 6224,c1(C(=O)NC(CN(C(COCCOC)=O)CC)C)cc2n(n1)CC(C)NC2=O 6225,C1(CC=C)(NC(=O)COC(C)(C)C)CCN(C(=O)NC2CC2CC)CC1 6226,N1(C(c2c(CC)n(CC)nn2)=O)CC(C)CN(C(C23CC(C2)C3)=O)C(C)C1 6227,c1(CCC(=O)NC2(CN(C)C(C3CC(N(C)C)C3)=O)CC2)cccnc1 6228,C1(NC(c2nc(CC)oc2)=O)CC12CCN(C(=O)Cc1ccoc1C)CC2 6229,N1(C(C(CCN(C)C)NC(CC2C(C)C(=O)CC2)=O)=O)CC2CSCC2C1 6230,c1(CNC(CN(C(=O)C=C2CCC2)C(C)C)=O)ccc(CO)o1 6231,N1(C(C(CC)OCC)=O)CCN(C(=O)CCCOc2ccc(F)cc2)CC1CF 6232,C(=O)(C1=CCCCC1P(C)(C)=O)NCC(C)CNC(=O)CCC#N 6233,CCCCCC(C)(CC)C(=O)NC1CCCCC2CN(C1)C2=O 6234,N1(C(CCC(C)OC)=O)CCC(C)C(CNC(c2cccc(F)n2)=O)C1 6235,C(C(C)C)(C(O)C(=O)NC(C)C(C)(C)C(=O)NCC1CCOC1)OC 6236,C(CC(=O)NCCSCCCO)(C(F)(F)F)NC(=O)C(c1ccccc1)F 6237,CCC(C)(COC)C(=O)N1CC=CC(NC(=O)C(C)(C)C(F)F)C1 6238,C1(C(=O)NCC(C)(CO)NC(Cc2c(Cl)cn(C)n2)=O)CCCCC(F)(F)C1 6239,C(=O)(C(O)CC1CCOCC1)NCCN(C(=O)CCOC(C)CC(C)C)CCC 6240,Cn1nncc1C(=O)NCC1(NC(=O)CCN2CCCC2=O)CCOC1 6241,c1(C(=O)NCCN(CCC)C2CC2)cc(Cl)ncc1F 6242,c1(C(=O)NCC(C2CC2)NC(c2cccnc2S)=O)cc2ccsc2s1 6243,N1(CC)CC(C(=O)NC2CC3CCC2(NC(=O)CCn2ccnc2)C3)CCC1=O 6244,c1(C(=O)NC2C(NC(CC(CC)CC)=O)CC2)cnc2ccoc2c1 6245,C=CCCCCC(=O)NCC(O)CCNC(=O)C(CCCC)NC(N)=O 6246,N1(C(c2c(CC)c[nH]c2)=O)CC(NC(c2sc(Br)nc2C)=O)CC1C 6247,c1(C(N2CCC(CNC(CSc3cn(C)nc3)=O)C2)=O)cccc2oncc12 6248,CC(CCF)N=c1nc(N(C)C2CC2)c2cc(OCCOC)ccc2[nH]1 6249,C=C(C)CN=C(NCc1cccc(C(=O)N(C)C)c1)NC1CCCCC1C 6250,Cc1cc(OCC(=O)NC2CN(C(=O)CC(=O)N(C)C)CC2C)ccc1F 6251,c1(C(=O)OC)c(C)[nH]c(C(N2CC(NC(=O)C(C)CSc3ccccc3)C2)=O)c1C 6252,N1(C(=O)C(O)CC)CCCC1(CNC(c1c(OCC)scc1)=O)CC 6253,O=S(=O)(c1c(Cl)ccc(Br)c1Cl)Nc1cc(CO)cc(Br)c1 6254,c1(CC(=O)NC(C)C(C)NC(c2ncccn2)=O)ccc(N2CCCC2=O)cc1 6255,CCC(CC)C(C)C(=O)NCC(C1CCN(C(c2nc(C)n(C)c2C)=O)CC1)C 6256,C1(C(N2CCC(NC(C3CC(F)(F)C34CCC4)=O)C2)=O)Cc2ccccc2C1 6257,Cc1ccnc(C=CCNC(C2CCN(CC3CN(C)C3)C2)=O)c1 6258,N1(C(C2C(C)C2C)=O)CCCC(C2CCN(C(C3(O)CCCCC3)=O)C2)C1 6259,c1(NCC)ccc(Cl)cc1C(=O)NCC(F)CNC(C1CC2CC1CO2)=O 6260,N1(C(c2cccc(C(F)F)c2)C(=O)Nc2c(C)cccc2)CCS(=O)C(C)(C)C1 6261,C(=O)(CC=C(Cl)Cl)NCCC(C)N(C)C(c1ccccc1OCC1CCCO1)=O 6262,CSC1=C(C(=O)NCC(O)CNC(=O)CCCCCCCC2CC2)CCCC1 6263,N1(C(CC2CCN(OC)CC2)=O)CCCC(O)(CNC(c2ccncc2)=O)CC1 6264,N1(C(C(C)CN(C)C)=O)CC2CCC1C(CNC(C1(C3CC3)CCCO1)=O)C2 6265,c1(C(N2CCC(n3cccn3)C2)C(=O)NC(CC)C)cc2ccc(OC)cc2o1 6266,C(=O)(C(C(F)(F)F)C(F)(F)F)N1CC2(OCC(NC(C(CC(N)=O)O)=O)C2)C1 6267,c12ccc(c(C)c1)S(=O)(=O)N2.C1(C(=O)OC)C(Cl)(Cl)C12CC2 6268,c1(C(=O)NCCCOCC=C)cc(CNC(=O)CCCF)ccn1 6269,N1(C(c2cccc(C(F)(F)F)c2O)=O)CC2CN(c3ncccn3)CC2C1 6270,CCC(C(=O)NC(C)(CNC(C1CCOC1=O)=O)C1CC1)OC 6271,C(C(C(=O)N(CCN(C(=O)C(C)(C)c1cnn(C)c1)C)C(C)C)N(C)C)OC 6272,c1(C(=O)NCC2CCCN2C(C2(O)CCOCC2)=O)cccc(Br)c1F 6273,c1(CC)cc(C(=O)NC(C2CCCC2)CNC(C2CC3CCC3C2)=O)cc(O)n1 6274,C12(C(=O)OC)CC(C(=O)NCC(CNC(=O)CN3CCC3C)CO)(C1)OC2(C)C 6275,C(=O)(CCC(C)(C)N(C)C)N(CCCNC(Cc1c(C)n(C)nc1)=O)CCO 6276,c1(CC(=O)N(C)CC2CCN(C(=O)CC(F)(F)F)C2)cc(Cl)ccc1O 6277,N1(C(C2C(CC)C2)=O)CCN(CC(N2CCC(C3(C)N=N3)C2)=O)CC1 6278,Fc1ccc(I)cc1C(NC1(CCC(F)(F)F)CC1)NI 6279,C(=O)(C1=COCC1)NCC1(F)CC(CNC(C2(CC=C)CCC2)=O)C1 6280,CCCC(C(O)C(=O)N(OC)C(C)CC)NC(c1nccs1)=O 6281,c1(NC)cnc(C(=O)NC(C)(C)CNC(=O)C=C2CCC(C)C2)cn1 6282,Cc1ncccc1C(=O)N(C1CC(NC(c2cc(C(C)(F)F)n[nH]2)=O)C1)C 6283,c1(CC)ccc(S(=O)(=O)N2CCC(C)(C(=O)Nc3c(C)ccc(I)c3C)C2)cc1 6284,CC(CN(C)C)C(=O)NCc1occc1C(=O)NCC1(C)CCCO1 6285,C1(CNC(C)Cc2nccs2)CCN(c2ccccc2)C1 6286,C1(C(=O)NCc2cccc(NC(CNC(=O)NC)=O)c2)CCCCN(C)C1=O 6287,C1(NC(c2c(CC)nccc2)=O)CC2CC(NC(C3(CC)CCC3)=O)CC12 6288,c1(OCC(N2CC(CNC(N3CCCC(OCCO)C3)=O)C2)=O)ccc(Cl)cc1Cl 6289,c1(C(N2CCC(CC(=O)NCCc3ccco3)C2)=O)ccc(F)c(F)c1 6290,CCC(CC)(CC(=O)OC)C(=O)NC1CCCN(C(=O)CC(=O)NC2CC2)CC1 6291,c1(C(=O)NCC2CCCN2C(c2ccc(O)cn2)=O)cn2cccc(Br)c2n1 6292,c1(CCC(=O)NC(C)(CC2C(c3n(C)ncc3)C2)CO)nnc(S)nc1O 6293,CC1(NC(=O)CCc2ccc(F)cc2)CCN(C(=O)C(F)C2CC2)CC1 6294,c1(C(N2CCN(C(C3(CO)CCCO3)=O)CC2)=O)ncc(F)cc1F 6295,Cc1cc(Cl)c(C(=O)NCC2CC(NC(=O)CC3CCC4CC34)C2)cc1N 6296,C(=O)(C(C)C(=O)N1CCC(C)(C(=O)NCC2(CF)CC(F)(F)C2)C1)OC 6297,N1(C(CC(C)c2ccncc2)=O)CCC2(CC1)CC2CNC(=O)Cn1ccnn1 6298,C1(NC(C(F)=CCC)=O)(CO)CCCN(C(c2cc(C3CCCO3)n(C)n2)=O)C1 6299,N1(C(C2CC(CNC(CCc3n(C)ncn3)=O)C2)=O)CCC(CCO)CC1 6300,CC(F)(F)CCC(=O)NC1CC2(C1)CC2NC(C1(O)CN(C(=O)OC(C)(C)C)C1)=O 6301,C1(NC(CC(CC)SC)=O)C2CC3C1C3C2C(=O)NC(c1ccccc1)C 6302,C(=O)(CCS(C)(=O)=O)NCC1C(CC(=O)NCCC=C=C)C1 6303,N1(C(C(C)=C2CCCC2)=O)CCN(C(=O)C(=O)NC2CC2)CC1c1cnn(C)c1 6304,c1(-n2ncc(C(N(CC(C)NC(C=C(CC)C)=O)C)=O)c2)cccc(Br)c1 6305,C(C1=NOC2(CCC2)C1)N(C(C=C1CCN(C)C1)=O)C1CC1 6306,Cc1cccc(CN2C(=O)NC(Cc3ccsc3)C2=O)c1F 6307,C1(CC=C)(NC(c2csc(C(C)(C)C)n2)=O)CCN(C(=O)C(C2CC2)OC)CC1 6308,N1(C(C(C)C)=O)CCC2(CC1)CC2CNC(C1CCn2cncc2C1)=O 6309,C1(CC(=O)NCC(C2CC2)NC(C=C(CC)CC)=O)CCCOC1 6310,C1(OCC)(CN(C(=O)C=Cc2cn(C)cn2)C2CC2)CCSCC1 6311,N1(C(C(C(CC)(F)F)(C)C)=O)CC2CC(C1)C2N=c1cc[nH]cc1C#N 6312,Cc1cncc(C(=O)NCCC2(C)CCN(C(C3(Cl)CC3(F)F)=O)C2)n1 6313,C1(CNC(Cc2ccc(C)cc2)=O)CN(C(c2ncnc(O)c2F)=O)C(C)(C)C1 6314,C(=O)(C(F)(F)c1ncccn1)NC(CNC(c1ccoc1)=O)C1CC1 6315,C1(NC(CCCC)=O)CN(C(C2CNC(=O)O2)=O)CCC1C 6316,CC1CCN(C(C2CCCN2CC(F)(F)F)=O)C(CNC(=O)COCCCF)C1 6317,c1(C(=O)NCCCN(CCCNC(C(C=C)O)=O)C)cc(OC)cnn1 6318,C1(N(C(c2cc(CC)no2)=O)CCO)CCCN(C(c2n[nH]c(C)c2F)=O)C1 6319,C(CCN(C(=O)COC1(C)CCC1)C)(C(C)C)NC(CC1(OC)CCCC1)=O 6320,N1(C(C(CCC)C)=O)CC2CCC1C1CN(C(=O)CC3CCS(=O)(=O)C3)CC21 6321,Cc1ccc(C(N2CCC(CN(C)C(C3CC(=O)NC3(C)C)=O)C2)=O)cc1CO 6322,CCCCC(F)C(=O)NC1CCCCC1C(=O)NCc1cc(C)nn1C 6323,C1(OC)CC(F)CN(C(C2CCC(C)N2C(=O)CCn2cnccc2=O)=O)C1 6324,C1(CS(Cc2cn(C)nn2)(=O)=O)CCC(F)(F)CC1 6325,c1(NC2(CNC(C3C(C)CCCC3)=O)COC2)cc(C2CC2)nc(SC)n1 6326,C(=O)(CC(C)(C)CC(F)F)NC1C2CC(NC(Cc3c(C)n[nH]c3)=O)CC21 6327,C(C(C)(C)CC(=O)N(CC(C)(C)CNC(c1ccn(C2CCC2)n1)=O)C)N(C)C 6328,C1(CC=C)(NC(=O)CC2CCCCC2O)CCN(C(=O)C(O)CCSC)C1 6329,Cc1c(C(=O)NCC2C3CN(C(c4nccn4C)=O)CC23)ccn1C 6330,c1(C(=O)NC2CN(C(c3occ(C)c3C)=O)CC23CC3)ccc2c(c1)SCCN2 6331,N1(C(C(C)OC(C)=O)=O)CCC(C)(CC(=O)NCC(C)CC2CCC2)C1 6332,N1(CCNC(CCC)=O)CCN(NC(COCc2cccnc2OC)=O)CC1 6333,CC1(C)COc2cc(Br)ccc2C1NC(C1CCN(c2ccc(Cl)cc2)CC1)=O 6334,c1(N(C)C)ncnc(N2CCN(C(c3coc(C(F)F)n3)=O)C(C)C2)c1[N+](=O)[O-] 6335,c1(N(C(C)=O)C)ccc(N)cc1.C(CCC=O)NC1CC1(F)Cl 6336,N1(C(C(F)=CC)=O)CC(NC(=O)Cn2cnc(Br)n2)CC(O)C1 6337,C(=O)(C(C)(C)CCC#N)NC(C)CN(C)C(c1cn(-c2ncccn2)cn1)=O 6338,N1(C(CCc2ccc(SC)cc2)=O)CCCC(CO)(NC(=O)C(C)CF)C1 6339,CCCCCC(F)C(=O)NCC1CN(C(=O)COC2CCCCC2)CC12CCC2 6340,N1(C(CN(C)C2CC2)=O)CCN(C(C2CCN(C)S2(=O)=O)=O)CC1CC(F)F 6341,C1(O)(CNC(Cc2cc(C)[nH]n2)=O)CCN(C(C2CC2c2ccccc2)=O)CC1 6342,C1(N(C(C(CC(C)C)OC)=O)C)CC2CCC(C1)N2C(=O)C(C)C1CCCO1 6343,C1(C(C(N2CC(F)(CC)C2)=O)C)CCCN(C(c2cncnc2C)=O)C1 6344,c1(C(N(CCN(C(c2c(OC)n[nH]c2)=O)C(C)C)C)=O)cn2cc(C)ccc2n1 6345,c1(C(=O)NCC(C)NC(=O)CCc2ccccn2)cc(F)c(F)c(N)c1Cl 6346,N1(C(c2c(COC)noc2)=O)CC2(CCN(C(c3ccc(CN(C)C)[nH]3)=O)C2)C1 6347,N1(C(C(=O)NC(CC)C)c2cnn[nH]2)CC2(CC2)c2ccc(Cl)cc21 6348,N1(C(C2CC3C(C(=O)C(F)(F)C(F)F)C3C2)=O)CCC(F)(CC(C2CC2)OC)CC1 6349,c1(N2C3CC(CN(C(c4ccc(SCC)cc4)=O)C3)C2)nc2ccc(F)cc2o1 6350,C1(NC(=O)CN(C(=O)CCC2OCCO2)C2CCC2)CCC2CC12 6351,C1(NC(C(C2CCCCC2)OC)=O)CCNC(=O)CC1 6352,CN1CCc2cc(C(N3CCN(C(=O)C(O)C(C)(C)C)CC(C)(F)C3)=O)sc2C1 6353,c1(C(=O)N)cn(CCC2(CC=C)CN(C(C3CC(O)C3)=O)C2)c(C)cc1=O 6354,Cc1ncnc(C)c1C(=O)NC1C(C(=O)NCCc2cnn[nH]2)C1(C)C 6355,c1(CNC(c2ccc(OCCCC)nc2)=O)ccc2cccc(Br)c2n1 6356,c1(C(N(CC(CN(C(CSCCCC)=O)C)O)C)=O)oc(C2CC2)nc1C 6357,CC1CCC=C1C(=O)NC1(C(=O)NC(CCO)C2CC2)CCSC1 6358,CC1CN(C(c2nccnc2C(N)=O)=O)CC1NC(C1C2CCCCC12)=O 6359,c1(C(=O)NC(CCN(C(=O)CC(C)(C)O)C)(C)C)ccc(-c2cccs2)c(F)c1 6360,Cc1cc(CNC(=O)Nc2cc(-c3ccc(C(C)(C)C)cc3)nn2C)ccc1F 6361,Cc1cc(OCC(=O)NCC(C)N(C)Cc2ncsc2Br)no1 6362,N1(C(c2cccc(-n3cc(C4CCCCCC4)nn3)n2)=O)C2CCCC1CC(O)C2 6363,C1(C(C)NC(C(F)=C(C)C)=O)CCN(C(c2coc(CO)c2)=O)CC1 6364,C1(NC(=O)Cc2nccs2)CCN(C(C2CC3(CC3)C2)=O)C12CCCC2 6365,N1(C(C(CC)NC(C)=O)=O)CC2N(C(C3CCC(O)CN3C)=O)CCC2(C)C1 6366,CCCCC(C)CCC(=O)N(CCCCN(C(=O)CC(C)(C)O)C)C 6367,C1(NC(COC(CC)CC)=O)(CNC(=O)C(COC(C)C)N(C)C)CCOC1 6368,c1(C(N(C(C)C(C)C)CC)=O)cc(CNC(=O)C(OC)SC)no1 6369,c1(C(N2CCC(C)(CNC(C3C(C)=C3)=O)CC2)=O)ccccc1N=[N+]=[N-] 6370,N1(C(C=CCN(CC)CC)=O)CCC(F)C(NC(c2sc(COC)nc2C)=O)C1 6371,C=CC(O)(C(=O)NC1CCN(C(=O)C(n2ccnc2C)C)CC1)C(F)(F)F 6372,N1(C(C2N(C(c3c(C)csc3C)=O)C(C)C2)=O)CCC2CCCC12 6373,N1(C(C(CC)(F)F)=O)CCCC(C)(CNC(c2ccc(Br)c(OC)c2)=O)C1 6374,c1(CNC(c2n(C)nnn2)c2ncc(Br)s2)ccc2cnccc2c1 6375,N1(C(C(C2N(C(C(CCCC)=O)=O)CCC2)(C)C)=O)CCC2(CCCC2)C1 6376,C1(CC=C)(NC(c2cc(CC)on2)=O)CCN(C(C2COCCC2C)=O)CC1 6377,C(=O)(CCC(C)(C)[N+](=O)[O-])NC1CCN(C(C(C)(C)SC)=O)CC1F 6378,c1(OCC)cc(CNc2cccc(-c3cc(CC)n[nH]3)n2)cc(F)c1 6379,C12(C(=O)NC(CC)(CNC(c3cc(C#N)c[nH]3)=O)CC)CC(C)(C1)OC2C 6380,N1(C(c2cc(O)ncn2)=O)CCC2(CC1)CC(NC(=O)CN1CCCCC1)C2 6381,C(CC(C(=O)NC1(C)CC(O)C1)NC(C1CC2CCC2C1)=O)OC 6382,C(CCC(C)C)(C(=O)NC(C1CC1C(=O)OC)C)NC(c1cccc(CC)n1)=O 6383,c1(C(=O)NC(C)CCNC(c2scnc2Cl)=O)ccnc(O)c1 6384,c1(NC)ccc(C(=O)NCCN(CCCN(C)C)C(c2c[nH]nc2F)=O)nc1 6385,CS(=O)(=O)C1(C(=O)NCCN2CCC(NC(=O)CC3C=CCCC3)CC2)CCC1 6386,CCCCC(CNC(=O)Cc1cncn1C)NC(=O)CC(C)N(C)C 6387,Cc1nccnc1-c1cn(CC(=O)NC2CC(C(N)=O)C2)nn1 6388,C1(C(N(CC(=O)NCCC2(COC)CCC2)C)=O)C=C(C)CS1 6389,N1(C(CC(=O)N(C)C)=O)CCC(NC(=O)CN(C)S(=O)(=O)N(C)C)C(CO)C1 6390,N1(C(C(C)C(F)F)=O)CCC(CCN(C)C)(C(=O)N(CCC(F)(F)F)C)CC1 6391,c1(C(=O)NC2C(NC(C(C(=O)OC)(C)C)=O)CC2)c(Br)ccc(F)c1C 6392,CC1SCCCC1NC(c1ccc(CO)cc1)=O.C12(CCSC1)C(=O)N2 6393,C#CC1(F)CN(C(c2ncoc2CNC(=O)C(C(C)C)OC)=O)C1 6394,C1(CNC(=O)C2=CCCC2)CN(C(=O)C2=CSCCO2)CCCO1 6395,C(=O)(CCC(C)(C)C)N1C(C)CC(NC(C(Cc2ccc(C)cc2)N(C)C)=O)C1 6396,Cc1cnoc1C(=O)NCC(C)(O)CNC(c1[nH]cnc1C)=O 6397,C1(CCNC(c2ccc(F)cc2)c2n(CCC)nnn2)CCC(C)(C)O1 6398,c1(CN2CCC(CC(=O)N(c3ccc(Cl)cc3)CC)CC2)cccc(OC)c1Cl 6399,C1(F)(CNC(c2n(C)nnc2)=O)CCCN(C(=O)C(C)(C)CF)C1 6400,C1(NC(C=CC=CC)=O)CN(C(=O)Cc2ncc(C)[nH]2)C2CCCC12 6401,C1(NC(C(C)(C2CC2)OC)=O)CCCCC1C(=O)NCCC12CCCC1C2 6402,C(=O)(C(C)(C)CC(F)F)NC1C(NC(c2n(CC)cc(Br)c2)=O)CC1 6403,c1(CCNC(c2c(Br)cc(C)c(C)n2)=O)ccc2c(n1)OCCO2 6404,C1(C(N(C)CC2(C#N)CCC2)=O)CCCC(C(=O)NC(=O)OC(C)(C)C)CC1 6405,C1(CNC(C(Br)=C(C)C)=O)CN(C(C2CC2c2cncn2C)=O)CCCO1 6406,c1(CC(=O)NCC2N(C(C(C)n3cccc3)=O)CCC2)ccc2nc[nH]c2c1 6407,C(N(C)N1CC2(CC(C(F)F)=NO2)C1)c1ncc(C)nc1 6408,C(=O)(C(C)(C)Cc1ccc(O)cc1)NCC(CNC(c1n(CC)nnc1)=O)OC 6409,Cc1cc(CC(=O)N(C)C)sc1C(F)(F)F.N12CCC1C2=O 6410,O=C(N=c1[nH][nH]c2c1CN(C(=O)CCCCCO)C2)c1cc(F)c(F)cc1F 6411,N#CC1=C(C(=O)N2CCCC(CCNC(C34CCC(CC3O)C4)=O)C2)CCC1 6412,C(C(O)CC(=O)NC1CCCC(NC(=O)CSc2nc[nH]n2)C1)N(C)C 6413,N1(C(C2CCN(CC)C2)=O)CC2CC3CC2C1C3NC(=O)Cc1cnns1 6414,Cc1[nH]c(C#N)cc1C(=O)NCCC1CN(C(C2CCCOC2C)=O)CCCO1 6415,C(=O)(C(C)C(C)NC(c1cc(C)no1)=O)N(CC#C)C1CC1 6416,C1(C(N2CC3(C(NC(CCCOC)=O)CCC3)C2)=O)CCC2(CCCC2)CC1 6417,CC(CC(=O)NCc1ccccc1CNC(=O)C#CC1CCOC1)C(C)(C)C 6418,S(=O)(=O)(c1cc2sc(=NCc3cc4n(n3)CCCO4)[nH]c2cc1Cl)NCCC 6419,N1(C(C(CO)OC)=O)CC2CCC1CC2NC(=O)CC1CC=CCN1C 6420,C=CC1OCCCC1C(=O)NCCN(C(C1CCCCC1)=O)CC1CC1 6421,C(=O)(CS(=O)(=O)CC(=O)N(C)CCNC(C1CCCC2(CCC2)C1)=O)OC 6422,N1(CC(N2CC3CC(O)CC2C3)=O)Oc2ccccc2S1(=O)=O 6423,C1(CNC(CC(=C)I)=O)C(C)CCCN1C(=O)Cc1cnc[nH]1 6424,C1(NC(c2cc(-c3ccccc3)c[nH]2)=O)CCCN(C(=O)CC(F)(F)Cl)C1 6425,C1(C)(CCNC(C(c2ccc(O)cc2)OC)=O)COCCO1 6426,C(CCS(C)(=O)=O)(C(=O)NCCCN(C(C1CCC(C)CC1)=O)C(C)C)OC 6427,CC(CN=c1cc[nH]cc1S(=O)(=O)NCC1CCCC12CCOCC2)S(N)(=O)=O 6428,c1(C2CN(CC3C(c4n(C)nnn4)CCCC3)C2)cc(-c2ccccc2)ccc1F 6429,CC1=CCC(C(N2CC(COC)(NC(C3CCCC34CC4)=O)C2)=O)CC1 6430,N1(CC)CCC=C(c2cc(C(N3CCc4nncn4CC3)=O)cc3c[nH]nc23)C1 6431,C(CCCCC(=O)NC1CCC(C)(CNC(c2[nH]ccc2C)=O)CC1)=CC 6432,C1(CC)C(C(=O)NC2CC(NC(=O)C=CCNC(=O)OC(C)(C)C)C2)CCN1C 6433,N1(S(c2cc(NC(C)=O)c(N)cc2)(=O)=O)CCC2(C1)C(=O)NC(=O)N2C 6434,N1(C(C(C(C)O)C)=O)CCN(C2CCCN(C(c3c[nH]ccc3=O)=O)C2)C(=O)C1 6435,C(=O)(CC(C)(C)NC(C1CCC(=O)O1)=O)NC(c1ncn(C)n1)C 6436,c1(C(=O)NC(C(C)NC(c2cccc(C(C)C)n2)=O)CO)cc(Cl)c(F)cc1O 6437,c1(C(=O)NCCCNC(COCCOC)=O)csc(I)c1 6438,Cc1ccc(F)c(C(N2CC(O)(CNC(=O)C(C)C(C)C3CCCCC3)C2)=O)c1 6439,CC#CCCC(=O)NC(C)(CNC(=O)C(Cc1ccsc1)NC=O)C(C)C 6440,C(C(CC1CC1)C(=O)NCc1ccncn1)NC(C1(C)CC(=O)C1)=O 6441,N1(C(c2c(O)cc(C)nn2)=O)CC(NC(=O)CCC2CC2(Cl)Cl)CC12CCCC2 6442,c1(C(=O)NC(CCNC(C)=O)C(C)C)cc(O)nc2c(Br)cccc12 6443,C(=O)(C(O)C(F)(F)F)NC1(CCCNC(C2CN(C3CCN(C)CC3)C2)=O)CC1 6444,N1(C(c2ccc(OC)cc2I)=O)CC2OCCN(S(=O)(=O)c3cn[nH]c3)C2C1 6445,C(=O)(C(C)C(O)CC)N(CCC)CCNC(=O)CCOCCOC 6446,N1(C(c2c(C)ocn2)=O)CCC(C)C(CC(=O)N(C2CNC(=O)C23CC3)C)C1 6447,C(=O)(CC1COCc2ccccc21)NCCN(C(Cc1ccc(C)s1)=O)C1CC1 6448,C#Cc1ccc(F)c(C(=O)N(CC)CC2CCCN2C(C2CC(F)C2)=O)c1 6449,C1(NC(Cc2ccc(C)s2)=O)CC2(NC(=O)CCC3(C)CC3)COC1C2 6450,C1(C)(CNC(CC(=C=C)C)=O)CCN(C(=O)CCC2CCCC(O)C2)CC1 6451,c1(C(=O)Nc2nc(C)c(C)s2)cnc2n1CCN(C(C1(C(F)(F)F)CCC1)=O)C2 6452,c1(C(N)=O)cccc(CNC(C2CC(F)CN2C(C2CNC(=O)O2)=O)=O)c1 6453,N1(C(c2c(C)nccn2)=O)CCN(C(C2OCCCC2(C)C)=O)C2CC12 6454,C1(C(=O)NCC2(C)N(C(C(C)=C(C)C)=O)CCC2)CC2(C1)CC(C)(C)C2 6455,CN1CCOc2c(C(N3CC(CNC(C4(C)COC4)=O)CC3(C)C)=O)cccc21 6456,CC1CN(C(C23CCN(CC2)C3)=O)CCC1CNC(=O)CCc1ncc(F)cn1 6457,c1(NC(CSC(C)(C)C)=O)cc(N2CCOC(C3CCC3)C2)ncn1 6458,c1(CC(=O)NC(C#C)C)cn2cc(-c3c[nH]nc3C)ccc2n1 6459,CC1CC(C(=O)NCCC2(NC(=O)CSc3nnnn3C3CC3)CC2)CN1C 6460,N1(C(C2(CC#C)CCOCC2)=O)CCC2CN(C(=O)C(C)OCC(F)(F)F)C2C1 6461,N1(C(CCC=CC)=O)CCC(C)C(NC(c2ccc(O)c(C(N)=O)c2)=O)C1 6462,C12(C(N3CC4CC4(CNCc4snc(Cl)c4Cl)C3)=O)CCCN1CCC2 6463,c1(C(=O)NC2CCCN(c3ccccc3F)C2=O)cc2cccc(F)c2s1 6464,C1(C(=O)NC2CC(CCNC(c3c(CC)nccn3)=O)C2)CC2(CCC2OC)C1 6465,c1(C(=O)NC2CC(NC(c3cccc(C4CC4)c3)=O)C2)cnn2cccc(Cl)c12 6466,Cc1cn2c(C(N3CC(N(C(=O)CC(O)CC4CC4)C)C3)=O)c(Cl)nc2s1 6467,c1(CC)noc(CNC(c2ncnn2C)C2CC(F)(F)C2)n1 6468,C1(OC)CN(C(=NCCCSC)NCC2CCN(C(C)=O)CC2)CC1OC 6469,C(=O)(CCCCCn1cnnn1)NCCC(C)(C)NC(C1(C)CC1)=O 6470,CCCC(C(O)C(=O)NC(C)(CO)C1CCC1)NC(=O)C#CC1CCCC1 6471,C1(c2ccc(OCC)cc2)CCN(C(=O)C(F)C(C)C)CC1NC(=O)C(C)CC 6472,C1(C(N2CCCC2CCO)C(=O)NC2COC2)CC12CCC2 6473,C(CCC(C)C(=O)NCC1(NC(c2cn(CCO)nn2)=O)CCCCC1C)OC 6474,N#Cc1cc(S(=O)(=O)NC2CCCC23CCOCC3)ccc1Br 6475,C(=O)(C1=CC2CCC1C2)N1CCCC(NC(C=Cc2cccc(C)c2)=O)(CO)C1 6476,C12(C(=O)NCC(CC)NC(=O)CCN3CCCS3(=O)=O)CCCC(CO1)C2 6477,Cc1cc(N)c(C(=O)N(C2CN(C(C3CCN3C)=O)CC23CC3)C)cc1C 6478,c1(C(=O)NC(C)(C)CNC(C2CCc3n[nH]cc3C2)=O)ccc(F)c2ccoc12 6479,c1(C(N2C(Cn3cc(CNC=O)nn3)CCCC2)=O)nccc2c[nH]nc12 6480,CN(Cc1c(Oc2ccccc2)cccc1F)N1CC(COc2ccccc2)C1 6481,CC1CCCC(C)N(C(C23CC2CN(C(=O)CN2CC=CC2)C3)=O)C1 6482,C(=O)(C(O)C(C)(C)C)NC1(CNC(c2nccc(CC)c2)=O)CCCC1 6483,c1(C(C)C)nnc2cc(NC3CCN(C(=O)CC4CCCCC4)CC3C)ncn12 6484,N1(C(CN2C(C)CCC2)=O)CCOC2(CCN(C(=O)CC3CNC(=O)C3)CC2)C1 6485,N1(C(CCC2N(C(CC=C)=O)CCCC2)=O)CCOC(C(=C)C)C1 6486,CN1CC(C(N2CC(F)(CNC(c3cc(Cl)cc(Cl)c3)=O)C2)=O)OCCC1=O 6487,CON(CN1CC(=O)N(c2cccc(F)c2)C1=O)CCC(C)C 6488,Cc1cc(C#N)sc1C(=O)NCC1CC(CNC(c2nc(Cl)cs2)=O)CO1 6489,C1(NC(C(C2CC2)OC)=O)CCC(N(C(=O)C(CC#N)c2ccccc2)C)CC1 6490,C1(NC(c2scc(OC)c2)=O)CCS(=O)(=O)C12CN(C(C1(C)CC=CCO1)=O)C2 6491,C(=O)(CCC(C)SC)NCCN1CCC(NC(c2cc(CCC)on2)=O)C1 6492,C1(COc2cncc(OC)c2)CC(N=c2[nH]c3cc(C)nn3c3ccccc23)C1 6493,c1(C(c2nnnn2CC)NC2(C)CC(=C)C2)c(Cl)cc(Cl)cc1Cl 6494,C1(CC=C)CCN(C(=O)C(CNC(=O)Cn2nccc2C)OC)C1 6495,C1(F)(C(N2C(C(=O)NCC3OCC(=O)NC3)CC3CC32)=O)CCCCC1(F)F 6496,C1(CNC(C2(CC=C)CC=CC2)=O)C(C)CCN1C(c1nn(C)nc1Br)=O 6497,Cc1oc(C#N)cc1C(=O)NC(CC1CCC1)C(N1CCCC(C)(F)C1)=O 6498,c1(OC)ccnc(C(N2CCC(N(C)C(c3cc(Cl)cs3)=O)C(C)C2)=O)c1N 6499,c1(C(N2CCC(C(C)NC(c3c(CC)[nH]cc3)=O)C2)=O)cscc1S(C)(=O)=O 6500,C(CNC(=O)CN1CCCCC1=O)(C(C)C(C)C)NC(c1c(C)csc1)=O 6501,c1(CC(=O)NCCOCCCNC(CC(CCC)C)=O)ccc2c(c1)CCOC2 6502,C1(C(=O)NC2(CNC(=O)Cc3ncn4c3CCC4)CC2)CCc2ncccc2C1 6503,N1(C(c2c(=N)cc[nH]c2)=O)CC(F)(F)CC1CNC(c1ncc(Cl)cc1Cl)=O 6504,c1(OC)c(NC(=O)Nc2cc(OC)nn2-c2ncccn2)cc(Cl)cc1Br 6505,C=CCC(C)(C)C(=O)NCC(C)(C1CC1)NC(c1nccnc1N)=O 6506,N1(C(c2cc(C)sc2C)=O)CC2CCC1(CNC(c1n[nH]cc1C)=O)CC2 6507,N1(C(c2cc(C)nn2C)=O)CCOC2CN(C(c3conc3C(C)(C)C)=O)CC12 6508,c1(CN(C)CC2CN(C(=O)COc3cccnc3)C2)ccnc2ccncc12 6509,c1(C(=O)NCC(CNC(C(CC)c2cccnc2)=O)(C)C)cn(C)nc1COC 6510,c1(SCC(=O)NCC2CCC2CNC(=O)Cc2ccns2)nc2ccccc2[nH]1 6511,CCC(C)C(CC(=O)NCC(C)(F)C(C)(C)F)NC(c1cccc2ccnn12)=O 6512,c1(CNC(C2CCN(Cc3ncccc3F)C2)=O)ccccc1[N+](=O)[O-] 6513,N1(C(Cc2cc(C)ns2)=O)CC2CCCN(C(c3cccc4c3CCC4)=O)C2C1 6514,Cc1noc(C)c1C(=O)NCC(F)CNC(C1(C)CC(C)(C)C1)=O 6515,c1(C(=O)NCC2CC(C)N(C(=O)C(C)S(C)(=O)=O)CC2)ccc2cccnn12 6516,C(C)(C)(C(=O)N(C1CC(NC(c2coc(SC)c2)=O)C1)C)OC 6517,N1(C(C(C)C)C(=O)NCC2CCCO2)CCCCCC(N)C1 6518,c1(C(=O)NCC2(NC(C3CCC(N(C)C)CC3)=O)CC2)ccc(N)c(O)c1 6519,c12nnc(cc1C(F)(F)F)SC2.c1(CC)cccnc1CC 6520,c1(C(=O)NCC2N(C(C(C=CCCC)O)=O)CCC2)cccc2ccc(O)nc12 6521,c1(CNC(=O)CC2CCCN(C(=O)CC3CCC3)CC2)ccc2cc[nH]c2c1 6522,c1(C(C)C)sc2c(c1F)CCCC2.C#Cc1cc2nn1CC(=O)N1C2COCC1 6523,C(C(C)C(=O)Nn1cccn1)N(C(C1C(C)=CCS1)=O)C 6524,C(=O)(C=C1SCC(=O)N1C)N1C(CN(C(C(CN(C)C)O)=O)C)COCC1 6525,N1(C(Cn2ncc(C#C)c2)=O)CC(C)CN(C(=O)CCCCC=C)C(C)C1 6526,CCCC(CCC)=CC(=O)NC1CC(NC(=O)CCCn2cccn2)C(O)C1 6527,C1(C#N)(C(=O)OC2CC2)CN(C(=O)Nc2ccc(COC)cc2)C1 6528,c1(C(=O)NC(CC)CNC(=O)CC(C)CC)cc2c(OC)cc(OC)nc2[nH]1 6529,N1(C(CC(=O)NCC)=O)CCC2(CCCC2NC(=O)Cc2nccs2)CC1 6530,c1(C(N2CC(F)(CNC(=O)CN3CC4CC4C3)C2)=O)coc2ccc(O)cc12 6531,c1(OC(C)C)ccc(C(=O)NC2CC23CC(NC(c2c[nH]cc2CN)=O)C3)nc1 6532,C1(CNC(C(C)NC(c2ccoc2)=O)=O)C2CC1N(C(=O)CCC1OCCO1)C2 6533,C1(C(N(CC(C)(C)CNC(=O)Cn2ncnn2)C)=O)CC12CCS(=O)(=O)CC2 6534,CC1CC(C(=O)NC2(c3ccccc3)CN(C(C3CCC(=O)N3)=O)C2)CC(=O)N1 6535,c1(CC)cc(=NCC2CCCC(NC(C3CCN3C3CCCC3)=O)C2)[nH]cn1 6536,C12(CNC(CCCCC)=O)CCCC1N(C(=O)C(F)=C(C)C)CCC2 6537,C(C(=O)NC1CN(C(c2cc(O)nn2C)=O)CC1C(F)(F)F)(C(C)C)SCC 6538,N1(C(c2ccc(C(C)=O)cc2)=O)CCC(NC(c2n[nH]c(C3CC3)n2)=O)CC1C 6539,C12(NS(=O)(=O)CC3CCCCC34CCC4)CC(C3CCCC3)(C1)C2 6540,N1(C(c2ccc(F)cc2Br)C(=O)NCCOC)CCOC2(CCSC2)CC1 6541,c1(C(=O)NCC2(CNC(C(CSC)OC)=O)CC2(F)F)ncccc1O 6542,Cc1cc(C(C)(C)C)ccc1C(=O)NCCN(C(=O)CCn1ccnn1)C1CC1 6543,c1(C(=O)NC(CC)CO)ccc(=NCc2cc(F)ccc2Br)[nH]c1 6544,Cc1ccc(OCC(=O)NC2CC(F)CN(C(c3c[nH]nc3F)=O)C2)c(F)c1 6545,N1(Cc2cn(CCOC)nc2)CC2(CCC(CNC(=O)COC3CCCC3)O2)C1 6546,Cc1cnc(C(=O)NC(C)CCN(C)C(C2CC2F)=O)c(Br)c1 6547,Cc1ccc(C)c(C(N2CCC(O)C2C(N2CCCC(O)(C(N)=O)C2)=O)=O)c1 6548,C1(O)(C(C)NC(=O)CNC(N)=O)CCCN(C(C2(n3nccn3)CC2)=O)C1 6549,N1(CCN(C(C2(OC)CCCC2)=O)C)CCN(C(=O)CCS(C)=O)CC1 6550,c1(C(=O)NC(C(C)NC(c2c(C)oc(C)c2C)=O)C)ccc2c(c1)COC2 6551,C1(CCC)CN(C(=O)Cc2nocc2C)CCN1C(c1cc(C)n(C(F)F)n1)=O 6552,c1(OC(=O)NCCc2cc(C(N(C(C)C)C)=O)no2)ncc(Cl)cc1Cl 6553,c1(N(C2(C#N)CCNC2)Cc2c(C)noc2C)ncnc2cnn(C)c12 6554,O=C(C1=NOC2(CCOC2)C1)NCc1ncoc1C1CCN(C(c2cocn2)=O)C1 6555,C1(C(N2CC(C3(NC(c4c[nH]nc4C(F)F)=O)CC3)C2)=O)CCC2CCC(=O)N12 6556,C1(O)(CNC(c2cc(I)c(Cl)cn2)=O)COCCC1O 6557,C12(CNC(C(C)N(C(=O)C(C)O)CCC)=O)CC(CO)(CO1)C2 6558,c1(C(=O)NC2CC(O)(CNC(C(C)(C)CO)=O)C2)cccc2c1OCC2 6559,N1(C(C2(CC=C)CCCC2)=O)CCCC(C(C)NC(=O)C(N)=O)C1 6560,Cc1csc(CCCC(=O)NC(C2CCN(C(c3cn(C4CC4)nn3)=O)C2)C)n1 6561,N1(C(Cc2cc(C)on2)=O)CC(C(=O)N(C)Cc2nccn2C)OC(C)C1 6562,C1(CNC(c2c(C)cn(C)c2)=O)CC2(CC2)CN1C(c1cc(F)n(C)n1)=O 6563,N1(C(C(=O)Cc2ccccc2)=O)CCC2(C1)CN(C(C1CC(O)C1)=O)C2 6564,C12(C(N3CCC(C)(CNC(Cc4nnc(C)s4)=O)CC3)=O)CCC(CC1)C(C)O2 6565,N1(C(C(C)CSC(F)(F)F)=O)CCC(NC(c2cc(C3CC3)[nH]n2)=O)C(F)C1 6566,c1(OC)ncc(C(N2CCC(CNC(c3cc(=O)n(C)o3)=O)C23CC3)=O)cc1Cl 6567,C1(CNC(C=CCN(CC)CC)=O)CN(C(C2(CCOC)CCCC2)=O)CC1C 6568,CC1(C(N2CCCCC(NC(c3snnc3C3CC3)=O)C2)=O)COC(=O)OC1 6569,N1(C(c2ccnc(C)n2)=O)CCN(C(c2cc(C3(C)CC3)on2)=O)C(C2CC2)C1 6570,c1(C(N(C2CN(C(=O)CC=CC(C)(C)C)C2)C)=O)ccc2c(c1)OC(F)(F)O2 6571,N1(C(C(C(C)(C)O)(F)F)=O)CCC2(COC(CNC(=O)C=CI)C2)C1 6572,CCCCC(F)C(=O)NCC1CC1CC(=O)NC(C)C(=O)N1CCCC1 6573,C1(c2n(C(CC)C)nnn2)(Nc2cc(C)n(C(=O)NCCO)c2C)CCCSCC1 6574,Cc1ccc(C(N2CC3(CC3C(N3CCC4(CCC4)C3)=O)C2)=O)nc1C 6575,c1(-c2cn(C(C)C(=O)NCc3cc(F)c(F)c(F)c3)nn2)ccc(S(N)(=O)=O)cc1 6576,C1(NC(c2c(C(C)NC(C(C)NC(CC)=O)=O)noc2)=O)CCS(=O)CC1 6577,CC1(NC(=O)CCC2CC2(Cl)Cl)CN(C(c2cnoc2C2CCOCC2)=O)C1 6578,C(CC(C)(C)C)(C(=O)N1CCCCC1CCC(C)(C)NC(c1cocn1)=O)OC 6579,C(=O)(CC(O)CC(C)(C)C)NC1(COC)CCN(C(=O)CN(C)S(N)(=O)=O)CC1 6580,c1(SC)cccc(C(=O)NCCCOCCCNC(C2(N(C)C)CCC2)=O)c1 6581,CCCC(C)(C)CC(=O)N1CC2OCC(NC(=O)C(C)(C)CN3CCOCC3)C2C1 6582,c1(C(N2C(C)(C(N(CC(C)(C)O)C)=O)C=CC2)=O)n[nH]c2c1CCC2 6583,CCC(C(=O)NCC(CNC(c1ccc(CN(C)C)s1)=O)OC)C(F)(F)F 6584,Cc1cc(C(=O)NCC2CC(NC(C3CC(C)(C)O3)=O)C(O)C2)ccc1F 6585,CCCCCC(CC)C(=O)NC1CN(C(c2ccc(N)c(SC)c2)=O)CCC1C 6586,c1(OC)ccc(C(=O)NCC2(F)CN(C(=O)C(F)C3CCOC3)C2)c(F)c1 6587,c1(C(N(C)CC2CCCN2C(=O)CCC2(C)CC2(F)F)=O)cc2cccn2cn1 6588,C(C)(C(C)(C)C)=CC(=O)NCC(c1ccccc1)NC(C(c1cccs1)SC)=O 6589,C1(C)(CNC(c2cnc(OCC)s2)=O)CCC(NC(=O)C(CC)SC)CC1 6590,CC1(C)OC(C)(C)C1C(=O)NCC1CN(C(C2CCS(=O)(=O)N2)=O)CC1O 6591,c1(-n2cc(C3(O)CN(C(=O)Sc4ccc(C(=O)O)cc4)C3)nn2)ncc(Br)cn1 6592,N1(C(=O)Cn2nccn2)CC2CCCC(Nc3ncncc3Br)C2C1 6593,C#CCCCCCCCC(=O)NC12CCC(CC1n1cc(-c3cnsc3)nn1)C2 6594,c1(CC(=O)NCC2CN(C(=O)CCn3ccnc3)C2)nc(F)c(F)cc1F 6595,N1(C(c2cncc(NC(c3cc(C)cc(C)c3)=O)c2)=O)CCC(C)(CO)C(O)C1 6596,C#CCCC(C(=O)NC(C)CCC(=C)C)NC(c1nnn(C)c1N)=O 6597,CC(CCC(C)(C)C)C(=O)NC1CCCN(C(=O)CS(=O)(=O)C2CC2)C1C 6598,c12ccc(F)cc1Cn1cc(nn1)CC1CCN1C2=O.S(C)(=O)(=O)N(C)C 6599,N1(C(=O)NC2CCS2(=O)=O)CCC(NCC(N2CC(OCCO)C2)=O)C1 6600,Cc1n[nH]cc1CCC(=O)NCC1(CNC(C2(C3CC3)CC2)=O)CCCC1 6601,c1(CNC(c2n(CCC)ncn2)c2nnnn2CC)ccnc(C(C)C)c1 6602,CCCC(C)(C)C(=O)N1C2CCC(C2)C1CC(=O)N(C)CCOC(F)F 6603,N1(C(C(CC(=C)C)OC)=O)CC2(CC(NC(c3ccn(C)n3)=O)CO2)C1 6604,CC1CN(C(C2C=CC=CC=C2)=O)CCCN1C(c1cc(O)nc(Cl)c1)=O 6605,C1(C(C(=O)NC2CC(F)(F)C2)N(C(C2CCN(C)CC2)C)C)CCCOCC1 6606,N1(C(c2cncc(OC)n2)=O)CC(O)C(O)C1CNC(=O)CSCc1cscn1 6607,c1(C(c2n(CCCSCC)nnn2)NCCCS(C)=O)ccnc(N(C)C)c1 6608,C(=O)(CCCCC(C)(C)C)N1CCC(NC(C(CCCCC)O)=O)C12CC2 6609,C1(NC(C2N(CCC)CCC2)=O)CN(C(c2ncn(C)c2C)=O)CC1OC 6610,N1(C(CC2CC(OC)C2)=O)CCCN(C(C2C(C#N)C2(C)C)=O)C(C)C1 6611,Cc1nn(CC(F)F)cc1C(N1CCC(O)(CNC(C2COC(=O)N2C)=O)C1)=O 6612,c1(C(=O)NCCN(C(C(CC)O)=O)CC2CC2)ccc(-n2cnnc2)cc1 6613,c1(NC(=O)NCCc2c(C)occ2C(F)(F)F)cccc(F)c1I 6614,C1(C(N(CCNC(=O)C=CCOC)CC)=O)CCn2c(cnc2Br)C1 6615,c12cc(no1)NC(=O)C(C)(C)C1CCCN1CC2.C(CCS(C)=O)N(C)C(N)=O 6616,c1(NC(C=CC)=O)cc(CC)cc(Cc2ccc(OC)c(C(C)=O)c2)c1OC 6617,c1(CC(=O)NCCC2CN(C(=O)C(F)n3cccn3)C2)cc(-c2ccco2)on1 6618,N1(C(C(C)N(C(C)=O)C)=O)CC(CNC(c2cn(C3COC3)nn2)=O)C(C)(C)C1 6619,N1(C(CN(CCC)C)=O)CC(C2CN(C(c3sc(COC)nc3C)=O)C2)C1 6620,C(C(N=c1cc(NCc2nc(Br)cs2)nc(C(F)(F)F)[nH]1)c1ccco1)N(C)C 6621,c1(COC)cc(C(C(=O)N(C(C)C)C2CC2)N(C2COCC2O)C)ccc1Br 6622,C1(C(=O)NCC2CC(NC(=O)CCc3ccsc3)C2)CC2(F)CC1C2 6623,c1(C(=O)NC2(C3N(C(c4ccc(CSC)o4)=O)CCC3)CC2)ccnnc1S 6624,N1(C(C2OCCOC2C2(C(=C)F)CCC2)=O)CC2(CC2)CC1CNC(=O)CC 6625,C12(C(=O)NCC3(NC(C4CC45CCCC5)=O)CCC3)CC(CO)(C1)OC21COC1 6626,C1(NC(C2(C)COC2)=O)CCN(C(C23CCC(C2)OC3)=O)CC1F 6627,Cc1ccc(C(=O)NC2CC(NC(c3cc(N)c(F)cn3)=O)C2)cc1S(N)(=O)=O 6628,C1(CC=C)(C(=O)NCC2NC(=O)NC2=O)CCCN1C(c1snnc1C)=O 6629,Cc1nc(-c2cnn(C)c2)oc1C(=O)N(C)CC1(NC(=O)CC2C=CCC2)CC1 6630,N1(C(CNC(CC#N)=O)=O)CCN(C(=O)C(F)(F)F)CC1c1ccccc1Cl 6631,c1(N2CC(C)(CC(C)C)OCC2)nc2cccnc2c(=NCCCSC(F)F)[nH]1 6632,N1(C(C2N(C(CC3(CC)CCC3)=O)CCSC2)=O)CCc2oc(C)nc2C1 6633,c1(C(=O)NCC2CN(C(CCc3c(C)ncs3)=O)C2)cc(F)cc2ccncc12 6634,Cc1nc(C(C)C)nc(O)c1C(N1CC2CC1(CNC(C1(C)CCCO1)=O)C2)=O 6635,CCC(C)C(O)C(C)C(=O)NC1C2CN(C(c3cccc(F)c3F)=O)CC12 6636,C#CCC(CC(=O)NCC(C)(C1CC1)OC)NC(c1c[nH]c(=NC)s1)=O 6637,C1(C(=O)OC)C2CC(CN(C(=O)C(=O)C(C)C)C2)N1C(=O)C(N)CN.C1CN1 6638,C(CCCCCCCCO)n1cc(C(=O)NCC2(CCO)CC2)nn1 6639,n1(CC(N2CC(N(C(=O)C=Cc3ccoc3)C)C(F)C2)=O)ccc2ccccc12 6640,C1(CC(=O)NC2CC3(CC(NC(C(C(CC)C)O)=O)C3)C2)CS(=O)(=O)CCN1C 6641,c1(CC)cc(F)c(C(N2CCN(C(=O)CC=C(C)C)C(CF)C2)=O)cc1F 6642,CC1(C)CCN(C(c2cc(F)ccc2F)C(=O)NCc2ccco2)CCS1=O 6643,CCCCC(CCCC)C(=O)N1CCCC2(C1)CN(C(=O)C(F)CN(CC)CC)C2 6644,Cc1oc2ccccc2c1CC(=O)NC1CC1CNC(C1(C)CC1(F)F)=O 6645,C=CCC(CC(F)F)NC(C12CC1CN(C(c1ccn(C)c1)=O)C2)=O 6646,CCC(C)CC(=O)C(=O)NCC(CNC(C1CCCN1C(C)C)=O)OC 6647,C(=O)(CCCCCSC)NC(CN(C(c1cnn(C2CC2)c1)=O)CC)C 6648,c1(C(=O)NC(C)CNC(=O)C(C)(C)C2CCOC2)cc2c(cn1)OCCO2 6649,CCCC(C(=O)NCC1CCN(C(=O)C=C(C)c2ccco2)CC1C)C(C)C 6650,S(=O)(=O)(CC(=O)N(C1CCC(NC(=O)C(C)OCC2CC2)CC1)C)NC 6651,N1(C(C(C)OCC#C)=O)CCCC1CNC(=O)C(C)n1cccn1 6652,C1(CC(=O)NC(CNC(CCOCC)=O)CO)CCC2(CC1)CCC2O 6653,N1(C(C2CN(CC)C(=O)C2)=O)CCC=C(C(=O)Nc2c(O)cccc2Cl)C1 6654,CN1CCc2[nH]nc(C(=O)NCC3CN(C(C4CC5CC4CC5(F)F)=O)C3)c2C1 6655,CCC(C)CCCC(=O)NCCN(C(=O)C(C)(O)C1CC1)C 6656,C1(N(C)C(c2cnc(Cl)s2)=O)CC2CCC1N(C(c1ccc(Br)cc1)=O)C2 6657,c1(OC)ccc(C(=O)NC(C)C(C)NC(C2NC(=O)OC2C)=O)c(Br)c1 6658,Cc1ccn(CCC(=O)NCC2CCN2C(=O)CCCNC(N)=O)n1 6659,Cc1ccc(C)c(C(N2CCC23CN(C(=O)COc2ccccc2O)C3)=O)c1 6660,c1(C(N(CCCNC(=O)C=Cc2cc[nH]n2)CCC)=O)cc(CCCC)oc1C 6661,c1(NC(C2CCN(C(C3CCC(F)(F)C3)=O)CC2O)=O)cc(O)ccc1Cl 6662,c1(C(N2CC3CC(NC(CC=C)=O)CC3C2)=O)ccc2cnc(C)n2c1 6663,c12ccc(Br)cc1NC(=O)CO2.c1(C(C)C)ccc(NC2CC2)cc1 6664,C1(C(=O)NCc2cnc(C3CCC3)[nH]2)CC2(CNC2)CO1 6665,C(CCCC(=O)N1CC2C=CC2C1)N(C(C(c1ccnn1C)C)=O)C 6666,N1(C(c2c(F)cc(NC(=O)OC(C)(C)C)cc2F)=O)CCCC2(CCCCO2)C1 6667,Cn1ncc2cc(C(=O)NCCC3(NC(=O)CCc4ccccc4)CC3)cnc12 6668,C1(C(N(C(CC(=O)NCCOCC(=O)OC)C)C)=O)CCCC(C)(C)C1 6669,N1(C(Cc2c(C)n[nH]c2C)=O)CC2(CCN(C(c3ccc(CN(C)C)s3)=O)C2)C1 6670,CC(CC(=O)NC1CC2(C1)CC(CNC(=O)CCC(=O)C1CC1)C2)CC(C)(C)C 6671,c1(CC(N2CC(F)(CNC(C=C(C)C(C)(C)C)=O)C2)=O)c(C)nc(O)nc1C 6672,C(=O)(C#Cc1ccccc1Cl)NC(C(=O)OC)Cc1ccc(OC(F)(F)F)cc1 6673,C(CC(O)CNC(c1csc(C2CCCO2)n1)=O)NC(C1(C)CSC1)=O 6674,N1(C(C2CCCSC2)=O)CCC2COC(C(N3CCC(CO)C(O)C3)=O)C2C1 6675,C1(NC(CC(CC)(C)C)=O)CN(C(c2c[nH]ccc2=N)=O)CC1S(C)(=O)=O 6676,c1(C2CN(C(=O)NC3CCC3F)C2)ccc(F)cn1 6677,CC1(C)CC(CNC(=O)CC2(C)OCCO2)N(C(=O)CCC2OCCO2)C1 6678,CC1CC=C(C(=O)N2CC(CCNC(=O)C(C)(C)c3ccn(C)n3)C2)CC1 6679,c1(CC)[nH]c(=N)sc1C(N1CCC(Nc2cccnc2)CC1)=O 6680,CCCC(CCCO)C(=O)NC1CC2CN(C(c3cnc(C)nc3O)=O)CC2C1 6681,C1(NC(CCC=C(C)C)=O)CN(C(C2(F)CCCCC2)=O)CC2(CCOCC2)C1 6682,c1(N(C(C23CC(C(=O)NCC)(C2)C3)=O)C)ccc2cnccc2c1 6683,C(=O)(C(F)(F)CN(C)C)NCC(c1cccc(C)c1)NC(C1C(C=C)C1)=O 6684,c1(C(COC)(C)O)cn(CCCN(C(=O)C(CN(C)C)N(C)C)C)nn1 6685,CN1CCC(CC(=O)NC(Cc2ccccc2Br)C(=O)NC2CCC3CC23)CC1 6686,N1(C(CN(C(=O)OCC)C)=O)CCN(C(=O)C(C2CC2)SC)CC1COC 6687,C1=CC(=O)N2CCC1CC2.O(C=CC(=O)OC)CC 6688,Cc1cc(C)nc(S)n1.C1(F)(CNC(=O)CC2(CC3CCC3)CC2)CC(C(=O)N)C1 6689,CCC(COC)C(=O)NCCCN(C(C1(c2cccs2)CC1)=O)CC 6690,c1(C(=O)OC)cccc(-c2ncc(C(=O)NCCc3cc(Br)c(Br)s3)s2)c1 6691,c1(C(N(CC(C)N(C)C(C2CCC(C)(C)O2)=O)C)=O)cc2cnccc2o1 6692,C1(C)(C(=O)NC(C)CN(C)C(c2sccc2C2CC2)=O)CC2CC2C1 6693,C1(C(N2C(C(=O)NCCCC#C)CCC2)=O)CCC2(CCC2)O1 6694,N1(C(=O)NCC)CCC(C(=O)NCCCCCN(C(=O)Cc2cncs2)C)CC1 6695,Cc1cc(C(=O)NCCCCNC(=O)C(C(C)C)N(C)C)cc(C)c1N 6696,N1(C(CSCCC)=O)CCN(C(=O)CC2OCCOC2(C)C)C(C(F)F)C1 6697,c1(C(N2CCN(C(C=CCC)=O)C(c3ccccc3)C2)=O)cc(C)c(F)cc1N 6698,C1(NC(=O)CCc2ccnc(Cl)c2)COC2(C1)CN(C(c1cn(CCO)nn1)=O)C2 6699,c1(C(N(CCNC(C2CC2(Cl)Cl)=O)CC2CC2)=O)cc(Cl)ccn1 6700,c1(N2CCN(C(COC(=O)C(C3CCCCC3)F)=O)CC2)cccc([N+](=O)[O-])c1 6701,Cc1c(C(N2CCC3(CCC3NC(C3C=CCC3)=O)CC2)=O)nn2c1CCCC2 6702,C(=O)(C1COc2ccccc21)N1C(C)CCN(C(Cc2c(C)scc2)=O)CC1 6703,C(C(C(=O)N1CCC1CC(=O)NCCCCCO)OC)OC 6704,c1(C(N2CCC(COC(F)F)C2)=O)ccnn1C(F)(F)F 6705,C12(CNC(c3cc(C)no3)=O)CN(C(C3CCS(=O)CC3)=O)CC1CCO2 6706,c1(C(=O)NC(C)C(C)C(=O)NCCCC(O)CO)nccc2[nH]ccc12 6707,N1(C(C=C(C)I)=O)CC=CCC1C(F)(F)F 6708,C(=O)(CCC(C(=O)Nc1cccc(Cl)c1C)N1CCSCC(C)C1)OCC 6709,N1(C(C(c2ccc(CC)s2)=O)=O)CCC2C(CCCN2C(c2cccnn2)=O)C1 6710,N1(C(C(CC2CCC2)NC(c2c[nH]nc2Cl)=O)=O)CC2CCCC2C1 6711,CN1CC(NC(=O)CC2CCN(C(C3CS(=O)(=O)C3(C)C)=O)C2)C(C)(C)C1 6712,N1(C(CC(C(C)C)O)=O)CCC(O)(C2(NC(=O)CC3CCC(=O)NC3)CC2)CC1 6713,c1(NC(CC=C)=O)ccc(=NCc2cccc(OC(F)(F)F)c2O)[nH]c1 6714,c1(CC)c(C(=O)NCCCNC(C2COC(C)C2)=O)cccc1F 6715,C(CCCC(=O)NCC(C)C(=O)NC(c1cncs1)C)OCC 6716,C1(C(C)NCC(c2ccsc2)C)CCN(c2cc(NS(C)(=O)=O)ncn2)CC1 6717,C1(NC(c2c(CC)cccc2)=O)(CNC(=O)CCP(C)(C)=O)CCCCC1C 6718,N1(C(C(c2ccc(F)cc2F)OCC)=O)CCCCC(C2CN(C(=O)CO)C2)C1 6719,C(CN=c1[nH]nc(O)s1)NC(c1ccc(C(C)(C)C)cc1)=O 6720,c1(CN2CCC(CC(=O)OC)C2(C)C)ccc2cc(F)cc(Br)c2n1 6721,c1(CCC(=O)NC(CNC(C2C(C#C)C2)=O)(C)C2CC2)ccc(C)c(C)c1 6722,CCCCC(O)CC(=O)NC1CCN(C(c2cnc(C3CCOCC3)s2)=O)CC1 6723,C12(C(=O)NCCC(C)(C)NC(=O)CC3CCS(=O)(=O)C3)CCCN1S(=O)(=O)CC2 6724,C1(C(N(C2CCN(C(=O)Cc3cc(C)no3)C2)CC#C)=O)CC(C)(F)C1 6725,C12CCCC(CC1)NC2=O.C(=O)(C(O)C(F)(F)F)NC1CCCC1.O=C1CN1 6726,C1(NC(C2Cc3n(cc(C)n3)C2)=O)CCC2CCN(C(=O)Cc3cscn3)C1C2 6727,C(C(=O)O)(C(F)(F)F)N(C)CC(C1C(C)(C)C1(C)C)SC1CCOC1 6728,N1(C(C2(CC)CCC2)=O)Cc2ccccc2C(NC(C2(N(C)C)CCSC2)=O)C1 6729,C1(CC(=O)NCC(CC)NC(=O)COCc2ccnn2C)CCCCC1(C)C 6730,C=C1Cn2c(C(N3CCCC(CCNC(=O)C(C)CC(C)C)C3)=O)nnc2S1 6731,N1(C(c2c(CC)ccs2)=O)C2CCC1(CNC(=O)C=CS(C)=O)CC2 6732,c1(C(N(C)CC2COCCN2C(=O)CC2CCCOC2)=O)nnc(O)cc1O 6733,N1(C(c2c(N)nccn2)=O)CC2COCC2(C(=O)NC2CCOC2C2CC2)C1 6734,C(=O)(C1CCc2cccc(O)c21)N1CC2CCCC(NC(CC(C)(C)O)=O)(C1)C2 6735,Cc1cn2cc(C(N3CCC(NC(=O)CN(CC(C)(C)C)C)CC3C)=O)nc2s1 6736,N1(C(Cc2c(C)cc(C)s2)=O)CCCCC(NC(=O)CCCF)C1 6737,C(C(=O)NC(c1ccc(Br)cc1)C(F)F)(C(C)(C)C)NC(C)=O 6738,N1(C(=O)COc2ccsn2)CCN(C(c2csnn2)=O)C2CS(=O)(=O)CC12 6739,c1(CNc2nnc(C)n2C)[nH]c(=NCC2(OC(C)C)CCOC2)nc2scnc12 6740,N1(C(CC(OCC)OCC)=O)CC(C)(C)CC1NC(=O)Cc1cc(O)nnc1O 6741,N1(C(C2(C=C)CCC2)=O)CC2CCC1C(CNC(c1ccnc(C)n1)=O)C2 6742,c1(OCC(N2C(CNC(c3c[nH]ccc3=O)=O)C=CC2)=O)cccc(Cl)c1 6743,n1(CC(C)C)ccc(=NC(=O)C(=O)NCCCc2ccnc3cc(Cl)ccc23)[nH]1 6744,C(=O)(C1=NNC(=O)CC1)N1CC(NC(c2cnn(C)n2)=O)(CO)C1 6745,c1(C(C)C)cc(C(=O)NC(C)(CNC(=O)C(F)CC2CC2)Cn2cccn2)on1 6746,c1(CCCNC(CC2CC(NC(C(C)OC)=O)C2)=O)nnnn1C 6747,c1(NC(N(C)Cc2cc(C)nn2C)=O)cc2c(cc1[N+](=O)[O-])N(C)CCO2 6748,Cc1[nH]nc2ccc(C(=O)NCC(C)CNC(=O)COCC3CCCO3)c(Cl)c12 6749,C1(C(=O)NC2CCCN(C(c3cnn(C4CC4)c3)=O)C2)Cc2nncn2C1 6750,N1(C(c2coc(Cl)n2)=O)CCCC(N=c2c(Cl)c[nH]cc2[N+](=O)[O-])C1 6751,C(=O)(C(C)(F)C(C)(C)F)NC1C(C(=O)NC(C23CCC(CO2)C3)C)CC1 6752,CC(C)CC(C(=O)N1CC(F)(C(=O)NC2CC(C)(C)OC2(C)C)C1)C(N)=O 6753,Cc1sc(NC(C2CCOC2c2ccnn2C)=O)nc1C(=O)O 6754,Cc1ccc(F)c(N(C)C(N2CCC(N3CCCCCC3)CC2)=O)c1F 6755,CC(C)C(CNC(C1COCC(C)O1)=O)C(=O)Nc1c[nH]ccc1=O 6756,CN1CCN(C(c2ccc(C(N)=O)o2)=O)CC1CNC(C12CCC(C)(C1)OC2)=O 6757,C(CCC(=O)NC1CCCC1C(=O)OC)N(c1cn(C(=O)OC)cn1)CC#C 6758,C1(CC(C)Nc2nc(C(C)(F)F)cs2)CCCCN1 6759,C(C(=O)N1CCC(C(=O)Nc2cncnc2N(C)C)C1)(C(C)C)NC(C)=O 6760,c1(N(c2ccnc(OC)n2)C(c2ccccn2)=O)ccc2c(c1)CCNC2 6761,Cc1ccc(C(C)C)c(C(=O)NCC2CC(NC(C3(C)CC4CC4C3)=O)C2)c1 6762,CC(CCC(C)(C)C)C(=O)N1CC2CC1C2NC(=O)CNC(=O)CC(F)(F)F 6763,C12(C(N3CCCC(CN(C)C(c4ccn(C)n4)=O)C3)=O)CC(C3COC3)(C1)C2 6764,C1(C(N2CCC(O)(CN(C)C(c3cc(Cl)c[nH]3)=O)C2)=O)(OC)CCS(=O)(=O)C1 6765,C1(N(C(CCC(C)NC(=O)CC2(N(C)C)CC2)=O)C)CCOC(C)(C)C1 6766,c1(CCC(=O)NCC2(NC(C3CCN(C)C3)=O)CCCC2)ccc(N(C)C)cc1 6767,C1(C(N(CCNC(c2c(C)oc(Br)c2)=O)C(C)C)=O)Cc2ccccc2CO1 6768,C1(CNC(C(C)=C2CC2)=O)CC(NC(c2cnn(CCC(F)(F)F)c2)=O)CC1O 6769,N1(C(c2c(CC)c[nH]c2)=O)CCC2(CCCN2C(C2CCCS2)=O)C1 6770,c1(N(C)C)ccc(F)c(C(=O)NCCC2CCC(NC(C3C4COCC34)=O)C2)c1 6771,c1(NCC(C)N(C(C(=O)NCC(C)N(C(C)=O)C)=O)C)ccccc1 6772,CCC(C)C(C(=O)N1CCCCC1C(=O)NC1(CF)CC1)N(C)C 6773,C(=O)(C1=CC2C=CC(C1)C2)NC1CC2(C(NC(c3n(C)cc(Br)c3)=O)C2)C1 6774,C(CC(=O)NC(CCO)C(F)F)(C(F)(F)F)NC(CN(C(=O)OCC)C)=O 6775,C=CCCCCC(O)CNC(c1ncsc1CC)=O 6776,Cc1ccc(OCC(=O)NCC2CN(C(C3CCCN3N=O)=O)CC2O)cc1C 6777,c1(C(N2CCC(O)(C(C)NC(C(CSC)O)=O)CC2)=O)cc(F)c(C)cc1F 6778,c1(C(=O)NC2(CC)CCN(C(=O)C(C)CC(=O)OC)CC2)ccc(S(C)(=O)=O)o1 6779,C=CC(O)C(=O)N1CCC1CNC(c1cc(C2(C)CC2)n[nH]1)=O 6780,c1(C(=O)NC(CSC)CO)ccc(S(=O)(=O)Nc2nc(C)cs2)cc1 6781,N1(C(COC(CNC(CCC=C)=O)(C)C)=O)CC(COC)CC1(C)C 6782,C(CCN=c1[nH]ncs1)NC(C1CC(c2cccc(Cl)c2)(C(F)(F)F)C1)=O 6783,C(=O)(C(C)(C)CC(C)(C)C)N(CC(CC)NC(c1cnc(C)c(C#N)c1)=O)C 6784,C(CN=C(NCC(=O)NC(C)C)NC1CCN(S(C)(=O)=O)C1)c1ccc(C)cc1 6785,N1(C(C2CC2c2ccccn2)=O)CCC(C2CC2NC(C2(F)CCCC2)=O)CC1 6786,Cc1oc2ccccc2c1CC(N1CCC(NC(C2(CCF)CC2)=O)C(F)C1)=O 6787,C(=O)(CS(=O)(=O)CCC(F)(F)F)N1CCCC(NC(C(N2CC(C)C2)C)=O)C1 6788,C(=O)(NNc1ncnc2sc3c(c12)CCC3)C(C)C(N1CCCCC1C)=O 6789,n1(CC(=O)NCCC(C(C)C)NC(C2CCC(C)(C)C2)=O)cc([N+](=O)[O-])cn1 6790,CC(C)(C(F)(F)F)OCC(=O)NCCCCNC(C1CCCN1C=O)=O 6791,c1(C(=O)OC)cc(Cc2cn(Cc3cc(CO)cc(I)c3)nn2)ccc1Br 6792,N1(C(C(CC(=C)C)NC(c2ccc(C)c(F)c2)=O)=O)CCC(O)C(F)(F)C1 6793,CC(C(=O)NC(C1CCN(C(C2CCCN(C(N)=O)C2)=O)C1)(C)C)S(N)(=O)=O 6794,CCCCCCC(=O)NC1CC(CCNC(c2cc(Br)co2)=O)C1 6795,C1(C(C)C)CCC(C)CC1C(=O)NC(CNC(C1(CCO)CC1)=O)C(C)(C)C 6796,CC1(O)CN(C(=O)CCC2CCN(C(=O)CN3CCOCC3)CC2)CCC1O 6797,C(=O)(C1=NOC(C)C1C)NCCn1cc(NC(CSCCC)=O)nn1 6798,CCC(C)C(C(=O)NC1(C(C)O)CC1)N(C)C(C1CCCCN1C)=O 6799,c1(C(N2CC(C)C(C(=O)Nc3cc(S(N)(=O)=O)cs3)C2)=O)csc2ccccc12 6800,C=CCCC(C)NC(C1(CNC(c2occc2CSC)=O)CCC1)=O 6801,c1(OC)ccc(C(=O)NCC2(NC(=O)Cc3ccsc3Cl)CCOC2)cc1OC 6802,C(CCCCC(=O)NCCCN(C)C(C1(NC(N)=O)CCCCC1)=O)=CC 6803,C1(C(=O)OC(CC#C)c2ccco2)OCCC12CN(C(=O)OC(C)(C)C)C2 6804,C1(C(N2C(C)CCCC2)=O)N(C(c2ccco2)=O)CCCC1(C)C 6805,c1(OC)ccccc1C1CC1C(N1CC(NC(C2COCCOC2)=O)C(C)C1)=O 6806,CC1(C)OC(=O)CC1C(N1CCC(CCC(=O)NCCc2cnccn2)C1)=O 6807,C1(C(N2C(CN(C(=O)CS(N)(=O)=O)C)CCC2)=O)CCC2(CC1)CC2(F)F 6808,C1(NC(C(CC=CC)C)=O)CC2(C1)CC(C(=O)N(C)CC1(CO)CCC1)C2 6809,Cc1cc2ccc(C(=O)N(CC(C)N(C(=O)CCc3ccco3)C)C)cc2o1 6810,c1(CCC(=O)N(CCN(C(c2c(C)nn(C)c2)=O)C)C)ccc(Cl)cc1F 6811,c1(C(=O)NC(C2CCCCN2C(c2cnc(Cl)s2)=O)C)cc2cccc(Cl)c2o1 6812,c1(CC(C)(C)CO)nc(C2(C3CCCNC3)CCC2)n(C2CCSCC2)n1 6813,CCC(CC(=O)N1CCC(N(C)C(C23CSCC2C3)=O)C1)C1CCC1 6814,c1(C(=O)NC2C3(CN(C(C4C(C)C4)=O)C3)CCC2)coc2c1C(=O)NCC2 6815,C1(NC(C(C)NC(CC)=O)=O)CCCCN(C(=O)CCC=CC(C)C)C1 6816,C1(C)(NC(C(CCC)OC)=O)CCCN(C(c2c[nH]cc(Br)c2=N)=O)C1 6817,C(=O)(C1=C(C)OCCC1)N(C1CCC(CNC(c2c(OC)scc2)=O)CC1)C 6818,c1(CC(=O)NCCCN(C(=O)CSCc2ccccc2Cl)C)ccc(O)nc1 6819,CC1CCN(C(=O)CCN(CCO)C(c2ccc(C3CC3)o2)=O)CCS1 6820,c1(C(N(C2CCN(C(C(CC)F)=O)C2)C)=O)ccc([N+](=O)[O-])cc1Br 6821,N1(C(C=Cc2cn(C)nn2)=O)CCC(NC(c2cc(C3CCC3)no2)=O)C12CC2 6822,CCCCCCCCCC(O)C(=O)NC1(C)CC(NC(c2cc(C)n(C)c2)=O)C1 6823,C1(CNC(C2C(NC(COCC(=C)C)=O)COC2)=O)CCCCN1C 6824,C1(NC(c2c(OC)noc2C)=O)CCCCN(C(=O)CC(C)c2cccnc2)C1 6825,C(C1C(C(=O)NCC2(F)CC(NC(=O)COCC(C)(C)C)C2)C1(C)C)=C(C)C 6826,C1(F)(C(N2CC(C)(CC)C2)=O)CCCN(C(c2ccc(Cl)cn2)=O)C1 6827,C1(CC(=O)Nc2cccc(CNC(=O)C(F)(F)C(F)F)c2)CCS(=O)(=O)CC1 6828,C1(O)(CC(=O)NCC(CNC(c2c(C)nc(C3CC3)[nH]2)=O)(C)O)CCCCCC1 6829,C1(CCOC)(NC(c2scc(C)c2C)=O)CCN(C(=O)CC2COCCN2C)C1 6830,c1(OCC(=O)NCC2CCCN2C(=O)CC23CCCC2C3)ccc(C(F)(F)F)nc1 6831,c1(SCCC)ccc(C(=O)NC2CCC(NC(C3CC(CC(F)F)C3)=O)C2)cc1 6832,C(=O)(C1=CCCCC1P(C)(C)=O)NC1CN(C(C=CC=CC)=O)C(CCOC)C1 6833,CCC(CC(=O)N1CCC(C)(NC(c2ccc(C(F)F)cc2)=O)C1)OC 6834,N1(C(c2cccc(CC)n2)=O)CC2CC1CC2N1CC(C(N)=O)(C(N)=O)C1 6835,CC1COC(CNC(=O)N(C2CCN(Cc3ccccc3)C2)C)C1 6836,c1(C(=O)NC2CCN(C(C#CC3(C)CC3)=O)C23CCC3)ccc2c(c1)CCC=C2 6837,c1(C(=O)NCc2cccc(C(N(CC(C)C)CC)=O)n2)cccc2ccoc12 6838,n1(CC(C(N2C(CNC(CSCC)=O)CCC2)=O)C)ncc2ccccc12 6839,c1(OCC(=O)NCCNC(c2cccc(COC3CCC3)c2)=O)ccc(Cl)cc1 6840,C(=O)(CCCCC(C)(C)C)N(CC(CC)NC(c1cncc(OC)n1)=O)C 6841,n1(CCC(=O)NC2C(CNC(c3c(C)ocn3)=O)CCC2)c(C)cc(O)cc1=O 6842,CCCCCC(C)(C)C(=O)NCC(CO)NC(=O)C(c1cccc(F)c1)O 6843,c1(N2CCC(CC(=O)NCCC=C)C2)cc(OC)nc(OC)n1 6844,C1(NC(c2nc(COCC)sc2)=O)C=CCN(c2nccc(CO)n2)C1 6845,N1(C(COC)=O)CCC2(CCCN2C)C1.C1(C)C(=O)N(C)C2CC(C2)O1 6846,C1(CNC(c2cc(O)ncc2Br)=O)CCCN(C(c2cnc[nH]2)=O)CC1 6847,C1(COC)(NC(c2cc(Cl)c[nH]2)=O)CCN(C(=O)Cc2ccc(F)cn2)CC1 6848,c1(C(=O)NC(C(C)(C)NC(c2cc(COC)on2)=O)C)ccc2c(c1)CCCS2 6849,N1(C(CN(CCC)C)=O)CC(NC(C2(O)CCSC2)=O)CC2(CC2)C1 6850,N1(CC(=O)NC(CC=C)CNC(=O)C(C)OC)C(=O)c2cc(Cl)c(Cl)cc2C1=O 6851,C(=O)(CS(=O)(=O)C(C)(C)C)N1CCC(NC(c2cccc(OC)c2C)=O)C2C1C2 6852,c1(C(=O)OCC)ccc(S(=O)(=O)N2CCC(O)(c3ccccc3Br)C2)c(F)c1 6853,C(CCN(C)C(C1(C)CSC1)=O)(C(C)(C)C)NC(C(CCC)NC(N)=O)=O 6854,N1(C(CNC(=O)OC)=O)C2CCC1CC(CNC(=O)CC1CCCOC1)C2 6855,N1(C(C(=O)NC(c2nccn2C)C)C)CCC(C(N2CCCC2)=O)CC1 6856,c1(C(C(=O)N(C(C)CNC(c2ccsc2)=O)C)C)ccc2ccccc2c1 6857,C1(CC)CN(C(=O)C(CC)SC)CC1NC(C)=O.n1(CC)cncn1 6858,c1(C(=O)NCC2(CNC(CC(=C=C)C)=O)CCOCC2)ccc(Cl)c(CC)c1 6859,C1(CC(=O)NC(C(=O)NCc2nc(CC)[nH]n2)C2(O)CCC2)C=NN(C)C1=O 6860,N1(C(C2(C#N)CC=CC2)=O)CC(NC(C2CC(F)(CO)C2)=O)C(N=[N+]=[N-])C1 6861,CCC(CCO)NC(=O)CNC(=O)C(c1cnn(C)c1)O 6862,C1(NC(c2c(CC)onc2)=O)CCCN(Cc2cc(F)ccc2F)CC1 6863,N1(Cc2cc(OC)c(Br)cn2)CCOCC2(COCCN2C)C1 6864,C1(C(=O)NCC(=O)OCC=C)CC2CCC1N2C(C1CC(=O)C1)=O 6865,N1(C(c2cc(OC)no2)=O)CCCN(C(=O)C2=CCC(C)CC2)CC1CO 6866,C(=O)(C1=CCN(C)C1)C(C1CC(CCN)OC1)=O.N1(CC)CCCC1(C)C(C)(C)C 6867,C(=O)(CC(C)CC(C)(C)C)NC1C2CCN(C(CCS(=O)(=O)NC)=O)C2C1 6868,c1(CCC(=O)NCC2CCN2C(c2cnn(C(F)(F)F)c2)=O)nnc(C(F)F)o1 6869,C1(C)(CNC(c2c(C)nn(C)c2C)=O)COCCN(C(=O)CC(F)(F)Cl)C1 6870,C(C(CNC(c1ccc([N+](=O)[O-])[nH]1)=O)C(F)(F)F)NC(C1N(CC)CC1)=O 6871,Cc1ccc(C(C)(F)F)cc1NCc1cc(F)ncc1F 6872,C(=O)(C(C)C(C)S(C)(=O)=O)NC1(CCNC(c2ccn(CCC)n2)=O)CCCC1 6873,CCCC(C(=O)NC1CCCN(C(=O)Cn2cnnn2)C1)c1cccc(Cl)c1 6874,Cc1ccc(C(=O)NC2CC(CNC(c3cc(=O)n(C)cn3)=O)C2)c(C2CC2)n1 6875,NS(=O)(=O)C1(C(=O)NC2CC(NC(=O)C=Cc3cocn3)C23CCC3)CCC1 6876,CN1C(=O)CCC1C(=O)NCC1CCCCC1NC(c1cccc(C2CC2)c1)=O 6877,CC(CCCCN=c1[nH]cc2ccnc-2[nH]1)NC(c1cc(C(F)F)on1)=O 6878,N12CCC(CC1)CCC2=O.N1(CCOCCOC2CN(C(C)=O)C2)CC2(COC2)C1 6879,CC1CCCC1N=c1[nH]c(N2C3CCC2COC3)nc2c1CCCC2 6880,C1(C(=O)NC2CC2)C2C3CC4C1C2C34C(N(C)Cc1ccc(C)cc1)=O 6881,C(=O)(CCC(C)(F)F)N(CC(C)NC(=O)CC1(C)CC(F)(F)C1)C 6882,C1(NC(=O)C=CC(N2CCOCC2)=O)CCN(C(N(C)C)=O)CC1 6883,c1(C(=O)NC(CNC(c2c(C#N)ccs2)=O)C2CC2)cccn2c(O)nnc12 6884,N1(C(CC(C)F)=O)CCC2(CC(C(=O)Nc3ccccc3C3CC3)C2)C1 6885,C1(CNC(CC=C=C)=O)(CO)CCCN(C(=O)Cc2c(C)nn(C(C)C)c2C)C1 6886,c1(C(N(CCCNC(=O)C(C)C(F)F)CCC)=O)cccc2ncnn12 6887,C(C(=O)NC1CCN(CC(=O)Nc2cccc(C)c2)CC1C)(C(C)(C)C)OC 6888,CC1(C)C(C)(C(=O)NC2CCC(NC(=O)CC(=O)NC3CC3)CC2)C1(C)C 6889,Cc1cc(=NCC2CC(NC(=O)C3COc4ccccc43)C2)[nH]c(S(C)(=O)=O)n1 6890,C(C(CC(=O)NCC(C)C(=O)OC)SC1CC1)NC(CN(CC)CC)=O 6891,C1(NC(C(=Cc2ccccc2)OC)=O)CN(C(C2(O)CC2)=O)CC1(C)C 6892,C(CC(N)=O)(C(=O)N1CCNC(=O)C1)NC(C1OCCN(C)C1)=O 6893,C1(C(N)=O)(NC(C2(O)CN(CCCc3nn[nH]n3)C2)=O)CC2CCC1C2 6894,CC1COCC(C(=O)N(C)CC=CC(=O)N(C2CCCC(O)C2)C)O1 6895,N(C1CCC2(CC2)c2cc(Br)ccc21)C1CCC2C(F)(F)C2C1 6896,c1(SCC)cc(Cl)ccc1C(=O)NC1CCC(NC(=O)C(C)n2cccc2)CC1 6897,N1(C(C2(c3cccc(-c4cnn(C5CCOC5)c4)c3)CCC2)=O)CC(O)C(O)C1 6898,CC1(C)CC(C)(C(N2CCC3(CCC3)C2)=O)CN1C(=O)CC#N 6899,N1(C(C2C(CCC)CCC2)=O)CC(F)CC1CNC(=O)CNC(=O)OC 6900,C1(NC(c2c(C)nccn2)=O)CCCC12CCN(C(=O)C1=CCS(=O)(=O)C1)C2 6901,Cc1nc(S(=O)(=O)NCC(=O)NCC(C)(O)CNC(=O)CC=CC(C)(C)C)cn1C 6902,C(=O)(C1=CCCCCC1)NC1CC(F)(CNC(=O)CC2CCCNC2=O)C1 6903,CCCCCC(O)CC(=O)N(CCCN(C)C(c1ccnc(F)c1N)=O)C 6904,C1(NC(C2N(C)CCCC2)=O)CCC2CC1CN2C(C1CCC(O)CC1)=O 6905,C(CCCCCNC(=O)C(C1CCN(C(=O)C(CO)NC(N)=O)C1)F)N(C)C 6906,N1(C(N(C)Cc2c(CC)cccc2)=O)CCCC2(CCCO2)C1 6907,c1(NCC)ccc(Cl)c(C(=O)NC2(n3cc(C#N)cn3)CC2)c1 6908,CC(C)(CCC(=O)NC1CCC(NC(c2cnc(N)cn2)=O)CC1)[N+](=O)[O-] 6909,CC1(C)CCC(CCNC(=O)C(CNC(=O)C(F)=CC2CC2)CC2CC2)O1 6910,N1(C(C=CCCC)=O)CCCC2(C1)CN(C(=O)Cc1nc(C)c(C)[nH]1)C2 6911,C1(NC(C2(C)CCCN(C)C2)=O)CCCCCN(C(c2ccsn2)=O)C1 6912,Cc1cc(N)c(C(=O)NC2CC(CNC(c3cn(C)c(O)n3)=O)C(O)C2)c(F)c1 6913,c1(C(N(CC(CC)NC(c2ncc(OC)cc2F)=O)C)=O)c(C)cc(C)nc1S 6914,N1(C(CC2(CNC(C(C)SCC)=O)CC2)=O)Cc2c[nH]nc2C1 6915,C12(NC(C3CCCCC3)=O)CCCC1N(Cc1cscn1)CC2 6916,c1(CC(=O)NCCCCC2CCCN(C(C(C)(C)O)=O)C2)cccc2nsnc12 6917,C1(C(=O)NC(CCN(C(COCC)=O)C)C(C)C)CC2(C1)C(F)(F)C21CC1 6918,N1(C(C(C2CCCC2)OC)=O)CCC(NC(=O)C(N)=O)C(C)(C)C1 6919,C1(NC(c2c(COC)ncs2)=O)CN(C(C2COCCN2C)=O)CCC1O 6920,C1(C2CC2)(NC(CCC(C)(C)F)=O)CCN(C(c2cc(Cl)c[nH]2)=O)C1 6921,C1(CNC(c2n(C=C)ncc2)=O)CCN(C(c2ccc(F)cc2C)=O)CC1C 6922,N1(C(c2n(CC)ncc2)=O)CCOC(C)C1C(N1CC2(CO)CC2(CO)C1)=O 6923,C(CC(=O)NOCCOC)(C(F)(F)F)NC(C1(CC=C)CCCC1)=O 6924,c1(NC(C2(C)N(C(CC)=O)CC2)=O)ccccc1S(=O)(=O)C(C)C 6925,N1(C(c2c(C)nn[nH]2)=O)CCN(C(=O)Cc2ccc(Cl)s2)C(C)C1C 6926,CC1CCN(C(=O)C(O)Cc2cn(C)cn2)C(CNC(c2cnccn2)=O)C1 6927,N1(CC(=O)O)CCN(C(c2ccc(SC3(C(F)(F)F)CCOC3)cc2)=O)CC1 6928,CC1(C)CCC(C(=O)NCC2CC3(C2)CN(C(c2csc(C(F)F)c2)=O)C3)CC1 6929,C1(NC(C2C(C)C2C)=O)CN(C(=O)CC2CC3(CCO2)CC3)C2(CCCC2)C1 6930,Cc1ccc(Br)cc1C(c1nnnn1C1CC1)NC(Cc1cnn(C)c1)C(=O)O 6931,C(=O)(C(C)(C)COC)NCC(CC)NC(c1cccc(F)n1)=O 6932,C(=O)(CN=c1cc[nH]cc1)N(CCOCCC(=O)NC(C)CCn1cncn1)C 6933,Cc1cnc(O)c(NC(C2(O)CCN(Cc3ccc(Br)c(O)c3)C2)=O)c1 6934,N1(C(CCCC(C)c2cn(C(C)C(=O)O)nn2)=O)CCC2COC(=O)NC2C1 6935,C(=O)(CC1CCOc2ccccc21)N(C(CCNC(CC(=O)NCC)=O)C)C 6936,c1(OC)cc(C(=O)NCC=CCC(=O)N(C)CCc2cnccn2)n(C)n1 6937,CC1CN(C(C2(CCNC(c3n[nH]c4ccccc34)=O)CC2)=O)CC(C)(C)O1 6938,N1(C(CCCCOCCC=C)=O)CCN(C(=O)CCC(C)SC)CC1CC(F)(F)F 6939,C1(CC(=O)NCC(F)CNC(C2(C)CCOC2)=O)(CC=C)CCCC1 6940,N1(C(C(CCNC(CCc2c(C)noc2)=O)O)=O)CCC2(CCC2)C(O)C1 6941,C(C)(C(=O)OCCC(=O)N(C)C)N(C1CCCC1)C(CNC(C)=O)=O 6942,C1(F)(C(=O)NCCc2c(C(N(CC)CC3CCCO3)=O)c[nH]n2)CCOCC1 6943,CN1CC(NC(C2CCC3(CC3)N2C(=O)CC2C=CCC2)=O)C2(CC2)C1 6944,Cc1cccc(C(C)N(C2(C3CCCO3)CCC2)C(=O)OC(C)(C)C)c1 6945,CN(C)S(=O)(=O)N1CCC(CN2CC3(CCC3)C2c2ccsc2)CC1 6946,N(C(=Nc1ccc(OC)cc1CC)N1CCC(O)C(C)(C)C1)C(C=C)C 6947,S(=O)(=O)(c1cccc(F)c1)NCC1C(C(N2CCCNCC2)=O)C1 6948,CC1(C)CCN(C(C2(O)CCCCC2)=O)CC1CNC(c1c[nH]nc1Br)=O 6949,C1(CN(C(=O)C(O)COC)CC)CCCN1C(c1cnn(C(F)F)c1)=O 6950,N1(C(CCSC)=O)CCC(CN(CC(C)NC(=O)C=CC(F)(F)F)C)C1 6951,c1(-c2nc(C(C)C3CC3)nn2C2CCCOC2)ccnc(O)c1Br 6952,c1(OC)c(Cl)cc(NC(C2CC(O)CN2S(=O)(=O)c2cccs2)=O)cc1Cl 6953,Cc1cnc2n1CCCC2C(=O)N1CCN(C(C2C=CC=CC=C2)=O)C(CO)C1 6954,CC(C)C(N=[N+]=[N-])C(=O)N1CCC(C)(NC(c2ncn3ccccc23)=O)C1 6955,C(C)(CNC(=O)C(C1CCCCCC1)C)(CC(C)C)NC(C=C=C(C)C)=O 6956,Cc1ccc(C(N2CC(F)(C(N3CCN4CCOCC4C3)=O)C2)=O)c([N+](=O)[O-])c1 6957,c1(CC(C(=O)N(CCC)CCNC(=O)Cc2csc(S)n2)C)c(C)n[nH]c1C 6958,N1(C(C(C2CCN(C(c3ccnc(O)c3)=O)CC2)C)=O)CCc2ncccc2C1 6959,C1(O)(CN(C(C(CC=C)C)=O)C)CCCN(C(c2cnc(C(C)(C)C)o2)=O)C1 6960,C(=O)(CCC(C)(F)F)NC(CC(=O)NC1(C#C)CC1)COC 6961,CC(C)(C(=O)NCC=CC(=O)N(C1CC(C#N)C1)CCO)C1CCCC1 6962,c1(CCC(=O)N(CC#C)CC2CC2)ncc(F)cn1 6963,Cc1[nH]nc(C(N2CCCN(C(=O)CCCSC(C)(C)C)CCC2)=O)c1[N+](=O)[O-] 6964,n1(CCCC(C)O)cc(C#CCN(C(N)=O)CCC(=O)NC(=O)OC(C)(C)C)nn1 6965,N1(C(c2ccc(C3C(C)C3)o2)=O)CCC(F)(CNC(=O)C(O)CC(N)=O)CC1 6966,C1(NC(=O)NCC2(CCOC)CCC2)CCC(C)c2ccccc2C1 6967,CC1CC(F)(F)CN1C(C1(NC(=O)C(O)C2CCCC2)CCSC1)=O 6968,CC(C)C(F)(CNC(=O)C1=CCCC1C)C(=O)NC(CO)C(=O)N(C)C 6969,c1(OC)cc(N2CCC(NC(C3(C4CCOCC4)CC3)=O)C2)c(F)cc1[N+](=O)[O-] 6970,C1(C(=O)NCC2(OC)CCCCC2)CN(C)CCN1C(c1cc(C)n(C)c1C)=O 6971,C1(C(N(CC(CN(C(C2(SC)CCC2)=O)C)O)C)=O)CC(C)(C(C)(C)C)C1 6972,C1(NC(C(C(=O)OC)C)=O)CC(F)(F)CC1NC(c1conc1C)=O 6973,N1(C(c2ccc(C#C)cn2)=O)CC2(CCN(C(=O)C(C)S(N)(=O)=O)CC2)C1 6974,Cc1ccc(F)cc1CC(=O)NCC1CC(NC(c2cc(=O)n(C)o2)=O)C1 6975,O=C(CCC(=O)NC1C(NC(c2ccns2)=O)CCOC1)Nc1cccs1 6976,N1(C(c2c(C)nns2)=O)CC(NC(c2occc2F)=O)CC(O)C1 6977,Cc1cc(C(=O)NCC(=O)NC2COCCC2NC(=O)CC2CCCO2)n(C)n1 6978,c1(OC)c(C(=O)NC(C)(C)CCCNC(C2CCC(=O)O2)=O)cc(F)cc1F 6979,C1(NC(C(C)COCc2cccc(C)c2)=O)CCCN(C(=O)C(C)(F)F)CC1 6980,C12(NC(CCCC=C)=O)CCC(F)(F)CC1CN(C(=O)CCC(C)CC)C2 6981,N1(Cc2onc(CC)n2)CCC(CO)(NC(C2CCCN2C(C)=O)=O)CC1 6982,Cc1c(Cl)ccnc1NNC(=O)CN1CCCCC1=O 6983,n1(CC)nc(C)cc1C(=O)NC1C=CCN(C(c2ncoc2Br)=O)C1 6984,c1(CCC)c(C(N2CCC2CNC(c2nccnc2N)=O)=O)nnn1CC 6985,C1(CNC(C2C3(CCN(CC(=O)OCCC)CC3)C2)=O)CCC2(CCCC2)CC1 6986,n1(CC(=O)N(CC(CN(C(=O)CC2C=CCCC2)C)O)C)ccc(Br)n1 6987,c1(C(N2CC(NC(CCN(C(C)=O)C)=O)C2)=O)cc(F)c(Br)cc1F 6988,N1(C(CC2(OC)CCCC2)=O)CCN(C)CC1CNC(=O)CC(C)CN(C)C 6989,C1(C(=O)NC(C2CCCC2)C)CN(C(c2[nH]ccc2C2CC2)=O)CCN1C 6990,c1(CC(=O)NCC(C)N(C(=O)CC2CC(=O)NC2=O)C)c[nH]c2c(F)cccc12 6991,Cn1ccc2c(N3CC4CC4(CNC(=O)Cc4noc(C(C)(C)C)n4)C3)ncnc12 6992,C1(c2n(-c3c(SC)cccc3)nc(-c3cncnc3)n2)CC(=O)NC1(C)C 6993,c1(C2(NC(=O)NCC(F)C3CNC3)CCC2)ccccc1 6994,C1(CNC(C=CCOC)=O)CCN(C(c2ccc(F)cc2Br)=O)C1(C)C 6995,C(C(CC)CC(C)C)NC(C(=O)NC(CC#CC)C)=O.C1CN1 6996,C1(C(N)=O)CCC(C(=O)NC2CC(F)(CNC(=O)CC3COCCO3)C2)CC1 6997,C1(NC(Cc2cc(C)c(Cl)cc2)=O)COC2C(NC(C3(C)CCCC3)=O)COC12 6998,c1(OC)cc(CN2CCN(C)CC2C(C)C)ccc1OC(F)F 6999,N1(C(C2(C(=O)OC(C)(C)C)CCOC2)=O)CC2(COC(CNC(=O)C3CC3)C2)C1 7000,C(=O)(C(O)CCCNC(C1CCCSC1C)=O)NCc1cc(C)ns1 7001,CC(CCP(C)(C)=O)(c1nnnn1C1CCC1)NCCCCn1cnnc1 7002,N1(C(C(CC(C)C)N(C)C)=O)CCCC(NC(c2cn[nH]c2)=O)CCC1 7003,c1(CC(C(=O)O)NC(c2cc(C3CC(F)(F)C3)no2)=O)ccc(Cl)nc1 7004,N(C(=NCC1CC1)N1CCN2C(=O)CCC2C1)CC(c1ccc(C)cc1)O 7005,C(C)(CCCC(=O)NC(c1cn(C)nn1)C)NC(c1c(C)cccc1)=O 7006,C1(CCC#C)CCCN1C(=O)CCC1CCN(C(=O)CC2CCCSC2)C1 7007,C=C1CC2CCC(C1)N2C(=O)C(C(C)CC)N(C)C(c1ncc(F)cc1F)=O 7008,c1(OC)cc(CN2CCOC(C(=O)NCc3ccn(C)n3)C2)ccc1C 7009,CC1CC(NC(c2ccccc2-n2cncn2)=O)CN1C(=O)CC1(C)CCCC1 7010,Nc1cc(C(N2CC(F)(CNC(C3C(F)(F)C34CC4)=O)C2)=O)c(F)cc1F 7011,C1(CNC(CC(CC)OC)=O)CCC2(CCC2)CN1C(C1CC1C1CCC1)=O 7012,C1(C)(CO)CN(Cc2cn(CCC3CCCNC3)nn2)CCO1 7013,N1(C(C2N(CC)CCC2)=O)CCN(C(c2c(Cl)cnn2C)=O)CC1CC(=O)NC 7014,c1(-c2scc(C(=O)Nc3ncc(-c4ccccc4)cn3)n2)ccc2sccc2c1 7015,c1(C(N2C3CCC2CC3)=O)cc(NC(c2ccc(C(=O)OC)s2)=O)n(C)n1 7016,CC1(C)CN(C(c2cccc(OC3CC3)c2)C(=O)NCC2CCCC2)CC1CO 7017,C(=O)(C(C1=NOC2CC12)N(C)Cc1ccc2c(c1)CCO2)NCCCOC 7018,N1(C(C(=O)NC2CC3(CC(OC)C3)C2)=O)CC2(CCC2)CC1CO 7019,Cc1cnoc1C(=O)N(CCC(C)C)C(C)(C)C.C12CCN(C1)N(C)C(=O)C2F 7020,N1(C(CC(CC)SC)=O)CCC(CNC(c2cnc(O)c(F)c2)=O)C(O)C1 7021,C12(NC(C(C)CN(C)C)=O)CCOC(CNC(c3ncccc3C(F)F)=O)(C1)C2 7022,c1(C(N2CCC(CNC(CNS(NC)(=O)=O)=O)CC2)=O)cc(F)c(Cl)cc1F 7023,c1(C(C(=O)N2CC(NC3CC(N4CCN(C)CC4)C3)C2)(C)C)c(F)cccc1F 7024,c1(CNC(c2c(NC(CC(=O)OC)=O)ccs2)=O)ccc2c(c1)COC2 7025,CN1CCC(CC(N2CC(c3ccccc3)(NC(C3C=CCC3)=O)C2)=O)CC1 7026,N1(C(CN2CCC(C)(O)C2)=O)CCN(C(=O)C(C)(C)O)CC12CCC2 7027,c1(CC(=O)N(C)CC2N(C(CCCCSC)=O)CCC2)cccc(F)c1O 7028,C(CNC(C1CN(C2CCC2)C1)=O)(CC(F)(F)F)NC(c1c(CC)nccn1)=O 7029,C(=O)(C(C)CS(C)(=O)=O)N1CCC(NC(c2sc(CC)c(C)c2)=O)C1 7030,CC(C)(C(=O)N(CCN(C)C)Cc1cn(-c2ccc(Cl)cc2)nn1)C(F)(F)F 7031,N1(C(C2N(CC)CC2)=O)CCOCC(F)(CNC(=O)C(=Cc2cnc[nH]2)C)C1 7032,CCC(C)(C#N)C(=O)NCC1(NC(=O)Cc2cnn(C(F)F)c2)CCC1 7033,S(=O)(=O)(c1ccc(C(=O)NC2CC3CCCCN3C2C)cc1)NC 7034,C1(C)(C(=O)NCCN(CC(C)O)C(c2cn(C)nc2O)=O)CC=CCC1 7035,C1(CNC(c2cnc(C3CC3)s2)=O)CCCN(c2cc(-c3ccccc3)ncn2)C1 7036,N1(C(CC(C)OC)=O)CCC2(CC1)CN(Cc1ccc(Cl)cc1C)CCO2 7037,c1(O)ccccc1Cl.C(C)(C(=O)OC1CN(C(=O)OCCOC(C)(C)C)C1)OCC 7038,C1(NC(C2CCCS2)=O)CCSC12CN(C(=O)CCc1nc3ncccn3n1)C2 7039,CC#CCCCC(=O)NCCN(C1CCCC1)C(c1cncc(CC)c1)=O 7040,c1(N(C)Cc2cccc(OCF)c2)nc(N2CCC(S(C)(=O)=O)C2)c2c(n1)COC2 7041,Cc1cc(=NCC2CC2(C)C(F)F)[nH]c(N2CCC2c2cc(C)oc2C)n1 7042,n1(CC)cc(CC(=O)NC2(CCNC(C3CC(CC(F)F)C3)=O)CCCC2)cn1 7043,c1(CN(C(C)C)C(=O)Nc2cccnc2Oc2ccccc2)cc(Br)ccc1F 7044,Cc1onc(C(=O)NC2CC2CNC(=O)CSc2ccccc2)c1Br 7045,C1(CNC(C2CC(=C)C2)=O)COC(C)(C)CN1C(=O)Cn1cnnc1O 7046,c1(OC)cc(-c2cc(C(=O)NCc3cc(Cl)ccn3)ccn2)ccc1CO 7047,C(=O)(CC(CC)C(C)C)NCC(C1CCC1)NC(CCN(C(CC)CC)C)=O 7048,Cc1oc(C)c(C(=O)NC(C2CCN(C(=O)C(c3cccc(O)c3)C)C2)C)c1C 7049,C1(C(=O)NC2CC(N(C(CSCCCC)=O)C)C2)CCc2nc(O)[nH]c2C1 7050,c1(CCC(=O)NC2(CNC(=O)CNC(=O)CC3CCCCO3)CC2)cccnc1 7051,Cc1nnn(NC(=O)CC23CCC2CN(C(=O)CCCOCCN(C)C)C3)c1C 7052,C1(NC(c2cc(C(N)=O)[nH]c2)=O)(CO)CCCN(C(C2CCCCS2)=O)C1 7053,C1(CNC(c2ncc(CC)cn2)=O)CN(C(c2sccc2F)=O)CCC1(F)F 7054,c1(CN2C(C(N3CCC(F)(F)C3)=O)CSCC2)cnc(Cl)cc1Cl 7055,C1(C(=O)NCC2N(C(=O)CCN3CCC(O)CC3)CC2)CCCC2NCCC12 7056,C1(CNC(C(c2n(C)ncc2)(F)F)=O)CN(C(c2ccsn2)=O)CCO1 7057,Cc1cnncc1C(=O)NCC(C)(C)CN(C(=O)COCC(=O)N(C)C)C 7058,N1(C(C(CC)=CC)=O)CCOC(C(C)NC(c2ccc(Cl)cn2)=O)C1 7059,c1(CCNC(=O)NC(CC(=O)OC)C2CCCCC2)nccc(C(F)(F)F)n1 7060,N1(CC)CC(C(=O)N(C)CCC2CCCCN2C(=O)CCSC)CC1=O 7061,C(=O)(CC(C(=O)NC1(C)CN(C(c2scnc2C(C)C)=O)C1)N(C)C)OC 7062,C1(C(N2CCC(NC(C=NOC)=O)C2(C)C)=O)CCc2nccn2C1 7063,N1(C(C2CC(SC)C2)=O)CCC2C(NC(=O)COCCOCCO)C12 7064,C#Cc1ccc(C(N2CCC(c3n[nH]cc3CNC(=O)C(O)C(C)C)C2)=O)nc1 7065,C(=O)(C1CCc2c[nH]nc21)NC1(CCCCNC(c2cnccc2Cl)=O)CC1 7066,C1(CCCCC)CCC(C(N2CCN(C(=O)CC3CCCCO3)CC2)=O)CC1 7067,CN1CCN(C(c2cc(Br)c[nH]2)=O)C(CNC(C2C3CCC(=O)C23)=O)C1 7068,C(c1cccc(C(F)(F)F)c1)=CC(=O)N(C1CN(C(C(F)OC)=O)C1)C 7069,C1(CC(C)NC(C(C)OC)=O)CCN(C(c2ccncc2)=O)CC1 7070,Cc1cc(C)c(C(N2CC(CNC(c3ccon3)=O)C(C)C2)=O)cn1 7071,C1(=CC(=O)NCC(CNC(c2nccc(Cl)c2F)=O)OC)CCCCC1(C)C 7072,CCC(C)(CNC(C1CN(S(=O)(=O)CC)C1)=O)NC(=O)C(C)(C)c1csc(C)c1 7073,c1(OC)cc(CC(N2CCN(CCNC(C3(O)CCCC3)=O)CC2)=O)ccc1C 7074,N1(C(CC(CC)(O)c2ccccc2)=O)CC2CN(C(=O)C(F)=CC3CC3)CC2C1 7075,c1(C(=O)NC2CN(C(c3cc(C)cc(O)n3)=O)C(C)CC2)[nH]cc2c1CCCC2 7076,C1(C(=O)NCC2C(C(N3C(C#C)CCC3)=O)C2(C)C)CC2COCC2C1 7077,c1(CNC(C(CC)C)(C)c2nnnn2CC2CC2)cn2c(C)cccc2n1 7078,C(=O)(C(F)(F)C(F)(F)F)NCC(CNC(c1ccnc(C)c1C)=O)(C)F 7079,c1(CC)[nH]c(=N)sc1C(=O)NC1CC(CNC(c2c[nH]cc2Br)=O)CC1O 7080,N1(C(C2C3CN(C(CC4(NC(C)=O)CC4)=O)C2C3)=O)CCCCCCC1C 7081,N1(C(C(C(C)OC)N(C)C)=O)CC(C)(C)CC1CC(=O)N(CC(C)(F)F)C 7082,c1(CN(C)CC2CN(C(c3cn(CC)nc3)=O)C2)c(F)ccc(OC)c1Br 7083,O(NC(=O)C(c1cccs1)NC(c1coc(CO)c1)=O)CCCC#C 7084,C(C)(C)(CC(=O)NCC(Cl)C(C)(F)F)N(C(CN1CCC(C)C1)=O)C 7085,N1(C(c2scc(OC)c2)=O)CCC2(CCCN2C(C2(O)CCC(C)(C)CC2)=O)C1 7086,c1(NC(c2nccs2)C)nccc(N2CCC(N3CCOCC3=O)CC2)n1 7087,N1(C(C(c2cccc(F)c2)(C)C)=O)CCOC(CNC(c2csnn2)=O)C1 7088,c1(C(C(N2CCC(NC(C(C)OC(C)(C)C)=O)C2)=O)(C)C)cc(Cl)cc(Cl)c1 7089,C(C(CC(C)C)C(=O)NC(C)C(C)NC(c1csc(SC)n1)=O)OC 7090,c1(C(N2CC(NC(CCc3n(C)cnn3)=O)C3C2C3)=O)cc2sc(Cl)cc2s1 7091,N1(C(c2n(C)ncc2Cl)=O)CCC(NC(=O)Cc2c(O)ncnc2O)CC(O)C1 7092,CCC(CCC(=O)NC(C1CCCOC1)(C)C)NC(=O)CN=[N+]=[N-] 7093,N1(C(CCSCC)=O)CCCOC(CCNC(=O)Cn2ccc(C)n2)C1 7094,Cc1c(C(C)NC(C2(c3ccccc3)CCOC2)C)cnn1-c1ccccc1 7095,C(=O)(C1=Cc2ccccc2C1)NC1(CNC(C(C(CC)O)C)=O)CC(F)(F)C1 7096,c1(NC(CC(CC)NC(c2cnn(C(C)C)c2)=O)=O)cc(CO)ccc1C 7097,CCC(C)(C)CC(=O)Nc1cccc(NC(C2CCCS(=O)(=O)N2)=O)c1 7098,c1(C(N2CC(C)(C(C)C)OCC2)C(=O)Nc2ccccc2)noc2ccccc12 7099,N1(C(CCOCCC)=O)CCC2CCCC12C(=O)NC(CO)C(C)(C)CO 7100,C1(C(=O)NCC2N(C(C3N(C(CC)=O)CSC3)=O)CC2)CC(S(C)(=O)=O)C1 7101,S(=O)(=O)(c1ccn(-c2ccccc2)n1)NC1C([N+](=O)[O-])C1 7102,O=C(N=c1ccn(CCC(=O)N2CCCC2)[nH]1)c1ccnc(F)c1 7103,C1(N(C(CN(C(=O)CCOC(C)C)CC)=O)C)CC2CCC1O2 7104,n1(CCC)cnc(C(=O)NC2(CNC(=O)C(CC)N(C)C)CCOC2)n1 7105,C1(CN(C(C=CC=CCC)=O)C)CCCN1C(=O)C(F)(F)c1cnn(C)c1 7106,c1(C(N(C2CCN(C(C3CCC(=O)C3)=O)C2)CC)=O)cnn2cccc(Cl)c12 7107,c1(CC(N2CCC(F)(CNC(C(CCC#C)O)=O)C2)=O)ccc([N+](=O)[O-])cc1F 7108,c1(CC)nccnc1C(N1CC(OC)C(C(=O)NCCCCCO)C1)=O 7109,C1(C)(C(=O)NCC2CCN(C(C)C)C2)CCN(C(C23CC(CO2)C3)=O)C1 7110,CC(C)CC(C)C(=O)N1CCC(N(C)C(C2CC3C=CC2CC3)=O)CC1 7111,C(=O)(CC(=O)NC(C)C(=O)NCCCc1cscn1)OC 7112,Cc1nn2c(C(=O)NC3CN(C(c4cc(CF)on4)=O)CCC3C)c(C)nc2s1 7113,c1(C(=O)NC2CCN(C(CNC(C)=O)=O)CC2C)cc2c(nn1)CCCO2 7114,N1(c2n(CC(C)C)c(C3CCS(=O)(=O)C3)nn2)CC2C(C1)C2(F)F 7115,N1(C(C2(C#C)CC2)=O)CCC2CCN(C(C3CC4(C3)CC4F)=O)CC2C1 7116,C(C1=NOC(C)C1)NC(C(Cc1ccoc1)NC(CC(C)SC)=O)=O 7117,CCCCCC(O)CC(=O)NC(C1CCN(C(=O)C(C#N)CC)C1)C 7118,c1(C(C(=O)NCCSC)NC(=O)CN(C)C)cncn1C 7119,c1(C(=O)NC(CN(C(=O)CCc2cncn2C)CC)C)cc(N)cc(F)c1 7120,C1(NC(N(CCN(C(=O)Cc2ccc(C(=O)OC)s2)CC)CC)=O)CC2CC2C1 7121,c1(CC)cccc(C(N2CC(N(C(=O)C(F)C(F)(F)F)C)C3(CC3)C2)=O)c1N 7122,C1(NC(C(Cc2ccsc2)NC=O)=O)CCN(C(=O)C(=O)NC2CC2)CC1(F)F 7123,C1(C(=O)OC)CCN(C(=O)C(CC(N)=O)NC(=O)CSC(F)F)O1 7124,c1(C(C)O)ncc(C(=O)NCC2(CNC(c3ccc(CO)s3)=O)CCC2)s1 7125,C1(C(N2CCN(C(COCC)=O)CC2CC(F)(F)F)=O)Cc2cc(C)ccc2S1 7126,C1(CCNC(C(C)Cc2cnn(C)c2)=O)CN(C(c2ccc(Cl)[nH]2)=O)CCO1 7127,C(c1ccco1)=CC(N1CCC1C(N1CCCC1C(O)CO)=O)=O 7128,c1(C(=O)NCC(CNC(c2c(C(C)C)nns2)=O)F)cccn(C2CC2)c1=O 7129,C(=O)(CC(CNC(C1CCCC2CC12)=O)C1CC1)NCCSC(C)C 7130,c1(CCNC(C(C2CC(NC(C3(C)CC3(F)F)=O)C2)F)=O)ccccc1O 7131,N1(C(c2c(CC)occ2)=O)CC(F)(F)CC1CNC(C1CC1C(=O)NCCO)=O 7132,Cc1nn(C)cc1NC(=O)CNC(=O)NC(c1ccccc1C(C)C)C 7133,Cc1c(C(=O)NC2CCN(C(=O)C=CCO)CC2CO)cc(C2CC2)n1C 7134,C(C(C)(C(=O)NC(C)C(=O)NCC(c1ccsc1)O)OC)OC 7135,N1(CC(C)CN(C)C(=O)NCC2CC2c2ccc(N(C)C)cc2)CCCS1(=O)=O 7136,C=CC(CC)CC(=O)N(C1CCCN(C(=O)Cc2ccn(C3CCCC3)n2)C1)C 7137,C1(C(=O)NCC2(CC)CCCC2)(CC)CCCN1C(=O)C1CC1 7138,c1(C(N2CCCN(C(C(C)(C)OC)=O)CC2)=O)ccc2c(c1)C(=O)NCC2 7139,c1(OCC)ccc(Cl)nc1C(N1CC2C(C1)N2C(=O)CCC(=O)N1CCCC1)=O 7140,N1(C(C(C)C2CC2)=O)CC2CC1CN(C(=O)CC1CSC1)C2 7141,c1(C(=O)NC2(C)CCN(C(CC(C)C3CC3)=O)C2)ccc2c(c1)CCCCC2=O 7142,c1(C(N2CC(CNC(CC(CC)O)=O)C(C(F)(F)F)C2)=O)cccc2cnnn12 7143,C1(C(=O)Nc2ccc(C)nc2)CCN(C(=O)C(O)C2CCC2)C12CC2 7144,c1(CC(=O)NCc2csc(C(N3CC4CC4C3)=O)n2)cccnc1F 7145,c1(OCC)cccc(C(N2CCCC(c3nn[nH]n3)(c3nn[nH]n3)C2)=O)c1CC 7146,C(=O)(C1=COCCO1)N(CCNC(c1cncc(OCC)c1)=O)CC1CC1 7147,c1(C(N(c2nccc(OCC)n2)CC2CCCN2)=O)ccc(F)nc1C 7148,CCCC(O)C(=O)N1CC(NC(c2conc2-c2ccc(Cl)cc2)=O)C(O)C1 7149,CCC(CC)(CO)C(=O)NCC(CC(F)(F)F)NC(c1c(C)ccn1C)=O 7150,C1(NC(C2(OCC)CCOC2)=O)CCCCC1CNC(=O)CCC1CCOCC1 7151,c1(-c2cn(CC3N(C(C(CCC)N(C)C)=O)CCC3)nn2)ccc([N+](=O)[O-])o1 7152,CC(CN=c1[nH]cnc(Cl)c1Br)N(C)C(c1cnc2[nH]cncc1-2)=O 7153,N1(c2n(CCCOCC)c(-c3occc3C)nn2)CCCC2(CCCO2)C1 7154,N1(C(C2CCCC(NC(Cn3c(C)ccn3)=O)CC2)=O)CCC2CCN(C)CC12 7155,CCCCC(CN=c1ccc(C(F)(F)F)n[nH]1)NC(=O)CNC(C)=O 7156,C12(C(=O)NCCCC(C)(C)C)CCC(CN(C(c3cc(=N)[nH][nH]3)=O)C1)C2 7157,N12CCCC1(C)c1cn(nn1)CC2=O.Cc1ncsc1OCc1ocnc1CO 7158,N1(C(c2nc(C)c(C)s2)=O)CCCCC12CC(NC(C1CC1C(F)F)=O)C2 7159,c1(C(N2C(C(=O)NCCCS(C)(=O)=O)CC(O)C2)=O)cc(F)c(Cl)c(C#N)c1Cl 7160,C1(CNC(C2(CCC)CC2)=O)CN(C(=O)C(C2CC2)OC)CCC1(C)C 7161,c1(-c2ccn(C)c(=O)c2)nc2ccc(C(N3CCN(C4COC4)CC3)=O)cc2s1 7162,c1(C(N2CC(CNC(C(CSC)O)=O)C(F)(F)C2)=O)cc(C)c(Cl)c(C)c1 7163,c1(OCCC)cccnc1C(=O)N(CCCCN(C)C(c1cccs1)=O)C 7164,C#Cc1ccc(CC(=O)NC(COC)C(=O)NCc2nc(COC)n[nH]2)cc1 7165,C#Cc1cnc(C(N2CCCC2C(C)(C)NC(C2CC3CCC2C3)=O)=O)c(C)c1 7166,N1(C(c2ccc(C)cn2)=O)CCCC(C)(CNC(C2(C)CCOC(C)C2)=O)C1 7167,C1(CNC(C(=Cc2ccco2)C)=O)CCN(C(=O)CCC2CC2(Cl)Cl)CC1 7168,c1(C(CNC(C(=O)N(c2ncccc2F)CCOC)=O)SC)ccc(OC)cc1 7169,CCCCC(CNC(c1c(C)noc1C)=O)NC(c1cc(C(C)(C)C)n[nH]1)=O 7170,c1(CCC(=O)NCC2C3CN(C(C(=C(C)C4CC4)F)=O)CC32)cccc(Cl)c1Cl 7171,N1(C(c2ccsc2Br)C(=O)NCc2c(OC)cccc2)CCc2cc(Br)ccc21 7172,N1(C(CCOCCC)=O)C2CCC1CC(CNC(C1CCN(C)C1)=O)C2 7173,Cc1nn(C(C)C)c(C)c1CC(=O)NCCNC(c1cc(C(C)(C)C)no1)=O 7174,Nc1cccc(Cl)c1C(N1CCCC(N(C(=O)C#CC2CC2)CCF)C1)=O 7175,c1(C(=O)NC2(C)CCN(C(c3cncs3)=O)C2)cc([N+](=O)[O-])ccc1N 7176,N1(C(C(C(C)C)C2CCC2)=O)CCC(NC(=O)CCC2(C)CC2(F)F)C12CC2 7177,n1(CC(N2CC(C(=O)NC(COC)CO)(SC)C2)=O)cccnc1=O 7178,C(=O)(C(C#N)C(C)(C)C)NC(CCC(=O)NC1CC(OCC)C1)C 7179,C(C(C)N=c1[nH]c2c(c(=NCC=CCl)[nH]1)COC2)Oc1cc(C)oc1C 7180,n1(C2CN(C(C(N3CCSCC3)C)=O)C2)cc(-c2ncccn2)nn1 7181,CCCCS(=O)(=O)NC(C)C(=O)OCCc1ccnc(C)c1 7182,CCC(C)(CO)C(=O)N1CCC(C(C)NC(c2cccc(C3CC3(F)F)c2)=O)C1 7183,C1(COC(C)(C)C)(NC(=O)CCC2CCCC2)CCN(C(=O)CCC2CC2)C1 7184,c1(C(=O)NC(CC)(C)CNC(=O)C=Cc2cscn2)ccn2ncnc2c1 7185,C1(C(N(C2C(C)C2)C)=O)CCCCN(C(C2CCC2)=O)C1 7186,C1(C)(NC(C2C(C)CN(C)C2)=O)CCC(NC(C2C3CC4C(C3=O)C24)=O)CC1 7187,CCCCC(C)(F)C(=O)NC1CCC(C(=O)NCC(C)N(C)C)C1 7188,C1(NC(=O)CCC2(NC(c3cc[nH]n3)=O)CCC2)CC12CCCC2 7189,n1(CC(=O)OC)cc(C2CN(C(C3CC(n4ccnn4)C3)=O)C2)nn1 7190,c1(C(=O)NCC(CCCC)NC(c2c(C)cnn2C)=O)nnc(Cl)cc1N 7191,C1(NC(=O)Cn2cnnc2O)COCCC1NC(c1ccn(C(F)F)n1)=O 7192,c1(SC)ccc(C)c(C(=O)NCC2COCCN(C(=O)Cc3cc(C)ns3)C2)c1 7193,c1(C(N)=O)ccnc(C(N2CC(OCCNC(=O)C(O)C3CC3)C2)=O)c1 7194,N1(C(C(C=CC)O)=O)CCCC(C2(NC(c3cc(=O)n(C)cn3)=O)CC2)C1 7195,N1(C(C2CCN2C(C2(n3cccn3)CC2)=O)=O)CCC(CO)C(O)C1 7196,C(C(=O)N1CCC(O)(CNC(=O)C(N)=O)C1)(C(C)C)NC(=O)OCC 7197,C(C(C)(C(=O)NCC(c1ccsc1)O)NC(=O)CCC(C)N(C)C)SC 7198,c1(COC)cc(NNC(=O)NCC(c2c(C)n[nH]c2C)C)ncn1 7199,C1(C(N2CCC(CCNC(c3n(C)cnn3)=O)CC2)=O)CCc2nc(O)[nH]c2C1 7200,C(=O)(C1=NNC(=O)CC1)N1CC(NC(C2CCN(C(CC)=O)C2)=O)C(C(F)F)C1 7201,c1(C(=O)NN(C(C2(CC)CC2)=O)C(C)C)cn(CC2CCCOC2)nn1 7202,c1(CN2CCN(c3ncc(-c4cnc(SC)nc4)cn3)CC2)c(Cl)ccnc1Br 7203,N1(C(C2CN(C(C(C=C=C)C)=O)CC23CC3)=O)CCc2ccccc2C1 7204,CC1CC(CNC(C2CC(=O)NC(=O)N2)=O)CCN1C(c1cnc(N(C)C)o1)=O 7205,CC1(C)COC(CC(N2CC(NC(=O)C(F)(F)CO)C2)=O)CO1 7206,c1(CNC(C2CC(CNC(=O)CN3CC=CC3)C2)=O)ncc(F)cn1 7207,Cc1cc(CC(=O)NCc2cc(C(=O)NCC(C)C(C)O)cs2)on1 7208,c1(CNC(C(C)N(C(C2CCN(CC)CC2)=O)C2CC2)=O)cc(C)nc(O)c1 7209,C1(c2n(CCC)nnn2)(Nc2cc(C)c(C)c(C)c2)CCCN2CCSCC12 7210,C1(C(=O)NCCCN(C(C2C(=C)C2)=O)C(C)C)CCc2nc[nH]c2C1 7211,C1(CNC(CNC(CC(C)(C)C)=O)=O)CN(C(C2CCNC(=O)C2)=O)CCCO1 7212,N1(C(C2C(=C)CC2)=O)CCC(C(C)(C)CNC(=O)Cc2cccnc2OC)CC1 7213,c1(NCc2nc(C(=O)NCC)cs2)cccc(NC)c1.C(N)(=O)N 7214,N1(C(C(=O)NC(c2scc(-c3ccc(C)s3)n2)=O)=O)CCOC(C(C)(C)C)CC1 7215,C(=O)(CC(C)CCC=C(C)C)NCC1C2CN(C(C3(COCC)CC3)=O)CC21 7216,C1(CNC(c2n(C)nc(C(F)F)c2)=O)CC2CCC1N2C(=O)CN1CC2CC2C1 7217,N1(C(C2CC(CC)(CC)C2)=O)CCCC2C1CCCN2C(C1CCC1)=O 7218,C1(C(N(CCC)CCC)=O)CC12CCN(C(=O)C(C)n1ccnn1)CC2 7219,N1(C(CC(C(F)F)c2cccc(OC)c2)=O)CCC2(C1)OCCO2 7220,Cc1ccc(CNCC2CCN(C(C3CNC(=O)N3C)=O)C2)cn1 7221,c1(C(C(=O)NCC=C)N(CC)Cc2ccc(C)c(C)c2)csc2ccc(C)cc12 7222,C1(NC(C(C)n2ccnc2)=O)CN(C(=O)COC2(C)CCOCC2)CC1C1CC1 7223,N1(C(C(c2cn(C)nn2)NC(=O)C=Cc2ccnn2C)=O)CC(C)(C)OCC1C 7224,c1(CNC(=O)Cc2cccc(F)c2)ccnc(OC2CCOC2)c1 7225,C1(NC(C2(C(C)C)COC2)=O)CN(C(=O)C(O)c2cnc[nH]2)CC1(C)C 7226,N1(C(CC=CCC)=O)CC(NC(c2c(C)noc2CC)=O)CC12CCCCC2 7227,C1(C)(C(N(CC(C)(C)NC(=O)CSC(C)(C)C)C)=O)CC(C#N)C1 7228,N#Cc1ccc(CNCC2CCCC3(CCC3)C2O)c2ccccc12 7229,N1(C(C(CCSC)(C)C)=O)CCC2CCN(C(=O)Cc3ncc(C)o3)CC2C1 7230,CC1CCCCC1C(=O)NC(C1CN(C(c2cncnc2)=O)CCO1)C 7231,C(=O)(C1=CC2(CCOC2)C1)N1C(C)(CC(=O)NCC(N)=O)CC1 7232,N1(C(C(C)CNC(=O)CCCN(C)C)=O)CCCC(O)CC1 7233,c1(C(=O)NC2(CCOC)CCN(C(=O)CC(C)SC)C2)cc2ccncc2s1 7234,Cc1ccc2ncccc2c1NC(C1CCN1C(c1cccc(C(F)F)c1O)=O)=O 7235,C1(NC(C2CN(CC(C)C)C(=O)C2)=O)CCN(c2nnco2)C(C)C1 7236,C1(CNC(c2c(C)coc2)=O)CCN(C(=O)CSCC(F)(F)F)CC1C 7237,N1(C(c2c(OC)cc(C)cc2C)=O)CC2OCCN(C(=O)C(C)NC=O)C2C1 7238,N1(C(CC(CC)C)=O)CCN(C(c2ccc(-c3ncccn3)cc2)=O)C(C#N)C1 7239,C1(C(N(CC(C)NC(c2c(N)ccc(CC)c2)=O)C)=O)CC2CC(O)CC(C1)C2 7240,CC#CCCCC(=O)N(C1CCCC(NC(c2nccc(F)c2Cl)=O)C1)C 7241,c1(OC)cccc2c(C(=O)NC3CCCCN(C(c4cnc(O)o4)=O)C3)csc12 7242,C1(NC(c2c(C)nc[nH]2)=O)CC(CNC(c2nc(Br)c[nH]2)=O)C1(C)C 7243,c1(SCC)cnc(O)c(C(=O)NCCC(C)N(C(=O)C(C)N(C)C)C)c1 7244,C=C(C)CC(C(=O)N1CCCC1C(N1CCC(n2cnnn2)C1)=O)OC 7245,C1(C(N2C(CCCNC(C=NOC)=O)CCCC2)=O)CCC=CCCC1 7246,C(=O)(C(C)(O)CC(F)(F)F)NC(c1ccc(Br)cn1)C 7247,C12(C(N3CCC(CCNC(c4ncn(C)c4)=O)CC3)=O)CC=CCN1CCC2 7248,O=C(NN1CCCCC1)NCCOCCC1CCCC1 7249,c1(OC)nc(N2CC(C(C)NC(c3snnc3C(C)C)=O)C2)cc(C)n1 7250,N1(C(c2c(C)c(C#N)[nH]c2)=O)CCOC2CN(C(=O)CC(C)C(C)(C)C)CC12 7251,CCC(C)C(C(=O)NCCC1CC(NC(C2(C)CC(F)C2)=O)C1)NC(C)=O 7252,c12nc(C)c(o1)CNC(=O)C(c1ccccc1)NC2=O.C1(CC)CCCC2CC12 7253,c1(CN2CCN(C(N3CC(OC)C(O)C3)=O)CC2)oc2ccccc2c(=O)c1C 7254,c1(OC)ccc2c(=NCCC#N)[nH]c(N3CCC(Cn4cccn4)C3)nc2c1 7255,CC1CC(NC(c2ccnc(C3CC3)n2)=O)CN1C(c1cnn(C)c1Br)=O 7256,CC1(C)CCCOC1CNC(=O)CC12CCC1CN(C(=O)CC(F)(F)F)C2 7257,C1(CNC(C(CC)OCC)=O)(CO)CCN(C(c2csc(SC)n2)=O)CC1 7258,c1(C(=O)NCC#CCNC(CC(C)O)=O)cc(Br)ccc1Cl 7259,Cc1ccc(N)c(C(=O)NC2CC(NC(=O)CC3CCCC4(CC4)C3)C2)c1 7260,c1(C(N2CC(C)N(C(=O)CCc3cc(Cl)no3)CC2)=O)cccc2oc(=N)[nH]c12 7261,N1(CC)CC2CN(C(=O)C=CCC3(NC(C4CC(=O)OC4(C)C)=O)CCC3)CC2C1 7262,c1(C(N2CC(NC(C(c3ccccc3F)(C)OC)=O)C2)=O)cnc(C(F)F)nc1 7263,C(CO)(C(C)(C)CO)NC(C1C(C)CN(C(=O)C(O)Cn2cncn2)C1)=O 7264,C1(C(N(CCCN)CCO)=O)CCCN1C1CCC(c2ccccc2)C1 7265,c1cc(-c2noc(-c3cc(OC4CCCC4)ccn3)n2)c2c(c1)CCCC2 7266,N1(C(C2CN(CCC)C(=O)C2)=O)CCCN(C(c2cncc(O)c2)=O)C(C)C1 7267,c1(N2Cc3c(C)cnn3CC2)nc(=NCC2CCO2)[nH]c2c1CCCCCC2 7268,C1(NC(C2C(C(=O)OC)C2)=O)CCC(NC(=O)Cc2ccccc2C)CC1 7269,C(C(=O)NC1CC2CCC1(NC(C1CCCCC1)=O)C2)(C(C)(C)C)NC(N)=O 7270,C(=O)(C(CCO)N(C)C)NCC(CC)NC(c1sc(C)nc1CC(C)C)=O 7271,C=CC1(NC(C2CC2NC(=O)COC(C)CC)=O)CCCCC1 7272,c1(CNC(CCN(C(=O)C=Cc2ccccc2)CC)=O)cc2ccccc2[nH]1 7273,C(=O)(C1CCCc2scnc21)NC1CCN(C(C2(CN(C)C)CC2)=O)CC1F 7274,C(=O)(C1=C(C)OCCS1)NC(COCC)C(=O)Nc1ccc(C)c(CC)c1 7275,C1(NC(C(C(C)C)OC)=O)CN(C(=O)CCc2ccc(F)nc2)CCC1C 7276,C1(C(=O)Nc2c(OC)noc2C2CC2)CCN(C(=O)CC(C)OC)CC1O 7277,c1(OC)ccc2[nH]c(C(N3CC4CC4(CNC(=O)C(C)CF)C3)=O)cc2n1 7278,NS(=O)(=O)c1cc(C(=O)NCC2CCC(NC(=O)Cc3ccco3)C2)co1 7279,C1(C2(O)CCN(C(C3COCCN3C)=O)CC2)(NC(C(C)SC)=O)CC1 7280,C=CC1(CC(=O)NCCC(C)NC(=O)C(O)Cc2ccccc2)CCCCC1 7281,CC(C)(C)C(CC(=O)N1CC(NC(c2ccc3c(c2)nnn3C)=O)C1)C(F)F 7282,c1(C(N(C2CN(C(=O)Cc3csnn3)CC2F)C)=O)cc2cncn2c(O)n1 7283,Nc1cc(C(=O)NC2CC(C(=O)O)C(C(=O)O)C2)sc1C(=O)O 7284,N(C(=NCCN1CCOCC1)NCC1CN(C2CC2)C(=O)O1)C(C#C)C 7285,C1(C(NOCC#C)=O)(COC)C=CCN1C(=O)C(C)C1CC1 7286,C(C(C)(C)C(=O)NCC1(F)CCC(NC(C2(C)CC2)=O)C1)N(C)C 7287,CC1(C2(C(=O)NCc3cc[nH]c3C(N3CCC(O)(CC4CC4)C3)=O)CC2)CC1 7288,C1(NC(C2(C#N)CC2)=O)(CF)CCN(C(=O)Cc2ccccn2)C1 7289,C#CCC(C)(C)C(=O)NCCOC1CCN(C(=O)CC2CCOC(CC)C2)C1 7290,S(=O)(=O)(c1cc(C(F)(F)F)ccn1)NC(CN(c1ccccc1)C)=O 7291,Cc1cccc2[nH]cc(C(N3CCC(C)(CNC(C45CSCC4C5)=O)CC3)=O)c12 7292,N1(C(C2CC(C)N2C(c2ccn(C)n2)=O)=O)CCc2cnccc2C1 7293,C1(C(C)NC(=O)COC2CC2)CCCN(C(C2(c3cccnc3)CCCC2)=O)C1 7294,C1(C(N(CCCCO)CC)=O)CCC(C)N1Cc1ccc(C(=O)OC)cc1 7295,C(=O)(C(=O)N=c1[nH]occ1-c1ccc(F)cc1Cl)N(C)CC1COC(C)(C)O1 7296,c1(C(N(CC(C)(C)NC(C2C(C)C2)=O)C)=O)cnn(-c2nccs2)c1 7297,C(=O)(CS(=O)CCC(F)(F)F)NCC1(NC(c2cc(C#N)[nH]c2)=O)CCCC1 7298,c1(C(N2CCC3(NC(C(C(=O)OCC)CC)=O)C(C2)C3)=O)cn2cccnc2n1 7299,c1(CNC(CCN(CC#C)C(C2CC2(Cl)Cl)=O)=O)ccc(NC)nc1 7300,S(=O)(=O)(c1cnc(NC(c2nccnc2C)C)c(Cl)c1)NCC=CCCC 7301,N1(C(CN(CC(C)C)C(c2cnn[nH]2)=O)=O)CC(C)C(F)(F)C1 7302,C(=O)(C(C)C(F)(F)F)NCCCCCNC(C(c1cccc(C)c1)F)=O 7303,C1(NC(C(c2cccnc2)OC)=O)COC2(C1)CN(C(c1csnn1)=O)C2 7304,n1(CC#C)c(C(=O)NCCNC(c2cc([N+](=O)[O-])c[nH]2)=O)cc2ccccc12 7305,Cc1ccc(C)c(CN(C)C(C2CCCN2C(=O)C(O)CC(C)C)=O)c1 7306,Cc1cc(C)c(C(=O)NC(C2CCCC2)CNC(=O)CC2CCC(C)C2)c(C)c1 7307,Cc1cccc(Br)c1S(=O)(=O)NC(Cc1ccccc1)C(=O)O 7308,C1(C(=O)NC2(C)CN(C(CCN(C)CC)=O)C2)CCc2ncnn2C1 7309,N1(C(CSCC)=O)CCN(C(=O)CC2C(=O)NN=C2C)C(CS(C)(=O)=O)C1 7310,O=S(=O)(c1ccc(NC2C=CCCCC2)c(Cl)c1)NCC(CC1CC1)CO 7311,C1(CNC(CCN(C(C)=O)C)=O)CN(C(c2coc(Cl)n2)=O)C2CCN1C2 7312,Cc1cc(NC(=O)C(C2CCN(C(=O)CC3CCCC3O)C2)C)cc(O)c1 7313,C(=O)(C(O)CC(F)(F)F)N1C(C(N2CCCC(CC=CC)C2)=O)CC(F)C1 7314,N1(C(c2c(C)nc(Br)o2)=O)CCN(C(C2(C)CCOC2)=O)C2(CC2)C1 7315,N1(C(C2N(C)CCCC2)=O)CCN(C(c2cccnc2F)=O)CC1C(F)(F)F 7316,C12(NC(c3nnnn3CCOCc3ccccc3)C3(C)CSC3)CC1CS(=O)(=O)C2 7317,C1(=CCNC(c2ncsc2C2CC2)=O)CCN(C(C2C(CC)(COC)C2)=O)CC1 7318,C=CC(C)(CC)C(=O)NC(c1ccccc1F)CNC(=O)C=Cc1cnc[nH]1 7319,c1(C(=O)NCC(C(C)(C)C)NC(CN(C)CCO)=O)ncc(Cl)cc1Cl 7320,c1(C(=O)NC2COCC2C(N2CC3CC2C3)=O)ccc2cc[nH]c2c1 7321,N1(C(C(C)(C)OC(C)=O)=O)CC(CNC(=O)CN(C)C2CC2)C(C)(C)C1 7322,C(C)(C(F)(F)C(F)(F)F)NC(CCCCOC(C)(C)C)=O 7323,CC1CCC(C)N(C(C2CN(C(=O)CNc3ncccn3)CCO2)=O)C1 7324,C12(NC(=O)OC(C)(C)C)CCCN(Cc3c[nH]c(-c4ccccc4)c3)CC1C2 7325,Cc1cc(N)c(C(N2CC3=C(C2)CN(C(C2(C)CC(F)(F)C2)=O)C3)=O)cc1C 7326,C1(=CCNC(C(C)(C)OCC(F)(F)F)=O)CCN(C(=O)C=CC(F)(F)F)CC1 7327,N1(C(C2(OC)CCOCC2)=O)CCCC(C)(NC(=O)Cc2csc(C3CC3)n2)C1 7328,C1(C(=O)NC(C(=O)NCCNC(C(C)(C)C)=O)CC2CCCC2)CC12CCCC2 7329,N1(C(c2cc(OC)n(C)n2)=O)CC2(COC(CNC(c3ccc(SC)o3)=O)C2)C1 7330,Cc1nccn1C(C)C(=O)NC1CC(CCNC(c2cnc(C3CC3)o2)=O)C1 7331,N1(C(C(CC)NC(c2ccco2)=O)=O)CCC(CNC(=O)C(C)OC)C(C)C1 7332,C(=O)(C1=Cc2ccccc2C1)NCC1C(C)CN(C(=O)CCP(C)(C)=O)C1 7333,O=C1CCC(CC(N2CCCC(CCNC(c3cc(=O)cc[nH]3)=O)C2)=O)CN1 7334,c1(C(C)NC(=O)CC2C=CC(NC(C3CC34CCC4)=O)C2)nccc(O)n1 7335,C1(NC(c2cnccn2)=O)CCN(C(c2c(F)cccc2I)=O)CC1F 7336,Cn1cc(S(N)(=O)=O)c(CNC(C2(c3nncs3)CC2)=O)n1 7337,C1(C(N2CC(O)(C(C)NC(=O)Cc3cncc(O)c3)C2)=O)CC2(CCCO2)C1 7338,C(=O)(C1CCCn2cnnc21)NCC1(CN(C)C(c2cn(CCO)nn2)=O)CC1 7339,CC1(C)CCC(C(=O)NC2CCC(NC(=O)C=CC=C(Cl)Cl)CC2)CO1 7340,C(CC#CC)(C(=O)NC1CCCSC1)NC(CC1CC(=C)C1)=O 7341,c1(C(N(CC(C)NC(C2(NC(N)=O)CC2)=O)CC)=O)ccc2c(c1)CCS2(=O)=O 7342,c1(N(c2ccn(C3CNC3)n2)C(c2scc(C)c2)=O)ncnc2c1c(Br)cn2C 7343,N1(C(C2CC(C)OC2=O)=O)C2CCCC1CN(C(=O)C=CC1CCC1)C2 7344,c1(CC)cc(C(=O)N(C(C)CNC(=O)CCCC2CCCO2)CC)ccc1F 7345,O=S(=O)(c1ccc(NC2CCCC2CO)cc1Cl)N1CCC(C2CCCCC2)C1 7346,C(=O)(C1=C(Cl)CCOC1)NCC(CC)(C)NC(c1cccc2sncc12)=O 7347,c1(OC)ccc2c(c1)NCCN(Cc1ccccc1OC1CC1)C2 7348,N(C1CCCc2cc(F)cc(F)c21)Cc1cncc(O)c1 7349,CC1(C)C2CC(C(=O)NCC#CCNC(C3(F)CCCOC3)=O)CC12 7350,C1(C(=O)NCC23CC(NC(CCCOC)=O)(C2)C3)CCC(OCCCOC)CC1 7351,N1(C(C2C(CNC(Cn3c(=N)nc[nH]3)=O)CC2)=O)CC2CCCC2C12CC2 7352,N1(C(C(CC)OC)=O)CCN(C(C2(C#N)CC2(C)C)=O)CC1C 7353,c1(C(=O)NCC2CCN(C(C34COC(CCO3)C4)=O)CC2)cccc2occc12 7354,C1(C(=O)NCC2C(NC(c3n(C=C)nnc3)=O)CCC2)SC2C=CC1CC2 7355,Cc1ccc2ncc(C#N)c(N3CCN(C4CC4)C(C)C3)c2c1 7356,CCS(=O)c1ccccc1C(=O)NC1CN(C(c2cncnc2)=O)CC1C1CC1 7357,C1(C(C)C)CN(C(=O)CO[Si](C)(C)C)CCN1C(=O)CC1CCC1 7358,CCCCC(C)CCC(=O)NOCC(N1CC2(CCCO2)C1)=O 7359,c1(C(=O)NCCC(C)NC(C(CC)CC2CCCC2)=O)cc(OC)cc(C)c1 7360,N1(C(C(C)OCC(F)(F)F)=O)CCC(NC(=O)CCCC(N)=O)C(O)C1 7361,c1(C(C)NC(=O)NC2(c3ccccc3)CC2C(F)(F)F)cnc2ccccn12 7362,C=CC(C)(C)CC(=O)N1CCCC1C1CCCN(C(=O)CCN(CC)CC)C1 7363,c1(CCN(C)C)c[nH]cc1C(N1CCCC1C1(C(=O)N)N=N1)=O.C(F)(F)F 7364,CC1CC2CN(C(=O)CC#N)CC2N1C(c1cc(C(C)(C)C)on1)=O 7365,N1(C(C(c2ccccc2)OC)=O)CC2CN(C(c3ccc(C#N)cn3)=O)CC2C1 7366,N1(C(C(=O)NCC(F)(F)C2CCC2)=O)CCN2C(=O)OCCC2C1 7367,S(=O)(=O)(c1ccc2[nH]c(=NCC3CCN(C)C3)ccc2c1)NC1(COC)CCC1 7368,C1(C(N)=O)(CNC(C2C(CNC(C(N3CCOC3=O)C)=O)COC2)=O)CCCC1 7369,C(=O)(C1CCCc2cc(O)ccc21)N1C(C)(CNC(CNC(=O)NC)=O)CCC1 7370,C(=O)(N=c1[nH]n(C)c2ncc(I)cc12)C1N(C(C(CC(C)C)O)=O)C2C(C1)C2 7371,N1(C(COCCOCC#C)=O)CCCC(C)C1CCNC(=O)Cn1ccnc1C 7372,c1(C(C(N2CC(OC)C(NC(=O)COCCOC)C2)=O)C)cc(C)ccc1F 7373,C1(CNC(C2CCC(n3cc(CN4CC5CC5C4)nn3)C2)=O)C2CC3C(C2=O)C13 7374,CC(C(O)C(=O)NC1C=CCC1)c1ccccc1F 7375,CCCCCCC(=O)NC(Cc1cn[nH]c1)C(=O)N(C)CCC1CCCO1 7376,c1(CC(=O)NC2C(NC(C(c3cscn3)OCC)=O)C2)ccnc(C(F)(F)F)c1 7377,C(=O)(C(C)(F)C(C)(C)F)NC1C(CNC(C(CC)(F)F)=O)CC1 7378,c1(C(N2CC(NC(C(C)=CC)=O)C(F)C2)=O)cc(=O)n2ccccc2n1 7379,C1(CNC(c2c(CC)con2)=O)CN(C(c2ccc(Cl)cn2)=O)CC12CCC2 7380,C1(C(C)(C)C)CCN(C(c2ccncc2)=O)C1.C12(C)CCN1C(=O)C2 7381,N1(C(CN(CCOC)C)=O)CC2CC(NC(c3c(C)nn(C)c3Cl)=O)C(C2)C1 7382,N1(c2cc(C)cc(C)c2)C(=S)NC(c2cccc(Br)c2)C2=C1C(C)CN(C)C2=O 7383,Cn1ccnc1C(F)(F)C(=O)NCCN(C(C1CC(C(F)(F)F)C1)=O)CC1CC1 7384,N1(C(C=CC(C)C)=O)CC(C)(C)CCC1CNC(C1CC(=C(F)F)C1)=O 7385,C(=O)(C1=CCCN(CCCc2cc(O)c(O)cc2O)C1)N1C(C)CCC(O)C1 7386,C1(NC(C2(C)CC(F)(F)C2)=O)CCN(C(=O)CSC2CC2)C(C2CC2)C1 7387,c1(C(=O)NCC2(C(NOCCCC=C)=O)CC(=C)C2)ccc2cc[nH]c2n1 7388,N1(C(c2nc(=O)cc(N)[nH]2)=O)CCC2(CC1)CN(C(=O)CCc1cc(Cl)cs1)C2 7389,C1(CCNC(c2nocc2Cl)=O)CCCCN1C(c1ccsc1-n1cnnn1)=O 7390,C12(C(N(C(C)C(C)(C)O)C)=O)CC(CO1)N(C(C1CC3CCCC3C1)=O)C2 7391,C(CCCC(CO)NC(=O)CCc1cn(C)cn1)NC(C1OCCC(C)C1)=O 7392,C1(C(=O)NCCCC(=O)NC2CC2)CC2CC2N1C(=O)CC1NC(=O)NC1=O 7393,C1(N(C(C(C2(O)CN(C(COCCCC#C)=O)C2)F)=O)CC)CC=C(C)CC1 7394,N1(C(C(CC#C)(C)NC(c2ccn(C)c(=O)c2)=O)=O)CCC2(COC(=O)N2)C1 7395,C(C(F)C(=O)NC(CSC)C1CC1)N(C(C1(CC2CCC2)CC1)=O)CC 7396,N1(C(C=CC)=O)CCCC1(CNC(C1CN(CC)C(=O)N1)=O)COC 7397,CC1(C)CC(CC(N2CCCC2(C)CNC(c2coc(Cl)n2)=O)=O)CO1 7398,O=C(C1CCc2c[nH]nc21)NC1CC(CC(=O)NCCN2C(=O)C(=O)NC2=O)C1 7399,C(=O)(CC(CC)C(F)F)N1CCC(=CCNC(C(CC)C)=O)CC1 7400,c1(C(N2CCN(C(C3CC(CC)OCC3)=O)CC2C)=O)ccc2c(c1)CCCS2 7401,Cc1ccc(OCCCC(=O)NCc2nc(C)c(-c3ccc(Cl)cc3)o2)c(C)c1 7402,N1(C(c2c(C)cccc2O)=O)C2CCC1CN(C(c1cn3c(n1)SCC3)=O)C2 7403,Cc1c(-n2cc(C3CCN(C(=O)CC(C)C4CC4)C3)nn2)cccc1F 7404,c1(OCC(N)=O)cccc(C(=O)NC2CCC(NC(=O)CSC3CC3)C2)c1 7405,C1(C(=O)NC(CCC)CCCNC(C2(CF)CCC2)=O)CCc2nc(C)cn2C1 7406,Cc1ccc(N)cc1C(N1CCCC(F)(CNC(=O)CNC(=O)CC(C)C)C1)=O 7407,CCC(CC(C)C)C(=O)NC1(C)CC(C(=O)NC(C2CCCCC2)CO)C1 7408,CC1COc2ccccc2C1C(=O)N1CC2(C1)CN(C(c1cccc(O)n1)=O)C2 7409,C1(NC(CC(C)c2ccncc2)=O)(CO)CCN(C(C2(CF)CCC2)=O)C1 7410,C(=O)(C(F)C(=O)N1CCC(NC(=O)CC=C(C)C)C1C(C)(C)C)OCC 7411,c1(NC(=O)CCCCBr)ccc(CNCc2ccc(F)nc2F)cc1F 7412,c1(NC(=O)N(C2CC2c2ccc(Cl)cc2)C2COC2)ccccc1Cl 7413,C(=O)(CCC(F)(F)F)NC1C(C)CN(C(=O)CCc2nnc(S)n2C)C1 7414,C(C(=O)NCCc1cnc(C)[nH]1)(C(C)CC)NC(c1cccc(CC)n1)=O 7415,n1(CC(N2CC(NC(C(C)CC(F)(F)F)=O)C(F)C2)=O)nc2n(c1=O)CCOC2 7416,C(=O)(C1CCCc2nc[nH]c21)N(CC(C)N(C(c1nc(OC)c(F)cn1)=O)C)C 7417,C1(C2CCCN(C(c3scnc3C(C)C)=O)C2)(NC(C(CSC)OC)=O)CC1 7418,Cc1cc(C(=O)NCC(O)CNC(C2(S(N)(=O)=O)CCCC2)=O)ccc1[N+](=O)[O-] 7419,C1(C(N(CC(C)O)CCNC(C)=O)=O)CC(O)C(O)CC1C(=O)OC(C)(C)C 7420,N1(C(Cn2nnc(=N)[nH]2)=O)CC2(COC(CNC(C3CC(C4CCC4)C3)=O)C2)C1 7421,C(CCC(C(=O)N1CCCC(C)C1)NC(c1ccc(C2CC2)cc1)=O)OC 7422,c1(C(N2CCC(OC)(CNC(c3cncc(Cl)c3)=O)C2)=O)cnnc(C)c1C 7423,C(=O)(CCCCC(C)CC)NCC(CN(C(C1CC(CCC)OCC1)=O)C)C 7424,C1(CCC)CN(C(c2oc(C)cc2C)=O)CC1NC(C1(CO)CCOCC1)=O 7425,N1(C(C(C(CC)C)NC(=O)CCS(N)(=O)=O)=O)CC2OCCOC2C1 7426,c1(C(=O)NC2C(CNC(C=COCC)=O)COC2)ccc(F)cc1Cl 7427,CC1CN(C(c2cn(CC3CCCO3)nn2)=O)CCN1C(C1CC1CF)=O 7428,C(=O)(CC(C)C(=O)NCC1(CNC(c2ncc(Br)cn2)=O)CCCC1)OC 7429,CC1CN(C(C2CCCNS2(=O)=O)=O)CC(C)C1N=c1nc[nH]n2c(Br)ccc12 7430,c1(C(=O)NCCC(CNC(=O)C(C)CC(N)=O)OC)c(C)nc(O)nc1C 7431,C1(C)(NC(CC(CC)C2CCC2)=O)CCC(NC(=O)CCCC(OC)OC)CC1 7432,Cc1ccccc1CC(C)C(=O)NCC1CCCN1C(=O)CCc1ccccn1 7433,C(=O)(CCP(C)(C)=O)N1CCC(NC(Cc2n[nH]c(=NC)s2)=O)(CO)C1 7434,C1(CNC(C2C(C)CCC2)=O)CCC2(CCN(C(=O)C#CC(C)(C)C)CC2)CO1 7435,C1(CNC(CC#N)=O)CC2(CC(NC(c3ccccc3C(F)(F)F)=O)C2)C1 7436,Cc1nn(C)c(=O)c(C(=O)NCCC2(NC(C3CCCS3(=O)=O)=O)CCC2)c1C 7437,n1(CC)nnnc1C(c1cc(C2CC2)no1)NC1CCCC1COC(C)(C)C 7438,N1(C(c2ccc(OC)cc2)=O)CCOC2(C1)CN(S(=O)(=O)CC1CCC1)C2 7439,N1(C(CCCNC(C(CCC)OC)=O)=O)CCOCCC1C 7440,N1(C(CC=CC)=O)C2CCC1CN(C(C1(CO)CCC(C)C1)=O)C2 7441,c1(C(=O)NC2CN(C(C(C)n3ccnn3)=O)C(C)(C)C2)cc(F)c(F)cc1F 7442,CCC(O)C(F)(F)C(=O)NCC1CC(F)(CNC(C2(CCOC)CC2)=O)C1 7443,C1(C(=O)NC2CCCN(C(c3cncc(CC)c3)=O)CC2)CC(C2CCCC2)C1 7444,c1(C2(C(NCCCC3CC3)=O)CCC2)ccccc1C.c1(C(=O)OC)cnc(C)cn1 7445,C(=O)(N1Cc2ccccc2CO1)C1(NC(c2cc(C(C)C)on2)=O)CC1(C)C 7446,c1(C(=O)NCC2N(C(COC(CC)C)=O)CC(O)C2)cc(F)cc(F)c1 7447,C1(NC(C=CC=CCC)=O)CN(C(=O)C=C(C)C(F)F)Cc2ccnn2C1 7448,C1(N(C(C2C(CNC(C(c3ccc(C)o3)C)=O)C2)=O)C)CCOCC1C 7449,CCC(CNC(=O)CCCC1CCCO1)(CC)C(=O)NC1(C)CCC(C)(C)C1 7450,N1C(=NCC2CC2)N2CCCC(C2)C1.CC1CN(C2CCNCC2)CC(C)O1 7451,C1(C(=O)NCC(CC)NC(C2CCC3CC23)=O)(Cc2cnn[nH]2)CC(F)(F)C1 7452,C1(N(C(C(CC)CC)=O)C)CCN(C(c2cnc(-n3cccn3)cn2)=O)CC1C 7453,N1(C(CC=C(C)C)=O)CCCC(F)(CNC(c2coc(-c3cnn(C)c3)n2)=O)C1 7454,C1(CCC)(NC(=O)CC2CCCS(=O)(=O)C2)CCCN(C(=O)C2=COCCO2)C1 7455,N1(C(C2CC(CNC(=O)OC(C)(C)C)CCO2)=O)CCCCC(CO)C1 7456,C12(C(N)=O)C3C4C1C1C2C3C41C(=O)NC1CC2(C1)CN(C(c1cnn[nH]1)=O)C2 7457,c1(CC(=O)NCC2(C(N)=O)CN(C(CCCC=C)=O)C2)cc(O)nnc1O 7458,C1(NC(C2(NC(c3ncccn3)=O)CCN(C)C2)=O)CC2(CCCO2)C1 7459,n1(C2CCN(C(C(CC)(F)F)=O)CC2)ncc2c1CN(C(c1cnc(C)o1)=O)C2 7460,N1(C(C(C)(C)CC#N)=O)CCC2(C(N3CCC3CN=[N+]=[N-])=O)CCCC12 7461,C(C(C(=O)N1CC2CC(C1)N2C(=O)CCC(C)(C)N(C)C)C(F)(F)F)OC 7462,c1(C2(NNC(c3cc(C(C)(C)C)oc3C)C)C(=O)N2)cc2c(s1)CCCC2.C(C)(C)(C)C(=O)C(C)=O.C 7463,C12(NC(c3ccn(C4CC4)n3)=O)CCC(CC1NC(C1(n3cncn3)CC1)=O)C2 7464,CC1(C)CCC(CC(=O)NCCC(O)CNC(=O)CN2C(=O)CNC2=O)CC1 7465,c1(C(N(C(C)C)CCNC(c2cccs2)=O)=O)cnc2n1CCC2 7466,C#Cc1ccc(NC(C2CCC(CN(C(=O)CCOC(C)=O)C)CC2)=O)cc1 7467,N(C1CCCc2n[nH]cc21)C(=O)CC1CC(C(N(C)Cc2cncn2C)=O)C1 7468,C1(F)(C(=O)NC(CC(C)NC(C(CC)(C)C#N)=O)C)CCC(F)(F)CC1 7469,C(=O)(C(C)CCC(C)(C)C)NCC(C)CNC(C1(c2cccnc2)CC1)=O 7470,c1(C(N(CCC(C)NC(=O)C(C)N2CCC2)C)=O)cccnc1 7471,c1(OCC)ncc(OCC2CCN(C(=O)Nc3ccc(CC)cc3)C2)cn1 7472,CCC1=NOC(C(N2CCOCC2C(=O)NC(C)Cc2nc[nH]n2)=O)C1 7473,c1(C(c2n(CCCC)nnn2)NCC2(CO)COC2)ccc(F)cc1I 7474,CC1CCC(C(=O)N(C2CC3CC3C2)C)N(C(=O)Cc2ccon2)C1 7475,N1(C(C(C=C)OC)=O)CCCc2c1ccc1nc(C)[nH]c21 7476,C1(F)(C(N(C)Cc2cnco2)=O)CN(C(=O)CC2CC(F)(F)C2)C1 7477,CC1(C)CN(C(c2coc(C3CC3)n2)=O)CCC1NC(=O)CCCNC(=O)C1CC1 7478,C1(C(N(CCNC(c2c(C)n(C)nc2)=O)C)=O)CCCCC(C)(C)C1 7479,c1(CC)cccnc1C(=O)NC(C)(CNC(=O)CCC1C(=O)NN=C1C)C1CC1 7480,N1(C(c2cc(CNC(C3CC(C)C3)=O)oc2)=O)CC2CCCC2C1 7481,CP(C)(=O)C1(C(N2CC(O)(C3CCCN3C(=O)CC3CC3)C2)=O)CC1 7482,CC(C)(C)CC(F)C(=O)N1CCC(F)(c2cn(CC3CC4CC4C3)nn2)C1 7483,c1(OC(C)C(=O)NCC2CC(C)N(C(=O)CC(O)C3CC3)C2)ccc(F)nc1 7484,CC1(C)CCC(C(=O)NC2CC(C(F)C(=O)NCCNC(=O)C3CC3)C2)C1 7485,N1(c2nnc(COC)s2)CC2CC1CCC2NC(C1(O)CCSCC1)=O 7486,C1(C(N2C(CNC(C(CSC)C)=O)CCC2)=O)(NC(=O)OC(C)(C)C)CCCCC1 7487,C12(NC(C3C(CC)C3(F)F)=O)COC(C1)C(NC(c1cnn(C)n1)=O)C2 7488,c1(C(C)(C)CN2CCCC2)cnc2nc(C#N)ccn12.c12conc1CS(=O)C2 7489,CC1CN(C(c2cn(C3CC3)nn2)=O)CC1(C)CNC(=O)CCNC1COC1 7490,N1(C(C2CC(OCC)C2)=O)CCCC(C)(CNC(c2[nH]c(C3CC3)nc2C)=O)C1 7491,c1(C(N2CC(C(C)OC(C(=O)OC)OCC)C2)=O)ccc(C(=O)CC)cc1 7492,Cc1n[nH]c(C)c1C(=O)N(C)CC1(O)CN(C(=O)C(C)(C)C2CCOC2)C1 7493,CCC(C)(C)CN(C)C(=O)N(c1cccnn1)CCOC(F)(F)F 7494,C1(NCCCCCC(C)(C)N)CCc2ncccc2C1 7495,C(=O)(C1=CC2CCCC12)N(CC(CNC(c1cccc(SC)n1)=O)C)C 7496,Cc1nc(C(=O)NC2CCCC2NC(c2cccn2C)=O)c2ccccn12 7497,CC1C2C(CCN2C(C2CCC3CC23)=O)CN1C(C1CC(=O)CCO1)=O 7498,Cc1cc(C(=O)NCC(O)CN(C)C(C2OCC3CCCC23)=O)ccc1Cl 7499,N1(C(COc2cc(C)on2)=O)CCCC(CCNC(=O)Cc2ncn(C)c2C)C1 7500,CC(C)C(C)(O)CNC(=O)CNC(=O)CNC(c1nc(Cl)cs1)=O 7501,c1(C(N2CC(NC(c3nn(CC)c(C)c3)=O)C(C)(C)C2)=O)c(C)cc(O)cc1C 7502,CCC(CC)C(C(=O)NCc1occc1C(=O)NCC1(CO)CC2CC2C1)OC 7503,c1(C(C)C)[nH]nc(C(=O)NC(CNC(=O)CCC2CCCO2)CO)c1[N+](=O)[O-] 7504,C1(CCC(=O)NCC(C)=CC(=O)NCc2cccc(Cl)c2)CCCN(C)C1 7505,c1(OCCC)cc(F)ccc1NC(C1C2CC3C(C1)C2C3)=O 7506,C12(CNC(C(C=C)OC)=O)CN(C(c3c[nH]nc3CC)=O)CC1CCO2 7507,N1(C(C2CCC3CCCCN23)=O)CCCCC1C1CCCN1Cc1cncs1 7508,C1(CNC(=O)C(O)C2CN(C(=O)COC3CCC3)C2)CCC(O)C1 7509,c1(C(N(CCC(C)NC(=O)Cc2cnn(C)c2)C)=O)ccc2nccnc2c1 7510,c1(C(N2CC3C(NC(CN(C)CC)=O)C(CC3)C2)=O)cc2c(cn1)OCCC2 7511,CC1=C(C(=O)NC2CN(C(c3ccc(C)nc3)=O)CCC2C(F)(F)F)CCO1 7512,C(=O)(C1CCc2c[nH]nc21)N1CC(C)(NC(CC(C(=O)OC)(C)C)=O)C1 7513,C#CC1(C(=O)Nc2cnc(C3CC3)nc2)CCN(C(=O)CC=C(C)C)C1 7514,C1(C(=O)NC(c2n(CC)ccn2)C)COCCN(C(=O)CCc2ccnn2C)C1 7515,N1(C(c2c(CC)onc2)=O)CCOCC(NC(c2cc(C(C)C)ccc2N)=O)C1 7516,c1(CC)c(C(=O)N(C)CC2CN(C(=O)C=CC(=O)NC3CC3)CCO2)cnn1C 7517,C(=O)(CCCn1ccnc1)NCCCOCCC(=O)NC(c1cncnc1)C 7518,N1(C(CNS(CC)(=O)=O)=O)CCC(C2CC2NC(C2CC=CCC2)=O)CC1 7519,C1(CNC(CC(=C)C)=O)CN(C(=O)CCc2ccco2)C2CC12 7520,C12(C(=O)NC(CNC(c3ccc(N)c(Cl)n3)=O)CO)CCCCC(=O)N1CCC2 7521,CCC(C)(CCNC(=O)CC1CC=CCN1C)NC(=O)CSC 7522,Cc1ccccc1C1(C(=O)NCC=CCNC(=O)C(F)n2ccnc2)CCC1 7523,N1(C(COCc2ccc(C)cc2)=O)CCC2CC(NC(=O)C=CCF)CCC2C1 7524,N1(C(c2c(Cl)sc(C)c2C)=O)CCC2(CC1)COC(CNC(c1cn[nH]c1)=O)C2 7525,C(CNC(C1CC12CCCC2)=O)(CC(=O)N1CCOC(C)C1)OC 7526,C1(C(=O)NCC2(C#C)CCCC2)CCC(O)CN1C(C1CC(OC)(OC)C1)=O 7527,N1(C(C(=O)N(C(C)C)CCNc2ccc(-n3ccnc3)nn2)C)C(C)CCC1C 7528,C1(CNC(CCC=CC)=O)C2CN(C(c3nocc3C(C)(C)C)=O)CC12 7529,N1(C(CS(CC)=O)=O)CC2(CCN(C(c3ncc(C(F)(F)F)cc3Cl)=O)CC2)C1 7530,C1(C(=O)NCC(C(=O)OC)OC)CCN(C(=O)CCOCC(F)F)C(C(C)C)C1 7531,c1(C(CC)=O)cc(C(=O)N(C2CC(NC(c3ncc(F)cn3)=O)C2)C)ccc1F 7532,N1(C(C(C2CCCN(C(C(CC)(C)C)=O)C2)C)=O)CCC12CCCSC2 7533,Cc1cc(Cl)ccc1NC(=O)CN1CCN(CCC(C)(C)C)CC1 7534,CCCC(C)(CCC)C(=O)OC1CN(Cc2ccccc2)CC(F)(F)C1 7535,C1(CCCC)CCCCC1C(=O)NC1CN(C(=O)CCC(=O)OC(C)(C)C)C1 7536,C1(NC(c2c(SC)csc2)=O)CC2(C1)CC(NC(c1coc(C3CC3)n1)=O)C2 7537,O=C(CC1=CCCCC1)N1CC2CCCC1C2c1cn(Cc2cccs2)nn1 7538,Cc1ccc(C(=O)NC2CC(CCO)C2)cc1-c1cn(CC2CCC(=O)O2)nn1 7539,C(CC1CCC1)(C(=O)NC(C1CCCC1)CNC(c1coc(C)n1)=O)OC 7540,c1(OC)c(C(=O)NC2CC(O)CN(C(C3CCN(C)CC3)=O)C2)cc(F)cc1F 7541,c1(C(N(CCC)CCNC(=O)C2=CC(C)(C)C2)=O)c[nH]c2cc(C#N)ccc12 7542,C(=O)(CC(F)(F)C(F)F)NC1(CCCNC(c2cc(C)no2)=O)CC1 7543,C(=O)(C(CC(C)C)N(C)C)N1C(CCC(=O)N(CCCF)CC)CCCC1 7544,N1(C(c2n(C(C)C)ncc2)=O)CC2CCCC2(NC(=O)C(=O)NCC(F)(F)F)C1 7545,N1(C(c2cc(CCC)[nH]n2)=O)CCCN(C(C23CSCC2C3)=O)CC1C 7546,C1(N(C(Cc2nnc(C)s2)=O)Cc2ccccc2)CCCN(C(C2CC2F)=O)C1 7547,N1(C(c2c(C)oc(C(C)C)c2)=O)CCN(C(=O)CC2(C)CCCO2)C(C(C)C)C1 7548,C1(C(=O)NCC(C(C)C)NC(=O)CC(C)(C)N(C)C)CCCC(F)C1 7549,c1(C(=O)NC2CN(C(C(CC)F)=O)C3(C2)CCC3)ccc2c(c1O)CCC2 7550,N1(C(C2(CC(C)=O)CC2)=O)CCC(C(=O)NCc2nnc(O)o2)=C(F)C1 7551,C12(C(=O)NCC3(NC(=O)C4=CSCCO4)CCC3)CCCC1CS(=O)(=O)C2 7552,C1(CCNC(CN2CC(C)C2)=O)CCCN1C(c1cc(-c2ccccc2)[nH]n1)=O 7553,C1(CNCc2ncn(C(C)C)n2)CCC2(CCC2)CO1 7554,N1(C(CC(COC)C)=O)CC(C)OC2(CCN(C(C3(CO)CCCCC3)=O)C2)C1 7555,c1(C(=O)NC2C3(CN(C(C(C(C)C)F)=O)C3)CC2)cnc(O)n(C2CC2)c1=O 7556,C(CC(C(C)(C)C)NC(=O)CC1CC=CCC1)N(C)C(c1sccc1C1CC1)=O 7557,Cc1ccc(Cl)cc1C(N1CC(C)C(C)(CNC(=O)CC2CC23CC3)C1)=O 7558,C1(C(N(CC(C)N(C(C)=O)C)C)=O)CCN(C(=O)C(C)Cn2ccnc2)C1 7559,N1(C(CC(C)(C)c2cn(C3CCC(OC)CC3)nn2)=O)CC2C(C1)C2(F)F 7560,C1(NC(c2cc(C(=O)OC)ncc2)=O)CN(C(C2CC(C)=NO2)=O)CC(C)(C)C1 7561,c1(C(C)Sc2n(CC)c(CCc3ccco3)nn2)ccc(Cl)cc1F 7562,N1(C(c2c(OCCC)cccn2)=O)CC(NC(C2CC2CC)=O)CC2(CCC2)C1 7563,c1(SC(C)C(=O)Nc2cnc(NC(=O)C=CC3CC3)s2)ccc([N+](=O)[O-])cc1 7564,N1(C(C(C2CC2)OCC)=O)CCCC(C)(C)C1C(=O)NC1CC(CC(N)=O)C1 7565,N1(C(C(n2cc(Cn3c(C)ccc3C)nn2)C)=O)CCOC(C2CC2)CC1 7566,C(=O)(C(C)(C)S(C)(=O)=O)N1CC(CC(C)NC(c2ccc(S(C)=O)cc2)=O)C1 7567,C(C(=O)NCC1CC(NC(C2CCN2C(C)=O)=O)C1)(C(C)C)NC(=O)OCC 7568,N1(C(C(C(C)C)OCC)=O)CCC2(CCC(NC(=O)C3=CCC3)CC2)CC1 7569,CCC(C(=O)NC1CC(C(=O)Nc2ccc(CO)c(F)c2)=CC1O)C(F)(F)F 7570,Cc1nn(C)c(NC2CC(C)CC(C)C2)c1C#N 7571,N1(C(c2ccc(COC)o2)=O)CC(CC(=O)NCCN(C)C(C)C)CC1(C)C 7572,N1(C(c2ccc(Cl)s2)=O)CCN(C(=O)C=CC2CCCO2)C(CF)C1 7573,CCC(C)(CN(C)N1CC(O)CC1CO)Oc1ccccc1 7574,c1(C(=O)NCC2CN(C(CS(CC)(=O)=O)=O)CC23CC3)cnc2c(C)cnn2c1 7575,C1(CC(=O)O)(NC(N2CCC(C(C(N3CCC(C)C3)=O)F)C2)=O)CCOCC1 7576,C12(NC(CN3CC(C)(C)C3)=O)CCCC1CN(C(C1(C)CCCNC1=O)=O)C2 7577,C1(NC(CCSCCC)=O)C=CC(C(=O)NC(C)Cc2cnccn2)C1 7578,C1(NC(C2(C)ON=C(C)C2)=O)CN(C(=O)CC2(O)CCCC2)CC1(C)C 7579,Cc1ccc2c(c1)C(C(=O)NCC(F)CNC(c1ncccc1CO)=O)OCC2 7580,N1(C(c2c(OC)csc2)=O)CCCC1CCNC(=O)C(C(C)C)OCC(C)C 7581,CC1CCC(NC(=O)C(O)C2CCC2)CN1C(=O)CCCC1CC1 7582,N1(C(c2ccc(SC)o2)=O)CC(NC(=O)CCc2ccc(O)nn2)C(C)(C)C1 7583,C1(C#N)(C(=O)NCCC(C)N(C)C(c2cc(-c3cccs3)on2)=O)CCSCC1 7584,N1(C(Cn2ncn(C)c2=O)=O)CCC2CC1CN(C(=O)CCC1CC1(C)C)C2 7585,C1(CNC(CCN(C(=O)C(CSC)OC)CC=C)=O)CCN(CC)C1 7586,c1(NCC)ccc(CN2CC(CCN)C(O)C2)cc1 7587,c1(N2CCN(C(=O)NC(c3c(C)noc3C)C)CC2)ccc(C#N)nc1 7588,N1(C(C2(CC)CCCC2)=O)CCN(C(=O)COCCSC)C(C2CC2)C1 7589,c1(SCC(=O)NCCC(C)N(C)C(C2COC3(CCC3)C2)=O)ccsc1[N+](=O)[O-] 7590,S(=O)(=O)(c1cnn2ccc(=NCc3csnn3)[nH]c12)N1C(CCC)CCC1 7591,C12(C(=O)NCCNS(N)(=O)=O)CCCC1N(C(C1CCNC(=O)C1)=O)CC2 7592,N1(C(CC=C)=O)CC(NC(c2cccc(-c3cscn3)c2)=O)C2(CCC2)C1 7593,c1(C(=O)NC2CCN(C(CCC#CC)=O)CCC2CO)cc2c(Cl)ccnc2s1 7594,C1(O)(C(C(=O)N(C2CCOC2=O)C)F)CN(C(=O)C=CC(=O)NC2CC2)C1 7595,C1(C(=O)NC2C(CNC(c3ncc(C)c(C)c3)=O)CC2)CC(C)CC(C)(C)C1 7596,n1(CC)ncc2c1CCCC2NC(=O)NC(c1ccccc1)(C)C 7597,C(=O)(C(C)S(C)(=O)=O)NCC=CCNC(C1CCN(c2cc(C)ncn2)CC1)=O 7598,C1(S(C)(=O)=O)(C(=O)NC2C(CNC(c3[nH]cc(CC)c3)=O)C2)CCCC1 7599,C12(CNC(CCCSC)=O)CC(NC(=O)CC3CSCCS3)(CO1)C2 7600,CC(C)CC(C(=O)N1CCCC1C(C)C)C(N)=O 7601,N1(C(C)C)N=C(C(=O)N2CCCC(C)C2CNC(=O)COC(F)F)CCC1=O 7602,C1(CC(=O)NC2CCC(N(C(C(CC)N(C)C)=O)C)CC2)C(=O)N(C)N=C1C 7603,N(C(=NC1CCS(=O)(=O)C1)N1CCC2(CC1)CC(C1CC1)=NO2)CC(C)(C)C 7604,N1(C(c2cnc(C)nc2)=O)CC(NC(=O)C=Cc2cc[nH]c2)C2(CC2)C1 7605,N1(Cc2c(-c3c(C)c(F)ccc3)c(Cl)n(C)n2)CCCc2sc(N(C)CC)cc2C1 7606,c1(C(N2CC(COC)(CNC(=O)C(C)C3CCC3)C2)=O)cccc(CO)c1 7607,c1(CNCC2CCC(NC(c3c(C)cc(Br)cn3)=O)CC2)cc2ccncc2[nH]1 7608,CCC(C(=O)NC1CCN(C(c2cc(O)nc(O)n2)=O)C12CC2)C(F)(F)F 7609,N1(C(C(N2C(=O)CCC2=O)C)=O)CCC2CN(C(=O)CCc3ccoc3)C2C1 7610,C(=O)(C(CNC(=O)CC(O)C1CCCC1)C(C)(C)C)NCCC=CCCC 7611,C(=O)(C1=CCCN(C(=O)CC(F)(F)F)C1)N(CC(N)=O)C 7612,Cc1ccc(C(N2CCC(CN(c3ncnc(Cl)c3F)C)C2)=O)cc1C 7613,CCN=c1[nH]c(CNC(=O)N(C2CC(O)C2(C)C)CC)cs1 7614,Cc1cccc(SC2(C(=O)NC3CC(NC(C4CC4F)=O)C(O)C3)CC2)c1 7615,N1(C(c2ccnc(C)n2)=O)CC2CC(NC(c3ccc(C)c(F)n3)=O)C2C1 7616,C(=O)(C(CC)CC(F)F)NC1(CN(C(c2cc(CC)c(F)cc2)=O)C)CC1 7617,Cc1cc(C(=O)NC2CC(NC(C3(Br)CC3)=O)C2)[nH]c1C 7618,N1(c2snc(C(C)C)n2)CCC(CC(N)=O)(NC(=O)CCc2cnccn2)CC1 7619,c1(CN(C(C2C(OC)CCCC2)=O)C2CC2)c(C)cccc1[N+](=O)[O-] 7620,n1(CC(=O)NCCN(CCC)C(C2OCC2(C)C)=O)cnc(Br)n1 7621,CC1(C)CCC(OC2CN(C(=O)C(=O)OC(C)(C)C)C(C)(C)C2)OC1 7622,N1(C(C(n2cc(C)nc2)(C)C)=O)CCC2(CCC2)C(NC(C2CCCC2O)=O)C1 7623,c1(CNC(C(C)CO)=O)ncccc1CNC(=O)CSC(F)(F)F 7624,c1(C(=O)NCC(n2cc(C(C)(C)NC(C)(C)C)nn2)C)cc[nH]c(=N)n1 7625,CC1C(C)N(C(=O)COC(C)(C)C)CCN1C(C1C2CCC1(C(F)(F)F)C2)=O 7626,c1(C(N2CCCC(CCNC(c3ncn(CC)n3)=O)C2)=O)cnc2cc[nH]c2c1 7627,C1(NC(C(=O)N(C)CC2OCC(C)C2)=O)CCC=CCCC1 7628,C(=O)(C(C(C)(C)C)c1ccccc1)N1CC(NC(CCCSC)=O)C(C)C1 7629,Cc1nc(N2CC(NC(=O)CCC(C)(C)[N+](=O)[O-])C(C)C2)c(Cl)cc1C#N 7630,c1(C(=O)NCC(C)(CNC(C2C=CCCC2)=O)OC)cn(C)nc1C(C)C 7631,CC1C(NC(=O)CCc2cn[nH]c2)CCN1C(=O)CN1CCOCC1=O 7632,C(C1CCOCC1)=CC(=O)NCCC1CS(=O)(=O)C1 7633,CCCC(O)CCNC(=O)CN(C(=O)CCCOC(C)(C)C)C 7634,Cn1ccc(=O)c(C(N2CCC(O)(CNC(=O)C(F)n3ccnc3)CC2)=O)c1 7635,c1(CC(=O)NC2CN(C(c3cn(Cc4onc(C)n4)nc3)=O)C2)cccc(F)c1 7636,N1(CC(=O)N(c2nccs2)CCN2CCCC2)CCc2cccc(F)c21 7637,C1(C(C)C(=O)NCCn2cnnn2)CCCN(C(C2SCCS2)=O)C1 7638,c1(C(=O)OC)cc2c(cc1OC)CN(CCNCc1ccc(C)cc1Cl)CC2 7639,c1(OC)cc(Br)cc(CN2CCCC2(C)C(=O)Nc2cnc3cc[nH]c3c2)c1O 7640,C=C(Cl)CC(C(=O)NCC(C)(C)C1CC1)NC(C1CC(=O)OC1(C)C)=O 7641,c1(CC)noc(C(N2CCSCC2CCNC(c2cnc(C)nc2)=O)=O)c1C 7642,N1(C(C2SCCN(C(c3c(C)ccc(OC)c3)=O)C2)=O)CCC2(CC1)CC2(F)F 7643,c1(NCCCC(CO)O)cnc2c(Br)c[nH]c2n1 7644,c1(N2CCCC(C(C)NC(CCOCC)=O)C2)cc(-c2ccco2)nc(C)n1 7645,Cn1cnc(I)c1C(c1nnnn1CC(F)F)NC1(C2CCCO2)CC1 7646,C(=O)(CC(F)(F)C(F)(F)F)NC1CCCN(C(C(CCC)c2ccccc2)=O)C1C 7647,C1(NC(C(CC)C(C)O)=O)C(C)CCN(C(=O)C=C2CCN(C)C2)C1C 7648,c1(CNc2cc(CO)c(OC(F)(F)F)cc2)cc(F)c(F)cc1Br 7649,C1(C(C)(C)C)(C(N(CCN(C(=O)CC2CSCCS2)C)C)=O)CCCC1 7650,C1(NC(C(=O)NCC)=O)CCSC12CN(C(=O)C(C(C)C)NC=O)C2 7651,c1(NC(C2N(C(C3C(C(=O)OC)C3)=O)CCOC2)=O)ccc(F)c(C(N)=O)c1 7652,n1(CC(=O)OCC)nc(-c2cccc(F)c2)nc1-c1c[nH]c(=O)cn1 7653,c1(C(=O)NCC=CCNC(C2C(C=C(C)C)C2(C)C)=O)cc(N)c(Cl)c(O)c1 7654,c1(C(=O)NCC2C3CN(C(c4snc(O)c4Cl)=O)CC23)cn2cccnc2n1 7655,C(CC(=O)NCC1CC(NC(=O)C(C)n2ccnc2)C1)OCCCOC 7656,CC1(C)CCC(C(=O)NCCC2CCCN2C(c2cc(O)cs2)=O)C1 7657,c1(OC)ccc(C(=O)NCC2CC2NC(=O)C(C(C)C)OC)c(OC)n1 7658,Cc1ccc(C(N2CC3(C2)CN(C(=O)C(=O)N(C)C)CC3CO)=O)c(N=[N+]=[N-])c1 7659,c1(OC)cncc(C(=O)N(C(C)CNC(=O)CC2CCC(=O)O2)C)c1C 7660,Cc1c(C(N2CCCN(C(c3sccc3Cl)=O)CCC2)=O)nn2ccccc12 7661,CCCCCC(F)C(=O)N1CCCC(C)C1CNC(=O)C(F)CCCC 7662,c1(N(CCC)C)ccc(C(N2CC(CC(C)NC(=O)C(F)C(C)C)C2)=O)cc1 7663,C1(NC(CC(=C)C)=O)CCC2(CC1)CN(C(=O)C1=COCCO1)CCO2 7664,c1(C(=O)NC2C3CN(C(C(CCC)OC)=O)C2CC3)sc(=NCC)[nH]c1C 7665,c1(-c2nc(CC(CC)C)nn2C(C)C(F)(F)F)cc2nccnc2cc1C 7666,CC(C)CS(=O)(=O)CCC(=O)NC1COC2CN(C(C3(C)CNC(=O)C3)=O)CC12 7667,c1(C(=O)NC2(CN(C(CCC(C)OC)=O)C)CC2)ccc(Cl)c(C)c1 7668,N(C1CCCc2c(Br)cccc21)C(c1n(C(C)(C)C)nnn1)CCCC1CC1 7669,N1(C(COc2cccc(NC(C)=O)c2)=O)CCC(O)C(NC(c2cscn2)=O)C1 7670,C1(CC)CCN(C(c2ccc(=N)[nH]n2)=O)C(C(=O)NC(C)CCCO)C1 7671,CC(C)CC(O)C(C)C(=O)N(CCC(=O)NCCCC(C)CO)CC1CC1 7672,C1(NC(c2c(CCC(=O)OC)cccc2)=O)CN(C(=O)CC2CC2)CCC1(C)C 7673,C(N=c1cc(C(F)F)nc[nH]1)C1(NC(=O)CCCc2cccs2)CCOCC1 7674,N1(C(=O)Cc2ccc(Cl)s2)CCC(O)(C(N2CCC(CN3CCCC3)CC2)=O)C1 7675,C(=O)(C1CCCc2nn(C)cc21)NC(CC(C)C)CNC(=O)CSS(C)(=O)=O 7676,C1(C(=O)NC2(CCOC)CCN(C(=O)Cn3cncn3)C2)C2CCC(C2)C1(C)C 7677,N1(C(c2ccc(C#C)cc2)=O)CCCC2CN(C(=O)C(n3ccnc3C)C)CC12 7678,N1(C(C2c3cc(OC)cc(c3)CN2C2CC2)=O)C2CCC1CC(=O)NC2.CC.OC 7679,c1(N2CCC=C(C(=O)OC)C2)ncnc2c1ncn2C1CCC(CO)O1 7680,N1(C(c2c(CC)occ2C)=O)CC(NC(=O)CP(C)(C)=O)CC(O)C1 7681,C=CCCCC(C)(C)C(=O)NC1CCOCC1NC(=O)C(c1ccnn1C)O 7682,Cc1cc2[nH]c(C(N3CC4CC3CC4CNC(C3CCCN3N=O)=O)=O)cc2s1 7683,Cc1c(C(N2C3CCC2CN(C(=O)C(O)C(C)C)C3)=O)sc2ccnc(O)c12 7684,CCC(CN(C)C)CC(=O)NC(C(=O)N(C1CCSCC1)C)C1(O)CCC1 7685,c1(C(N(CCCN(C)C(C2CC2(F)F)=O)C)=O)ncccc1Br 7686,C1(NC(C2CC23CCC3)=O)COCCC1NC(C1CCS(=O)CC1)=O 7687,N1(C(C23C(C)(C)C(CC2)C3)=O)CC(NC(c2cc[nH]n2)=O)C2(CCCC2)C1 7688,C(C1CN(C(C2(C)CC2(F)F)=O)CC1C(N1CCC(C)(C)CC1)=O)=CC 7689,Cc1cc(F)sc1C(=O)NC1(CC=CC(=O)NCC(O)CC(C)C)CCC1 7690,c1(C(=O)NC(CNC(C(C2CCC2)OC)=O)C)cc(O)c2cnn(C)c2c1 7691,N1(C(C(C)NC(COC)=O)=O)CCCCC1C(N1CC2CC2(CO)C1)=O 7692,CCC(CC(=O)NCC1CCCCCN1C(=O)COCc1nnc(C)s1)C(C)C 7693,c1(CC(=O)NC(C)CCS(C)=O)ccc(Br)c(C#N)c1 7694,C(=O)(CC(CC#C)c1ccccc1)N1CCCC(N(C(C(F)=CC)=O)CCOC)C1 7695,C1(CN(C(=O)CC2CCOCC2)CC)CCN(C(c2cnn(CC)c2)=O)CC1 7696,C1(CNC(c2cc[nH]n2)=O)(NC(c2ccc(-c3ccccc3)o2)=O)CCCCC1 7697,C1(NC(c2[nH]nnc2C2CC2)=O)CN(C(c2cncc(F)c2)=O)C2CC12 7698,c1(C(=O)NC(CC)CN(C)C(C2(CF)CCOCC2)=O)ncc(C)cc1Br 7699,C(C(C(C)(C)C)CC(=O)O)NC(=O)NC1CC(OCCOC)C1 7700,C(=O)(C1=CC2(CCN(C(c3cc(=N)[nH][nH]3)=O)C2)C1)NCC(C(=O)NC)(C)C 7701,Cc1cccc2[nH]c(=NC3CCC(Nc4ncc(C(F)(F)F)cc4Cl)CC3)sc12 7702,CC1(C(F)F)CC1C(=O)NO.C1(=O)CCN1c1cccs1 7703,c1(C(N2CCC(NC(C3CC(C)(CC)C3)=O)C(C)C2)=O)ccc2c(c1)CC(=O)N2 7704,C1(N(CCC)C(C2CCN(c3nccn3C)C2)=O)CC2OCCC12 7705,C1(CNC(c2cc(CC)n(C)n2)=O)CCC(C)CN1C(=O)CSc1ccncc1 7706,C(=O)(C(C)C(C)C(C)(C)C)NCCC(=C)CNC(c1ccc2c(c1)nnn2C)=O 7707,CC(C)CCC(c1nnnn1Cc1ccccc1)NCCC1(C)CC1(Cl)Cl 7708,N1(C(CNC(c2c(CCC)n[nH]c2)=O)=O)CC2CC1CS2 7709,c1(C(=O)NC(C(C)NC(CCc2ccc(C)o2)=O)C)ccccc1C#CC1CC1 7710,C(=O)(C1=CC(C)(CC)C1)NCC(C1CCN(C(CC)=O)CC1)O 7711,c1(C(N2CCC(NC(C(CC)C)=O)C(F)C2)=O)nn(C)c2ccc(Br)cc12 7712,c1(C(=O)NC2CCN(C(C3(OCC)CCOC3)=O)C2)cc(F)cc(C)c1N 7713,c1(C(=O)NCC=CCNC(=O)CC2CC(F)C2)ccccc1C#CC1CC1 7714,Cc1[nH]cc(C(=O)NC2CC(CO)N(C(=O)CCCN(C)C(C)C)C2)c(=O)c1Cl 7715,c1(OC)ccc2c(=NCC3CN(C(C)=O)C3)[nH]c(=NC(C)CS(C)=O)[nH]c2c1 7716,N1(C(CC=C)=O)CCCCC(C2CN(C(c3ccc(O)c(N)c3)=O)C2)C1 7717,C1(NC(CC(CC)C)=O)CCN(C(=O)C(C)NC(=O)CC(C)(C)C)C1(C)C 7718,N1(C(C(C(C)O)NC(C(CC#C)O)=O)=O)CCCCC1C#C 7719,c1(OCCCC)ccc(C(=O)NCC(CNC(=O)CCn2ccnc2)OC)cc1 7720,C1(NC(C2(C(N(C)C)=O)CC2)=O)CC2CCC1N2C(C1CCOC1(C)C)=O 7721,C1(C(=O)NCCCC(=O)NC)(CO)CCOCC1.C1(C=O)CC12CCCC2 7722,n1(CC(=O)NCC(C)(C)c2nc[nH]n2)cccc(N)c1=O 7723,c1(C(N2CCC(CNC(c3c(C)nc(C)s3)=O)C2)=O)oc(P(C)(C)=O)cc1C 7724,c1(NC(C(N2CCC(O)CC2)C)=O)cncc(-c2ccc(F)cc2)c1 7725,C1(C)(C(=O)NCC(C)CN(C(=O)CNC(c2ccncc2)=O)C)CCCO1 7726,c1(CN(C)C)cccc(C(=O)NCC=C2CCN(c3ncc(Br)cn3)CC2)c1 7727,C1(CC(=O)N(CCCCCNC(=O)Cc2nn(C)cc2Cl)C)COCC(C)(C)O1 7728,C1(CC(C)C)(C(=O)NC2(C(=O)OC)CCC2c2ccccc2)CCNC1=O 7729,CCC(C(=O)NC(c1cnn(C)c1)C)NC(c1ncc[nH]1)=O 7730,C1(CO)(CNCc2cn(-c3cccnc3)nn2)CCCC1 7731,C#CCC(CC(=O)NCc1c[nH]nc1C1CC1)NC(=O)CCN(C)C 7732,N1(C(CN(CC(C)C)C(C2CC(C)CC(C)C2)=O)=O)Cc2cccnc2C1 7733,c1(C(=O)NCC(CNC(c2[nH]cc(CC)c2)=O)C)sc(CC(F)(F)F)nc1C 7734,c1(C(N2CC(CC=C)(NC(=O)Cc3ccc(O)nc3)C2)=O)ccc(Cl)c(C)c1O 7735,c1(C(=O)NC(C(C)NC(CCCC#CC)=O)CO)ccc2c(c1)COC2 7736,n1(CC(=O)NCCNC(C)=O)cc(C(N2CC(C)(NC3CC3)C2)=O)c(O)nc1=O 7737,c1(C(N(CCCCN(C(CCCC(C)=O)=O)C)C)=O)[nH]c2c(c1C)CCCC2 7738,C1(O)(CCNC(CCC2N(C)CCC2)=O)CCN(C(C2(C)CCCCO2)=O)C1 7739,Cc1cc(S(=O)(=O)NCCC(c2cccc3c2OCCO3)=O)cnc1C(F)(F)F 7740,c1(CC)ccnc(C(N2CCCC(c3n[nH]c(CNC(=O)COC)n3)C2)=O)c1 7741,C=CCC(C)(CC)C(=O)N(CCC(C(C)C)NC(=O)CN(C)CCC)C 7742,c1(OC)ccc(F)cc1C(N1CCC(CNC(=O)COC2CCC(C)CC2)C1)=O 7743,Cc1conc1C(=O)NCC1(CNC(C2CCC(=O)O2)=O)CCC1 7744,Cc1ccccc1C=CC(=O)NCC1C2CN(c3nccc(CO)n3)CC12 7745,c1(CN2CCC(CC(=O)Nc3c(CN)nc(Br)cn3)C2)ccc(F)c(F)c1Cl 7746,C=CCC(CC(F)F)NC(C1C(CC)CCN1C(c1cccc(F)c1)=O)=O 7747,N1(C(C2(CC)CCC2)=O)CC2CCCC2(NC(=O)CCN2CCCCCC2)C1 7748,C1(OC)CC(CNC(C2CC(F)(F)C2)=O)N(C(=O)C(F)C2CCCC2)C1 7749,C12(NC(C(CCSC)NC(N)=O)=O)CCCCC1CN(C(=O)C1CC1)C2 7750,N1(C(C2C(C=C(C)C)C2(C)C)=O)CC(COC(=O)C2=CCCCO2)C(C)(C)C1 7751,C(=O)(C(CNC(=O)C(C)NC(N)=O)OC)N(CCCF)CC 7752,C(=O)(C1=CCCOC1)N1C(CNC(c2ccc(C#N)n2C)=O)CC(OC)C1 7753,C1(C(N2C(CN(C(=O)CCc3ccoc3)C)CCC2)=O)CC(F)C(=O)N1 7754,N1(C(=O)CNc2ccccn2)CC(C(N2CC(N3CCNC3=O)C2)=O)C2(CC2)C1 7755,c1(OCC(N2CC(NC(C3CCCOC3)=O)C2)=O)ccc(F)c(Br)c1 7756,C1(NC(C2(CNC(=O)CC3CNC(=O)O3)CC=CC2)=O)CC2CCCCN2C1 7757,CC1(CC(=O)NC(CO)CCCO)CCN(C(c2ccc(C(N)=O)o2)=O)C1 7758,C1(C(=O)NC(COC)C)CN(C(c2cnc(C(C)=O)cn2)=O)CCN1 7759,CC1CC2CN(C(C3CN4CCN3CC4)=O)CC2N1CC(F)(F)F.C(C)(C)C 7760,C1(CNC(Cc2ccc(C)cc2)=O)CC(C(=O)N(C)Cc2scnc2C)=NO1 7761,C#CCCC(C(=O)NC1CC(O)C(O)C1)NC(c1snc(C)c1N)=O 7762,c1(CCC(=O)NC2CC(O)CN(C(=O)C(O)C3CCC3)C2)c[nH]c2ncccc12 7763,C(=O)(C(C(C)(C)C)NC(c1cnc(OCC(F)(F)F)c(Cl)c1)=O)OCC 7764,Cc1c(C(=O)NC(CNC(C2CCCN2C(N)=O)=O)CO)oc2ccc(Cl)cc12 7765,N1(C(C2C(C)CC2)=O)CC2CCN(C(=O)CCC3CCC3)CC12 7766,N1(C(C(C)(F)F)=O)CC2(CCCN(C(=O)C=Cc3ccc(C(F)(F)F)cc3)C2)C1 7767,c1(N(C(C(=O)NC(COCC)C(C)C)=O)C)cc(Br)cn1C 7768,CC(C)CC(CNC(c1cncc(C2CC2)c1)=O)NC(=O)C(C)c1ccco1 7769,c1(CC(=O)NC(C2CN(C(c3n[nH]c(=N)[nH]3)=O)CCO2)C)cn2c(n1)CCCC2 7770,Cc1nc(C(C)C)sc1C(=O)NCC1(O)CN(c2nc(CC3CC3)ns2)C1 7771,C#Cc1ccc(C(=O)N(CCC(=O)NC(CC2CCCC2)CO)C(C)C)c(C)c1 7772,c1(C(=O)Nc2nc(C)c(C(=O)NCc3ccccn3)s2)cc(C(F)F)ccc1F 7773,c1(C(=O)NCC2COCC2CF)cnn(CC(N2CC(N3CCOC3=O)C2)=O)c1 7774,C1(CNC(C2(CC#C)CCCO2)=O)CCC2(CO1)CC(NC(=O)CC=C(C)C)C2 7775,c1(CC(N2CC(F)(CNC(C34CC(C)C3C4)=O)C2)=O)ccc(S(C)=O)cc1 7776,CC1CN(C(=O)CCN=[N+]=[N-])CC(C(N2CCC2CC2CCCC2)=O)O1 7777,C1(C(=O)NC2C(=O)NCCCC2)CC2CCC(C1)N2C(=O)C(F)C1CCCC1 7778,CCC(C)(CNC(=O)Cc1cc[nH]n1)NC(c1nocc1C)=O 7779,CN1CCN(CCC(N2CCC(NC(C3(CC(F)F)CC3)=O)C2C2CC2)=O)CC1 7780,C(=O)(CC(C)CCCCCC)NCC1(O)CN(C(C(C=C)(C)CCOC)=O)C1 7781,CC(C)C(O)C(C)C(=O)NCC(CO)NC(=O)CS(=O)(=O)Nc1ccccc1 7782,CCC(CC)CCC(=O)NCCCCNC(C1CCCN(C(=O)C(C)CC)C1)=O 7783,C1(O)(CCNC(C2CCCC(OC)C2)=O)CCN(C(C2NC(=O)CC2C)=O)CC1 7784,c1(C(=O)NCC2(CN(C(c3nc(COC)oc3)=O)C)CC2)n[nH]c2ccccc12 7785,C1(C(C)NC(=O)OC(C)(C)C)CC(NCCCC(C)(C)C)C1(C)C 7786,c1(OCCC)ccc(C(=O)NC(C)CCCNC(=O)Cn2ccc(C)n2)cc1N 7787,c1(C(=O)NC2(CO)CN(C(C=C(CC)CC)=O)C2)cc(C)ncc1C 7788,C1(F)(C(=O)NC2CC(OCC(=O)N(CCN(C)CCO)C3CC3)C2)CCCCC1 7789,N1(C(CCSCCC)=O)CCN(C(=O)C(C(C)(F)F)c2ccccc2)C(CC)C1 7790,NC(=O)CCCC(=O)NCCC1CCCCN1C(=O)CCNC(c1ccsc1)=O 7791,N1(C(C(C)NC(CC)=O)=O)CC(C)C(C)(CNC(c2nsnc2O)=O)C1 7792,C1(NC(C(C(CC)C)N)=O)COC2(CCN(C(c3cc(C)n(C(F)F)n3)=O)C2)C1 7793,c1(C(N2CC(O)(CNC(CC(=C)C)=O)C2)=O)cc(C)c(F)c(S(C)(=O)=O)c1 7794,c1(C(=O)NCC2(O)CCN(C(C(C)C#N)=O)C2)c(C2CC2)nc2sccn12 7795,Cc1nccnc1C(=O)NCC(C(C)C)NC(=O)C=CCN1CCCC1 7796,C(C(C)(C)C(=O)N1CC(OCC(=O)NC2(C)CCOC2C)C1)SC 7797,N1(C(CNS(CC)(=O)=O)=O)CC(NC(c2ccc(C(F)F)c(F)c2)=O)CC(F)C1 7798,N1(C(C2(COC)CCC2)=O)CC(CNC(=O)C(C)Cc2cnn(C)c2)C(C)C1 7799,Cc1cc(C)c(OCC(=O)NC(C)C(C)NC(c2cccc(=S)n2O)=O)c(C)c1 7800,C(=O)(CCCCCCS(N)(=O)=O)NC1CC2CN(C(C(CC)(F)F)=O)C1C2 7801,C1(C(F)F)(CNC(CN(CC(C)C)C(C2(CO)CC=CC2)=O)=O)CCN(C)C1 7802,c1(C(=O)NC2CCC(CNC(c3n(CC)nnc3C)=O)C2)cc(OC)ccc1Cl 7803,c1(C(=O)OCC)sc(N2CCCC2CC(=O)OCC)nc1C.C123CC1CN(C2)C3 7804,C1(CC=C)(C(=O)N(CC)Cc2nccs2)CCCN1C(=O)CC1CC2(CCC2)C1 7805,N1(C(C(C)NC(C)(C)C)=O)CCCN(C(C2CN3CCN2CC3)=O)CC1C 7806,N1(C(C2C(NC(C3(CC#C)CCOC3)=O)CCC2)=O)CCOC(CCF)C1 7807,N(C(=NCC(C)(C)CS(N)(=O)=O)N1CCC(Cc2ccccn2)CC1)C(C=C)C 7808,C(C(=O)NC1CN(C(C2CSCC(=O)N2)=O)C1)(C(C)C)c1cnc(C)s1 7809,c1(C(=O)OC)cc(S(=O)(=O)N2CC(CC#N)C2)c(F)cc1C 7810,N1(C(C2C3CCN(C(CC(CC(C)C)O)=O)CC32)=O)CCC2CCN(C)CC12 7811,CCC(CC(C)C)C(=O)NCC1(NC(c2cnc(SC)s2)=O)CCOC1 7812,c1(CC(=O)NC2C(C)N(C(=O)CC(C)(C)O)CCC2)nnc2n1CCOC2 7813,c1(C(C)=O)cc(C(N2CCCC(C)(CNC(=O)C(O)C(C)C)C2)=O)ccc1C 7814,N1(C(c2cc(OC)no2)=O)CCCN(C(C2(CC(C)C)CC2)=O)CC1C 7815,c1(C(=O)NCC(C(=O)NCCCC(CC)C)(C)CC)cc2ccccn2c1 7816,C(C(CC(C)C)C(=O)N(CCC(=O)N(C)CCN1CCCCC1)C)OC 7817,C1(NC(c2nnc(C)s2)=O)CN(C(=O)Cn2cnc([N+](=O)[O-])n2)CCC1O 7818,Cc1nc2c(o1)CCN(C(=O)CC(C(C)(C)C)NC(=O)C=Cc1cn(C)nn1)C2 7819,c1(C(N(CC(C)C)C)=O)ncn2cc(CCN3CCCC(CCO)C3)ccc12 7820,N1(C(c2c(CC)nns2)=O)CC(Nc2ncc3c(n2)CCCC3)CC2(CCC2)C1 7821,C1(OC)CC2(C1)CC(C(c1nnnn1CCCSC)Nc1ccccc1)C2 7822,N1(C(CC)(C)C)CCN(C(=NCC2CC2)NCC2(O)CCS(=O)(=O)C2)CC1 7823,c1(CC(C)N(C(=O)NC2CC(COC)C2)C)ccc(Br)cn1 7824,C1(C)(CNC(C2(SC)CCCCC2)=O)CCN(C(c2ccc(=N)[nH]n2)=O)CC1 7825,C1(NC(CN2CC(C)(C)C2)=O)CCN(C(C2CCC(C)(C)OC2)=O)CC1(C)C 7826,C1(CCCC)CN(C(c2ccc(CC)nc2)=O)CCN1C(=O)C#CC(C)C 7827,C1(NC(COCCOCC)=O)CCCC1NC(C12CC(CO1)C2)=O 7828,CC1(C)CC2(CC2NC2CCC2c2cccnc2)C1 7829,c1(OC)cccc(C(N2CC(CNC(=O)Cc3ccc(OC(F)F)nc3)C2)=O)n1 7830,CCC(C)(C)C(=O)C(=O)NCC=CCC(=O)NCC12CC(CO)(CO1)C2 7831,c1(C(C)NC(C(=O)NC2CC(C(F)F)(OC)C2)=O)cc(Cl)c(C)cc1O 7832,c1(NC(c2cnc(C)[nH]2)=O)cccc(NC(=O)CC(C)(F)F)c1 7833,CCC(N(C)N1CCN(C(c2ccc(F)cc2)=O)CC1)c1cc(Cl)cc(Cl)c1 7834,C(=O)(C1=CS(=O)CCC1)N(CCCCCCNC(C1CC1C1CC1)=O)C 7835,C(N=c1cc(C)nc(C)[nH]1)C1(C)CCCN(C(CS(CC)(=O)=O)=O)C1 7836,C#CCCC(C(=O)NCCc1ccn(C)n1)NC(C1CC2(CCC2)CO1)=O 7837,N1(C(c2cc(SC)oc2)=O)CC2CC1CCC2NC(=O)Cc1ccc(F)cc1F 7838,N1(C(C=CC=C)=O)CCC(F)(C(=O)NCCOOC2CCC2)CC1.CC=C 7839,C1(C(=O)NCC(CC)NC(C(CC)c2ccccc2)=O)CC(C)CC(=O)N1 7840,N1(C(=O)NCC2CCC(C)O2)CC(CNC(=O)OC(C)(C)C)C2(CC2)C1 7841,c1(NC(C(C(=O)OC)C)=O)ccc(C)c(C(=O)NC2CCCC(O)C2)c1 7842,N1(C(C(C)OC)=O)CC(O)CC1CNC(C1CCC(=O)N1C(C)C)=O 7843,C1(CC)CCOC1C(=O)NCCCC(=O)NCC1CCCCO1 7844,C1(C)(CNC(C(CC)(C)CO)=O)COCCN(C(=O)CCc2cnn(C)c2)C1 7845,N1(C(c2n(CC)cnn2)=O)CCC(C2CC2)C1CNC(c1nc(F)ccc1Cl)=O 7846,N1(C(=O)CC2CC2)CCC2CCCN(C(c3ccccc3C3CCC3)=O)C2C1 7847,C(CNC(=O)C(F)(F)C(C)(C)O)(CC(=O)N1CC(O)CCO1)OC 7848,N1(C(C(CC#C)NC(=O)C(O)C(C)(C)C)=O)CC2C3CCC(C3)C2C1 7849,C(=O)(C1COc2ccc(F)cc21)NC1C(NC(=O)Cc2ccc(Cl)cc2)C1 7850,C#Cc1cc(C(N2CCCCC(NC(=O)CS(=O)(=O)C(C)C)C2)=O)cc(Cl)c1 7851,N1(C(C(C)Cc2cnc[nH]2)=O)C2CCC1CN(C(=O)C(F)Cc1ccccc1)C2 7852,c1(C(N2C(CO)CC(NC(C3=NOC(C)C3)=O)C2)=O)cncc2ccccc12 7853,C1(N)(C(=O)OC)CCS(=O)(=NC(=O)C(C)(C)c2ccn3ccnc3c2)CC1 7854,N1(C(CCCOCCC)=O)CCCC2(NC(c3nncn3C)=O)CCCC12 7855,C(CC(C)(C)CC(=O)NCc1ccc(C(=O)NCC2CCC(C)(C)C2)nc1)OC 7856,C1(CCC(C)(C)NC(C2(N3CCCCC3=O)CC2)=O)CCN(C(=O)C2CC2)CC1 7857,CC1CCCCC1Cc1nc(-c2cccc(Cl)c2)nn1-c1cnn(C)c1 7858,C=CC(C)(CCOC)C(=O)NCC1(NC(=O)CNC(C)=O)CCCC1 7859,Cc1c[nH]nc1C(=O)NCCN(C(=O)C(F)n1cccn1)C1CC1 7860,N1(C(CCCc2n(C)cnn2)=O)CCCC(C(C)(O)CNC(C2(SC)CC2)=O)C1 7861,C1(NC(c2nncs2)=O)CC2CC(NC(C34CCCC(CO3)C4)=O)C1C2 7862,Cc1cc(Cl)ncc1CC(=O)NC1CC2CCC1(NC(=O)C=Cc1ccoc1)C2 7863,CCC1=NOC(CNC(=O)Nc2ccnc(OC(C)C)c2)C1 7864,Cc1nc(C)n(CC(=O)NC(CN(C)C)C(=O)NCCCN=[N+]=[N-])n1 7865,c1(C(N2CCC(CC(C)NC(C3(C=C)CC3)=O)CC2)=O)ccc(F)c(Cl)c1N 7866,C1(NC(c2c(F)c(F)cc(F)c2F)=O)CN(C(=O)CCF)C2CCCCC12 7867,C(c1ncc[nH]1)=CC(=O)NCC(C)(C1CC1)NC(C1CC(CC2CC2)C1)=O 7868,C1(C(=O)N(CC(C)C)CC(C)C)(CCCNC(c2cc(C)[nH]n2)=O)CC12CCC2 7869,c1(C(N2CCN(C(CC(C=C)CCC)=O)CC(C)C2)=O)cccn2cc(C)nc12 7870,N1(C(C(n2c(C)ncc2)C)=O)CC(NC(=O)CC(F)(F)C(F)F)CC12CCC2 7871,C1(CN(C(CC(=C)Br)=O)C)CCN(C(C2CCCC(OC)C2)=O)CC1 7872,c1(C(N2CCN(C(C(C)(C)C3CC3)=O)CC(O)C2)=O)cc(F)cc2nc(S)[nH]c12 7873,Cn1c(O)nc2cc(CNC(=O)NC(C)(C)CCNS(C)(=O)=O)ccc12 7874,c1(CCC2(C(=O)N(C(CN(CCCC)C)C)CC3CCC3)CC2)ccsc1C#N 7875,N1(C(CC2(OC)CCC2)=O)C2CCCC1CN(C(C1CC(O)C1)=O)C2 7876,n1(C(CC)CC)nccc1C(=O)NCC(C)(C1CC1)NC(=O)C(CO)N(C)C 7877,c1(C(=O)NCCCC2N(C(C3CCN(C)CC3)=O)CCC2)n[nH]c2c1CCC2 7878,C1(CC(=O)N(CC(C)N(C)C(c2cc3sccc3s2)=O)C)CCC(C)(C)CO1 7879,c1(C(=O)NC2CC(C)(NC(C3CC3C(F)(F)F)=O)C2)cccn2nccc12 7880,c1(C(NNCC=C)=O)sc2cc(Cl)ccc2c1Cl 7881,C=CCC(C)C(=O)NCC(C(=O)N1CCC(COC)C1)N(C)C 7882,Cc1c(F)ccc(C(=O)NC23CC2CN(C(C2CCC(=O)N2C2CC2)=O)C3)c1Cl 7883,N1(C(COC)=O)CCN(C(=O)CP(C)(C)=O)C(CO)C1 7884,Cc1cc2[nH]c(C(=O)NC3CC4CC3N(C(c3ccsc3)=O)C4)cc2o1 7885,N1(C(c2nc(NC(C)=O)sc2)=O)C2CCC1C(NC(=O)CC1CC3CCC1CC3)C2 7886,C(CCN=c1ccc(C(F)(F)F)c[nH]1)NC(c1cccc(Br)c1Br)=O 7887,Cc1nc(F)ccc1NC(=O)CCC1CCC(NC(=O)CCCC#N)C1 7888,N1(C(c2c(OC)ccc(Br)c2)C(=O)NC2CC2)CC(C)OC2(CCC2)C1 7889,c1(NCCCN(C(=O)Cc2ccc(O)nc2)C)ncnc2c1cnn2C 7890,C1(C(C)(CNCCCOCCO)OC)CCOCC1 7891,CC(CN(C)C)CCC(=O)N1CC(CNC(c2cccs2)=O)CC1(C)C 7892,N1(C(CC2C(C)CCN(C(CC=CCC)=O)C2)=O)CC(C)(CO)CC1(C)C 7893,C1(NC(c2ccc(OC3CCC3)cc2)=O)CN(C(c2ccccn2)=O)CC12CC2 7894,N1(C(c2ccc(C#C)o2)=O)CC2CCC1CN2C(=O)Cc1cc(C)on1 7895,C1(CNC(C(c2ccccc2F)C)=O)CCN(C(C23CC(C)(CO2)C3)=O)CC1C 7896,C(=O)(C(C)CC(F)F)NCC(CC=C)NC(c1ccnc(OCC)c1)=O 7897,Cn1c(C(N2CC(O)(C(F)C(=O)NC3CC(=O)N(O)C3)C2)=O)ccc1C#N 7898,CC1CCCC1CC(N1CC(CCCCNC(=O)CNC(c2ccsc2)=O)C1)=O 7899,c1(C(=O)NC2CCCN(C(C3CN(CC)C(=O)C3)=O)C2)ccc2c(c1)CCCN2 7900,C1(OC)CCC12CC(C(=O)NCCn1cc(CSC34CCN(CC3)C4)nn1)C2 7901,C(c1ccc(F)cc1)=C(C)C(=O)N1CCC1n1cccn1.C12CCN1CC(=O)C2 7902,C(=O)(C(C)S(N)(=O)=O)N1C(C(N2CC(CO)C2)=O)(COC)C=CC1 7903,N(C(=NCCC(=C)C)NC1CCN(c2ccc(-n3cncn3)cc2)CC1)C1C(=C)C1 7904,N1(C(CC(C(C)C)c2ccon2)=O)CC2CCC1C(CNC(C1(CO)CC1)=O)C2 7905,c1(C(=O)NCC2C(C)CN(C(C3(CO)CC3)=O)C2)ccc2c(O)ncnc2c1 7906,C(=O)(C1=CC2(CCOC2)C1)NCCN(C(=O)CCc1cnc[nH]1)C 7907,c1(CNC(c2n(C)cnc2)=O)nc(CNC(C2CCC3(CCC3)C2)=O)cc(O)n1 7908,c1(CC)cnc(C(=O)NC2CCC(C(=O)N(C(C)CC(C)C)C)C2)nc1 7909,Cc1cc(=NC(=O)C(=O)NCC2(NC(=O)C(O)C3CCCC3)CCC2)[nH]o1 7910,c1(C(=O)NC2C(NC(C3(CC)CCOCC3)=O)CC2)cncc(C)c1C 7911,C1(NC(C2(C)CC=CC2)=O)CC2CCCC(C1)N2C(c1cnc(Cl)s1)=O 7912,O=S(=O)(c1c[nH]c2cc(Cl)c(Cl)cc12)Nc1cccc2c1CCOC2 7913,N1(C2CCN(C(C3CN(C)C3)=O)CC2)Cc2cccnc2N2CCCC2C1 7914,C1(CNC(C(c2cnn(C)c2)OC)=O)CN(C(c2c(Cl)cnn2CC)=O)CCO1 7915,c1(N2CCN(CCN(C(=O)CC3CC(=O)NC3=O)C)CC2)ccccc1[N+](=O)[O-] 7916,N1(C(C2(CC#C)CCOC2)=O)CCCC(C)(NC(=O)CC(C)(C)OC)C1 7917,c1(-c2cn(C3CCN(CCNC(CCCC)=O)CC3)nn2)cc(F)ccc1Cl 7918,c1(SCC(=O)NCC(C)(C)NC(C(CO)N(C)C)=O)nc2ccccc2o1 7919,N1(CC)CC(NC(=O)C(C(C)(C)C)NC(=O)C=Cc2cncn2C)CCC1=O 7920,C1(CC)CCC(C(=O)NC2CC23CC(NC(=O)COCc2ccncc2)C3)CC1 7921,C(=O)(C(CCNC(c1cccn1C1CC1)=O)OC)NC1(CC#C)CC1 7922,N1(C(C2(OC)CCN(C(=O)C=CC(C)C)C2)=O)CC(=O)NC(C)C1 7923,N1(C(COCC(=C)C)=O)CCC2C(NC(=O)COC(F)(F)F)C2C1 7924,N1(C(C2(CC)CCCCC2)=O)CC(CN(C)C(c2ccoc2)=O)C2(CC2)C1 7925,C(=O)(C(CC(C)C)NC(=O)C(C#N)C(C)C)N(c1ccc(C)cc1)CC 7926,c1(NC(CCC(=O)C2CCCCC2)=O)nc(F)c(I)cc1F 7927,C1(O)(C(N2CCCC(CC(=O)NCC(CC)n3cccn3)C2)=O)CCCCCC1 7928,C1(NC(C2ON=C(C)C2)=O)CCCC2CN(C(c3csc(C(F)(F)F)c3)=O)CC12 7929,CC1(CNC(=O)CC2NC(=O)NC2=O)CCN(C(=O)CCc2ncccn2)C1 7930,c1(CC)ccc(F)cc1C(=O)NCC(C)(CO)NC(c1cc(F)ccc1O)=O 7931,N1(C(C(C)SCC)=O)CCN(C(=O)CCOC(C)=O)CC1CC(F)F 7932,C12(C(N(C)CCOCCNC(C3CSCCS3)=O)=O)CCC(C1)C(C)(C)O2 7933,c1(C(N2CC(CCNC(C(C)OC)=O)C2)=O)ccc2nc(O)[nH]c2n1 7934,N1(C(=O)Cn2cc(C(F)F)cn2)CC=CC(NC(C2(c3ccsc3)CC2)=O)C1 7935,C(CC(C(C)(C)C)NC(C1CCCN1C1CCCCC1)=O)N(C(C)=O)C 7936,N1(C(CCOCC(C)C)=O)CC2(CCCC2)C1C(=O)NC(C1(O)CCC1)C 7937,N1(C(CNC(C(C)(C)C)=O)=O)CCC(N=[N+]=[N-])(C(=O)NCC2(O)CCCOC2)C1 7938,C1(NC(C(C)n2cncn2)=O)COCC1CNC(c1csc(C(F)F)n1)=O 7939,C1(N(C(C(C)SCCCC)=O)C)C2CN(C(c3cc[nH]c(=N)n3)=O)CC12 7940,c1(C(=O)NCC2CN(C(CCC3C(C)=NOC3=O)=O)C2)nc(O)nc(O)c1N 7941,Cc1cc(C(N2CCC(OC(C)C(N)=O)CC2)=O)c(Br)cc1F 7942,CCC(C)C(O)CC(=O)NC(CNC=O)CC(C)C.C(CC(F)(F)F)O 7943,C1(OC)CCC(NC(=O)CCN(C)C(c2ccc(C)o2)=O)C1 7944,c1(OC)ccc2cc(C(N3CCC(NC(=O)Cc4cnc(C)o4)C3C)=O)[nH]c2c1 7945,C=CC(O)C(=O)NC(Cn1cccn1)C(=O)N1CC(C)(C(N)=O)C1 7946,N1(CC)CC(C(=O)NCC2CCCC2NC(=O)CC2CCCOCC2)CCC1=O 7947,N1(C(C(CC=CC)NC(=O)CC2(O)CCCC2)=O)CCC12CCCSC2 7948,C1(C)(CNC(c2cnc(NC(C)=O)o2)=O)CCCN1C(c1cnn(C)c1Cl)=O 7949,Nc1ccc([N+](=O)[O-])cc1C(N1CCC2C(NC(=O)CCC(F)F)C12)=O 7950,C(=O)(CC(CCC)CCC)N1CC(CC=C)(NC(=O)C=Cc2cn[nH]c2)C1 7951,C(=O)(C1=CC(C)(C)C1)N(C)CC1CCN(C(c2cnc(C)nc2)=O)C1 7952,C(=O)(C(C)(C)C(=O)NCC=CCNc1cn(CC2CCOCC2)nc1C)OCC 7953,CC1(NC(=O)C=Cc2cncnc2O)CCCN(C(c2cccc(=O)o2)=O)C1 7954,c1(CNC(c2cnc(C)s2)=O)ccc(C(=O)NCC2(F)CCOCC2)nc1 7955,C1(O)(Cn2cc(-c3n(C)ncc3)nn2)CCN(C(=O)COc2ccccc2)C1 7956,C(C1=CCN(C(c2cnc(-c3ccco3)s2)=O)CC1)NC(C1(C=C)CCC1)=O 7957,C1(C(N(C)Cc2c(C)cco2)=O)C2CC3C(C2NC(C2CCC(F)C2)=O)C13 7958,C(=O)(C1=CC2CCCC12)NCCC1CN(C(=O)CCc2ccco2)C1 7959,CC(CC(N)=O)C(=O)NCC(C)CNC(C1(C(F)(F)F)CC=CCO1)=O 7960,c1(C(N2CC(NC(C3CC(O)(CC)C3)=O)CC2(C)CC)=O)ccn2nncc2c1 7961,N1(C(C2C(OCC)CC2)=O)CC2OCC(NC(=O)C(F)(F)C(C)(C)O)C2C1 7962,c1(C(N2C3CCC2CC(C(N2CCC(CO)C2)=O)C3)=O)c(F)cc(Cl)cc1Cl 7963,N(C(=NCc1ccoc1)NCc1ccccc1-c1ccc(F)cc1)CC(C)(C)C 7964,C=C(Br)CCC(=O)NCC(CC)NC(=O)COC(F)F 7965,C(N=c1ccnc(CO)[nH]1)C12OCC(NC(C3CCC(C)CC3)=O)(C1)C2 7966,c1(C(=O)NCC2(OC)CCCC23CC3)ccc2c(c1)C(C)(C)CCN2 7967,c1(C(C(=O)NC(CCN(C)C)C(=O)OC(C)(C)C)=O)c(C)nn(C)c1C 7968,c1(-c2c(C(N(CCC(C)NC(C3CC3(C)C)=O)C)=O)c[nH]n2)ccccc1Br 7969,C(=O)(CCCCC(F)(F)F)N1CC(OCC)C(CNC(c2cnc(O)c(F)c2)=O)C1 7970,c1(C(N(CC(C)(C)NC(C2C(CCC)C2)=O)C)=O)cnsc1C 7971,N#Cc1ccc(Cl)nc1NC(C1C2CN(C(C3CC3(F)F)=O)CC12)=O 7972,C=Cc1ccccc1-c1ccc(CNC(c2sc(C)nc2C)=O)cn1 7973,S(=O)(=O)(c1cccnc1NCC1CC(C)OC(C)C1)NCCS(CCC)=O 7974,c1(N(CCCNC(C2CNC(=O)N2C)=O)CC)ncnc2c1ncn2C 7975,c1(C(=O)NC2CC3(CCN(C(C(COC)O)=O)C3)C2)nc2ncc(Br)cc2[nH]1 7976,C(=O)(C1CCCn2ccnc21)NC(CC)(CNC(=O)C(C(C)C)C1CCC1)CC 7977,N1(C(=O)CC(F)(F)CBr)CC2CCN(C(c3cncnc3)=O)CCC2C1 7978,N1(C(C)=O)CCCC1CC(=O)NC(C1CCCN1C(=O)CC1(C(F)F)CC1)C 7979,Cc1ccc(Cl)cc1OC(c1ccc(N2CCOC(C)C2)cc1)=O 7980,N1(C(C2CC(C)(C)C2)=O)CCC2CN(C(c3cc(C(C)(F)F)n[nH]3)=O)C2C1 7981,N1(CC(=O)N(C(C)C)CCN(C)C(c2ccc(Cl)s2)=O)CCc2ccccc21 7982,C(=O)(C(CO)NC(c1cn(C)cn1)=O)NCC(C)NC(=O)OC 7983,c1(C(N2CCC(C(N3CC4CC4(CO)C3)=O)C(O)C2)=O)ccc2cncn2c1 7984,c1(C(N2CCN(Cc3cc(OCC)cc(F)c3)C3C2C3)=O)ccc2cnoc2c1 7985,C1(C(=O)Nc2ccsc2CO)CC2(CC2)CN1S(=O)(=O)c1cccs1 7986,C1(C(N2CCCC(CCC)(NC(C=CCCC)=O)C2)=O)CCC2C(C1)C2(F)F 7987,C(=O)(C(C)(F)C(C)(C)F)NC(C)CC1CN(C(C2CCCS(=O)(=O)C2)=O)C1 7988,c1(C(N2C(CCNC(C3CCCCS3)=O)CSCC2)=O)ccc2c(c1)OCO2 7989,Cc1nc(C(=O)NCC(C)(C)NC(=O)CC2C=NN(C)C2=O)sc1C 7990,C1(CNC(Cn2c(C)c(Cl)cn2)=O)CN(C(=O)C2=NOCC2)CC(C)(C)C1 7991,N1(C(Cn2ncc(CC)c2)=O)CC(C2CC2)(C(N2CC(C3CC3)OC(C)C2)=O)C1 7992,C1(CC(C)NC(=O)Cc2cnccc2Cl)CCN(C(c2cc(Br)n[nH]2)=O)CC1 7993,c1(OC(C)C(=O)NC(CNC(=O)Cc2csc(Br)c2)C2CC2)cccnc1 7994,N1(c2cn(CC3N(C(=O)NC4C5OC(=O)OC54)CCC3)nn2)CCC(F)(F)CC1 7995,Cc1cc(C(=O)NCC(C)CNC(c2cnc(-c3ccoc3)s2)=O)cc(N)c1O 7996,C1(C(=O)NCCN(C(=O)CSC(F)(F)F)CC)CC2CC(OC)C2C1 7997,Nc1cc(C(=O)NC23CC(CNC(C4CC=CCC4)=O)(C2)C3)ncc1Cl 7998,N1(C(CCC=CC)=O)CCC(C2CCN(C(=O)Cc3c[nH]nc3O)C2)C1 7999,c1(C(N2C(CN(C(c3ccnn3C)=O)CC)CCC2)=O)ccnc2ccnn12 8000,N1(C(c2nc(N)c(Br)cc2)=O)CC2(CCN(C(c3ccnn3C3CC3)=O)C2)C1 8001,c1(CNC(c2n(CCCC)nnn2)c2conc2C)nc(C)c(C)cn1 8002,CCC(C)CCC(=O)Nc1ccc(NC(=O)CC2(C)CCOCC2)cc1C 8003,N1(C(C)(C)C)CCC(C(=O)NC2CC(n3cc(C4CCOC4)nn3)C2)C1 8004,C(=O)(C(CNC(C1(CCCF)CC1)=O)CC(C)C)N(C)Cc1c(C)nn(C)c1 8005,Cc1ccsc1CN(C(c1ccc(F)s1)C(=O)NCCCF)C 8006,C1(NC(c2c(CCCC)ocn2)=O)(COC)CCN(C(c2ccc(C#N)o2)=O)C1 8007,n12cc(cn1)CNCCc1cc[nH]c1-2.C(=O)(C(=O)NC)N(C(C)(C)C)CC#C 8008,c1(C(N2C(CCCC)CN(C(c3nccn3C)=O)CC2)=O)cnc2sccc2c1 8009,C1(C)(C(=O)NCC(CNC(c2cnc(Cl)s2)=O)OC)CCCCCC1 8010,C#CCCCCCCCC(=O)N1CC(C)CCC1CNC(C1C2CC(=O)CC12)=O 8011,CCCCC(CN)NC(=O)C(N1CCC(c2nccs2)CC1)=O 8012,CC(C)S(=O)(=O)C(C)C(=O)N1CC(C)(C)OCC1CNC(C1(CC2CC2)CC1)=O 8013,c1(C(C)=O)ncccc1C(=O)NCC1CCN(C(=O)C(C(C)O)NC(N)=O)C1 8014,N1(C(C2C(CC)C2)=O)CCC(C)C(NC(c2cc(-c3ccco3)on2)=O)C1 8015,C(C)(C(=O)N1CC(O)CO1)N(CCC)C(C1CN(C)CCO1)=O 8016,C1(OC)(CNC(=O)C(C2CC=CCC2)NC(=O)Cc2cc(C)no2)CCCCC1 8017,Cn1cnc2c3c(ccc12)N(Cc1ccccc1C(N)=O)C(C)C3 8018,C1(CC)CN(C(c2c(C)noc2N)=O)CCN1C(c1nn(CC)nc1C)=O 8019,C1(C(N(CCOCC)C)=O)CCC(C)CN1C(c1ccc(C)nc1C)=O 8020,Cc1ccc2ccccc2c1NC(C1CC(F)CN(c2ncnc3n[nH]cc23)C1)=O 8021,CC(C)C1=NOC(C(=O)N(CC(=O)NCC(C)(O)C2CCCC2)CC2CC2)C1 8022,c1(C(=O)NC2CC(CNC(CCNC(=O)CO)=O)C2)cc(C2CC2)cs1 8023,C1(NC(c2cncc(C)c2)=O)CCCN(C(c2cc3ccccc3[nH]2)=O)CC1F 8024,C(CCCC(C)(F)F)(C(=O)NCCc1ccc(F)cc1)N1C(C)CCCC1C 8025,Cc1nn(C)c(=O)c(C(=O)NCC(C2CC2)NC(c2ccnn(C)c2=O)=O)c1C 8026,C1(CN(C(C2(C)CSC2)=O)CC)CCN(C(=O)CC2(N(C)C)CC2)CC1 8027,CC(CN(C)C)CCC(=O)N1CCC1CNC(c1ccc(Cl)cn1)=O 8028,C1(CNC(CCC)=O)N(C(C2CC(C3CCC3)C2)=O)CCCC1(C)C 8029,C=C(C)CCCC(=O)N1CCC(NC(C2(C)CC(C)(C)C2)=O)C(F)C1 8030,C1(C2CC2)(NC(c2c(CC)ocn2)=O)CCN(C(=O)COCC(C)C)C1 8031,CC(C)CC(C(=O)O)N(C(=O)C=Cc1ccc(N2CCOCC2)nc1)C 8032,C1(NC(C(C)N=[N+]=[N-])=O)C2CCC(C2)C1C(N1CCC1C(C)O)=O 8033,Cc1cc(F)ccc1C(N1CC2CCC1C2NC(C12CCC(C)(C1)OC2)=O)=O 8034,C(C(C)CN=c1ccnc(C)[nH]1)c1n(Cc2c(C(=O)OC)c(F)ncc2)nnn1 8035,C#CCC(CC(F)F)C(=O)NCC(C1CCCCC1)NC(c1c[nH]nc1CC)=O 8036,C#CCC(C)(CC)C(=O)NC1CCC1NC(C1CCN(C(C)C)CC1)=O 8037,n1(CC(=O)NC2CN(C(Cc3cc(C)on3)=O)CC2C)nc(C)c(Cl)c1C 8038,C12(NC(COC)=O)CC1CN(C(C1(CC3CC3)CC1)=O)C2 8039,FCCCN=C(NCCCN1CCCCC1)NCc1ccccc1 8040,c1(OC)ccc(NC(=O)C(CCNC(=O)CN(C2CC2)C)OC)cc1O 8041,CC(=O)CCCC(=O)NCCNC(C1CN(C(c2ccc(F)o2)=O)C1)=O 8042,N1(C(C2CC(C)(C)CN2C(=O)CC2OCCCO2)=O)Cc2ncsc2C1 8043,C(=O)(CCCCCC(C)C)NCC(C)(C)NC(C1(C(=O)OC)CC1C(F)(F)F)=O 8044,C1(NC(c2cc(-c3n(C)ccc3)[nH]n2)=O)CCCCC1NC(=O)C(=O)NC1CC1 8045,Cc1cccc(CSCC(N2CC(N(C)C(c3ncoc3C(F)(F)F)=O)C2)=O)c1 8046,c1(OC)cc(Cl)ccc1CNC(=O)C=CC(=O)NC(c1nccs1)C 8047,C1(NC(C(c2cccs2)N(C(C(=O)OCC)C)CCCF)=O)(CO)CCSC1 8048,c1(C(N2CCCC(O)(CNC(c3cncc(C)n3)=O)C2)=O)cnc2ccnn2c1 8049,c1(C(=O)NCCC2N(C(Cc3c(C)ccnc3)=O)CCC2)ccc([N+](=O)[O-])s1 8050,CC1(C)COC(C(N2CCCC(c3cn(-c4ncc(F)cn4)nn3)C2)=O)CO1 8051,N1(C(CCC#N)=O)C(CNC(=O)CNS(=O)(=O)c2ccccc2)CC2CCCC12 8052,C(CC(=O)NC(C)(CNC(=O)CC1(C)CCCCC1)CC)(C1=CCCC1)OCC 8053,C(C(C)(CC(C)C)NC(=O)CC(c1ccc(Cl)cc1)O)NC(CCCOCC)=O 8054,N1(CC(=O)NCC(CN(C(c2c(C(=O)OC)[nH]nn2)=O)C)C)CC(=O)NC1=O 8055,CCCC(C)CCCC(=O)N1CCN(CCNC(=O)C(C)S(N)(=O)=O)CC1 8056,N1(C(CCC(=O)N(C)C)=O)CC2CCCC2(CNC(C23CCC(C2)OC3)=O)C1 8057,N1(c2cc(C(C)=O)nc(Cl)n2)CCC2(CC1)CN(C(=O)COC(F)F)C2C(C)C 8058,C1(NC(c2c(CSCC)cccc2)=O)CN(C(=O)CCC2CCOC2)C(C)(C)C1 8059,C(=O)(C(CO)C(C)(C)C)NC1(C)CN(C(c2csc(I)c2)=O)C1 8060,N1(C(C2C(C)(C)C2C(F)F)=O)CCN(C(=O)CN2CCS(=O)CC2)C2CCC12 8061,Cc1ccc(C=CC(N2CCC(CO)C(NC(=O)C(C)S(N)(=O)=O)C2)=O)cc1Cl 8062,c1(CC(=O)NC2CC(NC(c3cc(C(=O)OC)[nH]c3)=O)C2)ccc(F)cn1 8063,c1(CC(C)C(=O)NCC2CN(C(c3ncc[nH]3)=O)CCO2)ccccc1Cl 8064,N1(C(CC(C)c2ccccc2)=O)C(C(=O)N(CC#N)CC#N)CC2CC12 8065,c1(NC(c2cccc(-n3cccc3)c2)=O)ccnc(-n2cc(C(=O)O)nn2)c1 8066,CCCC(C(=O)NC(C)CC(=O)OCC)NC(c1nnn(C)c1N)=O 8067,CCCCCC(O)CC(=O)NC1CCN(C(=O)CC2CCCOC2)CC1 8068,C(=O)(N=c1[nH]ccnc1C(N)=O)C1C(C(=O)Nc2cc(C)nn2C(C)C)C1.C(C)C 8069,C1(C)(NC(CCCOC)=O)CCN(C(C2CCOC2C(F)(F)F)=O)CC1 8070,Cc1c(C(=O)NC(C)CNC(C2CCC(C)O2)=O)sc2ccc(Cl)cc12 8071,N1(C(C2(OCC)CCC2)=O)CCCC(C(C)(O)CNC(c2cccnc2C)=O)C1 8072,C1(NC(N2CC(C)(CC(=O)Nc3ccc(C)nc3)C2)=O)Cc2ccccc2C1 8073,C1(CNC(C(C2CC2)OC)=O)CN(C(c2ccc(F)cc2Cl)=O)CC1(F)F 8074,C(=O)(C1=NOC(C(C)(C)C)C1)NCCCCC1(NC(C=Cc2ccn(C)c2)=O)CC1 8075,C1(CC(F)F)(C(=O)NCCCNC(C2CC2c2ccccn2)=O)CCOCC1 8076,c1(NC2CCCN(C(c3cccc(C)c3)=O)C2)nc(Cl)nc2c1ncn2C 8077,c1(C(C(C)C)C(=O)NCCC(N2CCN(C)CC2)=O)cccc(C#N)c1 8078,N1(C(c2c(COC)cco2)=O)CCCC(N=c2[nH]ncs2)CC1 8079,N1(C(C(C)OCC)=O)CCC2(CC1)CC2CNC(=O)CC1CCCCCCC1 8080,c1(CCC(N2CC(CC)C2)=O)nc(C)cs1.C(=O)(CCn1cccn1)N(C)C 8081,Cc1ncccc1C=CC(N1CCN(C(=O)C=CC2CCOC2)CC1C(C)C)=O 8082,c1(C2(C(N3CCC(N(C)C(c4ccncc4F)=O)C3)=O)CC2)cccc(F)c1 8083,c1(C(=O)NCC(CCNC(c2ccc(OC)cc2F)=O)O)csc2ccccc12 8084,c1(C(=O)NC2COCCN(C(CN3C(C)CCC3C)=O)C2)c(O)nnc(C)c1C 8085,n1(CCC(=O)N(CCCNC(=O)Cc2cc[nH]c2)CC)ccnc1C(C)C 8086,c1(C(N2CC(C(=O)OCC)OCC2)C(=O)NC2CCC2)cc(F)cc(Cl)c1 8087,Cc1cc(C(N2CCC(CCC(=O)NCCCC3CCOC3)CC2)=O)[nH]c1C 8088,C1(NC(c2ccn(C3CC3)n2)=O)CN(C(c2cnn(C3CCC3)n2)=O)CC1F 8089,C(=O)(C1=NOC(C(C)(C)C)C1)NC1C(C)CN(C(C2CC2(C)Br)=O)C1 8090,C1(C(=O)NC2CC(NC(c3c(CC)sc(=N)[nH]3)=O)C2)C2CCCCCCC12 8091,C(c1nncn1C)=CC(=O)NCCN(C(C(CC)N(CC)CC)=O)CCCN(C)C 8092,C(CN=C(NCC(F)(F)C1CC1)NC1CCCC1)C1(COC)CCOCC1 8093,C1(CC(=O)NC)(CC(=O)NCC2C=CC(NC(C3CC(SC)C3)=O)C2)CCCC1 8094,c1(C(N(C2CCN(C(=O)C(CO)N(C)C)C2)CC)=O)cnn(-c2cccnc2)c1 8095,C1(OC)CN(C(C2(OC(C)C)CCOC2)=O)CCC1NC(c1sccc1C)=O 8096,c1(CCNC(=O)Nc2n(C)nc(C3CCC3)c2)nc2ccccc2n1C 8097,c1(C(N(CC(CC)NC(=O)CCC2CCCC2)CC)=O)nc(OC)ccc1C 8098,Cc1cc2[nH]c(C(N3CCCCC3C3CCN(c4nnn(C)n4)C3)=O)cc2s1 8099,c1(CC)nn(C)cc1C(=O)NCC1CCCC1NC(=O)COc1ccsn1 8100,C1(CC)CN(C(C2CC2c2nc[nH]n2)=O)CCN1C(=O)Cc1ccc(C)o1 8101,Cc1ncccc1C=CC(=O)N(C)CCOCCCN(C)C(C1CCOCC1)=O 8102,N1(C(C(C(C)OC)N(C)C)=O)CCC(CNC(=O)CC2OCCCO2)CC1C 8103,C1(NC(C(C)NC(N)=O)=O)C(C)(C)C(NC(C2SCCCS2)=O)C1(C)C 8104,C12(C(=O)NCCOC3CN(C(C4(CC#C)CCC4)=O)C3)CCCCN1CCC2 8105,N1(C(c2[nH]cc(C#N)c2)=O)CCC(CNC(c2cccnc2C(F)F)=O)C12CC2 8106,CC1(NC(=O)CC(F)(F)F)CCC(NC(c2cnc(-c3ccccc3)[nH]2)=O)CC1 8107,c1(C(=O)NCC2N(C(C(C)SC)=O)CCCC2)ccc(NC(C)=O)cc1OC 8108,S(=O)(=O)(c1cc(F)ccc1F)NS(CC1Cn2c(C)nnc2CC1)(=O)=O 8109,N1(C(C(CC=C)(F)F)=O)CCN(C(c2ccccc2SCC(N)=O)=O)CC(O)C1 8110,N1(Cc2onc(C)c2NC(=O)CC2COCCO2)CCCOC(CCN(C)C)C1 8111,C(=O)(CCCC(=O)CNC(c1cc(OC)ccn1)=O)OC 8112,c1(C(=O)NCC(C2CC2)NC(COC(CC)(C)C)=O)cccc(CNC(C)=O)c1 8113,c1(C(N(C2CCC(NC(CSC)=O)CC2)C)=O)ccc(=O)n(CCF)n1 8114,N1(C(c2c(CCC)cccc2)=O)CC(NC(=O)CCn2cccn2)CC(O)C1 8115,O=C(N1CC(O)CCO1)NCc1ncc(Br)cc1Cl 8116,c1(OC)ccc(CC(=O)NCC(C)CNC(=O)C(O)C2CCC2)c(Cl)c1 8117,N1(C(c2ccn(CCC)n2)=O)CC(C2(NC(=O)CC3CCCSC3)CC2)C1 8118,C(C(C)(C)CC(F)(F)F)(c1nnnn1C1CCC1)NCC(C(C)C)CO 8119,CC1CN(C(=O)C(C2CCN(C(c3[nH]ccc3C3CC3)=O)CC2)C)C(C)C1C 8120,C1(CNC(=O)CC(C2CC2)NC(C2(C(F)(F)F)CCC2)=O)CC2CC1CC2O 8121,C(C)(N=c1[nH]c(Cl)ncc1F)C1OCCN(C(C(CCC)CCC)=O)C1 8122,C=Cc1cc(C(=O)NCC2(NC(c3c(CSC)noc3C)=O)CCC2)cc(F)c1 8123,C=CCC(C1CC1)NC(C1CCN1C(=O)CSC1CC1)=O 8124,C1(NC(CC(=C)Br)=O)CN(C(c2cccc3c2CCN3)=O)CC2(CCC2)C1 8125,N1(C(CCC2C(C)C2)=O)CCOCC1CCNC(C1CN(C)C1)=O 8126,N1(C(C2CCN(C(C)=O)CC2)=O)CC(Nc2ncnc(Cl)c2CO)CC(C)(C)C1 8127,c1(CCC)c(C(=O)NCCN(CCOC)C(C2CCOC2C2CC2)=O)cnn1C 8128,C1(C(N(C2CC3CC(NC(=O)C(=O)NCC4CC4)C3C2)C)=O)CCC2CC1CO2 8129,N1(C(C2N(C(c3coc(C(F)F)c3)=O)CCC(=C)C2)=O)CCC12CCCSC2 8130,C=CCC(C(=O)NCC1(C(C)(C)C)CCN(C(=O)CCCCCC)C1)C(C)C 8131,CP1(=O)CCCC(N=c2[nH]c(=NCCCCc3ncc[nH]3)c3c(F)cccc3[nH]2)C1 8132,C#CC1(NC(C2(CNC(=O)C(C)Cn3cccn3)CC3(CC3)C2)=O)CCCOC1 8133,C1(C(=O)NC2C(C)N(C(=O)COC3CC=CC3)CC2)CC2(CC2)CN1C 8134,C12(C(=O)NCCN(C(C(C)OCC)=O)CC3CC3)COC(CC3CC3)(C1)C2 8135,c1(N2CCC(COC)CC2)nc2ccccc2nc1N1CCOC(C)CC1 8136,N1(C(c2ccc(SC)o2)=O)CC2CCCC2(CNC(=O)CC2CC=CCC2)C1 8137,C#Cc1ccc(C(=O)NCC2CC(CNC(c3ccc(C)cn3)=O)CO2)cn1 8138,c1(C(N(CCN(C(C(C)OC)=O)C)C)=O)ccnn1C1CCC1 8139,C1(C(=O)NCCCOC)CN(Cc2c(F)cc(F)cc2Br)CCC1(F)F 8140,C(CCC(C)(F)F)N(C(Cc1cccc(F)c1)C(=O)NC1CC1)C 8141,CCCC(C)CCNC(=O)CCNC(=O)C(C)(C)C1CCOC1 8142,c1(C(=O)NC2(CNC(C34CC3CCC4(F)F)=O)CCC2)cccc2ccccc12 8143,C=C(I)N=c1cccc(S(=O)(=O)NC2CCN(C)C3CCCC23)[nH]1 8144,Cc1cc(-n2cc(CSCCNC(=O)CC3CCC(C)(C)CC3)nn2)ccc1N 8145,c1(NCC(C)(C)C2CCCC2)ccc(C(=O)Nc2n[nH]cc2N2CCCC2)cn1 8146,C12(CNC(c3cc(C)on3)=O)CCC(CC1)N(C(c1cc3ccccn3c1)=O)C2 8147,c1(C(=O)NCCN(C)C(C2CC(S(C)(=O)=O)C2)=O)ccc(N)c(Cl)n1 8148,Cc1ccnc(NC(=O)C(C(C)C)NCCC2CC3CC3O2)n1 8149,c1(C(N(CC(C)CNC(C2C(C)(C)C2(F)F)=O)C)=O)cn2cccnc2n1 8150,c1(CC(=O)NCCc2ccc(CNC)cc2)c[nH]c2cccc(C)c12 8151,n1(C(=O)NC2(C)CC(NC(=O)COc3ccc(F)cn3)C2)ncc2cccnc12 8152,C1(NC(CC2(C)CCCCC2)=O)Cc2ccccc2N(C(=O)C=CC(N)=O)C1 8153,CC1CCSCCN1CC(=O)Nc1ccc(Sc2cccc(F)c2)cc1 8154,C1(C(=O)NCC(C)CN(C)C(C2(O)CCSC2)=O)CC2(CCC2)C1 8155,C(C)(C)(CC(=O)NC(c1ccc(F)cc1)CNC(=O)CSC1CC1)SC 8156,n1(CC)ccc(CNC(=O)C(C)N(C(=O)CCC2(C)CC2)C2CC2)n1 8157,N(C1CCCc2occc21)C(C(CC)N(C(=O)C(C)N=[N+]=[N-])C)=O 8158,c1(OC)ccccc1C(CNC(=O)CCC(C)SC)NC(C12CC(CO1)C2)=O 8159,N1(CC(=O)NC2CN(C(CCCc3nnc(C)n3C)=O)C2)CCc2sccc2C1 8160,c1(CC(=O)NCC(CN(C(CCC(CC)C)=O)C)C)ccc2c(c1)ncn2C 8161,Cn1c(O)nc2cc(C(=O)Nc3cc(Cl)cc(Br)c3F)ccc2c1=O 8162,CCCC(C)N(CCC(=O)NCC1(CC2CCC2)CC1)C 8163,C12(NC(C3CC(C)OC3)=O)CCCCCC1N(C(c1cc(O)ccc1N)=O)CC2 8164,c1(C(=O)NC(CC)CNC(=O)Cc2cncnc2O)ccnc(Cl)c1Cl 8165,N1(C(CC2(C=C)CCCCC2)=O)CC2CCN(C(C3SCCS3)=O)C2C1 8166,c1(-c2cn(CC(=O)NCC3(O)CC3)nn2)ccc(C(F)(F)F)cc1 8167,C(=O)(C(CC)C(=O)N1CCCC(NC(=O)CCCc2ccc(C)cc2)C1)OCC 8168,N1(C(Cc2nnc(C)o2)=O)CCN(CCNC(=O)C=Cc2cncs2)CC1 8169,c1(C(=O)NC23CN(C(C(CCCC)C)=O)C(CC2)CC3)c[nH]c2c(F)cccc12 8170,C1(C(=O)NC(COC)C)C2CC3C(C2NC(c2cc(C)nnc2C)=O)C13 8171,N1(C(CN(C2CC2)CC)=O)CC2(C1)CN(C(=O)CCC1CCCO1)C2 8172,Cc1c[nH]c2ncc(C(=O)NCC3(CNC(=O)CN4CC5CCC4C5)CC3)cc12 8173,C=CC(C)(C)C(=O)N(CC(O)CN(C)C(C1(CC)CCOC1)=O)C 8174,C12(NC(=O)CCF)CCCC1CN(C(c1ccc(-c3ccsc3)nc1)=O)C2 8175,c1(C(=O)NC2CCC(NC(C3(SC(C)C)CC3)=O)C2)cccnc1NC1CC1 8176,c1(C(=O)NC2C(CNC(=O)CCF)COC2)ncccc1C1CC1 8177,c1(OC)ncc(C(=O)NC2(CN(C)C(c3ccn(C)c3)=O)CC2)cc1C 8178,C1(C)(C(=O)NCC2CC(NC(c3n(CC)ccc3)=O)C2)CCC(=O)N(C)C1 8179,CC1CN(C(=O)COC2CCC2)CCCN1C(C1C2COCC12)=O 8180,C1(N(C(Cn2nnc(=N)[nH]2)=O)CCO)CCN(C(=O)CC2CC(OC)C2)CC1 8181,c1(CC)nc(OC(C2CN(C(=O)COCC3CCCC3)C2)C)cc(C)n1 8182,C1(NC(c2coc(Cl)n2)=O)CCC2(CC1)CCN(C(c1ccc(I)c(O)c1)=O)C2 8183,C(C)(N=c1[nH]c(=N)[nH]c(=NCC(C)C)[nH]1)c1c(OC)cc(F)c(OC)c1 8184,c1(C(=O)NC2C(NC(C(C)Sc3nc[nH]n3)=O)CCC2)cccc(C(F)(F)F)c1 8185,C1(C(N2CCC(O)(CNC(C=C(C)Cl)=O)CC2)=O)CC1C1CC(F)(F)C1 8186,N1(C(c2cnc(CCC)s2)=O)CC(NC(=O)C(C)(CC)CO)C(C2CC2)C1 8187,CC1(C)COCCN(C(C2CC(O)CN2C(C2(C)CC=CCC2)=O)=O)C1 8188,Cc1nnc2n1C(C(=O)N1CC(C)(NC(C3CCc4nccn4CC3)=O)C1)CC2 8189,C1(C(=O)NC(C(=O)OCC)CC)CN(C(C2(Cl)CCC2)=O)CC12CC2 8190,C1(NC(C=CCCC)=O)CCC2(CCN(C(C3(C)CCCC3O)=O)C2)C1 8191,C1(O)(CNC(c2n(C(CC)C)ncc2)=O)CCN(C(C2CCCOCC2)=O)CC1 8192,Cc1cnn(C)c1C(=O)NCC=CCNC(C1CCCN(c2ncccn2)C1)=O 8193,C1(NC(=O)CBr)CCC(CNC(C2(n3cccn3)CC2)=O)C1 8194,C(C(C(=O)N(C)CC1CCN(C)C1)C(C)(C)C)NC(C(C)(C)SC)=O 8195,c1(OC)nc(C)cc(C)c1-c1noc(C2CCCN(C(C)=O)CC2)n1 8196,C(C)(C)(CCCC(=O)Nc1cnn(C)c1C)NC(C1CCC(CC)O1)=O 8197,C12(C(=O)NC3CCN(C(CC(C=C)C)=O)C3C)CCC(CC1)C(C)O2 8198,C1(NC(=O)CN2CCCC2=O)CC2CC1N(C(c1nccc(F)c1Cl)=O)C2 8199,c1(SCC(=O)NCC(C)NC(c2ccc(OCCF)cc2)=O)ccc(O)cc1 8200,N1(C(CC=C(C)C)=O)CCC2(CC1)C(NC(=O)CCC(C)N(C)C)CS2(=O)=O 8201,N1(C(=O)NC2CN(C3CCCCC3)C2)CCC(C2CCCC23OCCO3)C1 8202,c1(CC)c(C(C(=O)NCc2nnn(C)n2)N(CC(C)CO)C)cccc1C 8203,N1(C(c2coc(Br)n2)C(=O)NC2CC(C(=O)OC)C2)CC2CC1CS2=O 8204,N1(C(C(CC2CCC2)NC(C(OC)OC)=O)=O)CCCN(CCO)CC1 8205,Cc1cc(C(N2CC=CCC2C(N2CC=CC2)=O)=O)[nH]c1C 8206,CC(C)(C#CC(=O)N1CC(O)C(C)(C)C1)CNC(C1CCC(=O)CC1)=O 8207,Cc1cc(C(=O)NC(C2CCN(C(c3ccccc3Br)=O)C2)C)ccn1 8208,c1(NC(CNC(C(N2CCC(C)C2)=O)=O)=O)c[nH]c2cccc(Cl)c12 8209,N1(C(CCC#N)=O)CCN(C2CCCC2NC(=O)CC(O)CC2CC2)CC1 8210,c1(COC)cc(C(N2CC=CC2C(=O)NCC(n2ccnn2)C)=O)n[nH]1 8211,C1(CCCC)(C(N2CCC(C(=O)OC)C2)=O)CN(C(C2CCC2C(=O)OC)=O)C1 8212,c1(C(=O)NCC2CCC(CC(=O)OC)CC2)cc2cccc(Br)n2c1 8213,C1(C(=O)NC(C)CC(=O)N(C)CCOCCCO)CC2CC(=O)C1O2 8214,C1(C(N(c2nccs2)CC)=O)CCN(Cc2ccc(F)s2)C1 8215,c12ccc(Cl)c3cc([nH]c13)CCOC2=O.C(C)(C)(C)OCCN(C)NC(=O)NC 8216,C1(CC(=O)NCC2(NC(C3CCC4(CCC4)O3)=O)CCCC2)CCC2(CCC2)O1 8217,C(=O)(CCC(=O)NCCC1COCCN1C(=O)Cn1cc(C2CCC2)nn1)NC 8218,C(C(C)(C)N=c1[nH]nc(C#N)s1)N(C)C(c1cc2c(=O)[nH]ccn2n1)=O 8219,C12(CN)CCCC1CN(CC1CC3(CO1)CN(Cn1ccncc1=O)C3)C2 8220,N1(C(c2ccc(NCC)cc2)=O)CCC2(CNC(=O)C(O)C(C)C)CCCCC12 8221,c1(C(=O)OC)cc(C)cnc1NC1CC(C)N(C(c2cnn(C3CCC3)c2)=O)C1 8222,C(CC(C)C)(C(=O)N1CCC(C(C)CO)CC1)N(C(CSCCC(C)C)=O)C 8223,N1(CC2C(C)(C)C(NC(=O)NCCc3ccccc3)CC2)CCC2(CC1)COC2 8224,C1(C(=O)NCCCC(C)NC(c2cccnc2OCCO)=O)CC(=O)OC1(C)C 8225,C(=O)(C1=C(F)CN(C(C2CC23CCOCC3)=O)CC1)NC(C#C)C(C)C 8226,c1(SC)cc(C(=O)NC2COCCN(c3ccnc(C)n3)C2)ccc1[N+](=O)[O-] 8227,c1(C(N2CC(c3ccccc3)C2(C)C)C(=O)NC(C)C)cc(C2CC2)ccc1F 8228,C1(NC(C2CCN(CC(C)C)C2)=O)CN(C(=O)CCCC2CC2)CC1O 8229,C1(CNC(c2c(C)cc(C)s2)=O)CCC12CCN(C(C1CCCOC1)=O)CC2 8230,N1(C(c2cc(I)cn2C)C(=O)NCCCC)CCOc2cccc(F)c2C1 8231,c1(C(=O)NCC(CCC)NC(c2sc(C)cc2OCC)=O)cnc(OC)cn1 8232,Cc1ccc(-n2cc(CC3CCN(C(C4C=CCCC4)=O)C3)nn2)cc1Cl 8233,c1(C(N(CCOC)CCNC(C2CN(c3nncs3)C2)=O)=O)cc(CO)n(C)n1 8234,Cc1c[nH]nc1C(=O)NC(C)CC(C)NC(=O)C(c1cncnc1)C 8235,C(=O)(C1=CCCCO1)NCCN(C(C1(O)CCN(C(=O)OC(C)(C)C)C1)=O)C1CC1 8236,c1(C(NNC(C2C(c3cn(C)nc3)OCCC2)=O)=O)c(F)ccc(Br)c1F 8237,C1(CCC(=O)NC2CCCC2CNC(C2CC(=O)N2)=O)CCCCO1 8238,C(=O)(CC(C)CNC(C1C=CCCN1C(=O)CSC(C)(C)C)=O)OC 8239,c1(C(n2cc(C3C(C)CCN3C(=O)C3=CCN(C)C3)nn2)C)cnc2nccn2c1 8240,Cc1cn(C)nc1C(N1CCC(CCNC(C2CCOC(C(C)C)C2)=O)CC1)=O 8241,C(=O)(C(C)(C)c1cccnc1)NCCN(CCC)C(c1nocc1C(C)(C)C)=O 8242,C1(NC(c2c(OC)csc2)=O)C2CC(O)C1N(C(=O)C=CC1C(C)C1(Cl)Cl)C2 8243,c1(C(=O)NCCCCCCNC(C2N(CC)CCC2)=O)[nH]c(=N)ccc1C 8244,CN1CCN(C)C(CN(C=O)Cc2ccc(-c3cccc(Cl)c3)o2)C1 8245,C1(C(N2CC(NC(c3cncnc3)=O)C(O)CC2)=O)CC2CC1CC2(F)F 8246,N1(C(c2c(CC)con2)=O)CC=CC(C(=O)NCC#CC2CC2)C1 8247,c1(CC(N2CCC(C(CNC(C(CC#C)C)=O)(C)C)CC2)=O)ccc(Cl)c(F)c1 8248,c1(C(N2CCC(C3N(C(COC)=O)CCC3)C2)=O)ncc(Cl)cc1Cl 8249,CC1COCC(C(=O)NC(C)(C(=O)NCC2(N(C)C)CCCC2)C2CCC2)O1 8250,C1(C(=O)NCCN2CC(=O)NCC2)C2CCC(C2)C1NC(C1CC(=C2CCC2)C1)=O 8251,c1(C(CCC)NCc2c[nH]nc2C(C)C)ccc(Cl)cc1Cl 8252,C(=O)(C(CNC(C1OCC2CCCC12)=O)CC(C)C)NC(CC)C(F)(F)F 8253,C(=O)(CCCC(C)(C)NC(=O)C(C#N)C(C)C)NC(CC#CC)CO 8254,c1(CN2CCC(O)(C(N3CCCCC(F)(F)CC3)=O)C2)cncc2ccccc12 8255,C=CCC(CC=C)C(=O)NC(C)(C)CCNC(c1cn(C)nc1C(F)(F)F)=O 8256,Cc1ccc(CCNC(=O)CCOCCCNC(C2CCOC2)=O)nc1 8257,CC1CCC(CNC(=O)CCc2ccoc2)CN1C(=O)COCC1CCCOC1 8258,O=S(=O)(CCN1Cc2ccccc2CC1CO)c1ccccc1 8259,C1(CNC(C(F)=CCC)=O)CC(NC(c2coc(CC3CC3)n2)=O)C1(C)C 8260,C(CC(C)(C)C(=O)NCC(c1ccccc1)CNC(C1(F)CC1C)=O)SC 8261,NC(CCOc1ccccc1)C(=O)NNc1nc(C(F)(F)F)no1 8262,C(CCC(C)(C)NC(=O)CC1CCC(C)C1)NC(CSc1nc(C)[nH]n1)=O 8263,C(CS(=O)(=O)CC(=O)NC(C1CC(NC(=O)CN2CSCC2=O)C1)C)OC 8264,N1(C(C2(C#N)CC(C)C2)=O)CCN(C)C(CNC(c2cncc(Cl)n2)=O)C1 8265,C(C(=O)NOC1CC2CCC1C2)(c1ccco1)NC(C1CC1(Cl)Cl)=O 8266,C1(NC(CCC=C)=O)CC2CCCC(C1)N2c1cc(SC)ncn1 8267,C1(NC(CC2CC(SC)C2)=O)C=CCN(C(c2ccc(C)cn2)=O)C1 8268,CCCCC(C(=O)NCC1CCCN(C(c2ncccc2CO)=O)CC1)C(C)C 8269,C(CCCCCCCO)=CC(=O)NC1CN(C(C(CN(C)C)(C)C)=O)CC2C1C2 8270,C1(NC(C2(CC)CCC2)=O)CN(C(c2ccc(C(N)=O)cn2)=O)CC1C 8271,c1(C(N2CCCC(O)(CNC(C(C(C)C)C#N)=O)C2)=O)sc2cccnc2c1Cl 8272,N1(C(C(C)O)=O)CCCC(C2CCCN(CCCOc3cccc(Cl)c3)C2)C1 8273,C1(C(=O)NCC=CCNC(C2(CC)CCOC2)=O)CC2(C1)CC(C)C2 8274,C1(C(N2CC(C(C)OC)C2)=O)(CCNC(=O)C(C)C2CC2)CCCC1 8275,c12cccnc1C(=O)NC1CC(C)(C1)CN2.C(C)(C(=O)NC(C)(C)C)NC(C)=O 8276,c1(OC)cc(OC)cc(NC(=O)NCCC2CCN(CC(C)O)CC2)c1 8277,C1(NC(CN(C(COC)=O)C)=O)CC(F)CN(C(=O)C(F)(F)CO)C1 8278,c1(CCNC(C(N2CCC(C(N)=O)CC2)c2cn(C)nn2)=O)cccc(F)c1 8279,C1(CNC(C2(CCC=C)CC2)=O)CC2CC1CN2C(=O)COC(C)CC 8280,c1(C(=O)NC2CC3(C2)CN(C(=O)COCC2CC2)C3)cc2cccc(F)c2s1 8281,CN1CCC(=CC(=O)NCC2CCN(C(=O)CC3CCC(=O)N3)C2)CC1 8282,C(=O)(C(C)(C)C(F)F)N(CC(C)(C)NC(C1CC12CC2)=O)C 8283,c1(C(N2C(C)CN(C(C3CCCC(=O)N3)=O)CC2)=O)ccc2ccccc2n1 8284,N1(C(C2CN(C(c3c(C)nsc3C)=O)CC2C)=O)CCCc2occc2C1 8285,C1(CNC(C(C)OC)=O)Cc2ccccc2CN1C(=O)C(N)=O.C(CCCCC)N 8286,C12(NC(C3SCC=C3C)=O)CC(NC(COCCOCCOC)=O)(C1)C2 8287,C1(CNC(C(CSC)(F)F)=O)CC2CCC(C1)N2C(c1cccc2c1COC2)=O 8288,Cc1ccsc1CC(=O)NCC1C=CC(NC(=O)C(O)CC2CCCCC2)C1 8289,c1(OCC)ccc(-c2nc(C3CCCC(n4cccc4)C3)n(CC)n2)cn1.C1(C)CC1 8290,C(C(CC(F)(F)F)NC(C1(O)CC1)=O)NC(c1nc(CC(C)C)sc1)=O 8291,N1(C(C2(COC)CCCO2)=O)CCC(n2cc(C3CCCCC3O)nn2)CC1 8292,N1(C(CN(C2CCC2)C)=O)CC2CCC2(CCNC(=O)C=Cc2nccs2)C1 8293,c1(C(N2CCC(CN(C)C(c3ccnnc3O)=O)C2)=O)cncc(C(C)(F)F)c1 8294,N(C(=NCCC(C)SC)NC1CC1NC(=O)OC(C)(C)C)C1CC(OC)C1 8295,Cc1ccc(CC(=O)NCC23CC(CO2)N(C(C2CCC(C)C2)=O)C3)cc1C 8296,C1(C#N)(C(=O)NCCC(=O)NCC2N(C(CSC)=O)CCCC2)CCCOC1 8297,C1(CC(=O)NC(C)C(C)n2cccn2)C(NC(=O)Cc2cncs2)CC1O 8298,N1(C(c2n(CC#C)cnn2)=O)CCC(C)C1C(=O)NC(C)(C)C#CCC 8299,c1(CC)ccc(C)c(C(N2CCC(CCNC(C3SCC=C3C)=O)CC2)=O)c1 8300,c1(C(=O)NC2C(CNC(c3ccc(O)cc3)=O)C2)cccc(Cl)c1[N+](=O)[O-] 8301,C1(CC(=O)NC)CCCN1C(C1(C(=O)OC(C)(C)C)CCC1)=O 8302,c1(OC(F)F)ncc(CN2CCOCC2Cn2cccn2)cc1F 8303,N1(C(CCCc2c(C)ccs2)=O)CCC(C)C1CNC(c1ccccc1CO)=O 8304,Cc1cnc(C(=O)NC2C3CC4C(C3)C24C(=O)NC(C)Cc2nc[nH]n2)c(C)c1 8305,c1(C(N2CCC(CC)C2CNC(C2CC2(C)C)=O)=O)ccc(F)c(Cl)c1 8306,N1(C(c2cc(C3CC3)ccn2)=O)CC2OCCN(C(c3sccc3Cl)=O)C2C1 8307,N1(C(CCOCC(C)C)=O)CCC(O)C1C(=O)N(C)CCOC(F)F 8308,C(CC(CC)(CC)NC(c1ccnc(OC)c1)=O)NC(C(C)OCC=C)=O 8309,N1(C(c2ccc(CNC(C(CCCC)F)=O)o2)=O)CCC2(CCCOC2)C1 8310,c1(C(=O)NCC(CC)NC(c2oc(C3CC3)nc2C)=O)cnc2c(c1)CCOC2 8311,C1(CNC(=O)NC(C(C)c2ccccc2)(C)C)CC(C)(C)CO1 8312,C12(C(=O)NCC(C)(C)N(C)C)CC(CCO1)N(C(=O)CN1CCNC1=O)C2 8313,C(=O)(C(C(=O)N1CC2CC(C1)N(C(c1cccc[n+]1[O-])=O)C2)C(C)(C)C)OCC 8314,c1(C(N(C2CCCC(N(C(=O)C(F)F)C)C2)C)=O)ccnc(-c2ncc[nH]2)c1 8315,c1(C(=O)NCC2C3CN(C(CCC(=O)NCC)=O)C(C3)C2)csc2c1CCCC2 8316,N1(C(C2(OC)CC(C)C2)=O)CCN(C(=O)CCn2nc(C)cc2C)CC12CCC2 8317,C(=O)(CS(=O)(=O)NC(C)(C)C)NC1(CO)CN(C(C(=O)NCC)C)C1 8318,C1(CNC(CC2(C)CC2(Cl)Cl)=O)C2CN(C(c3ccc(C(N)=O)nc3)=O)CC12 8319,N1(C(C2OCCN(C)C2=O)=O)CCC2(CCC2)C(NC(c2ncccn2)=O)C1 8320,c1(OC)c(C(N2CCCC(CCNC(=O)C(O)P(C)(C)=O)C2)=O)cccc1Cl 8321,C1(C(=O)NC(c2ccc(O)nc2)C)CC(NC(C2(C)CNC(=O)C2)=O)C(O)C1 8322,c1(C(=O)NC2CCN(C(CCCCNC(N)=O)=O)C2)ccc(N)cc1C(F)(F)F 8323,C1(CNC(C(C)OCCC#C)=O)CN(C(=O)Cc2csnc2C)CCC1(F)F 8324,C(=O)(CC(C)(C)C#N)N(CCC(C(C)C)NC(c1cc(C2CC2)ns1)=O)C 8325,N1(C(C(C(C)C)SC)=O)CC2(CCCN(C(=O)C(c3nc(C)cs3)C)C2)C1 8326,N1(C(CC(C)n2cccn2)=O)CCCC(CC(=O)NCc2ccc(Cl)cn2)C1 8327,C1(NC(C(C)N(C(=O)CC2CCOC2)CCC)=O)CCc2c[nH]nc2C1 8328,C(=O)(CC(C)(C)CC(=O)NCC(C)NC(=O)C(c1cc(C)ccc1C)C)OC 8329,N1(C(c2ncsc2C(F)(F)F)=O)CC2(CCN(C(C3(O)CC4CCC3C4)=O)C2)C1 8330,CC(C)C(O)CC(=O)NCC1CN(C(=O)CCNC(N)=O)CC1C(F)(F)F 8331,CC(C)CC(O)C(C)C(=O)N(C)CCOCCNC(=O)CCC(F)(F)F 8332,C(=O)(C#CC(C)(C)CNC(c1c[nH]cc1C(C)C)=O)NCc1n(CCC)ncn1 8333,N1(C(C(C)c2ccsc2)=O)CCCC(CO)(NC(=O)CO)C1 8334,C1(NC(CNC(N)=O)=O)CN(C(=O)COCc2ncc[nH]2)C2(CCOC2)C1 8335,CC(C(=O)NCC1CCC1C(N1CCN(C)CC1C1CC1)=O)C(C)(C)C 8336,C(=O)(CN=c1cc[nH]cc1)NC1(C)CC(C(N2CC[Si](C)(C)C2)=O)C1 8337,c1(CNC(C(=O)NCCc2cccc(OCCO)c2)=O)cc2cccnc2[nH]1 8338,Cc1cc(Br)cc(C(=O)NC2CC(NC(=O)CCS(C)=O)C2)c1F 8339,C1(C(=O)NC(C2CCN(C(=O)C(F)=CCCF)CC2)(C)C)CC2(CC2)CO1 8340,Cc1onc(Br)c1C(=O)NC1CCC1NC(=O)CC1CCN(C)C1=O 8341,N1(C(=O)CCCCBr)CC2CN(C(C3(c4ccc(F)cc4)CC3)=O)C2C1 8342,N1(C(c2n(C=C)ncc2)=O)CCCC2(C1)CN(C(C1CN(C)CC(C)O1)=O)C2 8343,c1(C(C)=O)ccc(NC(=O)CC2CC(NCCc3c(Cl)cccc3Cl)C2)c(Br)c1 8344,C1(C(NOCC=C(C)C)=O)CCC(NC(C2C=CCCC2)=O)CC1 8345,CC1CN(C(c2cc(C(F)F)cs2)=O)CC(C)CN1C(c1ccc(N)c(N)n1)=O 8346,CCCCCC(C)CC(=O)NC1CCN(C(c2cccc3c2CCC3)=O)C1(C)C 8347,C1(C(N2CC(C(N3CC(COC(C)=O)C3)=O)OCC2)=O)CC2(CCC2O)C1 8348,NC1CCC2(CC1)CN(Cc1cn(CCc3cccnc3Cl)nn1)C2 8349,CCCCC(CC)CC(=O)NC(C)C(CO)NC(=O)C(C)CC(C)C(C)=O 8350,c1(OC)cc(OC)cc(CC(=O)NC2(CN(C)C(C3COC(C)C3)=O)CC2)c1 8351,c1(NC(=O)NC(C=C)C)ccncc1-c1cccc(C(=O)NC)c1 8352,c1(C(=O)NCC2CCCN2C(C2CC2c2cnc[nH]2)=O)ccc(C(F)(F)F)cn1 8353,CN1CCC2CN(C(C3CCN(Cc4nc(Br)cs4)CC3O)=O)CC12 8354,c1(C(=O)NC2CC(C(=O)NC(CCCC)CO)OCC2)ccc(=NC)[nH]c1 8355,CCC(O)C(C)C(=O)NCCC1(OC)CN(C(C2CC2F)=O)C1 8356,CC1(C)Cc2cccc(C(N3CC(NC(=O)C=Cc4ncc[nH]4)C(O)C3)=O)c2O1 8357,CCC(C(=O)NCCCCCN(C(=O)C(C)c1cccs1)C(C)C)C(C)C 8358,N1(C(=O)OC(C)(C)C)C(CCNC(c2c[nH]nc2C(F)(F)F)=O)COC1(C)C 8359,C1(C(N2C(CN(c3nn(CC)c(C(F)(F)F)c3)C)CCC2)=O)CC(C2CCC2)C1 8360,C1(OC)CC2(C1)CC(C(=O)NCC(c1ccc(C)cc1)NC(=O)C(O)C(C)C)C2 8361,n1(CC)cc(C(=O)NCC2CC(NC(C3CC3C3CC3)=O)C2)c(C(C)C)n1 8362,c1(C(=O)NCC2(COC)CCCN2C(=O)C(C)NC(N)=O)c(F)ccc(N)c1F 8363,c1(C(=O)NCCCCCN(C(C(COCC)C)=O)C)cc(OC)n(C)n1 8364,Cc1cc(C(=O)NC2CC(CCNC(C3(O)CCC(C)CC3)=O)C2)nc(C)n1 8365,c1(C(N2CC(O)(CNC(C3CC4CCC3O4)=O)C2)=O)cc2n(n1)CC1(CC1)C2 8366,N(C(=NCC(=C)C)NC(C)COC(F)F)C(c1ccccc1)C#C.CCCC 8367,C(=O)(C1OCCc2c(Br)cccc21)NC1(CNC(c2cocn2)=O)CC1 8368,O=C(C1CCc2ccccc21)N1C2CC1CN(Cc1c(Cl)cncc1Cl)C2 8369,Cc1cc(C(=O)N(CC(C)O)CCNC(=O)CCC2CCCN(C)C2)cc(Cl)c1 8370,c1(CC)occc1C(=O)NC(C(=O)NCCC(O)C1CC1)C1(C)CC1 8371,C1(CNC(COCCCC(C)C)=O)(NC(=O)Cc2csnn2)CCCCCC1 8372,Cc1cc(Cc2cnc(N(C3CCNCC34CC4)N(C)C)cc2C)nc(C)c1 8373,N1(C(c2ccc(CSC)o2)=O)CCC2(CC2NC(=O)CCCCN(C)C)C1 8374,N1(C(c2c(CC)nc(C)nc2)=O)CC2CC(NC(=O)Cc3csc(C)c3)CC2C1 8375,c1(C(N2CC(CNC(C(CC)C)=O)OCCC2)=O)cc(Br)c(F)cc1F 8376,c1(C(=O)NCC(C)NC(=O)C(c2ccc(Br)cc2)O)cc2c[nH]nc2s1 8377,c1(C(N2C3CCC(CNC(CC(C)O)=O)(C3)C2)=O)cnn2c1OCCC2 8378,CCC(=O)CCC(=O)N1CC=CC1(C)C(=O)NC1CNC(=O)C1(C)C 8379,C=CC1(CC(N2CCC(C)C2CNC(c2cc(C)cc(C)c2)=O)=O)CCCCC1 8380,C1(CC(=O)NCC2(C=C)CCC2)CN(C(C2CCC2(F)F)=O)CC12CC2 8381,C1(NC(c2cc(C(=O)OC)sc2)=O)CC12CC(NC(=O)Cc1cnn(C)c1)C2 8382,O=C1CCC(C(=O)NCC2(C(F)F)CCN(C(=O)Cc3cccnc3Cl)C2)CN1 8383,Cc1ccc(Cl)cc1NC(=O)C(=O)NC1CC1NC(C1C(C)(C)C1(C)C)=O 8384,C1(C(N(CCNC(CC(C=C)C)=O)C2CC2)=O)CC1C1CCOCC1 8385,CCCC(C)(CCC)C(=O)NC(C)CN(C(=O)Cc1ncoc1C)C 8386,CC(CS(C)(=O)=O)NC(c1ccc(CNC(C2CCN(C)C2)=O)nc1)=O 8387,c1(C(N(CCNC(C(CCC)C(C)C)=O)CCC)=O)cnc2ccccn2c1=O 8388,C1(C2CCN(C(C3CC34CC(C)(C)C4)=O)C2)(NC(C(C)OC)=O)CC1 8389,N1(C(C(C(C)C)C)=O)CC2(CCCCN(C(=O)C(C)(C)C(C)(F)F)C2)C1 8390,Cc1ccc(Br)c(C(=O)NCC2(F)CN(C(C3OCCCO3)=O)C2)n1 8391,N1(C(c2cn(CCC)nc2C)=O)CCC(NC(c2ncccc2C)=O)CC1C 8392,CC(C)(C)C(C(=O)N1CC(CNC(=O)CC2CSC2)C(C(F)(F)F)C1)NC(N)=O 8393,c1(OC)ccc(NC(=O)C(C2CN(C(=O)CC3CNC(=O)O3)C2)SC)cc1C 8394,c1(CNC2CC(CC(=O)Nc3ncc(Br)nc3I)C2)ccc(Br)c2cccnc12 8395,Cc1cc(C(=O)NC(CNC(=O)C=CC2CC2)C2CCC2)cn(C)c1=O 8396,N1(C(C(=O)NCc2cc(OC)c(C(C)(C)C)cc2)=O)CCC2(CNC(=O)C2)C1 8397,C1(NC(c2csc3nnsc23)=O)CCCCCN(C(C2CCCCC2)=O)C1 8398,CCCCCCCCS(=O)(=O)NC1CCN(S(=O)(=O)CCC(=O)OC)CC1(C)C 8399,c1(COC)cc(C(=O)NCC(=O)NC(c2ccccc2)(C)C)n[nH]1 8400,C1(C(=O)NCC(COC)NC(=O)CC(C)F)CCC2CC1CO2 8401,c1(OC)cnc(C(N2CC(F)(C(=O)NCc3ccc(C)cc3OC)C2)=O)c(F)c1 8402,C(CCCCNC(=O)CC(C1CC1)NC(C1(F)CCOC1)=O)N(C)C 8403,C=CCC(CC=C)C(=O)NCC1CCC1NC(C12CCC(CC1)CO2)=O 8404,c1(C(C)C)cncc(C(N2CCC(F)CC2)C(=O)NC2CCOCC2)c1 8405,c1(CNC(=O)NCc2ccc(CNC(C)=O)cc2)ccc(S(C)=O)cc1 8406,C1(C(N2C(CC(=O)O)COCC2)=O)C2CCC1C(F)(F)C2 8407,C(=O)(C1CS(=O)(=O)c2ccccc21)N(CCN(C(C(CC)C#N)=O)C)C 8408,C1(=CCNC(C2CC=CCC2)=O)CCN(C(c2cccnc2C(F)(F)F)=O)CC1 8409,C(=O)(C1=C(Cl)CCOC1)NCC1C(C)CN(C(=O)Cn2nccc2N)C1 8410,C12(C(N3CC(O)(CCNC(C(C4CCOC4)OC)=O)C3)=O)CCC(CC1)CO2 8411,c1(CNC(N(C2CCC2O)CC)=O)csc(C2CCCO2)n1 8412,C(CCC(C)C)=CC(=O)N(CC(CNC(C(C)OCC=C)=O)C)C 8413,CC(C)CC(C)(O)c1cn(C2(C(=O)NCC3CCCC3(F)F)CC2)nn1 8414,N#CC1(C(=O)NCc2nc(C(N3CCC(C(F)F)CC3)=O)co2)CCCOC1 8415,C1(NC(CC(n2c(CC)ncc2)C)=O)CCN(C(=O)C2=CCCOC2)C(C)C1 8416,C(=O)(C1=CC2C=CC(C1)C2)NCC(CC(C)C)NC(c1ccccc1C(N)=O)=O 8417,c1(C(N2C3CCN(C(COCCCOC)=O)CC3C2)=O)cnc2c(c1)CCCO2 8418,CCCC(C(O)C(=O)NCC1CC(O)C12CCC2)NC(c1cc(C)[nH]c1C)=O 8419,Cc1noc(N)c1C(=O)NCC(C)C(=O)NC(c1cncc(F)c1)C 8420,c1(C(N2CCCC(CNC(C(C)OCC=C)=O)C2)=O)c(OC(F)F)cccc1Cl 8421,c1(NC(=O)NCCC(N2CCOCC(N3CCCC3)C2)=O)nc2ccccc2s1 8422,c1(C(N2C(C)(C(=O)NC(CCOC)C(C)C)C=CC2)=O)cc(C)cc(O)n1 8423,N1(C(c2n(C3CN(C)C3)ccc2)=O)CC(NCc2nc(C3CC3)cs2)C2(CC2)C1 8424,c1(OC)ccccc1C(C)C(=O)N(CC(C)CNC(c1nocc1C)=O)C 8425,N1(C(C(=O)N(C(C)CO)CC=C)C)CCC(C(=O)Nc2ccco2)CC1 8426,C1(=O)CS(=O)(=O)CCNC(=O)NCCN1CCOC.CCC(C)C(=O)C(=O)OCC 8427,N1(C(CCN(CCCCC)C(C)C)=O)CC(NC(=O)Cc2ccccc2)C(O)C1 8428,C1(c2cn(CC(O)CNC(=O)C3CC3)nn2)CCN(C(C)(C)C)CC1.CC1(C)CC1Cl 8429,C12(NC(Cc3cn(CC)nc3C)=O)CCCC1CN(C(C1(CC)CCCO1)=O)C2 8430,C1(CC(=O)OC(C)(C)C)CCCN(C(c2cnsn2)=O)C1 8431,C1(CNC(C2CC3C=CC2C3)=O)CC2(CC2)CN1C(=O)COc1ccc(Cl)nc1 8432,Cc1cc(S(=O)(=O)NCCCN2C(=O)CNC2=O)sc1C 8433,CCCCCC(F)C(=O)N1CC(CC(F)C(=O)NCCN2CCC(CO)C2)C1 8434,C(=O)(CC(C)P(C)(C)=O)N1C(CN(C)C(C2(N3CCCCC3=O)CC2)=O)CCC1 8435,O=S(=O)(N(CC(O)C1CCC1)C1COC1)N1CCN(CC(F)(F)F)CC1 8436,N1(C(c2nnc(CC)s2)=O)CC(NC(=O)C(C(C)C)N2CCCCC2)C(C)C1 8437,n1(CC)ccnc1CNC(c1noc(C)n1)c1nnnn1C1CCCC1 8438,N1(C(C=NOC)=O)CCN(C(=O)CCc2ccc(Cl)nc2)CC1CC(F)(F)F 8439,N1(C(C(C)SCC)=O)CC2CN(C(=O)C=Cc3cccc(Br)c3)CC2C1 8440,c1(C(CNC(C=CC(C)NC(=O)CNC(=O)CN(C)C)=O)C)ccccc1 8441,N1(C(C(CC(N)=O)NC(c2cc(CC)ncn2)=O)=O)CCCC2(C)CCCC12 8442,c1(C(=O)NCC23CC(NC(C4CCCO4)=O)(C2)C3)ccc2ccsc2c1 8443,C1(CC)C(C(N2CC(C(C)NC(c3ccc(SC)o3)=O)C2)=O)CCN1C 8444,Cc1ccc(C)c(C(=O)NC2CN(C(c3nnn(C)c3C)=O)CCC2F)n1 8445,C1(C(N2CC(C(N3CC(CCNC(C4C(=C)CC4)=O)C3)=O)C2)=O)CCCCC1 8446,CC#CCCC(=O)NCCCCCN(C(=O)CC(c1ccccc1F)C)C 8447,C(CCCCN=c1[nH]c(=N)[nH]c(=NC2CCCN(CC)C2)[nH]1)OC 8448,C(=O)(C#CC1CCOC1)N1CCC(CCNC(C2CCCN(CCF)C2)=O)CC1 8449,C1(COC)(NC(C2(C)C=CCC2)=O)CN(C(c2ccn(C)c2)=O)C1 8450,c1(NC(=O)NC(C)Cc2cncs2)cc(Cl)ccc1OCC(=O)C1CC1 8451,N1(C(CCCSC)=O)CC2(CCC2)CC1CNC(C1CCCCC1N=[N+]=[N-])=O 8452,N1(C(c2ncc(N)nc2)=O)C2CCC1CN(C(C1CCN1C1CCCC1)=O)C2 8453,c1(O)ccc(OC(CC)CNC(C2(OC(C)(C)C)CC2)=O)cc1.C(C)(=O)N 8454,C1(C(=O)NCC(CC=C)NC(=O)CC(CCC)NC)CCC2(CCCC2)C1 8455,Cc1cc(C(=O)NC2(CNC(=O)C(C3CCCCCC3)O)CC2)oc1C 8456,N1(C(C2=CCN(C(C3C(C(C)=O)C3(C)C)=O)CC2)=O)CCc2ccncc2C1 8457,C1(O)(CC(=O)NC(CN(C(c2ccc(O)cc2)=O)CC)C)CCCOC1 8458,C1(NC(C2N(C)CC(O)C2)=O)C2CCC1CN(C(c1ccc3c[nH]nc3n1)=O)C2 8459,N1(Cc2c(COC)noc2)CC2CN(C(=O)C(c3ncc(F)cn3)OC)CC2C1 8460,C1(C(=O)NCC(c2ccccc2)CNC(c2cc[nH]n2)=O)(CC)CC1(F)F 8461,N#Cc1cccc(N2CCN(CCCO)CC2)c1.C12CC1NC2CF 8462,c1(CCNC(C(N2CCC(CO)CC2)=O)Cc2ccccc2)c(O)cccc1Cl 8463,c1(CC(N2CCC(NC(CC=C=C)=O)C2(C)C)=O)ccc2oc(O)nc2c1 8464,C1(C)(NC(Cc2cc(C)on2)=O)CCCN(C(c2cc(C(C)(C)C)oc2C)=O)C1 8465,C1(=CC(=O)NC(CC(C)NC(COC(C)=O)=O)C)CC2CCC(C1)N2C 8466,N1(C(C)=O)CCc2cc(C(=O)CC(=O)C(N3C4CCC3CC4)=O)ccc21 8467,C1(NC(C(C)CO)=O)(CF)CCN(C(=O)COCCCF)C1 8468,N1(CC(=O)NCCOCCOCCCNC(=O)C=CI)CC2CC2C1 8469,Cc1ccc2c(c1)CCC2(C)NC(c1c(F)cc(I)cc1F)=O 8470,N1(C(C(CCSC)O)=O)CC2CC(N(C)C(c3cccc(CSC)c3)=O)C1C2 8471,C(CCCCC(=O)NC1COCCN(C(c2csc(Cl)c2)=O)C1)OC 8472,CC(C)CC(C(=O)NC(c1ccc(Cl)cc1)C)SC1CC1C(C)C 8473,C1(CNC(CN(C(=O)OC)C)=O)CC2CCCC(C1)N2C(=O)CCC1CCCO1 8474,C(=O)(CC(CC(C)C)NC(=O)CC1CC2CC2C1)NCCc1cc(CC)no1 8475,Cc1c(C(N2CCCC2C(=O)NCC(=O)O)=O)c(Cl)nn1C 8476,N1(C(C(C)CC(N)=O)=O)CC(C)(C)OCC1NC(C)C(=O)NCCc1ccc2c(c1)CC2 8477,C(=O)(CP(C)(C)=O)NC(C)CC1CN(C(=O)CCN2CCCC2)C1 8478,N1(C(C2CC(OC)C2)=O)CCOCC1CNC(C1(C(F)F)CCOCC1)=O 8479,N1(C(c2c(CC)c[nH]c2)=O)CCC2C(CCCN2C(c2ccc(N)cc2Cl)=O)C1 8480,c1(N(C(=O)NCCOC)C)coc(OCCCCO)n1.c1(O)ccccc1 8481,c1(C)cc(Br)ccn1.C1(C(C(=O)NC)N(C2(CCF)CC2)C)CCC(C(=O)O)C1 8482,C=CC(CC(=O)NC(COC(F)F)CO)C1CNC1 8483,c1(-c2cc(N(C)C)sc2)cccc2c1CN(C(=O)CN1C(=O)CSC1=S)CC2 8484,Cc1cc([N+](=O)[O-])cnc1C(=O)NCCNC(c1csc(-c2ccco2)n1)=O 8485,C(=O)(CCCS(C)(=O)=O)NC1CCCC(NC(C2(O)CC(C)(C)C2)=O)C1 8486,N1(C(C2N(C(c3cc(OC)n[nH]3)=O)CC(F)C2)=O)CCC2(CCN(C)C2)C1 8487,c1(CNC(c2nnnn2C(C)CC)CCOCC)ccc(OC)c(C)c1 8488,Cc1cc(NC(c2cn(Cc3ccn(C)n3)nn2)=O)ncc1Br 8489,C1(CC)CN(C)CCN1C(=O)CC(CNC(=O)CS(C)(=O)=O)OC 8490,N1(CCC#C)CCCC1CC1CCCC1.C1(=O)C(C)N1C(C)=O 8491,N1(C(CC(CC)C(C)C)=O)CC(NC(c2cscn2)=O)C2(CCCC2)C1 8492,C1(C(N2CC3C=CC3C2)=O)(OC)CCN(C(c2csc(C#N)c2)=O)C1 8493,C(=O)(C(C(C)C)OC)OCCNC(C(C)OC1CCN(C(COCC)=O)C1)=O 8494,c1(NCC2CCN(C(CCNC(C)=O)=O)CC2C)nc(Cl)nc2[nH]c(O)nc12 8495,C1(C(=O)NCC2C(CC(=O)NC(C#C)C3CC3)C2)CC2(CCC2)C1 8496,C1(C(=O)NCCCNC(C(C(C)C)n2ccc(C)c2)=O)CC2OC1C1CC21 8497,Cc1cc(C)c(C(N2CCC(C3CC3)C2CNC(=O)CP(C)(C)=O)=O)cc1C 8498,CCCCC(O)C(C)C(=O)NC(C)CCCC(=O)NC1(CO)CC(O)C1 8499,C1(CNC(C2CC(C)(O)C2)=O)CN(C(c2ccn3ccccc23)=O)C2(CCC2)C1 8500,c1(C(N2CCCC2C(=O)O)=O)cccc(C2(C(=O)O)CCC2)c1 8501,c1(C(=O)NCC(c2cccc(Cl)c2)NC(C=CCCC)=O)ccccc1C1CC1 8502,N1(C(CNS(CC)(=O)=O)=O)CCC(C)(C)C1CNC(C1CC2(C1)CC(O)C2)=O 8503,N1(C(C(C)SC)=O)CCCN(C(c2ccc(CSC(F)F)o2)=O)C(C(C)C)C1 8504,c1(CNC2C(C(N(C)Cc3ccc(C)cc3C)=O)CCC2)ccc(F)c(F)c1C 8505,N1(CCC(=O)N(C)Cc2ccccc2)CCCCC(NC(=O)CCC2CCC2)C1 8506,CC(C)(C)C(C)(O)C(=O)NCC1(C)CCCN1C(c1cnc2n1CCS2)=O 8507,C(=O)(CC1=NN(C)C(=O)C1)NC1CN(C(C(C)n2ccnc2)=O)CC1C 8508,C(C)(C)(CCCF)NC(CCN(C)C(c1cnc(S)nc1)=O)=O 8509,c1(C(=O)NCC2(c3ccccc3)CC(F)C2)ncc(C(F)(F)F)cc1Cl 8510,CCC(CNC(=O)Cc1cn(C)nc1C(F)(F)F)(CC)NC(C1CSCCS1)=O 8511,CC(C)(F)CC(=O)NCc1cccc(CNC(C2CCC(=O)O2)=O)c1 8512,N1(C(=O)C2=COCCC2)CCOC2(C1)CN(C(c1cscn1)=O)C2 8513,S(=O)(=O)(c1ccc(=NCCCCCNC(C)=O)[nH]c1)NCC(CCC)OCC 8514,CCCC(CNC(=O)CC(C)C)C(=O)N1CC(=O)NC(CC)C1 8515,C(C)(C(=O)NCc1ncnn1CC)(C1CCC1)NC(C(C)OCC#C)=O 8516,C1(NC(CC(CC)OC)=O)CCC2CN(c3nnc(-c4ccon4)s3)CC12 8517,Cc1c(C(=O)NCC2(F)CC(CO)C2)cc(C(F)(F)F)cc1[N+](=O)[O-] 8518,C#Cc1cnc(C(=O)NCc2ccc(C(=O)N(C)Cc3cocn3)s2)c(C)c1 8519,c1(OC)ccc2cc(C(=O)NCC(C(C)C)NC(=O)C3=CCC3)nnc2c1 8520,C1(NC(C2(C(CC)(F)F)CC2)=O)C2CC(NC(=O)CCC3CCN(C)C3)CC12 8521,CCCCCC(O)CC(=O)N1CC2CC1CN2C(C1CCc2nccn2CC1)=O 8522,c1(C2(C(=O)NCC(C)N(C(c3n[nH]c(C)n3)=O)CC)CCC2)ccccc1C 8523,Cc1cc(C(F)(F)F)ccc1C(=O)NCC1CN(C(=O)CCC2(C)CC2)CC1C 8524,C1(NC(c2ccnn2C2CC2)=O)CC(CNC(c2n[nH]cc2)=O)C12CCC2 8525,N1(C(c2cc(C)sn2)=O)CCC(NC(=O)COC2CCOCC2)C(CO)C1 8526,N1(C(c2c(C)csc2)=O)CCC2(CCN(C(C3CN4CCN3C(C)C4)=O)C2)C1 8527,c1(C(N2CC3CN(C(CCc4scc(C)c4)=O)C3C2)=O)ccc2ccoc2c1 8528,c1(C(N2CC(NC(C(C)(C)N(C)C)=O)C(F)CC2)=O)ccnc2c1ncn2C 8529,c1(CNC(C(C(CC)O)(F)F)=O)nnc2n1CCN(C(=O)CS(=O)(=O)CCOC)C2 8530,C1(OC(NNC(CCOc2cccc(OC)c2)=O)=O)Cc2ccccc2C1C 8531,Cc1c(C(N2CCC(N(C(=O)Cc3ccon3)C)C2)=O)c(O)nc2ccccc12 8532,C12(C(=O)NC(C3CN(C(C4CC(C)(O)C4)=O)C3)C)CC3CC1C2C3 8533,C(=O)(C(O)(CN(C)C)C(F)(F)F)NC1CC2CC(NC(C=CC=CC)=O)C1C2 8534,C1(NC(c2cccc(CNC(CCC=CC(C)C)=O)n2)=O)(CO)CCCCC1C 8535,C1(C(C)C)CCN(C(C2CC3(C2)CC3F)=O)C(CNC(C2CCOCC2)=O)C1 8536,C(=O)(C1=CCCCCC1)NC1(C2N(C(CN(C(=O)OC)C)=O)CCC2)CC1 8537,N1(C(Cc2ccc(OC)cn2)=O)CCC(CNC(C2(C)CC=CCC2)=O)CC1C 8538,N1(CC(=O)OC(C)(C)C)CCC(C)CC1.CCC1CN1C(C)=O.C1CCN1CCO 8539,c1(C(N(C2CCCN(C(=O)CCOCC(F)F)C2)CC)=O)cnc2nccn2c1 8540,N1(C(C(C)O)=O)CCN(C)C(CNC(c2cc(C3CCC3)nn2C)=O)C1 8541,C1(NC(C(OC)OC)=O)CCN(C(=O)C(F)(F)C=Cc2ccccc2)CC1 8542,C(c1ccccn1)=CC(=O)NCC(CNC(C=CCOCCOC)=O)(C)C 8543,c1(CNC(C2C3(CCN(CC(=O)NCC)CC3)C2)=O)cc2cc(C)ccc2s1 8544,N1(C(CN2CCN(C)CC2)=O)CCN(C(c2nc(=O)n(C)[nH]2)=O)CC1CC1CC1 8545,C(CC(=O)NCCC(C)(C)F)(C(F)(F)F)NC(c1ccc(C#C)cn1)=O 8546,c1(C(C)NCc2ccsc2C(F)(F)F)cc2ccccc2oc1=O 8547,C=CCCCC(C)(C)C(=O)NC1CC(C)(NC(c2ccc(C(=O)OC)n2C)=O)C1 8548,c1(OC)ccc(C(N2CC(NC(=O)CCNC(N)=O)C(F)C2)=O)c(F)c1F 8549,c1(C(=O)NC2COCC2NC(C2CC2(F)F)=O)cc(C(F)F)cc2ccccc12 8550,C1(C)(OC)CCCN(C(=O)CCCC(C)NC(=O)C(C)=CC2CC2)C1 8551,c1(C(=O)NCC(C(=O)N(C2C(C)C2)C)O)ccc(CO)cn1 8552,CC1CCCC=C1C(=O)N1CC(C)(C)CC1C(=O)NCCc1ccncc1 8553,c1(CC(=O)NC2(C)CCN(C(c3ccc(C(C)=O)o3)=O)C2)csc2ccccc12 8554,CC1(C)CC(NC(=O)C(O)CCCNC(C2CC2C#N)=O)C(=O)O1 8555,C1(CNC(c2cc(CC)no2)=O)CN(C(=O)C(C)N2CCCC2)CCC1(C)C 8556,C1(C(=O)OCC)(C(=O)NC2CN(C(=O)Cc3ncc(C)s3)C2)CC12CC2 8557,CC1CC(C(=O)NC2CN(C(=O)C=Cc3cc[nH]n3)CC2n2ccnn2)CN1C 8558,N1(C(CC=C)=O)CCC2(CCC2)C(CNC(c2nc(CC)oc2C)=O)C1 8559,C1(C#N)(C(=O)NCC2(C)CCN(C(c3c(COC)cccc3)=O)C2)CC2CC2C1 8560,Cc1cc(C(=O)NCC(C)(O)CNC(=O)C(C)C(C)(F)F)cc(C)c1F 8561,S(=O)(=O)(c1[nH]c(=NC(CO)c2ccccc2)ccc1Br)NCc1c(C)cccn1 8562,C(C(C(C)(C)C)NC(=O)Cc1cccc(C(C)C)c1)NC(C(C=C)O)=O 8563,c1(C(=O)NCCCC2(NC(=O)Cc3ccnc(Cl)c3)CC2)ccc2nccn2c1 8564,CCC(C)(CC)C(=O)NCCCCC(=O)Nc1cn(C)nc1Cl 8565,N1(C(C(C)(C)O)=O)CCN(C(c2ccnn2CC(F)(F)F)=O)CC(O)C1 8566,Cc1cc(C)c(C(=O)NCCC2CN(C(C3CC(C)C3)=O)CCS2(=O)=O)cc1C 8567,c1(CN(C(CCN(C(C(CO)OC)=O)CCO)=O)C)cccc(C)n1 8568,c1(C(=O)NC(C(C)NC(=O)COCCSCCO)CO)cccc(CC2CC2)n1 8569,CC1CCCN(C(=O)C=CC=C(Cl)Cl)C1CCNC(=O)CCC(N)=O 8570,C(=O)(CC(=O)NC1CCCC1CNC(c1coc(Br)n1)=O)NCC 8571,CCCCCCCCC(=O)NC1CCCCC1NC(=O)CNc1nccs1 8572,c1(C(=O)NCC(C)CNC(C2(Cl)CC2(C)C)=O)cc2ccoc2cc1F 8573,CCCCC(O)C(=O)NC1CCC(C)(CNC(c2ccnc(SC)c2)=O)CC1 8574,C1(C(=O)NC2CN(C(CCCNC(C)=O)=O)CC2C)CCn2ncnc2C1 8575,C1(C(N(C(CNC(CCCC)=O)C)C)=O)CC(=O)N(CCC)C1 8576,C(c1cn(C)cn1)=CC(=O)NC(C)C(CO)NC(c1cnc(C(F)(F)F)nc1)=O 8577,Cc1ccc(CC(N2CC(N(C(=O)Cc3cc(C4CC4)nn3C)C)C2)=O)c(Cl)n1 8578,C1(C(N(CC(C)(C)CNC(c2cn(CCO)nn2)=O)CC)=O)C2CS(=O)(=O)CC12 8579,c1(C(N2CCC(C)C2CNC(=O)CC2CCNC2=O)=O)ccc2cc[nH]c2c1 8580,C(=O)(C(C)CC#N)NCC#CC(=O)NC1C=CC(C(=O)NC)C1 8581,c1(C(=O)NC2C(NC(C(CC)C)=O)CCOC2)cc(C)nc2c(C)c(C)nn12 8582,c1(CC(=O)NCCN2CCN(C(C3CCC4CC34)=O)CC2)ccnc(C2CC2)n1 8583,c1(N2CCC(NC(C(C)C)=O)C2)cc(P(C)(C)=O)ccn1 8584,c1(C(C(=O)N(C(CNC(C(C)C(C)(C)C)=O)C)C)=O)c[nH]c2ccc(F)cc12 8585,Cc1ccc(C(=O)N(C(C)C(=O)Nc2ccc(C(C)C)cc2)C)cc1 8586,CCCCCC(CC)C(=O)OCCOCc1nc(C)no1 8587,C#CC1(CNC(=O)OCCN2CCC(OC)CC2)CCOCC1 8588,C1(CNC(c2c(CC)noc2)=O)CN(C(=O)CC2CCC23CCC3)C2(CCC2)C1 8589,Nc1cnc(Cl)c(C(=O)NC2CCCCCC2NC(=O)CC23CCCC2C3)c1 8590,Cc1ccc(OC(F)F)cc1C(N1CCC(NC(=O)C=CC(C)(C)C)C1C(C)C)=O 8591,CC(C)CC(C(=O)NCc1cnn(C)c1C(N1CC2(CSC2)C1)=O)N(C)C 8592,CC1CC1S(=O)(=O)NCC1(c2ccc(F)cc2)CCCCC1 8593,CC(=O)CC(C)(C)CC(=O)N1CC(OCCNC(c2ccn3c2CCCC3)=O)C1 8594,C(=O)(C(C)(C)C1CCCN1C(COC1CN(C(C)=O)C1)=O)NC1CCSCC1 8595,C(c1ccc(Cl)s1)=CC(N1CC(=C(CNC(c2c(C(C)(C)C)n[nH]c2)=O)F)C1)=O 8596,C1(NC(C(C(C)C)C)=O)CCN(C(=O)C(C)n2cccn2)CC1C(N)=O 8597,C1(CNC(CC=C=C)=O)CCCCN1C(c1ccc(C(N)=O)nc1)=O 8598,c1(NC(C)=O)ncc(S(=O)(=O)N2CCCC3(CO)CCCC23)s1 8599,Cc1nnc(N2CC(O)(CNC(c3ccnn3C(C)C)=O)C2)c(C#N)c1C 8600,C12(C(=O)NC(C)C(CO)NC(c3cnco3)=O)C3C4C1C1C2C3C41C(N)=O 8601,c1(OC)ccc2c(c1)C(C)CN(C(C1COCC(C)N1)=O)CC2 8602,Cc1cc(C(=O)NC2CCOCC2C(=O)NCCC2CC(C)(C)C2)nnc1C 8603,c1(NC2CCCN(C(C3CCCSC3)=O)CC2)ncc([N+](=O)[O-])cc1F 8604,CC1CN(C(C2(C)CCCO2)=O)CCC1CNC(=O)CC(C1CC1)C1CC1 8605,C1(CC)CN(C(c2cc(Cl)ccn2)=O)CCC1NC(C1CC(=O)N(CC)C1)=O 8606,C1(NC(C(C)SC)=O)CN(C(=O)C(C)CC2CCC2)CC(F)(F)C1 8607,CC(CS(C)(=O)=O)C(=O)N1CCOCC(NC(c2cnoc2)=O)C1 8608,CCC(CNC(=O)CN(CC(C)C)C(=O)C=CC1CCCC1)C(C)C 8609,C(=O)(C1CSc2ccccc21)N(C1CN(C(=O)CCCn2ccnc2)C1)C 8610,N1(C(c2cnc(NC)o2)=O)CCCC12CCC(NC(=O)CC(C)OC)CC2 8611,N1(C(CN(C)C(c2ncccc2N)=O)=O)CCC2CC2C1 8612,CCCCCCN=c1cc(NCc2ccc(-c3ccncc3)cc2)nc(C)[nH]1 8613,c1(COCCN(C2CCOC23CCC3)CCOC)ccc(S(=O)(=O)N(C)C)o1 8614,C1(CNC(CN(C2CCC2)C(C2C(C)CCOC2)=O)=O)CC2(CCO1)CC2 8615,CCCCCC(CC)C(=O)NCC(CCCC)NC(c1ncoc1C1CC1)=O 8616,C1(NC(CCC(=O)OC)=O)CN(C(c2cc(Cl)ccc2C)=O)CC1C#N 8617,Cc1cn2cc(C(=O)NC3CCC(NC(C4CSCC(=O)N4)=O)CC3)ccc2n1 8618,c1(C(N2CC3C(CNC(c4c(COC)cc[nH]4)=O)C3C2)=O)nc(C)ncc1Br 8619,N1(C(C=Cc2c(C)ccnc2)=O)CCCC(O)(CNC(c2cnnn2C)=O)CC1 8620,c1(-c2nc(C)c(NC(=O)CCn3cncn3)s2)ccc2nn(C)cc2c1 8621,C(C)(CC(=O)NC1(C)CC(C(=O)NCC2(CSC)CCC2)C1)OC 8622,c1(C(=O)NCCCOCCNC(C(C)O)=O)cncc2c(O)nccc12 8623,C1(C(N2CC(O)C2)=O)(NC(C=CCN(C)CC)=O)CCSC1 8624,C(C(C)(C)C(=O)N1CCC1CNC(=O)Cc1coc(-c2ccccc2)n1)N(C)C 8625,C#CC(CNC(=O)CSCCNC(c1cc(F)c[nH]1)=O)CC1CC1 8626,c1(CC)[nH]nc(C(=O)NC2(CO)CN(Cc3ccn(CCF)n3)C2)c1F 8627,C(=O)(CCCCCCCCS(C)(=O)=O)NCC=C1CCN(C(CCC#C)=O)CC1 8628,N1(C(C2CC(=O)NCC2)=O)CCC(O)(CNC(C2(c3ccccc3)CC2)=O)CC1 8629,C(=O)(C(Cc1cn[nH]c1)NC(=O)CN1CCCC1)N(C)CCc1cccs1 8630,N1(C(C2N(C)C(=O)C(F)C2)=O)CC2CC1CN(C(c1cncc(C(F)F)c1)=O)C2 8631,c1(C(N2C(CNC(c3cn[nH]c3)=O)COCC2)=O)cc(F)c(Cl)nc1Cl 8632,c1(C(N2CC3CCCC(C2)N3C(c2cccs2)=O)=O)cc2c(cn1)OCCO2 8633,c1(CCNC(CNC(CNC(C2CC(=O)NC2)=O)=O)=O)nccc(O)n1 8634,CCCC(C(=O)OC)C(=O)N1CCC(C)(NC(c2oc(C(F)F)cc2C)=O)C1 8635,C1(C(N2CCC(CCNC(c3cc[nH]c3)=O)C2)=O)CCC2(CCC2)O1 8636,CC(C)CC(C(=O)N1CC(CNC(=O)CNS(N)(=O)=O)CC(C)C1)NC(N)=O 8637,C1(CCC)(NC(=O)C=Cc2cnccn2)CCCN(C(c2sc(O)nc2C)=O)C1 8638,C(=O)(C1=CS(=O)(=O)CCC1)N1CCN(CCCNC(CC2C(C)CCC2)=O)CC1 8639,C(C)(CCC(=O)N(CCC(N1CCC(F)(C(N)=O)C1)=O)C)OC 8640,c1(CC(=O)NCCC2CC(NC(C3CC3Cl)=O)C2)noc2ccccc12 8641,C1(CNC(C(C)OCCOC)=O)CCCCN(C(c2ccc(O)nc2Cl)=O)C1 8642,C(=O)(C(C)(F)c1ccccc1)NCCN(C(=O)C(=CC1CCCC1)C)CCOC 8643,CCC(CC)(CO)C(=O)N1CCCCC(CNC(c2cc(C(C)(C)C)no2)=O)C1 8644,C(=O)(C(C)(C)C1=CCN(C(=O)C(C)n2ccnn2)C1)NC1CCN(CC)CC1C 8645,C1(C(=O)NC2C(CCOC)C2)CC(C)(C)CCN1C(c1cnncc1OC)=O 8646,C#CCCCCCC(=O)NC1CCC(C)N(C(c2ccc(F)cc2)=O)C1 8647,C1(C(=O)NCCCO)CCCCCCN1C(c1ccc(C(F)F)o1)=O 8648,C#CC(C)(C)C(=O)NCC(C)NC(c1cc(C)[nH]c1C)=O 8649,CCC(C)C(C(=O)N1CCC(CNC(c2ccc(NC(C)C)cc2)=O)C1)OC 8650,N1(C(c2cc(COC)on2)=O)CCN(C(=O)CC2(C)CC2(Cl)Cl)CC1CO 8651,N1(C(C(C2CCC2)OC)=O)CCN(C(=O)CCc2nccn2C)C(CC2CC2)C1 8652,c1(C(C(=O)N(CC(C)NC(C2CC3CC3C2)=O)C)(C)C)ccc(C#N)cc1 8653,c1(CNCCC(C)P(C)(C)=O)cccc2cn[nH]c12 8654,C(N=c1[nH]c(N2CC3CC2CO3)nc2c1CSC2)c1nnc(CC)s1 8655,n1(CC)cc(Cl)c(C(N2CC(NC(c3cccnc3C)=O)C(SC)C2)=O)n1 8656,CC1CCCC1(c1nnnn1C)NCCc1ccccc1 8657,O=S(=O)(c1cc2ccccc2s1)NCC1(O)CCCN(Cc2ncccc2Cl)C1 8658,C1(NC(c2ccc(COC)o2)=O)CN(C(=O)C(=O)NCCC(N)=O)C2CCCC12 8659,C=CC1(C(=O)NCC(C2CC2)N(C)C(c2cc(C)c[nH]2)=O)CCCCC1 8660,CC(C)(F)C(=O)NC1COCC1C(=O)NCC[Si](C)(C)C 8661,CCCC(C)CC(=O)NCCCCC(C)NC(c1ccn(C(C)C)n1)=O 8662,C1(CCC(=O)NCC(CSC)OC)CCCCN1C(=O)CCCC1CC1 8663,Cc1cnc(NCc2ncccc2Cl)c(S(=O)(=O)N2CCOC(C3CC3)C2)c1 8664,n1(CC(=O)NC2C(C)CCN(C(C34CCC(C3)C4)=O)C2)ccc(=O)c([N+](=O)[O-])c1 8665,C1(CNC(c2ccc(Cl)nc2)=O)CN(Cc2cc(Br)c[nH]2)CCO1 8666,S(=O)(=O)(c1ccc2nc(O)oc2c1)N1CCCN(C(C(C)n2cccn2)=O)CC1 8667,C(CCC(C)(C)C)NC(c1c(CNC(C(C)=C(C)C)=O)n[nH]c1)=O 8668,Cc1ccc(C(=O)NCC2(F)CN(C(C3CC3c3ccc(C)s3)=O)C2)cn1 8669,N1(C(C(C)C2CC2)=O)CCCC2(NC(c3cncc(F)c3)=O)CC2C1 8670,c1(C(C)=O)c(C)[nH]c(C(=O)NCC2(O)CC(NC(=O)CCC3CC3)C2)c1C 8671,N1(C(=O)Nc2c(Cl)cc(C(=O)OCC)c(F)c2)CCc2c(O)noc2C1 8672,c1(OCC(=O)NC2(F)CN(C(=O)COC3CCCC3)C2)cc(F)c(Br)cc1F 8673,N1(C(C(C(COCC)C)C)=O)CCc2sc(CNC(=O)COC(C)C)nc2C1 8674,CC1CN(C(c2cncnc2C(C)C)=O)CC1(C)CNC(C1COCCO1)=O 8675,c1(C(=O)NC(CN(C(=O)CSCCN(C)C)C)(C)C)coc(-c2ccccc2)c1 8676,C1(C(N2C(CN(C(CN(C)C)=O)C)CCC2)=O)CCC(F)(F)CC1 8677,C#CCCCC(C)C(=O)NCC(C(=O)NC1CC(O)C(F)C1)N(C)C 8678,CCCS(=O)(=O)CC(=O)NCCCC(C)NC(C1(CC)CCOCC1)=O 8679,c1(CN2CCC(CC(=O)Nc3c(OC)ccnc3)C2)ccnc(Cl)c1Cl 8680,C(CCN=c1[nH]c2cc(Br)cnc2s1)N(C(CC(C)C1CC1)=O)CC1CCCC1 8681,C1(C(C)=O)CC(CC(N2CCN(C(=O)C(F)=C3CCC3)CC2)=O)C1(C)C 8682,C1(CNC(Cc2c(SC)cccc2)=O)CCC2(CN(C(=O)CC3CN(C)C3)C2)O1 8683,CC(C)(CC(F)(F)F)C(=O)NCC(C(C)(C)C)NC(C1C2(CC2)C12CC2)=O 8684,C1(NC(C(C)=C2CC2)=O)CC2(C1)CC(CNC(=O)CSC(C)C)C2 8685,N1(C(CCNC(C)=O)=O)CCCC2(C1)CN(C(C1C(C#N)C1(C)C)=O)C2 8686,C12(CNC(c3cc(C)sc3)=O)CCC(CC1)N(C(C1CC1C1CCCO1)=O)C2 8687,C(=O)(CS(=O)C(F)(F)F)N(CC(C)N(C(CNC(C)=O)=O)C)C 8688,C(N=c1[nH]c(=NC)[nH]c(=NCc2cccc(F)c2F)[nH]1)C1CCN(CC)C1 8689,n1(CC(=O)NCC#CCNC(C2(C)CCOCC2)=O)cnc([N+](=O)[O-])c1 8690,C1(C(=O)NCC2(COC)CN(C(c3ccco3)=O)C2)C2CCCCC12 8691,C1(C(N2CCC(C)(CNC(c3cc(C(C)=O)oc3)=O)C2)=O)CC(C)CC(C)C1 8692,N1(C(COCCCC(C)C)=O)Cc2nccn2CC(NC(c2cscc2F)=O)C1 8693,C12(CNC(C(C)SC)=O)CC(NC(=O)CCSc3ccc(Cl)cc3)(C1)C(C)O2 8694,C(=O)(C1CCc2c[nH]nc21)NC1CC2CN(C(c3cc(C)[nH]n3)=O)CC1C2 8695,N1(C(C#CC(C)C)=O)CC2COCCC2(NC(c2ccc3nc(S)[nH]c3c2)=O)C1 8696,C1(NC(c2cnn(C)c2F)=O)CC12CCN(C(c1ccc(S(C)(=O)=O)[nH]1)=O)CC2 8697,Cc1cc(C(N2C3CN(Cc4cccnc4Br)CC23)=O)c(F)cc1F 8698,N1(C(C(C)=CC)=O)CCN(C(=O)CCSCc2ccccc2)C(C)CC1C 8699,C(C(=O)N=c1ccn(CCC)[nH]1)c1nccc(CNC(CCCCC=CC)=O)c1 8700,N1(C(c2c(CC)cccn2)=O)CCN(C(c2cccc(N)c2C(F)F)=O)CC1C 8701,C1(C(N(C2CCC2)CC#C)=O)CC2CCC(C1)N2C(=O)Cc1ccon1 8702,c1(C(=O)NCC(CC=C)NC(=O)C(n2ccnc2C)C)nc(C)ccc1OC 8703,c1(C(=O)NC2C(C(=O)NC(c3cnc[nH]3)C)COC2)cnn(C)c1Cl 8704,CC1=C(C(=O)NCC2CCCCN2C(c2cccc3nonc23)=O)CCCC1 8705,c1(C(=O)NC23CC(CNC(C4C(OC)CCC4)=O)(C2)C3)nnc(S)n1C 8706,C1(F)(CNC(c2ccc(CO)nc2)=O)CCC(NC(C23COCC2C3)=O)C1 8707,C#CCCCCCC(=O)NCC1(CNC(C2CC2(Cl)Cl)=O)CC1(F)F 8708,C12(NC(C3CC(=O)NC3)=O)CCC(C(=O)Nc3nccnc3CO)(CC1)CC2 8709,c1(C(N2CCC(NC(C(C=CCCC)O)=O)C(O)C2)=O)cnc2n1CCOC2 8710,O=S(=O)(c1ccc2c(c1)CC2)N1CCN(CC2C3CCCCC23)CC1 8711,N1(C(c2c(CC)cco2)=O)CC(NC(c2cncc(F)c2)=O)C(C(F)(F)F)C1 8712,c1(CN2C(C(N(C3CC3)CC)=O)CC3(CC3)C2)cc(OC)c(O)c(Br)c1 8713,c1(OC)ccc(C(=O)NC(C)CC(C)NC(=O)Cc2cnc(C)o2)cc1C(F)F 8714,N1(C(C(C)=C(CC)C)=O)CCC2(NC(C3CS(=O)(=O)C3)=O)CCCCCC12 8715,N(C(=NCCOC)NCC1(COc2ncccc2F)CCC1)CCOCCOC 8716,C1(NCc2[nH]c(=N)sc2)CCCCC1C(=O)NCc1ccccc1N1CCCC1 8717,N1(C(=O)NCCC(=O)N(c2ccc(F)c(Cl)c2)CC)CCC2CN(C(=O)NC)CC12 8718,C12(NC(c3ncn(CC)n3)=O)CC(C1)N(C(=O)CCC1CC1)C2 8719,C1(NC(c2ccc(SC)s2)=O)CC2CC(NC(=O)C=Cc3cc[nH]n3)CC2C1 8720,c1(-n2cc(C(N(C(C)CCNC(C3CC(C#N)C3)=O)C)=O)nn2)ccccc1Cl 8721,c1(OC)cnc(C(N2CCCCC2CCCNC(=O)Cc2c[nH]nc2C)=O)cn1 8722,C1(NC(c2cnsn2)=O)CN(C(c2sccc2OCCF)=O)CCC1C(F)(F)F 8723,C1(C2CCCN(C(C3CC(F)C3)=O)C2)(NC(C(C)NC(=O)CC(C)(C)C)=O)CC1 8724,c1(-c2ccc(OCC)cc2)ccc(=NCc2ccc(OC(C)C)cc2)[nH]c1 8725,c1(OCCN(C)C)ccccc1C(=O)NC1C2CC1N(C(=O)CN1CCSCC1)C2 8726,c1(OC)ccc(C(N2CCC(C(C)NC(=O)Cc3cc[nH]c3)C2)=O)c(O)c1 8727,C=C1CCC(C(N2CCCCC2C(=O)NC(C)C)=O)CC1 8728,C1(N(CC(=O)OC(C)(C)C)C)CC(C(N)=O)C1.C1CC(=O)N1Cc1cccs1 8729,C1(C(=O)NC(C2CCN(C(COC(CC)C)=O)C2)(C)C)CC2CCC(C1)S2(=O)=O 8730,N1(C(C2C3(CCN(C(c4cc(C)c(O)cc4)=O)C3)C2)=O)CCC2(CCCCO2)C1 8731,c1(OCC(=O)NCC2CC(CNC(=O)C(F)C3CC3)C2)ccc2c(c1)CCCC2 8732,N1(C(CC(C)(C)N(C(C(C)NC=O)=O)C)=O)Cc2ccccc2C1 8733,c1(OC)cc(C(=O)NCCC(O)CNC(=O)C(C)(C)C)ccc1[N+](=O)[O-] 8734,C(=O)(C1=CS(=O)CCC1)N1CC(OCCNC(=O)Cc2cocn2)C1 8735,CC(N=c1cccc(S(=O)(=O)NCC23CCCC2C3)[nH]1)C1CCOCC1 8736,C1(O)(CN(C(C(F)=C(C)C)=O)C)CCN(C(=O)C(C(C)(C)C)C2CCCC2)CC1 8737,N1(C(c2ccc(Br)cc2)C(=O)NCCSC)CCc2cc(F)cc(F)c2C1 8738,N1(C(CNC(C2CCC2)=O)=O)CCN(C(=O)C(O)c2ccsc2)CC2(CC2)C1 8739,C(CN=c1[nH]c2c(c(=NC(C)c3cncc(F)c3)[nH]1)CCC2)(C1CCCC1)OC 8740,c1(CNC(C(=O)N(C2CCN(CC(F)(F)F)C2=O)C)=O)c(S(C)(=N)=O)cnn1C 8741,N1(C(C2(C)CCCCC2)=O)CCS(=O)(=O)CC1.n12cc(nn1)NC(=O)N(C)C(C)C2 8742,c1(CCC)noc(CCC(=O)NC2CCCC2NC(C2CC2C)=O)n1 8743,N1(C(C=C2CCN(C)C2)=O)CC2CC(C1)CN(C(C1CC(=O)N(C3CC3)C1)=O)C2 8744,C(N=c1nc2ncn(C)c2c(NCC2Cc3ccccc3O2)[nH]1)c1n(C)ccc1 8745,c1(SCn2cc(C3N(C(CC(COC)C)=O)CC=C3)nn2)cn(C)c(C)cc1=O 8746,c1(C(N(C(C)CN(C)C(C2CCOC2)=O)C)=O)cc2c(nn1)OCCS2 8747,C(=O)(C1CCc2c[nH]nc21)NCCN(C(=O)C(F)(F)C(O)C1CC1)CC 8748,c1(C(=O)NCC(CNC(C2C(=C)C2)=O)O)cc2cc(Br)ccc2c(OC)n1 8749,C1(NC(c2cccc(CC)c2)=O)CCCN(C(=O)CSc2cnn(C)c2)C1CC 8750,C(CCC(C)(C)C(=O)N(CCC1CC1)CC1CC1)NC(C1C(C)OCCC1)=O 8751,C1(NC(=O)CN2CC=CC2)COC2(CCN(C(C3CC34CCSCC4)=O)CC2)C1 8752,CC(CC(F)(F)F)C(=O)NCCCCN(C)C(C1(C)CCNC1=O)=O 8753,Cc1ccc(F)c(C(=O)NCC(C)CN(C)C(C23CCC(C2)OC3C)=O)c1 8754,c1(C(=O)NC2CCC(N(C(c3ccc(OC)nn3)=O)C)C2)cc(F)c(F)cc1Cl 8755,c12ccc(cc1)C(=O)N1CCN(CC1)C(=O)C(C)(C)O2.C1(OC)CCC(OC)C1 8756,Cc1nc(O)c(Br)cc1C(=O)NCCCN(C(=O)Cc1ccc(O)nc1)C 8757,C(=O)(C(F)(CC)C(=O)OC)NCC1C(NC(c2c(CC)occ2C)=O)CC1 8758,c1(SC)ccc(C(=O)NCC(C(C)C)NC(=O)Cc2cnc(C)[nH]2)c(Cl)c1 8759,N1(C(c2nc(CC)sc2)C(=O)NCc2nnn(C)n2)CCOC(C2(C)N=N2)C1 8760,CCCCC(CNC(=O)C(C1CCOC1)OC)NC(=O)CSC(C)(C)C 8761,N1(C(Cc2cn(CC)nc2)=O)CC=C(CNC(=O)CNC(=O)CC(C)(C)C)CC1 8762,c1(CC(=O)Nc2ccc(C(F)F)c(Cl)c2)c(Cl)cccc1Cl 8763,C12=NC(=N)NC(=NCC(=O)N(C)CCCOC3CCCN1C3)N2.C(C)(=O)OCCN.CO 8764,Cc1sncc1C(=O)NC(C)CCNC(=O)CC1(C)CC1 8765,N1(C(C2(CC)CCN(C(C3CN(CC)C(=O)C3)=O)C2)=O)CC2(C1)NC(=O)NC2=O 8766,N1(C(c2c(C)occ2)=O)CCN(C(c2ccc(N=[N+]=[N-])cc2)=O)CCC1C 8767,c1(N2CC(CC)SCC2)nc(=NCC(C)C(C)(C)C)[nH]c2c1CSC2 8768,Cc1nnccc1C(N1CC2CC1C2C(=O)NCCc1nccs1)=O 8769,c1(C(=O)NC2CC(CNC(=O)C3=COCCO3)CC2O)nsc2c(Cl)cccc12 8770,C1(C(=O)NC2C(C)(CC)C2)COCCN1CCNC(=O)C1CC1 8771,c1(C(=O)NCC(C(C)C)NC(C2CC(CN(C)C)C2)=O)ccc(Cl)nc1 8772,c1(SCCCNC(c2ccccc2Cl)C)cc(Cl)nn(C)c1=O 8773,Cc1ccnc(C(=O)N(C)CC2CCCN2C(C2C3CCCC23)=O)c1 8774,C(=O)(C1=NNC(=O)CC1)NC1C(C(=O)NC(c2ccccc2)Cn2c(C)ncc2)C1 8775,N1(C(c2ncc(OC)s2)C(=O)NC)CCC(c2ccsc2)CC1 8776,CCC(CC(F)F)C(=O)NC1CCCCC1NC(c1c[nH]cc(Br)c1=N)=O 8777,CC(O)CCCCCC(=O)NC1CN(C(c2cnn(CC3CCOC3)c2)=O)C1 8778,CC(C)CCC(N)C(=O)NCC(c1ccco1)N1CCCC1 8779,C#CCCC(O)C(=O)N1CCCC1C(C)NC(=O)Cc1ncc(Cl)s1 8780,C1(NC(C(C(C)C)c2cccnc2)=O)CN(C(=O)Cc2cccs2)CC12CCC2 8781,C1(C(N(CC(C)(C)NC(c2c(CC)nco2)=O)C)=O)CCCCC1(F)F 8782,C1(CNC(Cc2scc(C)c2)=O)CN(C(c2cnn(C(C)(C)C)c2N)=O)CCO1 8783,C(=O)(CC1=CCCC1)NCC(CC)NC(c1ccccc1C(=O)NC(C)(C)C)=O 8784,C1(CC)(CNC(C2OCCC2CNC(=O)CC2(OC)CC2)=O)CCCO1 8785,CC(C)(C)C(O)CC(=O)N1CC(CNC(c2ccc(C(F)(F)F)[nH]2)=O)C1 8786,C(=O)(C1Cc2ccccc21)N(C1CCCN(C(c2nnc(CC)o2)C)CC1)C 8787,C1(N(C)C(C2CC(C)(F)C2)=O)CCCN(C(=O)CCc2ccc(Cl)cc2)CC1 8788,CN1CCCCC1CC(N1CC(CO)(NC(C2(F)CCOC2)=O)C1)=O 8789,C1(NC(NCc2cc(C)on2)=NCc2ccccc2C2CC2)CC(C)OC(C)C1 8790,c1(C(N2CCC(N(C(=O)CC(=O)N(C)C)CCC)C2)=O)c(Cl)ccc(O)c1Cl 8791,Cc1cc(F)cc2c1N(C(c1cnc(C)n1-c1ccccc1)=O)CC2 8792,Cc1ccn(C(C)(C)C(=O)NC2(C)CC(NC(=O)C(C3CCCOC3)OC)C2)n1 8793,c1(C(=O)NCCN(C(=O)CC2CC3CCC(C2)C3)CC)nc(C)ccc1OC 8794,c1(CC(N2C(CNC(C3C(CC)OCC3)=O)CC2)=O)cccc(F)c1O 8795,Cc1cnc(NCc2c(C)cccc2C)c(S(=O)(=O)N2CCC(C3CCC3)C2)c1 8796,C(=O)(C#CC1(C)CCCO1)NC1CC(CCNC(c2c(C)nn(C)c2Br)=O)C1 8797,c1(C(=O)NC2(CNC(=O)CSc3cn[nH]c3)CCOC2)cn2ccccc2n1 8798,C1(C(=O)NC(C(N2CCCC(OCC)C2)=O)C)CCC2(CCC2)C1 8799,N1(C(c2c(C)ccs2)=O)CC(CNC(c2ccccc2C2CCC2)=O)C(C)C1 8800,C(=O)(C1SCCc2ccccc21)N1CC(C(C)NC(=O)CC2(C)CC2)C1 8801,C1(N(C(=O)CCCCC2CC2)C)CCCN(C(c2cccc(F)c2N)=O)CC1 8802,c1(C(N2CC3C(CNC(C(C)c4cccs4)=O)C3C2)=O)coc2cccc(O)c12 8803,c1(C(N2CCCC3(NC(C=CCCC)=O)C(C2)C3)=O)cc2c(cc1O)CCCC2 8804,CC(C)C(O)C(C)C(=O)NCC12CC1CN(C(=O)CCc1ccccc1)C2 8805,CN1CCN(C2CCN(C(=O)CC3CCCCN3c3ccncc3)CC2)CC1 8806,c1(C(N(CC(=O)N(C(C(N)=O)C2CC2)C)CCC)=O)ccc(N)cn1 8807,C1(c2cn(CCNC(c3cn(C(C)C)nc3)=O)nn2)(N(C)C)CCCOC1 8808,N1(C(c2cn(CC)nn2)C(=O)NCCCC2CC2)CCC(C)(C)C2=C(CCO2)C1 8809,c1(-c2cn(CC3N(C(C(C=C)CC)=O)CC3)nn2)cc(N)cc(F)c1 8810,Cc1ncc(NC(C2CC(C)(NC(=O)CC3COCCO3)C2)=O)c(C)c1C 8811,c1(C(=O)NC2C(C)CN(C(=O)C3=CCCC3)C2)cccc2cnccc12 8812,c1(CC(=O)NCCOCCOCCNC(C2(O)CCC2)=O)ccc2c(c1)CCO2 8813,C1(C(=O)NCCOCCCN(C)C(c2cnsn2)=O)CC2CCC1O2 8814,c1(C(=O)NCCC(CNC(C2(CN(C)C)CC2)=O)O)cccc2ccn(C)c12 8815,N1(C(c2c(C)cno2)=O)CCCCC(CNC(=O)Cc2cn(C)nc2C)C1 8816,c1(NCc2c(C(=O)Nc3c(C)cnc(Cl)c3)cccn2)ccc2ncccc2c1 8817,C(=O)(C(O)CCC(F)(F)F)NCC1C(NC(C2(OC)CCC2)=O)CCC1 8818,C1(C(=O)NC(c2c(C)cccn2)C)CC2(CC(NC(=O)Cn3nccn3)C2)C1 8819,C(CCF)(C(=O)NCCC1CCCO1)NC(CCCOCC)=O 8820,Cc1nc(C2CCN(C(=O)NC3COC(C4CC4)C3)CC2)nc2c1CCCC2 8821,C1(CC)CCCN(C(=O)CC(C)(C)C2CC2)C1C(N1CC2(CC2)CC1CO)=O 8822,Cc1onc(CO)c1C(=O)NCC1CCN1C(C1CC(C)(CN2CCCC2)C1)=O 8823,C1(CC(=O)NC2CN(C(c3ccc(SC)s3)=O)CC2C)CCC2(CCCC2)CC1 8824,C1(C(=O)NC(C)C)CCCC(C(=O)Nc2cc(C3CCOCC3)nn2C)C1 8825,C(=O)(C1Cc2c(Cl)cccc21)NCCN(C)C(c1cnc(CCC(F)(F)F)s1)=O 8826,c1(C(=O)NC2C(NC(C(CCSC)N(C)C)=O)COCC2)ccnc2[nH]ncc12 8827,c1(C(N(CCC)CCNC(C2CC2(F)Cl)=O)=O)nc(C)c(C)nc1C 8828,N1(C(C(C)(C)C2CCCO2)=O)CCC(O)(CNC(=O)CC2CSC2)C1 8829,CC(C)CC(C)(CO)NC(=O)C(C)C(C)NC(c1c[nH]nc1C(C)C)=O 8830,N1(C(CCSc2n(C)nnn2)=O)CCN(C(C2(C)COC2)=O)CC1CCO 8831,N1(C(C=C(C(=O)N(CCC)CCC)F)=O)CCC(C)C1CSC 8832,c1(C(N(CCCC(=O)NC2CCSCC2)C)=O)ccc2[nH]nc(Cl)c2c1 8833,N1(C(C)=O)CCC(N(C)C)CC1.N12CCCCC1c1nnc(o1)CS2(=O)=O 8834,c1(CN2C(CC)CN(C(=O)Nc3cccc(F)c3C)CC2)cc(I)cc(I)c1O 8835,c1(C(C(=O)NC(C)(C)CC)N(C(C#C)C2CCC2)C)cnc(C)nc1 8836,C12(C(N)=O)CCCC1(C(=O)NCCOCCCNC(=O)CC1(O)CCC1)C2 8837,N1(Cc2cccc(C(=O)NCC(C)C#N)c2)C(=O)CN(C)C1=O 8838,c1(C(=O)NC(CC(=O)NC(CCCC)C)CC2CC2)cccc(C)c1F 8839,c1(C(N2CCC(NC(c3cnc(C)nc3)=O)C2C)=O)cc2c(Cl)cccc2[nH]1 8840,C1(C(N2CCC(NC(CC(C)n3cccc3)=O)CC2)=O)CC2CCC(C1)C2F 8841,C(C(=O)NOCC1CC1)C(C)(C)CNC(C1COCC1C(N)=O)=O 8842,C(C1CCCN1C(c1cc(F)c[nH]1)=O)=CC(=O)NC1(C(C)O)CC1 8843,C(=O)(CC(C)CC(=O)OC)NCC#CC(=O)NCC(CC)NC(=O)OC(C)(C)C 8844,n1(CCC)ccnc1C(F)(F)C(=O)NC1CC(C(C)NC(=O)C(F)CSCC)C1 8845,c1(C(=O)NC2(C)CC(NC(COCCN(C)C)=O)C2)cc(O)nc(Cl)c1 8846,C(C(=O)N1OC2CCC1CC2)(N(C)C(c1c[nH]nc1Cl)=O)C1CC1 8847,Cc1cccc(F)c1C(=O)NCCNC(=O)C(C)(C)N(S(C)(=O)=O)C.C12CC1N2 8848,C1(O)(C(=O)NCC=C=C)CCN(CC(C)CO)CC1 8849,c1(NCc2scc(CC)c2)ccc(SC)cc1.C1(C)C(=O)N1C(C)C 8850,C(=O)(C(F)CC(C)(C)NC(c1ncccc1O)=O)NC(CC)C(C)C 8851,C1(C(N2CCN(C(C)=O)CC2c2cnn(C)c2)=O)CCc2cnc(C)n2C1 8852,C(=O)(C1=Cc2ccccc2C1)NCC1(C)CN(C(c2cnc(O)s2)=O)CCO1 8853,C1(C(=O)NCCCN(CC)CC)C=CCC(NC(c2cnn(CCO)c2)=O)C1 8854,c1(C(=O)NC2CN(C(C=COCC)=O)CC(O)C2)[nH]c2c(c1C)CCCC2 8855,C=CC(C)(C)CC(=O)N1CCN(C(c2[nH]ccc2C2CC2)=O)CC1C(F)F 8856,c1(C(=O)NCCCN(C(COCC(=O)NC)=O)C(C)C)cscc1SC 8857,C1(CN(C)C(c2cnn(C(C)(C)C)c2)=O)COCCN1C(=O)CC(Cl)Cl 8858,Cc1cc(C(=O)NCCNC(c2cc(C(=O)C(C)C)c[nH]2)=O)nn1C1CC1 8859,c1(N2CC(C)CC(NC(c3ccc(OC)c(C)c3)=O)C2)ncc2sccc2n1 8860,N#Cc1ccc(C(N2CCSC3CCC23)=O)cc1O 8861,C(=O)(C(CCSC)NC(C)=O)NCC(C1CCC1)NC(C(=O)NC)=O 8862,c1(C(N2C(C(=O)NCC34CC(CCO3)C4)CC2)=O)coc2ccccc12 8863,n1(CC)ccc(C(=O)NCC2(F)CCN(C(=O)C(c3ccnn3C)O)C2)cc1=O 8864,Cc1cc(C(N2CCCCC2C2(NC(=O)CC(C)F)CC2)=O)cc([N+](=O)[O-])c1Cl 8865,c1(C(N2C(C)CC(CNC(C=C(CC)C)=O)C2)=O)ccc2c(c1)C(=O)NCC2 8866,Cc1nc(CC(N2CC(C)(C(=O)NC3CONC3=O)C2)=O)co1 8867,C(=O)(C1CSc2ccccc21)NC1CCC(CNC(c2ncncc2F)=O)CC1 8868,c1(C2C(C(=O)NCCCN(C(c3cnc(C(C)O)s3)=O)C)C2)ccc(F)cc1F 8869,n1(CCOC)ccc(=NC(=O)C2C(CNC(c3[nH]ccc3C)=O)C2(C)C)[nH]1 8870,NS(=O)(=O)c1cnn(CC(N2CCCCC2CCNC(C23COCC2C3)=O)=O)c1 8871,N1(C(C2CN(C(C)=O)C2)CC)CCN(Cc2n[nH]c(C3CC3)n2)CC1C 8872,C1(CNC(CCOCC)=O)COCCN1C(C1CCSC1)=O 8873,n1(CC)nnc(C(N2CCC2CNC(=O)CNc2nccs2)=O)c1C 8874,c1(N(C(CNc2ccc(Oc3ccccc3)cc2)=O)SC)c(C)cccc1C#N 8875,C(=O)(C(CC)C(=O)N1CC(CNC(C2CC3(CC(OC)C3)C2)=O)(OC)C1)OCC 8876,CC1CN(C(=O)CCCC#N)CC(C)N(C(c2cc3sccc3[nH]2)=O)C1 8877,C1(O)(C(=O)NCc2ccc(OCC=C)cc2)CCCNCC1 8878,CN1CCN(C(C2C3COCC23)=O)CC1C(N1CC(CC(N)=O)C1)=O 8879,C(=O)(CCCCC(N)=O)N(CCNC(c1c(C)ccnc1)=O)C1CC1 8880,C1(NC(CCC(CC)OC)=O)(CNC(C2CCCN2N=O)=O)CCC(F)(F)CC1 8881,c1(C(N2CCN(C(c3[nH]cc(C#N)c3)=O)CC2CCO)=O)nccc2nn[nH]c12 8882,c1(C(=O)NCC#CC(=O)N(C2CCCOC2)CCC)ccc(F)c(F)c1 8883,C1(NC(c2c(CCC)n(CC)nn2)=O)CCCN(C(c2conc2C)=O)CC1 8884,C1(NC(C(C)Cc2ccc(F)cc2)=O)CC2CC(NC(c3ccsc3)=O)C2C1 8885,C1(CNC(C(CC=C)CC)=O)CN(C(=O)CCC(=O)OCC)C2COCC2O1 8886,C1(C(N(C)CC2CCCN2C(=O)Cc2cn[nH]c2)=O)CCCC(C(N)=O)C1 8887,c1(-c2scc(CN3CCN(CCCCC)CC3)n2)ccc(F)c(OC)c1 8888,c1(C(N2C(C(=O)NC3CONC3=O)CSCC2)=O)ccc2sccc2c1O 8889,C1(CC=C)N(C(c2cccc3c2CCO3)C(=O)NCCSC)CCCC1(C)C 8890,C1(C(=O)NC(C)C2CC2)CCN(C(=O)C2=NOCC2)C(C)(C)C1 8891,c1(C(=O)NC(C(C)(C)C)CNC(c2cscn2)=O)c[nH]nc1S(N)(=O)=O 8892,c1(C(C)C2CC2)nc(C2CCN2CC2CCCC2)n(-c2cncc(Br)c2)n1 8893,N1(C(C(C)=C(CC)C)=O)CC(C(=O)NCCC2(C)CC2(F)F)C(C(C)C)C1 8894,C1(NC(NCc2sccc2)=NCC2CCCO2)CCCC12CCC2 8895,C(C(C)(C)C#CC(=O)N(C(C)C)CC)OC(CCSc1ccc(OC)cc1)=O 8896,O=C1OC(C(=O)NCC2CCN2C(=O)Cc2cn[nH]c2)Cc2ccc(Cl)cc21 8897,Cc1ccc(C)c(CC(=O)NC(CNC(c2cncc(C)c2C)=O)C2CC2)c1 8898,c1(C(=O)NC2C(C(N(C)C)=O)CCCC2)c(C(F)(F)F)oc2ccccc12 8899,N1(C(CSCC(N)=O)=O)CC(S(=O)(=O)N2CCN(C(C3CCCSS3)=O)CC2)C1 8900,C1(CCCC(=O)NCC(CNC(c2n(C)ccn2)=O)CO)CCCC(=O)N1 8901,S(=O)(=O)(c1ccc([N+](=O)[O-])cc1OC)N1CC(C(=O)OC)C(N)C1 8902,C(C(C(C)(C)C)NC(c1c[nH]nc1C1CCCCC1)=O)NC(CC1(C)CC1)=O 8903,c1(CCC(=O)N(CC(C)NC(C2CC2(Br)Br)=O)C)cncnc1 8904,c1(OC(c2ccccc2)C(=O)OCC(c2ccsc2)=O)ccc(Br)cc1Cl 8905,N1(C(C(C)OCCOC)=O)CCC(CNC(=O)C(COC)CC(C)C)C(C)(C)C1 8906,C(=O)(C(CO)C(C)(C)C)N(CC(C(N1C2(CC(COC)C2)CC1)=O)C)C 8907,N1(C(CCSCCCC)=O)CCC(CC)C1CNC(C1(C(=O)NC(C)C)CC1)=O 8908,CCCC(C(=O)NCCn1cc(C(N2CCC(N3CCC3)CC2)=O)cn1)OC 8909,N1(C(c2c(CCC)cccc2)=O)CCC2(CCCCN(C(=O)C3CCCS3)C2)C1 8910,N1(C(c2cc(CC)nc(O)c2)=O)CC2CN(C(=O)CN(C)S(N)(=O)=O)CC2C1 8911,C1(CC(=O)N(C)CCNC(=O)CC2(C)CCC2)COCC1(C)C 8912,C1(C(=O)NC2(CN(C)C)CC2)CCN(C(=O)C23CCC(C)(C2)OC3)O1 8913,Cc1nnc2c(C(N3CCC(CNC(C4CCC4)=O)C34CCC4)=O)cccn12 8914,CC(C)(N=[N+]=[N-])C(=O)NC1CCC(CNC(=O)Cc2cc[nH]n2)C1 8915,C=CCCCC(=O)NC(CC1CC1)C(=O)NC1(CO)CC1(C)C 8916,C1(O)(CC2C(Cn3cc(NC(C(CC)OCC)=O)nn3)CCC2)CCCN(C)C1 8917,C(c1c(F)ccc(Cl)c1F)=CC(N1CC2C(NC(CC(C)C(F)F)=O)(C2)C1)=O 8918,c1(C(=O)NCC(CC(C)C)NC(Cc2c(C)nc[nH]2)=O)cc(S(N)(=O)=O)c(C)o1 8919,N1(C(CCCC(CC)CC)=O)CCOC2(CCN(C(=O)CSC(F)F)CC2)C1 8920,C(=O)(CC(=O)NCc1nc[nH]n1)NC(C1(C(=O)NC2CC2)CC1)C 8921,Cc1cncc(C(N2CC(NC(C3CNC(=O)N3C)=O)C(C)C2)=O)c1 8922,N1(C(C(CCC)C)=O)CCN(C(c2n[nH]c(C)c2F)=O)C(CC(C)(C)C)C1 8923,C(=O)(C1CCCn2ncnc21)N1C(C(=O)NC2CN(C(C)=O)C2)CC2COCC21 8924,N1(C(C2CC(C)=C(C)CC2)=O)CCC(C)N(C(=O)C(c2cnn(C)c2)C)CC1 8925,C1(CC(=O)NCCC2(OC)CN(C(c3c(C)nsc3C)=O)C2)CCC(F)(F)CO1 8926,C1(N(CC#C)C(C2(CCC)CC2)=O)CCN(C(c2ncn(C)c2C)=O)CC1 8927,c1(CC(=O)N(CC(C)CNC(=O)CC2CCCN2C)C)cnccc1Cl 8928,C1(O)(CNC(c2c(CNC(CC=C=C)=O)n[nH]c2)=O)CCCOC1 8929,C1(F)(C(=O)NC2CC(OCC)C2)CCN(C(c2sc(C)nc2C(F)(F)F)=O)C1 8930,C(C1CCOCC1)=CC(=O)NC1CC1NC(c1cnn(CC(F)(F)F)n1)=O 8931,C1(C)(C(=O)NCC2CN(C(c3c(CC)onc3)=O)CC2O)CCCCC1(F)F 8932,C1(NC(c2c(C)ccnc2)=O)CN(C(c2ccc(Br)nc2)=O)CC1C#N 8933,CC(C)(C)C(C)(C)C(=O)N1CCC(CF)(NC(=O)CC2CCC(=O)NC2)C1 8934,CC(C)CC(CNC(=O)CC1CCC(C(F)(F)F)O1)NC(C1(C)CCOCC1)=O 8935,c1(C(N(C)CC2OCCN(C(c3cc(C)c(C)o3)=O)C2)=O)cccc(=S)n1O 8936,N1(C(CSCCCC)=O)CC2CCC1CN2C(C1(CCCC)CCCC1)=O 8937,c1(C(=O)NC2COCC2NC(C2CCCOC2)=O)ccnnc1S 8938,N1(C(c2nc(CCCC)sc2)=O)CC2CCC1C(CNC(=O)C(CO)N(C)C)C2 8939,C1(O)(CCNC(C(C)C2CCOC2)=O)CCN(C(c2coc(C(F)F)c2)=O)CC1 8940,C1(C(N(CC=CC(NOCC2CC(=C)C2)=O)C)=O)C2CCC(C2)C1C 8941,c1(CN2C3CN(C(=O)OC(C)C)C(C3)C2)ccc([N+](=O)[O-])cc1F 8942,C1(CC(=O)NCCCCCN(C)CC)CN(C(=O)C(C)OCC(C)C)CC1C 8943,N1(C(C2CCCN(Cc3c(OC)cccc3)CC2)=O)CCn2cccc2C1 8944,N1(C(CCNC(COC)=O)=O)CCC(C(C)NC(=O)Cc2sccc2Cl)C1 8945,c1(C(=O)NCCC2N(C(Cc3cnc(C)s3)=O)CCC2)ccccc1F 8946,C1(C(=O)N(c2ccccc2)CC(C2CC2)NC(CSCC)=O)CCC(C2CC2)CC1 8947,N1(C(c2cnc(Cl)s2)=O)CCCC(NC(=O)CSCc2ccc(F)cc2)C1 8948,c1(C(=O)NCC(CN(C)C(c2c(Cl)cccc2Cl)=O)O)coc2c1C(O)CCC2 8949,c1(C(=O)NC2CC3(CN(C(c4c(C)nc(C)o4)=O)C3)C2)cc(Cl)cc2c1CCC2 8950,c1(C(N(CCCC(=O)OC)C(=O)CCNC(C)(C)C)C)c(Cl)cnn1C 8951,CCC(CC(F)F)C(=O)N1CCC(NC(c2cc3ccccc3s2)=O)C1C 8952,c1(C(=O)NCc2csc(C(=O)NC(C(F)(F)F)C3CC3)c2)cnncc1O 8953,N1(C(C2(C)C(C)C2)=O)CCC2(CC1)CN(C(=O)CNC(C1CCCC1)=O)C2 8954,C(CC)(C(C)(F)F)NC(CC(C)N(C(CCSCCCC)=O)C)=O 8955,C(CC(O)C(F)(F)F)NC(C(CCN(C)C)NC(C=CCOC)=O)=O 8956,c1(N2CCC(OCC(C)C)C2)ccc(S(=O)(=O)NCC(O)CF)c(Cl)c1 8957,C1(C(=O)NCC2(NC(C(C)C3CCOC3)=O)CC2)CC(=O)c2ccccc2O1 8958,C1(C(N(C)CC2CN(C(=O)CCc3n[nH]c(=N)s3)C2)=O)CC12CC(C)(C)C2 8959,c1(CNC(C2CC23CN(Cc2ccnc(Cl)c2)C3)=O)cc(Br)ccc1O 8960,C1(C(N2CC(NC(c3n[nH]c(CC)c3Cl)=O)C3(C2)CC3)=O)CC=C(C(C)C)CC1 8961,CCC(C)(COC)C(=O)NC1CC2C(NC(c3ccnc(C(C)C)n3)=O)C2C1 8962,c1(C(=O)NCC2CCC(NC(C(CC)OCC)=O)C2)c(C)c(C)cc(C)c1C 8963,N1(C(CSCC)=O)CCC(CC(=O)NC(C2CCCCO2)(C)C)C1 8964,C1(CC=C)(NC(=O)Cc2ccco2)CCN(C(=O)C(F)OC(F)(F)F)C1 8965,N1(C(C2CN(C(=O)NC)C2)=O)CC2CCCC2(C(=O)NC2CCCC2)C1 8966,N1(C(C2C(OCC)CC2)=O)CC2CCC(C1)N2C(=O)CCc1ccon1 8967,Cc1cc(=O)ccn1CC(=O)NC1CC(NC(c2scnc2Cl)=O)C1 8968,C(C)(CCCCCO)NC(C(CSC)(C)NC(C1CC=CCC1C)=O)=O 8969,C12(C(=O)NC3C(NC(C=C(C)c4cccs4)=O)COC3)CCN(CC1)S(=O)(=O)C2 8970,N1(C(c2c(OC)cncc2)=O)CC2CC(NC(C3CCN(C)C3)=O)CC1C2 8971,C(=O)(CCCC(=O)C(C)SCC(C)C(=O)Nc1ccccc1C(F)(F)F)OC 8972,CCC(C)C(C(=O)NC1CCOCC1C)N(C(=O)CC(=O)NC1CC1)C 8973,Cc1[nH]nc2ncc(C(=O)NCC3(F)CCN(C(C4CC(N(C)C)C4)=O)C3)cc12 8974,N1(C(C(C)n2cncn2)=O)CCC2(CCC2CNC(C2CC(C#N)C2)=O)CC1 8975,CC1(C)CC(CNC(=O)CNC(=O)OC(C)(C)C)CN1C(=O)CCS(C)(=O)=O 8976,c1(C(CC)NC(=O)NCc2ccc(Cl)nc2C)cccc(S(N)(=O)=O)c1 8977,C1(NC(c2ncn(CC)n2)=O)COCCC1C(=O)N(C)CCOC 8978,c1(C(=O)NCC2(F)CC(NC(c3cnns3)=O)C2)ccc([N+](=O)[O-])cn1 8979,c1(C(=O)NC2CN(C(C=CC)=O)C(CC)(CC)C2)cc(Cl)cc(Cl)c1OC 8980,CC1CCN(C(C2CC23CCSCC3)=O)CC1NC(C1CN2CCN1CC2)=O 8981,CC(F)(F)CC(=O)NCC1CC1CNC(c1cnc(Cl)[nH]1)=O 8982,C1(NC(Cc2cc(C)no2)=O)CC(C)CN(C(C2CC(C)(C)CN2C)=O)C1 8983,CC(CO)(CO)C(=O)Nc1ccccc1OCC1CCCO1 8984,c1(OC)cccc(C(N2CCCC(C(C)NC(=O)Cn3ccnn3)C2)=O)c1Br 8985,C(=O)(C(C)CC(=O)N(CCC(N1CC(N=[N+]=[N-])C1)=O)C)OC 8986,C1(CC(=O)NC2C(CC)N(C(c3cc4n(n3)CCC4)=O)CC2)CCS(=O)(=O)CC1 8987,C1(NC(=O)NC(CC(=C)Cl)CO)CCOC2(CCCC2)C1 8988,c1(C(N(C(C)CCNC(c2cnc(Cl)[nH]2)=O)C)=O)ccc(C(F)F)cc1F 8989,c1(CCC(=O)NCC(COC)(C)CO)ccc(F)cc1C(=O)OC(C)(C)C 8990,CC1(C(=O)NC2CN(C(=O)C(F)(F)C3CC3)CC2CC2CC2)CCCS1(=O)=O 8991,C1(NC(C(Cn2ccc(C)n2)C)=O)CN(C(C23CC(CO2)C3)=O)CC1(C)C 8992,C1(S(C)(=O)=O)CN(C(=O)OC(C)(C)C)CCN1C(C(C)C(=O)NCC1CCC1)=O 8993,C=CC(C)(CC)C(=O)N(C)CCOCCN(C)C(c1cc(O)cc(F)c1)=O 8994,C(=O)(C(C)C(O)C(C)CC)NC1(C)CN(C(C2(C#C)CCCCC2)=O)C1 8995,c1(CC)ccc(OC)cc1C(=O)NC(C)C(C)NC(c1cnn(CC)c1C)=O 8996,C(=O)(CC1OCc2ncccc21)NC(C)CNC(C1C2(CC2)C12CC2)=O 8997,C1(CC=C)(NC(=O)CC2(CO)CC2)CCCN(C(=O)CNc2ccc(Cl)cc2)C1 8998,Cc1ccc(S(=O)(=O)NC2CCS(=O)(=O)C23CNC3)cc1Cl 8999,C1(C)(OC)CCCN(C(C2(C)CN(C(=O)C(N3CCNC3=O)C)CC2C)=O)C1 9000,c1(C(C)CC2CCCCO2)nc(-c2ccc(Cl)nc2)nn1CCSC(F)(F)F 9001,C1(C(N2CC(CC(C)NC(CCOCC)=O)C2)=O)COC2(CO)CC1C2 9002,Cn1nccc1C=CC(=O)NCC1CCC(C(N2CC(O)C(O)C2)=O)CC1 9003,C1(C(=O)NC(C)CN(C(=O)CC2CC(C(=O)OC)C2)C)(CC)CCOC1 9004,CC(=O)CCCC(C)C(=O)N1CCC(C(N2CC3C(C(N)=O)C3C2)=O)C(C)C1 9005,C1(C(=O)OC)CCN(C(C2CNC3CCOCC3C2)=O)C2(CC2)C1 9006,C1(CCC)CN(C(=O)CN(C)C(C)=O)CCN1C(=O)C(C1CC1)OC 9007,CCC(CC(=O)NCC(C)(C(C)C)NC(c1cnn(CC)c1)=O)C1CC1 9008,C(=O)(CCS(=O)(=O)C1CCCC1)NCC(CC)NC(C1CC(OC)C(OC)C1)=O 9009,C1(CNC(CSCC)=O)CCN(C(=O)CCn2cc(Br)c(C)n2)C12CC2 9010,Cc1nc2ncccc2cc1C(=O)NCC(O)CN(C)C(c1nsnc1O)=O 9011,c1(OC)ccc2[nH]c(C(N3CCC(CNC(=O)CCc4cnc[nH]4)C3)=O)cc2c1 9012,Cc1coc(C(c2nnnn2CCCOCC2CC2)NCC2CCCC2O)c1 9013,C=C(C)C(O)CC(=O)N1CC=C(CNC(=O)C(CO)NC(N)=O)CC1 9014,c1(C(N(C)CC2(N(C)C)CC2)=O)c(Cl)nn(C)c1Cl 9015,C1(NC(c2ccc(OC)cc2Br)=O)CC2CCCC(C1)N2C(=O)C(C)O 9016,c1(C(N2CC(C)C(NC(c3cccc(Cl)c3)=O)C2)=O)ccc2c(c1)CCCCS2 9017,C#CCCC(C(=O)N1CCC1C(C)O)NC(c1cnccn1)=O 9018,C1(C(N2C(CNC(c3c(C)cccc3Cl)=O)CCC2)=O)CC2CCCN2C(=O)N1 9019,N1(C(C(CC(C)C)NC(N)=O)=O)CCC2CCC(NC(=O)CCc3cnn[nH]3)C12 9020,c1(C(=O)NC2(CC=C)CCN(C(CCOCC#C)=O)C2)ccnc2[nH]c(O)nc12 9021,C1(CC(=O)NCC(C(C)C)(C)NC(=O)CCC2CCCCC2)NC(=O)CNC1=O 9022,C(C)(CN=C(NCC(F)F)N1CCC(C(N)=O)CC1)C1CCC(C)CC1 9023,c1(CCC(=O)NC(CCNC(COC(C)C)=O)C)cnc2cc(Br)ccn12 9024,c1(C(=O)NCC2CN(C(c3ccc(NC)cn3)=O)C2)oc(S(N)(=O)=O)cc1C 9025,C1(C(=O)NCC(c2nccs2)C)CCN(C(=O)CN2C(=O)CCC2=O)O1 9026,CC1=Nc2ccccc2C12CCN(C(C1CC3(CC3)CN1C)=O)CC2 9027,c1(OC(C)C)ccc(Cl)c(C(=O)N(C(CNC(C2(O)CCSC2)=O)C2CC2)C)n1 9028,c1(C(=O)OC)nc(C)n(C)c1NC(C1CC2(CC(NCc3cncs3)C2)C1)=O 9029,C1(C(=O)NC(C(=O)NC(CN(C(C)C)C)C)Cn2cncn2)CCCSC1C 9030,c1(CC(=O)NC2CCC(CNC(CCCC#C)=O)C2)ccc(OCC)c(OC)c1 9031,C(CC(CNC(=O)COCCOC)OC)NC(CC=CCC)=O 9032,C1(NC(c2cc(C(=O)OC)nn2C)=O)CN(C(c2ncncc2F)=O)CC12CC2 9033,N1(C(C2C(C)CC2)=O)CC(NC(=O)COc2ccon2)C(F)C1 9034,c1(C(N2CCC(C3N(C(COC)=O)CC3(C)C)CC2)=O)cc(F)cnc1O 9035,c1(COCC)nc(C)c(C(=O)NCC(C2CC2)NC(=O)CCCC2(C)N=N2)s1 9036,Cc1ccc(NC(=O)C(F)CC2CN(C(c3cocn3)=O)C2)cn1 9037,C12(C(=O)NCC(C#C)CC3(NC(C)=O)CC3)CC(CN(C(=O)OC(C)(C)C)C1)C2 9038,C=CCCCCCC(=O)N1CCC(C)(C)CC1C(=O)NCC1CCC(C)(C)CC1 9039,N(C(=NCC)N1CCN(C(C)=O)C(C)(C)C1)C(C#C)(CC)CC 9040,C1(F)(CNC(C(C)OC2CCCC2)=O)CCCN(C(C2CC3CC3C2)=O)C1 9041,C(=O)(C(C(C)C1CCCC1)N1CCCC1)NCCCSC 9042,c1(C(=O)NC(CC(C)NC(C2CCCC(C(F)(F)F)C2)=O)C)cc(N)ccn1 9043,Cc1cccc2[nH]cc(CC(=O)N(C)CCNC(C3CC4(C3)CC(C)C4)=O)c12 9044,c1(C(=O)OCc2cc(Cl)cc(Cl)c2Cl)ccc(S(=O)(=O)NC2CC2)o1 9045,Cc1nc2cc(C(N3CC4CC(NC(c5cccc(Cl)c5F)=O)C4C3)=O)[nH]c2s1 9046,S(=O)(=O)(c1ccc(C(=O)NC2CCN(C(C34CC(C)(C3)C4)=O)C(C)C2)cc1)NC 9047,C(c1c(C)nn(C)c1Cl)=CC(N1CCCC(NC(CC)=O)(CO)C1)=O 9048,C(N=c1[nH]c(=NCc2cc(C(F)F)n[nH]2)c2ccccc2[nH]1)C1(C(N)=O)CC1 9049,c1(C(N(C)CC2(CNC(=O)C(C)(Cl)Cl)CC2)=O)cc2cccnn2n1 9050,C1(O)(C(=O)OCC)CCN(C(=O)CCN2CCN(CCO)CC2)CC1 9051,c1(C(=O)NC(CCNC(Cc2c(C)ccc(C)c2)=O)C)ncc(Cl)c(N)c1Cl 9052,c1(CN2C(CC(=O)Nc3ccc(F)c(O)c3)CCC2)cnc2ncccn12 9053,c1(C(C)C)ccc(SNCc2cnn(C)c2)cc1OCC(F)F 9054,N1(C(C(C)C2CCC2)=O)CC2CC(NC(C3C4CCCCCCC34)=O)CC1C2 9055,C1(C(=O)NCC2C(CNC(c3ccn(C)n3)=O)C2)C2CCN1CC2 9056,C1(NC(CC2CCC(C)(O)CC2)=O)CN(C(=O)C(C)(C)F)CCC12CCC2 9057,c1(CC)ccc(OC)c(C(=O)N(CCNC(=O)CC(=O)OC)C(C)C)c1 9058,Cc1cc(NC(=O)CN2C(=O)CNC2=O)ccc1NC(=O)CP(C)(C)=O 9059,CC1CN(C(=O)CC2CCCN(C)C2)CCCN1C(=O)CC(C)(C)CN(C)C 9060,C1(CC)CCN(C(=O)C=CC2CCCC2)C1C(=O)NCC1(C(C)(C)O)CC1 9061,C1(CNC(C2CCN(CC(F)(F)F)C2)=O)CC2CC2N1C(=O)CCc1ccccc1 9062,c1(N2CC(c3ccccc3)(CC)OCC2)nc(=NCc2cc[nH]n2)[nH]c2cc[nH]c12 9063,c1(C(=O)NC2C(CNC(=O)C=Cc3ccncc3)CCC2)ncc(Cl)cc1Cl 9064,C#Cc1ccc(F)c(C(N2CCCC2CN(C)C(C2CCCCC2(C)C)=O)=O)c1 9065,n1(CC(=O)N(C)CC2N(C(C(C)OC3COC3)=O)CCC2)cc2ccccc2n1 9066,C(C(CC(=O)N1CCC(F)(CNC(C2COCCOC2)=O)CC1)C(F)F)N(C)C 9067,C1(CNC(C2(C(=O)OC)CC2)=O)CCCC1C(=O)N(C)CCn1cncn1 9068,c1(C(=O)NC2CCCC(CNC(c3ccoc3)=O)C2)ccnc2[nH]nnc12 9069,C1(C(N2CCN(C(CN(C)C(c3cncnc3)=O)=O)CC2)=O)CC2C=CC1CC2 9070,C1(NC(c2c(CC)scc2)=O)C2CC3CN(C(c4c[nH]c(Br)c4)=O)C1C3C2 9071,N1(C(C2SCC=C2C)=O)CCCC(CCC(=O)NCC2(C)N(C(C)=O)CCC2)C1 9072,CN1C(=O)CCCC1C(N1CC(C2(NC(=O)CC3(N(C)C)CCCC3)CC2)C1)=O 9073,C1(OC)CC2(C1)CC(C(=O)NCC(C)(CC(C)C)NC(c1nc(C)oc1C)=O)C2 9074,n1(CC)nnnc1C(C1(COC)CCC1)NCCc1cccn1C 9075,CC1(CNC(=O)CCCCC2CC2)CN(C(C2NC(=O)OC2(C)C)=O)CCO1 9076,c1(OC)c(C(=O)NCC2CCN(C(=O)Cc3csc(=N)[nH]3)C2)[nH]c2ccccc12 9077,N1(C(CC=C=C)=O)Cc2cnn(C3CCN(C(c4coc(Br)c4)=O)CC3)c2C1 9078,C(C(CC)(CC)C(=O)NCCN1CCCC1=O)NC(C(CC#C)O)=O 9079,C(=O)(CC(C)C(C)C)NCC(C1N(C(c2c(C)nc[nH]2)=O)CCCC1)(C)C 9080,N1(C(C2CN(C)C2)=O)CCC(NC(c2cnc(C(F)F)nc2)=O)C(F)C1 9081,c1(N(C(CCNC(C(C)N(CC(F)(F)F)C)=O)C)C)nc2cccnc2s1 9082,C1(N(C)C(C2CC(O)C2)=O)CN(C(C2CC2OC(C)(C)C)=O)CC1C(F)(F)F 9083,c1(OC)ccc(CCCC(=O)OC(C)C(=O)NC2(C(=O)O)CCCCC2)cc1 9084,c1(C(=O)NCC2(OC)CCN(C(c3ccnc(Cl)c3F)=O)C2)c(C)oc(C)c1C 9085,C(CNC(=O)CCCOC1CCOCC1)(C(C)(C)C)NC(Cc1c(C)cco1)=O 9086,C(c1ccc(F)cc1)=C(C(=O)NCCC(CC)(C)O)C 9087,CCC(C)C(C(=O)N1CCC(C)(C)C1C(=O)NCC1(O)CCCCC1)N(C)C 9088,c1(NC(C)=O)ccc(C(=O)NC2(C)CN(C(c3nnn(C)n3)=O)C2)c(Cl)c1 9089,N1(C(C=C=C(C)C)=O)C(C(=O)NCC(=O)NC(C)(C)C)CCC12CC2 9090,N1(C(CCCCOC)=O)CCC=C(CNC(=O)C(C)Cc2ccncc2)C1 9091,Cc1ccc(Cl)c(OC(C)C(=O)NC(C)(C)CCNC(=O)C(C)CF)c1 9092,c1(CCC(=O)NCC(CC)NC(c2cnn(C)c2)=O)ccccn1 9093,O=S(=O)(Oc1ccc(Br)c2c1CCC2)C1COCC1O 9094,N1(C(c2c(CC)non2)=O)CC=C(CNC(=O)CCC2CC(OC)C2)CC1 9095,c1(C(C)=O)cc(NC2CCCN(C(=O)C(C)=CC3CC3)C2)ncn1.C(C)(C)O 9096,C1(NC(C(CC)=CC)=O)CC2CN(C(=O)COc3ccc(SCC)cc3)CC12 9097,CC1(C)C(NC(C2CC=CC2)=O)CCN1C(=O)Cc1cc(-c2ccccc2)on1 9098,C=CCN=c1[nH]cc(C(N2CCN(C(=O)CNC(=O)C(C)SCC)CC2)=O)s1 9099,C1(C(N2CCCC(NC(C(C(C)C)(C)O)=O)CC2)=O)CCC2CCCCN12 9100,C1(NC(C(N2CCN(C)CC2)C)=O)CC(C)CN(C(=O)CCc2cnn[nH]2)C1 9101,C(c1ccco1)=CC(=O)NC(C(=O)NCCOCC#C)C1CCOC1 9102,CN1CCN(C(C2(c3ccon3)CCC2)=O)c2cc(C(F)(F)F)ccc21 9103,Cc1cc[nH]c(=N)c1C(=O)NCC1(NC(=O)CC2CCCC2)CC1 9104,N1(C(COC2CN(C(C)=O)C2)=O)CCC(CCCNC(c2cnc(Cl)s2)=O)CC1 9105,c1(C(=O)NC(c2nnc(C)s2)C)ccc(CNC(C2CCOC2)=O)cn1 9106,Cc1scc(C(=O)NC2CCOCC2C(=O)N(C2CCOC2=O)C2CC2)c1C 9107,C(=O)(C(CC(C)C)N(C)C)N(CCCSc1ccc(C(F)(F)F)o1)CC(=O)OC 9108,c1(NC(=O)NC2N(C(CNC(c3nc(C)sc3C)=O)=O)CC2)cc(Cl)ccc1C 9109,CC(C)(CC(F)F)C(=O)N1CCN(C(N2CCN(C(=O)C(C)(C)C)CC2)=O)CC1 9110,O=C1CCN(Cc2cncc(Br)c2)C(=O)C(CC2CC2)N1 9111,C1(NC(c2cc(C)[nH]n2)=O)C2CC3CN(C(c4ccnnc4)=O)C1C3C2 9112,C(CC(C(=O)N(C)Cc1nc(C)no1)NC(=O)C=CC1CCOC1)OCC 9113,c1(C(C)C(=O)NC2CC2NC(C2COC2)=O)ccc(C(F)(F)F)cc1 9114,C(=O)(CC(C)Cc1cccc(OC)c1)NCC(CC)(C)O 9115,n1(CC(=O)NCCNC(c2c(CC)c(F)ccc2)=O)nnc2ccccc2c1=O 9116,C1(CC)CCCN(C(=O)C=CC(C)(C)OC)C1C(=O)N(C)Cc1ccccn1 9117,C1(C(=O)NCc2c(CCNC(C3CCN(C)C3)=O)ocn2)CCC2(CC2)C1 9118,c1(NC(CN(C(=O)NC(CO)CCO)CCO)=O)csc(O)n1 9119,Cc1c(C(=O)N(CCCNC(C2COCCN2C)=O)C2CC2)c[nH]c1C#N 9120,C(=O)(CC(O)CC(C)C)NC1(CC(=O)NC2CC(CC)C2)CC1 9121,C1(CNC(c2ccc(OC(C)C)cn2)=O)C(C)CCCN1C(=O)C=C(C)C(F)F 9122,C1(C#N)(C(N2CC(C)C(NC(C3(CF)CCC3)=O)C2)=O)CC2C=CC1C2 9123,C1(C(=O)NC(C2CN(C(=O)C(C)Cn3ccnc3)C2)C)CC2(C1)CC21CCC1 9124,C(=O)(CCCCN=[N+]=[N-])NC(C(=O)NCC(C#C)CC)COC(C)C 9125,N1(C(C)C(=O)NCCOCCNC(N)=O)CCCC(c2cn[nH]c2)C1.C1(=O)COC1 9126,c1(-c2n(CCNC(=O)OC(C)(C)C)nc(C3CC3)n2)ccnc(S(N)(=O)=O)c1 9127,N1(c2nc(C)nc(O)c2)CCC2(CCOC2)C(CNC(=O)C#CC(=O)N(C)C)C1 9128,C1(C(=O)N(C)C(c2cncn2C)=O)(C2CC2)CCCO1.CN(CCO)CC1CC1 9129,C1(C(=O)NCCCN(C(C(C)c2cncs2)=O)C)Cc2nccnc2C1 9130,N1(C(C(C=CC)O)=O)CCC(C)(C)C1C(N1CCC(C)(NC(C)=O)CC1)=O 9131,N(C(=NCCCCl)NCC(c1cccc(F)c1)C)Cc1c(C)cc(N(C)C)cc1 9132,C(N=c1[nH]c(=NCC(F)F)[nH]c2cccnc12)c1c(C)nc2ccccn21 9133,Cc1ccc(C(N2CCOC(CC(N3CCN(CCO)C(C)C3)=O)C2)=O)nc1C 9134,Cn1ccc2cnc(N3CCNCC3C(=O)Nc3nc(Cl)ccc3F)nc12 9135,CC1(C)CN(C(=O)COC(F)F)CC1N=c1cc(Cl)nc(C(F)(F)F)[nH]1 9136,C1(N(C(C2CC(C(=O)OC)C2)=O)C)CCC(NC(=O)C(N2CCOCC2)C)CC1 9137,CCC(CNC(=O)CC1CCCCC1NC(=O)CC1CCN(C)C1=O)CC(C)C 9138,CC1(C(=O)NCC2CCCCN(C(c3cncc(Cl)c3)=O)C2)CCCCNC1=O 9139,C1(S(C)(=O)=O)(CNC(=NCCc2cc(C)no2)NCc2cc(C)on2)CCC1 9140,Cc1ccnc(CNC(C23CC(NC(=O)OC(C)(C)C)C2C3)=O)c1 9141,c1(CC)cnoc1C(=O)NC1CC(O)(CNC(=O)CC(C)O)C1 9142,C1(NC(C2CC3(CC(=C)C3)C2)=O)CCC2CC1CN2C(=O)C(c1cnn(C)c1)=O 9143,c1(OC)ccc(CCC(N2CC(F)CC2CN(C(=O)C(C)CO)C)=O)cc1 9144,C(CNC(C1(C#N)CC1(C)C)=O)(CC(C)C)NC(Cc1n(C(C)C)ncc1)=O 9145,CC(=O)C(C)CC(C)C(=O)N1CCC(N(CC(C)C)C(C2CC(C)(C)C2)=O)CC1 9146,N1(C(CC2(C(=C)F)CCC2)=O)CCN(C(=O)Cc2cccc(C)c2)CCC1C 9147,C1(N(C(C23CC(C(C)C)(C2)C3)=O)CC)CC(F)CN(Cc2ccc(OC)cc2)C1 9148,c1(C(=O)NC23CC(C(=O)O)C(C2)C3)ccc2c(c1)nc(O)n2C1CC1 9149,Cn1ccc(C(=O)NC(C2CCN(C(c3cn(CC(F)(F)F)cn3)=O)C2)(C)C)c1 9150,c1(C(=O)NCCCN(C(C2C(C)C2)=O)CCO)cc(F)c2ncccc2c1 9151,CC(C)(O)C(F)C(=O)NCCCCNC(C1CCC2(CCC2)O1)=O 9152,C1(C(C)(C)NC(NOCCCN(C)C)=O)CC2CCC1C2 9153,Cc1nc(C(=O)NC(C)CCCCNC(c2occc2Br)=O)[nH]c1C 9154,C1(OC)CN(C(=O)CC2CCN(C)C2=O)CC1C(=O)NCC1CCC1CO 9155,N1(C(c2c(C(C)C)nn(C)c2)=O)CC(CNC(=O)CN(C)C2CC2)C(C)(C)C1 9156,N(C1CCc2ccc(F)cc21)C(=O)C(F)(F)c1csnn1 9157,N1(C(C2C(C3C(C)C3)C2)=O)CCC2(CCCC2NC(C2CCCO2)=O)CC1 9158,CC(CNC(c1ccnn1Cc1ccccc1)=O)(CO)NC(=O)CC1CCCO1 9159,N1(C(C(C(C)C)(C)O)=O)CCC2CCC(C1)N2C(=O)CCc1nnc(C2CC2)o1 9160,c1(C(=O)NCC(CC)(C)NC(C2CS(=O)C2)=O)nc(Cl)c(Cl)s1 9161,C=C(C)CC(C(=O)NCC=Cc1ccccc1)NC(C1CCOC(C)(C)C1)=O 9162,c1(N2CCC(=C)CC2)ncccc1S(=O)(=O)N1CC2CC3CC2C1C3O 9163,c1(C(=O)NCCC(C)NC(C2CC2C2CCC2)=O)ccnn(C)c1=O 9164,N1(C(C2N(C(c3cc(OCC)n[nH]3)=O)CCC(O)C2)=O)CC(O)CC(C)(C)C1.O 9165,N1(C(c2n[nH]c(C(C)C)c2Br)=O)CCN(C(=O)CC(C)F)C(C)C1 9166,c1(CC)cc2c(NC(C)COC(c3cccc(Cl)c3)C)ncnc2s1 9167,C1(CCNC(=O)Cc2cc[nH]n2)CC(F)(F)CN1C(c1cc(Cl)c(Cl)s1)=O 9168,C12(C(=O)OC)CCC(NC(c3ccnc(-n4ccc(O)nc4=O)c3)=O)(CC1)C2 9169,C(=O)(CN=c1cc[nH]cc1)NCC(c1ccccc1)NC(c1c(C)cnn1C)=O 9170,C12(CNC(C3CC34CCCC4)=O)CCC(CC1)CN2C(=O)COCC1CCCO1 9171,c1(C(C)=O)ccc(C(N2CCN(C(=O)CCCF)C(C)C2)=O)cc1C 9172,C#CCC(CC#C)C(=O)NCC(F)CNC(C1(O)CCCCC1)=O 9173,c1(NC(c2nnnn2C2CCC2)(C2CCCOC2)C)ccccc1SCC(N)=O 9174,Cn1cnnc1CC(=O)N(C1CCN(C(=O)COc2cccnc2)C1)CC1CC1 9175,c1(C(=O)OCC2(OCC)CCOC2)[nH]c2cc(F)cc(F)c2c1C 9176,c1(C(=O)NCC2C(C(=O)NCc3c(OC)cccc3)CCC2)ccc(C)cc1O 9177,C1(OC)(CNC(N2CCCC2C(F)(F)F)=O)CCCCC1 9178,N1(C(c2c(C)snn2)=O)CCC(O)(CN(C(=O)CN2CCCCC2=O)C)CC1 9179,c1(C(=O)NC(CN(C(=O)CC2COCCO2)CC)C)cnc(OC)c(Br)c1 9180,c1(C(=O)NC2C(CNC(C3(CC)CC(C)(C)C3)=O)CC2)nsc2ccc(C)cc12 9181,c1(C(=O)NCC(CC)NC(C2CCCC2(C)C)=O)ncc(F)cn1 9182,Cc1cc(C(=O)NCC2CC(C)CN(C(C3(C)SCCCS3)=O)C2)c(O)nn1 9183,c1(C(=O)NCCCNC(CC2C=NN(C)C2=O)=O)cc[nH]c(=N)c1[N+](=O)[O-] 9184,N1(C(C2(C)N(C(C(CC)N(C)C)=O)CCC2)=O)CC2CC1CN2C(C)=O 9185,c1(C(=O)NC(CNC(c2nc(C)oc2C)=O)C)ccc(F)c2cccnc12 9186,c1(C(=O)NCCC(C)NC(c2c(COC)scc2)=O)cc(C(F)(F)F)nn1CC 9187,c1(C(=O)NC(c2cc(F)ccc2F)CC(=O)OC)ccc(C(N)=O)c(Cl)c1 9188,c1(C(=O)NCCNC(C2CCCCS2(=O)=O)=O)c(F)cc(OC(F)F)cc1F 9189,N1(C(c2c(Cl)cc(C)s2)=O)CCC2(CCCC2NC(c2coc(C#N)c2)=O)C1 9190,c1(OC)cccc(C(=O)NC2CN(C(c3csc(Cl)c3)=O)CC2C)c1 9191,Cc1ccn(C)c1C(=O)N(CC(C)CNC(c1nn(C(C)C)cc1Br)=O)C 9192,C(=O)(CCC(=O)NC1(CF)CCN(C(c2cnoc2SCC)=O)C1)NCCC 9193,C1(C(=O)NCCCNC(C(C(C)(C)C)O)=O)CC(=O)c2cc(Cl)ccc2O1 9194,C1(C(=O)NC(CC=C)CNC(c2n[nH]cc2C2CCC2)=O)COCC1(C)C 9195,C(CC(CC)C(=O)N1CCN(C(c2cc(C)c(Cl)s2)=O)C(C2CC2)C1)=CC 9196,c1(C(N(C)CC2(NC(COCCCCC)=O)CC2)=O)ccnn1CCCC 9197,c1(C(N2CCCC(NC(C(CC)F)=O)(CO)C2)=O)nnn2ccccc12 9198,c1(C(N(C2CCN(C(=O)CC3CCC3=O)CC2)CC)=O)cccc2ccccc12 9199,C1(NC(C=C(C)C)=O)CC2CN(C(C3CCS(=O)CC3)=O)CCN2C1=O 9200,CC(C)CC(C(=O)N1CCC(CNC(c2ccsc2)=O)C(O)C1)C(C)C 9201,N1(C(c2ccc([Si](C)(C)C)s2)C(=O)NC2CC2)CCn2c(cc3ccccc23)C1 9202,c1(C(=O)NC2CN(C(CCN3C(C)CCCC3)=O)CC2O)ccn2nnnc2c1 9203,CC(F)(F)CCC(=O)N(CC(=O)NC1CCC12CCCC2)C1CCC1 9204,C1(NC(c2cn(CCC)nc2)=O)C2CCC1CN(C(C1(CF)CCOCC1)=O)C2 9205,C1(OCC)COCCC1CC(=O)NC1(C)CN(C(c2ccc(COC)o2)=O)C1 9206,c1(CC)nn(C)cc1CNC(=O)CC(C)CNC(=O)CSc1cn[nH]c1 9207,c1(C(=O)NC2CC(NC(C=Cc3c(C)n[nH]c3)=O)C2)nn(C)cc1S(N)(=O)=O 9208,Cc1cc(C(N2CCC(O)(CNC(C3(O)CCOCC3)=O)CC2)=O)cc(C)n1 9209,C1(F)(CNC(Cc2ccc(CCCC)cc2)=O)COCCN(C(=O)CCC#N)C1 9210,C1(C(=O)NCC#CCNC(C2(OC)CCSCC2)=O)CC2(C)CCC1(C)O2 9211,C1(CNC(=O)CSC(F)F)CN(C(C2CC2Br)=O)CC1O 9212,c1(OC)cc(N)c(C(=O)NC2CCCC(N)CC2)cc1Cl 9213,C1(C(=O)NC2CN(C(C(C)(C)c3ccno3)=O)C2)CC1C1CCCC1 9214,N1(C(c2cc(C(C)(F)F)on2)=O)CC2CC1CN2C(C1CCCCO1)=O 9215,c1(C2(C(=O)NCC(CC=C)NC(C3COCCO3)=O)CCC2)ccccc1C#N 9216,Cn1ncc2c(C(=O)NC3(CNC(c4sc(Cl)nc4Cl)=O)COC3)cc(Br)cc12 9217,CC1CN(C(C2CCCS2)=O)CC2(CCN(C(c3ccn(CC#N)n3)=O)C2)O1 9218,N1(C(C2CCC(=O)O2)=O)CCC2(CC1)CC2C(N1CCC(F)(F)C1)=O 9219,C1(CNC(C2CCCCN2C(c2ccc(-c3ccco3)o2)=O)=O)CCC(O)CC1 9220,N1(C(C#CC(C)(C)O)=O)CC(NC(C2CC3C=CC2C32CC2)=O)CC(F)(F)C1 9221,CN1C(=O)CN(CC(N2CC(CNC(=O)CC3CCCOC3)CC2(C)C)=O)C1=O 9222,c1(C(=O)NCC(C)CN(C(=O)CCSC(F)(F)F)C)[nH]cc2c1CCS2(=O)=O 9223,C1(SC)CCN(C(=NCC(C)C)NC2CC(NC(=O)OC(C)(C)C)C2(C)C)C1 9224,c1(C(N)=O)cc2cc(C(N3CCC(OC4CCNC4)CC3)=O)ccc2[nH]1 9225,c1(OC)c(C(=O)N(C)CCN(C)C(c2ccc(N(C)C)cc2)=O)cc(F)cc1F 9226,CCCCCCNC(=O)C(c1cnc(C)[nH]1)N1CCC(c2ccnn2C)C1 9227,Cc1ccc(C(N2CC3C(N(C(=O)CC4CC5CCC4O5)C)C3C2)=O)cc1C 9228,C1(CC(=O)NCc2cnc(CC)[nH]2)CCCN(C(=O)Cc2cnc(C)o2)C1 9229,C1(O)(CCNC(COCC(=O)OC)=O)CCN(C(C2CCCCC(=O)N2)=O)CC1 9230,C(=O)(CC(C)(F)F)N(C1CCC(NC(c2c(C(C)C)occ2)=O)C1)C 9231,C1(C(N(CCNC(C=CCC)=O)CCOC)=O)CCCCN1Cc1ccc(Cl)nc1 9232,CC1(C)C2CN(C=O)C(C(=O)O)C12.C1(NC(C)(C)C)C2C3CCC(C3)C12 9233,C1(C(=O)NCC2CCCCC2NC(C2(CO)CCCC2)=O)CCn2ccnc2C1 9234,C1(C(C)C)(C(=O)N(C(C)CCO)C)CCN(C(C2CCC2C)=O)C1 9235,C1(CC(N)=O)(NC(c2ccc[nH]2)=O)CCN(C(c2n[nH]c(C(C)(C)C)n2)=O)CC1 9236,N1(C(c2ccc(F)cc2)=O)CCCC(C2CCCCN2C(=O)Cc2cc[nH]n2)C1 9237,c1(OC)nc(C(=O)NC(CCN(C(=O)C(O)C(F)(F)F)C)C(C)(C)C)ncc1F 9238,C1(C(=O)NCCC2(NC(Cc3cn(C)nc3)=O)CC2)CNC(=O)CC1C(F)(F)F 9239,N1(C(COC2CCN(C(C3(CO)CC(C)(C)C3)=O)C2)=O)CC2CC3CC2C1C3 9240,C(C)(C(=O)NCC(C)(C1CCC1)NC(=O)C=CC(C)(C)SC)OCC=C 9241,C1(CNC(c2ccn(C)n2)=O)CN(C(=O)CCc2cc[nH]n2)CCC12CCOC2 9242,c1(C(N2CCC3(C(C(=O)Nc4ccnc(O)c4)C3)C2)=O)ccc2occc2c1 9243,N1(C2CCN(C(CN(C)CCO)=O)C2)CCC(NC(=O)CC2(C3CC3)CC2)CC1 9244,Cc1cc(C(=O)NC2C=CCN(C(C3COC(=O)O3)=O)C2)nn1C1CCCCC1 9245,C(C(=O)NCC1(C(=O)NC2(C)CCCS2)CCC1)(C(C)C)NC(C(C)C)C1CC1 9246,N1(C(Cc2nc(C)on2)=O)CCC2(CC1)CC2C(N1CCCC(C)C1)=O 9247,Cc1nccc(C(=O)NCC2COC(CNC(=O)CSc3n[nH]c(=N)s3)C2)n1 9248,N1(C(C(CC)F)=O)CC23CCCC2(C1)CN(C(c1c(C)cc(C#N)cc1C)=O)C3 9249,C1(C(=O)OCC)C(C(=O)OCCCNC(=O)OC(C)(C)C)C2CC1C(O)C2O 9250,C1(CC)CN(C(C2(C(=O)Nc3ccc(COC4CC4)cn3)CC2)=O)CCO1 9251,c1(C(=O)NC(CC#C)C(=O)NC(C)(CC)CCC)cc(C#C)ccn1 9252,c1(OC)cc(C(=O)NC2CC(CNC(C3CN(C4CCOC4)C3)=O)C2)ccc1C 9253,C#CCC(C)(C(=O)NC(c1nnc(O)o1)C)NC(=O)CCOCC(F)F 9254,c1(C(N2CCN(C)CC2C(=O)NC2CCCCC2C#N)=O)ccc2[nH]ccc2c1 9255,n1(CCCOC)c(N2CCCC(OCCOC)C2)nnc1C 9256,C1(C)(NC(CSCCCC)=O)CCN(C(c2nnn(C)c2C)=O)C1 9257,c1(C(=O)NC2(C(=O)NCc3ccncn3)CCSC2)cn2ccccc2n1 9258,c1(C(N2CCC(O)(CNC(c3ncc(C)nc3)=O)C2)=O)cccc(O)c1C 9259,N1(C(Cc2ccn(CC)n2)=O)CCC(NC(c2cnn(C3CCC3)c2)=O)C(O)C1 9260,c1(C(C(=O)NC2CC(F)(CNC(CCC(C)C)=O)C2)(F)F)cc(Cl)ccc1Cl 9261,N1(C(c2n(CC)ncc2)=O)CC(CC(=O)NC(c2cnsc2)C)C(C)C1 9262,N1(C(c2cc(C)sc2)=O)CCC2(CCCN(C(c3n[nH]c(C)n3)=O)C2)C1 9263,C(=O)(C1=CCCCO1)N(CC(c1ccccc1)NC(CCNC(=O)C=CCl)=O)CC 9264,C1(C#N)(C(=O)NC2CCN(C(C(C)(C3CC3)OC)=O)C2)CCSCC1 9265,c1(CN(CCCNC(c2cc(CO)on2)=O)C(C)C)ccncc1Cl 9266,Cc1nn(C)c2ncc(CN3CCCC3c3ccc(Br)cc3)cc12 9267,C=CCC(C)(O)C(=O)NCCC(O)C(N1CCCC2(C1)N=N2)=O 9268,Cc1ccc(CS(N2CC(NC(c3oc(C)nc3C)=O)C(F)C2)(=O)=O)cc1 9269,C1(C)(C(=O)OC)CC(C(=O)OC)CN1C(c1cc(Br)ncc1Cl)=O 9270,CS(=O)(=O)c1ccc(O)c(C(=O)NC2(CNC(C3CCC4CC4CC3)=O)CC2)c1 9271,CCC(CC)C(=O)N(CCNC(=O)CCCc1cc(C)sc1C)CCOC 9272,C1(c2nnnn2CCCF)(NC2C(C(N)=O)CCCC2)CCC2(CC1)CSC2 9273,C=CCCCC(=O)NCC(C)CN(C(=O)C=C1CCC(C)CC1)C 9274,c1(C(N2CCC(NC(CCCC(=C)C)=O)CC2C)=O)cnc2[nH]nnc2c1 9275,c1(OCC(=O)NC(CC)(C)CNC(=O)CN2CCCC2C)cc(F)ccc1F 9276,c1(C(N(CCC)CCNC(=O)CC2C(=O)NN=C2C)=O)cccc2c1COC2 9277,C1(F)(CNC(c2cnn(CCN(C)C)c2)=O)CC(CNC(C2CC23CC3)=O)C1 9278,N1(C(C2(OC)CCCCC2)=O)CCCC(O)(CNC(=O)CCn2ccnn2)CC1 9279,c1(C(N2CCC(C3(NC(C4CCCSC4)=O)CC3)C2)=O)[nH]c2ccccc2c1Cl 9280,N1(C(C2CC(c3cccc(O)c3)C2)=O)CCC2(CC1)CN(C(c1ccns1)=O)C2 9281,c1(OC(C)C)ccc(S(=O)(=O)NC2CCNC2CO)cc1F 9282,C1(C)(C(=O)NCC#CCNC(c2n(CC)ccc2)=O)CCCC1O 9283,c1(C(=O)NCC(N(C(C(C)S(N)(=O)=O)=O)C)C2CC2)c(Cl)ccc2ccncc12 9284,C1(c2ccccc2)(N)CCCCC1.c1nnnn1C1(C2CCCO2)CC1 9285,c1(CNC(CC(CC)C2CC2)=O)ccc(CNC(=O)CC2CCCC2C)c(F)c1 9286,c1(C(CCSN2CCCC2=O)NC(N(CCCO)CC)=O)ccc(F)cc1 9287,CON(C)C(=O)CC(C)(C)N(C)C(C1CC(=O)NC1(C)C)=O 9288,CCCCCC(C1CC1)NC(C1CCCCN1C(=O)CSC(C)C)=O 9289,C12(N)CCCC1(C(=O)OC)C2.CCCC(C)=CC(=O)NCCCN(CC)CC 9290,c1(C(=O)NC2C=CC(CNC(c3noc(CC)c3C)=O)C2)ccc(N)c(N)n1 9291,N1(C(COCC)=O)CC2CC2(CNC(=O)C(C)NC(c2cc(C(C)C)no2)=O)C1 9292,C(C(C)CC(=O)N1CCC(C2CCCN2c2nnc(CC3CC3)s2)C1)SC 9293,CC(C)CC(O)C(=O)N1CCN(C(=O)CCNC(c2ccco2)=O)C(C(F)F)C1 9294,C1(C(N2C(C(=O)NC(CNC(=O)OC)C)CC(C)C2)=O)CN(C)CCN1C 9295,C(=O)(C1=CC2(CCN(C(=O)C(CO)OC)C2)C1)N(CC(=O)NC)CC=C 9296,c1(C(=O)NCCC2N(C(CNC(=O)OC)=O)CCSC2)cn(C)c(=O)cc1C 9297,C1(CNC(C(C)C)=O)CCC12CN(C(=O)CC(C1CC1)NC(=O)OC(C)(C)C)C2 9298,C1(C(=O)NCCCN(C)C(C2CN(C(=O)C=CC(=O)NC)C2)=O)CCC=CCCC1 9299,C1(CC(=O)NC(C2CCN(C(C=CSC)=O)C2)C)COCCOC1 9300,C12(C(N3CCC(NC(C4(COC(C)C)CC4)=O)CC3C)=O)CCCN(CCC1)C2 9301,C(=O)(C1SCCc2ccccc21)NC1CC(C)N(c2cc(Cl)ncn2)C1 9302,CC1(C)CN(C(c2ncc(F)cn2)=O)CCC1NC(c1sc(F)cc1Cl)=O 9303,C1(NC(=O)COCCF)CCC(NC(C2CCOC2)=O)CC1 9304,CCC(C)C(O)C(C)C(=O)NCC(C(=O)NCC1(N(C)C)CCCC1)N(C)C 9305,c1(C(=O)NC23CC(CNC(C=C4CCC(C)C4)=O)(C2)C3)cccc(S(C)=O)c1 9306,c1(C(=O)NCC2CCN(C(CS(=O)(=O)NC)=O)C2(C)C)cc2ccsc2c(O)n1 9307,CCC(CC(C)C)C(=O)NCC1(c2ccccc2)CC(NC(=O)CS(=O)(=O)CC)C1 9308,c1(CNCC2C(c3ccc(C)cc3)OCCC2)cccn(C)c1=O 9309,C=CCCCCC(=O)NCCC1CSCCN1C(c1cc(C)n(C(C)C)n1)=O 9310,CC1CCCN(C(c2cncc(CO)c2)=O)C1CNC(=O)C(F)=CC1CC1 9311,C=CCC(C(=O)NC1(C)CSC1)NC(=O)Cn1ncnn1 9312,CCC(CC(=O)N(CCNC(C1(C#N)CC2C=CC1C2)=O)C(C)C)CC(F)(F)F 9313,C12(CC(=O)NCC3CCN(C(C45CC6CC4C5C6)=O)CC3)CCC(CC1)C2 9314,N1(C(CSCC=C)=O)CC2CN(C(c3cccc(C4CC4)c3)=O)CC2C1 9315,C(=O)(CCCCCNC(N)=O)NC(C1CN(C2CCC2)C1)C.c12cc(no1)SC2 9316,C1(N(C(C2C(C)CC=CC2)=O)C)CN(C(=O)C=CCN2CCCC2)CC1(C)C 9317,N1(C(C(C)OC)=O)CCCN(CCc2cn(-c3nc(Br)sc3C)nn2)CC1 9318,c1(C(=O)NC2CCC(CNC(C3(CC=C)CCOC3)=O)C2)cnn2ccncc12 9319,Nc1ccc(C(N2CCC(F)(CNC(=O)CC3CC4(CC4)C3)CC2)=O)nc1N 9320,C(CC(C(=O)N(CC(O)CN(C)C)C)NC(c1ccc(C(C)=O)[nH]1)=O)=CC 9321,c1(C(N2CCC(NC(c3ncccc3Cl)=O)C(F)C2)=O)cc(O)c(O)c(O)c1 9322,C(=O)(C1=CS(=O)CCC1)N1CCCC(F)(CNC(=O)Cc2ccno2)C1 9323,c1(C(=O)NCC(C)N(C(=O)C(C)n2cncn2)CC)nn(C)c(=O)cc1C 9324,Cc1coc2ccc(C(=O)NC(CNC(c3ccc4n[nH]cc4c3)=O)CO)cc12 9325,C1(C(=O)NCC2CC(CC)C2)CC(C)(C)CN1C(=O)C(=CC1CCCC1)C 9326,N1(CC)CC(C(N2CC(O)(CCNC(=O)C=CC(C)C)C2)=O)CC1=O 9327,C1(CC(N2CCCCC2)=O)COCCN1C(=O)C(OCC)OC.C1(CCC)CC1C=O 9328,C1(NC(CN2CCC(C)C2)=O)CC2CCC1N(C(C1Cc3ccccc3N1)=O)C2 9329,CCCCCCCNC(C12CC(NC(=O)C=C=C(C)C)(C1)C2)=O 9330,O=C(C1=CCCS1)NCCOC1CCN(C(=O)C(F)=C2CCC2)CC1 9331,Cc1nn(CC(N2CCC(N(C)C(c3cc(F)c[nH]3)=O)C(C)C2)=O)c(=O)n1C 9332,C1(O)(CNC(c2cc(Cl)cs2)=O)CCN(C(c2sccc2C(F)F)=O)C1 9333,CCC(CC(=O)N1CC(OC)C(NC(=O)C(C)(C)n2cccn2)C1)OC 9334,c1(C(N2CCCC(n3ccnc3CC)C2)C(=O)NCC(=C)C)sc(Br)nc1Cl 9335,C1(C(N2C(CCNC(C3(F)CCOC3)=O)CC(OC)C2)=O)CCc2nnnn2C1 9336,N1(C(C=C(CC)C)=O)CC(C2(NC(c3ccc(N(C)C)cc3)=O)CC2)C1 9337,N1(C(c2n(C)c(=O)ccc2)=O)CCC2(CCOC2)C(CNC(C2(F)CC2)=O)C1 9338,c1(-n2c(C(c3nc(C)sc3)C3CCCCC3)nc(C3CCC3)n2)ccc(F)c(C)c1 9339,Cc1ccc(OCC(=O)NCC2(F)CCN(C(=O)CCC#N)C2)c(F)c1 9340,c1(OC)ccc(CCC(N2CCC(CNC(=O)C=CC3CC3)C(C)C2)=O)cc1N 9341,CC1CC(C(=O)NCC2CC(NC(c3nc(N(C)C)nc(=N)[nH]3)=O)C2)=NO1 9342,N1(C(C(CC=C)NC(C)=O)=O)CCCC12CCN(C(C1CCCN1C)=O)CC2 9343,N1(C(CC(C)C2CCCC2)=O)CC2(C1)CN(C(c1cc(C#N)c[nH]1)=O)CC2CO 9344,c1(C(=O)NCC#CCNC(C(CCCC)CC)=O)cc(S(=O)(=O)CC)cnc1O 9345,c1(OC)ccc(C(N2CC(C(F)Cn3cc(CC(O)C(C)C)nn3)C2)=O)cc1 9346,CC(CCCCCO)NC(=O)C(C1CCCC1)NC(=O)C=CC1(C)COC1 9347,C1(C(=O)NC(CC)CNC(=O)C(c2cnn(C)c2)=O)CCCCC1(F)F 9348,C(=O)(CCC(=O)NC)NCC1N(C(CC2(C=C)CCC2)=O)CC1 9349,C1(NC(C2CC2C(N)=O)=O)CC2CN(C1)C2=O.c1(C(=O)OC)sccc1C 9350,N1(C(c2cc(C)nn2C)=O)CCOCC(C(N2CC3CC2C3)=O)C1 9351,c1(C(CC)C)cc(C(=O)N(C2CN(C(c3cc(Cl)no3)=O)C2)C)on1 9352,c1(C(=O)NCC(O)CNC(c2cc(C(F)(F)F)ccn2)=O)cc2sccc2[nH]1 9353,C(=O)(N=c1ccn(CCF)[nH]1)N1C(C)(C)CC(NC(=O)CCc2cn[nH]c2)C1 9354,c1(C(N(C2CCN(C(c3ccnnc3O)=O)C2)C)=O)cc2scc(Cl)c2[nH]1 9355,Brc1cc(CNCC(N2CCc3sccc3C2)c2ccccc2)cc2c1OCO2 9356,c1(OC)cccnc1C(=O)N(C1CCCC(C)C1)C1CC2CC1CN2 9357,C1(C(=O)NCCCN(C(CCCC(CC)C)=O)CC)CCOC2(CCOCC2)C1 9358,C12(NC(=O)CCNc3ccccn3)CCN(C(=O)CCC3CCOCC3)CC1C2 9359,Cc1nc(C2CC2)nc(C)c1C(=O)NCCNC(=O)CC(C)(C)c1ccccc1 9360,c1(C(N2CC(O)(CNC(c3c(OC)cccc3)=O)C2)=O)cnc(C)nc1C 9361,c1(NC(=O)NCC2CCN2C(=O)C(O)CN2CCCC2)ccc(N2CCC2)nc1 9362,Cc1c(-c2cn(CC3(O)CCN(C(C4CC=CCO4)=O)C3)nn2)cnn1C 9363,C(CCC(=O)NC1CC(F)(C(=O)NOCC(N)=O)C1)SC 9364,c1(C(=O)NCC(CC)NC(=O)Cc2ccc3sccc3c2)cccc2c1NCC2 9365,c1(NC(CSCc2nc(C(C3C=CCCC3)C)on2)=O)ccc(F)cc1 9366,C12(C(=O)NC3CCN(C4CCN(C(CSC)=O)C4)CC3)CC=CC(C1)OC2 9367,N1(C(C2(C=C)CCC2)=O)CCN(C(=O)CCn2cccnc2=O)C2CCCCC12 9368,C(=O)(C(=O)C(F)(F)F)N1C(C(C)(C)NC(C(CC)OCC)=O)CCC1 9369,c1(C(N2CC(C)N(C(c3cncc(Cl)c3)=O)CC2)=O)cc2cccc(O)c2[nH]1 9370,c1(C(N(CC(C)NC(=O)Cc2cc[nH]n2)C)=O)nc(=N)[nH]c2ccccc12 9371,C(=O)(CC(C)(C(F)(F)F)N(C(C)=O)C1CC1)N1CC(C)C(CCN(C)C)C1 9372,C1(c2n(C)ccn2)CCCC(c2nnnn2C2CC2)(NCCn2cccn2)C1 9373,c1(-c2cnc(C(=O)Nc3c(C(C)C)cccc3)nc2)cccc2c[nH]nc12 9374,N1(C(C(c2ccccc2)C)=O)CC=C(CNC(C2CC2Cl)=O)CC1 9375,c1(N2CC(Cl)(Cl)N(CC)CC2)nccc(=NC2CC3CSCC3C2)[nH]1.C1CC1 9376,N1(C(CN2CC(C)C2)=O)CCCC1C1(O)CN(C(=O)C=CC2CCC2)C1 9377,N1(C(CSCC#C)=O)CCC(C(F)Cl)C1.C1(CC(F)F)(C(N(CC=C)CCO)=O)CC1 9378,n1(CC)nnc(C(=O)NCCC2(NC(c3ccnn3CCF)=O)CC2)c1C 9379,N1(C(C2C3N(C(C(COC)(C)OC)=O)C(CC3)C2)=O)CC2CCCC(O)C2C1 9380,c1(CC)cc(NC(=O)NCC(N2C(=O)CCC2=O)OC)ccc1F 9381,c1(OC)ccc(CN2CCC(NC(N(C)CC3CNCCOC3)=O)CC2)cn1 9382,Cc1ccc(CC(C(N2CC(NC(C3CCC3)=O)CC(C)C2)=O)N(C)C)c(C)c1 9383,S(=O)(=O)(c1ccc(=NCCC2CC2C(F)(F)F)[nH]c1)NCC(n1cccn1)C 9384,c1(CCN=C(NC(CC)C)NCC2CCOC2)c[nH]c2ccc(OC)cc12 9385,c1(OCC(=O)NC(CNC(CN(CCCCCC)C)=O)CO)cc(Cl)ccc1C 9386,Cn1[nH]cnc1=NC(=O)NCc1ccc(OC(F)F)cc1 9387,C1(N(C)C)CCC(C(=O)NCCNC(=O)Cn2ccnn2)C1 9388,C12(NC(C(C)O)=O)CCC(CC1)N(C(c1cnncc1C(F)(F)F)=O)C2 9389,c1(CC2CN(C(c3ccon3)=O)C2)ccc(COOC(F)(F)F)cc1 9390,C1(NC(Cc2n(C)nc(C3CC3)c2)=O)CCCCC1N=c1ccnc(C2CC2)[nH]1 9391,C(=O)(CCC(C)(C)[N+](=O)[O-])NC1(C(N(C2CC(CO)C2)C)=O)CC1(C)C 9392,Cc1ccc(CNC(CN(CC(=O)OCC2NCC2(C)C)C)=O)cc1.C(C)(C)(C)O 9393,C#CCCCC(C)C(=O)N1CC2CC2(C(N2CC(O)CC2C(C)C)=O)C1 9394,c1(OC)cnc(F)c(C(N2CC(F)(F)CC2CNC(=O)C=CC2CC2)=O)c1 9395,C(=O)(C1CCCc2n[nH]cc21)NC(CCNC(CCOCCOC)=O)(C)CC 9396,C(=O)(C(C)(O)C(C)(O)C(=O)N(CC(=O)NOCCC1CC1)c1ccccc1)OC 9397,C(C(C)C(=O)N(C(c1ccccc1)CNC(c1cnc(C)s1)=O)C)OC 9398,C1(CNC(c2c(C)nn[nH]2)=O)C(C)CCN1C(=O)CSCc1cccc(Cl)c1 9399,Cc1cc(C(=O)NCC2CC(NC(=O)C(c3ccc(Cl)cc3Cl)O)C2)nc(O)c1 9400,N1(C(CC(CC)c2ccc(C)cc2)=O)CC2CC1CC2NC(C1(C)CCC1)=O 9401,c1(OC)c(F)ccc(F)c1C(N1CCC(NC(C2CCc3ncsc3C2)=O)C1)=O 9402,C1(C)(CNC(C2OCCN(C(c3cc(C(C)C)[nH]n3)=O)C2)=O)CC2CCC1C2 9403,C(C1CC1)(C1CC1)=CC(N1CCC(O)(CNC(C2(c3ccno3)CCC2)=O)C1)=O 9404,C(=O)(C(C)C(C)C)N(C1CCN(C(c2ccc(Br)cn2)=O)CC1)CCC 9405,N1(C(C(CC)OCC)=O)CCC2(CC1)CC2NC(=O)CCc1cccnc1Cl 9406,C12(CC(N3CCCN(C(C4(C)C(C)CCCC4)=O)CC3)=O)CCC(CC1)C2(C)C 9407,CC1CC(=O)NC1C(N1CC(CO)(NC(c2cnc(Cl)cn2)=O)C1)=O 9408,Cc1cn2c(CC(=O)NCC(C)C(F)C(=O)NC34CCC(CC3)CC4)csc2n1 9409,Cc1cc(C(N2CC(NC(c3c(C)n[nH]c3C)=O)C3CC23)=O)sc1C 9410,N1(C(C(CCCCC)O)=O)CC2(C1)CN(C(c1cnn(CC)c1)=O)CC2CO 9411,c1(CN2CCC(C(C)OC)CC2)c(C)cc(F)cc1C.C(=O)C(C)(C)C 9412,c1(OCCC)cccc(CNC(=O)C(=O)Nc2cnccc2SC(C)CC)c1 9413,C1(NC(C2(C)COCCO2)=O)CC2CCC1CC2NC(=O)C(c1cccnc1)O 9414,CC(C)(CN1CCOCC1)C(=O)NCC1CC1NC(=O)CCCc1cnccn1 9415,C(=O)(CS(=O)(=O)N1CCOCC1)NCCCN(C(c1cc(C)ns1)=O)C1CC1 9416,CN1C(=O)CC(C(=O)NC2(CNC(=O)CCC(C)(C)C)CC2)C1c1cccs1 9417,C1(N(C(CCN(C(C)=O)C)=O)C)CCN(C(=O)CCc2ccc(O)cc2)CC1C 9418,C(=O)(CCC(F)(F)F)NC1CCCC(CNC(c2c(C)cnnc2)=O)C1 9419,c1(C(=O)OC)oc(C(=O)NCC2CCC(F)C2)cc1C 9420,C(=O)(C1(C)OCCc2ccccc21)NCC(CNC(COCCCC(C)C)=O)C 9421,O(C1CCc2cc(Br)ccc21)C(c1c(C)cccc1F)=O 9422,c1(C(=O)NCC(CNC(=O)CCC2CCCOC2)F)ccc(N(F)F)cn1 9423,C(=O)(CC(C(C)(C)C)NC(=O)C=CC(F)F)NC(C1CCCCC1)C 9424,C1(=O)C(CC2CCCC2)CN1.C(=O)(C(N)c1ccns1)C1(C)CC1 9425,C1(O)(CC(=O)NCC(C)(O)CNC(C2(F)CC=CCC2)=O)CCOCC1 9426,C#CCCCC(C)C(=O)N1CC2CC1CN2C(=O)CC1(O)CCC1 9427,N1(C(C(C=C)O)=O)CCC(C(C)(C)CNC(C2CCCC(CF)C2)=O)CC1 9428,N1(C(CC2(N(C)C)CCC2)=O)CCCCC1CNC(C1C2CCCC12)=O 9429,Cc1cc(C)c(C(=O)NC(C2CCN(C(=O)CCOCCN(C)C)C2)C)c(N)c1 9430,C1(C(=O)NC2(CNC(c3sccc3F)=O)CCC2)CC2C=CCC(C1)C2 9431,N1(C(C(C)=C2CC2)=O)CCC(NC(=O)CN2CCC(C)(C)C2)C(C)C1 9432,C1(C2CC2)(C(=O)NCc2occ(C)c2)CN(C(=O)C(C2CCCCC2)O)C1 9433,c1(COC)nocc1C(=O)NC1CCC1NC(=O)CC1CN(C)C1 9434,C1(C)(CNC(CCc2ccc(C)s2)=O)CCN(C(C2CC(F)(F)C2)=O)C1 9435,N1(C(c2cc(COCC)[nH]n2)=O)CC2(C1)CN(C(=O)C(C)n1cccn1)C2 9436,CCCCCCC(C)(F)C(=O)N1CCC2(CCCOC2)C1 9437,c1(C(N(C)CC2CCN(c3nnc(C(C)(C)C)s3)C2)=O)cccc(N)c1O 9438,C12(C(=O)NCC(C(=O)NCC(C#C)C(C)C)C)CCC(C1)OC2C 9439,N1(C(c2n(CCC)ncc2)=O)CCC(C)(CNC(C2(C)CC2(F)Cl)=O)CC1 9440,N1(c2nc(C(C)C)nc(Cl)c2)C(CNC(=O)C(C)(C)S(C)(=O)=O)CC2COCC12 9441,CCC(C)C(O)C(C)C(=O)NCCC1CN(C(=O)CC2(C)CCCC2)C1 9442,c1(C(N(C2CCN(C(=O)C(C)OCCN(C)C)C2)CC)=O)cc(O)nc(O)n1 9443,c1(C(N2C3CC(CNC(C4CCC(C)C4)=O)(OC3)C2)=O)cc2cccnn2n1 9444,c1(C(=O)NCCOCCCNC(C2(CC)CC2(F)F)=O)cnc(N(C)C)nc1 9445,C1(C(N)=O)CCCCC1NC(=O)C(c1cnn(C)c1)NC(=O)CC1CCCCO1 9446,c1(NC(=O)NCC2CC2(F)F)cc(Cl)ccc1OCc1cccnc1 9447,C=C(C)C1OCCCC1C(=O)NC1CCC(C)(NC(C2OCCO2)=O)CC1 9448,N(C(=NCCCCl)NCC1Cc2ccccc2C1)CC1CCC(C)O1 9449,c1(C(=O)NC2(CCC)CCCN(C(=O)CC(C)CC)C2)ccn2ncccc12 9450,c1(C(=O)NC(CCNC(C(C(CC)CC)C)=O)C)cc(Cl)c2ccncc2n1 9451,C1(NC(C2(CC)CCCCC2)=O)CC2CC1N(C(c1cncc(COC)c1)=O)C2 9452,Oc1ccc(OCCCSc2ccccc2Br)cn1 9453,c1(OC2CC(OCC)C2)ccccc1.C12CC(C1)NC(=O)CC1C(C1)C(=O)NC2 9454,CCCC(CCNC(C1(F)CCN(C(=O)CCC2(C)CC2)C1)=O)C1CC1 9455,C1(NC(Cc2c(C)con2)=O)CCN(C(=O)C(C)N2CCCC2)CC(C)(C)C1 9456,C1(CNC(=O)C(C2CCC2)C2CCC2)C2CN(C(c3occc3F)=O)CC12 9457,C(CC)(C(=O)NCC(COC)NC(c1nnsc1C)=O)OCC 9458,C#Cc1cccc(C(=O)NC2CN(C(c3cc(OC)ns3)=O)CC2C)c1C 9459,Cc1sc(C(=O)NC2(C)CC(NC(C3CN(C4CCOCC4)C3)=O)C2)nc1O 9460,n1(CC)nnc2c1CCC(C(=O)NCC1CCCCN1C(=O)C(C)NC(N)=O)C2 9461,c1(C(=O)NCCC2N(C(C3CC(OC)C3)=O)CCC2)nc2nccc(C)n2n1 9462,c1(SCC)cncc(C(N2CC3CC3C2c2ccccc2)=O)c1 9463,C(=O)(CC(CC)CC(F)(F)F)N(CCNC(CC(CCC)CC)=O)C 9464,N1(C(C)=O)CCC(O)CC1C(=O)NCc1c(-c2cccc(CO)c2)cc[nH]c1=O 9465,CC(C)C(C(=O)N(C)C)NC(=O)C=CCN(C(=O)CCC1CC1(C)C)C 9466,CC1CN(C(c2nc(Cl)c(Cl)s2)=O)CC1NC(c1cccn1C1CC1)=O 9467,N1(C(C=CC=CCC)=O)CCC(C)(CNC(c2cc(C(C)(C)C)n[nH]2)=O)C1 9468,c1(CNC(=O)NC(C(=O)OCCCC)C)ccc(N(C)CCO)nc1 9469,O=C1NC2CSC(CCCCCN3CCC(NC(C4CCCC(O)C4)=O)C3)C2N1 9470,CCC(O)(CNC(=O)N(C1CCCN(CC(F)(F)F)C1=O)CCO)CCCO 9471,CC1SCCCC1C(=O)NCCNC(c1ncncc1Cl)=O 9472,c1(C(CO)NC(c2c(C)nc(CO)s2)=O)cc(F)c(F)c(F)c1.C(C)(C)(C)NC(=O)O 9473,C(=O)(C(C)S(N)(=O)=O)NCC1(OC)CCN(C(C2CC(C)(O)C2)=O)C1 9474,c1(C(N(C(=O)C(=O)C2(c3cncnc3)CC2)C)=O)ccc2n[nH]cc2c1 9475,C(=O)(NNC(=O)c1cccc(Cl)c1)NC(c1cn(C)nn1)C 9476,c1(OC)ccc(C(=O)NC2CC2CNC(=O)Cc2ccon2)cc1OC1CC1 9477,c1(CN2C(C(=O)Nc3n(C)nc(C(F)(F)F)c3)CC(F)C2)cc(Cl)c(O)cc1F 9478,N1(C(C(c2ccnn2C)C)=O)CCCC(CNC(=O)Cc2ccns2)CC1 9479,C1(CC(=O)NCC#CCOC)C2CCCC2N1C(=O)CCc1cnco1 9480,CCCC(C(=O)N1CCOC(CC(=O)NCCC(=O)N2CCCC2)C1)N(C)C 9481,CC(C)(CN=c1nn[nH]n1-c1ccccc1)NC(=O)C1=COCCO1 9482,c1(C(N(CC(CC)NC(=O)C(N2CCC(O)CC2)C)CC)=O)cc(O)n(C)n1 9483,C1(NC(c2c(Cl)cn(C)n2)=O)CN(C(C2CC3(C2)CC3F)=O)CCC1CO 9484,Cc1cccc2c(=O)c(C(=O)NC3CC(CN=c4[nH]nc(C(C)C)o4)C3)c[nH]c12 9485,C(CCC(=O)N1CCCC1C(C)(C)CNC(c1coc(SC)c1)=O)OC 9486,O=C(CC(O)c1ccccc1)NCC(=C1CN(C(=O)CC(O)C2CC2)C1)F 9487,C#CCC(CC(=O)Nc1ccc(CO)c(F)c1)NC(c1cnn(C(C)C)n1)=O 9488,C1(C(=O)NCC(CC)N(C(=O)C(CC(C)C)OC)C)Cc2nnc(C)n2C1 9489,N1(C(=O)C=Cc2cscn2)CCC(F)(C(=O)NCCc2c[nH]nc2O)CC1 9490,CC(C)C(C(=O)NC1CC(Cn2cc(-c3cnn(CCl)c3)nn2)C1)n1cnnc1 9491,Cc1cncc(CC(=O)N(CC(C)CNC(=O)CC2CCN(C)CC2)C)c1 9492,O=C1CCC(C(=O)N2CCC(C(F)F)(CNC(c3c(F)cncc3Cl)=O)C2)=NN1 9493,N1(C(C(C)OCCOC)=O)CCCN(C(C2(C(C)(C)O)CC2)=O)CC1C 9494,c1(C(=O)NC2CCN(C(C(CCC)O)=O)C(C)C2)nc2ccccc2cc1C 9495,C12(COC(CSCCC)=O)CCC(CC1)OC2 9496,N1(C(C(CCO)N(C)C)=O)CCC2(CCCN2C(=O)CS(C)(=O)=O)C1 9497,C12(C(=O)NCCC3(CNC(C=CCOC)=O)CC3)CCCN(CCC1)C2 9498,N1(C(CNC=O)=O)CC2(C1)OC1(CNC(C3CCCCC3O)=O)CC2(C(N)=O)C1 9499,c1(CC(=O)NC2CCCN(C(CCC(C)(F)F)=O)C2)csc2cccc(F)c12 9500,C1(NC(=O)Cn2ccc(C(F)F)n2)CC(O)CN(C(=O)C2=CCCCO2)C1 9501,C#CCC(C)(C(=O)NC(CC(=O)OC)SC)NC(=O)C(CC)CCOC 9502,Clc1ccc(CN(C2CCCC2)CC(c2ccccc2I)O)cc1 9503,c1(C(=O)NCC2(O)CCN(C(c3cc[nH]n3)=O)CC2)scc2c1CCCC2 9504,CC(CN=c1ccnc(N(C)Cc2ccc(Cl)cc2F)[nH]1)Oc1ccccc1 9505,c1(C(=O)NCC23C(CN(C(C4CC(CC)OCC4)=O)C2)C3)cc(F)c(O)c(Cl)c1 9506,c1(CC)nc(C)c(C(=O)NC(C)CC(C)NC(=O)C(c2ccccc2)NC(C)=O)o1 9507,C1(NC(C2(OC)CC(C)C2)=O)CCC(N(C(=O)C(O)Cc2ccccc2)C)CC1 9508,C1(C(=O)OC(C)(C)C)C2CC3C(C2CN(C2CC2)C)C13.C12(OC)CCC(C1)C(=O)O2 9509,C1(NC(C2CN(C(Cn3c(C)ccn3)=O)CC23CC3)=O)CN2CCC1(F)CC2 9510,C=CC(C)(C)C(=O)NCc1cn(CC(=O)NCC2(C)CC2(C)C)nn1 9511,N(C1CCCn2nccc21)C(C(C1CC(C(=O)NCc2cccnc2F)C1)F)=O 9512,N1(C(C(CNC(C=CC=CC)=O)CC2CCCC2)=O)CC2CC(CO)C(C2)C1 9513,CC1CC(N=c2nc(-c3ccccc3)[nH]s2)CCN1C(=O)C(F)n1cccn1 9514,C(=O)(C1COc2ccc(Cl)cc21)NC1C(NC(c2cnc3scnc3c2)=O)C1 9515,C1(NC(Cc2cccc(OC)n2)=O)CCN(C(=O)C2=NNC(=O)C2)C(C)C1 9516,CC1=CCC(C(=O)NN(C(C2C3(CC(CC4CCCC4)C3)C2)=O)C)CC1 9517,N1(C(C2(COC)CC2)=O)CCC(C2CCN(C(C3(S(C)(=O)=O)CC3)=O)C2)C1 9518,c1(OC)cncc(CNC(=O)CC2CCN2C(c2oc(C)cc2C)=O)n1 9519,N1(CC(=O)NCCC2CCN(C(C3(c4cc[nH]n4)CCC3)=O)C2)CCCNC1=O 9520,NCCS(=O)(=NC(=O)c1ccc2cc[nH]c2n1)c1ccccc1 9521,C(=O)(CCC(N)=O)N1C(CC(=O)NCC2C(CC)C2)CC1 9522,C1(C(N(C)CCOc2ccccc2CO)=O)CCCOC12CCC2 9523,C(C(F)(F)C(=O)N(C)CC1CN(C(=O)COCC(C)C)CCO1)OC 9524,C(C(CC(C)C)NC(=O)C(C)OC(C)C)NC(C1(CC)CC1(F)F)=O 9525,c1(N(C(=O)CCc2nc(=N)[nH][nH]2)C(C)=O)cc(Br)ccc1C(=O)NCCNC1CC1 9526,c12ccc(cc1)NC(=O)C(C)=NOCC2.C1(NC)CCC1 9527,Cc1cnn(C)c1C(N1CC(O)(CCNC(c2cnn(C)c2CC(C)C)=O)C1)=O 9528,CC1C(C)N(C(c2cc(C3CCOCC3)[nH]n2)=O)CCN1C(c1cnn(C)c1)=O 9529,c1(COC(C2C(C(=O)OC)COC2)=O)cnc(OC)c(Br)c1C 9530,N1(C(CC2C=CCN(C(=O)C=CC3CCCCC3)C2)=O)CCc2cccnc2C1 9531,C1(F)(C(=O)NCC(C)N(C(=O)CO)C)CS(=O)(=O)CC12CCC2 9532,C1(N(C(=O)C=CC2(C)COC2)C)(C(=O)NCCCC(F)F)CCC(C)(C)C1 9533,CCCC(C)CCCC(=O)N1CCCC1CCNC(C1CCC(=O)N1C(C)C)=O 9534,N1(C(c2ccc(C)cc2)=O)CCC2(CC2C(=O)N(C)CCN(C)C)C1 9535,c1(SCC)cnc(O)c(C(N2CC(NC(C3CC(=O)N(C(C)(C)C)C3)=O)C2)=O)c1 9536,CC(C)CC(F)C(=O)N1C2CCC1(CNC(=O)Cn1ncn(C)c1=O)CC2 9537,N1(CCC(=O)NCC(CCOC)NC(c2nc(CC)oc2)=O)CCP(C)(=O)CC1 9538,N1(C(c2cc(CC)[nH]n2)=O)CCCC(C)C1CCNC(c1cnc(C2CC2)[nH]1)=O 9539,c1(C(=O)NCCCN(C(c2cc(OC)n[nH]2)=O)CC)coc(COC)c1 9540,N1(C(=O)CCN2CCCC2)CCC2CCN(C(C3CSCCS3)=O)CC2C1 9541,C(=O)(CC(C(C)(C)C)NC(=O)CNc1ncccn1)N(CC(C)CO)C 9542,C1(C(N2CC(CNC(C3(c4ccccc4Cl)CCC3)=O)C2)=O)CC(C2CC2)C1 9543,CC1CCc2[nH]c(=NCC3CCCCS3)[nH]c(=NCCC(F)F)c2C1 9544,CCC(CC)C(F)C(=O)NCC1CC(C)CN(C(C2CC3CCC(C2)N3C)=O)C1 9545,N1(C(C2C(=C)C2)=O)CCN(C(c2coc(C(C)(C)C)n2)=O)C(CCO)C1 9546,N1(C(C2(C)CCOCC2)=O)CCC2(CC1)OCCC2NC(=O)CC1CS(=O)(=O)C1 9547,C(C(C)C(F)(F)F)NC(C(CC)NC(C1CCN(C)C1)=O)=O 9548,C1(NC(C2(OCC)CCOC2)=O)COC2CN(C(c3cnn(C)c3C)=O)CC12 9549,c1(C(=O)NC2CN(C(C3CCC(=O)O3)=O)CC(F)C2)ccc2nnc(O)n2c1 9550,C=C1CCN(C(=O)C=Cc2ccn(C)c2)C(C(N2CCC(c3ccon3)C2)=O)C1 9551,C=C(CNC(C1(CC)CCCN(C(=O)C(C(C)C)SCC)C1)=O)c1ccccc1 9552,CC(C)(C)C(C(F)F)NC1COC2(CCC2)C1 9553,c1(C(N2CC(C)CC(NC(CC3(C=C)CC3)=O)C2)=O)ccc(C)c(S(C)(=O)=O)c1 9554,C(=O)(CCC(=O)N1CCC(C)(CNC(c2cc(=O)cc[nH]2)=O)C1)N(C)C 9555,N1(C(CNC(CNC(C)=O)=O)=O)CCCCC1CNC(C1(C#N)CC=CC1)=O 9556,n1(CC(=O)NC(CC(C)NC(C2(C)CC(C)C2)=O)C)cccc(C(F)(F)F)c1=O 9557,N1(C(C=C(C)CNC(C2COC(=O)N2C)=O)=O)CCC(CO)C(O)C1 9558,CC(=NO)C1CC(C(N2CC(NC(c3nc(N(C)C)ccc3Cl)=O)C2)=O)C1(C)C 9559,C1(NC(C2(C3N(C(C=CCC)=O)CCC3)CC2)=O)CCCN(CC)C1 9560,CC1CCC=C1C(=O)NC1(CCNC(c2cn(C)c(=O)n2C)=O)CCC1 9561,c1(C(C(=O)NCC)N(CC2CCCCC2)Cc2ccccc2)nc(CC)cs1 9562,C12(CNC(c3nc(CC)oc3)=O)CC1CN(C(=O)C(C)Oc1ccc(C)cc1)C2 9563,CC1CN(C(C2CN(C(=O)CCc3ccncc3)CCO2)=O)CC1N(C)C 9564,CC1CN(C(=O)CCS(N)(=O)=O)CC(C)N(C(c2ncccc2OC(F)F)=O)C1 9565,c1(C(=O)NCC2(C)N(C(CC3CC(=C)C3)=O)CCC2)cc2n(n1)CC(C)NC2=O 9566,c1(C(N2C(CNC(CCCOCC)=O)C=CC2)=O)noc(C2CC2)c1C 9567,C(=O)(C1=NOC2COCC12)NCC1ON=C(C(=O)NCc2c(C)cncc2)C1 9568,C1(C(N(C2CCCN(C(C=NOC)=O)CC2)C)=O)CC2(CCC(F)(F)CC2)CO1 9569,N1(C(c2cc(C)n(C)c2C)=O)CC(C(=O)NCC2CCC(C)C2)CC(C)(C)C1 9570,c1(C(N2C3CN(C(c4n(C)nnc4)=O)C(C3)CC2)=O)c[nH]c2cccc(Br)c12 9571,c1(C(N2CCC(NC(=O)CC3CCCS3(=O)=O)CC2)=O)ccc(O)c([N+](=O)[O-])c1 9572,CC(C)CC(C(=O)N(C1CCSC1)C)ONC(=O)CC1CCC(C)CO1 9573,c1(N(C)Cc2ccc(C)cc2Br)nc(NCc2cccnc2Br)c2ccsc2n1 9574,C(=O)(C1=CC(C)(C)C1)NC(c1c(C)cccc1)C.C12CCCCC1C(=O)N2 9575,c1(C(=O)OCC)c[nH]ccc1=NCC1CCCCN1C(=O)CC1CC2(CC2)CO1 9576,c1(C(=O)NC2CCCC(N(C(C=C(C)C3CC3)=O)C)C2)csc2c(F)cccc12 9577,C1(Nc2c(CC)cccc2)(NC(N2CCOCC2)=O)CC2(CCC2)C1 9578,c1(CC(N2CC(N(C(CC3N(C)CCC3)=O)C)C(O)C2)=O)cnc2cccnn12 9579,C(=O)(CCS(N)(=O)=O)N(C)Cc1cn(Cc2ccnc(Cl)c2)nn1 9580,C1(N(C)C)CN(C(C2CCCN(CC(=O)OC(C)(C)C)C2=O)=O)CC1(C)C 9581,C(=O)(C#CC(C)(C)CNC(C1(C)CCC(=O)C1)=O)NCCCNC(=O)NC 9582,N1(C(C(C(=O)OC)C)=O)CC2OCCN(C(c3cc(C4CC4)no3)=O)C2C1 9583,C12(C(=O)NC3(CC=C)CCOC3)CC(C)(CN1C(C1(Cl)CCC1)=O)C2 9584,n1(CC)ncc(Cl)c1C(=O)NCC(O)CNC(c1cnn(CCC(C)C)c1C)=O 9585,C1(N(C(=O)C(F)(F)c2cscn2)CCN(C2CCCC2)C(C)=O)CCN(C)C1=O 9586,C1(CN(C(=O)C(O)CSC)CC)CCCCN1Cc1ccc(N2CCCC2)nc1 9587,C1(OC)CC2CCC1CC2C(=O)NC(C)CNC(C1CCCCN1S(C)(=O)=O)=O 9588,C(C(CO)CC(C)C)NC(C1CC(CNC(C=CCOC)=O)C1)=O 9589,N1(C(CCN(C)CC)=O)CCOCC(NC(=O)CCCOc2ccccc2)C1 9590,C(=O)(CS(=O)(=O)C(C)C)N1CCC(NC(C2CN(C(=O)NC)C2)=O)C(F)C1 9591,n1(CC)cnc2c(NCCC(C)NC(=O)OC(C)(C)C)[nH]c(=NC(C)C(F)F)nc12 9592,c1(-c2cc(C)c(CO)cc2)cn2c(n1)CN(C(=O)C(c1cccn1C)=O)CC2 9593,C1(CN(C(C(CC)OCC)=O)C)CN(c2nccc(CC#N)n2)CCO1 9594,N1(C(C2(Cl)C(C)(C)C2)=O)CCN(C(=O)Cc2cncn2C2CC2)C(CO)C1 9595,Cc1cncc(NC(=O)C(N2CCCC(CCNC(=O)C(C)(C)C)C2)C)n1 9596,C(=O)(N1CC(O)C(O)CO1)C1CCC(CNC(c2c(N)c(F)ccc2)=O)C1 9597,C1(OCC)CCCCN(C(=O)CCCC(C)C)C1.c1(CC=O)ccc(C=O)cc1 9598,c1(C(N2CCC(C)(NC(c3c(COC)cccn3)=O)C2)=O)ccc(N)c(Cl)c1O 9599,Cc1ccn(CC(=O)NC(C)CNC(=O)C(C)Cn2cccn2)c(=O)c1 9600,C1(CCNC(C(=Cc2cnc[nH]2)C)=O)CCN(C(=O)Cc2sccc2C)CC1 9601,N1(C(=O)CN2CCCC2)CC2CC1CN2C(C1(C(F)F)CCCO1)=O 9602,C1(CC(=O)NCCSCC=C)CN(C(c2cnc(C)cn2)=O)CCC1C 9603,Cc1ccccc1CCC(N1CCC(CNC(c2cnnn2C)=O)C1)=O 9604,C=C(Cl)CC(C(=O)NCC1(SC)CCC1)NC(=O)CCc1nncs1 9605,Cc1ccc(C(=O)OCCc2nnn(CC(F)(F)F)n2)c2ccccc12 9606,C1(C)(CCNC(c2ncn(C(C)C)n2)=O)CCN(C(=O)CC2CCCC2)C1 9607,c1(C(N2CCC(O)(CCNC(C(C)(C)C(N)=O)=O)C2)=O)ccc(C#N)cc1O 9608,c1(N(C)C)ncnc(Cl)c1F.CC1CC2CN1C(=O)c1cncc(c1)OCCN2 9609,CC(C)(C)CC(O)CC(=O)NCC1CC(C)(C)CN1C(c1cnn(CCF)c1)=O 9610,c1(C(N2CC(NC(C=CC)=O)C(c3ccccc3)CC2)=O)cc(F)c(F)cc1Cl 9611,CC(C)CC(F)C(=O)NCCC(C)NC(=O)CCC(=O)c1cccc(Cl)c1 9612,c1(CNC(c2cccnc2)CC)cc(F)c(C(F)(F)F)cc1F 9613,c1(OC)ncnc(C(=O)NC2(CCCNC(C3CCOC3C)=O)CC2)c1F 9614,Cc1ccccc1C(C)NC(c1oc(CNC(c2ncncc2N)=O)cc1C)=O 9615,Cc1ccc(CCNC(=O)CC2CC(C)N(C(=O)CNC(C3CC3C)=O)C2)cn1 9616,C(=O)(C(C)(C)C(C)(C)C)NCC(CC1CCCCC1)NC(CCCCC=CC)=O 9617,N1(C(C(c2ccc(F)cc2)(C)O)=O)CC2(CCC(CNC(=O)C3CC3)O2)C1 9618,C1(O)(CCNC(=O)NCc2ccc(-c3csnn3)cc2)CCCOC1 9619,c1(C(=O)NC(C(c2ccccc2)NC(C=CCOC)=O)C)ccc(C(N)=O)cn1 9620,N1(C(C(CC#C)C)=O)CCC2(CCC(CNC(C3(C(F)(F)F)CCC3)=O)O2)CC1 9621,CCCC(C)(O)CC(=O)N1C2CCC1CN(C(=O)CN1C(=O)NC(C)(C)C1=O)C2 9622,C1(C)(NC(C2C3C(NC(C(C)C4CCCO4)=O)C4C(C3)C42)=O)CCC(C)(C)CC1 9623,S(=O)(=O)(c1ccc(NCCc2nncs2)c(Cl)c1)NC(CC(C)C)CN(C)C 9624,N1(C(C(CCC=C)(C)C)=O)CCC2CN(C(c3cnc[nH]3)=O)CC2C1 9625,c1(NCC(CC)CO)ccc(S(=O)(=O)N2CCC(C3CCCCC3)C2)cc1Br 9626,C1(C(=O)NCC2(CCC=C)CC2)CCN(C(=O)C2CC3OC2C2CC32)O1 9627,N1(C(c2cnn(C)c2N)=O)CCC(CO)(NC(=O)COCC2CCCC2)CC1 9628,N1(C(c2ccc(CSC)o2)=O)C2CCC1CC(NC(=O)C(O)C(F)(F)F)C2 9629,CC1COCCN1C(c1n[nH]cc1CNC(=O)CCC1CCCOC1)=O 9630,c12ccc3cc(c(F)cc3n1)N2.N1(C(C)=O)CC2CCCC(C1)N2CCN(C)C 9631,Cc1cc(C(=O)NC(C2CCOC2)CNC(=O)COCCF)c2sc(=N)[nH]c2n1 9632,c1(OC)cccc(C(=O)N(CC(C)(C)NC(C2CN(C)CC(C)O2)=O)C)c1OC 9633,CC(C)C(O)C(C)C(=O)N1CCC(CNC(c2coc(CO)c2)=O)C(O)C1 9634,C1(CC)(NC(=O)C(C)CC2CC2)CCCN(C(c2ccc(C)c(C)n2)=O)C1 9635,C=C(Cl)CCC(=O)N1CCCC(C(C)NC(c2cccnc2CC)=O)C1 9636,N#Cc1cc(CNC(C2(F)CCCN(C(=O)CC3CCSC3)C2)=O)ccn1 9637,C1(C(=O)NCC(CC)NC(c2ncnn2C)=O)CN(C)CCN(C)C1 9638,C(=O)(CCN=[N+]=[N-])N1CCC(OCC(=O)N(C2CCCC2)C)C1 9639,CCC(C(=O)N1C2CCC1C(CNC(C1(C3CCC3)CCC1)=O)C2)C(C)C 9640,C=CCCC(CC(C)C)C(=O)NC1(C)CN(C(=O)CC(C)(C)O)C1 9641,C1(C(=O)NCc2noc(-c3cccs3)n2)CCCC2CC12 9642,C1(C(=O)OC)(COC)CCN(c2nnnn2CCCOC2CCCCC2)C1 9643,C1(NC(c2cc(CC)ncn2)=O)CCC(C)N(C(=O)CNC(=O)C(F)(F)F)C1 9644,Cc1ncc(Cl)cc1C(N1CC(N(C)C(C2CCCCC2(C)C)=O)C(O)C1)=O 9645,C=C1CC2(C1)CC(C(=O)NC1CC3(C1)CC(NC(=O)COCC1CCCC1)C3)C2 9646,N1(C(C(n2ncc(C)c2)C)=O)CCC(N(C(=O)C=Cc2cn(C)nn2)C)CC1 9647,C1(C(=O)NCC2(CCOCC)CC2)COC2(C1)CN(C(=O)COCC(C)C)C2 9648,c1(C(N2CCOCC(C(=O)NC3(C)CCC(C)C3)C2)=O)cc2c(s1)CCCC2 9649,c1(C(C)C)nnc2cc(N3CCC(NC(C4(F)CCOC4)=O)C3)ncn12 9650,C(=O)(C(CC(C)CC)NC(C1CCC(=O)O1)=O)N(CC(=O)NCC)C 9651,C1(C(N2C(CC)CCCC2)=O)COC2(C1)CN(C(=O)CCC(CF)CF)C2 9652,c1(NC(C(C)NC(C(CCCOC)C)=O)C(C)C)cc2nncn2cn1 9653,CC(C)CC(C)(C)CNC(C1COCCC1NC(=O)CCCn1ccnn1)=O 9654,O=C(Nn1cnc2ccccc12)C1CCCCN1C(C1C2COCC12)=O 9655,C1(C(N2CC(OCC(=O)NC(COC)CO)C2)=O)C2CCCCC12 9656,c1(C(N(C(C)CN(C(=O)COC2CCOC2)C)C)=O)[nH]cc2c1CCC2 9657,CN=c1[nH]cc(C(=O)OCc2cnccc2C(F)(F)F)s1 9658,c1(CCNC(C2(C(C)C)CCC2)=O)nc2ncccn2n1 9659,c1(C(N(CCNC(=O)Cc2cc(F)cc(Br)c2)CC)=O)ccc2[nH]ccc2n1 9660,N1(C(c2cc(OCC)no2)=O)CC(C)CC1C(=O)NCC(C)CN(C)C 9661,CCC(CC)(CCNC(c1c[nH]c(=N)s1)=O)NC(=O)CC1(C(F)F)CC1 9662,Cc1cc(NC(=O)C(N2CCC(NC(=O)CC3C=CCC3)C2)C)ccc1F 9663,c1(OC)c(NCC2CCN(C(=O)OC(C)(C)C)CC2C)cc(F)cc1Br 9664,c1(C(=O)NC2CCCN(C(CCC=C=C)=O)C2)ccc(N)c([N+](=O)[O-])c1 9665,CC1(CC(=O)NCCOCCNCCN=[N+]=[N-])CCS(=O)(=O)N1 9666,C(=O)(C(C)(C)CC(F)(F)F)NCC(N(C(C(C)OCC#C)=O)C)C1CC1 9667,N1(C(C2CC(C)(C)C2)=O)CCC(C(N2C3CCC2CC(CO)C3)=O)CC1(C)C 9668,Cc1ccc(C(N)=O)cc1C(=O)NC1CC(NC(=O)C(C)(C)CC#N)C1 9669,Cc1ccc(=O)n(CC(N2CCN(C(C3CSC3)=O)C(CC(C)(C)C)C2)=O)c1 9670,c1(C(N2CC(CNC(C3(CC=C)CC3)=O)OCCC2)=O)c(C)nc2ccccn12 9671,C(CN=c1cccc(S(=O)(=O)NC(C2CCCO2)C)[nH]1)c1cccc(OC)c1 9672,Cc1cc(C(N2CC3CC2(CNC(C2(C)CC(O)CN2C)=O)C3)=O)nc(C)n1 9673,c1(C(=O)NC(CCCCNC(c2cccc(C)c2)=O)C)cc(O)ncc1Br 9674,N1(C(C(CC#C)C)=O)CC2CCCC2(NC(=O)CSc2ccc(C)cc2)C1 9675,c1(C(=O)NC(CCOC)C(=O)NC2CCOCC2O)cc(C)nnc1C 9676,C1(C(=O)NCC2CCN(C(c3nnn(C)n3)=O)CC2)CCC2(CCCC2)CC1 9677,n1(C(CC)C)nc(C2OCCc3ccccc32)nc1-c1coc2c(F)cccc12 9678,CC(=O)CCC(=O)N1CCCCC1C(=O)NCC(C)(O)C1(C)CC1 9679,N1(C(=O)NC)CCN(C(c2occc2CNC(C23CC(CO)(C2)C3)=O)=O)CC1 9680,N1(C(CNC(CC)=O)=O)CCCC1C(=O)NCc1ncc(C)[nH]1 9681,O=C(C1CCCc2ncnn21)N(C(CC(F)(F)F)c1cccc(C(F)(F)F)c1)CO 9682,c1(C(N2C(C)(CNC(c3ccc(C(N)=O)s3)=O)CCC2)=O)cc(F)c(F)c(O)c1F 9683,C1(CC(=O)NC)CCN(C(c2cnncc2OC)=O)CC1.C12(NC)CC1C2 9684,c1(OCC)cccc(CC(=O)NCC2(OC)CCN(C(C3CC(OC)C3)=O)C2)n1 9685,C(=O)(C(CC=C)C(C)C)NC(C(=O)NC1CCCC(C#C)C1)CC=C 9686,C1(CNC(COC)=O)CCN(C(c2cc(-c3ccccc3)cs2)=O)C(C)C1 9687,N1(C(=O)CC2CCN(C(c3n[nH]cc3I)=O)CC2)CCC(F)(F)CC1 9688,c1(C(=O)NCCCN(C)C(C2(O)CCSC2)=O)cc(Cl)ccc1Cl 9689,CC1(CCNC(C2(O)CCSC2)=O)CCN(C(=O)COCc2nc[nH]n2)C1 9690,n1(CC(=O)N(C2CN(C(C3CCOC(=O)CC3)=O)C2)C)[nH]cc2c(=O)ncnc1-2 9691,CC1CC(C(N2CCCC(C)(NC(c3ccc(C(C)(C)C)[nH]3)=O)C2)=O)CCC1=O 9692,c1(CN2CCC(NC(c3cc(OC)cc(Cl)n3)=O)C2)cc2cn[nH]c2cn1 9693,N#Cc1ccc(C(=O)NC2CCCN(C(c3csnn3)=O)C2)c(F)c1 9694,N1(C(C=CC(=O)OCC)=O)CC(CNC(=O)C2=C(C)OCC2)CC1(C)C 9695,Cc1oc(C)c(C(=O)NCC2CN(C(=O)CC34COC(C)(C3)C4)CCN2C)c1C 9696,C12(NC(c3c(OC)c(F)ccc3)=O)CCOCC1CN(C(=O)C1=CCCCC1)C2 9697,C12(CNC(c3cc(OC)ncc3)=O)CC3CC(C1)C(O)C(C3)C2 9698,C12(C(N(C)Cc3cn[nH]c3)=O)CC1CCN2C(C1CCSC1)=O 9699,N1(C(C(CCC)CC)=O)CC2CCC(C1)N2C(=O)C(F)Oc1ccc(Cl)c(F)c1 9700,C1(C(=O)NCCN(C2CCOC2)C(c2cncnc2)=O)CC12CCCC2 9701,C1(NC(=O)COCC2CCCC2)CCC(CNC(c2cnnc(O)c2)=O)CC1 9702,C1(NC(CC2(OC)CN(C(C3(C)CC(C(F)(F)F)C3)=O)C2)=O)CC2CCC1CC2 9703,C(=O)(C1=NNC(=O)C1)NC(C)C=CC(=O)NC(C)(C)CCCO 9704,C=CCC(CC(=O)NCCC(O)C(F)(F)F)NC(=O)CC(=O)N(C)C 9705,C#CCCC(C(=O)NCc1ccnc(OC)c1)NC(=O)C(COC)COC 9706,C1(C)(C(=O)NC(CC)CN(C(=O)CCCc2ccc(C)cc2)C)CCCN(C)C1 9707,c1(C(=O)NCC(C)N(C(C(CCCC)C)=O)C)cc(=O)c2cc(F)ccc2o1 9708,C=CCN=c1[nH]cc(C(=O)NC2CCCC(NC(=O)CC3(OC)CCCC3)C2)s1 9709,c1(C(C)(C)OC)ccc(C(=O)NCCC(C)N(C)C(c2nocc2C)=O)cc1 9710,C12(C(N(CCCC)CCCC)=O)COCC1CN(C(C1(C)CNC(=O)C1)=O)C2 9711,c1(OC)cc(F)c(C(c2nnnn2C2CC2)NC2(C)CCSCC2)c(F)c1 9712,C1(C(=O)NC(CC)(C)CC)CN(C(=O)C(O)C(C)C)CC1(F)F 9713,C1(NC(CNC(=O)OC)=O)CC2CCC(C1)N2C(c1sccc1C(C)C)=O 9714,C(=O)(C(CCOC)OC)NCC(C)N(C(c1onc(CC)n1)=O)C 9715,N1(C(CC(C(F)F)NC(CC2C(C)(C)C(O)C2)=O)=O)CCC(O)(C2CC2)CC1 9716,C(C(C)(C)C(=O)NC1CCCC(N(C(=O)C(c2csc(C)n2)=O)C)C1)OC 9717,c1(C(=O)NC(Cc2ccc(Cl)cc2)C(O)C(F)(F)F)ccc2c(n1)CCCC2 9718,C1(C(N(C2CC2)Cc2n(C)ccn2)=O)CCCN(C(c2cc(Br)ccc2Cl)=O)CC1 9719,c1(CC)cnc(C(=O)NCC2COCC2NC(=O)Cc2sc(O)nc2O)cn1 9720,CCCCCC(C1CC1)NC(c1cccnc1CNC(=O)CC1CCOC1)=O 9721,c1(C(=O)NCCC(C)NC(=O)CCc2cnco2)csc(=NC2CCCCC2)[nH]1 9722,C=CCC(C)C(=O)NCC1(C(=O)NC(C)CC(N)=O)CCC1 9723,N1(C(C(CC#C)CC#C)=O)CC2CC3CC2C1C3NC(=O)CC1C=CCCC1 9724,C1(C(=O)NC2CCC(CNC(c3cc(COC)sc3)=O)CC2)CC2CC1CC2O 9725,C1(CC=C)(NC(=O)C=CC(F)(F)F)CCN(C(C2CC(C(F)F)C2)=O)CC1 9726,C1(CCOC)(C(=O)NC(C)CF)CCN(C(=O)CC2CCC(=O)C2)CC1 9727,C1(NC(c2nc(CCC)sc2)=O)CN(C(C2(OC)CCCCC2)=O)CC1O 9728,c1(C(=O)NCCCCNC(c2n[nH]c(C)c2F)=O)cn2c(n1)C(C)CCC2 9729,C(=O)(C(C)(C)C(C)C)NCCC1CC(NC(c2c(CCC)n(C)nn2)=O)C1 9730,c1(C(N2CCC(COC)(CNC(=O)C(F)C(F)(F)F)C2)=O)c(C)cc(C)nc1C 9731,CC(C)(C)CC(O)CC(=O)NC1CCN(C(=O)Cc2n[nH]c(=N)s2)CC(O)C1 9732,C1(OCC(=O)N(CCCNC(C(CCSC)O)=O)CCO)CCC(F)(F)CC1 9733,Cc1cc2c(N(C(c3cnc(Br)c(F)c3)=O)C(C3CCCNC3)C)ncnc2[nH]1 9734,CC1(C)CN(C(=O)C(F)F)CC1C(N1CCCC1c1ccon1)=O 9735,c1(C(=O)C(C2CC3C=CC2O3)=O)cnn(C)c1C.C=CCC(CC)O 9736,N1(C(CC(C)(F)F)=O)CCC(NC(=O)CCn2cc(Br)ccc2=O)C(F)C1 9737,CC(CCC(C)(C)C)C(=O)N1CCOCC1CCNC(=O)C(N1CCCCC1)C 9738,N1(CC)CCC(C(=O)N2CC(O)CO2)C1(C)C.N1C(=S)NCC1=O 9739,N1(C(Cc2c(C)ncs2)=O)C2CCC1CN(C(=O)C(C(C)O)OC(=O)N(C)C)C2 9740,C1(C)(C(=O)NCCc2ccnc(C)n2)CCCN(Cc2c(C)noc2C)C1 9741,Cc1ccc(I)c(COC(=O)Cc2csnn2)c1 9742,c1(C(N2CCCC(N(C(c3c(C)coc3)=O)CCF)C2)=O)cc(Cl)c(N)cc1F 9743,N1(C(c2nc(CC)sc2)=O)CC2CCC1CN2C(=O)CC1CCCC(C)C1 9744,n1(CC(=O)N(C(C)C(=O)NCCC2CCOC2)CC)cc(CC)cn1 9745,N1(C(c2ccc(CC)o2)=O)CCC(O)(C(C)NC(c2cc(C(C)(F)F)n[nH]2)=O)C1 9746,c1(CC(=O)NCC2CCC(NC(C3C(C=C)C3)=O)CC2)ccnc(O)c1Br 9747,N1(C(c2coc(C3CC3)n2)=O)CCC(C(N2CCC(CO)C2)=O)C12CC2 9748,C(C(C)C)(C(O)C(=O)NCCCCCC(N1CC(O)(c2cc[nH]n2)C1)=O)OC 9749,c1(CNC(c2cc(CO)[nH]n2)=O)nc2c(s1)CN(C(C1CCCCC1F)=O)CC2 9750,Cc1cnc(S(C)(=O)=O)nc1N(C(=O)CC1(O)CCC1)CC1(F)CCNCC1 9751,S(=O)(=O)(c1ccc(Cl)c(C(=O)NC(C)CNC(c2ccc[nH]2)=O)c1)NCCOC 9752,N1(C(C(C)(C)F)=O)CCC2CN(C(C3CC4CCC(C3)C4O)=O)CC12 9753,c1(C(N2C(C)CC(NC(=O)C=Cc3ccsc3)C2)=O)nccc2ncncc12 9754,N1(C(C2(C)CCN(C(c3c(CC)ncs3)=O)C2)=O)Cc2nn3nccnc3c2C1 9755,C1(CNC(C2(C(N(C)C)=O)CC2)=O)CN(C(C2CCC(C)(C)O2)=O)CCN1C 9756,Cc1nc(-c2csc(-c3ccc(C)o3)n2)n(CCS(N)(=O)=O)n1 9757,C#CCCCCC(=O)N(C)CC1CCN(C(c2ccncc2)=O)C1 9758,C#Cc1cccc(C(=O)NCC(C(C)(C)C)NC(c2cn(C)cn2)=O)c1C 9759,C(=O)(CCCC(C)(C)C#N)N1CC(C2N(C(C(C)NC(CC)=O)=O)CCC2)(O)C1 9760,C1(NC(=O)C=CC(F)(F)F)CCCCC12CCN(C(c1cscc1C(F)F)=O)C2 9761,C1(OC)(CNC(c2cnc(O)cc2C)=O)CCN(C(=O)Cc2ccsc2Cl)CC1 9762,C(C)(C)(CCCCNC(C1CCOC1)=O)NC(COCC=C)=O 9763,C(=O)(C(CC1CC1)NC(c1ccc(C(C)C)o1)=O)NCCCSC 9764,c1(CS(N2CCN(CC3CCCNC3)CC2)(=O)=O)csc2nccn12 9765,C1(NC(C2CCN2C(C2CC2(Cl)Cl)=O)=O)CC(Cl)(Cl)C1 9766,n1(CC(N2CC(CC3CC(F)(F)C3)C2)=O)cc(Br)c(=O)c(I)c1 9767,N1(CC(N2CC(C(C(=O)N(C)C3CC3)OC)C2)=O)CCCC1=O.C(C)=O 9768,C1(CC(CNC(=O)CC2COC(=O)C2)NC(C=CC(CC)C)=O)CCOCC1 9769,c1(C(=O)NCC(CC)NC(=O)C2=CCCS2)ccc(=N)[nH]c1 9770,C1(NC(C(CC)n2ccnc2)=O)CC2CC1CN(C(c1cc(Cl)sc1Cl)=O)C2 9771,c1(SC)ccc(Cl)c(C(N2CC(NC(=O)CCc3cccs3)CCC2C)=O)c1 9772,c1(C(N2CCOCC(NC(C3C(C)CC(=O)N3)=O)C2)=O)cc2n(n1)CCCN2 9773,CC1CN(C(C2(C(N)=O)CCC2)=O)CC1CC(=O)NCCCCO 9774,C1(CCOC)COCCC1Nc1cncc(CO)c1 9775,N1(C(c2cn(CC)nc2C)=O)CCCC(C(=O)NC2CN(C)CC23CC3)(CC)C1 9776,C1(NC(C(=C)CN(C)C)=O)(CN(C)C)CCCCC1C 9777,C12(CO)CCCN(C1)C(=O)C1C(C)(C1)C(=O)N2.c1(C(=O)OCC)ccc(F)cc1 9778,C1(C(N(CC(N2CC(c3ccon3)C2)=O)CCOC)=O)CC2CCC(C1)O2 9779,C1(NC(C2CCC(=O)O2)=O)CCCCCC1NC(c1ccn(CC(F)F)n1)=O 9780,C(=O)(C(CCC1CCCO1)N(c1nc(Cl)cs1)C)NCCCSC 9781,c1(CC(C(=O)NC(c2ccccc2)Cn2ccnc2)O)ccccc1Br 9782,c1(C(=O)NC(C2(O)CN(C(=O)COC3CCOC3)C2)C)cnc(-c2ccsc2)s1 9783,c1(C(=O)NC2CC(NC(=O)CC3CC3)C23CCC3)c(C2CC2)nc2sccn12 9784,C(=O)(NNc1cc(F)cc(Br)c1)c1n(CCC)cnc1 9785,C1(CNC(=O)C(=O)NCC2CC2)(CNC(C2CC3C=CC2C3)=O)CC12CCC2 9786,C(C(C(C)C)NC(c1cc(CNC(=O)Cc2coc(C)n2)[nH]n1)=O)OC 9787,CC1=NNC(=O)C1CC(=O)NCC12CC(NC(c3cc(C4CCC4)on3)=O)(C1)C2 9788,c1(CN2CCC(N(C)C(c3ccoc3)=O)CC2)cccc(Cl)c1C#N 9789,c1(OC)ccc2nc(C(=O)NC3(C)CCN(C(=O)Cc4csnn4)CC3)cn2n1 9790,Cc1sc(C)c(C(=O)NC2CN(C(C3CC(=O)N(C4CC4)C3)=O)CC2C)c1C#N 9791,C=CC(C)(CC)C(=O)NC1C2CN(C(=O)CCOc3ccccc3C)CC12 9792,C1(NC(c2cccs2)=O)CCOCC1C(=O)N(C)C1CC1.c1(C2CC2)ccncc1 9793,C1(CNC(c2n(C=C)ncc2)=O)CN(C(C2(C)CC(F)C2)=O)CCN1C 9794,Cc1cc(C)c(C(=O)NCC2(O)CCN(C(C3CCCN(C)C3)=O)C2)c(=O)o1 9795,N1(C(=O)OC(C)(C)C)CCCOC(CCOC(C2CC(O)C(F)C2)=O)C1 9796,C1(C#N)(C(N2CCC(N(C(=O)Cn3ccnn3)CCC)CC2)=O)CCCOC1 9797,O=C(C1CCc2c[nH]nc21)NC1CN(C(c2cnco2)=O)C2(CCCC2)C1 9798,C(c1ccsc1)=CC(=O)NC1(C(=O)NC2C=CCC2)C(C)C1 9799,CC(C)(C(=O)NC1CCCC1NC(=O)CC1COCC1O)NS(C)(=O)=O 9800,Cc1nccn2ncc(C(=O)NC3(CNC(C45CCCN4CC(O)C5)=O)CC3)c12 9801,N1(C(=O)NC(C)C)CCCC(C(=O)NC2CC(NC(c3cc(C#N)cs3)=O)C2)C1 9802,C12(COC)CC(NC(=O)C=Cc3ccc(C)nc3)(CN1C(c1cnc(C)[nH]1)=O)C2 9803,c1(C(=O)NC(C(CO)NC(C(COCC)C)=O)C)cccc2nc(O)n(C)c12 9804,c1(OC)cn(C)c(C(N2CCC(C(F)CNC(C3CC3C)=O)CC2)=O)cc1=O 9805,c1(OC)cc(COc2c(Cl)nc(Cl)n2C)ccc1C 9806,c1(CNC(=O)COc2ccsn2)ccccc1-n1cncn1 9807,CC1CN(C(=O)CC2CCCN2C(C2CC(=O)OC2(C)C)=O)C(C)C1C 9808,C1(CNC(CN(C)CC2CCCC2)=O)CCN(C(C2CCSC2)=O)CC1(F)F 9809,N1(C(CN(C)C)=O)CCC2CC2(C(=O)N(C)C2CC2)CC1 9810,c1(CC(=O)NC2CCCCN(C(C=COCC)=O)C2)nc2ccccc2s1 9811,c1(C(=O)NC(C(=O)NC(CNC(=O)OC)C)C)ccc(C)cc1 9812,NC(CCC1CC1)C(=O)c1cccc(-c2ccon2)c1 9813,N1(C(COCCCOC)=O)CCCN(C(=O)CSCc2cccs2)C(C)C1 9814,n1(CC)c(CCNC(C2CNCCC2(F)F)=O)nc2ccccc12 9815,C1(CNC(C(C)OCC#C)=O)CCC(CNC(=O)C(CC2CCC2)OC)CC1 9816,N(C(=NCCCCl)NCC(c1nc2c(s1)CCC2)SC)CC1CCC(OC)CC1 9817,C(=O)(C1=NOC(C)C1)NCC(Cc1ccccc1)NC(C1OCCN(CC)C1)=O 9818,C1(C(=O)NCC(C)Cn2cccn2)CN(C(C2(O)CC(CF)C2)=O)CC1C 9819,c1(CNc2c(C)nc(N3CCOCC3)cc2)cnn2c1CNCC2 9820,CC1=C(C(=O)NC2(C)CN(C(=O)CC3=CCOCC3)C2)COCC1 9821,c1(N2CCC(CC)C2)nnc(C(O)CC)n1Cc1nc(C2CC2)cs1 9822,CC1CC(CNC(c2cncn2C)=O)CCN1C(=O)Cc1cc(Br)cs1 9823,C1(O)(CC(N2C(CCCC)CCC2)=O)CCN(C(c2ccc(F)nc2C)=O)CC1 9824,c1(OC)ccc(C(CNC(=O)CC2CC23CC3)NC(=O)C(C)=C2CCCC2)cc1 9825,c1(NCCC2CCC(C)O2)ccc(S(=O)(=O)NCc2c(F)cccc2F)c(Cl)c1 9826,C1(C(=O)NCC(C(C)C)NC(C2C(=C)C2)=O)CCN(C2CCSC2)CC1 9827,C=C(Cl)CC(C(=O)NCC1(CC2CC2)CC1)NC(C1C=CC1C(=O)OC)=O 9828,N1(C(COCC=C)=O)CCC(=C)CC1C(=O)NCC(=O)N(C)OC 9829,N1(C(C2CN(C(C)=O)C2)=O)CC2CCCC(NC(C3(C)CCC(C)C3)=O)C2C1 9830,N1(C(C(c2ccccc2)C)=O)CCCC(NC(=O)C(F)(F)C2(O)CCC2)CC1 9831,c1(C(N(C2CCCN(C(c3ccnc(C)c3)=O)C2)CC)=O)ccc(C)c(Cl)c1 9832,C(=O)(C(C)C(C)NC(c1oc(CNC(=O)CC(C)(C)C)nc1C)=O)OC 9833,C(=O)(C#CC1CCCOC1)NC1(C)CN(C(c2c(C)ncn2C)=O)C1 9834,C1(C(C)(C)C)(CNC(c2c(C)coc2)=O)CCN(C(C2(F)CCCOC2)=O)C1 9835,c1(C(=O)NCCCCNC(c2coc(O)n2)=O)ccc2occc2c1 9836,N1(C(COCC=C)=O)CCN(C(=O)COCC(C)(C)C)CC1CCOC 9837,c1(C(=O)NC23CC(NC(CCc4cc(C)[nH]n4)=O)(C2)C3)ccc2c(n1)CCCC2 9838,CC1CC(NC(c2cnc(Cl)[nH]2)=O)CN1C(=O)CCNC(c1ccco1)=O 9839,C1(NC(C2C(CC)C2)=O)CCC2(CC1)CC2NC(c1cc(S(C)(=O)=O)cs1)=O 9840,C1(C(=O)NC(CC)(CC)CCNC(c2cccs2)=O)CCc2nn(C)cc2C1 9841,C1(CC(=O)NCC2(OC)CCOC2)CN(C(c2sncc2C)=O)CCC1C 9842,c1(NC(C(C)OCC)=O)ccc(OCC2(NC(=O)CN3CC(C)C3)CCC2)cc1 9843,CCCCS(=O)(=O)NC(C)C(=O)NCC12CC1CN(C(C1CCN1CC)=O)C2 9844,C12(OC)CCC(C(N3CCC(C)(CNC(C4C(C)(C)C4(F)F)=O)C3)=O)(CC1)C2 9845,C1(C(=O)NC(CC)(C)CC)CN(C(=O)C(C)Nc2ccccn2)CCC1O 9846,c1(C(=O)NC2(CO)CCN(C(CC(C)SC)=O)C2)ccc(Cl)c(F)c1N 9847,c1(NC(CCC)SC)ncc(C)cc1S(=O)(=O)NCC1(c2cccc(Br)c2)CC1 9848,C(=O)(C(CCC(C)C)N(C)C)N1CCC(C)(N(C)Cc2cc(SCC)on2)C1 9849,C1(CNC(CCc2ccc(C)nc2)=O)CN(C(=O)Cc2nc[nH]n2)CC(C)(C)O1 9850,c1(CN2CCC(NC(c3ccc(C(N)=O)cc3)=O)C2)ccc(O)c(F)c1 9851,C1(C(=O)NCCCc2ncc[nH]2)(CC)CCN(C(c2cc(Cl)no2)=O)C1 9852,C1(NC(C(C)O)=O)CN(C(c2cccc3ccccc23)=O)C2(CCCC2)C1 9853,C#CC1CC2(C1)NC(=O)N(c1ccc(OCC)c(Cl)c1)C2=O 9854,N1(C(C=CC)=O)CCN(C)C(CNC(=O)C=Cc2ccc(SC)cc2)C1 9855,C(C)(CCC(=O)NC1CN(C(c2ccncc2C(F)(F)F)=O)C1)OC 9856,Cc1nc(N)cnc1C(N1CCN(C(C2(N(C)C)CC2)=O)CC1C)=O 9857,C1(C(N(C)CC2N(C(CCC(C)C#N)=O)CCC2)=O)CCS(=O)(=O)C12CCC2 9858,CCN=C(NCC1(c2ccsc2)CC1)NCC12CC(C1)C(C)O2 9859,C12(NC(c3c[nH]c(C(F)F)c3)=O)CC(C1)N(C(c1cnc[nH]1)=O)C2 9860,C1(Nc2cc(OC)ncn2)CN(C(C23CC(C2)C3)=O)CC12CC2 9861,c1(OCC(=O)NCC(C2(O)CN(C(=O)C(O)C3CC3)C2)(C)C)ccccc1C#N 9862,c1(C(=O)NCCOCCCNc2ncccn2)ccc2nc(O)[nH]c2c1 9863,CC(CC(F)(F)F)C(=O)N(CC(C)(C)CNC(c1cnc2sccn12)=O)C 9864,N1(C(C(C)O)=O)CC2CC(NC(c3c[nH]nc3C(F)(F)F)=O)CC1C2 9865,CCCCC(C)C(=O)N1CC(C(N)=O)(CNC(C2CCC=CO2)=O)C1 9866,c1(C(N2CCN(C(C3(CC)CC3)=O)CC2CO)=O)cccc2c1CCS2(=O)=O 9867,CC1CC(CC(=O)NCC2C3CN(C(C4CS(=O)(=O)C4)=O)CC23)CCC1C 9868,Cc1ccc(CC(N2CCC(F)(CNC(C3(C)CC3(F)F)=O)C2)=O)cc1Br 9869,C1(NC(C2CC23CC(O)C3)=O)CCN(C(C2(C(F)F)CC2)=O)CCC1CO 9870,c1(C(=O)OC(C2CCN(C(=O)CC3C4CN(CC)CC34)C2)=O)cc(F)cc(Cl)c1 9871,N1(C(C2N(C)CC(O)C2)=O)CCC2(CCN(C(=O)C=Cc3nccs3)C2)C1 9872,N1(C(COCc2c(C)cccc2)=O)CCN(C(=O)Cc2ncoc2C)CC(O)C1 9873,N1(C(C(C2CCOC2)NC(C2C(CC(C)C)C2)=O)=O)CCC2(C=CCO2)CC1 9874,Cc1cc(C)c(C(=O)NCCOC2CN(C(C3(CCO)CC3)=O)C2)c(S)n1 9875,C(CN=C(NC1CCC1)N(C)CC1CCCN1C)c1ccc(OC)cc1 9876,n1(CC)nc(C)c(CC(=O)N(C)CCNC(=O)CN(c2ccc(Cl)cc2)C)c1C 9877,N1(C(C=C(CCC)C)=O)CCC(C)(C)C(CNC(=O)CS(=O)CC)C1 9878,c1(COCC(=O)NC(CN(C(C=CC=CC)=O)CC)C)ccccc1.OC.CC 9879,CC1C(C(=O)NC(C(=O)NCC(C)(C)CN=[N+]=[N-])C2CCOC2)=NOC1C 9880,Cc1cc(C(N2CCCC(C3CCCCN3C(=O)C#CC(C)C)C2)=O)[nH]c1C 9881,N1(C(C2CC=CC(NC(CCOCCOC)=O)C2)=O)CC2CC(C1)N(C)C2 9882,C(=O)(CC1OCc2ccccc21)NCC1CC(NC(c2c(CC)csc2)=O)C1 9883,C12(C(N3CCC(F)(C(=O)NCC4N(C)CCCC4)C3)=O)CCCC1C2(F)F 9884,C1(NC(=O)CCc2ccncn2)C2CC3CN(C(=O)C4=COCCC4)C1C3C2 9885,Cc1ccccc1C(CC(=O)O)NC(=O)C(C1CCCC(=O)C1)(F)F 9886,c1(NC)snc(C)c1C(N1CC(CNC(=O)C=CSC)C1)=O 9887,C1(c2cccc(OC)c2)CN(C(=O)C=C2CCC(C)C2)CCN1C(=O)C1CC1 9888,C1(NC(C2(c3nn[nH]n3)CN(Cc3ccccc3)C2)=O)COC2COCC12 9889,C(=O)(CC(C)(C)c1ccccc1)N(CCCNC(=O)C(C1CCC1)C1CCC1)C 9890,c1(OC)ccc(OCC(N2CCC(CN(C(=O)Cc3cn(C)nn3)C)C2)=O)cc1 9891,N1(C(CC(C(F)F)NC(c2cc(C(N)=O)[nH]n2)=O)=O)C(CO)CC2CCCC12 9892,Cc1ccncc1C(C)(C)C(=O)NC1CCC(NC(C2CCCOC2)=O)CC1 9893,c1(C(=O)NC2C(C(N(CC)Cc3cccc(Cl)c3)=O)C2)ccc(Cl)c([N+](=O)[O-])c1 9894,N1(C(CC(C)C)=O)CCCC2C1CCCN2C(c1ccn(C2CCOCC2)n1)=O 9895,c1(N2CCC(C3(OC(CC(CCC)C)=O)CC3)C2)cc(OC)c([N+](=O)[O-])cc1Cl 9896,c1(C(C(=O)NCCC(CCNC(C2(OC)CCCC2)=O)C)=O)cc(F)cc(Cl)c1 9897,C1(CNC(C(c2scc(C)n2)(F)F)=O)CN(C(C2CCCS2)=O)CC(C)(C)O1 9898,C12(F)COCCN(C1)CNC(=O)N2.c1(SCC=C(C)C)ccc(F)cc1 9899,c1(OC)ccc(C(CNCc2cc(C(F)(F)F)n(C)n2)N(C)C)cc1 9900,N1(C(c2cccc3ccn(C)c32)=O)CCOC2(CCN(C(c3cnns3)=O)C2)C1 9901,N1(C(C)=O)CCOC(C(N2CCC(NC(=O)Cc3ncc(C)o3)C2C)=O)C1 9902,CC1(C)CCCCC1(C)NC(=O)CNC(C1CCC(C#N)CC1)=O 9903,CCC(CNC(=O)CCCCCn1cc(CCSC)nn1)CC(F)F 9904,C12(n3c(CN4C(C)C(c5ccccc5)CC4)nnn3)CC1COC21CCC1 9905,C=CC1(C(=O)Nc2ccc(OC)cc2)CCN(C(C2CC3(C2)CC(C)C3)=O)C1 9906,c1(CC)ccc(C(N2CC(OC)C(NC(=O)CC3CCC(C)(C)C3)C2)=O)c(Cl)c1 9907,N1(C(C(C)CO)=O)CCC2(CCCCC2NC(c2cc(F)cc(Cl)c2)=O)CC1 9908,Cc1nn[nH]c1C(C(=O)NCCCOCC1CC1)N(C1C2CCCC12)C 9909,N1(C(C(CC)OCC)=O)CC2CCC(C1)C(NC(c1c(C)nn(C)c1Cl)=O)C2 9910,C1(CO)CCC(CNC(c2nnnn2CCCF)CC2CCOC2)CC1 9911,CC1CCCCC1(CNC(=O)CCC(=O)c1ccccn1)NC(c1cnsc1)=O 9912,c1(C(N2C(CCNC(C(C(C)O)N(C)C)=O)CCC2)=O)ccc(Cl)c(N)c1 9913,c1(C(N2CCC(CNC(C3C(F)(F)C34CCC4)=O)C2)=O)cc(C2CC2)ccc1F 9914,c1(C(=O)NCC(O)Cc2nn[nH]n2)ccc2c(c1)CCCC2 9915,c1(CC)cccc(C(N2CC(O)(C(F)C(=O)N(C3CC(O)C3(C)C)C)C2)=O)c1 9916,NC1CCCC2CN(CC(=O)NC3CCN(c4nncs4)CC3)CC12 9917,C1(NC(C2CC(C(C)C)C2)=O)CCCN(C(c2sccc2CC#N)=O)C1C 9918,c1(OC)csc(C(N2CCC(F)(CNC(C3(C)CCCS3)=O)C2)=O)c1OC 9919,c1(C(=O)NCC2(C(C)NC(c3cc(C(C)=O)oc3)=O)CC2)cc(C)ccc1C 9920,C(=O)(C(CC(C)C)CC(C)C)NC1C(CNC(CCc2ccc(C)o2)=O)CC1 9921,n1(C(C)C)c(O)nc(N(C)CCOCCNC(C2CCN(C)C2=O)=O)cc1=O 9922,c1(NC(c2c(C)nc(CC)o2)=O)ccc(NC(c2cncc(C)n2)=O)c(C)c1 9923,CCC(CC(C)C)C(=O)NCC1CCC(NC(=O)Cn2nnnc2C(C)C)CC1 9924,CC(CCN(C)C)C(=O)NC1CCCC1C(N1CCC1(C)CCO)=O 9925,c1(C(=O)OCc2c(C)ncn2C)cc(S(=O)(=O)N(C)C)ccc1F 9926,N1(C(c2cc(C)c(Br)o2)=O)CC2(COC(CNC(c3ccncn3)=O)C2)C1 9927,N1(C(C2(Br)C3COCC23)=O)CC2(C1)CN(C(C1(C3CCC3)CC1)=O)C2 9928,N1(Cc2ccc(OC)c(-c3ccncc3F)c2)CCCC2(C1)OC(=O)NC2=O 9929,C1(C(N2CCCC3COCC23)=O)CCCCC1C1CCNCC1 9930,C#CCC(C)(CC)C(=O)N1CCC(O)(CNC(c2ccoc2Br)=O)C1 9931,Cc1ncn(C)c(=O)c1C(=O)NCC1(NC(=O)C(N2CCCC2)C2CC2)CCC1 9932,CN=c1[nH]cc(C(=O)NC2C=CC(C(=O)NCC(CO)OC)C2)o1 9933,C1(NC(=O)Cc2cn[nH]c2)CC12CCN(C(c1ccc(O)cc1Cl)=O)CC2 9934,N1(CC)CCN(C(=O)C(C)CNC(=O)C(F)C(C)(F)F)CC1C 9935,CC1=C(C(=O)NC2COCCC2NC(=O)C=Cc2cnc[nH]2)CCC1 9936,C(=O)(CCCCCC(=O)N1CC(NC(=O)C(F)=C2CCC2)C(C2CC2)C1)OCC 9937,c1(C(=O)NCCN(C(=O)CCNC(=O)NC)CCC)c(C)ccc(Cl)c1F 9938,N1(C(c2cc(C)nn2CC(F)F)=O)CCC(F)C(NC(C2CCCC2)=O)C1 9939,Cc1c(C(N2CC(CNC(=O)C(C)CCO)CC2C)=O)[nH]c2c1C(=O)CCC2 9940,N1(C(C(C)C)=O)CCC2CCN(C(c3ccc(NC(C4CCC4)=O)cc3)=O)C2C1 9941,C1(CC(=O)NC(C)CSC(F)F)CC(F)CN1C(=O)CCC1OCCO1 9942,N1(C(C=C(C)Cl)=O)CCN(C(c2cccn(C)c2=O)=O)C(C(C)(C)C)C1 9943,CCCCC(C(=O)N1CCC(CNC(=O)CC2CN(C(C)=O)C2)(OC)C1)N(C)C 9944,C1(C(N(C(CNC(CN(C)C2CC2)=O)C2CC2)C)=O)CC2CC1CO2 9945,c1(C(N2C(C)(CNC(=O)CC3(O)CCCOC3)CCC2)=O)cccc(N=[N+]=[N-])c1 9946,Cc1[nH]nc(C(F)(F)CO)c1C(=O)NCCOCCNC(=O)C=Cc1ccoc1 9947,C(=O)(CC(C)C(F)F)NC(CC)(C)CCNC(=O)Cc1n[nH]c(C)n1 9948,N1(C(c2cc(C)c(F)cc2)=O)CC2CC1CCN2C(=O)Cn1cncc1C 9949,S(=O)(=O)(c1ccc(C=CC(=O)NC(CCc2nn[nH]n2)C(=O)O)cc1)NCC 9950,C1(NC(C2CC3CCC(C2)C3)=O)CC2CN(C(c3cscc3C(F)F)=O)CC2C1 9951,CC1CCC(C(N2CC(CO)CC2CO)=O)CN1C(=O)Cc1cc[nH]c1 9952,N1(C(c2ncc(CC)cn2)=O)CCC(C(N2CCCCC(C)(F)C2)=O)CC1(C)C 9953,N1(C(=O)C=C(Cl)Cl)CCC(C2CCN(C(C3CC3[N+](=O)[O-])=O)CC2)C1 9954,C1(C(=O)NCC(C)OCCO)CC2(CC(NC(=O)CC3(O)CCOC3)C2)C1 9955,c1(C(=O)NCC2CC(F)(CNC(CC3CC(=O)NC3)=O)C2)csc2nnsc12 9956,C1(NC(C2C(=C)CC2)=O)CCC2CC1CN2C(c1c[nH]ccc1=O)=O 9957,C1(C(=O)NCc2c(CC)n[nH]c2)CCC(C)(C)N(C(C23CCC(C2)C3)=O)C1 9958,C1(CC)CN(C(=O)Cc2cccc(C)c2Cl)CCC1NC(c1ncc(C)cn1)=O 9959,N12C3CCC1CN(CC3)C(=O)Nc1c(cccc1)N(CC)C(=O)C2.C(C)(C)OC 9960,C12(CNC(=O)CC3CC3)CCCC1N(C(=O)CN1CCCCC1)CCC2 9961,C=C1Cn2c(C(=O)NCC3(C)CCN(C(=O)C(=Cc4c[nH]cn4)F)C3)nnc2S1 9962,CCC(C)CC(C(=O)Nc1ccc(OC)cc1C)NC(=O)CC1(O)CCOCC1 9963,C(C)(C(C)(C)CO)NC(C1C(CNC(C2(CC)CCCC2)=O)CCC1)=O 9964,Cc1nn(CC(N2CCC(NC(=O)COCC3CCOC3)C2C)=O)cc1[N+](=O)[O-] 9965,C1(NC(c2cnsc2)=O)CC2CCC1N2C(=O)COc1ccc(Cl)nc1 9966,c1(C(=O)NC(c2cncnc2)C)cccc(CNC(C2CCC3(CC3)C2)=O)n1 9967,C(=O)(C1=CCC(C)(C)CC1)NC1CC(CNC(c2c(C)[nH]nc2C(F)F)=O)C1 9968,N1(C(CCCOCCC)=O)CC(C)CCC1CNC(=O)CNS(=O)(=O)CC 9969,N1(C(C(C)C#N)=O)CC(F)(F)CC1CNC(c1ccc(C(F)(F)C(F)F)cn1)=O 9970,C(CCCC(CO)NC(c1cnn(C)c1)=O)NC(CCN(CC(F)(F)F)CC)=O 9971,N1(C(c2n(CC=C)ccn2)C(=O)NCC=C)CC2CCC1C(C(=O)OC)C2 9972,C=CCN=C(NCC(N1CCOCC1)c1nccn1C)NCCSCCOC 9973,Cc1cc(C)n(C(C)CC(=O)NCCC(C)NC(=O)CSCc2ccccc2)n1 9974,C(=O)(CC(=O)N(CCNC(C1(C2CCCCO2)CC1)=O)C1CC1)NCC#C 9975,N1(C(c2c(CC)oc(C)c2)=O)CCCC(NC(=O)C=C2CCCCC2)C1CC 9976,C(=O)(C1=CC2(CCOC2)C1)N(CC(C(=O)CCCn1cncn1)=O)C1CC1 9977,c1(C(N2CC(NC(CCC=CC)=O)C(O)C2)=O)ccc2sncc2c1 9978,CCC(CC(=O)N(C1CC1)CC1CCCN1C(=O)CCc1nc(C)cs1)SC 9979,C(=O)(C1=CC2CCCCCC12)NCC1(CN(C(c2ccc(C)o2)=O)C)CC1 9980,N1(C(CCCN(C)C)=O)CC(C2CCCN(C(=O)C=CS(C)=O)C2)C1 9981,Cc1cc(C(=O)NC(C2CCCN2C(c2ncn(C(C)C)n2)=O)(C)C)n[nH]1 9982,N1(C(CN(C2CCCCC2)C)=O)CC(F)(F)CC1(C)CNC(c1csc(Cl)n1)=O 9983,c1(CNC(c2cc(C)ncc2)c2nnnn2-c2ccccc2Cl)cc(Cl)cc(Br)c1 9984,c1(C(N2CC(CNC(C3(CF)CCC3)=O)C3(CC3)C2)=O)cnc2n1CCCC2 9985,C1(CNC(C(CC)(C)F)=O)CN(C(c2cccc(C)c2)=O)CC1(C)C 9986,CCC(C)(C)C(O)C(=O)N1CCC(NC(=O)Cc2scnc2C)C1 9987,N1(C(CCN(CC)CC)=O)CCCC12CCN(C(C1CCCCC1C)=O)CC2 9988,c1(OC)ccc(C=CC(=O)NCC2CN(C(C3OCCC3C(C)C)=O)C2)nc1 9989,C(=O)(CC1CCC(=O)c2ccccc21)NCCNC(C(C)C1CCC1)=O 9990,c1(C(N2CC3(CC(CNC(C4(CC)CC4)=O)OC3)C2)=O)cnc2c(c1)CCCO2 9991,c1(CC(=O)NC(CCN(C(C2N(C(C)=O)CCC2)=O)C)C)cccc(Br)c1 9992,CC(C(=O)N(C1CN(C(c2nn(CC(F)(F)F)cc2Cl)=O)CC1O)C)C(C)(F)F 9993,CCCC(CCC)C(=O)NC1CCC(C)N(CC2(c3cccc(C#N)c3)CC2)C1 9994,C1(C(=O)OC)C(NC(=O)NC2(c3nnc(C)o3)CCC2)C2CC1C(O)C2O 9995,N1(C(C2OCCC(C)(C)C2)=O)CCC2(C=C(C(=O)N3CCC3C3CCOCC3)C2)C1 9996,C(CCCC(=O)N1CCC1CNC(C1(F)CCCOC1)=O)N(C)C 9997,c1(CC)c(N2CC(NC(C3CC(=O)N(CC(C)C)C3)=O)CCC2C)ncnc1Cl 9998,c1(NC(C2(C)N(c3cc(NC(C)=O)ncn3)CCC2)=O)ccnn2cccc12 9999,N1(C(C2(COC)COC2)=O)CC(C(N2CCCCCC2)=O)C(C2CC2)C1 10000,c1(N(C)Cc2ccncc2F)cccc(S(=O)(=O)NC2CSC2)n1 10001,C1(CC(=O)NC2C(NC(=O)CC3(O)CCOCC3)CCCC2)CC(F)(F)C1(F)F 10002,c1(CCNC(=O)C(O)C2CCCO2)ccccc1Sc1nc[nH]n1 10003,C(=O)(CS(=O)(=O)C(C)(C)C)NC1C(C)CN(C(c2scnc2C(C)(C)C)=O)CC1 10004,c1(C(N2CCOCC(NC(c3cccc(SC)c3)=O)C2)=O)ccc2c(c1)CCC2 10005,N1(C(c2cc3nc(C)oc3cc2)=O)CCc2ccccc2C1CNC(=O)C(C)O 10006,C12(C(=O)NC(CC(=O)NCCC3CCCC(C)C3)C)CCC(C1)C2(C)C 10007,N1(C(C2(CC)COC2)=O)CCCCC1C1(NC(=O)CN2CC(C)(C)C2)CC1 10008,c1(C(=O)NC2CC(NC(c3ccccc3O)=O)C2)cc2ccc(Br)cn2c1 10009,N1(C(CCOCCCSC)=O)CCCC1C1(CNC(=O)Cn2cccn2)CC1 10010,C1(C)(C(=O)NCC)CCCN1c1nccc(OCC)n1 10011,Cc1cnccc1C(C)C(=O)N1CC(CNC(=O)CC2CCOC(C(C)C)C2)C1 10012,c1(C(=O)NC(C)C)ccc(CNC(=O)NC23CC(C2)NC3=O)cc1 10013,C(CCCC(C)NC(=O)C=CCC1CCCCC1)NC(C(C)Cc1cnco1)=O 10014,c1(C(C(=O)NCCCN(C(=O)C2=COCC2)C(C)C)C)ccc(C(F)F)cc1 10015,C(=O)(C1=NOC(CNC(C2(CC(C)C)CC2)=O)C1)N(C)CC1CCN(CC)C1 10016,C(CC(=O)NC(C)C(C)(C)NC(c1cc2c(s1)CCC2)=O)(C(N)=O)NC(C)=O 10017,C(=O)(CC(C)(C)C(=O)NC1COCCC1NC(c1cc(CC)c(C)s1)=O)OCC 10018,c1(CCC(=O)NCCC(O)CNC(C2(CO)CCCC2)=O)ccc(Cl)cc1Cl 10019,N1(C(C=CCCC)=O)CCCN(Cc2cn(CCCC(=O)O)nn2)CC1 10020,N1(C(CCC2CCN(C(C3(OC)CCOC3)=O)CC2)=O)CC2C(C1)C2(F)F 10021,C1(CNC(c2cn(C3CC3)cn2)=O)C2CN(C(c3c[nH]cc3Br)=O)CC12 10022,C1(NC(CNC(c2nncc(OC)c2)=O)=O)C2C=CC(C2)C1CO 10023,c1(C(=O)NC2C(CNC(CC(C)c3ccncc3)=O)C2)nnc2n1CCCCC2 10024,n1(CC(=O)NCCOC2CCCCC2)cccnc1=O.C12CCC(C1)NC2=O 10025,CCC(CC1CCCC1)C(=O)NCCNC(=O)CNC(=O)Nc1ccc(Cl)cc1 10026,CS(=O)(=O)C(CNC(=O)C=CC1CCOCC1)CNC(C1(F)CCCCC1)=O 10027,n1(CC)nnc(C(=O)N(CC(C)(C)C(=O)NCCc2nnc(C)n2C)C)c1C 10028,C1(C(=O)NCc2c(C(=O)NCC(C3CCC3)OCC)n[nH]c2)CCCCC1C 10029,N1(C(c2c(C)ccs2)=O)CCOC(C(N2CCC(C(C)(C)O)CC2)=O)C1 10030,N1(C(C2C(C=C(C)C)C2(C)C)=O)CCN(C(c2c(C)ncnc2C)=O)CC1C 10031,C1(CC#C)(C(=O)N(CC(=O)NC2CC2NC(N)=O)C)CCCC1 10032,N1(C(CC2(C)CCOC2)=O)CCC2(CCCN2C(=O)CS(=O)C(F)(F)F)C1 10033,c1(COC)nc(CNC(=O)C(=O)NC(c2ccccc2)c2ccco2)cs1 10034,c1(CC)cccc(CC)c1CC(=O)N(C)CC1CCCN1C(C1CCOC1C)=O 10035,N1(C(c2c(CC)nco2)=O)CC2OCCN(C(=O)C(C)C(O)C(C)C)C2C1 10036,CC1(c2cn(C3(C(N)=O)CC3)nn2)CCN(C(=O)CC2CCCCC2O)CC1 10037,Cc1cc(NC(c2ocnc2C2CC2)=O)n(C2CCOC2)n1 10038,N1(C(C2(NC(C)=O)CC2)=O)CCCC(N(C(=O)C(C)C)CC(C)C)C1 10039,CC1(CNC(c2ccnc(S)c2)=O)CN(C(c2cccc(Cl)c2Cl)=O)CCO1 10040,C1(C)(CC)C=C(C(=O)NC2CC2NC(C2(C(=O)OC)CC2)=O)C1 10041,C1(C2(NC(c3c(OC)scc3)=O)CC2)CCCCN1C(=O)COC1CCCOC1 10042,c1(C(=O)NC(C)CCN(C)C(C2CC2F)=O)cc(Br)ccc1O 10043,C1(C(=O)NCCNC(=O)OCC)CC=CCN1C(c1ccsc1C)=O 10044,C(=O)(CCCCCCC(=O)N1CCC1C(=O)Nc1c(Cl)ccc2c1OCO2)OC 10045,c1(-c2cc(C(N(C(CCNC(CN3C(C)CC3)=O)C)C)=O)on2)cccc(F)c1 10046,C1(C)(CNC(C(C(C)C)OCC)=O)CCN(C(=O)C(C2CCCCC2)F)CC1 10047,O=C1CCC(C(=O)NC2CCCN(C(=O)C3=COCCO3)C2)c2ccccc2N1 10048,N1(C(=O)C(F)(F)C2CC2)CCC2(CC1)CCN(c1nc(O)c3c[nH]nc3n1)C2 10049,C(C#CC(=O)NC1CC(C(=O)OCC)C1)NC(C=CCCC)=O 10050,CC1(C)CN(C(=O)CC2(CO)CC2)CC1NC(C1(C)CCCS1(=O)=O)=O 10051,C1(NC(c2c(CC)onc2)=O)CCCN(CC(O)COc2ccc(Cl)cc2)CC1 10052,C(CO)(C(C)(C)C)NC(CC1CC(NC(c2c(OC)ccs2)=O)C1)=O 10053,C(C(C)C(=O)N(C)CCC1CN(C)C1)NC(CCOC(C)=O)=O 10054,CCCCC(C)CCC(=O)NCCCN(C(=O)C(c1ccccc1)F)C(C)C 10055,C1(CNC(COCC#C)=O)CCC2CN(C(c3ccncc3CC)=O)CCC2C1 10056,C1(=CC(=O)NCC2(C)CC(NC(=O)Cc3cnns3)C2)CCOc2ccccc21 10057,c1(CC)ccc(C(C)C(=O)NCC(O)CNC(=O)CCc2cncs2)cc1 10058,c1(CC(=O)NC(CNC(c2c(CC)n[nH]c2)=O)C2CC2)cc(C)ccc1Br 10059,c1(C(=O)NC2CN(C(c3cc[nH]n3)=O)C3CC23)ccc2c[nH]nc2c1 10060,N1(C(c2c(C)cc(CNC(CC3ON=C(CC)C3)=O)o2)=O)C2CCC1CC(F)C2 10061,C#CCCCC(C(=O)NCCSC)N1CCC(CCn2cccn2)C1.OC 10062,C(CCCCC(=O)N1CCC(N(C)C(c2ccnc(C3CCC3)c2)=O)C1)OCC 10063,c1(NC(C)=O)cccc2c1CCCN2C(C1OCCC1C(=O)O)=O 10064,C1(NC(C)=O)CCC12CN(C(C1CCC(C(N)=O)CC1)=O)C2 10065,Cc1nc2ccc(C(=O)Nc3cc(Cl)c(OC(F)F)c(Cl)c3)cc2n(C)c1=O 10066,C1(C)(OC)CCCN(C(C2(F)CCN(C(=O)CCCC(=O)OC)CC2)=O)CC1 10067,c1(-n2cc(CCCC)nn2)cccc(C(=O)NCC(=O)N(CCC)CCNC)c1 10068,C(=O)(C(C)(C)NC(=O)C(F)(F)F)NCC(C)NC(=O)C(C(C)C)n1ccnc1 10069,N1(C(c2ncccc2F)=O)CC(F)(F)CC1C(N1C2CCC1COC2)=O 10070,N1(C(c2nc(C(N)=O)sc2)=O)CC(CNC(C2CS(=O)C2)=O)N2CCC1C2 10071,CC1(C)CC(NC(c2ccc(C(C)(C)C)o2)=O)CC(O)C1 10072,c1(C(N(C)CC2CCC(CNC(C3CC4CCC34)=O)CC2)=O)ccc(F)c(Cl)c1 10073,c1(C(N2CC3C(NC(C4CCC(C)O4)=O)(C3)C2)=O)cc2c(Cl)cncc2s1 10074,CS(=O)c1ccc(CC(=O)NCC(O)CNC(c2coc(Cl)c2)=O)cc1 10075,C1(NC(CCC2CCCN(C(c3c(CC)occ3)=O)C2)=O)CNC(=O)C12CC2 10076,CCCC(O)CC(=O)N(CC(O)CN(C)C(c1nc(C)ncc1Br)=O)C 10077,C1(COC)(NC(=O)CC2CCCN2C)CCN(C(=O)C=CC(C)C)C1 10078,c1(C(=O)NC2CC3(C(=O)NC45CCC(CC4)C5)COC2C3)cn2ccccc2n1 10079,CC(CCCc1ccccc1)C(=O)N1CCCC1CCNC(C1COC(=O)N1)=O 10080,C(c1ccc(F)c(OC)c1)=CC(N1C2CC(NC(C(CCOC)C)=O)C2CC1)=O 10081,N1(C(C(C)NC(CC)=O)=O)CC2CC1C2NC(=O)C(C)=CC1CC1 10082,c1(CC(=O)N(CCCCN(C(C(C)=C2CC2)=O)C)C)nc2nc(C)cc(C)n2n1 10083,C#CCC(CC(=O)NC1CCCCCC1)NC(c1cccc(C)c1C)=O 10084,C(C(C)(C)C(=O)NCC1CCN1C(C1(CN)CCCC1)=O)SC.c1(C)cnn[nH]1 10085,c1(N(C)C)ccc(F)c(C(=O)NCCCCn2cc(-c3cccnc3F)nn2)c1 10086,N1(C(c2c(C)cc(SC)o2)=O)CCC(C)C(NC(=O)C=Cc2cn(C)cn2)C1C 10087,N1(C(c2c(C)oc(C)c2Br)=O)CCN(C(=O)C(C)N(C)C)CC(C)(F)C1 10088,N1(C(CNC=O)=O)CCCC(O)(c2cn(Cc3cnc(OC)c(F)c3)nn2)CC1 10089,c1(C(=O)NC2CC2)cccc(-n2cncn2)c1.C12(F)CN(C1)C(=O)C1CC(C1)C2 10090,C1(C(=O)NC(CC)CNC(C2(OC(C)C)CCCC2)=O)CCC(F)(F)C1 10091,c1(CN2C(C(N3CCC(C(F)(F)F)C3)=O)CC(O)C2)cc([N+](=O)[O-])cc(Br)c1O 10092,Cc1ccc2nnc(C(=O)N(C)CCNC(C3(C)CCOC(C)C3)=O)n2c1 10093,N1(C(CC2CN(C(c3ccc(CC)s3)=O)CC23CC3)=O)CCn2ncc(C)c2C1 10094,C1(C#N)(CC(=O)N(CC(C(=O)N(CCCOCC)C)C)C)CCOCC1 10095,C(=O)(C(CC(C)C)NC)N(CCN(C(=O)C(O)C1CC1)Cc1ccccc1)CC 10096,C1(F)(C(=O)NCCCN(CCCCNC(C=C(C)C)=O)C)CCCC1 10097,c1(-n2cc(C3(OC(C)C)CCC3)nn2)ccnc(Br)c1F.N12CCCC1C2=O 10098,N#CC1CN(C(c2cc(Cl)ccc2Cl)=O)CCN1C(c1cnnc(Cl)c1)=O 10099,CCCCC(O)CC(=O)NCC1CC1CNC(C1CCC(CC)O1)=O 10100,C1(CS(C)(=O)=O)C2CCC1CN(CC(=O)NCC1CCC(=O)N1)C2 10101,C(C(F)(F)C(=O)NCCOC1CCN(C(=O)CCc2ncc[nH]2)CC1)OC 10102,N1(C(CCC2C(C)(C)C2)=O)CCN(CCNC(C2CC(=C3CC3)C2)=O)CC1 10103,N1(C(C=COCC)=O)CCCC(O)(CNC(C2(CC)CCOCC2)=O)C1 10104,N1(C(Cn2c(C)ccn2)=O)CC2(C1)CN(C(=O)Cc1ccnc(F)c1)CC2CO 10105,c1(OC)ccc(-c2nc(C)c(C(C)NC3(Cc4ccccc4)CCCC3)s2)cc1 10106,c1(OC)cc(C)cnc1C(=O)NC1(C(=O)O)CC(OC)C1 10107,N#Cc1c(F)cc(C(=O)NC2CC(CNC(=O)C3=CSCCO3)C2)cc1F 10108,C12(CNC(C(C)=C(C)C)=O)CC(CO1)N(C(=O)C(c1ccccc1F)O)C2 10109,C(C(C)(C)CCCc1ccccc1)NC(N(C1CC1(C)C)C)=O 10110,Cc1ccc(CNC(C)Cc2ccnc(O)c2)cc1.C12(CC1)C(=O)N2 10111,N1(C(CC(CC)OC)=O)CCC2(CC(NC(c3csc(O)n3)=O)C2)C1 10112,C(=O)(C1=C(CCl)N(CC2CC2)C(=O)NC1c1ccc(-c2ccccc2)o1)OCC 10113,C(=O)(C#CC1CCOC1)NCC1C(C(=O)NC2C(C)(C)C2(C)C)CC1 10114,C(=O)(C1=CN(C)S(=O)(=O)N=C1C)NCC(CNC(C(C(CC)O)(C)C)=O)CO 10115,C(=O)(C(CO)NC(=O)C(c1cn(C)nn1)NC(c1cnn[nH]1)=O)N(C)C 10116,CCCC(C(=O)NCCCN(C)Cc1csc(C(C)C)n1)OC 10117,N1(C(CC(=C)Br)=O)CC2CCCC2(NC(=O)CCc2ccccc2Cl)C1 10118,Cc1cc(P(C)(C)=O)oc1C(=O)NC(C)CNC(c1cc(C2CC2)cs1)=O 10119,N1(C(C2C(C)(C(=O)OCC)C2)=O)CCC2(C1)CN(C(c1n[nH]c(C)n1)=O)C2 10120,N1(C(C=C(COC)C)=O)CC2ON=C(CNC(c3csnc3Br)=O)C2C1 10121,C1(NC(CCC#CC)=O)CC2(NC(c3scnc3COC)=O)COC1C2 10122,C1(C)(CCNC(C(C)O)=O)CCN(C(c2ccc(-c3cccnc3)cc2)=O)C1 10123,c1(C(=O)OC)cccc(C(N2CCC(NC(=O)CC3CC(SC)C3)C2C)=O)c1 10124,Cc1ccc2c(CCC(=O)N3CC(N(C(=O)CCCS(C)(=O)=O)C)C3)c[nH]c2c1 10125,C1(NC(C(C)=CC)=O)CCN(C(C2CC(NS(C)(=O)=O)C2)=O)CC1CO 10126,C=C(C)CCC(=O)NC(C1CN(C(=O)C(CCC)c2cccc(Cl)c2)C1)C 10127,C1(N=[N+]=[N-])(C(=O)Nc2c(CC)nn(C)c2)CCN(C(=O)CSc2nc[nH]n2)C1 10128,N1(C(C(C)(C)n2cccn2)=O)CC2(C1)CN(C(=O)CC1CCCCC1)CC2CO 10129,C1(C(N2CC=C(C)C2)=O)(C(C)C)CCN(C(=O)CCC2CCC2)C1 10130,CC(C)CC(O)CNC(=O)CCCCN(C)C(C1(CO)CCCCO1)=O 10131,c1(C(N2CCCCC2C2CCCC2O)C(=O)NCC)cc(Br)ccc1F 10132,CC1(C)C(c2cccc(Cl)c2)CCN1C(c1nn(CC(F)(F)F)cc1Cl)=O 10133,c1(C(=O)NC2CC(NC(c3c(CC)nccn3)=O)C2)nc(C2CC2)ncc1Cl 10134,CN1CCCC1(C)C(=O)NCCOC1CN(C(=O)CC2CCCS2(=O)=O)C1 10135,C(=O)(C#CC1CCCO1)NCC(CC(C)C)NC(=O)CSc1nncn1C1CC1 10136,C1(C(=O)NCCCCNC(C(C)CN2CCOCC2)=O)Cc2ccc(F)cc2O1 10137,C1(c2ccccc2)(NC(CCN(CCCCC)C)=O)CCN(C(=O)CC2CC2)C1 10138,c1(C(=O)NCCN(C(c2cc(C)oc2C)=O)C)ccc(C)c(S(=O)(=O)C(C)C)c1 10139,c1(C(N2CC(NC(C3(O)CCOC3)=O)CC(C)(C)C2)=O)cnnc2ccccc12 10140,C1(NC(c2c(C)nns2)=O)CCCN(C(=O)CC2CCN(C)C2)C1C 10141,c1(C(=O)NC(C2C3CNCC23)C(=O)OC)csc(Cl)c1OC 10142,c1(OC)ccc(O)cc1C(=O)NCC1CCCC(NC(C2CC(F)C2)=O)C1 10143,c1(C(N2CC(N(C(c3c(C)nccc3)=O)C)C(O)C2)=O)cc(C2CC2)nnc1O 10144,c1(CC(=O)N(C2CCN(C(c3c(CC)cco3)=O)C2)CC2CC2)cncnc1O 10145,n1(CC(CC)CC)nc(C(C)C2CC2)nc1-c1ccc(C(=O)N(C)C)cc1 10146,CC(CCN(C(=O)CCc1nncs1)C)NC(C1CC1CN(C)C)=O 10147,Cc1cccc(N2CCC(NC3CC4CCC3O4)C2=O)c1 10148,N1(C(C(Cn2ccc(C)n2)C)=O)CCC2CN(C(c3cn(C)ccc3=O)=O)C2C1 10149,C1(c2nn[nH]n2)(CCN2C(=O)CCC2=O)CCN(C(=O)COC(F)F)CC1 10150,c1(C(=O)NCC(CN(C(c2ncc(C)c(C)c2)=O)C)C)ccc2ccnn2c1 10151,C1(C(N2CC(OC)(CNC(=O)C(C)C3CCCC3)C2)=O)COC(=O)N1C 10152,N1(C(C2CC(SC)C2)=O)CC(NC(c2csnc2C)=O)CC12CCCC2 10153,CC(=O)CCCC(=O)NCC1C(O)C(O)CN1C(c1c[nH]nc1Br)=O 10154,C1(NC(c2c(C(C)C)nns2)=O)CN(C(=O)C2=CSCCO2)CCC1CO 10155,N1(C(c2ncn(C)n2)=O)CC(NC(=O)C(F)(F)C2(O)CCC2)CC12CCCCC2 10156,CCC(C(=O)N(C)CC1(CNC(=O)Cc2ccncc2Cl)CC1)C(F)(F)F 10157,C12(NC(=O)COc3ccon3)CCCN(C(C3(CO)COC3)=O)CC1C2 10158,N1(C(c2n(CC)ccn2)=O)CC2CC1C2NC(=O)CCCN1C(=O)CCC1=O 10159,C1(C2CN(C(=O)C(F)(F)C3(O)CCCC3)C2)(NC(c2ccc(CF)cc2)=O)CC1 10160,c1(C(=O)NC(c2cccc3cc[nH]c23)CC)cnn2cc(-c3nn[nH]n3)cnc12 10161,c1(C(N(CC(CN(C(=O)CC2CCCC2)C)O)C)=O)cc(P(C)(C)=O)cs1 10162,CC1CC(C(=O)N(CCC(=O)NCC(C)S(C)(=O)=O)C(C)C)=NO1 10163,c1(C(=O)NCCN(C(=O)CCSCC(C)C)CC)cc(Br)c[nH]1 10164,c1(C(=O)NCC(CNC(CCCOCC=C)=O)C)ccc(S(=O)(=O)C(F)F)cc1 10165,Cc1cccc2c(C(=O)NCC34CCC(CC3)N(C(C3CCCS3)=O)C4)n[nH]c12 10166,c1(C(N2CC(F)CC(NC(=O)CSc3nncs3)C2)=O)cc2cn[nH]c2cn1 10167,c1(C(=O)NCC2C(C)(C)C(NC(=O)COC3CCC3)C2)ccccc1[N+](=O)[O-] 10168,CC1C(=O)CC2CCC1N2C(=O)NNc1nccs1 10169,Cn1cc(SCC(=O)NC2(CNC(=O)C(C)(c3cccs3)N(C)C)CCOC2)cn1 10170,c1(C(=O)NCC2(F)CC(CNC(C(F)=C(C)C)=O)C2)cccc(Br)c1C 10171,c1(C(N2C(CNC(C(C(C)C)C)=O)CC(O)C2)=O)cc(=O)n(C)cc1Br 10172,c1(OC)ncnc(C(N2CCN(C(c3csc(Br)n3)=O)C3CC23)=O)c1F 10173,C(=O)(C(O)C1=CCCCC1)N1C(C2(NC(CC(=O)NCC)=O)CC2)CCC1 10174,CCC(C)(CS(C)(=O)=O)C(=O)NCC(O)CNC(=O)CNC(=O)NC 10175,c1(C(=O)NC2(CN(C(C(CC)OC)=O)C)CC2)cc2c(C#N)cccc2[nH]1 10176,N1(C(COCC#C)=O)CC(C2CCCN(C(C3(CC)CCCO3)=O)C2)C1 10177,N1(C(Cc2c(C)nc[nH]2)=O)CCC(CO)C(NC(C2(C(C)C)CCC2)=O)C1 10178,CN1CCC(COC(=O)CC2(Cc3cccn3Cc3ccccn3)CC2)CC1=O 10179,c1(C(N(CCC(C)NC(=O)C(C)(C)C)C)=O)ccc2c(c1)OC(C)(C)OC2 10180,CC(C1OCCc2ccccc21)N(C(=O)Cc1csc(Br)c1)C 10181,O=C(C(CCC1CCC1)NC(C1CC=CC(O)C1)=O)NCc1ccc(O)nn1 10182,N1(C(Cc2c(C)scc2)=O)CCC(CC(=O)NCCC(C)(C)C)C1(C)C 10183,C1(NC(=O)COc2cccnc2)COCCN(C(C2C3CCCC23)=O)C1 10184,N1(C(CN(CCC(=O)NCC=C)NC(N)=O)=O)CC=CCC1C(=O)OC 10185,C1(NC(c2cncc(OC)c2C)=O)CC2(CCC(NC(=O)C(C)N(C)C)CC2)C1 10186,n1(CC)nccc1S(=O)(=O)NCC(=O)Nc1nc(C(=O)OC)ns1 10187,N(C)(S(=O)(=O)N(C)CC1CC1)CC#C 10188,c1(C(C(=O)NCC=CCl)NC(CN(C)CC)=O)cnn(C)c1 10189,C1(NC(n2cc(-c3ccn(C4CCC4)n3)nn2)=O)CCN(CC2CCCN2)CC1 10190,N1(C(C2C(C)(C)N(C(=O)CC3CC4(CC4)C3)CC2)=O)CCOCC2(CC2)C1 10191,C1(CNC(CN(C2CC2)CC)=O)CN(C(c2cscc2OC)=O)C2CC12 10192,C(N=c1[nH]c(N2Cc3cnn(C)c3C2)nc2c1CC(C)CC2)C1N(CC)CC1 10193,C(=O)(CS(=O)(=O)CCO)N1CC(NC(c2cncc(COC)c2)=O)C(OC)C1 10194,N1(C(C(COC)CC(C)C)=O)CC(C)OC2(CCN(C(=O)CCC(C)C)CC2)C1 10195,C1(C(=O)NCC2(CNC(c3c(CC)noc3)=O)CC2)CCCCC12OCCO2 10196,c1(OC)ccc(NC(c2ncsc2C(C)C)=O)cc1C#N 10197,c1(N2C(C)CC(NC(c3cc(C)nc(C)n3)=O)C2)ncnc2sc(C)c(C)c12 10198,C(CC(C)C(=O)NC1CCC(F)(CNC(c2c[nH]c(C(F)(F)F)c2)=O)C1)OC 10199,Cc1nsc(NC(N2CC(F)CC2C(C)(C)O)=O)c1Cl 10200,C(CC(C)C(F)(F)F)NC(CC1(O)CCN(C(Cc2cccc(C)c2)=O)C1)=O 10201,C1(CNC(C(CC=C)NC(C)=O)=O)CC(C(=O)NCC2(N(C)C)CCC2)=NO1 10202,N1(C(C(C2CC2)SC)=O)CC(NC(=O)CC2CN(C)C2)C(C)(C)C1 10203,C1(NC(C(N)=O)=O)CC2(CCN(C(C3CCCOC3)=O)C2)C1 10204,C1(NC(C2(OC)CCSC2)=O)CCN(C(=O)C(c2c(C)noc2C)C)CC1CO 10205,c1(C(N2CCC(O)(CNC(C3C(CCOC)C3)=O)C2)=O)ccc([N+](=O)[O-])o1 10206,C(=O)(C(C)(O)C(C)C)N(CCC(=O)NC1C2CCCC12)CC=C 10207,C=C(C)CCCC(=O)NCC1(O)CCCN(C(c2cc(CN(C)C)on2)=O)C1 10208,C1(NC(C(C)OCC)=O)CCN(C(=O)Cc2ccc(C(C)=O)s2)CC1(C)C 10209,CC(C)C(C(=O)NC(CNC(=O)Cn1cnnn1)C(C)(C)C)NC=O 10210,C(=O)(C1COc2ccccc21)NCCOCCN(C(=O)C1Cc2ccccc21)C 10211,N1(C(N)=O)CCCC(C)(NC(Cc2cn(CCSC(C)(C)C)nn2)=O)C1 10212,N1(C(=O)NCc2ncc(CC)o2)CCCCC1CCNC(C)=O 10213,c1(CCC(=O)NCC=CCNC(c2c(OC)nsc2)=O)cccc([N+](=O)[O-])c1 10214,N1(C(C(C)OCC)=O)CCC(COC(=O)NCCC2C(NC(=O)C3CC3)C2)CC1 10215,CC(C(=O)NCC1CC(NC(=O)CCCN2CCCCC2)C1)F 10216,Cc1ncc(NC(=O)NCCOc2ccc(Cl)nc2)cc1Br 10217,C(=O)(C1CCc2ccccc21)NC1(C(=O)NCC(c2cnc[nH]2)C)CCCCC1 10218,C1(C(=O)NC(c2ccns2)C)(CC)CCCN(C(c2cnn(C(C)C)c2)=O)C1 10219,C#CCCCCCC(=O)N1CCCC2(NC(=O)C(C)Cc3ccco3)CC2C1 10220,Cc1cc(C(=O)OC(C(=O)Nc2ccc(N(C)C)c(F)c2)C(C)C)ncc1N 10221,c1(NC(C(CCC)C)C)ccc(S(=O)(=O)N(C2(CCO)CCSCC2)C)cc1Br 10222,c1(C(=O)NCCC2CCCN(C(C3CC(F)C3)=O)C2)nccc2n[nH]cc12 10223,c1(C(C)=O)cncc(C(=O)NC(CNC(C2CCC2(F)F)=O)C2CC2)c1 10224,N1(C(CC(C)OC)=O)CC2(CCN(C(=O)C(C)Sc3ccc(N)cc3)C2)C1 10225,c1(NC(C2(C)CCN(C(C3CC3F)=O)CC2)=O)sc2c(c1C#N)CCCC2 10226,C1(C#N)(C(=O)NC2CCCN(C(C(CCC)=CCC)=O)CC2)CC2CCC1CC2 10227,N(C1CCCn2cnnc21)C(N1CCC(C(=O)OCC)C1)=O.CCC 10228,c1(NC(=O)NCc2cccc(-c3cccc(OC)n3)c2)ccc2sc(O)nc2c1 10229,c1(C(N2C(CNC(CNS(N)(=O)=O)=O)CC(O)C2)=O)cnn2c1CCC2 10230,O=C1CC2(CCCN(C(=O)C3=NOC(CO)C3)CC2)CN1 10231,CC(CSC(F)(F)F)C(=O)N1CCCC1CN(C)C(c1ccco1)=O 10232,C(=O)(C(CNC(C1CC1(F)Cl)=O)C(C)C)N1CCC(C(=O)NC)C1C 10233,C1(CNC(CSC)=O)CN(C(c2cc(C(C)(C)C)nn2C)=O)C2(CCC2)C1 10234,CCCC(CCC)CC(=O)NC1CN(C(C2CCCOCC2)=O)CC1OC 10235,C(C1c2ccccc2CN1C)NC(C(C)NC(c1ccc(O)c(N)n1)=O)=O 10236,c1(N2CC(NC(c3cnc(SC)nc3Cl)=O)C2)ncnc2sc(C(C)(C)C)cc12 10237,S(=O)(=O)(c1ccc(C(=O)NC2CCC(CNC(=O)C(C)C(C)O)C2)cc1)NCC 10238,n1(CC(=O)NCCCN(C(=O)CC2(O)CCC2)C)ncccc1=O 10239,c1(C(N(C2CCN(C(COC)=O)CC2)CCO)=O)cnn2cc(OC)ccc12 10240,N1(C(C(C)NC(N)=O)=O)CCN(C)C(CNC(c2nsnc2O)=O)C1 10241,C1(N(C(C(=O)Nc2ccccc2)=O)CCCO)CC2CC1CN2 10242,c1(C(=O)OCC)ccccc1NC(C1CC1CNC(=O)CCc1ccn(C)c1)=O 10243,CC(CNC(C1(F)CCN(C(c2ccc(Cl)cn2)=O)CC1)=O)CC(F)(F)F 10244,C1(C(=O)NCC(CNC(Cc2c(C)n[nH]c2)=O)C)CCCN(C(C)C)C1 10245,c1(N(C)CC2CCN(C(C3N(C(CCC)=O)CCCC3)=O)CC2)nnc(C)c(C)n1 10246,c1(N2CC(C)S(=O)CC2)ccc(Br)c(S(=O)(=O)N(CC(O)CF)C)n1 10247,CN1CCCC1C=CC(=O)NC1(C(=O)N(C2CSC2)C)CC(F)C1 10248,C12(CNC(c3ccccc3)=O)CCC1CN(C(c1ccc(=O)n(CCO)c1)=O)C2 10249,C1(Nc2nccc(OC)n2)(CO)CCN(C(C)=O)CC1.C12(CCCC1)C(=O)N2 10250,N1(C(CC2(N(C)C)CC2)=O)CC(NC(=O)Cn2cc(Cl)cn2)C(C(F)F)C1 10251,C1(CC(N2CCN(C(C3N(C)CC(O)C3)=O)CC2)=O)CCc2ccccc2C1=O 10252,c1(OC)nsc(OC)c1C(C)NC(C1(n2cc(F)cn2)CC1)=O 10253,C1(O)(CCNC(COCCOCC)=O)CCN(C(c2cccnc2N(C)C)=O)C1 10254,C12(CN)CCCN(C(=O)NCC=CCCC(C)C)C1C2 10255,C1(C(=O)OC)CCOC1C(=O)NCCN(C)C(C1CC(C(C)C)C1)=O 10256,C(CCCC(=O)N1CC2C(C)C2C1)NC(COCC)=O 10257,CCS(=O)(=O)CCNC(=O)C(C(C)C)c1ccn(C)n1 10258,c1(C(N2CCCC(CNC(C(C)(C)OCC)=O)C2)=O)cc(Cl)c(OC)cc1C 10259,C(=O)(C(C)(C)CS(C)(=O)=O)NCCCC(C)NC(=O)C(O)CC(N)=O 10260,C(=O)(CC(C(C)C)NC)N1C(N(C(=O)C(=O)NCCOC(C)C)CC)CCC1 10261,c1(C(N2C(C(C)(C)NC(C3CC3CF)=O)CCC2)=O)cc(O)ccc1Cl 10262,Cc1cnc(Cl)[nH]c1=NCC=Cc1ccc(C2CC(OC(C)(C)C)C2)cc1 10263,N1(C(c2c(Cl)ncc(C)c2)=O)CC2CCN(C(c3cc(Cl)c(Cl)cn3)=O)C2C1 10264,c1(C(=O)NC(C)C(C)(C)NC(=O)CCC(C)C#N)cc(N(C)C)ccc1F 10265,N1(C(C2CCN(C(=O)CCc3ccccc3)CC2)=O)CCOCC2(CCC2)C1 10266,c1(C(=O)NCC(CN(C(c2c(C)noc2N)=O)C)C)cc(Cl)ccc1Cl 10267,N1(C(CCC2C(C)C2)=O)C2CCC1CN(C(c1ccns1)=O)C2 10268,Cc1cc(C(=O)NCC2CN(C(=O)COCCF)CC2C)c2c(C)nn(C)c2n1 10269,c1(C(=O)NCC(C2N(C(C(CC)CC)=O)CCCC2)(C)C)cnc2ccnn2c1 10270,N1(C(=O)CCN(C(c2nsnc2O)=O)CC2CC2)CC23CCC2(COC3)C1 10271,c1(NC(C2(C)CCN(C(c3ccc(CF)cc3)=O)C2)=O)ccc(F)c(O)c1 10272,Cc1nn2c(C(N3CC4CC4(NC(=O)C(C)C(=O)OC(C)(C)C)C3)=O)c(C)nc2s1 10273,CCC(Cc1cccc(C)c1)C(=O)NCC(C(C)C)NC(=O)C(Cl)=CCl 10274,C(=O)(C(C(=O)N1CCCC(C(=O)NCOC)C1)OC)OCC.C1(=O)CC(SC)N1 10275,C(=O)(CC(C)C(F)(F)F)NCC1CN(C(C=C(CCC)C)=O)C(C)C1 10276,C1(CCNC(CCC#CC)=O)CN(C(C2CC3CCC3C2)=O)CCS1(=O)=O 10277,C1(C(=O)NC2(CCC)CC2)C(C2CC2)CCN1C(=O)COCCCF 10278,C1(N(S(=O)(=O)CC#N)C)CCCN(C(c2ccc(C(=O)O)cc2)=O)C1=O 10279,N1(C(CC2(C(=C)F)CCC2)=O)CCC(C(=O)NCC(Cl)C(C)(F)F)C(C)C1 10280,N1(S(CC)(=O)=O)CCC(C(=O)NCC2CN(C(=O)C=CCOC)CC2O)CC1 10281,C(=O)(CCC(=O)NCCCCCCNC(C1CC1(Br)Br)=O)NCC 10282,C1(NC(C2(C(=O)NC)CCC2)=O)CN(C(c2cc(Cl)ccn2)=O)C2(CCOC2)C1 10283,c1(C(N2C(C)C(NC(=O)CCc3ccnn3C)CC2)=O)cc2ncccc2s1 10284,C1(C(=O)OCC2C(Cl)(Cl)C23CC3)CNC(=O)CN1C(=O)NC(C)(C)C 10285,C#Cc1ccc(C(N2CCCC2CCC(N2CCOCCC2C(N)=O)=O)=O)cc1 10286,c1(CC(N2CCC(Cc3cn(CCF)nn3)C2)=O)ccc2c(c1)CCO2 10287,C(=O)(C(CC(C)C)C(C)C)N1CC(OCC)(CNC(c2cncc(N)n2)=O)C1 10288,Cc1c(CN2CCC(O)CC2C(N2C3CCC2CC3)=O)[nH]c2ccccc12 10289,N1(C(N2CCC(CNC)C2)=O)CCCCC1CC(C)C 10290,C1(CC)CN(Cc2cccc(-c3ccccc3)n2)CCN1C(C1CC1F)=O 10291,Cc1ccc(C(=O)NCC(=O)NCC(C2CC2)NC(=O)C=CSc2nc[nH]n2)s1 10292,N1(C(c2cnc(C)c(N)c2)=O)CCCC12CCN(C(=O)C(C)CC(C)(F)F)C2 10293,CC(N=[N+]=[N-])C(=O)N1CC(C(=O)NCCC2COCC2O)C(C)C1 10294,c1(C(=O)NC2CCC(S(C)(=O)=O)C2)csc2ccc(F)cc12 10295,c1(C(=O)NC2(CNC(C3=CCC(C)(C)CC3)=O)CC2)cc(Cl)cc2c1NCCC2 10296,N1(C(c2cc(CC)nc(O)c2)=O)CC2(CCN(C(=O)C(C)NC(=O)NC)C2)C1 10297,C1(CNC(c2cn(CCCC)nn2)=O)C(C)CCCN1C(=O)C#CC(=O)N(C)C 10298,c1(C(=O)OCC2(C(=O)O)C3CCC23)cnn2c(OC)cccc12 10299,C1(C(N2CCC(CCOC)(NC(CC=CC)=O)C2)=O)CC2COCC2C1 10300,C1(C(=O)NCC(CCC)OCC)CCC2CCC1N2C(c1ccccn1)=O 10301,N1(C(Cc2c(C)oc(-c3ccsc3)n2)=O)CCc2nncn2CC1 10302,CC(C)C(C(=O)NC1(C)CN(C(C2CCC(=O)C2)=O)C1)c1cccc(Cl)c1 10303,c1(C(=O)NCCNC(CCc2ccc(C)nc2)=O)nc(C)n(C)c1C 10304,c1(CC)cc(C(N2CC(NC(=O)CS(=O)CC)C(SC)C2)=O)nn1CCO 10305,c1(C(N(OC)Cc2cnn(C)c2)=O)ccc(C(=O)O)cc1Cl 10306,C12(CNC(c3cncc(COC)c3)=O)CCC(CC1)CN2C(=O)CC1CCC1 10307,c1(CC)ccoc1C(=O)N(CCNC(c1ccc(CS(C)(=O)=O)o1)=O)CC1CC1 10308,c1(CNCC2(C(=O)O)CCSC2)ncnc(O)c1F 10309,N1(C(C(C2CCCO2)SC)=O)CCC(N(C(=O)CCOC2CCC2)CC2CC2)CC1 10310,N1(C(c2cnc(Br)s2)C(=O)NCC=C)CCC(C)(O)C(C)(O)C1 10311,N1(C(c2nccc(C)c2O)=O)CCC2(CCC2)C(NC(C2CCCSC2)=O)C1 10312,C1(N(C(C2CC(=C)C2)=O)C)CCC(n2cc(CCc3nn[nH]n3)nn2)CC1 10313,S(=O)(=O)(c1ccc(NC2(C(=O)O)COC(C)(C)C2)cn1)NC(=O)OC(C)(C)C 10314,N1(C(CCCCCOC)=O)CC(CNC(C2(CF)CC2)=O)CC12CCC2 10315,N1(C(CC2C(=O)NC(=N)S2)=O)CC2=C(C1)CN(C(C13C4C5C1C1C3C4C51CO)=O)C2 10316,c1(C(=O)NC(CC2(CC)CCC2)=O)cc(CN2CCCC(NC(C)C)C2)ccn1 10317,C(=O)(C(C)(C)C(C)(C)O)N(C(C(=O)NCC(C)CN(C)C)CC(F)F)C 10318,Cn1c(C(=O)NC2(c3cccc(C#N)c3)CCOCC2)cc2cc(Cl)ccc12 10319,C(=O)(CCCC(=O)N1CCC(C(F)(F)F)C(OC)C1)NCCC 10320,C1(NC(c2c(CC)nc(C)nc2)=O)CN(C(=O)Cc2ccnn2C)CC12CCC2 10321,N1(C(CN(S(C)(=O)=O)C)=O)CCN(C)c2ccc(NC(=O)OC(C)(C)C)cc21 10322,Cc1c(C(=O)Nc2cc(OC3CCCCC3)ccn2)cnn1C1CC1 10323,C(=O)(N=S(=O)(c1ccc(F)cc1)C(F)F)C1(C)CCN(C)C1 10324,C1(CC=C)(NC(c2csc(CC)n2)=O)CN(C(=O)C(F)CC2CCCC2)C1 10325,N1(c2nc(OC)c(C)cn2)CCOC2(CCCN(C(=O)CC3CCC3)C2)C1 10326,Cc1ccc(C(=O)NCC(N2CCN(C(=O)C3=NOCC3)CC2)C)c(F)c1 10327,C1(COC)(NC(=O)CN2CCS(=O)CC2)CCN(C(C2(Cl)CC2(F)F)=O)C1 10328,C12(C(=O)NC(C3(C)C(C)CCC3)c3ccccc3)CC(CO1)N(c1cnccn1)C2 10329,c1(C(N2CC(OC)C(NC(C3C(Cl)(Cl)C34CC4)=O)C2)=O)cccc(F)c1F 10330,c1(C(C(=O)NCc2cn(CCSC)nc2)CC)cccc(Cl)c1 10331,C(=O)(CCCCCc1ccccc1)NCC1N(C(c2c(COC)cc[nH]2)=O)CC1 10332,N1(C(C2CC(N(C)C(C34CC(CO)(C3)C4)=O)C2)=O)CCC([N+](=O)[O-])CC1 10333,C(=O)(CCCCCC#N)N1CC(C(=O)NCC(C)C2CCC2)N(C)CC1 10334,C1(CNC(CS(CC)=O)=O)COCCN(C(C2CC(N3CCCC3)C2)=O)C1 10335,C(C(CC(=O)N(C1CCSC1)C)NC(=O)C=Cc1cc(C)no1)OC 10336,C1(NC(c2ccc(CC)c(Cl)c2)=O)COC2C(NC(=O)CC(=O)N(C)C)COC12 10337,C(=O)(CCC(C)(C)C)N1CC(C)C(CNC(c2cn(CCCF)nn2)=O)C1 10338,c1(C(=O)NCC(CN(C)C(C2COC3(CCC3)CO2)=O)O)cnc2cc[nH]c2c1 10339,N12CC3CCC3(C1)C2=O.Cc1cc(C(=O)Nc2ncc(C3OCCO3)s2)nn1C 10340,N(C1CCCn2ccnc21)C(C(CCNC(c1c(C)cn(C)n1)=O)O)=O 10341,c1(C(=O)NC(CC=C)CNC(=O)C=Cc2scnc2C)cccc(S(C)=O)c1 10342,N1(C(C(CSC)C)=O)CCC(O)(CNC(c2c(C)coc2C)=O)C1 10343,Cc1nsc(C)c1C(=O)NCC1CC(C)N(C(=O)Cc2ccc(C(N)=O)nc2)C1 10344,Cn1nnc(C(=O)NCCOCCNC(=O)CCCc2ccccc2)n1 10345,C12(NC(c3c(CC)ocn3)=O)CCN(C(c3cc(C(C)(C)C)no3)=O)CCC1C2 10346,N1(C(CSCCC(C)C)=O)CCCC2(NC(c3cncc4sccc34)=O)CC2C1 10347,c1(N2CCCC(N(C(COc3cccc(OC)c3)=O)C)C2)ccc2nnnn2n1 10348,CC12CCC(C(N3CCOC(CNC(=O)CSC4CC4)C3)=O)(CO1)C2 10349,C1(CNC(C(c2ccccc2)OC)=O)CCN(C(C2CC(N(C)C)C2)=O)C12CC2 10350,c1(C(N2CCC(C)(NC(C3C4COCC34)=O)C2)=O)cccc2c1OCCN2 10351,c1(C(N2CCCCC(NC(c3cc(OC)no3)=O)C2)=O)cnc2c(n1)CCCC2 10352,c1(C(N(C)CC2N(C(C(C(CC)C)O)=O)CC(F)C2)=O)cc(C)cc(C)c1C 10353,N1(C(C2N(C(C3C(C)C4CCC3C4)=O)CC(F)(F)C2)=O)CC(=O)N2CCCC2C1 10354,c1(C(=O)NC2(C)CC(OCC)C2)ccc(-c2ccccc2)c(C)n1 10355,C1(CNC(CN(C)C2CC2)=O)CCCC(NC(C2(O)CCOCC2)=O)C1 10356,C(=O)(C(C)C(C)S(C)(=O)=O)N1CC2C(CNC(CCCCC(C)C)=O)C2C1 10357,N(C1CCc2cccnc21)C(C1(NC(c2ccnnc2)=O)CCN(C)C1)=O 10358,C(=O)(NN=Cc1cccnc1)c1c(C)cc(C(=O)O)s1 10359,N1(C(C(C)(C)OC)=O)CCC2(CC1)COC(CNC(=O)C(C#N)C1CC1)C2 10360,C(=O)(N1CCCc2nccn21)c1ccc(CNC(=O)C=CCN2CCC2)cn1 10361,c1(C(=O)NC2(CNC(c3n[nH]c(C)c3Cl)=O)CCOC2)ccnc2ccsc12 10362,N1(C(c2cncc(C=C)c2)=O)CC2(C(=O)NCC3CCOC3)CCC1CC2 10363,c1(OC)cc(OC)cc(C(=O)NC2CCCC2CNC(C2CC(OC)C2)=O)c1 10364,C1(NC(c2c(OC)noc2C2CC2)=O)CCC(C)N(C(=O)C(O)CC(N)=O)C1 10365,CC#CCC(C(=O)NC(COC)C1(C)CC1)NC(=O)Cc1cnn(C)c1 10366,c1(C(=O)Nc2scc(-c3c(OC)ccc(Br)c3)n2)cc(C)c(C)cc1I 10367,c1(OCCC)cccc(C(c2nnnn2C)N(C2CCC2)C2CC2)c1 10368,CC1(NC(=O)C(F)CC2CCCC2)CC(NC(=O)Cn2ccc(C(F)(F)F)n2)C1 10369,c1(CC)cc(N)ccc1C(=O)NC(C)(C)CNC(C1(C(F)(F)CC)CC1)=O 10370,N1(C(c2c(C)nn(C3CCC3)c2)=O)CCC2(CCC2)C(NC(C2CC(O)C2)=O)C1 10371,n1(CC(=O)NCCC(C)NC(=O)CCOC2CCOC2)cnccc1=O 10372,c1(OC)ccnc(O)c1C(=O)NC1CCCCN(C(C2C3CC(=O)CC23)=O)C1 10373,N1(C(c2c(C)ccc(NC(COC)=O)c2)=O)CC(C)N(C(=O)CCF)C(C)C1 10374,N1(C(COCC(C)C)=O)CCC(N(C)C(C2CC3(CC(=O)C3)C2)=O)C(C)C1 10375,CC(CC1CCC1)C(=O)NCC1(NC(c2cnnn2C)=O)CCCC1 10376,C1(C(C(C)C)NC(Cc2nnc(C)o2)=O)CCN(C(C2(O)COC2)=O)CC1 10377,C(=O)(C1=CC2CCC1C2)N1CC2C(CNC(c3cn(CCOC)nc3C)=O)C2C1 10378,S(=O)(=O)(c1cccs1)N1C(C(=O)Nc2c(C(=O)OC)nc[nH]2)CC(OC)C1 10379,c1(CNC(CN(CC(C)(C)C)C)=O)nc(O)c2ccc(Cl)cc2n1 10380,c1(C2(C(=O)NCCN(CCC)C(C3CC3[N+](=O)[O-])=O)CC2)ccccc1 10381,C1(Nc2ccc(COC)cc2)CCC2CN(C(c3ccc(Cl)cc3Cl)=O)CC12 10382,N1(C(=O)OC(C)(C)C)CCC(NC(N(C(C)C(c2ccccc2)C)C)=O)CC1 10383,c1(OC)c(C(N2CC(=C(F)CNC(=O)CC(O)C3CC3)C2)=O)c(C)nn1C 10384,C1(NC(C23CC(C)C2C3)=O)CN(C(c2ccc(CS(C)(=O)=O)o2)=O)C(C)(C)C1 10385,N1(C(C)C)C(=O)CCC1C(=O)N(C1CCN(C(=O)CC2(C3CC3)CC2)C1)C 10386,c1(CC(=O)NC2(CC=C)CCN(c3nccn4nnnc34)C2)ccc2c[nH]nc2c1 10387,C(=O)(C(C)(C)CF)NC(C)C(c1ccccc1)NC(c1cnc(N)cn1)=O 10388,Cn1cnc2nc(N3CC=CC(NC(c4cc(C5CC5)[nH]n4)=O)C3)ncc12 10389,CC(C)(C)C(O)CCC(=O)N1CCN(C(=O)CCCCCC#N)CC1 10390,c1(SC)ccccc1C(=O)NC(C)CC1CN(C(=O)Cc2[nH]nnc2C2CC2)C1 10391,Cn1ccc2nc(N3CCC(O)C3C(=O)Nc3ccc(F)nc3)ncc12 10392,c1(CNC(C2CCCCCCN2)=O)ccc2c(c1)CCCN2 10393,c1(CC(=O)NC2C3CN(C(C(CC)=CC)=O)CC2C3)ccc2nsnc2c1 10394,CCC(C)(C(=O)NCC1CN(C(=O)Cc2cc(C)[nH]n2)C(C)(C)C1)C(N)=O 10395,C#CCC(C(=O)N1CC(C)(COC)C1)NC(=O)CCN=[N+]=[N-] 10396,c1(OC)cnc(C(=O)N(C)CCN(C)C(c2n[nH]cc2CC(C)C)=O)c(OC)n1 10397,C(C#Cc1ccccc1)N1CCN(C(=O)CC2(O)CCOC2)CC1 10398,C1(CC)CN(C(C2CC(O)C2)=O)CCC1NC(C1CN(C2CCOC2)C1)=O 10399,c1(C(=O)NC(CNC(C2(C)CCN(C)C2)=O)(C)CO)cccc2c1OCC2 10400,CC(C)CC(=O)C(=O)N(CCCCC(=O)NC(C)CCCCO)C 10401,N1(C(CCNC(=O)C2CC2)=O)CCC2(CC1)OCCCC2NC(=O)Cc1ccon1 10402,C1(CNC(c2cc(C)on2)=O)C2CN(C(=O)C(C)(C)N3CCOCC3)CC12 10403,C1(OC)CCC12CC(C(=O)NCCC1CCN(C(c3cnc(=N)[nH]c3)=O)CC1)C2 10404,C(CCF)(C(=O)N(CCNS(N)(=O)=O)CCO)NC(CCC1(C)CC1)=O 10405,C#CCCCCCCC(=O)NC(C(=O)NC1CCC(=O)NC1(C)C)C(C)OC 10406,C(=O)(CC(C)C(F)(F)F)NCC(C)NC(c1onc(CC)c1C)=O 10407,N1(C(CC2(COC)CC2)=O)CC(NC(c2ccc(-c3cscn3)cc2)=O)C(O)C1 10408,N1(C(c2cn(CC(CC)O)nn2)C(=O)NC(C)(C)CC)CCOC(C2(C)N=N2)C1 10409,C1CCNC(=O)C1.C#CC1(OCC(C(CCC2(N)CCC2)=O)=O)COC1 10410,C(c1ccc(CN(C)Cc2cc(Br)ccc2Cl)cc1)=CC(=O)OC 10411,CC(C(=O)N1CCCCC1CN(C)C(C1(C)C=CCC1)=O)C(C)O 10412,CCCCS(=O)(=O)CC(=O)NCC1(C2CC2)CCN(C(C2CCS(=O)(=O)C2)=O)C1 10413,c1(CN2CCC(C#N)(CC)C2)cc(Br)cc(F)c1O 10414,S(=O)(=O)(c1ccc(C(N2CC(CNC(=O)C(C)C#N)C(C)C2)=O)cc1)NC(C)C 10415,CC1CCCCN1CCC(=O)NCC1CCN(C(=O)C(c2ccccc2)=O)C1 10416,N1(c2nccc(OC)n2)CCC2(CC1)CC2NC(c1ccn(-c2ccccc2)n1)=O 10417,C1(NC(C2CC(OC3CCC3)C2)=O)CC2CN(C(C3CCC3)=O)CC2C1 10418,C1(C(=O)NC2(CC(=O)NCC3(C#N)CCCC3)CCCCC2)CC(C2CC2)=NO1 10419,C1(O)(CCNC(C(C)C#N)=O)CCN(C(c2cc(C(N)=O)n(C)n2)=O)CC1 10420,c1(C(=O)NCC(C)(CO)NC(CC(CC)C(F)F)=O)c(F)ccc2occc12 10421,c1(CNC(C2=NOC(C)(C)C2)=O)ccc2c(c1)CN(C(C13CC(CO)(C1)C3)=O)C2 10422,C(=O)(C1CCCc2sc(=N)[nH]c21)N1C(CNC(CNC(CC)=O)=O)CC(F)C1 10423,C(=O)(C(CCS(C)(=O)=O)OC)NC1CCN(C(CSCC#C)=O)CC(O)C1 10424,C1(C(Cc2nnnn2C)NC(c2ncnn2C)CC)CCC(F)(F)CC1 10425,C(CN=c1cc[nH]cc1S(=O)(=O)NCCN1CCCC(O)C1)N(C(C)C)C 10426,C12(NC(CNC(N)=O)=O)CC1CN(C(=O)CC(F)(F)Cl)C2 10427,c1(OC(C)C(=O)NC(C2CN(c3cncc(Cl)n3)CCO2)C)ccc(Cl)cc1 10428,N1(C(=O)NCC2CCSCC2)CCN(c2ccc(F)cc2F)C(=O)C1 10429,C1(C2(O)CCN(C(c3ccc(Br)c(O)n3)=O)CC2)(NC(C(N)=O)=O)CC1 10430,N1(C(C(CNC(C2CCC(=O)N2)=O)CC2CC2)=O)CCSC2(CCC2)C1 10431,C(=O)(C(C(=O)O)C(C)C)N(C1CCCN(C2CCC2)C1)CCOc1ccc(C)cc1 10432,CC1COC(C)CN1C(c1ccc(Cl)s1)C(=O)NCC1CC1 10433,C=C(Cl)C(C)(C)C(=O)N1CC2CC(NC(C3(F)CCOC3)=O)C1C2 10434,C1(C(=O)NCCCNC(c2ccc(C3(F)CC3(F)F)cc2)=O)CCCC12CC2 10435,C#CCC(CC(=O)Nc1cncnc1C)NC(C1OCCC1C(C)C)=O 10436,c1(NC(C(=O)N(C2CCOC2)CC#C)=O)cc(C2CCCCC2)ccc1C 10437,c1(C(=O)NC2CC2CNC(C2CC3COCC3C2)=O)ccc([N+](=O)[O-])cc1Cl 10438,C1(C(=O)NC2CN(C(CCc3n(C)ccn3)=O)CC2O)CNC(=O)CC12CCC2 10439,Cc1cc(C(N2CC3CCN(C(=O)COC4CCOC4)C3C2)=O)c2[nH]cnc2c1 10440,N1(CC=CC)C(=O)CCC1CC(=O)NC1CN(C(=O)Cn2cc(C(C)=O)nn2)C1 10441,c1(C(N(CCN(C(Cc2c(C)cco2)=O)C)C)=O)cc(Cl)sc1Cl 10442,C(C(=O)NC(CSC)C(=O)N(C1CCC(C)(C)C1)C)(C(C)C)SC 10443,N12CCC(O)C(C1)C(=O)N1CCC2C1.C(COCCO)OCC 10444,c1(C(=O)NCC2N(C(CCCOC)=O)CCC2C)ccc2c(c1)CCS2(=O)=O 10445,c12cnn3ccc(nc13)[nH]2.c1(C(=O)OCC)c[nH]nc1C(=O)N(C1CNC1)C 10446,c1(C(N(C2CN(C(c3ccc4c(c3)CC4)=O)C2)C)=O)cnc2sccn12 10447,N1(C(=O)CCCF)CC2CN(C(C3C4C=CC(C4)C3CO)=O)CC(C1)O2 10448,Cc1cnc(C(=O)NCc2cccc(NC(=O)C(CC#N)c3ccccc3)c2)nc1 10449,C#Cc1ccc(CCCC(=O)N(CC(C)CNC(=O)CC=CC(C)(C)C)C)cc1 10450,c1(C(N(CCC(=O)OC)Cc2ccccc2)=O)ccc([N+](=O)[O-])c(F)c1 10451,N1(C(CCC2CCC(NC(=O)C3=NOCC3)C2)=O)CCCCC(CO)C1 10452,N1(C(C(CCC)CCC)=O)CC2(C1)CN(C(C1CCC(NC)CC1)=O)CCO2 10453,CC1(C(=O)NCCCNC(C23CC(c4ccccc4)C2C3)=O)CCCS1(=O)=O 10454,C(CCCCCS(N)(=O)=O)NC(=O)OC(C)(C)C.c12cccc(c1)CN(C=O)C2 10455,C(CN=c1nc(OC(C)C)cc[nH]1)C1CCC(Cc2cc(OC)nc(C)c2)C1 10456,Cc1nc(C(N2CC3CC2C3NC(C2(C)CCCOC2)=O)=O)cn1C(F)F 10457,N1(C(C2CCN(C(C)C)C2)=O)CCN2C(C)COCC2C1 10458,c1(C(N(CC(CC)NC(C2C3CCCC23)=O)CC)=O)csc(-c2ccccc2)n1 10459,C(=O)(CCC(C)(C)F)NC1CCN(C(C(C)NC(CC)(C)C)=O)C1 10460,C(=O)(C(O)CC(C)C)N1C(COC)(CNC(=O)C(C)=C2CC2)CCC1 10461,C1(COC(C(=O)NC(CC)C(=O)OC)C)CCN(C(=O)NCCOC)CC1 10462,Cc1cc(NC(=O)CCC(C)NC(=O)CCCN(C)C)cc(CO)c1 10463,C(=O)(C(CC(C)C)C(N)=O)NC(CC)CNC(c1sc(F)cc1Cl)=O 10464,C=CCC(CNC(c1cn2c(n1)CCC2)=O)C(=O)NC(CN(C)C)CO 10465,C(=O)(C(C)C1=CCCC1)NCCCN(C(=O)CCC(=O)c1ccccc1)CC 10466,C1(OCC=C)CCN(C(=O)C(CNC(C2CC2(F)Cl)=O)N(C)C)C1 10467,C1(CNC(C(C)=CC)=O)CCN(C(C2CCn3cc(C)nc3C2)=O)CCC1(F)F 10468,Cc1cccc(OCC(=O)NCC(C)N(C(=O)C(F)C2CCOC2)C)c1 10469,c1(CNC(C2(C)CC=CCO2)c2n(CC=C)nnn2)cc(OC)c(OC)c(Cl)c1 10470,Cc1ncc(CCNC(=O)C(C2CCN(C(c3csc(C)n3)=O)C2)C)s1 10471,c1(OCC(N2CC(O)(CNC(C(c3ccc(F)cc3)C)=O)C2)=O)cncc(Cl)n1 10472,N1(C(C(C)(C)Cl)=O)C2CC1CN(C(C1(c3ccccc3F)CC1)=O)C2 10473,c1(OC)ccc2c(c1)C(C(=O)NC1(C)CN(C(=O)CCOC3CCCC3)C1)CC2 10474,N1(CCC(C2(CC(C)C)COC2)=O)CCC(N=c2nc(C3CCCC3)[nH]s2)CC1 10475,C1(CNC(c2c(OC)n[nH]c2)=O)CN(C(C2(F)CC=CCC2)=O)CCN1C 10476,C(c1ccncn1)=CC(=O)NC(CNC(CNS(NC)(=O)=O)=O)(C)CO 10477,c1(CNC)cn(C(C)C)nn1.N1(C(CC2(COC)CC2)=O)CC(CC=O)C1 10478,C(=O)(C1(C)CCn2ccnc21)NCC(C)CN(C)C(c1csnc1Cl)=O 10479,C1(CC)CCOCCN1C(=O)CC(C1CC1)NC(c1cc(C)no1)=O 10480,C(=O)(CCCS(C)(=O)=O)NC1CC2CC(NC(c3ccnn(C)c3=O)=O)CC21 10481,C=CC1(O)CCN(C(=O)Cc2ccc(F)cc2I)C1 10482,c1(C(=O)NCC2(O)CCN(C(Cc3n(C)nnc3)=O)C2)c2c(nn1C)CCSC2 10483,c1(C(=O)NCCCC(=O)N2CCC(c3nc[nH]n3)C2)ccc([N+](=O)[O-])o1 10484,Cc1cc(C(=O)NC2CC(NC(=O)CC3CSC3)C23CCC3)cc(Cl)c1 10485,C1(C(=O)NCC(CNC(C2(CSC)CCC2)=O)CO)CCC(C)(C)C1 10486,C1(C(N2CC(C)C(NC(COCCOC)=O)C(C)C2)=O)CCc2nnnn2CC1 10487,Cc1cc(=NCC(C)CNC(=O)C=C2CCSCC2)[nH]c(CO)n1 10488,C(=O)(C(C)S(=O)(=O)CCC)N(CCCNC(C1(C#C)CCCC1)=O)CC 10489,N1(C(C(COC)O)=O)CC=CC(NC(C2(C(F)(F)F)CCCCC2)=O)C1 10490,C1(NC(c2cn(CCNC(CC3CC(C)OC3)=O)nn2)=O)(CO)CC2(CCC2)C1 10491,Cc1nc(C2CC2)ncc1C(N1CCC(CN(C)C(c2ccsc2Cl)=O)C1)=O 10492,C#Cc1cnc(C(N2CCOCCC2C(=O)NCC(C(C)(C)C)OC)=O)c(C)c1 10493,C1(CC(=O)NC2CN(C(=O)CCc3nncs3)C2)COC(=O)C1 10494,C(c1ccc(CN2CCCC2=O)o1)=CC(N1C(CNC(C(CC)=CC)=O)CC1)=O 10495,C(=O)(C1=CCC(C)CC1)N1CCC(C(C)NC(=O)Cn2cnnc2O)C1 10496,c1(NC(N(c2c(C)ccc(C)c2)CCC#N)=O)nc2cccnc2s1 10497,c1(CC)cncc(C(=O)NCC(CCOC)NC(C2(C(=O)NC)CCC2)=O)c1 10498,C(=O)(CC(O)CNC(=O)Cc1cccnc1O)N(C1CCC(C)(C)C1)C 10499,c1(CC)cccc(F)c1C(N1CCN(C(c2ccc(OC)c(N)c2)=O)CC1C)=O 10500,c1(C(N(CCN(C)C(c2csc(C3CC3)n2)=O)C)=O)c(N)ccc(F)c1F 10501,c1(C(N(C(C)CNC(=O)CC2(C)CC2)C)=O)cc(F)c(F)c(O)c1F 10502,C(CCC(C)(C)C(=O)N1CC(O)CC1c1ccc2c(c1)OCO2)OC 10503,Cc1ccc(C#N)c(NC(N2CCCC2c2ncc(-c3ccc(CO)o3)[nH]2)=O)c1 10504,N1(C(C(CC)OC)=O)CCN(C(c2sc(N(C)C)nc2Cl)=O)C(C(C)C)C1 10505,Cc1cc(C(=O)NCC=CCNC(c2c(C)[nH]c(C)c2C)=O)ncc1Br 10506,C1(NC(C=CCC(C)(C)NC(CCOCCC)=O)=O)CCCCC1(C)O 10507,N1(C(C2CCC(C)(C)O2)=O)CCCC2CN(C(c3c[nH]nc3Br)=O)CCC12 10508,c1(C(N(CCOC)CCNC(C2CCC(OC)CC2)=O)=O)cc(C)nc(C)n1 10509,N1(C(Cc2cccc(NC(C)=O)c2)=O)CC2CC(NC(c3scnc3C)=O)C1C2 10510,CCCCC(C(=O)N1CCC(CCO)CC1)NC(c1cn(C)nc1OC)=O 10511,C1(C(N2CC3C(NC(c4ccc(=O)oc4)=O)C3C2)=O)COc2ccc(O)cc2O1 10512,Cn1cnc2[nH]c(=NCC3CCCN(C(=O)CSCC(F)(F)F)C3)nc(O)c12 10513,C(=O)(CCC(O)C(C)(C)C)N1CCC(C(C)NC(CN(C(COC)=O)C)=O)CC1 10514,N1(C(CN(CCC#C)C)=O)CC2CCC(NC(c3sc4ccsc4c3C)=O)(C2)C1 10515,c1(OC)ccc(COCC(O)CNC(C2(c3ccccc3)CC(C)C2)=O)cc1 10516,c1(C(=O)NCC(CO)NC(c2ccc(C(C)(C)C)nc2)=O)ccc(Cl)c(F)c1 10517,Cn1cc(C(=O)OC2CC(=O)N(CCOC(=O)OC(C)(C)C)C2)c(I)n1 10518,CCCC(CN=c1cccc(S(=O)(=O)NC2CCc3ncsc3C2)[nH]1)OC 10519,C1(CC(=O)N(CCOCCNC(c2c(C)csc2)=O)C)CCCC(=O)N1 10520,CCC(CC(F)(F)F)N=c1[nH]c(=NC)[nH]c(=NCCCCN2CC(C)OC(C)C2)[nH]1 10521,C1(C(=O)NCCCOCCNC(C(C)C2=CCCC2)=O)CCC2(CC1)CC2(F)F 10522,C1(C(=O)Nc2ccc(-c3c(C)ncs3)cc2)CCCC12CCOCC2 10523,CC(C)CN=C(NCc1cn(C)nc1C(F)(F)F)NCC1(COC)CCC1 10524,CC(CO)C(=O)N(C)CCOCCCNC(c1cnn(C)c1)=O 10525,C=Cc1ccc(C(=O)NCC(C)(O)CNC(=O)COCCc2ccccc2)cc1 10526,C(CC(C)N=c1ccnc(NCc2ccc(OC)nc2C)[nH]1)OC 10527,n1(CCC(=O)N(CC(C)NC(=O)C(Cl)=CCl)C)c(=O)nc(O)c2ccccc12 10528,c1(OC)c(F)cc(F)c(-c2cnc(C(=O)Nc3ccnc(Br)c3)nc2)c1F 10529,c1(C(N2CCC(OCc3ccccc3)C2)C(=O)NCC)cc(Cl)nn1C 10530,c1(C(C)NC(c2cn[nH]c2)=O)nocc1C(=O)NCC(CO)C1CCC1 10531,c1(OCC=C)ccc(C(=O)OC(c2ccc(C(C)(C)C)cc2)C)cc1 10532,c1(C(N2CC(NC(C3C(CC(C)C)C3)=O)C(C)C2)=O)ccc(=O)n2c1CCC2 10533,N1(C(C=C(C)C(C)(C)C)=O)CCC(C2(NC(C3CC4CC4C3)=O)CCC2)CC1 10534,C1(C(=O)NC2(CCCC)CC2)CN(C(=O)C(C)OCCOC)CC1(C)C 10535,Cc1ccccc1C(=O)NC(CCN(C)C)C(=O)N1CC(C)C(F)C1 10536,c1(CNC(NCC2CC(CC)C2)=NCCF)nnc2c(=O)[nH]ccn12 10537,c1(C(N2CCCCC2COC)C(=O)NCCC)ccc(C)c(OC)n1 10538,CC1CN(C(C2CC23CC(C)(C)C3)=O)CCC1NC(C1CC2(CCCO2)C1)=O 10539,CC1CC=C(C(=O)NCC(C)(CO)NC(=O)CN2CSCC2=O)CC1 10540,c1(OC)nc(N(C2(C#N)CCNC2)Cc2c(F)cccc2F)ncc1F 10541,N1(C(c2nc(C)n(C)c2C)=O)CC2CCCC2(NC(C2CCCC(=O)N2)=O)C1 10542,N1(C(c2n(OC)cnc2C)=O)CC(C)CN(C(=O)Cc2nn(C)cc2Cl)C(C)C1 10543,c1(OC)ncc(NC(C2(F)CCN(C(c3cc(O)ncc3Br)=O)CC2)=O)cc1F 10544,C1(CC(=O)NC(c2cnc(C)s2)C)(NC(c2cocn2)=O)CCCCC1 10545,CC(=NO)C1CC(C(=O)NCC(C2CCN(C(=O)CNC=O)CC2)(C)C)C1(C)C 10546,c1(C(N2CC(C(=O)OC)C(C)(C)C2)=O)ccc(Br)c(O)c1Br 10547,N1(C(c2c(C)cc[nH]2)=O)CCC2(CC1)CC2CNC(c1cnc(S)[nH]1)=O 10548,c1(C(=O)NC2CC(C)CN(C(=O)C=Cc3cccs3)C2)cncc(P(C)(C)=O)c1 10549,N1(C(C2CCCCN2C(C23CC2CNC3=O)=O)=O)CCOC2(CCC2)C1 10550,N1(C(CC2CCCC(OC)C2)=O)CCCC(NC(=O)Cc2cc(Cl)n(C)n2)C1C 10551,C(C)(CN=c1[nH]cncc1C)NC(C(c1ccc(C)cc1)C)=O 10552,c1(C(=O)NCCC(C)NC(c2c(C3CC3)cccc2F)=O)cn2cccnc2n1 10553,C(=O)(C(O)CCS(C)=O)N(C(C)C)CCN(C)C(c1ncc(F)cc1N)=O 10554,C(C(=O)NCCN(C(C1CCC12CCC2)=O)C(C)C)(C(F)(F)F)OC(C)=O 10555,C#CCC(O)C(=O)N1CC(C(=O)NCCCCC2CC2)C(F)C1 10556,N1(S(CCCC)(=O)=O)CCC(C(=O)NCCc2nccs2)(CO)CC1 10557,c1(C(N2CC(C(C(=O)N(C(C)C(C)C)CC)OC)C2)=O)ncc(F)cn1 10558,C1(C(=O)NC2CCCC(CNC(=O)C3=CCCSC3)C2)CCc2ccccc2O1 10559,C1(C(=O)OC)CC(C(=O)NC(C)CCNC(C23COCC(C2)C3)=O)C1(C)C 10560,C1(CC#C)(C(=O)NC(C2CCCC2)CNC(=O)C(C)COCC)CCCCO1 10561,C#Cc1ccc(NCC(CC(=O)N(CC(C)C(F)(F)F)C)C2CCC2)cc1 10562,c1(C(N2C(C(C)NC(c3c(C)nc(C)o3)=O)CCC2)=O)ccc(C)c(Cl)c1 10563,N1(C(c2cccc(C(CC)=O)c2)=O)CCN(C(c2cc(F)ccc2F)=O)C2CC12 10564,N1(C(c2ccc(CC)o2)=O)CCC(O)(CC(=O)NCC(c2ccncc2)C)CC1 10565,C1(OC)COCCC1CC(=O)N(CCCNC(=O)CNC(=O)NC1CC1)CCO 10566,Cn1cc2cccc(-c3cnc(CNCc4cccc(Br)c4O)nc3)c2n1 10567,CN1CCC(C(=O)NCCC2=CCCC2)(NC(=O)CC2CC3CCC2C3)C1 10568,CC(C)CC(CNC(=O)CCOC1CC1)NC(c1ccc(Cl)o1)=O 10569,CCC(C)(C)C(O)C(=O)N1CC(C(=O)NCc2nocc2C)C(C2CC2)C1 10570,C1(C)(CNC(C(=O)NCCOC)=O)CC(OC)CN1C(c1sccc1OC)=O 10571,c1(OC)ccc(F)cc1C(=O)Nc1ncc(CCSC)s1 10572,N1(CC(C)NC(C(COCC)n2cc(-c3csc(C)n3)nn2)=O)CCCNC1=O 10573,N1(C(Cc2ccc(OC)cc2Cl)=O)CC(=O)N2CCCC2C1 10574,N1(CCN(CCN(CC=C)C)C(=O)NC)CCCC(C)(OC)CC1 10575,C1(NC(C2C=CCN(C(c3n(C)c(=O)ccc3)=O)C2)=O)CC2(CCCCC2)C1 10576,c1(C(N2CCN(Cc3ccc(O)cn3)C3CC23)=O)cc(Cl)c(Cl)cc1Cl 10577,CCC(CC)C(C)C(=O)N1CC(C)(CNC(c2c(C)cccc2C)=O)CC1(C)C 10578,N1(C(CCNCc2ccc(-n3ccnc3)c(Br)c2)=O)CC2(CCCN2CC)C1 10579,c1(-n2cc(C3OCCN(C(C4(C#N)CC4)=O)C3)nn2)c(Cl)cc(F)cc1Cl 10580,N1(C(C=Cc2ccc(OC)cc2)=O)C2CCC1CN(C(c1cnncc1C)=O)C2 10581,N1(C(c2c[nH]c(=N)s2)=O)CCCC2C(NC(c3ccc(C4CCC4)cc3)=O)C12 10582,C=CCCCC(C(=O)N1CC(F)C(F)C1)NC(C1CC2CCC2C1)=O 10583,N1(C(c2ccc(Cl)o2)=O)CCCC2(CCC(NC(C3(C4CC4)CCC3)=O)C2)C1 10584,N1(CCCCNC(C(C(C)C)OC)=O)CCCN(C(c2csc(C)c2)=O)CC1 10585,C(=O)(C(C(C)O)N(C)C)NCC1(NC(C2OCC(C(=O)OC)C2)=O)CC1 10586,C1(C(C)C)CN(C(=O)CC2CCOC2(C)C)CCN1C(C1SCCCS1)=O 10587,c1(C(N2C(CCNC(C3(OC)CCC3)=O)CSCC2)=O)cccc2cnccc12 10588,c1(NC(C2N(C(COc3cc(C)on3)=O)CC(C)C2)=O)cc(F)cnc1Cl 10589,Cc1cc(S(C)(=O)=O)cc(C(=O)NC(C)C(C)(C)NC(=O)CC(O)C(C)C)c1C 10590,C1(C(=O)NC2(C)CC(=C)C2)CCCN(C(=O)C(C)c2ccco2)C1 10591,C(=O)(CC(C)C(F)F)N(CCN(C(CC1N(CC)CCC1)=O)C)C(C)C 10592,C1(NC(C=CCCC)=O)CCCC(NC(c2cncc(Cl)c2C)=O)CC1 10593,N1(C(CC)=O)CCOCC(NC(C2C(C)CCN2C(=O)OC(C)(C)C)=O)C1 10594,CN1CCN(C(c2ccc(-c3cnn(C)c3)o2)=O)C(CNC(=O)C2=COCC2)C1 10595,C1(NC(c2cnc(C)nc2)=O)CC12CCN(C(=O)CC(C)CF)CC2 10596,c1(C(N2CCC(NC(CC(C)n3cccn3)=O)C2C)=O)[nH]cc2c1CCCC2 10597,CCCCCC(C)CC(=O)NC(C1(C(=O)NC2CN(C)C(C)(C)C2)CC1)C 10598,CC1CCCC(CC(=O)NCCOC2CN(C(=O)C(C)Cn3ccnc3)C2)C1 10599,c1(C(N(CCNC(=O)C(C)OC)CC)=O)c(Br)nc2n1CCOC2 10600,N1(C(C=Cc2scc(C)n2)=O)CC2(CCN(C(c3cccc4sccc34)=O)C2)C1 10601,c1(C(=O)NC2(CNC(C(CCOC)OC)=O)CCOCC2)ncc(N)nc1C 10602,C1(C(=O)NC(CNC(c2n(CC)nc(C(C)C)c2)=O)C)Cc2ccc(F)cc2O1 10603,C#CC1(C(=O)N(C)CC2CC2(F)F)CCN(C(=O)CS(=O)(=O)CC)CC1 10604,c1(C(=O)NCCC2(NC(c3coc(C(F)(F)F)n3)=O)CC2)ccc2ncnn2c1 10605,CC1C(C)N(C(=O)CC2CCN(CCF)CC2)CCN1C(=O)CC1CCC1 10606,N#Cc1ccccc1OCC(N1CCC(CCNC(c2csnc2Cl)=O)CC1)=O 10607,N1(C(c2c(CC)noc2C)=O)CC(NC(c2cc(F)cc(I)c2)=O)C(F)(F)C1 10608,CC(C)CC(CNC(C12CC(F)(C1)C2)=O)C(=O)NC(C)CS(C)(=O)=O 10609,Cc1cc(C2(C(=O)N(C3CN(C(=O)CC4CCC(C)C4)C3)CCO)CC2)on1 10610,CC1CN(C(=O)CSc2nncs2)CC(C)N(C(C2(O)CCOCC2)=O)C1 10611,N1(C(Cc2cc(C)on2)=O)CC(NC(c2csc(C3CCCO3)n2)=O)CC1CO 10612,N1(C(C(CSC)C)=O)CCCCC(C(=O)NCc2nc(=O)o[nH]2)C1 10613,n1(CC)nc(C)c(C(N2CC(N3CCN(C(c4cnn(C)n4)=O)CC3)C2)=O)c1Cl 10614,c1(OC)cc(CCCOC(=O)C=CC(c2ccc(F)cc2)=O)cc(OC)c1O 10615,C1(C(N2C(C(C)NC(=O)C=C3CCN(C)CC3)CCCC2)=O)CC12CCCCC2 10616,Cc1ccc(S(=O)(=O)N(C2Cc3ccc(Cl)cc3C2)CCO)cc1 10617,c1(C(N2C(CCCNC(C(C)SC(C)C)=O)CCC2)=O)cc2n(c1)CCSC2 10618,Cc1cc(C)c(C(=O)NC2CC2CNC(c2nc(-c3ccco3)sc2C)=O)o1 10619,c1(NC(C)C)nnccc1C(=O)NCC1CN(C(=O)CN2CCC(C)C2)C1 10620,c1(C(=O)NCCC(CNC(c2nsnc2O)=O)OC)cc2ccncc2[nH]1 10621,C1(C(=O)NCC2(O)CCN(C(=O)CN3CCC(CO)CC3)C2)CC12CC(F)(F)C2 10622,N1(C(CC(C)SC)=O)CC(NC(c2cccc(C3(F)CC3)c2)=O)C(C)C1 10623,CC(C)(C)C#CC(=O)N1CCN(C(=O)C(=C2CCCCC2)F)C(C(F)F)C1 10624,C1(C(N2C(CN(C)C(C3CC4C=CC3O4)=O)CCC2)=O)NC(=O)C2CC12 10625,Cc1nc(C2CC2)[nH]c1C(N1CCC(NC(C2SCCC2C)=O)CC1)=O 10626,C1(CC(=O)NC2CC(NC(C3N(CCC)CCCC3)=O)C2)CCC(=O)NC1=O 10627,CCCCC(CNC(C1CC(=O)N(C)C1)=O)NC(=O)CC1COCCO1 10628,CC1(C)CCC(C(=O)NCC2(C)CC2(F)F)CN1C(C1CCC(=O)O1)=O 10629,C1(NC(=O)COc2cccc(F)c2)CN(C(C2(C(F)F)CCC2)=O)CCC1F 10630,Cc1ccc(CNC(=O)C=CCC2(NC(=O)C(C)CC#N)CCC2)cn1 10631,c1(C(=O)NC(c2cccnc2)CN(C)C)c[nH]nc1C1CCOCC1 10632,N1(Cc2n(CC)nnn2)CC(OC)C(NC(C)=O)C1 10633,C1(NC(CCSCCC)=O)CCC(N(C)C(c2coc(O)n2)=O)C1 10634,C(=O)(CCCCC(N)=O)N1C(CC(N2CCCC(C)C2)=O)C(C)(C)CC1 10635,c1(C(C(=O)NC(CC(C)NC(C(Br)=C(C)C)=O)C)O)cccc(C)c1 10636,C1(C2CCN(C(C3CCC4(CC4)C3)=O)C2)(NC(c2cn(C)c(=O)cc2)=O)CC1 10637,c1(CN(CC)CC)cc(CNCCOCC(=O)NC(CCOC)=O)no1 10638,c1(C(N2CC(F)(CNC(C3CC(C)OC3)=O)C2)=O)cc2c(s1)CCC2=O 10639,c1(C(=O)NC2(CC(=O)NCCC34CC(CO3)C4)CCCC2)ccc(Cl)cc1O 10640,C1(C2CN(C(C34CCCC3C4)=O)C2)(NC(CCCn2c(C)ncc2)=O)CC1 10641,C(=O)(C(CC)CC(C)C)NCc1cc(C(=O)NC(CCC(=C)C)C)on1 10642,c1(C(N2CCN(C)C(=O)C2)=O)nn2ccccc2c1C(=O)NC1CCCC(O)C1 10643,C(=O)(CC(CCCC)NC(C1CC(CC)=NO1)=O)N(CCC#C)CC 10644,C1(NC(CC=CCC)=O)COC2CN(C(C3CCCCC3)=O)CC12 10645,CCCCC(C)C(=O)N1CC(C(C)NC(=O)C(c2cnn(C)c2)O)C1 10646,Cc1ncnc(C(=O)NC(C)(C)CC(N2CCOC(C)CC2)=O)c1C 10647,c1(C(N2CCN(CCNC(C(CC)(C)CC)=O)CC2)=O)cnn2c1CN(C)CC2 10648,C1(C(N(CCNC(C(C)OCCC=C)=O)CCC)=O)CC=CC(O)C1 10649,c1(C(=O)NCC(CNC(C(C)=C(C)C)=O)O)oc(-c2ccccc2)nc1C 10650,Cc1nc(C)c(CC(=O)NCC2CCCCN2C(=O)COc2cn[nH]c2)c(O)n1 10651,C(=O)CCC1=NNC(=O)CC1.C(=O)(CC(C(F)F)n1cccn1)N(C1(C)CCC1)CC 10652,N(C(=NCCN(S(C)(=O)=O)C)NCc1ccsc1C)Cc1cccc(C)c1 10653,c1(CC(C(=O)NCC(=C)CCNC(c2oncc2CC)=O)C)ccc(Cl)c(Cl)c1 10654,Cc1ccc(O)c(CNC(=O)CC2CCCN(C(=O)CC#N)C2)c1 10655,c1(C(=O)NCc2c(C(NOCC#C)=O)n(C)nc2)cc(C#N)ccc1C 10656,C1(C(=O)NC2CC(NC(c3cnc(SC)n3C)=O)CC2O)CCCCN1N=O 10657,c1(-c2nc(CSCCNC(CCc3ccnc(C)n3)=O)sc2)c(Cl)cccc1Cl 10658,CC1CN(C(C2CCN(C3CC3)C2=O)=O)CCN1C(c1cnc(N(C)C)cn1)=O 10659,C1(CNC(CCC#CC)=O)CC2(CC(NC(=O)C(c3cn(C)nc3C)C)C2)C1 10660,c1(C(=O)NCCCC(C)NC(Cc2cn(C(C)C)nc2)=O)cc2sccc2s1 10661,N1(C(c2c(C(C)(C)C)n[nH]c2)=O)C2CCC1CC(NC(C1CC3(CCC3)C1)=O)C2 10662,n1(CC(=O)N(CCNC(=O)C(c2ccc(C)cc2)C)CC)cnc2ccccc12 10663,c1(C(=O)NCC2CN(C(c3ccc(C)s3)=O)C2)ccc(Br)c2cn[nH]c12 10664,Cc1ccc(C)c(C(N2CC(F)(C(=O)NC(C)Cn3cc(C)cn3)C2)=O)c1 10665,C(=O)(C(CC)CC(C)C)NCCNC(c1cn(CC(OCC)OC)nc1)=O 10666,c1(C(n2cc(C3CCN(C(C4(CO)CC4)=O)C3)nn2)C)ccc2ccccc2c1 10667,C1(C(N2CCCC2CNC(C23CC4CC(CC2C4)C3)=O)=O)CCOC2(CCC2)C1 10668,c1(C(=O)NC2CCN(C(C(N3CCSCC3)C)=O)C2)nnn2c1CCCC2 10669,c1(C(N2CC3CC3C3CC23)C(=O)NCCCOC)ccc2c(c1)COC2 10670,c1(C(N(C2CC(NC(=O)C(=O)C(C)(C)C)C2)C)=O)cc(F)cc2ccoc12 10671,N1(C(C2C(OCC)C2)=O)C(CO)CSCC1c1ccccc1 10672,c1(C(N2C3CC(NC(CCCC)=O)C2CC3)=O)c(OC)cnc2ccccc12 10673,c1(CNC(C(C2(O)CCC2)NC(c2cccnc2S)=O)=O)ccc(CO)nc1 10674,C(=O)(CCCCC(=O)NC1CCN(Cc2nc(C(C)OC)no2)CC1C)NC 10675,c1(OCC)cccc(CC(=O)NC2CCCC2)c1.C1(CN(C)C)(NC=O)CC1 10676,C1(C(=O)NC(CCC)C2CCCC2)CCC(C)(C)N(C(=O)C(F)C2CCCC2)C1 10677,C12(NC(c3cc(C)c(C)o3)=O)COCCC1CN(C(=O)Cc1[nH]cnc1C)C2 10678,c1(C(N2CCC(Cc3ccccc3Br)C2)=O)ccnc2ncnn12 10679,C=CCC(C)(C)C(=O)N1CCN(C(=O)C(C2CC2)SC)C(C2CC2)C1 10680,N1(C(CSCCC)=O)CCC(CO)(NC(=O)CCCCCN(C)C)CC1 10681,CCC(C)(C#N)C(=O)N1CC2(NC(c3cc(-c4ccccc4)c[nH]3)=O)CC1C2 10682,c1(C(=O)NC(CCCC)CNC(=O)CCCCCO)ccc2c(c1)COC2 10683,Cc1oc(C(=O)NC2C3CC2N(C(=O)CCCN(C)C)C3)cc1S(C)(=O)=O 10684,N1(C(C(c2ccccc2)C)=O)CCC2(C1)CN(C(C1(F)CCCOC1)=O)C2 10685,C1(C(NOCC#C)=O)CCC(CNC(=O)CCc2cccs2)C1 10686,N1(C(Cc2c(C)ccs2)=O)CCCC2CN(C(=O)C=Cc3ccccc3)CCC12 10687,C12(NC(C3N(C(C)=O)CC(O)C3)=O)CCN(C(c3ccc(CO)nc3)=O)CC1C2 10688,c1(C(=O)NCC2(CCNC(C(C)(C)OCC)=O)CC2)cc(C#N)no1 10689,c1(CNC(C2CCCCS2)=O)ccccc1-n1cc(CN2CCCC2=O)nn1 10690,C1(n2cc(C(CCC)C)nn2)CON(C(=O)C(C)C(F)F)C1 10691,C1(C(N(C2CN(C(=O)OC)C2)C)=O)CCN(C(=O)CCc2ccc(Cl)cc2)CC1O 10692,c1(C(=O)NCC(C)N(C(=O)CC(O)C2CCCC2)C)cc(-c2ccccc2)no1 10693,Cc1oc([N+](=O)[O-])cc1C(=O)N(C1CCN(C(C2CC(F)C(=O)N2)=O)C1)CCO 10694,N1(C(=O)CCc2nc[nH]n2)C2CCC1C(F)C(NC(C1(CCNC=O)CC1)=O)C2 10695,N1(C(Cn2cc(C(=O)OC)nn2)=O)CCCC2(CCN(C(=O)C(C)C3CC3)C2)C1 10696,C(=O)(N=c1[nH]c(Cl)ncc1O)C1C2(CN(C(c3c(OC)csc3)=O)C2)C1 10697,C(=O)(C(O)C(F)F)N(CCN(C(C)C)C(c1ccc(NC(C)C)nc1)=O)C 10698,c1(OCC)cnc(C(=O)NCC2CC3CC3N2C(=O)C(C)(O)CC)cn1 10699,C1(C(=O)NC(c2nc[nH]n2)CC)CN(C)CCN1C(=O)CC(C)(C)C#N 10700,CCCCCC(O)C(=O)NCC1CCN(C(c2coc(C)n2)=O)CC1O 10701,C=CCCC(C(=O)N1CC(C)(C)C1COC)NC(C1(C)CCC2CC2C1)=O 10702,c1(C(=O)NCC(C)(C)NC(C2C(=C)CC2)=O)cc2ccc(Cl)cc2o1 10703,C1(NC(c2cc(C(F)F)ccn2)=O)CCN(C(C2C(Cl)(Cl)C23CC3)=O)CC1F 10704,c1(SC)nc(NCC2CCN(C(c3cnc(C(F)(F)F)s3)=O)C2)ncc1C 10705,N1(C(c2cncc(C)n2)=O)CCC2CC(C1)CN(C(C1CC1c1ccsc1)=O)C2 10706,Cc1onc(C(=O)NCC2CCCC(NC(C3CC=CC3)=O)C2)c1[N+](=O)[O-] 10707,Cc1ccc(C)c(CNC(c2nnnn2CCOCC2CC2)C23CCCC2C3)n1 10708,CN1CCCC(C)(C(=O)N(C)CC2(O)CCN(C(=O)CCc3cncs3)C2)C1 10709,C(=O)(CCN=C(NCc1nncs1)NC1CCCN(CC(F)(F)F)C1)N(C)C 10710,OCC(Cc1cccc(F)c1)CN=c1[nH]c2c(F)c(F)c(F)cc2s1 10711,c1(C(=O)NC2CC3CN(C(C(CC)OC)=O)C2C3)nccn2ccnc12 10712,N1(C(C(Cn2cccn2)NC(CC2(C)CC2)=O)=O)CCCC(F)(F)CC1 10713,N(C(=NCCCCl)NCCCN1CCCC1=O)C(C1CCOCC1)C#C 10714,c1(OC)cc([N+](=O)[O-])ccc1CNC(=O)C=Cc1ccc(Cl)cc1F 10715,C(=O)(C(C)(C)CC#N)N1C(CN(C(=O)Cc2cnc[nH]2)C)COCC1 10716,C1(OC)(CNC(=O)CC2CCC2)CCN(C(=O)CC(N2CCCS2(=O)=O)C)C1 10717,CS(=O)c1ccccc1-c1cnc(CNCc2ccccc2C(F)(F)F)nc1 10718,c1(OC)ncccc1NC(c1cc(CCNC(C2CCC2C(C)(C)C)=O)on1)=O 10719,C1(NC(N(C)CCc2ccncc2)=O)CCN2CCCCC12 10720,c1(C(N2CCC(NC(c3cncnc3)=O)CC2C2CC2)=O)cc([N+](=O)[O-])ccn1 10721,C=C1CC2(C1)CC(C(=O)NC1CCN(C(=O)C=Cc3cncs3)CC1C)C2 10722,C(=O)(C(C)(C)C1CCCN1C(=O)C(C1CCOCC1)O)NCC1CC(OCC)C1 10723,C1(OC)CCN(CC(O)COc2ccc(-n3cccn3)c(C)c2)C(C)C1 10724,C1(C(N(CCSC)CC)=O)CN(C)CCN1C(=O)Cc1cn(CC)nn1 10725,C1(O)(CCNC(C(CC)OCC)=O)CCN(C(c2cnccc2Br)=O)C1 10726,c1(C(N2C3CC(CC(NC(c4n(C)ccc4)=O)C3)C2)=O)coc2cc(O)ccc12 10727,CC1CN(C(C2(O)CCSCC2)=O)CCC1CNC(c1cnc[nH]c1=N)=O 10728,C(=O)(C1CCCc2ccnn21)N1CC(C2CN(C(CS(C)(=O)=O)=O)C2)C1 10729,Cc1nnc(CCC(N2CCCC(CNC(C3CCN3C(C)(C)C)=O)C2)=O)n1C 10730,C(=O)(C1=C(F)CN(C(C2CCCC(=O)C2)=O)CC1)NC(c1csnn1)C 10731,C1(NC(CCN(CCC)C)=O)CC2CC1CN(C(c1ccnn1CC1CC1)=O)C2 10732,C(=O)(CCCC(C)(C)C)NCC(CC=C)NC(c1coc(C)c1)=O 10733,C#Cc1cn(C)nc1C(=O)NC1CCC(CC(N2CCCC2C)=O)C1 10734,CC1(F)CCCCN(C(c2ccc(C(F)F)cc2)C(=O)NC2CCOCC2)C1 10735,C#CCCCCC(=O)NC1CCCC(NC(c2ccn(C)c(=O)c2)=O)C1 10736,N1(C(C2N(C(CC(=O)OC)=O)CCC2C)=O)CC2CSCC(C2)C1 10737,N1(C(C2C(CC)C2)=O)CCCC2(C1)CN(C(c1ccc(N)cc1F)=O)C2 10738,c1(C(=O)NCC2C(CNC(CSc3cn(C)nc3)=O)C2)ccnc(Cl)n1 10739,Cc1cnn(CCCNC(=O)C=CC(C)NC(=O)CCCC2CC2C)c1 10740,CCC(C)CC(=O)NC1CCCC1C(=O)Nc1ccc(NC(C)=O)cc1 10741,C(=O)(C(O)CCC(F)(F)F)N1CC(CNC(c2c(C)cccn2)=O)N(C)CC1 10742,CCC(CC)(C(=O)NC(C)C(C)NC(=O)Cn1ccc(C(F)F)n1)C(C)C 10743,C1(C)(COC)CC(NC(=O)CC2CC2)CN1C(=O)Cn1cnc([N+](=O)[O-])n1 10744,CC1OC2(CO)CC1(C(=O)NC(C)CN(C)C(c1cc(C3CCCC3)no1)=O)C2 10745,C(CCN=c1[nH]c(=NCCC(C)F)[nH]c2c1COCC2)N(C(C)=O)C 10746,CCCC(CC)C(=O)N1CC(NC(c2cc(Cl)cc(Cl)c2)=O)CC(F)C1 10747,c1(C(=O)OC(c2cn(C)nn2)c2ccccc2)ccc2ccnc(Cl)c2n1 10748,c1(C(N2C(CNC(c3cc(CCC)on3)=O)C=CC2)=O)n[nH]c2c1COC2 10749,N1(C(C(C(C)C)F)=O)CCCN(C(=O)CN2CCC(C(N)=O)CC2)C(C(C)C)C1 10750,C(CC(C)C)(C(=O)N1CC2(C1)CN(C(=O)Cc1cscc1Br)C2)OC 10751,CCC(O)C(C)C(=O)NCC1CCCN1C(=O)CN1CCCC(C(=O)OC)C1=O 10752,C(=O)(C1=COCCO1)NCC(C(C)(C)C)NC(c1c(Cl)cncc1Cl)=O 10753,C1(N(C(CCC=C)=O)C)CCN(C(=O)C(c2ccc(F)cc2)CO)CC1 10754,N1(C(Cn2c(C)cc(C)n2)=O)C2CCC1C(NC(=O)Cc1ccsc1)C2 10755,N1(C(c2c(CC)[nH]cc2)=O)CC2CC(C1)N(C(C1CCCN(CC(C)C)C1)=O)C2 10756,C12(C(=O)NCCC3OCCN(C(C(CCSC)O)=O)C3)CCC(CC1)C2(C)C 10757,Cc1ccc(C(=O)NC2CN(C(c3ccn(C4CC4)n3)=O)CC2C)cc1F 10758,C1(CC(=O)OC(C)(C)C)(NC2CC3CC3C2)CCOCC1 10759,N1(C(C2(OC)CC(c3cn(CCC(=O)OC)nn3)C2)=O)CC2COCC2(C)C1 10760,C(CC(=O)N(C(C)(C)CO)C(C)C)(C(F)F)NC(CSCC=C)=O 10761,c1(C(C)SCC(=O)N(C(CNC(CCC(=C)C)=O)C)C)nc2ccccc2[nH]1 10762,C1(OC(C)=O)CCc2nn[nH]c2C1.C(C1CNC1=O)OC.C1(=O)C(C)(C)CN1C 10763,C1(NC(=O)NCCS(=O)(=O)NC2CCCC2)CCCC1C1CCCC1 10764,c1(N2CC3C(CNC(C(C)Cc4ccco4)=O)C3C2)ncnc(Cl)c1Br 10765,C1(NC(C(F)=C(C)C)=O)CC2CCC1C1CN(C(=O)C=CC3CCCC3)CC21 10766,N1(C(C2N(C(c3nc(C)sc3)=O)CCC(C)C2)=O)CCCC(O)(C2CC2)C1 10767,C(c1ccc(C)cc1C)=CC(=O)NCC1N(C(C=C(C)C(C)C)=O)CC=C1 10768,N1(C(c2n(CC)cc(Cl)c2)=O)CCCN(C(=O)C(O)CC(F)(F)F)C(C)C1 10769,c1(C(=O)NCC2C(C)CCN2C(c2nnsc2SC)=O)ccc(OCF)cc1F 10770,C#Cc1ccc(C(N2CCN(C3CN(C(C4CC(F)C(=O)N4)=O)C3)CC2)=O)cn1 10771,Cc1cc(=O)n(CCCN2CCCC(N(CC(=O)O)C)CC2)cn1 10772,C1(NC(c2ccn(CCCC)n2)=O)CC(O)CN(C(c2ccc(CF)cc2)=O)C1 10773,N1(C(CCOC)=O)C2CC=C(C(=O)NC(c3cc(C)on3)C)C1CC2 10774,c1(CCC(=O)NC(CC(C)C)CNC(c2sccc2F)=O)c(F)cccc1F 10775,C(C(CC(C)C)C(=O)NC1CC2(C(=O)NCCCCS(C)=O)COC1C2)OC 10776,S(=O)(=O)(c1ccc(N2CCOC(C)(C(C)(C)C)C2)c(Cl)c1)N(C)CC1CC1(C)C 10777,S(=O)(=O)(c1cc(C)c(OC)cc1Br)N1C(CC)CNC(=O)C1 10778,C1(CC)COCCN(C(=O)C(=O)NCCn2cc(C(C)(C)N(C)C)nn2)C1 10779,c1(C(N2CC(NC(C3(SC)CC3)=O)C(F)C2)=O)ccc2nc(O)[nH]c2n1 10780,C(CCN=c1[nH]c2c(c(=NCCN3CCOCC3C)[nH]1)COC2)OCC(C)C 10781,c1(CC)noc(C)c1N(C)C(N1CCC(C2CCCCN2C(=O)C2CC2)C1)=O 10782,Cc1nc(C(=O)NCCC(C)NC(C2CC2C)=O)c2n1CCCC2 10783,N1(C(CCCOCC=C)=O)CCN(C(=O)C(O)CC)C(CC(=O)NCC)C1 10784,C1(N(C(=O)CCCc2cccc(Cl)n2)C)CN(C(=O)CC(F)(F)Cl)CC12CC2 10785,N1(C(C=C(CCC)C)=O)CCCC(C)(CNC(=O)CCc2cc(O)ccc2C)C1 10786,c1(C(=O)NCC(C)CNC(C23CC(C(F)F)(CO2)C3)=O)ncc2ccccn12 10787,C1(CC(=O)N(CCC(C(C)C)Nc2nccnc2C#N)C)CCCC2(CCC2)O1 10788,CCCCC(O)C(=O)NCc1cc(C(=O)NC2CCN(CC)CC2)on1 10789,N1(C(C(C)(C)NC(=O)NCC)=O)CCCC(CNC(=O)C(C)c2ccsc2)CC1 10790,c1(CC)c(C(N2CCC(NC(=O)COCC(F)(F)F)C(F)C2)=O)cccc1F 10791,c1(C(N(CCCNC(CC(CC)C)=O)CCO)=O)ncnc2cc[nH]c12 10792,S(=O)(=O)(c1ccc(=NCCc2ccc(OC)nc2)[nH]c1)N(CCOC)CC 10793,Cc1cnc(C(N2CCC(NC(C3CCS3(=O)=O)=O)C23CC3)=O)c(C)c1 10794,CC1=NNC(=O)C1CC(=O)NC(CNC(=O)C(C)N1CC(C)C1)C(C)(C)C 10795,c1(C(=O)NCC(C)NC(c2cccc(C(C)=O)c2)=O)cccc2c(C)cccc12 10796,C(C1CN(C(c2cc(C)c(O)nn2)=O)CC1C(=O)NCCC(O)C1CCC1)=CC 10797,c1(COC)ccc(C(=O)OC)cc1F.C1C(CO)NC(=O)CC2CC2NC(=O)N1 10798,c1(CC)noc(COCC(=O)N(C(C)(C)CNC(C)=O)C2CCC2)n1 10799,C=CC1(CO)CCN(C(=O)CCC(CC)NC(c2ccc(N)c(F)n2)=O)CC1 10800,C=CC(C)(C)CC(=O)NC(C1CCN(C(=O)CCS(C)=O)C1)(C)C 10801,C1(CC(=O)NCC(CC)NC(c2cccc(C(N)=O)c2C)=O)CCS(=O)(=O)CC1 10802,c1(C(=O)NCCC(C)N(C(CN2C(C)CC2)=O)C)nn(C)cc1N 10803,C1(CC)CCN(C(=O)CC(C)(C)O)C1CNC(c1cc(C)ncn1)=O 10804,C1(CN(C)C(C2(O)CCSCC2)=O)CC(F)CN1C(c1ccc(C(F)F)o1)=O 10805,c1(COC(c2ccc(OC3CCOCC3)cc2)=O)cc2c(s1)CCOC2 10806,C1(OC)CN(C(=NCCCCl)NCc2ccc(CSC)cc2)CC1O 10807,Cc1c(C(F)(F)F)n[nH]c1C(N1CC(CNC(c2cccc(N)n2)=O)CC1C)=O 10808,c1(C(=O)NC(c2cccc(C)c2)CNC(C(C)(C)SC)=O)nc(Cl)ccc1N 10809,FC(F)C(F)(F)CCN=c1[nH]c(N2CCOCC2)nc(=NCCc2cnn[nH]2)[nH]1 10810,c1(N(CC(N2CCC(C)(NC(CC(CC)(F)F)=O)C2)=O)C)ccc(Cl)cc1C#N 10811,C1(CNC(=O)CCCn2ccnn2)CC2(CC2)CN1C(=O)COCC1CCC1 10812,C1(C(C)C)C(NC(c2cnn(C)c2N(C)C)=O)CCN1C(c1cnn[nH]1)=O 10813,C(=O)(C1=CCCC1C)NCC(C1CCN(C(c2n(CC)c(O)nc2)=O)CC1)C 10814,C1(C(=O)NC2C(CNC(c3n(CC)ncc3Cl)=O)CCCC2)Cc2nccn2C1 10815,C(=O)(CC(C)CC(C)(C)C)N1CC(NC(c2c(C)ccc(C)c2)=O)C(F)C1 10816,c1(C(C(=O)NC2CCCN(C(C(CC)CC)=O)C2)C)c(F)cccc1F 10817,c1(N2CC3(C(C(=O)Nc4c(C)ccc(I)c4)C3)C2)ncnc2c(C)csc12 10818,S(=O)(=O)(c1ccc(Cl)cc1)CC(=O)NC(C)CCNC(=O)C(C)OC(C)(C)C 10819,C(=O)(CCN(OC)C(=O)c1coc2c1COC2)N1CC(COC)(OC)C1 10820,c1(CNC2C(C)CNCC2)nc(N(C)C)n(-c2ccccc2)c1Cl 10821,c12csc(n1)CNC2C.C1(CC(=O)OCC)(CC)CNC1 10822,C12CC(c3ccccc3)(C1)NC(=O)C(=O)N2.C(=O)(CC(C)C1CCCO1)OCC 10823,c1(CN2CCCC(C)(C(=O)NC3CNC(=O)C3)C2)ccc(F)c2ccoc12 10824,Cc1cccc(OCC(=O)Nc2ccccc2CNC(=O)CC(C)(C)C#N)c1C 10825,c1(OC)c(Cl)ccc(C(=O)NCCC2CCC(NC(=O)C(O)CSC)C2)c1F 10826,c1(C(=O)NCC(C)CNC(c2cnoc2C2CCC2)=O)cc(F)cc2nn[nH]c12 10827,c1(C(=O)NCCC(C)NC(=O)C(F)(F)c2csc(Cl)c2)cn(C)nc1Cl 10828,Cc1c(C(=O)NC(C2(O)CN(C(=O)CC(=O)N(C)C)C2)C)cnn1C1CC1 10829,C1(C)(C(=O)NCC(n2cc(-c3ccc(COC)cc3)nn2)C)COC(=O)OC1 10830,CC(C)(C)C(=O)N1CCCC1C(=O)N(CCC=CBr)CC1CC1 10831,C(CC(C(=O)NCc1cc(C)c(C)s1)NC(C1CC(F)C1)=O)=CC 10832,N1(C(=O)NCC2(CC(F)F)CCCO2)CCC(C2(O)COC2)CC1 10833,C1(CNCCc2cc(OC(=O)Nc3ccccc3)ns2)CN(OC)CCN1 10834,C1(CNC(CCCOC(C)C)=O)CC(C)(C)CN1C(=O)CC1(O)CCCOC1 10835,C1(SC)CN(C(=O)COC2CCC2)CC1NC(=O)C(O)Cc1[nH]cnc1C 10836,N1(C(c2csc(Br)n2)C(=O)NCC(=C)C)CCC(CO)(COC)C1 10837,C1(NC(CC=CCC)=O)CC(O)CN(C(=O)C(=O)Nc2ccccc2)C1 10838,N(C1CCSc2ccc(F)cc21)C(c1cc(OC)sc1Cl)=O 10839,c12ccc(c(O)c1)C(=O)NC1(CC)CCC(CC1)NC2=O.C1(CC)(COC)CC1 10840,CCCCC(C)CCC(=O)N(C1CC(C(=O)NCC(CC)SC)C1)C 10841,c1(C(N(C)CC2N(C(C(C)C3CCOC3)=O)CCC2)=O)cc([N+](=O)[O-])sn1 10842,CC1CC2(CC(C(=O)N(C(C)(C)CC(=O)N3CC(c4ncccn4)C3)C)C2)C1 10843,CC1CCN(C(c2cc(Cl)cs2)=O)CCN1C(=O)CC1OCCCC1(C)C 10844,C1(CNC(C2CC2CF)=O)CN(C(=O)Cn2ccnc2)CC12CC2 10845,CC(C)(CCC#N)C(=O)NCCOCCNC(=O)CC1CCC2CC12 10846,Cc1ccc(S)cc1.C12(C=O)CCC1CC2.n12cc(nn1)C1CC(C1)NC(=O)C2 10847,N#Cc1ccc(CSCC(=O)N(c2ncc[nH]2)CC(F)(F)F)cc1 10848,C1(NC(C=CS(CC)(=O)=O)=O)CCC2CCN(C(C3CC3(Cl)Cl)=O)C1C2 10849,C1(N(CCC)C(c2cc(C)co2)=O)CCN(C(=O)CSCC2CCCCO2)CC1 10850,C1(C(N2CC(C(C)OC)C2)=O)CC(C)(C)CCN1C(c1cccc(C)n1)=O 10851,Nc1c(C(=O)NC2CC(CCNC(=O)CN3CCCC3CO)C2)cc(F)cc1Cl 10852,c1(CC(C(=O)C(C(N2CCSCC2)C)=O)O)ccc(F)cc1.C1(N)CC(N)C1 10853,c1(NC(CCC2N(Cc3cn(C)nn3)CCC2)=O)ccc(S(N)(=O)=O)cc1 10854,c1(OC)cc(C)cc(C(=O)NCC=CCNC(c2cnc(C)nc2SC)=O)c1N 10855,C(=O)(C(C)(C)C(F)(F)F)NC1CN(C(c2noc(CC)c2C)=O)C(CC)(CC)C1 10856,Cc1cc(C(=O)NC(C)(CNC(C2CC2C(N)=O)=O)C(C)C)cc(C)c1C 10857,Cc1cc(C(=O)NCC2(CNC(=O)CC3COC(=O)C3)CCC2)n(CC(F)F)n1 10858,N1(C(C(CC)=CC)=O)CCC(C)C(NC(c2cc(Cl)cc(Cl)n2)=O)C1 10859,C1(CC(=O)OC)CC(C)(C)CN1C(=O)NC(C1(n2cccn2)CC1)C1CC1 10860,C1(NC(CCNC(N)=O)=O)CCCCC1NC(C1(CO)CC(F)(F)C1)=O 10861,C(=O)(C(=O)N1CCC(C(N2CCNC(=O)C2C(C)C)=O)O1)NCC 10862,C1(N(C)C(c2ncoc2C2CC2)=O)CCCC(NC(=O)C=Cc2cncn2C)C1 10863,c1(C(=O)NC2CC3CCC(C2)N3C(=O)Cc2ccoc2)nncc2c1CCCC2 10864,C1(C(N(C2CC3(CC3)C2)C)=O)CC2CC1CN(C(C1CC1C1(C)COC1)=O)C2 10865,C1(C(=O)OC)CCC2(CCC2)N(C(=O)CCC2CCOC2=O)C1 10866,CC1CN(C(=O)COCC2CC2)CC(C)N(C(c2ccc(-c3cccs3)s2)=O)C1 10867,C1(NC(C2CC(NC(C(C(C)C)O)=O)C2)=O)CC(C)CCC1O 10868,c1(CC)nc(N2CCC(NC(c3cnn(C(F)F)c3)=O)CC2C)c2ccsc2n1 10869,C(=O)(CS(=O)C(F)(F)F)N1CCC(CNC(CCOC)=O)C1(C)C 10870,Cc1cc(OCC(=O)NC2CC(NC(C3CCOC(=O)CC3)=O)C2)ccc1Cl 10871,C(=O)(CCC[N+](=O)[O-])N1CCC(C)(CNC(C(Cc2c(C)noc2C)C)=O)C1 10872,C1(CC(=O)NC(C(=O)NCC(C)C)c2cn[nH]c2)CC2C=CC1C2 10873,Cc1nn(C)c2c(NC3CCCCC3C)nc(=NCC3(C)NC(=O)NC3=O)[nH]c12 10874,C(N=c1[nH]c(N(C)CCOC(F)F)nc2ccccc12)c1cc2ncn(C)c2cc1 10875,c1(CN=[N+]=[N-])ccc2c(c1)CCO2.C(=O)C(C)(O)C(F)(F)F.CC(C)C1CC(=O)N1 10876,C1(NC(C(C)NC(=O)NCC)=O)C=CCN(C(c2cc(OCC)n[nH]2)=O)C1 10877,C1(n2cc(CNC(C(C)=C(C)C)=O)nn2)CCN(C(=O)CCc2cccs2)CC1 10878,C1(CNC(C2(OCC)CCCC2)=O)CN(C(c2c(C(C)C)n[nH]c2C)=O)CC1C 10879,c1(CC(N2C(CNC(C(C(C)C)(C)O)=O)COCC2)=O)cccc2c1OCCO2 10880,N1(C(CN(C(C)=O)C)=O)CCC(C2N(C(=O)CC3CC3(C)C)CC2(C)C)CC1 10881,N1(C(C(c2c(C)n[nH]c2C)C)=O)CCCN(C(c2cnns2)=O)C(C)C1 10882,C1(C(N2CC(CNC(=O)CSC)C(C(F)(F)F)C2)=O)(COC)CC=CCC1 10883,c1(OC)cc(CCC(=O)NC(C)CN(C)C(c2cc(C(F)(F)F)cs2)=O)on1 10884,Cc1ccsc1C(N1CCC1)=O.n1(Cc2ccccc2)cc(C(C)(C)N(C)C)nn1 10885,C12(C(=O)NC3CC(C)N(C(=O)CCC4CCCC4)C3)CC(C)(CCO1)C2 10886,CCC(C)CCC(=O)NCC1COCCN1C(c1cnc(-c2ccccc2)[nH]1)=O 10887,C1(C)(CNC(C(=O)NC(C)C)=O)CCC(NC(=O)C(c2ccccc2)=O)C1 10888,c1(CC(=O)NCCCCN(C(c2ccc(C#C)cn2)=O)C)cn2cc(C)sc2n1 10889,C1(C(C2CC2)NC(CCN(CC(F)(F)F)C)=O)CCN(C(=O)OC(C)(C)C)C1 10890,Cc1cccc(CCN(CCCNC(c2ccc(C3CCCCC3)cc2)=O)C)c1 10891,C(CCCCC(=O)NCCc1cnc(C)s1)NC(C1(OC)CCC1)=O 10892,N1(C(C(C(C)C)F)=O)CC2CCCC(Nc3cc(-n4ccnc4)ncn3)C2C1 10893,CC(C)CC(C)(C)C(=O)NCC(C)N(C(=O)Cc1cc(F)c(N)cc1F)C 10894,c1(CNC(N2CCN(CC(=O)Nc3ccccc3)CC2)=O)cnc(Cl)c(Cl)c1 10895,CCC(F)(F)CC(=O)N1C2CCC(C2)C1CNC(=O)C(C)Oc1ccccc1 10896,C1(C(N2CCC(NC(c3n(C)nnc3)=O)(CO)C2)=O)CCc2nccn2CC1 10897,c1(C(=O)NCC(N(C(C=C(CC)CC)=O)C)C2CC2)cc(F)ccc1Br 10898,c1(SC(C(=O)NCC2CC(NC(C(c3cnccn3)C)=O)C2)C)ccccn1 10899,C1(O)(CC(=O)N(CCC(N2CC(C)(CO)C2)=O)C)CCOCC1 10900,c1(OCC)ncccc1NC(C1CC(O)(CNC(=O)CN(C)CC)C1)=O 10901,Cc1ccc(C(=O)NCCOC(C)(C)CNC(c2nccnc2C)=O)c(Cl)c1 10902,c1(C(=O)NCCCN(CCO)C(C2CCCSC2)=O)ccc2nn[nH]c2n1 10903,N1(C(CC(C)F)=O)CCC(C)(C)CC1C(=O)NCc1cncc(C#N)c1 10904,C(c1ccccc1Cl)=C(C)C(=O)NC1CC(C)N(C(=O)CCn2ccc(=N)[nH]2)C1 10905,c1(C2(C(=O)NC3C=CC(CNC(=O)Cn4nccn4)C3)CC2)cc(F)cc(Cl)c1 10906,S(=O)(=O)(c1cc2c(Br)cncc2s1)NCCC1CCN(C(C)=O)CC1 10907,C1(C)(CC)CC(NC(=O)NC(C2(CC(=O)OC)CCOCC2)C)CCO1 10908,C12CCN(CC1)C2=O.C1(NC(CSCc2nnc(C)s2)=O)CC12CC(O)C2 10909,c12cnc(c(Cl)c1)N(CCCNC(CC)=O)C2.c1(C(=O)OC)cc(OC)ccn1 10910,c1(OC)cnccc1-c1noc(C2(C3CC3)CC2)n1 10911,C(=O)(CCCCC(=O)N1CC(CNC(=O)CN2CCCCC2)CC1C)OC 10912,c1(C(=O)NCC(CCC)NC(=O)CCN(C)CC)c(C)coc1CC 10913,c1(CN(CCOC)C(=O)NCc2cncs2)ccc(F)cc1Br 10914,CC(C)C(C(=O)NCCC(C)N(C)C(C1CCC(=O)C1)=O)N(C)C 10915,N(C1COc2ccc(Cl)cc21)C1(c2n(CCSC)nnn2)CCN(OC)CC1 10916,c1(N2CC3CC(NC(CC4(OC)CCC4)=O)C3C2)nc(C)nc2scc(C)c12 10917,c1(C(N2C(CC)CN(C(c3cc(Cl)n(C)n3)=O)CC2)=O)cccc2ccncc12 10918,c1(CN2CC3C(C(=O)Nc4nc(O)cs4)C3C2)cccc(I)c1F 10919,C1(C(N2C(CNC(CN(C)CC)=O)CCCC2)=O)CNC(=O)CC12CCOC2 10920,N1(C(c2cnn(C)n2)=O)CCCC(CCC(N2CCCC2C(C)(C)CO)=O)CC1 10921,c1(OC)ccc(C(=O)O)cc1CN1CCC(O)C(C(=O)Nc2nc(C)ccc2F)C1 10922,C12(CNC(c3n(CC)ncc3)=O)CC1CN(C(C1CC(C)(O)C1)=O)C2 10923,c1(NC(c2cc(-c3c(OCC)cc(F)cc3)ncc2)=O)cc(Br)cc2[nH]ccc12 10924,Cc1nc2ccc(C(N3CCC4CN(S(=O)(=O)c5nccs5)CCC34)=O)cc2o1 10925,CCC(C)(COC)C(=O)NC1CC2(C1)CN(C(c1csc(Cl)c1)=O)C2 10926,N1(C(c2cncc(NCC)c2)=O)CCC(NC(C2(CCCF)CC2)=O)C(CO)C1 10927,C1(CC)(CO)CCN(C(c2cccc(C(C)(C)C)n2)C(=O)NC2CCC2)C1 10928,c1(C(C)(C)C)ncc(C(=O)NCCC2CCN(C(c3cn(C4CC4)cn3)=O)C2)o1 10929,N1(C(c2c(C)nccc2Cl)=O)CCCC(NC(=O)C=Cc2ccsc2)C(F)C1 10930,N1(C(C(C)C2CCCC2)=O)CCC2CCC(C1)N2C(c1cc(=O)cc[nH]1)=O 10931,c1(C(C(=O)OCCOCCOCCC(=O)O)OC)cc(F)cc(F)c1 10932,N1(C(CC(=O)NCC#C)=O)CCC(C(=O)NCCCC(C)(C)O)C12CCC2 10933,N1(C(=O)CCc2cnco2)CC=CCC1C(N1CCSCC1C1CC1)=O 10934,N1(C(C2=C(C)OCCC2)=O)CCC2(CNC(c3cnc(C)n3C)=O)CCCCC12 10935,c1(OCC(C)OC)ccc(CNCc2ocnc2C)cc1 10936,c1(CC(CC2C(C(C)(F)F)C2)=O)ccc(C(F)F)cc1 10937,CCCCC(F)C(=O)NC1CCCCC1C(N1CCC(C(CC)CC)C1)=O 10938,c1(-c2nnc(N3CCCC(C)(NC(=O)CCCCCF)C3)o2)noc2ccccc12 10939,c1(NC(COCCOCC)=O)ccc(OCC(=O)N(CC(C)C)C(C)C)cc1C 10940,Cc1cc(C(=O)NC2CC3CN(C(=O)C(CO)C(C)C)CC23)cc2nn[nH]c12 10941,CCCC(C(=O)NC(C)CCNC(c1nn(CC)nc1Br)=O)NC(N)=O 10942,CN(C)S(=O)(=O)N1CCCC1COC(=O)CC(=O)NCc1nccs1 10943,C(=O)(C(O)C1=CCCCC1)NC(C(=O)NCc1c(C)cnn1C)Cc1cnc[nH]1 10944,c1(C(=O)NCC2C(NC(c3cccc(O)n3)=O)C2)cc(Br)ccc1[N+](=O)[O-] 10945,c1(C(N2CCC(O)(CNC(Cc3scc(C)n3)=O)C2)=O)ccc(C(N)=O)c(Cl)c1 10946,c1(C(=O)NC(C(C(C)C)C)CNC(c2ccn(C)n2)=O)cc2ccc(O)cc2[nH]1 10947,C1(CCNC(C2CN(C)C(=O)C2)=O)CN(C(c2cccc(Cl)c2F)=O)CCCO1 10948,c1(C(N2C(C3CCN(C(C(C)NC=O)=O)C3)CCC2)=O)cccc(=O)n1C 10949,n1(CCC)c(C(N2CCC(CF)(NC(=O)C3=CCCO3)C2)=O)cc2ccccc12 10950,C(=O)(CCCn1cc(NC(C)=O)cn1)NCC(COCC)O 10951,C1(CN(C(C2(Cc3ccc(Cl)cc3)CC2)=O)CC)CCN(C(=O)C(O)CF)CC1 10952,C(=O)(CC=CC(C)(C)C)NCC=CCNC(CC1(C)CC1)=O 10953,c1(C(N2C(C3(O)CN(C(c4ccn(CC)n4)=O)C3)CCC2)=O)ccc(=N)[nH]n1 10954,C(N=c1[nH]c(=NCC2CCCSCC2)[nH]c2c1CC(C)CC2)c1[nH]c(=NC)sc1 10955,C1(N(C(CCN(C(C(COC)O)=O)C2CC2)=O)C)CCCC(C)C1C 10956,N1(C(CCOCC#C)=O)CC2CCC1CN2C(C1CCCC(C)CC1)=O 10957,S(=O)(=O)(c1ccc(C(C)NC(C)CSc2cccc(C)c2)cc1Cl)NCCOC 10958,C(=O)(CCCCC(N)=O)N1CCC(NC(c2c(C)ccc(OC)c2)=O)(CF)C1 10959,C(=O)(CCCC(C)(F)F)N1CC(N(C(=O)C=Cc2ccnn2C)C)C(C)(C)C1 10960,c1(C(N(C(C)CCNC(=O)C(C)O)C)=O)c[nH]c2cccc(Br)c12 10961,c1(C(N2CC3CN(c4nccnc4F)CC3C2)=O)c(F)c(F)cc(F)c1F 10962,C(=O)(CP(C)(C)=O)NC1(CCNC(CCc2n(C)ncc2)=O)CCCC1 10963,c1(N(C(C#C)C)C)nnc(-c2ccc(C)nc2)n1CC(=O)NCCO 10964,c1(C(=O)NCC2(C)CCN(C(c3sccc3CC#N)=O)C2)cc2c(s1)CCC2 10965,N1(C(C2(COC)CC(=C)C2)=O)CC=C(C(=O)N2CCC(CC)C2)C1 10966,c1(CC)c(C(=O)NC(C)(CNC(=O)C(O)CC(C)C)CO)cccc1F 10967,C1(NC(C(CCCC)O)=O)Cc2ccccc2C1NC(C1(CC)CC1)=O 10968,C1(O)(CN(C(C(C)=C2CCCC2)=O)C)CCCN(C(C2CN(C3CC3)C2)=O)C1 10969,C1(C)(C(=O)NCC(CC(C)C)NC(=O)C(C)S(N)(=O)=O)CC2(CCC2)C1 10970,N1(C(CCOCC)=O)CCC2(CC1)COC(CNC(C1(C)C=CCC1)=O)C2 10971,c1(CCNC(=O)NC(CO)CCO)nc(-c2cccnc2)no1 10972,N1(C(C2N(C(=O)CC3CCCCC3)CCC(C)(C)C2)=O)CCC2(COC(=O)N2)C1 10973,c1(C(N(C(C)CNC(c2cccc(O)c2)=O)C)=O)cccc2nsnc12 10974,C(=O)(C1Cc2ccccc21)NC(CCC=C)C(=O)N(C1CCC2(CC1)CC2)C 10975,Cc1ccc(SCCCC(=O)NC2C=CCN(C(C3CCC(=O)NC3)=O)C2)cc1 10976,N1(C(C)C(=O)NCC(O)CNC(=O)CCCc2cccs2)CCc2sccc2C1 10977,c1(COC)nc(C)c(C(=O)NCCC(C(C)C)NC(c2n[nH]cc2C(C)C)=O)s1 10978,C1(NC(c2cnc(=N)[nH]c2)=O)C2CCC1N(C(=O)Cn1ccc(Br)cc1=O)C2 10979,c1(C(=O)NC2CN(C(C3CC3C3CC3)=O)CC2O)c(F)cc(C(F)(F)F)cc1F 10980,n1(SC(C)(C)C)cc(C2OCCC2NC(=O)NC2C(C(C)=O)C2(C)C)cn1 10981,C1(C(=O)NC2(C)CC(NC(c3cc(Cl)ccc3Cl)=O)C2)CCC2(CCC2)O1 10982,c1(SC)ncc(C(F)(F)F)c(N(C(c2cc(C)cc(F)c2)=O)CC2CCNC2)n1 10983,S(=O)(=O)(c1ccc(N(C)CCOc2ccccc2)c(C#N)c1)NCCSCC=C 10984,N1(C=O)CCC(C(F)C(=O)N(C)CC2CC2CC2CC2)C1.C(=O)(CC1(N)CC1)OC 10985,c1(CCC(=O)N(C2CCC(NC(c3ncoc3C3CC3)=O)C2)C)ccc(F)nc1 10986,O=C(C#CC1CCCO1)N1CC2(CCN(C(C3(C(F)(F)F)CC=CCO3)=O)C2)C1 10987,Cc1noc(C)c1S(=O)(=O)N1CCOC2CN(c3ncc4ccsc4n3)CC12 10988,c1(OC)cc2c(cc1CNC(=O)N(CC(C)O)Cc1ccco1)OCO2 10989,c1(C(=O)NC(CC)Cn2cncn2)c[nH]nc1CCNC(C1(C)CC1)=O 10990,c1(CNC2C(C(N3CCC(Br)CC3)=O)CCC2)c(F)ccc(Cl)c1F 10991,C#CC1CN(C(=O)C(C2CCCO2)NC(=O)C=CCCC(C)C)CCN1C 10992,C(c1ccccc1Cl)=C(C)C(=O)NCC1(CNC(=O)CCCCN(C)C)CC1 10993,c1(CC(N2CC(CNC(C=CC=CC)=O)OCC2)=O)ccc(C)c(OC)c1 10994,C(C)(C)(CCC(=O)N1CCN(C2CC2)CC1)NC(c1cncc(NC)c1)=O 10995,c1(C(N2C3C(NC(c4occc4Cl)=O)CC(C3)C2)=O)cccc2occc12 10996,C(=O)(CCCCCN=[N+]=[N-])N1CC(C)N(C(Cn2ccc(C)cc2=O)=O)C(C)C1 10997,C1(CNC(CC2N(C(C3CC(C(C)C)C3)=O)CC2)=O)CNC(=O)CO1 10998,c1(NC(C2C(C)CN(C(C3C4CN(C(=O)CO)CC34)=O)C2)=O)ccc(Cl)c(Br)c1 10999,C1(C(N(CCNC(c2cnc(COC)s2)=O)C2CC2)=O)C(C2CC2)C1(F)F 11000,c1(C(=O)NC(CC(C)NC(C(C)=C2CC2)=O)C)c(C)nc(C(C)(C)C)nc1S 11001,N1(C(CC=CCCCCC)=O)CCC2CCC(C1)N2C(=O)COCCC 11002,C1(O)(CCC)CCN(C(C2CCCN(C(C3OCCCC3(C)C)=O)CC2)=O)CC1 11003,Cc1nccnc1C(C)OC(c1csc(-c2ccccc2)c1)=O 11004,Cc1nnc2n1CC(C(=O)NCCN(CCCN(C)C)C(=O)Cc1cocn1)C2 11005,N1(C(c2cnc(CC)[nH]2)=O)CC(C(F)F)CC1CNC(=O)CCCN(C)C(C)C 11006,C(=O)(C(C)C(C)(C)C)NC1C(NC(Cn2c(C(C)C)nnn2)=O)CC1 11007,N1(C(c2ccc(SC)cc2)=O)CCC2(CC1)CC2NC(=O)C(C)NC=O 11008,c1(C(C(=O)NCCC(=C)CNC(c2cnc(N)cn2)=O)CC)cccc(Cl)c1 11009,C(C)(C(=O)NCC1C=CCCN1C(=O)CN)(C(C)(C)C)NC(=O)OC(C)(C)C 11010,c1(C(=O)NCC2(CN(C(C(c3cnn(C)c3)C)=O)C)CC2)cnn(CCO)c1N 11011,c1(C(C(=O)NC2CCN(CC(=O)NC)CC2)NC(CCC#C)=O)c(C)cccc1Br 11012,C1(C(N2CCC(O)(CCNC(CCc3nc(C)sc3)=O)C2)=O)CC12CC(C)(C)C2 11013,c1(C(N(CCCCCC)CCNC(=O)C=C(Cl)Cl)=O)n[nH]c(C)c1Cl 11014,N1(C(C(C)Oc2ccccc2)=O)CCC(CNC(C2CC2C2CC2C)=O)C12CC2 11015,C=CC(C)(C)CC(=O)N(C(CC(F)F)C(=O)N1CCC(OC2CCC2)C1)C 11016,c1(C(N2CC(C)(CCC(=O)NC3CN(CCC)C3)C2)=O)cc2ccccn2n1 11017,N1(C(c2nc(C(N)=O)sc2)=O)CCC(C2CCN(C(=O)COCCCF)C2)CC1 11018,c1(CCC(N2C(C)CCC(NC(C=C(C)Cl)=O)C2)=O)ccc2ocnc2c1 11019,c1(CC)ccc(C(=O)NCCN(C(C2CC23CCOC3)=O)CC)cc1C(F)(F)F 11020,N#Cc1cc2c(n(CC3CCCN3Cc3noc4c3CCC4)c1=O)CCC2 11021,C1(NC(CC(=O)OC)=O)C2CCCC1CC(NC(C1CN3CCN1CC3C)=O)C2 11022,N1(C(C2CCN(C(CCC)=O)CC2)=O)CCN(C(C2CNC(=O)C2)=O)C2CCC12 11023,C1(c2cn(CCCC(=O)OC)nn2)CCCN(C(C2CCC(F)(F)C2)=O)C1 11024,c1(NC(C2N(Cc3c(C)noc3)CCC2)=O)cc(Br)ncc1F 11025,C1(c2nnnn2CC2CCCC(C)O2)(NCC=C)CCN(C2CCCC2)CC1 11026,c1(C(N2CCC(CCNC(C3(COC)COC3)=O)C2)=O)ccc(C(C)C)nc1O 11027,C1(C(=O)NC2C(NC(c3cccc(C(F)F)c3)=O)COC2)CS(=O)(=O)CC12CC2 11028,C1(NC(C2CCO2)=O)CC2(CCCCN2C(c2nnn(-c3ccccc3)n2)=O)C1 11029,Cc1c[nH]cc(C(N2CC(NC(c3cncc(N(C)C)c3)=O)CC(O)C2)=O)c1=O 11030,C1(C(=O)NC(C=C)CO)(CC)CCN(C(=O)CC2CCCCN2C)C1 11031,c1(CCC)onc(C)c1C(=O)NCC1(O)CN(C(=O)Cn2c(C)nccc2=O)C1 11032,CC1(NC(=O)CCF)CCN(C(=O)C(C)(C)c2ncco2)C1 11033,C#CC1(NC(N2CC(C(=O)NC)(CC)C2)=O)CCCCC1 11034,c1(CC)cnoc1C(=O)NCCN(C(c1cc(C(C)(F)F)n[nH]1)=O)CC 11035,c1(CC(=O)NCC(O)CNC(c2csc(-c3ccoc3)n2)=O)ccc(F)cc1 11036,CC1(O)CCC(CC(=O)NCCNC(c2n[nH]c(C3CC3)c2Cl)=O)CC1 11037,c1(OC)cccc(S(=O)(=O)N2CCC3C2CCCN3C(=O)C(Cl)(Cl)Cl)c1 11038,N#CC1(C(=O)NCC2(CC(=O)NCC(O)C3CC3)CC2)CCOCC1 11039,c1(CN(C)C)cc(C(=O)NC2CCC(CNC(=O)C(F)CC3CC3)CC2)ccn1 11040,C(CCCC(=O)NCCC(C)N(C)C)NC(C(N1CCOCC1)C)=O 11041,C1(CNC(c2ccc(CSC)cc2)=O)CC(F)(F)CN1C(=O)C(C)S(N)(=O)=O 11042,C1(C(=O)NCC2CC3CCC(C2)S3)C2CCCCCCC12 11043,Cc1cccc(Cl)c1CC(=O)NC1CC(CNC(=O)C=C(Cl)Cl)C(O)C1 11044,C1(C(N2CCC(C)(O)CC2)=O)CC2(CCC2)CN1C(=O)CSCC(F)F 11045,c1(C(=O)NC2(CO)CCCN(C(C(CCC)(C)C)=O)C2)nc2cc(C)ccc2o1 11046,C1(N(C(c2cccn2CC)=O)CC)CCCN(C(C2CCC2(F)F)=O)CC1 11047,C1(C(=O)NC2(C)CCCN(C(c3cc(O)cc(=O)o3)=O)C2)CCC(C2CC2)CC1 11048,c1(-c2cn(CCCC(=O)NC3(c4ncc(Br)s4)CCC3)nn2)ccc(Cl)c(Cl)c1 11049,CN1CC=C(CCNC(=O)CCN(C(=O)CC2CC3CC3C2)CC2CC2)CC1 11050,C12(c3onc(C)n3)CCC(CC1)N2C(=O)C(c1cccc(O)c1)C 11051,c1(OCC)cnc(C(=O)N(C)CC2CCN(C(c3ccn(C(C)C)n3)=O)C2)cn1 11052,c1(C(=O)NCC2(F)CCCN(S(CC)(=O)=O)C2)cnc2[nH]c(C)nc2c1 11053,C12COCCN(C1)C2=O.C(C(=O)NC1CC1OC(C)(C)C)=CCNC(C)=O 11054,c1(C(N2C(C(C)N)CCCC2)=O)ccc2c(c1)C(=O)OC2(C)C 11055,O=C1CCc2cc(C(N3CC(N4CCCC4=O)C3)=O)c(F)cc2N1 11056,c1(OCCC(COC)OC)nc2ccccc2nc1N1CCCC(F)(CO)C1 11057,c1(CNC(C(=Cc2ccco2)C)=O)ncccc1C(N1CCCC2CC12)=O 11058,C1(C(N(CC(=C)C)CC)=O)CC=CCN1C(=O)Cc1csc(C)c1 11059,C12(NC(CCc3n(C)c(S)nn3)=O)CCC(CN(C(c3ccc(F)s3)=O)C1)C2 11060,c1(OC)nc(C)ncc1C(=O)NCC1CC2(CC2)CN1C(C1CCCS1(=O)=O)=O 11061,Cc1cc(C(=O)NCCC(=O)NCc2[nH]c(C)nc2C)c(O)nn1 11062,CC(C)C(C)(CNC(=O)CC1CCCC(C)O1)NC(=O)C1=CCCS1 11063,C1(C)(CNC(C2CCC(CC)O2)=O)CCCN1C(=O)CCc1ccccc1Cl 11064,C1(CNC(C(CC=CCC)C)=O)CC2CCCCC2N1C(=O)CCC(=O)C1CC1 11065,C1(CNC(C(C=CC)O)=O)CC(C)(C)CN1C(=O)Cn1cc(C(=O)OCC)nn1 11066,c1(C(=O)NC(C#C)CC2CCOC2)ccc(-c2ccc(Br)cc2)n1C 11067,C(=O)(C1=NOC2(CCC2)C1)NC(CC(C)NC(c1ccc(CC)c(OC)c1)=O)C 11068,C(c1ccc(Cl)cc1)=CC(=O)NCC1CC(OC)CN1C(=O)CCc1cnoc1 11069,Cc1nc(CC(N2CCC(C(=O)NCCC3CCCOC3)C2)=O)cs1 11070,Cc1cc(Cl)c(Cl)cc1C(=O)NC1CCCCC1NC(=O)C(C)(C)F 11071,c1(N(C(C)C(=O)NCCOc2ccccc2F)C)cc(C(C)(C)C)nc(Cl)n1 11072,N1(C(C(C)=CCO)=O)CC=CC1CO 11073,c1(OC)cc(C(=O)NC2(C)CCN(C(=O)C(C)NC=O)C2)cnc1O 11074,c1(C(=O)CNC(c2cccs2)=O)cc(Cl)ccc1OCC1CCCO1 11075,C1(C)(NC(C(CCN(C)C)NC(c2coc(CO)c2)=O)=O)CC2CCC1C2 11076,c1(C(N2C(C(=O)NC(C3CCOCC3)CC)CCCC2)=O)ncc(C)cc1C 11077,C(=O)(CCCN(C)N=O)N1CCC(C)C1CNC(c1cnn(-c2nccs2)c1)=O 11078,N1(C(C(CC)=CCCC)=O)CCC(N=[N+]=[N-])(C(N2CCC(CC3CC3)C2)=O)C1 11079,N(C1CCOc2cc(F)cc(F)c21)C(=O)NCC#CCCCCCC 11080,N1(C(c2c(C)[nH]nc2I)=O)CCOC2(CCN(C(=O)C(N)=O)C2)C1 11081,N1(C(C(C#N)CC2CC2)=O)CCN(C(c2cncc(Cl)c2)=O)CC1CCO 11082,C#CCC(C)(C(=O)N1CCN(C(C)C)C(=O)C1)NC(=O)CCCCCF 11083,C1(C(N(C2CCOCC2)C)=O)CC2C=CC1N(C(=O)CC(=O)OC(C)(C)C)C2 11084,CC1(C)C(NC(=O)CNC(C2CCOCC2)=O)CC1CNC(=O)CC1OCCO1 11085,c1(C(=O)NC2C(CNC(C(COC)N(C)C)=O)CC2)cnn2ccn(C)c12 11086,N1(C(C(C)(C)OCC)=O)C2CCCC1CN(C(c1ccc(C)c(C)c1)=O)C2 11087,CCC(C(=O)N(CC(=O)NCC1(CCO)CN(C)C1)C1CC1)N(C)C 11088,N1(C(C(SC)SC)=O)CCC(CCC2CCCN2C(c2cnns2)=O)CC1 11089,n1(CC)nc(C(N2CCCC2CC(=O)NC2CCC(O)CC2)=O)c(C)n1 11090,C(=O)(C1=CCCSC1)NC1C(CNC(c2ccc(CNC(C)=O)cc2)=O)CCCC1 11091,C(=O)(CCC(=O)N(OC(=O)CC1CCCN1C)CC)N1CC(OCC)(C2CC2)C1 11092,N1(C(CC(CNC(C2(CCCN=[N+]=[N-])CC2)=O)OC)=O)CCN(C)CC1C 11093,C(=O)(C#CC(C)(C)O)N1CCCC(NC(C(CC)(C)C)=O)C1 11094,C12(C(N3C(CC)CC(C)C3)=O)COCC1CN(C(C1CC1(C)C)=O)C2 11095,C(=O)(C(O)CC(C)C)N1CC(O)(C(C(N2CC(C#CC)C2)=O)F)C1 11096,c1(C(=O)NCC(CCOC)NC(=O)C=C(C2CC2)C2CC2)ccc2snnc2c1 11097,N1(C(CCCOCC=C)=O)C2CCC1C(NC(=O)CNC=O)C2 11098,C1(CNC(c2c(C)c(F)ccc2)=O)CCCCN(C(=O)Cc2n[nH]c(=N)s2)CC1 11099,C1(C(=O)NCC(C)OCC#C)C2CC3C(C2NC(C2(CO)CCOC2)=O)C13 11100,C1(NC(c2c(OCC)ccs2)=O)CCN(C(C2CCCCC2)=O)C1C(C)(C)C 11101,N1(C(C2(C)CSC2)=O)CCC(C(CO)NC(c2ccc[nH]2)=O)CC1 11102,C(=O)(CN=S(C)(C)=O)N1C(CN(C(=O)CSc2ccncc2)C)COCC1 11103,N1(C(c2cnc(COC)s2)=O)CC=CC(NC(C2C(C)C2C)=O)C1 11104,CCC(CO)CCNC(=O)CC1(C)CCN1C(=O)CC1CCC(=O)C1 11105,N1(C(c2cc(C3CC3)no2)=O)CCCC(CN2CCN(c3cnccn3)CC2)C1 11106,C1(CNC(c2c(C)cco2)=O)C(C2CC2)CCN1C(c1ncc[nH]c1=O)=O 11107,c1(CC)nnc(NC(C(=O)OCC)C2COC2)s1 11108,C=CCCCC(C(=O)NC(C=C)C(F)(F)F)NC(=O)CCNC(C)=O 11109,c1(C(N2CCC23CN(Cc2ccncc2)C3)=O)cccc(C(=O)O)c1F 11110,C1(CC(=O)N(C(C)C(=O)NC2C3CCCC23)CC)CCCC(C)O1 11111,c1(NC(C2C(CNC(C3CCC(N(C)C)CC3)=O)C2)=O)nccc2cccnc12 11112,C1(NC(C(CC)CC)=O)CCN(C(c2ccc(CC#N)cc2)=O)C(CC)C1 11113,CC(C)(CNC(c1nn[nH]c1C(=O)O)=O)CNC(=O)Cc1cncnc1 11114,Cc1cc(-c2ccnc(NC(=O)Nc3cc(C)c(Cl)cn3)c2)cc(C)n1 11115,C1(NC(C(=O)NC2CC(C)OC(C)C2)=O)CCCCC12CCCC2 11116,N1(C(c2cc(C(=O)OC)no2)=O)CCC(C(C)NC(=O)C=C2CCC2)CC1 11117,c1(C(N2CC(CC(C)NC(=O)CSCC#N)C2)=O)nc2c(s1)COCC2 11118,N1(C(c2cnn(CC)c2CC)C(=O)NCC)CC2(CC=CC2)C1C(C)C 11119,c1(COC(c2ccncc2NC(CO)CO)=O)ccc(F)cc1.C1(N)CCCCC1 11120,N#CC1CCN(C(C2CCOC2CNC(C2CCCC2O)=O)=O)CC1 11121,c1(C(=O)NC2C3CN(C(C4CCCN(C(CC)=O)C4)=O)C2C3)cnc(F)c(C)c1 11122,N1(C(C(CC=C)C)=O)CC(NC(=O)Cc2ccoc2)CC(C)C1 11123,CC1CNC2CC(C2)N(C)C(=O)CC1.C(=O)(C(O)Cc1ccccc1)NC1CC1 11124,C(=O)(CCC(=O)NN(C)C)N(C)CC1(O)CCN(C(C(CC#C)O)=O)CC1 11125,c1(C(=O)NC23CC(C(=O)Nc4cccc(C)n4)(C2)C3)nc2c(s1)CN(C)CC2 11126,C1(CC(=O)OC)CC2(CO1)CN(C(=O)NCc1cccc(SC)c1)C2 11127,C1(O)(C(C)NC(COCCCC)=O)CCN(C(=O)CCc2nc[nH]n2)CC1 11128,c1(C(C)O)cn(CC(F)CCNC(c2ccc(C(N)=O)[nH]2)=O)nn1 11129,C1(NC(CC2(C)CCOC2)=O)CCCCC1CC(=O)NCCCc1ccsc1 11130,c1(C(C)C(=O)Nc2nc(CNC(c3ccccc3)=O)cs2)cccc(Br)c1 11131,N1(C(c2cc(CC)[nH]n2)=O)CCC(CNC(=O)C(C)SC)C(C)C1 11132,c1(OC)ccc(Br)cc1C(N1C(C(N2CC(F)CC2C(N)=O)=O)CC2CC12)=O 11133,N1(C(CC(C)N(C(C(C(=O)OCC)CC)=O)C)=O)CC2(C1)NC(=O)NC2=O 11134,c1(C(N2CCCC(CCNC(CCC(C)OC)=O)C2)=O)ccc(C)c(Cl)c1 11135,N1(C(C=Cc2ncn(C)c2)=O)C2CCC1CN(C(c1cc(C3CC3)sn1)=O)CC2 11136,c1(OCC(=O)NCCC2N(C(CC#C)=O)CCCC2)ccc(Br)c(Cl)c1 11137,CCC(C)CC(=O)NC1CC(CNC(=O)CSCc2ccc(Cl)s2)C1 11138,c1(OC)nccc(C(=O)NC2CC(C(=O)N(C3CCOCC3)CCO)CC2O)n1 11139,N1(C(CCSC)=O)CCN(C(C23CCC(N=[N+]=[N-])C2C3)=O)C(C)C1C 11140,c1(OC)cc(C(=O)NC(C)CC2CN(C(=O)CN3CC4CC4C3)C2)sn1 11141,c1(OC)ccc(CC(=O)NCC2C=CCN2C(c2conc2C)=O)cn1 11142,c1(C(=O)NCC2(OC)CN(C(c3ncsc3C(F)(F)F)=O)C2)occ2c1CCC2 11143,C(=O)(C(C)(C)CS(N)(=O)=O)NCC1CN(C(C(CC)NC(C)=O)=O)CC1O 11144,Cc1ccc(NC2CCCN(C(C)C)C2)c(-n2cc(-c3cnsc3)nn2)c1 11145,N1(C(c2c(C)n[nH]c2C)=O)CCN2C(=O)C(NC(=O)CC(C)(C)C)CC2C1 11146,c1(OC)ccc(NC(c2ccccc2NS(=O)(=O)C2CC2)=O)c(OC)c1OC 11147,C(CC(C)C(=O)NCC1(F)CC(CNC(c2cc(Cl)cs2)=O)C1)OC 11148,Cn1oc(C(=O)NC2CN(C(=O)COC3CCCCC3)C2)cc1=O 11149,c1(OCC(N2CC(OC)(CNC(=O)CC3CCCN3C)C2)=O)cc(Cl)ccc1Cl 11150,c1(C(N2C(C)C(NC(=O)C(=O)N=S(C)(C)=O)CCC2)=O)cn2c(n1)C(C)CCC2 11151,N1(C(CCC=CC)=O)CCCCCC(NC(=O)C(C(C)O)N(C)C)C1 11152,Cc1ccc(C2CC2C(=O)N(CCCCCNC(C2(F)CCOC2)=O)C)cc1 11153,C1(CC)CN(C(C2CCN(C(=O)C(C)C(=O)OC)C2C)=O)CCS1 11154,CN1CCCCC1CC(=O)NC1CCCC1(C)CNC(c1c[nH]nc1C(F)F)=O 11155,c1(C(=O)NC23COC(CNC(C4(O)CCC4)=O)(C2)C3)cc([N+](=O)[O-])cnc1O 11156,C1(CC(=O)NC(C(C)(C)NC(c2cnc(C(C)C)s2)=O)C)CC(=O)NC1=O 11157,N1(C(CCC(C)(C)NC(=O)Cn2cnnc2O)=O)CC2CC(C1)C2(C)C 11158,c1(OC)ccc(C)c(C(=O)NCC2(CCCNC(=O)C=C(C)C)CCCC2)n1 11159,O=S(=O)(c1cccc(F)c1)NC1CN(Cc2ccccc2)CC2(CCC2)O1 11160,c1(OC)cc(C(=O)NCC2CCC2NC(c2cc(Br)n(C)n2)=O)ccc1C 11161,c1(C(N2CCC(N(C(=O)CC3CCC(=O)N3C)C)C2)=O)ccc([N+](=O)[O-])c(Cl)c1 11162,c1(C(N2CCC(CC)C2C(=O)Nc2cnccc2C)=O)ccc2n[nH]cc2c1 11163,c1(CNC(=O)N)cccc(Cl)c1Cl.CC(C)(C)OC(=O)NCC1CC1C(=O)O 11164,c1(N(C)CCc2ccccc2)nc(=NCC2CCC3CC23)[nH]c2cccc(F)c12 11165,c1(C(=O)NC2CN(C(C3CC(O)(CC#C)C3)=O)CC2O)cccc2c1OCC2 11166,C(=O)(C(CC(N)=O)NC(c1ccccc1)=O)NCC1CCN(C(CCC=C)=O)C1 11167,Cn1cnn(CC(N2CC(CNC(=O)CCc3ccc(Cl)cc3)C2)=O)c1=O 11168,C1(C(NOCC=C)=O)COCCN1C(c1ccc(C)nc1)=O 11169,c1(CCNC(C2(COC)CCCS2(=O)=O)=O)coc2ccccc12 11170,c1(C(N2C(COC)CN(C(=O)C=C(C)C)CC2)=O)cnn2ccc(OC)cc12 11171,c1(CC)cc(N(C)CC2(CNC(=O)C(C3CCOCC3)F)CC2)nc(CC)n1 11172,C1(C(N(CC(C2CC2)OC)C)=O)C2CCCC2CN1C(=O)Cn1ccccc1=O 11173,N1(CC)CC(NC(C2(CCNC(c3ncn(C)c3C)=O)CCC2)=O)CC1=O 11174,n1(CC(=O)NC2CC3CC2CN3C(c2ccoc2C2CC2)=O)nc(O)ccc1=O 11175,CCC(CNC(C1CC(=O)N(C2CC2)C1)=O)(CC)c1ccccc1 11176,Cc1c(C(=O)N(CCC(=O)NC(CO)CCF)C2CC2)ccn1C 11177,c1(-c2cn(CC3CCN(C(CN(C)C)=O)C3)nn2)cc(CO)ccn1 11178,CCC(C(=O)N(C1(C(=O)NCC(F)Cl)CC1)C)C(C)C 11179,c1(CC(=O)NCC(C)NC(c2c(CC)ocn2)=O)ccc(F)c(Cl)c1F 11180,CC1(C)C(C)(C)C1(F)C(=O)NCC1CCCN(C(c2nnc(O)nc2O)=O)CC1 11181,c1(C(C)N(C(C2CC3CCC2CC3)C(=O)NCC2CC2)C)nc2ccccc2s1 11182,C(CCNC(c1ccncc1)=O)(C(C)(C)C)NC(c1cc(C2(C)CC2)n[nH]1)=O 11183,CN1CCCCC(C(=O)NCC(C)(C)CNC(C2(C)CCC(=O)C2)=O)C1=O 11184,c1(CCC)noc(CCC(=O)N(C2CCN(C(=O)C=C(C)C(F)F)C2)C)n1 11185,C1(CNC(c2occ(C)c2)=O)CC(C)N(C(c2cn(C(C)C)cn2)=O)C1 11186,C(C)(CCC(C)(C)C)NC(c1nnnn1CC(F)F)C1CC(=C)C1 11187,CC(C)P(=O)(CC(=O)NCC1(C(C)(C)O)CN(C(=O)C(C)(C)F)C1)C(C)C 11188,C1(O)(CNC(CC2(N(C(CC3(OCC)CC3)=O)C)CC2)=O)CCCC1C 11189,CCCCC(CNC(=O)COCCCF)NC(=O)C(C)Oc1cccc(C)c1 11190,CC(=O)C(C)CC(C)C(=O)N(C)CCNC(c1n[nH]c2c1CCC2)=O 11191,c12ncc(F)c(n1)Nc1ccc(cc1)C(=O)N1CCN2CC1.C(C(F)(F)F)O.CO 11192,c1(C(N(C)CC2CC(F)CN2C(=O)C=C2CC2)=O)cccn2nnnc12 11193,c1(C(=O)NCC2(CN(C)C(c3ccc(Cl)cc3)=O)CC2)cnn(C)c1N 11194,Cn1nnc2ccc(C(N3CC(NC(c4ccc(=O)oc4)=O)C4(CC4)C3)=O)cc12 11195,N1(C(C2(SC)CCC2)=O)CCN(C(C2CCCCS2)=O)C(c2nccn2C)C1 11196,c1(C(N2CCC(N(C(C(COC)OC)=O)CCO)C2)=O)nnc2ccccc2n1 11197,c1(OCC)cccc(C(=O)NC2(C)CCN(C(c3n[nH]c(C4CC4)n3)=O)C2)c1 11198,c1(CC(C)C(=O)NCCCNC(C2CCCS2)=O)ccc(Cl)c(Cl)c1 11199,N1(C(C2C(C)(C(C)C)C2)=O)CC2CCC(NC(=O)Cc3cc(C4CC4)no3)C2C1 11200,N1(C(CCC2(NC(COCCOC)=O)CCC2)=O)CCC(CO)C(C)(C)C1 11201,Cc1cccc(C(CNC(=O)N(C(C)(C)S(C)(=O)=O)C)N(C)C)c1 11202,C(C(CCC(=O)O)CC(F)(F)F)N(CCC=C)CCCC 11203,N1(C(CC(COC)C)=O)CCCC(C)(NC(=O)CCCc2ccc(Cl)cc2)C1 11204,N1(C(C2CCC(C(=O)OC)C2)=O)CC2CC(C)N(C(c3ccsc3Cl)=O)C2C1 11205,c1(CC)cc(C(=O)NCC2(C(N3CC(O)C3)=O)CC(C)(C)C2)c(C)o1 11206,C1(C(=O)NCC2(F)CC(CNC(C3CCCO3)=O)C2)Cc2ccccc2S1 11207,CCCCC(O)C(=O)NC(CCC(=O)N(CCO)CCN(C)C)C(C)C 11208,C(=O)(CCS(=O)(=O)C(F)(F)F)N1CC(CCNC(Cc2cnn(C)c2CN)=O)C1 11209,CC1COCCC1NC(=O)C(CC1CCC1)NC(=O)CC=C(Cl)Cl 11210,C1(NC(COCCCCC)=O)CN(C(c2cnc(CC)s2)=O)CCC1CO 11211,CC(C)CC(C(=O)N1CC(C(=O)NCc2ncoc2C2CC2)CC(C)C1)C(N)=O 11212,CC(C)(C)C(CNC(=O)C(O)CC1CCOCC1)NC(C1(CF)CCC1)=O 11213,C1(C(N2CCC(N(C)C(c3cnc(C(F)(F)F)o3)=O)C2)=O)CCOC(C)(C)C1 11214,N1(Cc2nc(CCCC)on2)CCC2(CCN(C(=O)C(O)CC(C)(C)C)C2)C1 11215,N1(C(C2C(=C)C2)=O)CCC(CO)(CNC(=O)Cn2cccnc2=O)C1 11216,c1(NC(C2C3(CN(C(CC(CC)C)=O)C3)C2)=O)cc(F)c([N+](=O)[O-])cc1F 11217,c1(C(N(CC(CC)NC(C2(O)CCOC2)=O)C)=O)ccsc1SC 11218,c1(NC(N2CCCC(O)(c3ccc(Cl)cc3)C2)=O)ccc(S(=O)(=O)CC2CC2)cc1 11219,N1(C(Cc2c(C)ccnc2)=O)CC2CCC1C(NC(=O)CCn1ccnc1C)C2 11220,C1(CNC(c2ncn(C(C)(C)C)n2)=O)CC2CCC1N2C(C1(C)CCC(=O)C1)=O 11221,C(=O)(C1CCCc2ncccc21)NCC(CNC(c1c(C)onc1C1CC1)=O)C 11222,c1(C2N(C(C3N(c4ccnc(OC)n4)CCCC3)=O)CCC2)ccc(Br)cc1F 11223,CC1(NC(C2CC2(C)C(F)(F)F)=O)CC(NC(c2ccccc2)=O)C1 11224,C(N=c1cc[nH]cc1S(=O)(=O)NC(C)(C)C1CC1)c1cnc(CC)s1 11225,N1(C(C(C2CCCC2)NC(C2NC(=O)CC(C)C2)=O)=O)CCC2CCC(C1)N2C 11226,C1(C(=O)NCCC(C)N(C(C(C)OCC#C)=O)C)CC12CCOCC2 11227,CC(CN(C)C)CCC(=O)N(C(=S)Nc1nccs1)CC(=O)N(C)C 11228,N1(C(C(C)N(CCC)C(C2CCCCS2)=O)=O)CC2(COC(=O)C2)C1 11229,c1(NC(C)=O)ccc(C(=O)NC23CCN(C(=O)OC(C)(C)C)CC2C3)c(C)c1 11230,c1(C(N(CCNC(C2N(C(C)=O)CSC2)=O)C2CC2)=O)cnc(C2CC2)nc1C 11231,C1(C)(CNC(C(c2cccnc2)C)=O)CCCN1C(c1cccc[n+]1[O-])=O 11232,c1(C(=O)NCC(C)NC(=O)C(c2ccc(Cl)cc2Cl)O)nccc2[nH]ccc12 11233,c1(CN(C)C(c2cccc(-c3cc4ccccc4o3)c2)=O)ccc2c(c1)CCO2 11234,C(=O)(CC(CNC(c1csc(F)c1)=O)OC)NC(c1ncc[nH]1)CC 11235,Cc1nc(NCCc2nc3c(s2)CCC3)cc(=NC(C)c2cc(Br)no2)[nH]1 11236,N1(C(C2(C)COC2)=O)CC(C(N2CCCCC2CCCO)=O)C(C)(C)C1 11237,C(=O)(CC1OCc2ccccc21)NCC1CN(C(C(CCOC)C)=O)C(C)C1 11238,Cn1c(=N)[nH]c2ccc(C(N3CCCC4(NC(=O)CCC(N)=O)CC4C3)=O)cc12 11239,C1(CC(=O)NCC(CC)OC)CCCN1C(c1csc(NC(=O)C2CC2)n1)=O 11240,c1(CC(c2c(C)c(Cl)sc2Cl)Nc2cc(Cl)ccc2Cl)cnc2cccnc2c1 11241,c1(C(N(CCCCNC(C2CC2C2CCCO2)=O)C)=O)ccncc1Br 11242,C1(NC(C(CSC)C)=O)CC2CN(C(c3cc(-c4ccncc4)on3)=O)CC12 11243,N1(C(C(Cc2cn[nH]c2)NC(c2cc(OC)no2)=O)=O)CCOCC1CO 11244,CC1(C2(C(N3CCC(CCC(=O)N4CC(C(F)(F)F)C4)C3)=O)CC2)CC1 11245,N1(C(C(C)(C)NC(=O)C(F)(F)F)=O)CC2CN(C(C3CC(=O)C3)=O)CC2C1 11246,C1(N=[N+]=[N-])(C(=O)NCC(CCC)OC)CCN(C(=O)CCCC(C)(C)C)C1 11247,N1(C(c2nc(C)nc(O)c2)=O)CC2CCN(C(c3cc(C(F)F)n(C)n3)=O)CC12 11248,c1(CNC(=NCCOCC)NC2COC(C)C2)nc2cccc(Cl)c2n1C 11249,C1(NC(C(C2CCCCC2)N(C)C)=O)CCN(C(=O)CCF)CC1O 11250,c1(C(=O)OC)nccn1CC1CN(C(=O)CC2(NC(=O)C(C)(Cl)Cl)CCC2)C1 11251,N1(C(=O)CCC2CCOC2)CCCC2C1CCN2C(=O)C(F)F 11252,C(CC(F)(F)Cn1cc(CCC2CC2)nn1)NC(C1(CCCC)CC1)=O 11253,N1(C(C2CC(CC)N(C(c3ccccc3C)=O)CC2)=O)CCC2(CC=CCO2)C1 11254,N1(C(c2cncc(C)n2)=O)CCC2CN(C(=O)Cc3nc(C4CC4)cs3)CC2C1 11255,C1(C(=O)NCCCN(C(=O)CC2CCCCO2)C)(CC)CCOCC1 11256,c1(C(N(C2CCN(C(=O)CC3C=CCCC3)CC2)CCOC)=O)ccccc1C 11257,S(=O)(=O)(c1cccs1)N(C(C(N1CCC(N(CCCO)C)CC1)=O)=O)CCO 11258,N1(C(CC(=C)C)=O)CC(NC(=O)CCc2cc(Cl)no2)CC(C)C1 11259,c1(C(N2C3CN(C(C4C(CCC)C4)=O)C(C3)C2)=O)ccc(Br)c2cn[nH]c12 11260,c1(C(=O)NCC2N(C(C3C(C)C3)=O)CCCCC2)c[nH]c2nccc-2c1 11261,c1(OC(=O)Cc2csc3ccc(Br)cc23)ccc2c(c1)CCCO2 11262,N1(C(C(C)=C(C)C)=O)CCC(NC(c2cc(C)cnc2Cl)=O)CC1C 11263,C1(CC(N2CCC(OCCNC(C3C(OCC)C3)=O)C2)=O)CCCS(=O)(=O)C1 11264,c1(NCc2c(N)ncc(Br)c2)ccc(S(=O)(=O)NC2CCSC2)c(Br)c1 11265,Cc1cc(C)c(C(=O)NCC2(C(F)F)CCN(C(=O)C(CCO)N(C)C)C2)cn1 11266,CC(C)(CCCF)C(=O)NCC1CCN(C(C2CCCC(=O)CC2)=O)C1 11267,N1(C(c2c(C)cno2)=O)CCC(CNC(c2ccn(C3CC3)n2)=O)C12CCC2 11268,N1(C(C(Br)=C(C)C)=O)CC(CNC(=O)COC2CCCCC2)CCC1C 11269,N1(C(c2cnc(C)o2)=O)CC(NC(c2ccc(CC(C)(C)C)cc2)=O)CC1C 11270,C(=O)(CCS(C)(=O)=O)N1CCC(CC)C1C(=O)NCCc1cnc(C)[nH]1 11271,C1(C(=O)NC(C)CCF)CN(C(=O)CC#N)C2(CCC2)C1 11272,c1(OC)ncc(C=CC(N2CC(NC(C3CCCS3)=O)C3(CC3)C2)=O)cn1 11273,C=CC1(CC(=O)NC(c2ccnn2C)C)CN(C(=O)CCSC)C1 11274,Cc1onc(Cl)c1C(=O)NC(C)CC1CN(C(c2ccc(C#N)s2)=O)C1 11275,C1(C(N2CCC(CNC(CCNS(CC)(=O)=O)=O)CC2)=O)CCCCC1(F)F 11276,N1(C(c2c(Cl)cn(C)n2)C(=O)NC2CCOC2)CCCC2(CCCNC2=O)C1 11277,CC1CC=C(C(=O)N2CCC(CN(C)C(c3cccc(O)c3F)=O)C2)CC1 11278,Cc1cc2nc[nH]c(=NCC(C)N(C(=O)C(c3ccc(F)cc3)O)C)c2[nH]1 11279,C1(C(N(CCCCNC(c2c(C)ccc(Cl)c2)=O)C)=O)CCCC2CCCN12 11280,Cc1cc(N(C)CC2CS(=O)(=O)CCO2)nc(=NCC2(CS(C)(=O)=O)CC2)[nH]1 11281,C1(CN(C(C(C)O)=O)C)CCCN(C(=O)C=CCN2CCC2)C1 11282,c1(CC(=O)NC2CN(C(C3CCN(CCO)C(=O)C3)=O)C2)ccc(O)c(Br)c1 11283,c1(NC(C(CNC(=O)CCNC(N)=O)OC)=O)cccc(C(C)F)c1 11284,c1(NC2C(C(=O)Nc3c(OC)cc(F)c(C)c3)C2)ncnc2c(C)cccc12 11285,CC1=C(C(=O)N2CCCCC2CCN(C)C(C2(C#N)CC2)=O)CCC1 11286,N1(C(C2(O)CCCN(C(C)=O)C2)=O)CC2CN(C(c3c[nH]c(=O)cn3)=O)CC2C1 11287,c1(C(=O)NC2C3CN(C(CC4(C)CC4)=O)C2C3)cc(N(C)C)nc2ccccc12 11288,Cc1cc(O)ccc1CNC(C12CC(NC(=O)OC(C)(C)C)C1C2)=O 11289,c1(C(=O)NCC23C(CN(C(C(CC)COC)=O)C2)CC3)cnc2[nH]cnc2c1 11290,C1(N(C)C)CC(C(=O)O)CN(C(=O)CC2CC(SC(C)(C)C)C2)C1 11291,CC(C)C(O)C(C)C(=O)N1CC(C(=O)NC2CC(C3CC3)C2)CCC1C 11292,N1(C(COCCC)=O)CC(N(C(=O)CNc2cccnc2)C)C(C)(C)C1 11293,C1(C)(CNC(C2CN(CCC)C(=O)C2)=O)CCCN(C(c2cn[nH]c2)=O)C1 11294,C#CCC(C)(CNC(=O)NCc1cc(C(=O)OC(C)(C)C)c(C)s1)CO 11295,CC(CC(C)(C)C)C(=O)NCC12CCC(CN1C(c1cc(Br)n[nH]1)=O)C2 11296,N1(C(CC(C)F)=O)CCCC(CN2CCN(C(c3ccc(C(N)=O)s3)=O)CC2)C1 11297,N1(C(Cc2nc(C)oc2)=O)CC2ON=C(CNC(c3nnc(C)s3)=O)C2C1 11298,C1(C(N2CCC(COC)(NC(=O)Cc3cncnc3)C2)=O)CC2C(C1)C2(F)F 11299,C(=O)(C(C(C)(C)C)OCC)N(CCC)CCNC(C12CCCC1C2)=O 11300,N1(CC(N2CCC(C3CCCN3C(C34CSCC3C4)=O)C2)=O)CCC(F)CC1 11301,c1(N2CC(C(C)C)OCC2)nc(NC2CC2C(F)(F)F)c2cnn(C)c2n1 11302,c1(C(C)C)ccc(C(C)NC(c2nnnn2CC(F)F)c2ncco2)cc1 11303,Cc1cc(CC(=O)NCC(O)CN(C)C(c2nc(C3CC3)cs2)=O)cs1 11304,Cc1[nH]c(C(=O)NC(CCN(C(=O)CCC(N)=O)C)C(C)C)c(C)c1C 11305,CC1OC(C)C(C(=O)NC2(CCCCNC(=O)CC3CC(F)(F)C3)CC2)C1C 11306,c1(C(N2CCCC(N(C)C(c3ccsc3)=O)CC2)=O)cc(N)cc(O)c1F 11307,N1(C(C2C(COC)C2)=O)CCCC(CO)C1.C12CC(N(C(=O)OC)C1)NC2=O 11308,CC(C)C(CNC(=O)CC1CSC1)C(=O)NCc1ccon1 11309,N1(C(c2cc(OC)n(C)n2)=O)CC(C)(C(N2CC3C4CCC(C4)C23)=O)CC1(C)C 11310,O=C(C#CC1CCCCO1)NC1CCC2CCN(C(=O)CCC3CC3)C1C2 11311,Cc1cn2c(n1)CCC(C(=O)NC1CC(CNC(c3ccc(C)s3)=O)C1)C2 11312,C1(N(CCNC(C(CC)O)=O)C(c2cc(OC)ccn2)=O)CCCCCC1 11313,N1(C(CC=C(C)C)=O)CCC(N(C(=O)CCCN(C)C)CC2CCCC2)CC1 11314,Cc1ccnc(CNC(C2COCCN(C(c3ccncc3)=O)C2)=O)c1F 11315,C1(C(N2CCN(C(=O)C=C3CCSCC3)C(C3CC3)C2)=O)CC2CCC(C1)C2 11316,c1(C(N(C)CCNC(c2ccsc2Br)=O)=O)ccc2sc(=N)[nH]c2c1 11317,N1(CCCNC(c2sccc2NC(C2CCCCC2)=O)=O)CCS(=O)(=O)CC1 11318,Cn1nc(CNC(=O)NNC(=O)c2cc(Br)cs2)c2c1CCC2 11319,C#CC1(C(=O)NCCC2(C)CCCC2)CCN(C(C2CCC(N(C)C)C2)=O)CC1 11320,CC1(C)CCCN(C(=O)C2=CCCOC2)C1C(N1CCNC(=O)C1)=O 11321,C(=O)(CCCCCCC(=O)N1CCC(NC(c2ccc(SC)o2)=O)C(O)C1)OC 11322,C12(NC(c3ccc(OCC)cc3)=O)CCCC1CN(C(c1occc1F)=O)C2 11323,n1(CC(=O)NC2C(C)CN(C(C3CC34CC4)=O)C2)cnc2ccccc2c1=O 11324,c1(C(N2C(C3(NC(CCC=C(C)C)=O)CC3)CCC2)=O)ncc(Cl)cc1O 11325,Cc1cc(C(=O)NNC(=O)N2CCC(C(=O)N(C)C)C2)c(C)n1-c1ccc(F)cc1 11326,C=C(Cl)C(C)(C)C(=O)NCC1CC(CNC(C2CC2c2cccnc2)=O)C1 11327,C(=O)(C1=C(Cl)CCOC1)NCC1C(NC(CC2CCCC(C)(C)O2)=O)CCCC1 11328,C(=O)(C(CNC(c1c(Cl)cnn1C)=O)C(C)(C)C)NCC1(O)CCN(C)C1 11329,C1(NC(C2N(C(=O)NC)CCC2)=O)CCC2CC1CN2C(c1ncncc1Cl)=O 11330,C(C)(C)(CC(=O)N(C)Cc1ccccn1)N(C(C1C(C)C1C)=O)C 11331,c1(C(=O)NCCN(C(C)C)C(c2cc(Cl)cn2C)=O)nc2n(c1Cl)CCCC2 11332,N1(C(CC)=O)CCC(NC(C2CCCN(Cc3ccccc3)C2)=O)C12CC2 11333,N1(C(C2CN(C(N)=O)C2)=O)CCOC2(CCC(NC(C3CC=CC3)=O)CC2)C1 11334,c1(N2C(C3(NC(c4n[nH]cc4C4CC4)=O)CC3)CCC2)ccc([N+](=O)[O-])cc1 11335,CC(C)CC(CNC(=O)CCC(=O)c1ccccc1N)NC(=O)C=C1CC1 11336,C(=O)(C1=CC2C=CC(C1)C2)NC(C(=O)N(C(C=C)C)C)CO 11337,C1(NC(C=NOC)=O)C2CC3CN(C(=O)CCCCC(F)(F)F)C1C3C2 11338,CCC(CNC(c1cscc1C)=O)(CC)NC(c1ccc(C2COC2)cc1)=O 11339,N1(C(c2nc(CC)oc2)=O)CCC2(COC(CNC(=O)CCS(C)(=O)=O)C2)C1 11340,Cc1ccc(C2CCCCC2)n1NC(=O)OCC(=O)OC1CCCCC1 11341,CCCC(C(=O)OCCCc1nc(C)cs1)n1ccc(C2CC2)n1 11342,N1(C(CCC=CC(C)C)=O)CC2(CCCC2)C1 11343,CCC(COC)C(=O)NCCCN(C(c1cc(C(C)(C)O)ccn1)=O)CC 11344,O=C(CCc1ccco1)NCCN(C(=O)Cc1nc[nH]n1)C1CC1 11345,C(CCS(=O)(=O)NCC(=O)NC1CN(C(C2(C)CCCC2O)=O)C1)OC 11346,CCC(CC)C(=O)NCC(=O)NCCCC1(NC(=O)C(C)C(C)O)CC1 11347,CC1=C(C)CC(C(=O)NCC2CCN2C(c2c(C)noc2C(F)(F)F)=O)CC1 11348,n1(CC(=O)NC(CCOC)CNC(=O)Cn2ccc(C3CC3)n2)c(C)ccc1C 11349,Cc1ncc(F)c(N2CCC(C#N)(NC(c3n[nH]c(C)c3C)=O)C2)n1 11350,C1(NC(c2csc(-c3ccccc3)c2)=O)CC2(C1)CN(C(C1CCCCO1)=O)C2 11351,c1(C(=O)NC2CN(C(=O)C(F)(F)c3nccs3)CCC2F)cccc2nccn12 11352,N1(C(C(C)N(C)C)=O)CCCCC1CNC(=O)C(F)(F)c1cnn(C)c1 11353,c1(CCC(=O)NCC(C)(C2CC2)NC(C(CCC)OC)=O)ccc2ocnc2c1 11354,CCC1c2ccsc2CCN1C(c1cc(F)ncc1C)C(=O)NC(C)(C)C 11355,C(C(C)(C)C(=O)NC(C)CCCNC(=O)C(O)CCSC)OCC 11356,Cc1cc(CCC(=O)NCCCCNC(C2CC(OC(C)(C)C)C2)=O)cc(C)c1 11357,Cc1cc([N+](=O)[O-])cnc1C(N1CCC(C2(NC(c3csc(O)n3)=O)CC2)C1)=O 11358,CN1CCCC1C=CC(=O)NCCN(C(=O)C=Cc1cscn1)C1CC1 11359,c1(CCC(=O)N(C(CC)C)CC)ccc(OC)c(OC(=O)C(C)=CC(C)(C)C)c1 11360,C1(C(N2C(CN(C(c3ccc(C(C)C)cn3)=O)C)CCC2)=O)C(C)OC(C)C1C 11361,C(CO)(C(=O)NCc1cc(C(N2CCC(c3nn[nH]n3)C2)=O)co1)N(C)C 11362,c1(C(N(CC(CC)NC(CC(=C)I)=O)C)=O)n[nH]c(C)c1O 11363,Cc1cc(Cl)cnc1C(N1CC(O)(CCc2cn(C3CCCC3O)nn2)C1)=O 11364,Cc1cc(F)c(C(=O)CN2CCN(c3ccccc3)C(=O)C2)cc1F 11365,c1(NC(C2(O)CCC(CCC)CC2)=O)cc(F)ccc1C(F)(F)F 11366,CCC(CC(=O)NCCC1CC(C)C1)N(C)C(c1cnsc1C)=O 11367,c1(CNC(Cc2cn(CC)nn2)=O)ncccc1CNC(C1CNC(=O)C1)=O 11368,CCC(C(=O)OC)N(C(c1cnn(CCCl)c1)C(=O)NCC(F)F)C 11369,C=CC1OCCC1C(=O)NCCOC1CN(C(=O)CC(O)CN(C)C)C1 11370,C=CC(C)(C)CC(=O)NCC12CC(NC(c3cc(CC)ccc3F)=O)(C1)C2 11371,c1(C(=O)NCC(C(C)(C)C)OC)cc(CN)c2n1CCOC2 11372,NS(=O)(=O)c1cc(C(=O)NC2CC(F)CN(C(C3CC=CCO3)=O)C2)ccc1F 11373,Cc1ccc(C(=O)NCCN(CC(C)O)C(c2coc(Br)c2)=O)o1 11374,c1(C(=O)NCCOCCNC(C2CC(F)(C(=O)NC3CC3)C2)=O)cccc(Cl)c1 11375,C1(C(=O)NC2CCCCN(C(CC(C)C3CC3)=O)C2)Cc2ccccc2N1C 11376,c1(OC)cc2[nH]ncc2cc1NC(=O)CC1CCN(C(c2cncnc2)=O)C1 11377,c1(NC(=O)OCC2CCCC2C(=O)NCC)ccc2c(c1)OCCO2 11378,Cc1cnccc1C=CC(=O)NCC1(C(N)=O)CN(C(=O)CCC(N)=O)C1 11379,c1(C(N2CC(O)(Cn3cncn3)C2)=O)ccc(CNC(C2CC(O)C2)=O)nc1 11380,N1(C(=O)CCC2CC2(F)F)CC(O)C(O)C1CNC(C1(C(N)=O)CC1)=O 11381,C1(C(N(C(C(=O)NC2CCC(C)C2)(C)C2CC2)C)=O)CC(=O)CC(=O)N1 11382,N1(C(C2CCC(=C)CC2)=O)CCC2CCN(C(=O)C(C)SC(C)C)CC2C1 11383,c1(C(N2CC(NC(c3ccc(CO)o3)=O)CC(C)C2)=O)cc2c(cn1)OCCO2 11384,c1(C(=O)N)nc(C)n(C)n1.c1(CC(CCc2cccnc2)NC(C)=O)ccccc1 11385,C(C#CC(F)(F)F)OC1CCN(C(C(=O)NCCOC)=O)C1 11386,c1(NC2CCC(NCC(Br)=C(C)C)C2)ccc(S(=O)(=O)N(C)C)cc1C#N 11387,c1(C(N(C2CCCN(C(C3C4COCC34)=O)C2)C)=O)ccc2c(c1)C=CS2(=O)=O 11388,c1(-n2cc(Cn3cnc(C(=O)OC)n3)nn2)cccc(OCc2ccccc2)c1 11389,Cn1c(C(N2CCOC(C3CN(C(=O)C=CCO)C3)C2)=O)cnc1O 11390,C(N=c1cc(C)nc(NC(CC2CC2)C2CC2)[nH]1)C1(OC)CCSC1 11391,C(CCC(C)C)(C(=O)N1CCC(O)C(C)C1)NC(CCN(CC)CC)=O 11392,c1(NC(C2CC(C)CN2Cc2cncc(O)c2)=O)ccc(C(N)=O)c(F)c1 11393,C1(NC(CC(=O)OCC)CC#N)CC2COCC(C1)C2 11394,c1(C(=O)NCC(CO)NC(c2ccc(C3(C)CC3)cc2)=O)cccc([N+](=O)[O-])c1 11395,Cc1c(Cl)ccnc1C(N1CCC(CF)(NC(=O)CCc2ncc[nH]2)C1)=O 11396,c1(C(=O)Nc2cc(C(C)O)c(F)cc2)nc(O)c2ccccc2n1 11397,n1(CC(C)N(C(=O)CC2(c3ccccn3)CC2)CC)cc(CCC2CCOC2)nn1 11398,Cn1nccc1C(N1CCC(c2ccccn2)C1)C(=O)NC1(C)CC1 11399,N1(C(=O)Nc2n(C)c(=O)on2)CCN2C(=O)COCC2C1 11400,C(N=c1[nH]cnc2cc(C)[nH]c12)C1C(N(C(=O)CN2CCCC2=O)CC)CCC1 11401,N1(C(C(CC)C)=O)C2CCC1C(C(N1CCCC1c1ccncc1)=O)C2 11402,c1(C(=O)NC2(CC(NOC3CCN(C)CC3)=O)CC2)cccc2[nH]ncc12 11403,C12(C(N(CC(CN(C(CC3CCN(C)C3=O)=O)C)O)C)=O)CCC(CC1)CO2 11404,C1(NC(C(C)SCCCC)=O)CN(C(c2cc(CCOC)on2)=O)CC1C 11405,Cc1cc(C)c(C(N2CC3CCC2C(NC(c2cccs2)=O)C3)=O)c(C)c1 11406,C1(C(=O)NCCN(C(=O)C2=CCCOC2)CC(C)O)C(C)(C)CCCC1(C)C 11407,N1(C(c2c(CC)c(C)sc2)=O)CCCC2(C1)CN(C(C1CN3CCN1CC3)=O)C2 11408,Fc1cccc2cccc(CNCc3cc(F)c(F)cc3N)c12 11409,Cc1ccc(C(=O)NCC=CCNC(=O)C(=Cc2c[nH]cn2)F)cc1F 11410,C(C(C)(C)C#CC(=O)N1CCCC(C)(OC)CC1)NC(C(CC)C)=O 11411,C(C(C)(COC)C(=O)N1CCC(NC(=O)CC2CSC2)C(CO)C1)OC 11412,N1(C(C2C(C(=O)OCC)C2)=O)Cc2ccnn2CC1C.C1(=O)CCCC(C)(C)N1 11413,Cn1cnc(CCNC(C2(C3CCCN3C(=O)CNc3cnn(C)c3)CC2)=O)n1 11414,C1(CNC(C2(COC)CCCC2)=O)CC(C)(C)CN1C(=O)C1CC1 11415,c1(C(=O)NCC(CCCC)NC(=O)C2=CCCC2(C)C)ccc(Cl)c(C)c1N 11416,C(=O)(CCC(F)(F)c1ccc(Br)cc1)NCCC(CC)F 11417,S(=O)(=O)(c1cccc(F)c1C)N1CCN(C2CN(C(C=COCC)=O)C2)CC1 11418,C(CCCCCC(=O)NCCCC1(NC(c2csnc2C)=O)CC1)SC 11419,C1(CNC(=O)COC2CCCNC2)CCNC2(CC2)C1 11420,CN1CCCC1CCC(=O)Nc1cc(C(=O)NOCC(O)CO)on1 11421,c1(C2(C(N(C3CN(C(=O)CCc4cn(C)cn4)C3)C)=O)CC2)ncccc1F 11422,C1(C(C)C(=O)N(C2(C(=O)NC(C)C(=O)NC3CC3)CC2)C)CCC(=O)N1 11423,c1(OC)ncc(Cl)cc1C(=O)NC1CCN(C(=O)C(C)C(F)F)C1 11424,C#Cc1cccc(NC(c2cccc(C)c2C)C(F)(F)F)c1.c12ccccc1O2 11425,N1(C(C)=O)CCN(C(C2(F)CCN(C(C3CCC(=O)CC3)=O)C2)=O)CC1 11426,C#Cc1cc(C(=O)NC(Cc2cccnc2)CO)cc(C(F)(F)F)c1 11427,c1(NC(c2ccoc2)=O)ccsc1C(=O)NCCF 11428,c1(-n2c(C3C(c4ccc(C)cc4)CCC3)nc(CCN(C)C)n2)cc(Cl)ccc1C 11429,C=C(C)C1OCCC1C(N1CCC2(CC2NC(c2cccnn2)=O)C1)=O 11430,N1(C(c2cc(OC)ncc2)=O)CCC(C2CC2)(CNC(=O)CC2CC23CC3)C1 11431,c1(OCC)ccccc1NC(=O)C(N1CCC(C)(CNC(C2CC(C)C2)=O)C1)=O 11432,N1(C(CC2N(C)CC=CC2)=O)CC2(CCCC2NC(c2ccc(=N)[nH]n2)=O)C1 11433,c1(N(C)CC2(CN(C)C)CC2)ccc(S(=O)(=O)N(C2(C)CCOC2)C)cc1F 11434,C(=O)(C(CC)C(=O)OC)NCCN(C(c1nccc(CC)c1)=O)C(C)C 11435,CC1=C(C(=O)NCCN(C)C(C2CC2c2cnnn2C)=O)C(=O)OC1(C)C 11436,C1(C)(NC(C2(C(C)(C)OC)CC2)=O)CN(C(=O)Cc2cnc(C(C)C)o2)C1 11437,N1(C(COCc2c(C)ncs2)=O)CC2(NC(C3CCC(=O)N3)=O)CC1C2 11438,c1(C(CC)N(CC)CC2CCCN2C(c2cccc(CF)c2)=O)ccccc1F 11439,c1(CNC2CC(CC(=O)NCc3cccc(C(=O)OC)c3)C2)c(I)ccnc1Cl 11440,C1(C(=O)NCC(C2CCC2)OC)CN(C(=O)C(O)CSC)CCC1(C)C 11441,N1(C(COCCCOC)=O)CCOCC1CNC(c1conc1C(C)C)=O 11442,C12(C(=O)NC(CC(=O)NC(C)C)C)CCC(CN(C(=O)C(CO)N(C)C)C1)C2 11443,N1(C(C=CCCC=C(C)C)=O)CCOC(CNC(=O)C(C)(C)c2ccccc2)C1 11444,n1(C(C)C)cc(C(=O)NC2(CNC(c3cn(CC(F)(F)F)nn3)=O)CC2)nn1 11445,C12(C(=O)OC)CCC1(C(=O)OC)CN(C(=O)COC1CN(C(C)=O)C1)C2 11446,c1(SCC)ccc(CC(=O)NC(C)Cn2cc(-c3cnn(C)c3)nn2)cc1 11447,CCC(C)CC(C(=O)NCc1cccnc1)NC(c1cc(C(C)=O)[nH]n1)=O 11448,N1(C(=O)OC)CCC(CN2CCCC2)CC1.C=C1CC2(C1)C(=O)N2 11449,N1(C(CC2C(COC(C)=O)C2)=O)CCCC2(C1)CN(C(c1nccc(CC)c1)=O)C2 11450,C(C)(C)(CCCC(=O)N1CC(CC(C)C)C1)NC(c1cc(COC)on1)=O 11451,CCC(C(F)(F)F)NC(=O)C(=O)N(C1CCC1O)C 11452,N#CC1CCCCCN1C(c1[nH]nc(C(F)(F)F)c1[N+](=O)[O-])=O 11453,n1(COC)ccc(C(=O)NCC(C)N(C)C(C2CC2(F)F)=O)n1 11454,CC1CN(C(C2(C)CCCN2)=O)CCCN1C(c1cc(Cl)ccn1)=O 11455,C1(CNC(C=CCN(C)C(C2(C#N)CC2)=O)=O)CCC(F)C1 11456,C(=O)(C(C)(CC)C(F)F)NC(CN(C(c1coc(C)n1)=O)CC)C 11457,C12(CC3(CC3)C1)C(=O)NC2.Cc1ccc(C(C)C(=O)NC2(CN(C)C)CC2)o1 11458,Cc1cc(C(=O)NC2CCCC(NC(c3ccsn3)=O)C2)ncc1S(N)(=O)=O 11459,C1(CC)CC(C)CN1C(c1c(Br)ncn1C)C(=O)NC(C)C(=O)OC 11460,N1(C(c2cc(C)oc2)=O)CCC2(CC1)CC(C)N(C(c1ccc(CO)cn1)=O)C2 11461,C12(C(=O)NCC3(F)CCC(NC(=O)CN4CC=CC4)C3)CCCN(CC1)C2 11462,CC1(C)CCc2c1n[nH]c2C(=O)NC1CCSC12CN(C(=O)C1CC1)C2 11463,N1(C(Cn2cc(C(C)=O)nn2)=O)C2CCCC1CC(NC(=O)CC1CC13CC3)C2 11464,N1(C(CCC2CC(NC(c3c(NC)nccc3)=O)C2)=O)CC2CCC1C(CO)C2 11465,c1(C(N(C2CC2)CC2N(C(CCCCC)=O)CCC2)=O)cc2c(C)cccc2[nH]1 11466,Cc1nc(C#N)c(NCCC(=O)NC(C)C(C)NC(=O)CC2CCCCCC2)o1 11467,N1(C(C2(CC=C)CC2)=O)CCC(F)(C(=O)NC(c2nc(C)no2)CO)C1 11468,N1(C(C(CNC(c2cc(C(C)C)on2)=O)CC2CCCC2)=O)CCCCCC1C 11469,C1(NC(c2csc(C(F)F)c2)=O)CC(NC(c2ccc[nH]2)=O)C12CCC2 11470,c1(CC)cc(C(=O)N(CCn2cc(C(C)(C)N(C)C)nn2)CC)c(C)nn1 11471,CCC(CC)(CC(=O)OC)NC(c1ccc(Cl)cc1NC)=O 11472,N1(C(Cc2cccc(SCC)c2)=O)CCC(NC(=O)C2=COCCO2)C(F)C1 11473,c1(C(N(c2ccc(Br)cc2)C(C)C)=O)cc(Br)c2[nH]c(=N)sc2c1 11474,N1(C(C(C)SCC)=O)CCCCCC1CNC(=O)C1=CCOC1 11475,C1(C(N(C2CCCN(C(c3ccc(C(C)=O)o3)=O)C2)CC)=O)CC(=O)N(O)C1 11476,C1(C(=O)NCC(CCC)NC(c2cnns2)=O)(CC)CCOCC1 11477,C(=O)(C1Cc2ccccc21)NCC1N(C(CC=C=C)=O)CC1 11478,C1(C(=O)NC(C)CF)CN(C(c2cncc(N(C)C)c2)=O)CCC1(F)F 11479,N1(C(C2(CNC(c3ccc(NC)cn3)=O)CCCC2)=O)CCC2CN(C)CC12 11480,C1(OC)CN(C(=O)C=CC2CCCC2)CC1NC(C1CCN1S(C)(=O)=O)=O 11481,c1(CN(C(C2CC(CCNC(=O)CCCc3ncco3)C2)=O)CC)cccnc1 11482,c1(C(N2C3(CNC(C=C(C)C)=O)CCC2CC3)=O)ccc(Br)c(F)c1C 11483,C#Cc1ccc(C(=O)NC2(C(=O)NC(c3ncn(C)n3)C)CCSC2)cc1 11484,C1(COC)(CNC(c2nocc2C)=O)CCN(C(C2CCC(C)(C)C2)=O)C1 11485,C#Cc1ccc(C2CC2C(N2CCN(C(=O)C(C)CC(C)C)C(CC)C2)=O)cc1 11486,n1(CC)cnc(C(=O)NCC2CN(C(=O)C=Cc3cc[nH]c3)C2)n1 11487,C(=O)(C(F)C(C)(C)O)NCC(C)N(C(=O)CSCCC#N)CC 11488,C12(CNC(c3c(CC)nc(C)nc3)=O)CCCC(CN1C(=O)CS(C)(=O)=O)C2 11489,c1(C(=O)OC)sc(C(N2CC=CC(NC(C3(OC)CCCOC3)=O)C2)=O)cc1N 11490,Cc1cc(Br)cc(C)c1NNC(=O)Cc1ccnc(F)c1F 11491,c1(C(N(CCCCCNC(C(n2ncc(C)c2)C)=O)C)=O)cncc(C)c1O 11492,Cc1cccc(F)c1C(N1CCC(C)(CNC(=O)CC(F)(F)Cl)CC1)=O 11493,N1(C(CC(C)(C)O)=O)CCC(NC(=O)CCNC(=O)CO)C(F)C1 11494,C1(C(N(CCOC)CCNC(c2coc(COC)n2)=O)=O)CC2OC(C)(C)OC2C1 11495,N(C1CCc2cccnc21)C(C(C1CCCO1)NC(CSCC=C)=O)=O 11496,c1(CC)cc(C(=O)N(CCCNC(=O)CC2CCC(C)C2)C)no1 11497,S(=O)(=O)(c1ccc(N(C)CCC2CC2)cc1Br)N(C(C)CN)C 11498,C1(C(=O)NCC(F)(F)F)(NC(C2CN(C)C2)=O)CCCC1 11499,C1(CNC(CN(CCCCCC)C)=O)CCCC(NC(=O)CS(N)(=O)=O)C1 11500,c1(CC(=O)NCC2CC2NC(=O)C2=NOCC2)cccc(F)c1 11501,c1(OC)cc(C(=O)N(CCC(C)NC(=O)C(O)Cc2cn(C)cn2)C)[nH]n1 11502,c1(C(N2C(C(=O)Nc3ccc(F)c(I)c3)CNCC2)=O)cc(O)c(Br)c(O)c1 11503,CCCCC(CNC(=O)CC1CSC1)NC(c1n[nH]c(C)c1Cl)=O 11504,c1(OC)c(F)cc(CN2CC3(CNC(=O)OC(C)(C)C)CC2CO3)cc1F 11505,C1(N2CCN(CCOC)CC2)COC2(CCN(C(C3CCCO3)=O)CC2)C1 11506,N1(C(CC(=O)OCC)=O)CCC2(C=C(C(=O)N3CCOC(C)CC3)C2)C1 11507,C1(N=[N+]=[N-])(C(=O)NC(C(C)SC)C)CCN(C(c2oc(C)nc2C)=O)C1 11508,C1(NC(CC(CNC(C(c2ccn(C)c2)C)=O)O)=O)CCCCCCC1O 11509,c1(CC)nc(C)c(C(=O)NCCN(C(=O)C(C)C2CCC2)Cc2ccccc2)s1 11510,C1(CC)CC(C(=O)NC(CNC(=O)CC2CCOCC2)C(C)(C)C)CCO1 11511,Cc1ncc(C(N2CC(CNC(c3cccc(Cl)c3)=O)CC2C)=O)cc1Cl 11512,N1(C(c2ccnc(OC)n2)=O)CCCC2C1CCCN2C(c1cc(C)n(C)c1)=O 11513,CCCC(CCC)C(C)NS(=O)(=O)Cc1ccc(F)cc1Cl 11514,N1(C(CC=C)=O)CCCC(O)(CCNC(c2cc(CN(C)CCC)c[nH]2)=O)C1 11515,c1(C(=O)NCCCCSC)occc1CNC(=O)C=CC(C)(C)C 11516,C1(C)(C(=O)NCC2C(C(N(CC(=O)NC(C)C)C)=O)CCO2)CCC(=O)CC1 11517,N1(CCC)CC(C(=O)NCCCCCCNC(c2ccsc2C)=O)CC1=O 11518,CC1CN(C(C2CC2C(F)F)=O)CC1NC(C1CCC(N2CCCC2=O)CC1)=O 11519,C(=O)(CC1=CCOCC1)NC1(CO)CCN(C(C(C)Cc2cccnc2)=O)C1 11520,C(C)(CCCCNC1CCCC1(F)F)N(C(=O)OC(C)C)C(c1ccnn1C)=O 11521,N1(Cc2nccc(C)c2)CC(C(=O)Nc2ncc(CO)cc2Br)CC(F)C1 11522,CN1N=C(CC(=O)N2CCCCC(N(C)C(C3CC4(CCCO4)C3)=O)C2)CC1=O 11523,N1(C(c2cc(CC)ncc2)=O)CCCC(F)(C(=O)NCC(C)OCCOC)C1 11524,CC(C(C)(C)NC(c1ccnn1CCF)=O)NC(c1cnn(C(F)(F)F)c1)=O 11525,C(CC1=CCN(C(=O)C(N2CCCCCC2)C)CC1)NC(C=CC=CCC)=O 11526,C1(CNC(CC2CCC(=O)NC2)=O)(NC(C2CC2C(F)F)=O)CC2CCC1CC2 11527,c1(CC(=O)NCC2C(C)CCCN2C(c2ccoc2)=O)c[nH]c2cnccc12 11528,N1(C(c2c(C)scc2)=O)CC2CC2(NC(=O)CCc2cncc(O)c2)C1 11529,C1(CNC(c2nc(CC)[nH]n2)=O)CCC(CNC(=O)CCc2cccs2)CC1 11530,C12(C(N(C)CC3CCN(C(C4C(C)(C)OC4(C)C)=O)C3)=O)CCCC(C)(C1)OC2 11531,C1(O)(C(=O)NCC2C3CN(c4nccc(C(C)=O)n4)CC32)CCCC(C)(C)CC1 11532,O(NC(=O)CC1(CNC(=O)COC(C)C)CC1)CC(C)C 11533,Cc1cn2c(CC(=O)NC(C)C(C)(C)NC(C3CCCCC(=O)N3)=O)csc2n1 11534,N1(C(c2ccc(CC)nc2)=O)CCCC(NC(=O)C(C)NC(C)(C)CC)C1CC 11535,c1(-n2c(-c3cc(SCC)c(O)cc3)nc(CSC)n2)cnnc2ccccc12 11536,Cc1ccc2ccccc2c1NCC1CC(O)(CO)C1 11537,C1(NC(C2CN(C(C)=O)C2)=O)CN(C(C2(C)CC2(C)C)=O)CC1c1ccnn1C 11538,c1(C(=O)NCCC2CSCCN2C(=O)CC2CCOC2)cccc(C2CC2)c1F 11539,c1(C(=O)Nc2c(C)nc(C#N)cc2)n[nH]c2cc(CNC=O)ccc12.C(C)(C)C 11540,Cc1ccnc(C)c1CNC(c1coc(CNC(C2CC(F)C2)=O)c1)=O 11541,C(C(C)CC(=O)NC1CC(NC(c2coc(-c3ccccc3C)n2)=O)C1)OC 11542,c1(C(=O)OCCC2CCCCC2)cccc(N2CCOCC2)c1 11543,N1(C(C=CC=CCC)=O)CCC(C(F)CNC(C2CC2[N+](=O)[O-])=O)CC1 11544,c1(C(=O)NCC(CCCC)NC(=O)C(F)C2CCC2)cnc2c(C)cccc2c1 11545,N1(C(Cc2nc(C)[nH]n2)=O)CCC2CCCC12CNC(c1ccc(F)s1)=O 11546,N1(C(c2cc[nH]c(=N)c2Cl)=O)C2CCC1c1ccccc12 11547,C1(F)(C(N(CCO)CC)=O)CCN(C(=O)C(C2(O)CCCC2)F)C1 11548,C(=O)(NNc1cc(Cl)nc(N(c2cc(Cl)nc(Cl)c2)C(C)=O)n1)OC(C)(C)C 11549,C1(NC(C2CCCCC2)=O)CC2(C1)CC(NCc1cc(Cl)c(Cl)cn1)C2 11550,N1(c2cc(C)[nH]c(=NCC3CN4CCN3CC4)n2)CC2(C)CN(C)CC2(C)C1 11551,C1(CN(C)C(c2cnc(O)n2C)=O)CCC(NC(c2ncoc2Br)=O)CC1 11552,C1(NC(c2cccc(OC(F)F)c2)=O)CCN(C(C23C=CC(CC2)C3)=O)CC1 11553,C1(SCC)COCCC1NC(=O)N(C)CCN(C)Cc1ccccc1C 11554,N1(C(C=CC)=O)C(CNC(=O)C(c2ccc(Br)cc2)OC)CC2CCCC12 11555,C#Cc1cc(F)c(C(=O)NC(C(C)NC(=O)CC(=O)NCC)C(C)C)cc1F 11556,C(=O)(C1CCCc2ncccc21)NCC(C(C)C)(C)NC(=O)C#CC(C)(C)C 11557,Cc1cncc(-n2cc(CONC(C3C(C)=NOC3C)=O)nn2)c1 11558,C(C(CC(=O)NCC1CCC1NC(c1cccc(=O)o1)=O)CC(C)C)NC(C)=O 11559,Cc1ccc(C(=O)NC2(CO)CCN(C(=O)C(C)(O)C3CC3)C2)cc1Cl 11560,C1(NC(CCCC(=C)C)=O)(CNC(=O)CCC2CCC2)CC2CCC1CC2 11561,c1(OC)cc(C(=O)NCCCNC(=O)CSC(C)(C)C)c(F)cn1 11562,N1(Cc2cn(CC)nc2)CCCC2(CCN(C(c3cc([N+](=O)[O-])cs3)=O)C2)C1 11563,C(C)(C(CC(=O)NCC1CC(SC)C1)NC(=O)C(C)NC=O)OC 11564,C12(CNC(c3cn(CC4CCCO4)nn3)=O)CCCC1N(C(C1COC1)=O)CC2 11565,c1(NC(C(C2CCN(C(c3cccc(F)c3O)=O)CC2)C)=O)nc(Cl)ccc1O 11566,CC1(C2(C)CC2NCc2cc(Cl)nc(Cl)c2)CC1 11567,C12(NC(=O)CC=CCNC(=O)C(O)c3ccsc3)CC(CO)(C1)C2 11568,CC(C)(CCNC(C1CNC(=O)N1)=O)NC(=O)CCCc1ncco1 11569,c1(C(N2C(CNC(c3cnc[nH]3)=O)CCCC2)=O)cc2ccc(Cl)cc2c(=O)o1 11570,C1(CNC(C23CC(C2)C(C(F)(F)F)O3)=O)CC2(CCC2)CN1C(=O)C1=COCCC1 11571,C(=O)(CCCCCNCc1ccccc1)N(C1CC2CC2C1)C(C)(C)CO 11572,c1(NCc2n(C)c(Br)nn2)[nH]c(=NCC(Cl)(Cl)Cl)nc2c1cnn2C 11573,Cc1nn(C)c(C(=O)NCC(C)NC(C2CC2c2cnn(CCN(C)C)c2)=O)c1Cl 11574,N1(C(C(COCC)n2cc(CN(C)CCOC)nn2)=O)CCC(C(C)=O)CC1 11575,c1(OC)cnc(CNCCN(C2CCCC2)C(=O)C=Cc2ncc[nH]2)nc1 11576,c1(C(N2CC(NC(CCCOCCC)=O)C(OC)C2)=O)cc(=O)cc(Cl)[nH]1 11577,c1(OC)nccc(C(N2CCN(C(=O)C(Cl)=CCl)C(CS(C)(=O)=O)C2)=O)c1F 11578,CC(C)CC(C(=O)N1CCCC1Cc1ccccc1)NC=O 11579,c1(CC(C)C)c(C(=O)N(C2CCC(NC(C34CCC3CC4)=O)C2)C)cnn1C 11580,N1(C(C(C)SCC)=O)CCC2CN(C(c3cnc(C)o3)=O)CC2C1 11581,Cn1nc(Cl)cc1C(=O)NCC1(CNC(C2CC(F)C2)=O)CCCCC1 11582,C1(C)(NC(CC(C)C)=O)CCCN(C(=O)C(O)CN2CCCC2)C1 11583,c1(C(=O)NCCC(C)NC(C2CCCC(=O)CC2)=O)c[nH]cc(Cl)c1=O 11584,Cc1ccc(C(N2CCC(NC(c3ccncc3)=O)CC2C)=O)cc1OC(F)F 11585,CC1(C)CC(=O)OC1CNC(C1C=CCN(C(C2CCSCC2)=O)C1)=O 11586,C(CC(O)CC(=O)NC1C=CCN(C(=O)C(C(C)C)NC(N)=O)C1)SC 11587,c1(C(=O)NC2CC3CN(C(C4(C)CC4(F)F)=O)C2C3)ccc(Cl)c2ncccc12 11588,C1(C(=O)NC2C(O)CCN(C(CCNC(=O)NC)=O)C2)CC2CCCCCC12 11589,CCC(C(=O)NC1(C)CC(NC(=O)CCC2CCCOC2)C1)N(CC)CC 11590,Cc1[nH]c(C(=O)NCc2ccc(F)cc2F)c(C)c1C(=O)NCC1CCCN1C 11591,N1(C(CC2(C)CC2)=O)CC(C)(C)OCC1CNC(=O)Cc1sccc1C(=O)CO 11592,N1(c2c(Br)cnc(C)n2)CCC2C1CCCN2C(c1c(Cl)cccc1Cl)=O 11593,c1(CC)ncc(C(=O)NCC2CC(F)(F)CN2C(=O)CN2CC3CC3C2)c(O)n1 11594,N1(C(C=CCNC(C2CCOC2C2CC2)=O)=O)CCCC2CCCCC12 11595,N1(C(c2ccc([Si](C)(C)C)s2)C(=O)NCCCC)CCC2(C1)NC(=O)N(C)C2=O 11596,c1(SC)ccc(CC(=O)NCCCC2CCN(C(C3CCC(=O)N3)=O)CC2)cc1 11597,C1(CC(N2CC(CCNC(c3[nH]c(C)nc3C)=O)(OC)C2)=O)CCCNC(=O)C1 11598,Nc1cc(Cl)nc(Cl)c1C(N1CC2(COC(CNC(=O)Cc3cnoc3)C2)C1)=O 11599,Cc1ccc(C=CC(=O)NC(C2(O)CN(C(C3(C)CC3(C)C)=O)C2)C)cc1Cl 11600,C1(O)(CNC(CC(CC)c2ccccc2)=O)CCN(C(c2ccc(=N)[nH]n2)=O)CC1 11601,C(=O)(C1CCc2ccccc21)N1CC2C(NC(C(CC=C)OC)=O)(CCC2)C1 11602,C(=O)(CCCCN1CCOCC1)N(C(CNC(C(CC)O)=O)C1CC1)C 11603,c1(CNC(c2nnnn2C2CCC2)C2(OC)CC2)cc(Cl)nc(Cl)c1 11604,C1(NC(c2nnnn2C2CC2)(CSC)C)CCc2nncn2C1 11605,C1(CC=C)(C(=O)NC(C)CCC(=O)OC)CCN(C(=O)CSC(F)(F)F)C1 11606,C1(SCC)CCc2nc(NC(N3CCCC3C(=O)NCC)=O)sc2C1 11607,N1(C(c2[nH]c(=NC)sc2)=O)CCC2CC2(NC(=O)CC2CCOCC2)CC1 11608,CCC(CC)C(=O)NCC(C)NC(c1cnn(C(C)(C)C)c1C(F)(F)F)=O 11609,C(CC)(CC(C)CC)(c1n(CC(=C)C)nnn1)Nc1cc(SC(F)F)ccc1C 11610,c1(C(=O)NC2CC(NC(c3c[nH]c(=NC)s3)=O)C2)cccc(S(=O)(=O)C(F)F)c1 11611,C1(C)(NC(C=CC(C)NC(COC)=O)=O)CCC(C)=C(C)C1 11612,O=C(CCCCCCCCCO)NC1(CO)CCN(C(C2CCC(O)C2)=O)CC1 11613,c1(CC(=O)NC(C(C)NC(c2c(COC)nn[nH]2)=O)C)ccc(F)cc1 11614,C(CCCCCCCCCCCO)NC(C1C(NC(c2cccs2)=O)C1)=O 11615,C=CC1CN(C(c2n[nH]c(C)c2C)=O)CC1NC(c1ncoc1C1CC1)=O 11616,c1(C(=O)NC2(CCCNC(C(C)n3cnnn3)=O)CC2)ccc(Br)nc1N 11617,N1(S(CC)(=O)=O)CCC(C(=O)NC(C)CCN(C(=O)CN(C)C(C)=O)C)CC1 11618,N#CC1(CC(N2CCCCCC2CNC(=O)C(F)n2cccn2)=O)CCOCC1 11619,CC1(C)CN(C(=O)NC2(c3ccc(F)cc3F)CCCC2)C12CCOCC2 11620,C(CN(C)N1CCC(NC(=O)OC(C)(C)C)CC1)N(C)C(c1ccco1)=O 11621,c1(C(N2CCC(C)(C(N3CCC(CF)CC3)=O)C2)=O)ccc(Br)cc1S(C)(=O)=O 11622,N1(C(c2cc(C(C)(C)C)no2)=O)C2CCC1C(NC(c1ccc[nH]1)=O)C2 11623,c1(C2C(C(N(CC(C)CNC(=O)Cn3ncnn3)C)=O)C2)ccc(Cl)cc1Cl 11624,c1(CSCC(=O)N(C(C)CNC(C2CCO2)=O)C)ccc(Cl)s1 11625,O=C1Nc2ccccc2CC1CC(N1CC2CCCC2C12CC2)=O 11626,C(=O)(C(F)C(F)(F)F)N(CCNC(=O)COC1(C)CCCC1)CC 11627,CC(C)CCCCCC(=O)N1CC2CC1C2NC(c1cncc(CN(C)C)c1)=O 11628,C(=O)(CCCCCn1cnnn1)NC(C)(C)CCCNC(=O)CCC1CC1(C)C 11629,c1(C(N2C(C(C)NC(c3cn(CC=C)nc3)=O)CCC2)=O)cc(Cl)ccc1OC 11630,C(=O)(CC1=CCN(C(C2CC2C2CCC2)=O)CC1)NC1(CCC=C)CC1 11631,CCCCC(O)CC(=O)NCC1CN(C(=O)CNC(N)=O)CCCO1 11632,c1(CNC(C(C)=CC(C)(C)C)=O)cncc(C(=O)NC2(C(C)O)CC2)c1 11633,c1(C(=O)NC2CCCC(NC(C(C)(C)O)=O)C2)cnc(O)c2cnccc12 11634,CC12CC(C(=O)NC3CN(C(c4ccc5cnnn5c4)=O)CC3F)(C1)C(C)(C)O2 11635,CCC(O)C(F)(F)C(=O)N(CC(C)(C)Nc1ncnc2[nH]ccc12)C 11636,C(=O)(C1CCc2c(Cl)cccc21)NC1CC(CCNC(c2cc(=N)[nH]cc2)=O)C1 11637,c1(NC(=O)NCC2(NC(Cc3c(C)cc(C)s3)=O)CC2)cc2c(Cl)cccn2n1 11638,CCC(C(=O)Nc1ccc(N2CCC(C)CC2=O)cc1)C(C)(C)CC.C(C)(=O)OC 11639,c1(OC)cccc(F)c1CNC(=O)NCc1ccc(-n2cncn2)cc1 11640,N1(c2nnc(C(C)C)n2CCC#N)CCC(C2CCCCC2)C1 11641,C1(C(N(C)CC2(OC)CCC2)=O)CCC(C)N1C(=O)COc1cccnc1 11642,N1(C(c2c(C)coc2)=O)CC(NC(=O)C(F)(F)c2ccccc2)C(O)C1 11643,N1(C(=O)Nc2c(C)ncc(C)c2)CCC2(CC1)OC(C)(C)NC2=O 11644,C(=O)(CC(C)C(F)(F)F)N1CCC(N(C(=O)Cc2ncsc2Cl)CCC)CC1 11645,c1(C(=O)NC(CC(C)Nc2ncnc(Cl)c2F)C)cc2ccoc2cc1F 11646,C(N=c1cc[nH]c(=NCCCC2CCOC2)[nH]1)c1cnc(C)s1 11647,c1(OC)cc(C)cc(C(=O)NCCOCCNC(C2(S(N)(=O)=O)CCCC2)=O)c1O 11648,C(=O)(CC(=O)NCCCN(C(=O)Cc1cnn(C)n1)C)OCC 11649,Cc1nc(C)c(C(N2CCN(C3CCCN(C(=O)C=CC(N)=O)C3)CC2)=O)[nH]1 11650,C1(NC(C(CO)OC)=O)CCOC(CNC(c2ccc(C(F)F)cc2)=O)C1 11651,C(CC1=CCN(C(C2CCCC23CCC3)=O)CC1)NC(C1CCC2CC2C1)=O 11652,N1(C(CC2(C)CC2F)=O)CC2(CCN(C(c3cc(=N)[nH]cc3Br)=O)C2)C1 11653,N1(c2ncc(CC)cn2)CCC2CC1(c1noc(COC(=O)NC(C)(C)C)n1)C2 11654,N1(Cc2cnc(C)nc2)CCN(C(c2cccc(C(F)(F)F)c2)=O)CC1C 11655,Cc1sc(Cl)c(C(N2CCN(C)C(CNC(=O)C(c3cccnc3)O)C2)=O)c1C 11656,CCC(C)(C(=O)NCCC(Cc1ccccc1)NC(=O)C(CCSC)SC)OC 11657,N(C1CCNc2ccccc21)C(=O)CC1CCc2ccccc2C1 11658,c1(CC(=O)NC2(CO)CCN(C(C=C3CCC(C)C3)=O)C2)cccc(Cl)c1F 11659,Cc1ccc(=N)[nH]c1C(=O)NCC(CO)NC(=O)CCn1cncn1 11660,C(CC(=O)NC(C)C(=O)OC(C)C)(CC(C)C)NC(CC1ON=C(CC)C1)=O 11661,C(=O)(CC(F)(F)C(C)C)NCC(CNC(C(COCC)C)=O)CO 11662,CP(C)(=O)c1cc(F)ccc1NC(C1C(Cl)(Cl)C12CC2)=O 11663,c1(C(N(CCCN(C(CC2(COC)CCCC2)=O)C)C)=O)ccc(C)n(C)c1=O 11664,C(CCN=C(NC1CSC1(C)C)N1CCC(CC(C)C)CC1)SC 11665,C(=O)(C(C)C(=O)N1CCOCC1)N1C(COC(c2cnc(OC)s2)=O)CC1 11666,CC(C)C(C(=O)N(CC(O)CN(C(=O)C(C)Cc1ccccc1)C)C)NC(N)=O 11667,C1(C(=O)NCC2OCCCN(C(c3cc(C)sc3C)=O)C2)CCc2cnnn2C1 11668,c1(C(n2cccn2)CNC(N(C)CC2CCC2)=S)ccc(Br)cc1 11669,C1(C(=O)OCC)CC2(CC(NC(C3CCCN(CC(F)F)C3)C)C2)C1 11670,N1(C(Cc2ccc(C)o2)=O)CC2CC(NC(C3CC3CF)=O)CC(C2)C1 11671,c1(CC)cccc(CNC(=O)NC(c2cc(Br)ncc2F)C)c1C 11672,c1(C(=O)NC2CN(C(C3(C)CCOC3)=O)CC2F)ccc(F)c(O)c1 11673,N1(CCNC(C(COC(C)C)(C)C)=O)CCCN(C(C2COCCN2C)=O)CC1 11674,c1(NC(N(C)Cc2ccc(C(C)(C)OC(F)F)cc2)=O)ccc(OC(F)F)c(F)c1 11675,C1(CNC(CC2(C(C)NC(=O)C=C3CCCCC3)CC2)=O)CC12CCOCC2 11676,c1(C(=O)NC(c2cn(C)nn2)C(=O)N(CC(F)Br)C)ncc(F)cn1 11677,N#Cc1ccc(F)c(CNC(=NCCCF)NCc2cnccn2)c1 11678,CCC(C(=O)NC1(CO)CN(C(C2CC2c2ccncc2)=O)C1)C(C)O 11679,c1(OC)ccc2c(c1C(=O)NC1CN(C(=O)CC=C(C)C)CC(C)(C)C1)CCC2 11680,C(=O)(C(O)CC(=O)OC(C)(C)C)NCC(CN(C(CC(=C)C)=O)C)O 11681,C(C(C(=O)N1CC(NC(=O)C=CCN2CCCC2)C1)OC)OC 11682,C1(Cc2cn(C3(C(C)(C)C)CC3)nn2)COCCN1C(=O)COC1CCCCC1 11683,C(CC(C)P(C)(C)=O)NCc1nc(C(=O)OCC)nn1C 11684,C=CCC(C(=C)C)C(=O)N1CC2C(NC(c3cc(F)c(Cl)cc3F)=O)C2C1 11685,C=CC(C)CC(=O)N1CCCC1C1(NC(c2csc(C(C)(C)C)c2)=O)CC1 11686,C#CCC(C)(C(=O)NC1CCCCC1CO)NC(=O)CCOC1COC1 11687,c1(C(=O)NC(C(C)NC(c2cc(CCC)[nH]n2)=O)(C)C)c[nH]c2cc(F)ccc12 11688,N1(C(c2cc(C)nn2C(F)F)=O)CC2CCN(Cc3cccnc3C(=O)O)C2C1 11689,N1(C(c2cc(C)c(F)cn2)=O)CC(C(=O)NC(C2(O)CCC2)(C)C)CCC1(C)C 11690,C=CCCC(CO)NC(=O)CCCNC(=O)CC(C)N(C)C 11691,c1(-c2ccc(CC)s2)ccc(CNC(C2(CC)CCOCC2)=O)cc1 11692,c1(C(=O)NCC(CCCC)NC(C2(C(C)C)CCCO2)=O)nsc2ccccc12 11693,Cc1ccccc1C(=O)NC1(CF)CCN(C(=O)Cc2cccs2)C1 11694,C1(O)(C(N(CCCN(C(C2(C)CC(=C)C2)=O)C)C)=O)CCCC(C)(C)CC1 11695,N1(C(c2c(CC)noc2)=O)CC2(CCCC2NC(=O)C(c2ccccc2)C)C1 11696,CCCC(CC(=O)NCc1ccc(CO)o1)NC(c1c[nH]c(C#N)c1C)=O 11697,c1(C(N2CCN(C(C(CC)SC)=O)CC2CF)=O)coc2c(F)cccc12 11698,C=CCCC(C(=O)NC1(C)CC2CCC1C2)NC(=O)C(O)CC 11699,Cc1n[nH]c(C)c1CC(N1CC2C(NC(c3ccncc3O)=O)C2C1)=O 11700,Cc1cc(F)ccc1C(=O)NC1(C)CCOC1C 11701,CN=c1nc(C(=O)NC2CCN(C(=O)CCC(C)(C)OC)C(C)C2)cc(C)[nH]1 11702,Cc1ccn2nc(C(N3CCCC3CN3CCC(OC(C)C)CC3)=O)nc2n1 11703,C(C(=O)N(C)CCOCCN(C)C(c1cccc(C(F)(F)F)c1)=O)(C(C)C)SC 11704,N1(C(C2(CC)CCC2)=O)CC(C(=O)NOCCNC(=O)NCC(C)C)C(O)C1 11705,C=CCC(CNC(c1cnc[nH]1)=O)NC(=O)CC1COCC1O 11706,N1(C(c2ccc(C)cc2N)=O)CC2CC(C)N(C(=O)CC3CC(F)C3)C2C1 11707,C1(C(N2C(CC(=O)NCCC(C)OC)CCCC2)=O)CC(C)(C)CN1C 11708,C1(NC(Cc2cn(C(C)(C)C)nc2)=O)CC(NC(=O)C2=CCC2)C(O)C1 11709,C1(C(=O)NCC(C2CCCCC2)C)CCN(C(=O)CCC2CC2(C)C)C1 11710,Cc1ccc(OCCC(=O)NCCCCN(C)C(C2CCCS2(=O)=O)=O)cc1C 11711,CN1CCOC2CN(C(C3CC4CN(C(c5ccn(CF)n5)=O)CC4C3)=O)CC12 11712,c1(OCC=C(C)C)ccc(CNC(=O)Nc2n[nH]c(=N)o2)cc1 11713,CCC(C)(C#N)C(=O)NCCCN(C(=O)CSCC(N)=O)CCO 11714,CC(CC(=O)NCC1CCC1NC(=O)C=CSCc1ccco1)C(F)(F)F 11715,c1(C(C)F)ccc(C(=O)NCCC(C)NC(=O)CC=CCc2ccccc2)cc1 11716,C1(F)(C(=O)NC(CC(=O)OC)C)CCN(C(c2ccnn2C(F)F)=O)C1 11717,c1(CC)nn(C)c(C(=O)NC2CCN(C(c3cnc(O)n3C)=O)CC2O)c1Cl 11718,C(=O)(C1CNC(=O)c2ccccc21)OCC(=O)NCc1ccc(F)c2cccnc12 11719,N1(C(C(C(C)(C)C)n2ccnn2)=O)CCCC(NC(=O)CC(F)(F)F)CCC1 11720,N1(C(=O)Nc2cccc(OC)c2)CCC2(CCc3ccccc32)C1 11721,CCS(=O)c1ccccc1CC(=O)NCC(OC)OC 11722,C1(C2N(C(c3c(C)cc[nH]3)=O)CCC2)CCN(C(C2CN(S(C)(=O)=O)C2)=O)CC1 11723,C1(C(N)=O)(C(c2ccccc2)NC(C(C)SC(C)C)=O)CN(C(C2CC23CC3)=O)C1 11724,c1(OCC)cccc(C(C2CCCC2)CCNCCCc2n[nH]c(C)n2)c1 11725,N1(C(Cn2c(C)cc(C)n2)=O)CCC2C(C1)CN2C(C12CC(C)C1C2)=O 11726,N1(C(C(CN(C(CN(CCOC)C)=O)C)C)=O)CCCC2OCCC2C1 11727,c1(CC)ccc2[nH]c(C(=O)NCCNc3cc(C)nc4ncnn34)c(C)c2c1 11728,N1(CC(=C(Cl)c2ccccc2F)C)c2ccc(Cl)cc2NC(=O)C1C 11729,N1(C(C2CC(CCNC(C3CC4(CCC4O)C3)=O)C2)=O)CCOCC2(CC2)C1 11730,c1(SC)c(C(N2CCC(NC(C3CCC(C)(C)O3)=O)C2C)=O)cnn1C 11731,c1(CNC(C(C2(O)CCC2)NC(c2ccc(CO)s2)=O)=O)ccc(O)nc1 11732,CC1CC(O)CCN(C(=O)C(C)N(C(c2cccc[n+]2[O-])=O)C2CC2)C1 11733,C12(C(CNC(c3n(CC)nnc3)=O)NC(c3ccc(CO)o3)=O)CCC(CC1)C2 11734,C1(NC(Cc2nc(C)sc2)=O)C2CC1N(C(C1(Sc3ccccc3)CC1)=O)C2C 11735,C1(C(N(CC(CNC(C(=Cc2cnc[nH]2)C)=O)(C)C)C)=O)CC2(C1)CC1(CC1)C2 11736,C1(C(N(C2(C(=O)NCc3nc(CC)[nH]n3)CC2)C)=O)CCC(C2CC2)C1 11737,c1(NC(c2n(CC)nnn2)C23CCCC2C3)ccc(OC(C)C)cc1 11738,CC1(C)CC(C(N2CCC(C(N)=O)C2)=O)CN1C(c1cccc(CC#N)c1)=O 11739,C(=O)(C(C)CC(C)(F)F)NC(CC(C)C)(C)CNC(=O)C(F)(F)c1cscn1 11740,CC1CCOC1CNC(c1sccc1CNC(=O)CC1COC(=O)C1)=O 11741,c1(CC(=O)NC2C3(NC(c4cc(C)ns4)=O)CCC(C2)C3)ccc2sccc2c1 11742,C(=O)(CCCCCO)NCC12N(C(C3C(OC)CCC3)=O)CC(C1)C2 11743,c1(C(N2C(C)C(C)N(C(c3ccc(Cl)cn3)=O)CC2)=O)ccc2nn[nH]c2c1O 11744,C1(C(=O)OCC)CCCC(Nc2c(C(N3CC(CC(C)(C)OC)C3)=O)scc2)C1 11745,c1(NC(CC)=O)cc(C(=O)Nc2cc(SC)ncn2)c(F)cc1F 11746,c1(-c2cn(CC(C)NC(C3CC(C)OC3=O)=O)nn2)ccc(N)c(Cl)c1 11747,CN1CCN(CC(=O)N(CCCNC(=O)COc2ccc(Cl)cc2)C)CC1 11748,c1(SC)cc(C(=O)NCCN(CC(C)O)C(c2ccn(CCOC)n2)=O)co1 11749,C1(C2CCC2)(C(=O)NCC2CCCCN2C(=O)COCC2CCCOC2)CC1 11750,C(CCCCC(=O)N1CCCC1)NC(CN(C(C(C)n1cccc1)=O)C)=O 11751,N1(C(C(c2ccc(F)cc2)CC)=O)CC2C(CNC(c3cnn(CC)c3)=O)C2C1 11752,N1(C(C(CC)OC)=O)CCCCC1C(C)(C)CNC(C1(OC)CCOCC1)=O 11753,C(=O)(C(C(C)C)NC(c1cc[nH]n1)=O)Nc1c(C)scc1 11754,C=C=CC(C)C(=O)NCC1CCCCN1C(c1n[nH]cc1-c1ccccc1)=O 11755,c1(C(N2C(CNC(C(CCN(C)C)O)=O)CCC2)=O)c[nH]c2cccnc2c1=O 11756,N1(C(c2ccc(C#C)c(F)c2)=O)CC(CO)C2(C1)CN(C(=O)C(O)C1CCC1)C2 11757,Cc1ccc2cc(C(=O)NC(C)Cc3cc(Br)ccc3F)cnc2c1 11758,CC(C)(C)CN(CCO)C(C1(CNC(=O)CC2CC=CC2)CC1)=O 11759,C(=O)(CCC(O)C(C)(C)C)N1CCC(CN(C)C(c2cn(CCO)nn2)=O)CC1 11760,N1(C(COCCC#C)=O)CCN(C(c2nnc(C)cc2O)=O)C2CCCCC2C1 11761,c1(CC)nc(=N)[nH]cc1C(N1CCCCCC1CNC(C1CNC(=O)N1C)=O)=O 11762,N1(C(c2c(CC)cncc2)=O)CCCC(C)(NC(=O)CC2COC(C)(C)C2)C1 11763,c1(CC(N2CC(NC(C3C(C(C)C)CCO3)=O)C2)=O)cc2ccccc2cc1O 11764,CC(C)CCCC(C)C(=O)N1CCC(CC(=O)NCCC2(CO)CC2)C1 11765,N1(C(CCSCC)=O)CCC(NC(C23CCC(CC2)CO3)=O)C(F)C1 11766,C1(CC(=O)NC(c2c(C)ncs2)C)CCN(C(c2n[nH]c(C)c2C)=O)C1(C)C 11767,C(c1ccncc1)=C(C)C(=O)N(C1CCCN(C(C2C(C)C2(F)F)=O)C1)C 11768,c1(-c2cn(C)nc2)ccc(CNc2ncccc2NS(N)(=O)=O)c(F)c1 11769,c1(C(=O)NCC2=CCN(C(C3CC3F)=O)CC2)cc(F)cc2nc[nH]c12 11770,c1(OC)ncnc(C)c1C(=O)NCC1CN(C(C2(OC)CCCC2)=O)CC1C 11771,C12(C(=O)NC3COCCN(C(=O)CC4CSC4)C3)CC=CCN1CCC2 11772,C1(C(=O)N(C)C)CCN(CCNC2CC(NC(CCSC)=O)CC2O)CC1 11773,c1(C(=O)NCC=CCNC(=O)C=CC=C(Cl)Cl)cccc(CF)c1 11774,C1(C(=O)N(C)CC2(CNC(c3ccc[n+]([O-])c3)=O)CC2)(OC)CCC(C)C1 11775,C1(C(=O)NC2CC(CNC(c3c(C)ncs3)=O)CC2O)CC12CCS(=O)(=O)CC2 11776,CC(C)CC(CO)NC(C1C(CO)CCN1C(=O)CC1(CSC2CC2)CC1)=O 11777,O(NC(=O)C(COCC)NC(=O)CCC1CCOCC1)CC(CC)C 11778,c1(C(=O)NC23CC(NC(c4cccnn4)=O)(C2)C3)ccc(=O)n2c1COCC2 11779,N1(C(CCN(C)C)=O)CC(C(=O)N(C2CCSC2)C)C(F)(F)C1 11780,Cc1ccc(C(=O)NCC(C)CC(=O)NC(c2ncccc2F)C)cc1O 11781,C(CC(=O)N1CCC(CNC(c2nc(Cl)c(Cl)s2)=O)C1)(C(F)(F)F)OC 11782,CC(C(O)C(F)F)NC(C1(NC(=O)CCOCCN(C)C)CCCC1)=O 11783,c1(OC)ccc(S(=O)(=O)N2CCC(CNC(=O)CC3CCCC3)C2)c(F)c1 11784,N1(C(CC(C)(C)OC)=O)CC2(CCC(CNC(=O)C(C)(C)c3cc[nH]n3)O2)C1 11785,C1(NC(C=C(C)I)=O)CN(C(c2c(C)ccn2C)=O)CC1O 11786,N1(C(CCC2(C#N)CCC2)=O)CC2(CCN2C(C2CC(C3CC3)=NO2)=O)C1 11787,N1(C(C(CC)C(=O)OC)=O)CC2(CCC(NC(C3CCCOCC3)=O)CC2)C1 11788,C1(NC(C(CO)NC(C(C)C)=O)=O)CCCN(Cc2ccccc2)C1 11789,CC1CN(CC(Cl)=CCl)CCC1N(C)C.C12(CCC1)C(=O)N2 11790,c1(C(=O)NCC2CCCN(c3nccc(CO)n3)C2)cnc(O)c(C(F)(F)F)c1 11791,C1(C(=O)NN2CC3CC3C2)CCN(CCNC(CNC(CCC)=O)=O)CC1 11792,C(=O)(C1=CCN(C(c2cc[nH]n2)=O)C1)NC(c1ncc[nH]1)(C)C 11793,C(=O)(CC(C)(C(F)F)N(C)C)NCC(CC=C)NC(=O)Cc1cccc(Cl)c1F 11794,Nc1cc(C(=O)NC(CO)CCc2ccccc2)on1 11795,c1(CNC(CSC)=O)cc2cnccc2o1.c12ccc(cc1)[nH]c2=O 11796,c1(CC)nn(C)c(C(N2CCSC(C(N3CCOC(SC)C3)=O)C2)=O)c1Cl 11797,C(=O)(CCCN1CCCC1)NCC(CSC)C 11798,C(=O)(C1=CCN(C(C2(F)CCCC2)=O)C1)N(c1cnc(F)nc1)C 11799,N1(C(c2ccc3c(n2)NCC3)=O)CCCC2CN(C(C3(F)CCC3)=O)CCC12 11800,N1(C(C(C)OC)=O)CC(CNC(=O)C(c2ccc(C)cc2)C)C2(CCC2)C1 11801,Cc1cc(C(N2CC(NC(=O)C(F)F)C(F)C2)=O)c(C)n1-c1ccc(Br)cc1 11802,C1(NC(C(C=C)O)=O)CCC(NC(=O)C(C)NC(=O)COC)CC1 11803,C(CCCc1cccs1)(c1ccccc1)NC(C(n1cc(C2(O)CC2)nn1)C)=O 11804,CCC(O)CC(=O)NC(CC1CC1)C(=O)N(C)CC1CCCC2CC12 11805,CCC(C)(O)C(=O)NCC1(F)CCC(CNC(=O)C=C(C)I)C1 11806,c1(C(N2CC(CC(=O)N(CCCCCC)CC)(OC)C2)=O)ncn2c1CCC2 11807,CC1Cn2nccc2CN1C(=O)C1=C(F)CN(C(=O)CCc2ccnn2C)CC1 11808,CCC(CC(=O)NCCC1CCCCC1O)N(C(=O)C(C)N1CC(C)C1)C 11809,C1(NC(C2C(C)(CC)C2)=O)CCN(C(C2CC2C2CCCC2)=O)CC1(C)C 11810,c1(NC(N2C(CCNC(C3C4CCOCC34)=O)CCC2)=O)cnccc1CO 11811,c1(CC)cnc(C)nc1N1CCC(CF)(NC(c2cnn(C)c2Cl)=O)C1 11812,N1(C(C(C)(C)OC)=O)CC2(CCCN(C(=O)CC3CCCC(=O)C3)C2)C1 11813,c1(C(N2C(C)CC(NC(c3c(C)cc(C)nc3)=O)C2)=O)ccc2nc(S)[nH]c2c1 11814,c1(CC(=O)OC)cccc(CN2CC3CC3(C(N3CCC(C)C3)=O)C2)c1 11815,c1(CC)cc(F)ccc1C(=O)NC(C)C(C)NC(C1(C2CC2)CC1)=O 11816,c1(C(=O)NC(CN(C(C2(C)CCC(F)(F)C2)=O)CC)C)cnc(C(C)C)nc1C 11817,CC1CCN(C(c2n[nH]cc2Cl)=O)C(CNC(c2cc(-c3ccco3)on2)=O)C1 11818,N1(C(c2c(C)nc(Cl)s2)=O)CCc2sc(C(=O)NCC3CNCCO3)cc2C1 11819,N1(CC)CCC(C(=O)NC2CCCCC2CNC(c2cnsc2C)=O)CC1 11820,C(CN=C(NC(C)COC)NC1CC2(CC2)C1)OC 11821,N1(C(c2cc3c(s2)CCC3)=O)CCCN(C(=O)C(F)CC2CCC2)C(CO)C1 11822,N1(C(CNC(=O)NC)=O)CCC2C(CCCN2C(=O)CCn2cc(Br)cn2)C1 11823,C(CNC(c1ccccc1N(C)C)=O)(C(C)C(C)C)NC(Cc1cnc(C)s1)=O 11824,c1(C(N2CCCC(NC(C3CCC4CC3CO4)=O)C2)=O)nc2c(s1)COCC2 11825,C1(NC(C(C)(C)N2CCC2)=O)CC2(C1)CC2C(N1CCC(O)(C(F)(F)F)C1)=O 11826,c1(C(N2CC(n3cc(CCNC(C)=O)nn3)C2)=O)cc(Cl)cn1C 11827,C(C(=O)NC(C)(C)C)(C(C)CC1CC(F)(F)C1)N(C1CCC1)CC 11828,c1(C(=O)NC2C(NC(Cc3[nH]c(=N)sc3)=O)CCCC2)ccc2c(O)ncnc2c1 11829,CC1(C(=O)NCC2CC(O)(CNC(=O)CNC(C3CCC3)=O)C2)CCOCC1 11830,C#Cc1ccccc1CN1CCC(O)C(C(=O)Nc2cc(CC)nn2CCO)C1 11831,Cc1cc(NC2(CNC(=O)CCCC3CCC3)CCOCC2)nc(S(C)(=O)=O)n1 11832,Cc1ncsc1C(C)NC(=O)CN(C(=O)CCn1ccnc1C)C 11833,c1(C(N(CCCN(C)C)CCNC(C23CCC(C2)C3)=O)=O)cc([N+](=O)[O-])n[nH]1 11834,n1(CC(=O)NC2C(NC(Cc3c(C)n[nH]c3)=O)COC2)nc(C)n(C)c1=O 11835,C(=O)(CCCCCC(C)(C)C)NCCCN(C(C)C)C(C1CC12CCOCC2)=O 11836,c1(NC(c2cncnc2)COC)cnc(C(C)(C)Cl)s1 11837,C1(NC(CSCC(=O)OCC(C)C)=O)CN(C(=O)CCOC(C)C)CCC1C 11838,N1(C(c2c(C)nc[nH]2)=O)CC2CC(NC(c3cc(N)ccn3)=O)C(C2)C1 11839,C1(C(=O)NC2(CNC(CCC(C)C)=O)CC2)Cc2ccccc2N1C(C)=O 11840,c1(CNC(=O)NC2(C(=O)O)C(C)C2)cc(Cl)cc(Br)c1 11841,N1(C(C2(CCNC(CCC(C)OC)=O)CCCC2)=O)CCSCC(C)C1 11842,N1(C(c2cc(C)nc(O)c2)=O)CC(CNC(c2nccnc2Cl)=O)OC(C)(C)C1 11843,N1(C(C2CC(=C)C2)=O)CCCC2C1CCCN2C(c1cnc(OC)c(C)n1)=O 11844,Cc1nc(C(=O)NCC2C=CC(NC(=O)C(O)CC3CCOCC3)C2)sc1C 11845,N1(C(CSCC=C)=O)CCOCC1CNC(C1CCCC(CF)C1)=O 11846,Cc1ccccc1C(=O)NCC(N1CCOCC1CC(=O)NC1COC(=O)C1)=O 11847,N1(C(C(C(C)C)CNC(C2CCN2C)=O)=O)CC2(C1)CC(C)(O)C2 11848,c1(CC)cccc(C(=O)N(CC(C)N(C)C(c2ccc(Br)cc2)=O)C)c1 11849,CCCC(C)CCNC(c1nnnn1CCCF)c1cn[nH]c1 11850,N1(C(C(c2cccnc2)NC(C(C)n2ccnn2)=O)=O)CC(CO)C(C)C1 11851,Cc1c(F)cc(C(N2CC(NC(c3ccc(CO)cc3)=O)C(C#N)C2)=O)cc1Br 11852,N1(C(c2cc(CC)[nH]n2)=O)CCC(C2CCN(C(=O)CCCC(=O)N(C)C)C2)C1 11853,Cc1ccc(=O)n(CC(N2CC(NC(c3cc(C(C)(C)C)n[nH]3)=O)CC2C)=O)n1 11854,N1(C(C(CC=CC)CC)=O)CC(C2CCN(C(=O)CCNC(N)=O)CC2)C1 11855,CCCCCCC(C)C(=O)NC1CC2CN(C(=O)C(F)(F)C(F)(F)OC)CC2C1 11856,c1(NC(C2CN(C(=O)Cc3ncccn3)CCN2)=O)ncc(Br)cc1Br 11857,N1(C(C2(SC)CC2)=O)CC2CCCC2(CNC(=O)C(C)CNc2ccccc2)C1 11858,C#Cc1ccc(CC(=O)NCCC2(CNC(C3CC3C3CC3C)=O)CC2)cc1 11859,C(=O)(C1=CC2CCCC12)N1CC(COC)(NC(=O)C(=O)Nc2cc(C)ccc2C)C1 11860,CC(C)CC(=O)C(=O)NCC(C(N1CC(CO)CC(C)C1)=O)N(C)C 11861,C(=O)(CS(=O)(=O)C(C)(C)C)N1CC(C(N)=O)(CNC(Cc2c(C)nc(C)s2)=O)C1 11862,Cc1c(C(=O)NC(CNC(C2(n3cc(Cl)cn3)CC2)=O)CO)ccn1C 11863,C1(C(N(CCN(C(CC2C(C)=NOC2=O)=O)C)C)=O)SC2C=CC1CC2 11864,n1(CC)nc(C(N2CC3CC3(NC(C3CCC(C(F)(F)F)CC3)=O)C2)=O)cc1O 11865,CCC(c1cccc(Cl)c1)=CC(=O)NC1CCC(CNC(C2CNC(=O)N2)=O)C1 11866,C(=O)(C(CC(C)(C)C)OC)NCC(CNC(C1(OCC)CCCCC1)=O)OC 11867,C(CN=c1nc2[nH][nH]cc-2c(O)n1)N(C(c1ccccc1S(C)=O)=O)CC 11868,C1(C(C)C)C(NC(C2CCNC2=O)=O)CCN1C(=O)CCCn1ccnc1 11869,N1(C(c2n[nH]c(CC)c2F)=O)CCCC2(CCCN(C(=O)CCOC)C2)C1 11870,C1(NC(c2c(CC)nn[nH]2)=O)CC=CCC1C(=O)NC(C(C)C)C1CC1 11871,C1(C(N2CCC(N(CC#C)C(C3COCCO3)=O)C2)=O)CCCCC1(C)C 11872,c1(CN(c2n(C(C(CC)C)C)nnn2)C)ccc(Cl)cc1 11873,C#CC(C)(C)C(=O)NC(C1CN(C(=O)C=CCN(CC(F)(F)F)C)C1)C 11874,c1(C(=O)NC(CNC(c2cc(CC)n(C)n2)=O)C(C)C)c[nH]c2ccc(C)cc12 11875,c1(C(=O)NCCC2(CNC(c3cnsn3)=O)CC2)cc(=O)n(-c2ccccc2)[nH]1 11876,N1(C(C(C)(C)Oc2ccccc2)=O)CC2ON=C(CNC(C3CC=CC3)=O)C2C1 11877,Cc1cc(CN2CCC(C)(NC(c3cc(C)n(C)n3)=O)C2)c(C)s1 11878,N1(C(C(C)NC(CC)=O)=O)C2CCC1CN(C(c1c(C)nc(C)n1O)=O)C2 11879,Cn1cc(Br)cc1C(=O)NCCC1CN(C(c2cncnc2C2CC2)=O)C1 11880,c1(C(=O)NC2CC(CNC(C(C)O)=O)C2)ncoc1C1CC1 11881,c1(C(=O)NCCN(c2[nH]cnc3nc(Cl)cc2-3)CCC)cc(F)cc2nn[nH]c12 11882,c1(C(C)=O)ccc(C(N2CCOC(CNC(=O)C(C)=CC(C)(C)C)C2)=O)cc1 11883,Cc1cc(F)cnc1C(N1CCCC1C1(C(=O)NCCF)CC1)=O 11884,N1(CCNC(C2C=CCC2)=O)CCCN(C(=O)Cc2csc(C3CC3)n2)CC1 11885,N1(C(=O)C2=CCCO2)CC2CCCN(C(C3C=CCCC3)=O)C2C1 11886,N1(C(c2c(C)sc(O)n2)=O)CCCC(NC(c2ccncn2)=O)C(F)C1 11887,c1(CCC(N2CCCC(n3cc(COC(=N)O)nn3)C2)=O)ncc(Br)cn1 11888,C(=O)(C1=CCCC1C)NCc1cc(C(=O)NCC(C)OCC=C)on1 11889,N1(C(C(CCCC)(C)F)=O)CCC2(CCN(C(c3c(C#N)cnn3C)=O)CC2)C1 11890,c1(C(=O)NCC2N(C(CC3C(CC)C3)=O)CC2)cccc(Br)c1N 11891,C1(N(C(CC2(COC)CC2)=O)C)CCCN(C(c2c(C)ccn2C)=O)C1 11892,N1(C(C(=O)N(C)C)=O)CCC2CCN(C(=O)Cc3coc4ccccc34)CC12 11893,CCC(C)(CNC(c1ccc(F)s1)=O)NC(=O)CN(c1ncccn1)C 11894,N1(Cc2ncn(C)n2)Cc2[nH][nH]c(=NC(=O)c3ccn4ccnc4c3)c2C1 11895,C(=O)(C(CC(F)F)c1ccccc1)NCC(CC=C)NC(=O)OC(C)(C)C 11896,C(=O)(C1CCCc2nccn21)NC1CNC(CO)C1.C1(OC)CN2CCC12 11897,C(=O)(C1=C(F)CN(C(C2CC(n3ccnn3)C2)=O)CC1)N(C1CC2CC2C1)C 11898,N1(C(C2C(C)N(C)CC2)=O)CC2(CCNC(=O)CCC(N)=O)CCC1C2 11899,CC(Cc1ccc(Cl)cc1)CC(=O)NCC1CCN1C(=O)Cc1cnccn1 11900,Cc1ccc(OCC2CCC2)c2ccccc12.N1(C(=O)O)CCC2C(CCCN2CCC)C1 11901,N1(C(=O)Cn2ccnn2)CCCCC(C2CN(C(c3c(Cl)cccc3Cl)=O)C2)C1 11902,c1(C(CNC(CC2(C)CN(C(C3CNC(=O)C3)=O)C2)=O)=O)ccc(Cl)cc1 11903,N1(C(=O)C(C2CCOCC2)O)CC2CCCC2(Nc2cc(Cl)ncn2)C1 11904,C1(F)(CNC(C(CCC)(C)O)=O)COCCN(C(c2coc(C(N)=O)c2)=O)C1 11905,CC1COc2c(C(=O)NC3CCC3CNC(c3cnc(Cl)s3)=O)cccc21 11906,C(=O)(CC(=O)N(CC(C)C(=O)NCCCC(=O)NC)C)OCC 11907,C12(CNC(C(C)OCc3ccncc3)=O)CCCCC1N(C(=O)C(C)O)CC2 11908,N1(C(C(CC)C(F)(F)F)=O)CCC(C2CCN(C(=O)CCn3cnnn3)CC2)C1 11909,c1(C(N(C2CCN(C3CCN(C)C3=O)C2)CCC)=O)ccc2oc(O)nc2n1 11910,CC1(C)CC(CNC(=O)C(F)=CC2CC2)CN(C(=O)CN2CC3CC3C2)C1 11911,Cc1ccncc1C(=O)NCc1cn(CCNC(=O)Cc2ccns2)nn1 11912,C=CC(CC)CC(=O)N1CCN(CCCNC(C2(S(C)(=O)=O)CC2)=O)CC1 11913,N(C(=NCCC1CCCOC1)N1CCCC(S(C)(=O)=O)C1)Cc1c(C)nccn1 11914,c1(C(N2CC(c3cn(CC(=O)O)nn3)C2)=O)cc(Br)cc(I)c1F 11915,C1(CCNC(CC2(C)OCCO2)=O)CCCN(C(c2cnc(Cl)s2)=O)CC1 11916,c1(C(C(=O)NCC2CCC(NC(c3nsnc3O)=O)C2)(F)F)ccc(F)cc1F 11917,C=CCC(CC)C(=O)NCC1(CO)CCN(C(=O)CC2(C)CC2)C1 11918,Cc1cncc(C(N2CC(NC(c3cc(-c4cnn(C)c4)[nH]n3)=O)C(F)C2)=O)n1 11919,c1(C(=O)NC2C(C)CN(C(c3cccn(C)c3=O)=O)C2)cccc2c1CCCC2 11920,c1(C(N2CCCC(CCNC(C(CC)CO)=O)C2)=O)ccc2nonc2c1 11921,C1(CNC(CC(=O)OCC)=O)CCN(C(=O)CN(c2ccnc(Cl)n2)C)CC1 11922,c1(CN)ccc(C2(C(=O)NCCc3cn(CC(=O)OC)nn3)CC2)cc1 11923,N1(C(C(C2CCCCC2)NC(C(=O)NC(C)C)=O)=O)CCS(=O)(=O)CC1 11924,C1(C(=O)NCC2CCN(C(C3CCO3)=O)CC2(F)F)CCC2(CCCC2)CC1 11925,N1(C(CCCC#CC)=O)CCC2(CCC2NC(=O)CCc2nncn2C)CC1 11926,n1(CCOC)c(N(C)Cc2cccc(C(C)(C)C)c2)nnc1-c1cc(CO)no1 11927,C1(CC(=O)OC(C)C(=O)OC(C)(C)C)CCN(CC2(C#N)CCC2)C1 11928,N1(C(COCCCC#C)=O)CCC(C2N(C(=O)C=C(C)C)CC2(C)C)CC1 11929,C(=O)(C1=C(C)CCCC1)NCC12N(C(C(CCCC)O)=O)C(CC1)CC2 11930,C(=O)(C=CS(F)(F)(F)(F)F)N1CCN(C)CC(OC(F)F)C1 11931,c1(CNC(COCC(=C)C)=O)ocnc1C(=O)NC(C)Cc1cccnc1 11932,N1(CCC)CCc2cc(C(C)NC(C)CSCOC)ccc21 11933,C1(NC(c2c(SC)cn(C)n2)=O)CCN(C(c2cc(F)ccc2F)=O)C1(C)C 11934,CCCC(C(=O)N1CCN(C(c2ccc(OC)c(F)c2)=O)C(C(F)F)C1)C(C)C 11935,CC1OC2CCC1(C(N1CC(NC(c3cc(Cl)cs3)=O)C1)=O)C2 11936,c1(OC)ccc(C(=O)NCC(C(C)(C)C)NC(c2ccsc2)=O)cc1C(F)F 11937,C1(C#N)(C(=O)NCC(C2CCCC2)NC(C(C2CCOCC2)C)=O)CC=CC1 11938,C(=O)(CCCCCC(C)(C)C)NCC(CNC(CN1CC(CC)C1)=O)O 11939,C#CCCCC(C)C(=O)N1CCCN(C(c2ocnc2C2CC2)=O)CC1 11940,C1(C(N2C(C(C)(C)NC(=O)CC3CCCC(O)C3)CCC2)=O)CC(S(C)(=O)=O)C1 11941,C12(C(=O)NCc3nc(CNC(C4CCCC4C(F)F)=O)sc3)CCCN(CC1)C2 11942,N1(C(=O)CC2CCCO2)CCN(C(c2cnc(O)o2)=O)C(c2ccccn2)C1 11943,C1(CNC(C2N(CC)CC2)=O)CN(C(=O)Cn2cc(C3CC3)nn2)CCCO1 11944,c1(OCC=C)ccc(CCNC2CC(=O)N(c3ccccc3Cl)C2)cc1 11945,C1(C(=O)NC(C2(O)CN(C(Cc3cc(C)[nH]n3)=O)C2)C)CCc2nccn2C1 11946,C#CC(CNC(=O)C(C)N(C(=O)C(CCC)N(C)C)CCC)CC(C)(C)C 11947,C1(CCNC(c2cn(CC=C)nc2)=O)CCCN(C(=O)CCc2nc[nH]n2)CC1 11948,C1(O)(CCNC(C2CCOC2)=O)CCN(C(c2cnn(CC(F)F)n2)=O)C1 11949,c1(OCC)cc(C(=O)NC(C)C=CC(=O)N(CCCOC(C)C)C)[nH]n1 11950,c1(OCC(=O)NCC2(CNC(C3N(N=O)CCC3)=O)CC2)ccccc1[N+](=O)[O-] 11951,c1(N2CC(O)(CCNC(C=COCC)=O)C2)ncc2cccnc2n1 11952,N1(Cc2c(N(C)CC)nccc2)CCC(=O)N(Cc2cc(Br)c(F)cc2F)C1=O 11953,C1(NC(CC2ON=C(CC)C2)=O)CC2CCCC(C1)N2C(c1cccn1CC)=O 11954,c1(C(N2CCC(CC=C)(NC(C3COC(C)C3)=O)C2)=O)cc([N+](=O)[O-])cnc1O 11955,N1(C(CC(C=C)(C)O)=O)CCC2(CC1)CN(C(=O)C=CBr)CC(C)O2 11956,N1(C(C(C(CC)C)OC)=O)Cc2ccccc2-c2ccccc2C1 11957,C1(C(N2CC(OC)(CNC(C3CCCC3O)=O)C2)=O)C2(CCC2)C12CCC2 11958,c1(CN(C)C(c2ccon2)=O)ccccc1CNC(c1cc(Cl)ns1)=O 11959,N1(C(CCCOC(C)C)=O)CCCC(C(C)NC(=O)CCCCC2CC2)C1 11960,c1(-c2cn(CC(=O)N(CCC)C(C)C)nn2)ccc(C(=O)NC(C)C)nc1 11961,c1(CN=C(NC(c2sc(C(F)(F)F)cc2C)C)NC(C)C)c(F)cc(F)c(F)c1F.CO 11962,c1(C(=O)NC2CCN(C(C3CCN(C4COC4)C3)=O)C2)ccc2c(c1)NCC2 11963,N1(C(CCCCC=C)=O)Cc2ccnn2CC(NC(c2nc(CC)sc2N)=O)C1 11964,N(C1CCc2cc(Br)ccc21)C(=O)Cn1cc(COc2cccc(CO)c2)nn1 11965,Cc1ccc(C)c(C(=O)NC2CCN(C(=O)CSc3ccccn3)CC2F)c1C 11966,c1(C(=O)NC2C(C)CN(c3nc(C#N)ncc3Cl)CC2)ccc2ncccc2c1 11967,c1(OC)ccc2c(C(=O)NC(C3CCCCN3C(c3ccns3)=O)C)n[nH]c2c1 11968,CCC(CC)C(=O)NCCCCC(C)NC(=O)CO.c1(OCCO)ccccc1Br 11969,C1(NC(=O)CC2CCCCCO2)CC2CCC(C1)N2C(C1(CC(F)(F)F)CC1)=O 11970,O(N1CCC(c2nc(COC)nn2-c2cccnc2On2cncn2)CC1)CC 11971,c1(C(c2nnnn2C)NCC(CCCC)CO)ccc(S(=O)(=O)NC)cc1 11972,CC1(C)CC(C(=O)NC(C2CCC(F)(F)C2)=O)(CO)C1.c1(C2CC2)cc[nH]n1 11973,c1(NC(N2C(c3cn(CCC=C(C)C)nn3)C(C)CC2)=O)ncc(Cl)cc1Cl 11974,CC1Oc2c(F)cccc2C1NC(=O)C(N1CCCC(O)(C(N)=O)C1)=O 11975,CC1(C)CC(C(N2CCC2CC(=O)N(C)C)=O)N(C(=O)CC2CCC=CCC2)C1 11976,C(CCC(=O)NCC1(C(N2CC(CC)C2)=O)CC=CC1)=CCC=C 11977,C1(C(=O)NC(CNC(CC2CC(CC)C2)=O)CC)CCn2nnnc2C1 11978,CC(C)CC(F)C(=O)N1CC2CC1(CNC(c1csc3nnsc13)=O)C2 11979,c1(C(N(CC)CC2CCN(C(=O)C(C)SC)CC2)=O)cc2n(n1)C(C)CCC2 11980,c1(SC2C(C(=O)NCC(C3CCCCC3)NC(C)=O)C2)ccccc1 11981,CCCCC(C(=O)NCCC1(O)CCN(C(=O)C2=CCCC2)CC1)C(C)C 11982,O=C(CC(C(F)F)NC(c1cc(Cl)ns1)=O)NCCC1CCCCC1O 11983,n1(CC(=O)NCC(C)(CNC(=O)CCOC2CCC2)OC)nc(C)nc1C 11984,O=C(C1=CC2(CCOC2)C1)NCC1CCN(C(c2cc(=O)cc[nH]2)=O)C12CC2 11985,c1(N(C)Cc2ncccn2)nc(N2CCCC(CC(F)F)C2)nc2c1ncn2C 11986,c1(Sc2ccc(Cl)cc2)cccc2c1NC(=O)CN(c1n(CCC)nnn1)C2.CC 11987,O=S(=O)(c1cc(Br)cc(Br)c1)N1CCn2c(C3CC3)nnc2C1 11988,c1(C(=O)NCC(CNC(C(CC#C)C)=O)CO)cc(N2CCCC2)cc(Cl)c1 11989,C1(Nc2c(C(=O)OC)ccc(CO)c2)Cc2cccc(C)c2O1 11990,c1(C(=O)NC2(CC(=O)NCC3(C(=O)OCC)CCC3)CC2)cncc(C#N)c1 11991,c1(NC(=O)Nc2cn(C(F)(F)F)cn2)cc(C(F)(F)F)ccc1O.C12CN(C1)C2 11992,c1(C(=O)NC(CNC(C2(C#C)CC2)=O)CC(C)C)ccc(Cl)c(CCC)c1 11993,CC1(C)CC2(CC(C(=O)NCC(O)CNC(=O)CP(C)(C)=O)C2)C1 11994,S(=O)(=O)(c1ccc2c(c1)CCO2)N1C(C(=O)Nc2cccc(Br)c2F)CC(=C)C1 11995,C(=O)(C(CC(C)C)OC)N(C1CCC(NC(C2(CC)CC(C)(C)C2)=O)CC1)C 11996,N1Cc2ccccc2C1.N1(C(C(C2CC2)SC)=O)CCC(C)CC1C(=O)N 11997,Cc1cc2sc(C(=O)NCC(C(C)C)NC(=O)C(C#N)C(C)C)cc2s1 11998,CC(C)(Cn1nc(-c2nccs2)nc1CC1CCOC1=O)S(C)(=O)=O 11999,c1(OC)ccc(O)cc1NC(=O)CCC(C)NC(=O)C(C)(C)C(C)O 12000,CCC(O)(CC)CCNC(C1CC(NC(=O)C(C)c2cccs2)C(O)C1)=O 12001,c1(C(N2CCC(NC(C(CC=C)C)=O)(CO)C2)=O)cccn2c(CO)nnc12 12002,C1(N(C(CC2(C(=O)OCC)CCC2)=O)C)CCCCC1N(C(=O)C1=NOCC1)C 12003,c1(C(N2CC(CNC(c3nc(C)nn3C)=O)C(O)C2)=O)cc(Cl)cc2c1CCC2 12004,C1(NC(C2CC3CCC2C3)=O)CCCC(CC(N2CCC(F)CC2)=O)C1 12005,CC(C)C(Br)C(=O)c1ccc(C2CCN(C)CC2)s1 12006,C1(c2n(C(CC)C)nnn2)(Nc2cnn(CC(C)C)c2C)CSC(C)(C)C1 12007,N1(C(c2c(N)cncc2)=O)CC2(CCCC2NC(=O)COCC(F)F)C1 12008,C(=O)(C(C)S(C)(=O)=O)NCC1CCC(CNC(c2n[nH]c(C)c2Cl)=O)CC1 12009,C12(NC(C(CC#CC)NC(=O)C(COCC)N=[N+]=[N-])=O)CCC(CC1)C2(C)C 12010,c1(C(=O)NC(CN(C(c2ccc(OC)c(F)c2)=O)C)C)csc2c1CCC(C)C2 12011,c1(CNC(=O)Nc2ccnn2C2CC2)cccc(-n2cccn2)c1 12012,C(CC(C(=O)NC1CC(CNC(=O)OC(C)(C)C)C1)c1ccccc1)=CC 12013,c1(N2CCC(NC(=O)Cc3cccc(Cl)c3)C(O)C2)ncnc2ccc(O)cc12 12014,N1(C(c2cccc(OC)n2)=O)CCC(C)(C)C1C(=O)NOCCC(F)F 12015,c1(C(N2CCC(NC(c3nn(C)c(Cl)c3)=O)C2)=O)c(F)cncc1Cl 12016,C(=O)(C(O)CC(F)(F)F)N1CC(CCCCNC(c2ccc([N+](=O)[O-])o2)=O)C1 12017,c1(CNC(C=NOC)=O)ccccc1CNC(C1CC(=O)N(c2cn[nH]c2)C1)=O 12018,C(=O)(CCCCCC(C)C)N1CCCC(CCC(N2C(CC)CCC(C)C2)=O)C1 12019,c1(OCC)nc(N2CCCC2CNC(C23CCCC(C2)OC3)=O)ncc1Cl 12020,C1(C(=O)NC2CN(C(c3c(C(C)C)ocn3)=O)CC2C)CCC2(C1)CC2(F)F 12021,CC1(C)CN(C(=O)C(F)F)CCC1NC(=O)CCc1ccc(F)cc1Cl 12022,N1(C(C(C)SC)=O)CCC(C2CCN(C(c3cn(C)nc3C(F)(F)F)=O)CC2)C1 12023,CC1(C)COCC1CNC(C1C(NC(=O)CCc2ncccn2)CCC=C1)=O 12024,c1(C(=O)NC2CC3CN(C(c4ccc(Br)cn4)=O)CC23)cccn2cncc12 12025,C(=O)(C1=CCC(C)CC1)N1CCN(C(c2ccc(C)cc2F)=O)C(CF)C1 12026,Cc1cc(C)n(Cc2cccc(C(N3CCC(NCCN(C)C)CC3)=O)c2)n1 12027,c1(C(N(C)CC2N(C(C(C)NC(N)=O)=O)CCC2)=O)ccc(Cl)c(Br)c1 12028,C(=O)(C(C(C)(C)C)NC(C1CCN(C(=O)C=Cc2cncs2)C1)=O)OC 12029,C1(NC(c2c(SC)cccn2)=O)COC2(CCN(C(C3(C#N)CCCO3)=O)C2)C1 12030,C(=O)(C1=CSCCO1)N(CCCNC(=O)Cc1sccc1Cl)CC 12031,C(C(=O)N1CC(C(=O)NCC2CCC(C)(C)O2)C2(CC2)C1)(C(C)(C)C)OC 12032,C12(C(N(CC#C)C)=O)C(NC(=O)C=C(C3CC3)C3CC3)C3CC1C2C3 12033,CC1C(NC(C2CCN(C3CC3)CC2)=O)CCCN1C(=O)CN1CC2CC2C1 12034,C(C(C(=O)N(C1(C2CC2)CC1)C)NC(C1CCC(=O)O1)=O)N(C)C 12035,C1(C#N)(C(N2CCC(CN(C)C(c3ccnc(CO)c3)=O)CC2)=O)CCCC(=O)C1 12036,C1(CC(N)=O)CCN(C(C2CC(n3cnnc3)C2)=O)C2(CC2)C1 12037,Cc1[nH]nc2c(C(N3CCCCC(NC(C4(C)CCCOC4)=O)C3)=O)cccc12 12038,C1(C(=O)NC2CCC(NC(CCc3cc(C)on3)=O)C2)CCC2(CCCCC2)C1 12039,c1(SC)cc(C(=O)NCC2(NC(C3C=CC(CO)C3)=O)CCC2)ccc1N 12040,Cc1ccc(F)c(OCC(N2CC(NC(C3CCCS3)=O)C3(CC3)C2)=O)c1 12041,C(=O)(C#CC1CCOCC1)N1CCC(C(N2CCCC(CC(C)C)C2)=O)C1C 12042,c1(C(=O)NCCCCCN(C(=O)CC2(C)CC2(Cl)Cl)C)cc([N+](=O)[O-])cnc1N 12043,N#Cc1ccc(N2CCCC(NC(=O)NC(c3ccccn3)CCO)C2=O)cc1 12044,N1(C(CC=C)=O)CCCN(C(=O)C(c2ccc(OC)c(F)c2)C)C(CC2CC2)C1 12045,c1(CC)cccc(C(=O)N(C)CC2(NC(c3cc(C4CC4C)on3)=O)CC2)c1F 12046,Cc1cc(CC(N2CC(n3cc(CNC(N)=O)nn3)C2)=O)ccn1 12047,C1(N(C(C(COC)N(C)C)=O)C)CN(C(c2cn(C)nn2)=O)CC1O 12048,C(C(=O)CCC(=O)N=c1ccn(C2CCOC2)[nH]1)Oc1ccc(C)cc1 12049,C#Cc1ccc(CC(N2CC3(C)CC2C3NC(=O)C(C)n2cccc2)=O)cc1 12050,CCC(C)CCCC(=O)N1CC=CC1C(=O)N(C)CC1CN(C)CCO1 12051,c1(OC)ccc(CCC(=O)N(C(C)CNC(=O)C=CC(=O)NC(C)C)C)cc1C 12052,c1(CC)cc(C(=O)NCc2cn(C3CN(C(c4cc(C)co4)=O)C3)nn2)no1 12053,C1(NC(Cc2nc(C(C)(C)C)sc2)=O)CC2CCC(C1)N2C(C1(O)CC1)=O 12054,Cc1cc(=O)n(CCC(=O)NC23CC(NC(=O)CSc4n[nH]c(=N)s4)(C2)C3)cn1 12055,N1(C(CCCn2c(C)ncc2)=O)CCOC(CCNC(C2CC(F)C(=O)N2)=O)C1 12056,C(CN=c1cc(Cl)nc[nH]1)(c1ccccc1F)NC(c1cocn1)=O 12057,c1(CC)c(C(=O)NC(C)CC2CCN(C(C3CCN3CC)=O)CC2)cnn1CC 12058,C1(COC)(NC(=O)CCNC(N)=O)CCN(C(c2cc(F)cc(Cl)c2)=O)CC1 12059,c1(OC)cc(NC(=O)CC(n2nc(C)cc2C)C)cc(OC)c1C(C)C 12060,Cn1cc(C(=O)NC2CCC(CNC(C3(C)CCNC3=O)=O)C2)c(=O)n(C)c1=O 12061,N1(C(c2c(CC)cns2)=O)CC(O)CC1C(=O)NC(COC)C(C)C 12062,C1(NC(CCCC)=O)CC2(CCN(C(=O)C(C(C)C)N(CC)CC)CC2)C1 12063,c1(SCc2nc(C3(C(F)F)CCNC3)on2)ccc(Cl)c(Cl)c1 12064,CCCCCCCCC(=O)NCC(C1CC1)NC(=O)C(CC)C(=O)OCC 12065,N(C(=NCc1ccc(C)cc1)NC1CCOCC1)CC(C1CCOCC1)OC 12066,C1(OC)C(OC)CN(C(=O)C(C)C2CC2)C1CNC(c1nc(Cl)sc1C)=O 12067,C1(OCC)COCCC1CC(=O)NCC1CCN(C(C)C(=O)NC(C)(C)C)CC1 12068,C1(OC)CC2(CCC(C(=O)NC3CCCC(CNC(=O)CNC(N)=O)C3)CC2)C1 12069,Cc1ncccc1CC(=O)NC1CC1NC(=O)CCc1cn(C)nn1 12070,C1(OC)CC(CNC(=O)C=Cc2ccnn2C)N(C(c2cc(C)on2)=O)C1 12071,c1(C(=O)NC(C2CN(C(CC(C)SC)=O)C2)C)ncnc(C)c1C 12072,C(=O)(C(=O)CC(C)C)N1CCC(C(C(=O)N(C)CC2(OCC)CCC2)C)CC1 12073,C1(C(N(N2C(C)CCC2)CC)=O)CC12CC(F)(F)C2.c1(C=O)cnc(N(C)C)o1 12074,C12(C(CNC(CC3CC(C)C3)=O)NC(=O)CC3CCCOC3)CCC(CC1)C2 12075,N1(C(c2cc(C)c(C)o2)=O)CCC(CCNC(c2csnc2C)=O)C(F)(F)C1 12076,CC(C)(C)C(C(=O)NCC(O)CF)NC(c1ccc(CC#N)cc1)=O 12077,C1(CN)CCCCN1Cc1cccn1CC1CCC(C(=O)OC)O1.n1(C)ccnc1 12078,c1(-n2cc(CN(C)C(C3CCC(C(=O)O)C3)=O)nn2)ccc(OC(F)(F)F)cc1 12079,c1(C(=O)NCCN(C(C)C)C(C2(CN(C)C)CC2)=O)cc(C(F)F)ccn1 12080,C(=O)(C#CC1CCCCC1)N1CCCCC(NC(c2c(C(C)=O)cn(C)n2)=O)C1 12081,N1(C(CSCC=C)=O)CC2(CNC(C3(C)C=CCC3)=O)CCC1CC2 12082,c1(C(=O)NC2(C)CN(C(=O)Cc3ccsc3)C2)nc2n(c1Br)CCC2 12083,c1(C(N2CCCC(NC(c3ccco3)=O)(CO)C2)=O)c(F)cc(F)c(O)c1F 12084,CC(CC(C)(C)C)C(F)C(=O)N1CCC1CNC(=O)CC1CNC(=O)O1 12085,C1(NC(c2ccc(Cl)c(F)c2)=O)CCC2(CC1)CN(C(=O)CC1CSC1)C2 12086,c1(OCCCC)ccc(S(=O)(=O)N2CC(c3ccccc3)C3(CCC3)C2)cc1 12087,CC(CC(=O)NCCOCCCNC(=O)CN(C)C(c1ccsc1)=O)P(C)(C)=O 12088,C(=O)(C1CCc2nccn21)NCC(C)(C)OCC(=O)Nc1cccc(N(C)C)c1 12089,Cc1cc(C(=O)NC(CNC(c2ccc(CC(N)=O)cc2)=O)C2CC2)ncn1 12090,c1(-c2cn(CC3N(C(C(C4CC4)SC)=O)CC3)nn2)ccc(-c2cn[nH]c2)cc1 12091,c1(NC(C=CC(=O)N(C2(C)CN(C(C)=O)C2)CC2CC2)=O)ccc(F)c(Cl)c1 12092,c1(C(N2CCC(CC=C)(NC(C3CC(C)OC3C)=O)C2)=O)cnc2nccn2c1 12093,Cc1nnccc1C(N1CC2CC1C2NC(=O)CSCc1cccs1)=O 12094,N1(C(C2=CCCN(C(C3CCC(C)O3)=O)C2)=O)CCCC(C2(C)CC2)C1 12095,c1(OC)ccc2onc(CC(=O)NC(C)C(C)NC(c3c[nH]c(=N)o3)=O)c2c1 12096,C1(CCNC(C(C)(C)OC(C)=O)=O)CCCN(C(C2CCCN2S(C)(=O)=O)=O)C1 12097,c1(C(=O)OCCSc2cc(Cl)ccc2Cl)cc(Cl)c(Cl)cc1F 12098,N1(Cc2cc(C)n(CCC)c2C)CCS(=N)(=O)C(C)(C)C1 12099,c1(C(=O)NCCCOCCNC(c2c(C)ccnc2O)=O)cc2c[nH]cnc-2n1 12100,C1(N(C(C(CC)Sc2ccc(-c3nn[nH]n3)cc2)=O)C)CCC(=O)N(C)C1 12101,C1(=O)C(C(CC)CC)N1.C(C)(C(=O)NC)N(CC(C)C)CC=C 12102,N1(C(c2c(OC)cnnc2OC)=O)CC2ON=C(CNC(c3ccco3)=O)C2C1 12103,N1(C(C2CCN(CC)C2)=O)CC(C(=O)NC2CC(=O)N(O)C2)CC(C)C1 12104,CCC(C(=O)N1CC(O)(CN(C)C)C1)N(C)C(C1CCC1C#N)=O 12105,n1(CC(=O)NCC(C)N(C(CCC(C)SC)=O)C)c(=O)cnc2ccccc12 12106,c1ccc2cc(C3(N4CC4)CCC3)ccc2c1.C(CC1CC1)CO 12107,C1(CC(=O)NC)CN(C(c2ccn(C(C)C)n2)=O)CCN1C(=O)COCC(C)C 12108,c1(C(=O)NC2C(NC(COC(c3nccn3C)C)=O)CCC2)cccc[n+]1[O-] 12109,N1(C(C2(C)CC(C)C2)=O)CCC(O)(C(N2CCC(Oc3ccccc3)CC2)=O)C1 12110,c1(CC(=O)NCC2C3CN(C(=O)CC4CC(F)(F)C4)CC23)ccc(O)c(Cl)c1 12111,N1(C(CC=C)=O)CC(C(=O)N(CC2=CCSC2)C)C2(CCC2)C1 12112,C1(NC(C(C(C)C)O)=O)C2CC3C1C3C2C(=O)NCc1ccccc1F 12113,c1(C(N2C(C(C)(C)NC(C(C)=CC)=O)CCC2)=O)ccc(C(F)(F)F)cn1 12114,c1(C(=O)NCCOC(C2CC3(CC3)C2)=O)c[nH]c2ccccc2c1=O 12115,c1(OC)cccc(SCC(=O)NCCCCC(C)NC(=O)C(C)(C)OC)c1 12116,N1(N(C(C)=O)C)CCCC(C(=O)NC(C)CNc2scnc2CC2CCOC2)C1 12117,CC1(C)C2CC=C(CCNC(=O)NNC(=O)Nc3cc(Cl)cc(Cl)c3)C1C2 12118,N1(C(C2CC(NC(C=C(C)C3CC3)=O)C2(C)C)=O)CCN2CCCC2C1 12119,n1(CCNC(C2(C)ON=C(C)C2)=O)cc2ncccc2n1 12120,c1(C(N(CCCC)CCOC)=O)ccc(C(=O)NC2CNCCOC2)cc1Cl 12121,C1(O)(CNC(C2C(C)C(=O)C2)=O)CCCN(C(=O)CCc2ccccc2F)C1 12122,C1(CC)C(NC(C2CS(=O)C2)=O)CCCN1C(c1ccc(C)c(C)c1)=O 12123,CC1CCc2c(C(N3CCCCC3CNC(c3cccc(=O)n3C)=O)=O)n[nH]c21 12124,CC(C)C(C(C)NC(c1cscc1Cl)=O)NC(c1ncoc1-c1ccon1)=O 12125,CCCS(=O)(=O)C(C)C(=O)NC1CC(CNC(C2CN(C)CCN(C)C2)=O)C1 12126,c1(C(N2CCC3(NC(=O)CNS(=O)(=O)C4CC4)C(C2)C3)=O)n[nH]c2c1CCCC2 12127,C1(CNC(CCc2cc(C)no2)=O)CCN(C(c2cc(Cl)c(Cl)n2C)=O)CC1C 12128,N1(C(C(c2c(C)n[nH]c2C)C)=O)CC(NC(c2conc2C2CC2)=O)CC(C)C1 12129,c1(C(N2CCOCC2c2cccs2)C(=O)NC2CCCC2)cccc([N+](=O)[O-])c1 12130,CCC(Cc1cccc(C)c1)C(=O)NCC(O)CNC(=O)CC1CCCC1C 12131,C1(C(=O)NCCCCCCn2cc(-c3cncc(C)n3)nn2)(CC)CCCOC1 12132,C1(C(=O)NCC(=C)Br)COC2(C1)CN(C(=O)C(C)OC)C2 12133,c1(C(N2CCC(O)(CNC(CCC(C)OC)=O)C2)=O)ccnc(C)c1C 12134,C1(NC(C2CCC(O)C2)=O)CC2(CCN(C(C3(F)CC=CCC3)=O)CC2)C1 12135,C(=O)(C1=NN(c2ccc(F)cc2)C(=O)CC1)NCC(C)CN(C(=O)C(F)F)C 12136,n1(CCC)cc(C(=O)N(CCNC(=O)CC2OCCC2C)C(C)C)nn1 12137,c1(C(=O)NC(CC)CNC(=O)C(C)SC(F)(F)F)ccc([N+](=O)[O-])s1 12138,N1(C(C(C)(C)N(C)C)=O)CC23CCCCC2(C1)CN(C(=O)C(O)CC(N)=O)C3 12139,Cc1ncnc(C)c1C(=O)NCC1CCCCC1NC(c1cc2occc2[nH]1)=O 12140,c1(C(N(C2CN(C(CCCN(C(C)=O)C)=O)C2)C)=O)ccc([N+](=O)[O-])s1 12141,C1(NC(C2CCC(CC)O2)=O)CC(OC)CN(C(=O)CCc2ccn(C)c2)C1 12142,Cc1nc2cc(C(=O)NC(CNC(=O)CN3CCCCC3=O)CO)c(F)cc2[nH]1 12143,C=CCC(C(=O)NCC1C=CCCC1)NC(=O)Cc1ccnn1C 12144,Cc1cc(C(=O)NC2CC(CNC(C3CC3(C)C(C)C)=O)C2)c(F)cc1Cl 12145,c1(SC)cc(C(=O)OC(C)(C)C)c(NC(C)=O)s1.C1(=O)CC(C)N1C 12146,C1(CNC(c2ccc(Cl)o2)=O)CC(F)CN1C(c1ccc(OC2CCC2)cc1)=O 12147,C1(C(=O)Nc2c(OC)cc(Br)c(F)c2)CCC(N=c2nc[nH]n3cc(Br)cc23)CC1 12148,N#CC1(CC(N2CC=CC2CNC(C2CCCCS2)=O)=O)CCCCC1 12149,CC1(C)CC(CNC(C2CSCN2C(=O)CC=C(Cl)Cl)=O)CCO1 12150,C1(NC(C23N(C(CSCCOC)=O)CCC2C3)=O)CN2CCC1(C)CC2 12151,C(=O)(C(C)(C)C(C)C)NCC(C1(O)CN(C(C=C(COC)C)=O)C1)(C)C 12152,N1(C(C(CC=C)CC)=O)CC(NC(C2CC(C)(C)C2)=O)CC2(CCC2)C1 12153,N1(C(CCn2c(C)cc(C)n2)=O)CCC2CC1CN2C(C1CCCS(=O)(=O)C1)=O 12154,Cc1cc(C)c2[nH]c(=NCC(C)N(C(=O)Cc3c(F)cccc3Cl)C)sc2c1 12155,C(CO)(CC(C)CC)NC(CSCCNC(C(C=C)C)=O)=O 12156,c1(CCC(=O)NC(CN(C(=O)C(C)CC(F)F)CC)C)c(C)ncnc1O 12157,N1(C(COCC=C)=O)CC2C=CC1C(C(=O)NCC(CO)C(C)CC)C2 12158,N1(C(=O)CCOc2ccc(F)cc2)CCN(C(=O)Cn2ncnn2)C2CCCC12 12159,c1(C(N2C(CCNC(c3[nH]ccc3C3CC3)=O)CCC2)=O)ccc(O)nn1 12160,CN1CCC(C(=O)NCC=CCC(=O)NC2(C3CC3)CCCC2)CC1=O 12161,C1(CC)CCCC1C(=O)N(CC(C)CNC(c1csc(C)c1)=O)C 12162,Cc1ccc(F)c(N)c1C(N1CC(NC(C2(C3CCC3)CC2)=O)C(C)C1)=O 12163,Cc1sc(C)c(C(N2CCC(C)C(NC(c3cnc[nH]3)=O)C2)=O)c1C#N 12164,c1(CC)nc(-n2cccc2)sc1C(=O)NC1CN(C(c2cnoc2C)=O)CC1C 12165,CN=c1[nH]c(=NC(C)c2cccc(F)c2)[nH]c(=NC2CCC3(CC2)CC(O)C3)[nH]1 12166,c1(C(=O)NC2(CCNC(C3(COC)CC3)=O)CC2)ccc2c(c1)COC2=O 12167,N1(C(CC2(NC(C)=O)CC2)=O)C2CCC1CC(CCNC(c1ccnn1C)=O)C2 12168,Cc1occc1C(=O)OCc1cn(C(c2ccccn2)C)nn1 12169,Cc1[nH][nH]c2ncnc(=NCC3(C)CCC(NC(=O)C(CO)NC(N)=O)CC3)c1-2 12170,c1(C(C)C)nc(C(=O)NCC(O)CNC(c2cc(C(N)=O)no2)=O)cs1 12171,CS(=O)(=O)c1ccccc1CNCC1CC2CC1CC2O 12172,N1(C(c2ccc(Cl)cc2F)C(=O)NCC2CC2)CC=C(c2cccs2)CC1 12173,C(=O)(CC1COc2ccccc21)NC1C(CNC(CC2(C=C)CCOCC2)=O)C1 12174,c1(C(=O)NCCCC2(NC(=O)CCNC(N)=O)CC2)cnc(-c2ccco2)s1 12175,c1(-n2cc(C3(C(=O)O)CN(C(C4CCCC4O)=O)C3)nn2)cccc2n[nH]cc12 12176,C(C(=O)N1CCC(N2CCC2)C1)(C(C)(C)C)NC(C(C)=C(C)C)=O 12177,C(=O)(C(CC)n1cccn1)NCC1(CNC(CSCCC)=O)CCC1 12178,N1(C(C(CCOC)C)=O)CCC(NC(=O)Cc2ccccc2NC(C)=O)CC1C 12179,c1(C(C(=O)NCCSC)N(C)Cc2c(C(=O)OC)cccc2)ccc(F)cc1Cl 12180,CC1CN(c2cc(C(F)F)ncn2)CCC1NC(C1CCC2CC2CC1)=O 12181,C1(C(N2CC(NC(C3CC(C)(C)C3)=O)C(C(F)F)C2)=O)CCn2c(O)nnc2C1 12182,C1(CC(=O)OC)CS(=O)(=O)CCN1C(=O)C(=O)N=S(C)(C)=O 12183,c1(C(=O)NCC(CNC(=O)CN2CCNC(=O)C2)OCC)ccc(NC)c(Cl)c1 12184,C1(C(=O)NC(c2ncccn2)C)C2CN(C(=O)CCc3ccccn3)CC12 12185,CC1(NC(c2cnn(CCNC(=O)Nc3ccccc3C#N)c2)=O)CCC(O)CC1 12186,Cc1noc(C)c1C(=O)N(C1CCN(C(C2CN(CC(C)C)C2)=O)CC1)C 12187,C1(NC(CC2CCN(C(Cn3c(C)cc(C)n3)=O)CC2)=O)CC2CCCC2C1 12188,C12(NC(CCN(C(=O)CN3CCC(C)C3)CC)=O)CC=CC(C1)OC2 12189,C1(CNC(C2C(C)OC(C)C2C)=O)CCC2(CN(CCOC3CCCCC3)C2)O1 12190,C(c1ccc(C(=O)NC2CC2CNC(=O)C(C)(C)CO)o1)=CC(=O)OC 12191,N1(C(c2ccn(CCOC)n2)=O)CCN(C(c2c(C)ncn2O)=O)CC2(CC2)C1 12192,CCC(C(=O)OC)C(=O)NC1CCCCN(C(C2OC(C)CC2C)=O)C1 12193,N1(C(c2cn(C3CC3)cn2)=O)CCC2(C1)CN(C(C1CC=CC(O)C1)=O)C2 12194,N1(C(C2CCC(CNC(C3(c4ccno4)CC3)=O)CC2)=O)CC2CC1CS2=O 12195,CC1CCCc2nc(C(=O)NCC(C3CCC3)NC(=O)Cc3csc(S)n3)cn21 12196,c1(N(C(C2(COC)CCCO2)=O)CC2CCCCO2)ccc2c(c1)OCCO2 12197,C12(CNC(c3cnc(C)c(N)c3)=O)CCC(CC1)N(C(C13CCC(CO1)C3)=O)C2 12198,C1(CNC(C(=O)N(c2ccccc2O)C)=O)CC2CN(C(c3nncn3C)=O)CC12 12199,c1(-n2c(CCCCN(C)C)nc(-c3ccc(F)cc3)n2)ccc(F)c(Cl)c1 12200,C=C(C)C(CC(=O)NCC1(CN(C)C(c2cnn(CCO)c2)=O)CC1)OCC 12201,N1(C(C2CCC(CC)O2)=O)CCC2(CCC(NC(c3cn(C)nn3)=O)CC2)C1 12202,N1(C(C(CCC)C#N)=O)CC2CCC1C1CN(C(=O)COc3cccnc3)CC21 12203,C12(C(N3C(CCC(=O)NC)CCCC3)=O)CCC(C)(CC1)O2 12204,c1(CC(=O)NCC2CC2NC(=O)CCN(S(=O)(=O)C(F)F)C)cccc(OC)n1 12205,N1(n2c(-c3cccc(-c4cnc(C)[nH]c4=N)c3)ncc2)CC(C)CCCC1C 12206,N1(C(c2c(CNC(c3cnc(CC)s3)=O)ocn2)=O)CCCN(C)CC1 12207,c1(C(N(CCCNC(C)=O)C2CC2)=O)cnc[nH]c1=N 12208,c1(NC(CCC=CCC=C)=O)ccc(NC(=O)C(O)P(C)(C)=O)cc1C 12209,N1(C(c2c(CCC)[nH]cc2)=O)CC2CC(C1)N(C(=O)Cc1cc(O)nnc1O)C2 12210,c1(C(C)C)nc(Cl)cc(=NCC(C)NC(=O)CC2CC(F)(F)C2)[nH]1 12211,N1(C(=O)C(N2CCCC2)C2CC2)CC23COCC2(COC3)C1 12212,c1(OC)ccc2cc(C(=O)NCCCOCCNC(=O)C(C)OC3CC3)[nH]c2c1 12213,c1(CC(=O)N(CC)CC2CCCN2C(=O)CC2OCCCO2)ccc(F)c(C)c1 12214,CS(=O)(=O)c1ccc(CC(=O)NC2CC2(C(=O)O)C(=O)O)cc1 12215,C1(C(=O)NC(CCC)CCC)CCCCN(C(=O)CC2C=CCCC2)C1 12216,c1(C(=O)NCCCOCCNC(c2cc(CC)sc2)=O)nccn2nccc12 12217,c1(N(C(CSCC#C)=O)CCNC(=O)C(C)(C)OCCC)ccccc1NC 12218,N1(C(c2c(CC)noc2)=O)CCC2(NC(c3occ(C)c3C)=O)CCCCCC12 12219,C1(C(=O)NC2C(C(=O)NCC3(OCC)CN(C)C3)CCOC2)C2CCC(C2)C1C 12220,C12(C(N(c3cc(C)nn3C)C)=O)CCC(C(=O)NCc3ccccc3F)(CC1)C2 12221,C1(C(CCO)=O)(NC(C2CCCN(C(=O)CCN3CCC(F)C3)C2)=O)CCCCC1.CO 12222,C1(N(C(=O)C(C2CC2)N(C)C)CCOC)CCN(C(C2CS(=O)(=O)C2)=O)CC1 12223,C1(NC(CCSCC(N)=O)=O)CCN(C2CCN(C(C3CC=CCO3)=O)C2)CC1 12224,Cc1cccc(Br)c1C(=O)NC1CCCC1C(=O)Nc1c[nH]nc1C#N 12225,c1(NC(C2CN(c3ncnc4ccsc34)CCC2O)=O)ncc2c(n1)CCC2 12226,CC(C(=O)N(CCNC(C1CC(CC(C)(C)C)C1)=O)C1CC1)OCC1CCCO1 12227,C(=O)(C(F)CCC)NCC(c1ccccc1)CNC(CCOCCC)=O 12228,N1(C(C(CC)OC)=O)CCC(C(N2CC(C(C)C)C2)=O)C1(C)C 12229,CC(C)(C)C#CC(=O)NCC1CCCCC1C(=O)NOCCC(F)F 12230,c1(OC(C)C)ccc(NC(=O)NC(C2CCCCCC2)CO)c(C(C)C)c1 12231,c1(C(N(CCN(C(c2c(C)cns2)=O)C)C)=O)cnc2c(cnn2CC(C)C)c1 12232,CC1CCN(C(=O)C(c2ccc(F)c(F)c2)(C)C)CCN1C(C1CCCOC1)=O 12233,C(C(C)C(F)F)N(C(CCN(C(C(C)=CCC)=O)C)=O)CC(C)C 12234,N1(C(CCC(C)C)=O)CC(O)(C2(CNC(c3cccc4ccnn34)=O)CC2)C1 12235,Cc1c(C(=O)NCC(C)(C)NC(=O)C(C)C2CCOC2)[nH]c2c1CCCC2 12236,C(=O)(CC1=NNC(=O)C1)N1CCN(C(c2c(C)oc(CCO)c2)=O)CC1CO 12237,c1(C(N(CCCNC(=O)COC(C)=O)CC)=O)cc2n(n1)CCCNC2=O 12238,CC(CF)C(=O)N(C(CNC(c1ncc(C(F)F)s1)=O)C1CC1)C 12239,Cc1nscc1C(=O)NC(C1CCN(C(=O)CC2CCCN2C(C)C)C1)(C)C 12240,CC1CC2CN(C(C3CCC(NC(=O)CC4CCCO4)C3)=O)CCN2C1 12241,Cc1nc(=NCC2(CCNC(c3ccc(N(C)C)cn3)=O)CC2)[nH]cc1[N+](=O)[O-] 12242,c1(C(=O)NCC(C2CCCN2C(c2cc[nH]c2)=O)(C)C)nc(C2CC2)ncc1Cl 12243,C1(C(=O)NC2(CO)CN(C(c3ccc(C)c(Br)c3)=O)C2)CCn2ccnc2C1 12244,Cc1cnc2n1CCC(C(=O)N(CCNC(=O)C=Cc1cn(C)cn1)C1CC1)C2 12245,CC(CC(=O)NCC1(C(C)(C)O)CN(C(=O)CC2CC=CC2)C1)P(C)(C)=O 12246,[N-]=[N+]=NC1CCN(C(=O)C(C2CC2)NC(C2C=CCS2)=O)CC1 12247,c1(OCC)ccc(CN(c2ccc(C(=O)OC)c(C)c2)C)cc1OC 12248,C(=O)(CCN(OC)C(=O)CS(N)(=O)=O)N(c1cccc(OC)c1)C 12249,N1(C(c2ccc(C)c(C)n2)=O)CCC2(CCCN(C(c3cnc(=N)[nH]c3)=O)C2)C1 12250,C12(NC(C(c3cccc(Cl)c3)CC)=O)COC(C)(C1)C2 12251,C(=O)(C1=Cc2cc(Cl)ccc2OC1)N1CC(C)N(C(=O)C(N)=O)CC1C 12252,C1(C(=O)NCc2cc(C)on2)CCC(NC(=O)Cc2ccccc2Br)CC1 12253,C1(CC=C)(NC(=O)CNC(=O)OC)CCCN(C(=O)C=Cc2cccc(Cl)c2)C1 12254,C1(NC(C(C)C)=O)CCCCCC1C(=O)NCCCOC(=N)O 12255,C=C(Br)CC(C)(C)C(=O)NC1CCCN(C(C2(C#N)CCOC2)=O)CC1 12256,C1(NC(c2nc(CCC)oc2)=O)CCC(C(=O)NC2C(C)CCC2C)CC1 12257,C1(C(N(C)CC2CCN(C(C3CCN(C(C)=O)CC3)=O)C2)=O)CCC2(CC1)CC2 12258,N1(C(=O)CC2CCCC2)CC(C2CC2)(C(N2CCCC(CO)CC2)=O)C1 12259,c1(CC)cnc(C)c(NC(=O)C(CCNC(=O)CP(C)(C)=O)OC)c1 12260,c1(OC)nscc1C(=O)NC(CO)C(=O)NCCC1CC(C)(C)C1 12261,c1(C(N2CC3(CCCCN3C(c3ccns3)=O)C2)=O)cc2cc(F)cc(F)c2[nH]1 12262,C(=O)(N=c1cc2ccccn2[nH]1)C1N(C(Cc2c(C)n[nH]c2)=O)CCSC1 12263,C(CCN=c1ccnc(Cl)[nH]1)NC(c1coc(C2CCOCC2)n1)=O 12264,CCC(C)(C)C(=O)N(C)CC1CCN(C(c2cnc(SC)nc2)=O)C1 12265,C#Cc1ccccc1CC(=O)NCC(O)CNC(C1OCC1(C)C)=O 12266,N1(C(CC#N)=O)CCC2CCN(C(=O)CCn3ccnc3)CC2C1 12267,C1(C(N2C(C)C(NC(c3cc(O)nn3C)=O)CCC2)=O)CCc2cnn(C)c2C1 12268,N1(C(COCCC)=O)CCOCC1CCCNC(=O)COCc1ccc(C)cc1 12269,C(CC(F)F)(C(=O)NC(c1cccs1)C)NC(Cc1cc(C)nn1C)=O 12270,c1(NCc2cn(CC(=O)NCCN3CCC(OC)C3)nn2)ncc(N)cc1C.OC 12271,N1(C(C(c2ccccc2)NC(C)=O)=O)CCC(C)(NC(=O)CC2(O)CCC2)C1 12272,Cc1oc(Cl)nc1C(=O)N(C(C)CCNC(=O)Cc1ccccc1O)C 12273,C12(C(N3C(C#C)CCC3)=O)C(NC(C3CCC(N(C)C)C3)=O)C3CC1C2C3 12274,C1(C)(CC)CCC(C(=O)N(C2(CC(=O)NC(C)(C)CCCO)CC2)C)O1 12275,C1(C(NOCC(C)(C)C)=O)CSCCN1C(=O)Cn1ccccc1=O 12276,CN1CC(C(N2CCCC(NC(=O)CCCc3ccsc3)C2)=O)CC1=O 12277,C(=O)(C1=C(C)CCCC1(C)C)N1CC(CNC(C(CCCC)(C)F)=O)OCCC1 12278,c1(C(CC)C)ccc(-n2cc(-c3sc(C4CC4)cc3C)nn2)cc1 12279,C1(NC(c2c(CC)nn(C)c2)=O)C2CC3CN(C(=O)CC4CN(C)C4)C1C3C2 12280,c1(C(N(CCOC)CCNC(c2cccnn2)=O)=O)c(O)ncc(Br)c1C 12281,N1(C(C2C(C)(C)OCC2)=O)CCOC(C(N2CC(c3ncccn3)C2)=O)CC1 12282,C(C(=O)N(CCC(=O)N1CCC(F)(F)C(OC)C1)OC)(C1CC1)OC 12283,Cc1cc(C(=O)NC(C(N2CCCC2CF)=O)C2CC2)sc1C 12284,C1(N(C(c2cc(CC)on2)=O)C)CCCN(C(c2ccn(CC(C)C)n2)=O)CC1 12285,C1(NC(C(c2ccccc2F)(C)C)=O)CCN(c2nnc(CO)o2)CC(O)C1 12286,N1(C(c2ccn(C(C)C)n2)=O)CCCC(NC(=O)CC2COCCN2C)C1 12287,Cc1ccc(OCCNC(=O)Cn2nnc(-c3nc(C(C)C)no3)c2C)c(C)c1 12288,c1(CC)cc(C(=O)N(CCCN(C(=O)CSC(F)F)C)C)sc1C 12289,C1(NC(C(=O)NCCCOC(C)=O)=O)CCOCC1 12290,C1(CNC(C(COC)(C)O)=O)CC2CCC1N2C(c1cc(C)cc(C)n1)=O 12291,N1(C(C2(CC)CCC2)=O)CCOC(C)(CNC(=O)CC2CC(=O)NC2=O)C1 12292,Cn1c(NC(C2CCCC2C2CC2)=O)nc2cc(Br)ccc12 12293,N1(C(C(=O)NCC(F)C2CCC2)=O)CCC(O)C(F)(F)C1 12294,CCCCC(C(=O)NCCn1cncn1)NC(c1cn[nH]c1)=O 12295,S(=O)(=O)(c1cnc(N(C)Cc2ccnn2C)cc1C)NC1CC(CC)OCC1 12296,CCCC(CC)C(=O)NCC1(F)CC(NC(c2cc(O)ncc2Br)=O)C1 12297,c1(CNC(N2CCC(C(N(C)C)=O)C2)=O)ccc(N2CCCS2(=O)=O)cc1 12298,Cc1cc(C(=O)N(C(CNC(C2(CC3CC3)CC2)=O)C2CC2)C)n[nH]1 12299,N1(C(C2CCN(C3CC3)C2=O)=O)CC2(CCN2C(c2ccc([N+](=O)[O-])[nH]2)=O)C1 12300,CC1(CNC(c2cnn[nH]2)=O)CCN(C(c2c(Br)cnn2C2CCC2)=O)C1 12301,S(=O)(=O)(c1ccc2[nH]c(=NCCCF)sc2c1)N1CCN(C)C(CO)C1 12302,C1(CNC(C=CCC)=O)CCC2(CN(C(=O)C(c3ccccc3)SC)C2)O1 12303,C1(NC(CC(CC)C)=O)CC12CCC(NC(c1cccnc1C(F)F)=O)CC2 12304,c1(C(=O)NC2CC(NC(C(CCC)O)=O)C(O)C2)cccc2ccc(C)nc12 12305,c1(C(N2CC(O)CC2c2cccc(C(F)(F)F)c2)=O)cc2c(F)c(Cl)ccc2[nH]1 12306,c1(N2CC(NC(=O)NOCc3cc(Br)co3)C2)ccccc1 12307,N1(C(C2CC(C)(CC)C2)=O)CCCC(C(C)(C)C(=O)NCc2ccc(C#N)o2)C1 12308,N1(C(=O)CCN2CCCCC2)CCN(C(c2cn3ccnc3s2)=O)C2COCC12 12309,c1(C(C)OCC)nc(C)c(NC(=O)N(C(C)C(=O)N2CCCC2)CCC#N)s1 12310,C1(CCC)CN(C(c2cnns2)=O)CCN1C(=O)CN(C)C(c1cccs1)=O 12311,Cc1ccc2nc(SCC(N3CC4CCN(C(=O)C(C)CO)CC4C3)=O)[nH]c2c1 12312,c1(SC)nc(NC23CCC(CC2NC(=O)CCCCCSC)C3)cc(C(F)F)n1 12313,C(CCC(=O)NC(C)CN(C)C(c1cc(-c2cccnc2)[nH]n1)=O)N(C(C)C)C 12314,N1(C(C(C)SC(C)C)=O)CCC(C)(C)C1CC(=O)NCC1CCCCC1 12315,C1(C(=O)NC2CC(CCC)C2)(CCNC(=O)CCCc2sccc2C)CCCC1 12316,N1(CCC(=O)NCC2(CN(C(C(CC)C)=O)C)CC2)CCCCC1C 12317,N#Cc1ccccc1SC(c1cccc(NC(=O)N(O)Cc2cccc(Cl)c2)c1)=O 12318,C1(C)(C(=O)NCC2(C(C)NC(C(COC)OC)=O)CC2)CC(F)(F)C1.N(C)(C)C 12319,N1(C(C2(SC)CCC2)=O)CCC(O)(C(C)NC(=O)COC2CC(F)(F)C2)CC1 12320,C(c1cc2ccccc2o1)=CC(=O)NCC1CC(NC(CC=CC)=O)C1 12321,c1(CN2CCC(CNC(C(c3ccc(OC)cc3)O)=O)C2)ccc(F)c(F)c1 12322,CC1CCOCC1C(=O)NC1(C(=O)NOCc2ccccc2Cl)CCCCC1 12323,c1(CN(CCOC)C(=O)NCCSc2ccc(N)cc2)ccccc1Cl 12324,c1(CN2CCC(NCc3ccc(C(F)(F)F)cc3)C2)cc(N)c(Cl)cn1 12325,CCC(C(=O)NCCOCCNC(c1ccc(N)c(Br)n1)=O)C(C)(F)F 12326,C(=O)(CC(C)C(C)C)N1CCC(C(=O)NC(C(=O)OC)(C)CO)C1 12327,c1(C(=O)NC2CCN(C(c3cc[nH]c3)=O)CC2O)cnc2ccc(F)cc2c1 12328,c1(C(N(C2CCN(C(c3c(CC)nc[nH]3)=O)C2)C)=O)nc2cnccc2s1 12329,CCC(C)(C)C(O)C(=O)NC1(C(=O)NCC2CCC(C)(C)CO2)CCOCC1 12330,CCC(C)C(O)C(=O)N1CCCC(C)(CNC(=O)C(C2CCCCC2)C)C1 12331,c1(C(=O)NCC(C(C)C)NC(C2(C)CSC2)=O)cc2cc(F)cc(F)c2[nH]1 12332,C1(N(C(COCc2onc(C)n2)=O)C)CN(C(=O)C(C)CC2CCC2)CC1F 12333,CCC(CC(=O)N(C1CC(NC(c2cc(Cl)ns2)=O)C1)C)C(C)(C)C 12334,C(=O)(C(CC)(CC)C(=O)O)Nc1c(C(=O)OCC)cc(OCC)cc1.C(=O)OC 12335,c1(C(N(C2CCN(C(c3ccc(C)cn3)=O)C2)C)=O)ccc(C)c(F)c1N 12336,CCC(CC(F)F)C(=O)N1CC(OC)CC(NC(=O)CCNC(N)=O)C1 12337,N1(C(CN(CCCCCC)C)=O)CC(CNC(C2(CO)CC2(F)F)=O)C(O)C1 12338,N1(c2cc(NCP(C)(C)=O)nc(C)n2)CCN2C(=O)COCC2C1 12339,c1(C(=O)NC2CCN(C(c3c(C)ccnc3C)=O)CC2O)cccc2c1COC2 12340,c1(C(=O)NC2C(CNC(C(CCC)CC)=O)CC2)cc(C)c(Br)c(C)c1 12341,C(=O)(C(F)C(F)(F)F)NC1(CC(=O)NC2CCC(C(N)=O)CC2)CCOCC1 12342,C1(N(C(CC2CC(CC)C2)=O)C)CC2CC1N(C(c1csnc1C)=O)C2 12343,c1(C(N2CC(C(=O)NCc3ncccn3)C(F)(F)C2)=O)ccc2nccn2c1 12344,C1(C2CCN(C(C3CCCCCS3(=O)=O)=O)CC2)(NC(C2CCCC2)=O)CCC1 12345,N#CC1(c2ccc(CC3CCN(C(=O)C=C4CCC4)CC3)cc2)CCCC1 12346,N1(C(c2cc(OC)n[nH]2)=O)CC2COCCC2(NC(=O)Cn2ccc(C3CC3)n2)C1 12347,N1(C(C2C(COC)(COC)C2)=O)CCOC(C)(CNC(c2cc(CO)no2)=O)C1 12348,N1(C(C(C)CC2CC2)=O)Cc2ccccc2CC1CNC(=O)C(C)C(C)(F)F 12349,N1(C(C2C(=C)CC2)=O)CC2(CCC2)CC1CNC(=O)COc1ccccc1Br 12350,C1(C(=O)NC2CCCN(C(C=C(C)CN3CCOCC3)=O)C2)CC2CCC(C1)S2 12351,C1(CN(C(C2(CC)CN(C(=O)CCc3ccc[nH]3)C2)=O)C)CCCCC1O 12352,C1(C(N2CC(CC(C#C)C)C2)=O)CC2CCCC2N1C(=O)C(CC)NC(N)=O 12353,C1(OC)CCC(C(=O)N(C(C)(C(=O)NC(C)CC(C)C)C2CC2)C)CC1 12354,N1(C(C(C)C(F)F)=O)CCC(C)C(N(C)C(c2cc(C(F)(F)F)ccc2F)=O)C1 12355,O=C(CC(F)(F)C(F)(F)F)NC1CCCCC1NC(C12CCCC1C2)=O 12356,C#Cc1ccc(CC(N2CCN(C(C)=O)C(CS(C)(=O)=O)C2)=O)c(F)c1 12357,C=CC1(C(=O)NC(C)CN2CCCC2)CCN(C(C2OCCC2(C)C)=O)CC1 12358,N1(C(CCC#CC)=O)CC(NC(=O)C(O)Cc2ccc(F)cc2)CC12CCCC2 12359,N1(C(CSCCCC)=O)CCC2(CC1)OCCC2NC(=O)CSc1n[nH]c(O)n1 12360,C1(C(=O)NCC(C(=O)NC(C2CCOC2)(C)C)CC2CC2)CC2(CC(=O)C2)C1 12361,c1(C(N2CCC(N(C(CC3CCC(C)O3)=O)C)CC2)=O)cc(N)nc(Cl)c1 12362,N1(C(CCC=C=C)=O)CCCC(O)(CCNC(=O)CCN2CCC(F)C2)C1 12363,C1(NC(c2ccn(CCC)n2)=O)CCC12CN(C(=O)CCOCC)C2 12364,CCCC(C(=O)NC(C)CC(N)=O)NC(=O)C(C)N1CC(C)C1 12365,C(=O)(C1=CCCC1C)NC(C(=O)NC1CCCN(C(C)=O)C1)CCN(C)C 12366,C12(NC(c3cc(C)c(Cl)cn3)=O)CCCC1CN(C(C1CN(C(C)C)C1)=O)C2 12367,CCC(CC)C(C(=O)N(CCNC(C1(O)CCCC1)=O)C1CC1)N1CCOCC1 12368,N1(C(C(C)=C2CCC2)=O)CCN(CC(=O)N(CC(F)Cl)C)CC1 12369,N1(C(CNC(C2(CC(C)C)COC2)=O)=O)CC(C)(NC(C(N)=O)C2CC2)C1 12370,N1(C(CNC(C2C(CCC)C2)=O)C)CCN(C(=O)Cc2ccn(C)n2)CC1 12371,N1(C(c2cc(C)no2)C(=O)NCC(F)F)CCc2cc(C#N)ccc2C1 12372,c12ccc(cc1)OC2C.Cc1nccn1Cc1nccn1C 12373,Cc1nc(Br)cnc1NC(c1c(NS(=O)(=O)CCCN(C)C)cccc1F)=O 12374,N1(C(C2CCC(C)CC2)=O)CCC(NC(C2(n3cncn3)CC2)=O)C(O)C1 12375,c1(OC)cc(C(N2CCC(NC(=O)C(Cl)=CCl)CC2C)=O)ccc1[N+](=O)[O-] 12376,N1(C(CC=CC)=O)CCN(C(=O)C(C)C(=O)N)C(CC)C1.c1(SCC)ccc(C)cc1 12377,C=C(C)CN=C(NCC(C1CCCCCC1)(C)O)NCC1CCC(C2CC2)O1 12378,n1(CC(C)C)ncc2cc(C(=O)NC3CC3Sc3ccccc3)cnc12 12379,C(=O)(C(CC(C)(C)C)OC)N1CCCC(CC)C1C(=O)NCc1scnc1C 12380,N1(c2ccc(CNCCc3n(C)ncc3)cc2)CCCCCCC1 12381,C1(NC(CC=C(C)C)=O)CCCCCCC1NC(c1cc(C)nn1C)=O 12382,c1(C(N(CC(CC)C)C)=O)coc2c1CN(C(C1CC1C(F)(F)F)=O)C2 12383,C(=O)(C(O)C(C(C)C)OC)NC(CNC(C(CC)N(C)C)=O)COC 12384,C(N=c1[nH]c(N2CCCC(C(N)=O)(N(C)C)C2)nc(=N)[nH]1)C1(OC)CCCSC1 12385,C1(F)(C(N2C(C)(c3ccc(C(F)(F)F)cc3)CCC2)=O)CC2CCC1CC2 12386,C1(N(C(c2c(C)nccc2)=O)C)CN(C(C2CC3C=CC2C3)=O)CC1(C)C 12387,c1(NC(C2CC(OC)C2)=O)nc(C)cc(C)c1C(F)(F)F.C12CN(C3CC13)C2=O 12388,Cc1ccsc1CCCC(=O)NCC(CO)NC(=O)CN1CCCC1 12389,C12(CNC(CS(=O)(=O)NC)=O)CCCC1CN(C(c1cc(C)co1)=O)C2 12390,Cc1csc(=O)n1CC(=O)NC1C2CC1N(C(c1sccc1SC(F)F)=O)C2 12391,c1(C(N(c2ccc(C)c(C)c2)CCC)=O)ccc2cnccc2c1O 12392,C(CCC(=O)NCC1CC1CNC(c1cnn(C2CCC2)c1)=O)OCCOC 12393,Cc1cnn(C)c1C(=O)NC(C)C(C1CCCCC1)NC(c1ccsc1)=O 12394,C1(C(=O)NCCN(C(c2cc(C(=O)OC)nn2C)=O)C)CC12CCc1ccccc12 12395,N1(C(c2ccc(OC)s2)=O)CC(NC(C2CCN2C2CCCC2)=O)CC12CCCC2 12396,N1(C(C2(C)CCN(C(Cc3cccc(SC)c3)=O)C2)=O)CCCC(C)(O)CC1 12397,c1(C(=O)NCC2CN(C(C3C(C)OCCO3)=O)C(C)(C)C2)c[nH]c2ccccc12 12398,C(=O)(C1=NNC(=O)C1)NC(C(=O)NCCCCCOC)C1CC1 12399,O=C(C1=CCCOCC1)NC1CN(C(c2cc(Cl)ns2)=O)CCC1O 12400,CC1CC(NC(c2cn(CCCC#N)nn2)=O)CN1C(=O)CCC(F)F 12401,N#CCCCCCC(=O)NC1CC2CCC1CC2NC(C1CCS(=O)(=O)CC1)=O 12402,C=CC1CCCC(NC(C2CC(C)(NC(=O)C=CC(C)CC)C2)=O)C1 12403,N1(C(c2ccc(OC)c(C(C)(C)C)c2)C(=O)NC)CCN(S(C)(=O)=O)CC1(C)C 12404,C(=O)(CCCC(=O)N1CCC(C(C)NC(=O)CC2CCC(C)(C)CC2)C1)OCC 12405,c1(C2CCN(C(CSCCOC)=O)CC2)ccccc1NC(=O)C(C)C1CC1 12406,N1(C(COC(C2CN(C)CCC2O)C)=O)C2CCC(C2)C1C(=O)OC(C(C)(C)C)=O 12407,C1(CNC(=NCC)NCCC(C)(C)C)CC2(CC2)S(=O)(=O)N1 12408,Cc1ccc(C=CC(N2CCC3(CC3C(=O)NCC3(CC(N)=O)CC3)C2)=O)cc1 12409,C(=O)(C1CCOc2c(F)cccc21)NC(CC(C)NC(C1CC2C=CC1C2)=O)C 12410,C1(NC(COCCC#C)=O)CCCOC12CCN(C(C1(O)CC1(C)C)=O)CC2 12411,Cc1cccc2c1c(CNC1CC(NC(=O)C(O)C(C)C)C1)cn2C 12412,N1(C(C2(CNC(C3CC(=C)C3)=O)CCCO2)=O)CCN(C)C(CC)C1 12413,c1(C(N(C2CCN(C(=O)COc3ccccc3)C2)C)=O)c(N)cnn1C 12414,c1(C(N(CCC(C)NC(c2ccc([N+](=O)[O-])cc2)=O)C)=O)cc2c(ccn2C)[nH]1 12415,C(=O)(CC(CC)C(C)C)NC1C2(CN(C(c3nc(CC)sc3)=O)C2)CC1 12416,C(N=c1nc2c(ncn2C)c(NCc2ccoc2C)[nH]1)C1(CCC)CC1 12417,c1(C(=O)NCCCNC(CC(CCC)(C)O)=O)cc(S(=O)(=O)CC)cnc1O 12418,Cn1cc(C(N2CCC(OCC(=O)NC3(CCF)CCC3)C2)=O)cn1 12419,c1(OC)cc(C)ccc1OCC(=O)NCCC(C)NC(=O)C(C)S(N)(=O)=O 12420,CC(C)C(C(C)NC(c1c[nH]nc1C1CC1)=O)NC(=O)CCN(CC(F)(F)F)C 12421,N1(c2nnc(C)s2)CC2(C1)SCCC2NC(C1CC(=O)N(C(C)C2CC2)C1)=O 12422,CC1NC(=O)CCC1CNC(=O)CCN(C(=O)C1=NOC(C)C1)C 12423,C1(N2CCC(N(C(=O)CC3CCCCCC3)CC3CC3)CC2)CCC(=O)NC1=O 12424,C12(C(=O)NCC3=CCN(C(CSCCC#N)=O)CC3)CCCN1S(=O)(=O)CC2 12425,c1(CC(=O)N(CC(C)N(C(C(CCC)OCC)=O)C)C)cc(F)cc(Cl)c1 12426,N1(CC(C)C)N=C(C(=O)N2CCCN(C(=O)C(C)N(C)C)C(CO)C2)CCC1=O 12427,N#CC1(C(=O)NC2CC(CNC(=O)C=C(Cl)Cl)C2)CC2(CC2)C1 12428,Cc1c(C(=O)NCC2(F)CC(NC(=O)CN(C)C)C2)[nH]c2ccc(C(C)C)cc12 12429,Cc1cnc(C=CC(=O)NC2CCC(CNC(c3ccnc(C)n3)=O)CC2)[nH]1 12430,N1(C(c2ccnc(F)c2)=O)CCC(F)(F)C(CNC(C23CCCC2C3(F)F)=O)C1 12431,Cn1nc(C(N2CC(O)CC2(C)C(=O)NOCC(O)C(C)(C)C)=O)ccc1=O 12432,C1(CNC(C2(C)CC=CCC2)=O)CC12CCN(C(C13CC(CO)(C1)C3)=O)CC2 12433,c1(C(=O)NC2C(C)CCN(C(CCc3c(C)ncs3)=O)C2)ccc2n[nH]cc2c1 12434,c1(OC)cccc(N2CC3CCC2C(NC(C2CC(=O)N2)=O)C3)c1[N+](=O)[O-] 12435,CP(C)(=O)c1cc(C(=O)NCC2CCCN(C(=O)CNC=O)CC2)ccn1 12436,c1(C(N2C(CNC(c3cnc(C)s3)=O)CC(O)C2)=O)cccc(CO)c1C 12437,C1(NC(COCCSC)=O)CCCC1CNC(=O)CCC1CCN(C)C1 12438,Cn1cc(C(N2CC3CC3(C(=O)NCC(=C3CCCCC3)F)C2)=O)n(C)c1=O 12439,CCC(C)C(C)(O)CNC(C1CC(CNC(c2ncn(CC)n2)=O)C1)=O 12440,c1(C(C(=O)NCC(c2ccccc2)N(C)C(c2cnco2)=O)O)ccccc1Cl 12441,N1(C(CCCOc2ccc(C)cc2)=O)CC2(CCC2N(C)C)C1 12442,CC(=O)CCCC(=O)N(C)CC1CCN(C(=O)COCc2ccnc(O)c2)C1 12443,N1(C(=O)COC2CCCCC2)CCC(CNC(C2(F)CC2)=O)C12CCC2 12444,C12(C(=O)NCC(CNC(C3(CC(F)F)CCC3)=O)OC)CC(C(C)C)(C1)C2 12445,C1(O)(CC(=O)OCC)CCN(C(=O)C(C)c2ccsn2)C1 12446,c12cccc(c1)NC(=O)NC2.N1(CC(C)C)CCC(NC2CC2)C1 12447,C1(CC(=O)NC(Cn2cncn2)C(=O)NCC2CC2Cl)CNC(=O)O1 12448,CC#CCC(C(=O)NC(c1nc[nH]n1)CO)NC(=O)C(CC1CCC1)OC 12449,C(=O)(C(F)C(=O)NC1CN(C(=O)Cc2nncn2C(C)C)CC1C(F)F)OCC 12450,C(=O)(N=c1[nH]onc1C1CNC(=O)N1)c1ccc(C(C)Nc2ccc(Br)nc2F)s1 12451,N1(C(C)=O)CCN(C(=O)C(Cc2ccco2)NC(=O)Cc2coc(C)n2)C(C)C1 12452,C1(CC=C)(NC(c2cc(COC)on2)=O)CCN(C(C2CSCCS2)=O)C1 12453,C1(CC)C(NC(=O)COC2CCCC2)CCCN1C(=O)C=Cc1cnccc1C 12454,c1(OC)ccc(-c2ncc(C(=O)N(C)Cc3cnc(C)s3)s2)cc1 12455,C1(NC(CSc2n(C)ccn2)=O)CCC2(CC1)CCN(C(=O)CC1CC1(C)C)C2 12456,N1(C(C(CN=[N+]=[N-])NC(C2CC2OC(C)(C)C)=O)=O)CCn2nncc2C1 12457,CC1OC2(C(=O)NC3C=CCN(C(c4c(F)cccc4F)=O)C3)CCC1CC2 12458,c1(C(N2CC(C)C(CNC(c3cc(Cl)no3)=O)CC2)=O)ccc2ncccn12 12459,C1(C(N(CCCN(C(C(c2cccnc2)OC)=O)C)C)=O)CC1C1CC1 12460,c1(NCC(C)OC(F)F)ncccc1S(=O)(=O)NC1CCc2ncsc2C1 12461,c1(C(=O)OCC)c(NC(C2CCN(Cc3ccc(Cl)o3)CC2F)=O)cccc1Cl 12462,N1(CCNC(C(CC2CCCC2)OC)=O)CCN(C(C23CC(F)C2C3)=O)CC1 12463,C=CC1(CC(=O)N(C)Cc2scnc2C)CN(C(C2CC(C)(C)CO2)=O)C1 12464,C1(COC)CC2CC2N1N1CC(NC(=O)OC(C)(C)C)C(C)C1 12465,C(CCc1ccc(F)cc1)(C(=O)NCCCC1CC1)N(CCOCCC)C 12466,C=CC1(C(=O)NC(c2nn[nH]n2)C2CC2)CCN(C(=O)C=CCC)C1 12467,c1(C(CNC(C2N(C(c3ccccc3)C)CSC2)=O)(C)C)ncccc1F 12468,CC1CCC(C)(C(=O)N(CC(C)CNC(=O)C(O)Cc2ccccc2)C)C1 12469,c1(C(=O)NCC2CC(NC(c3cc(SC)c(C)o3)=O)C2(C)C)ccc(N)cc1Cl 12470,CC1C(C(=O)N(C2CCOC2=O)C)CCCN1C(c1ccc(F)cc1)=O 12471,c1(N2CCC(CC=C)C2)cc(Br)ccc1S(=O)(=O)N1CCOCCC1 12472,C1(NC(c2c(C)nco2)=O)CC2CCC(C1C)N2C(=O)C(C)S(N)(=O)=O 12473,c1(C(N2CC3C(CCNC(=O)CSC(F)(F)F)(CC3)C2)=O)cnc2cc[nH]c2c1 12474,N1(C(c2c(CC)nccc2)=O)CCCC(C)(C(=O)Nc2cc(Br)cnc2Br)C1 12475,CON(C)C(=O)CN=C(NCC(C)(C)C)NCC1CCOC1C 12476,c1(OC)cccc(C(C)NC(=O)NC(C(O)CO)c2ccccc2)n1 12477,CC1CSCCN(C(c2cnn(CCNC(=O)CC3CC(F)C3)c2)=O)C1 12478,CC1CC(CNC(C2(F)CCCCC2)=O)CN1C(=O)CCc1cscn1 12479,C(CC(O)C(=O)N1CCCC(NC(c2cnnn2-c2ccccc2F)=O)C1)SC 12480,c1(OC)ccnc(NC(c2cnc(-c3cc(O)cc(F)c3)cn2)=O)c1I 12481,C1(C(N2C(C(C)NC(c3ccc(Cl)cn3)=O)CCC2)=O)OCC2COCCC12 12482,C1(C(N2CC(c3cn(CC(=C)CC)nn3)(C(=O)OC)C2)=O)CC2C=CC1C2 12483,C1(NC(C=C(CCC)C)=O)CC2CCC(C1)N2C(=O)C(C(CC)CC)OC 12484,CC(C)C(CN(C)C)C(=O)NC1CCN(C(=O)CCC2CC2)CC1O 12485,C(CNCC(=O)OC)(CC(=O)N(C)CC1CN(C)CCO1)OCCCC#C 12486,C(CC(C)(C)C(=O)NCC1(C)CCN(C(=O)COc2ccc(Cl)cc2C)C1)OC 12487,N1(C(C(C(C)C)SC)=O)CCC(C)C(NC(c2cc(C(C)(C)C)n[nH]2)=O)C1 12488,N1(C(=O)C2=CSCS2)CCC2(CC1)CN(C(C1CC3(CCCC3)CO1)=O)C2 12489,C1(NC(c2ccc(CC)cc2O)=O)CC(NC(c2ccoc2)=O)C12CCOCC2 12490,CC1COC2(C1)CN(C(C1CC3CN(C(C4(C)CS(=O)(=O)C4)=O)CC3C1)=O)C2 12491,C1(CC(=O)NC(C(=O)OCC=C)(C)C)C2CCCC2N1C(=O)CCc1cnoc1 12492,N1(C(CC=C(C)C)=O)CCC2(CC1)CN(C(C1C3CCC1CC3)=O)CC(C)O2 12493,C(CC(C)C)(C(=O)N1CCCC(C)(C(N2CC(O)C(O)C2)=O)C1)NC(=O)OC 12494,C(C(C)(C)CNC(C1(OC(C)C)CCC1)=O)N(C(=O)CCc1conc1C)CC 12495,c1(-c2cc(OC)ncc2)nc(C(N2CCC(C(F)(F)F)C2)=O)ccc1F 12496,CCC(C)(CNC(C1(CNC(c2ccnnc2O)=O)CC2(CC2)C1)=O)C(N)=O 12497,O=C1CN(CC(N2CCC3CC23C(=O)Nc2cnccc2CO)=O)CCN1 12498,CC(C)C(O)C(C)C(=O)N1CC(NC(=O)C=CC(=O)NC2CC2)CC2(CC2)C1 12499,Cn1nc(C(=O)NCC2CC(NC(=O)C(c3ccc(Cl)cc3)(C)C)C2)ccc1=O 12500,c1(CC)n[nH]cc1C(=O)NCCC1CCN(C(=O)C(O)C2CCC2)C1 12501,Cc1cccc(N)c1C(=O)NC1CCC(NC(=O)CCC2CNC(=O)N2)CC1 12502,c1(C(=O)NCCN(C(=O)C2=CCCOC2)CCC)cc(C)ccc1OC.C(C)N 12503,C=CCC(C(=O)NCC1CN(C(=O)C(C(C)(C)C)NC(N)=O)CC1C)C(C)C 12504,CC1CC(NC(c2csnc2Cl)=O)CCN1C(C1CN2CCC1CC2)=O 12505,C1(C)(CNC(CS(=O)(=O)NCC)=O)CC(F)(F)CN1C(c1cc(C(C)=O)on1)=O 12506,c1(C(=O)NCC2C(C)(C)C(NC(=O)Cn3nccn3)C2)ccnc2ccnn12 12507,c1(C(=O)NCC2(C)CC(NC(C3COC(=O)O3)=O)C2)cc(Cl)cc([N+](=O)[O-])c1 12508,c1(C(=O)NCCCC2N(C(c3c(C)ccs3)=O)CCC2)ccccc1OC1CC1 12509,CC1=C(C(N)NC(C2CC(=O)N(C3CCCCCC3)C2)=O)NC1 12510,C1(C2CCN(C(c3ccsc3Cl)=O)C2)(NC(=O)Cc2ccc(F)cc2)CC1 12511,CC(C)CC(CNC(c1cscc1Cl)=O)C(=O)NCCNC(=O)N(C)C 12512,C1(N(C(c2cc(CCC)on2)=O)C)CCCN(C(=O)CC2C(CC)C2(F)F)C1 12513,c1(C(N(CCNC(Cc2cnc(C)s2)=O)C)=O)cc(F)c(C)cc1O 12514,C1(C)(C(N2CCC(CCNC(C3(C(=O)NC)CCC3)=O)C2)=O)CCCCO1 12515,N1(C(CSCCOC)=O)CCC2(CC(C(=O)N(C)Cc3ccc(F)cc3)C2)C1 12516,N1(C(C2C(C)CC2)=O)CCC(C(C)(O)CNC(c2nn(C)cc2Br)=O)CC1 12517,c1(OC)c(C)cc(C(=O)NCC2CCC(NC(=O)C(O)P(C)(C)=O)CC2)cc1C 12518,CC1CCc2nc(Cl)nc(N3CCCCC(NC(c4coc(Cl)c4)=O)C3)c2C1 12519,N1(C(C2N(C(C)=O)CSC2)=O)CCC12CN(C(=O)CN(C1CCCC1)C)C2 12520,C1(CC)CN(C)CCCN1C(C1COCC1NC(=O)C(F)C(C)(F)F)=O 12521,CC(C)(F)C(C)(F)CNC(C1COCCC1NC(=O)OC(C)(C)C)=O 12522,Cc1cc(C(F)F)n2ncc(C(=O)NCC(C(C)C)NC(=O)C3=CCCC3)c2n1 12523,C1(C(=O)NCC2CCS(=O)(=O)CC2)CC2C=CC1N(C(=O)Cn1cccn1)C2 12524,C1(C(N(CCNC(=O)CSC2CC2)CC)=O)CCn2ncnc2C1 12525,N1(C(CC2NC3CCC2C3)=O)CCCC2(CCC2)C1.CC1=C(C=O)CCC1 12526,c1(SC)c(C(=O)NC2CCC(NC(=O)C(N3CCCCCC3)C)C2)cccc1F 12527,c1(CC(C)NC(=O)C(N2CCC(N(c3ccccc3)C)C2)=O)ccccc1Cl 12528,C(=O)(C1CCc2snnc21)NCC1(CO)CCN(C(Cc2cnc(C)[nH]2)=O)C1 12529,N1(C(C(=Cc2cccnc2)C)=O)CCCC(C)(NC(=O)COC(F)F)C1 12530,N1(C(CCS(=O)(=O)NC)=O)CC2(C1)CN(C(=O)CC1CCC1C)CC2CO 12531,C1(NC(C2C3COCC23)=O)CN(C(=O)C=CCF)C2(CCC2)C1 12532,c1(CCNC(C=C(CNC(CCCOC)=O)C)=O)cccc(C)n1 12533,C1(NC(Cc2ncc(CC)[nH]2)=O)CN(C(=O)Cn2cnccc2=O)CC1CC 12534,c1(OC)c(Cl)cc(C(=O)N(CCC(C)NC(c2cc(C)oc2C)=O)C)cc1Cl 12535,N1(C(C(c2ccc(OC)cc2)CC)=O)CC(NC(c2occc2C)=O)CC(C)C1 12536,C(=O)(C(C)(C)C)NC(C)C(=O)NC(C1CCCC1)CNC(=O)C=Cc1ncco1 12537,c1(CC(=O)NCC2N(CC)CC2)ccc(S(C)=O)cc1 12538,CC1CC(NC(c2cc(N)ccc2Cl)=O)CCN1C(=O)C=Cc1ncc[nH]1 12539,C(c1ccc(C)c(Cl)c1)=CC(N1CCC(NC(C2C(C=C)CC2)=O)C(F)C1)=O 12540,N1(CC(=O)NC2CC(CCNC(C3(CO)CCCO3)=O)C2)CCCNC1=O 12541,c1(C(=O)OCCN(c2csc(C)c2)C2(CC)CC2)ccc([N+](=O)[O-])c(C(F)(F)F)c1 12542,CC(CCc1ccncc1)N=c1[nH]c2c(c(=NCCCCN(C)C)[nH]1)COC2 12543,N1(C(C(C)C)=O)CCCCC(C(=O)NC(=O)C(C)Sc2ccccc2)C1 12544,CCCCCCCCC(=O)NC1CC1NC(c1ccc(C(N)=O)s1)=O 12545,C(=O)(C1=C(Cl)CCOC1)NCCC1CC(NC(C=Cc2c(C)nccc2)=O)C1 12546,N1(C(CC(C)O)=O)CC(CNC(=O)CC2C=CCC2)C(F)(CO)C1 12547,C1(NC(CN(C)C(N)=O)=O)C2CCC1N(C(=O)Cc1cncc(F)c1)C2 12548,N1(C(c2c(C)noc2)=O)CCC2OCCN(C(c3cc4cccn4cn3)=O)C2C1 12549,n1(CCCC)nnnc1C(c1ccncc1)NCCSCC1CCCC1 12550,N1(C(c2c(CCC)n[nH]c2)=O)CC(CNC(c2ccn(CCF)n2)=O)CC1(C)C 12551,c1(NC(C(C2CCN(Cc3ccsc3)CC2)C)=O)cc(Cl)ccn1 12552,N1(C(C(C)OCC#C)=O)CCC(CNC(C2CCS(=O)(=O)CC2)=O)C(F)(F)CC1 12553,N1(C(CC2CC(C)N(C(=O)CC(C)(C)C3CC3)C2)=O)CC2C3CCC(O3)C2C1 12554,c1(OC(C)C(=O)NC(C)CC2CN(C(C3CSCN3C)=O)C2)ccc(F)nc1 12555,N1(C(c2cc(C)oc2C)=O)CCC(NC(=O)Cc2cc[nH]n2)C(CO)CC1 12556,c1(C(=O)NCC2CC(NC(=O)CSc3ccccn3)C2)cc2ccccc2o1 12557,C1(C(N(C)Cc2c(CNC(CSC)=O)cccc2)=O)CCOCC1(C)C 12558,C1(NC(c2cc(C)ncc2C)=O)CC2CN(C(C34CC(CO)(C3)C4)=O)CC2C1 12559,c1(N(C(CNC(C2(C)CC=C(C)CC2)=O)C)C)nc2cc(C)ccc2o1 12560,CC(C)(CCNC(C1CC2CC1CC2O)=O)C(=O)NCc1cnc(O)nc1O 12561,C1(OC)CC(NC(=O)C=CSc2ccccc2)CN(C(C2CCS(=O)CC2)=O)C1 12562,C(=O)(CCCC(=O)NC(=O)C=Cc1ccsc1)NC1C(CC(=O)OCC)CCC1 12563,Cc1ccc(C(=O)NCC2CC2NC(c2snnc2C2CC2)=O)c(Cl)c1C 12564,CC1(C(=O)NCC2CC(NC(c3cccc(CF)c3)=O)C2)CC2CC2C1 12565,Cc1ccc(CC(=O)NCC2CC2NC(=O)C(C)(C)c2ccns2)s1 12566,N1(C(CCc2c(C)cccn2)=O)CCC(CNC(C2CCCOC2)=O)C(C)C1 12567,C=CCC(CC(C)C)C(=O)NN1CC(O)CC1Cn1cc(CN(C)C)nn1 12568,C#Cc1ccc(C(=O)NC2CCC(NC(=O)Cc3cn(C)nc3C)C2)nc1 12569,N1(C(C(CN(C)C)N(C)C)=O)CCCC(CC(=O)NCC2CC(C)(C)CO2)CC1 12570,C(C1=NOC2CN(C(c3cccc4c3CCC4)=O)CC12)NC(C(CCC)(C)C)=O 12571,CC1CN(C(=O)Cn2ccccc2=O)CC(CCNC(C2CC(F)(CO)C2)=O)O1 12572,C(=O)(C(C)(C)C(C)(F)F)NCC1N(C(CC(CC)SC)=O)CCOC1 12573,c1(C(=O)NCC#CCNC(c2cc(CC)nnc2C)=O)cnc2ccnn2c1C 12574,N1(C(c2ccc(C)nc2C2CC2)=O)CCOC2(CCN(CC3CCC3)CC2)C1 12575,C1(C(=O)NC2CC(CNC(C3CC4(CCC4)C3)=O)C2)CC12CCCOC2 12576,C1(NC(C2CC=CCC2)=O)CC2CC1CN(C(=O)C=C1CCOCC1)C2 12577,CC1(C#N)CCN(C(=O)C(C2(O)CN(C(c3c[nH][nH]c3=N)=O)C2)F)C1 12578,N1(C(=O)OC(C)(C)C)CCCCCC1N=c1ccc(Br)n[nH]1 12579,CC1CN(C(=O)Cc2nc(C3CC3)n[nH]2)CC1NC(=O)CC1CC1 12580,CON1CCC(C(=O)NC(CN(C)C)C(=O)NCC2(F)CCOCC2)CC1 12581,C1(C(=O)NC2CC3(C(NC(c4c(C)nc(CO)s4)=O)C3)C2)COC2CCCCC12 12582,C(=O)(C(C)(C)C(C)O)NCCn1cc(CCNC(CSCCCC)=O)nn1 12583,c1(COC(C)C)ccc(C(=O)NCC2(C)CCCN2C(C2CC(C)=NO2)=O)cc1 12584,N1(C(C(C2(O)CCC2)NC(CCCC2C(C)C2)=O)=O)CC2CCC(C1)C2C#N 12585,C#CCC(C(=O)NCCCSC)NC(=O)C(=Cc1cn[nH]c1)C 12586,C1(SC)CCN(C(=O)CCOCCN(C(=O)C(C)Cc2cnc[nH]2)C)C1 12587,CN1CCN(C(c2sccc2CN)=O)C(CO)C1.C1(N2CC(=O)N2C)CCCC1 12588,C(=O)(C(C)S(=O)(=O)C(C)C)NCC(CNC(C(CC)(CC)CC)=O)C 12589,C1(c2nnnn2CCc2ccccc2)(NCC2(COC)CC2)CCCSC1 12590,c1(CC(=O)NCCN(C(c2cnccc2Cl)=O)CC)ccc(OC)c(C)c1 12591,C1(C)(N(C)C)CCCN(C(=O)C(c2ccnn2C)NC(=O)C=CCN2CCC2)C1 12592,N1(C(C2N(C(CC(C)=C(C)C)=O)C(C)CC2)=O)C2CCC1COC2 12593,CC1CCCC(O)(C(=O)NCC2(F)CN(C(c3ccc4cc[nH]c4n3)=O)C2)CC1 12594,c1(C(=O)NC2C(NC(c3c(C)cco3)=O)CC2)cc(F)c(F)c(O)c1F 12595,c1(C(=O)NC(C(=O)NCc2c(C)scn2)C2CC2)cnc(C)n1C 12596,CCCCC(S(=O)(=O)NC(=O)C(c1ccc(Br)nc1)(C)C)c1ccccc1 12597,CC(C)CC(C)(CNC(c1cc(Br)n[nH]1)=O)NC(c1ccc(Cl)o1)=O 12598,C=Cc1cncc(C(N2CCCC(O)(CNC(=O)OC(C)(C)C)C2)=O)c1 12599,c1(C(N2C(C(C)NC(C=CCCC)=O)CCCC2)=O)nc(C2CC2)ncc1Cl 12600,N#Cc1ccc(NC(CNC(c2ccc(C3CC3)cc2)=O)C2CC2)c([N+](=O)[O-])c1 12601,c1(C(=O)NCC2C3CN(C(CC4(C)CCCC4)=O)CC32)nncc2c1CCCC2 12602,N1(C(C(C)n2cncn2)=O)C2CCC1CC(NC(c1ncsc1Br)=O)C2 12603,c1(CNC(CC=C)=O)nc2c(s1)CCN(C(=O)CS(=O)(=O)N1CCOCC1)C2 12604,C1(F)(C(=O)NCC(C)NC(c2cc(-c3ccccc3Cl)no2)=O)CCCOC1 12605,C(CCC(=O)OC)SC1C(C(=O)OC)CC1.C1(=O)C(C)O1 12606,c1(OC)nc(Cl)ccc1C(N1CCC(NC(c2ncccc2C)=O)CC1C)=O 12607,N1(C(CCCn2cc(CC(C)(C)CO)nn2)=O)CC2CC2(CN2CCCC2)C1 12608,CCCCCC(CC)C(=O)NCC1CC1CNC(=O)Cc1c[nH]c2cccc(C)c12 12609,N1(C(c2cc(OCC)n[nH]2)=O)CCC2(C(=O)NC(C3CCOC3)C)CC2C1 12610,N1(CC(=O)NC2C3CC2N(C(c2snc(O)c2Cl)=O)C3)CCCCCCC1=O 12611,c1(C2(CNC(F)CF)CCCC2)ccc(Cl)cc1 12612,C=C(C)C(C)(C)C(=O)NC1COCC1NC(=O)CCC(=O)c1ccncc1 12613,N1(C(C(CC)OC)=O)C2CCC1CC(CC(C)NC(=O)CCc1ccnn1C)C2 12614,C(=O)(N1CCCc2ccnn21)C1C2(CCN(C(c3cc(OCC)no3)=O)C2)C1 12615,CC(C)CC(C)(CNC(=O)Cc1ccccc1)NC(C1CN(C)CC(C)O1)=O 12616,C(N=c1nc2c(c[nH]1)COCC2)C1CCCC(NC(c2ccc(C)c(F)n2)=O)C1 12617,C1(NC(C=C(C)C2CC2)=O)CN(C(C23CCCC(C2)OC3)=O)C2CCCCC12 12618,C(CCS(=O)(=O)c1ccc(F)cc1)NC(=O)NC(C1CC2CCC1C2)C 12619,c1(SC)cccc(N2CC(c3nc(-c4cnn(-c5ccccc5)c4)no3)CC2=O)c1 12620,C=CCC(C)(C)C(=O)N(CCCCCNC(c1ccnc(C(F)(F)F)c1N)=O)C 12621,C1(NC(C=CSC)=O)CS(=O)(=O)C2CN(C(c3cc(Cl)no3)=O)CC12 12622,Cc1nn(CC(=O)N(CCC(C)NC(c2cncc(F)c2)=O)C)cc1Br 12623,C1(C(N2CCC(O)(C(C)NC(=O)COCCF)C2)=O)CS(=O)(=O)CC(=O)N1 12624,c1(NCC2C(C)CCN(C(=O)C(C)CC3CCCC3)C2)ncnc2cnccc12 12625,C1(C(=O)NCCN(C)C(c2ccc3c(c2)OCC3)=O)C2C3CC4C1C1C2CC3C41 12626,N1(C(c2c(C)cnnc2)=O)CCC2(CC2)CC1C(=O)NCc1ncn(C2CC2)n1 12627,C1(C)(CNC(CC=C)=O)CN(C(c2coc(COC)n2)=O)CC1C 12628,N1(C(c2ccn(CC)c2C)=O)CC2(C1)CN(C(c1cc(C(F)F)[nH]n1)=O)C2 12629,C(=O)(C(F)(F)CCC)N1C(C(=O)NCCCCC#C)CSC1 12630,CC(CC(F)(F)F)C(=O)N1CC2(CC2)CC1CNC(=O)CC12CCCC1C2 12631,C1(C)(C(=O)NC(CCOC)C(=O)NCc2cc(C)nc(O)c2)CCCN(C)C1 12632,c1(C(=O)NC2CN(C(C(C(C)C)C(C)C)=O)CC2F)cccc2c1nc(O)n2C 12633,Cc1csc(CC2(C3CC3)CCCO2)n1.c1(C2(C)CNC(=O)N2)ccccc1 12634,c1(C(=O)OC(C)C(=O)N2CC(CC3CC3)C2)cc(Br)cs1 12635,N1(C(CCSC)=O)CCCC2(NC(c3ccc(CN(C)C)cc3)=O)CC12 12636,N1(C(C2(C3N(C(c4cc(C(C)C)[nH]n4)=O)CCC3)CC2)=O)CCC(C)(C#N)CC1 12637,C1(c2nc(CNC(c3ccn(C4CCC4)n3)=O)[nH]n2)CCCN(C(=O)C2=CCC2)C1 12638,c1(NC(C2(C)CCCN(C(C(C)OC)=O)C2)=O)cc2ccccc2cc1O 12639,C12(CNC(Cc3c(C)cccn3)=O)CCC(CC1)N2C(C1C2CC3C(C2=O)C13)=O 12640,C1(C(N(CC(C)NC(c2cc[nH]c2C2CCCC2)=O)C)=O)CC12CC(C)(C)C2 12641,Cc1ccn2ncc(C(N3CCN(C(=O)CN(C)C)CC(CO)C3)=O)c2n1 12642,N=c1[nH]c2c(s1)CCCC2C(=O)NCC1(O)CCCN(C(=O)C(O)C(F)(F)F)C1 12643,CC(C)(CCCO)NC(C1CSCCN1C(C1CC(=O)C1(C)C)=O)=O 12644,c1(C(=O)OC)cc2[nH]c(C(=O)NC(C)CC(C)NC(=O)CCP(C)(C)=O)cc2s1 12645,C1(C(=O)NC2(CC(=O)N(CC(C)N(C(C)=O)C)C)CC2)CCCC(F)C1 12646,c1(C(=O)NC2CC(N(C)C)C2)ccnc(CNC(C2(N3CCCC3)CCC2)=O)c1 12647,c1(NC(CC)=O)cncc(C(N2CC=CC2CNC(=O)C=C2CCC2)=O)c1 12648,CN1CC(CNC(=O)CC2CCCN(C(=O)CCc3ccnn3C)C2)CC1=O 12649,C12(NC(C3OCCN(C(C)C)C3)=O)CC(CNC(=O)C(C)C(F)F)(C1)OC2C 12650,N1(C(COCCCOC)=O)CC2C(NC(=O)CNS(=O)(=O)N(C)C)C2C1 12651,C1(C)(C(N(C)Cc2c(C)nsc2)=O)CCCN1C(=O)C(c1cncnc1)C 12652,C(=O)(CC1=CCOCC1)NC(COC)CC(=O)N1CC(OCC2CC2)C1 12653,C(C(=O)NCCC1(C)CCOC1)(C(C)(C)O)NC(C1CCC(CC)O1)=O 12654,c1(C(=O)NC(CN(C(=O)CCCc2ccc(C)s2)CC)C)cc(CC2CC2)on1 12655,CCCCCCCC1CN(C(=O)CCCn2cc(C(C)(C)CO)nn2)C1.C1C(=O)O1 12656,C1(NC(COC2(C)CCCC2)=O)CCN(C(C2CN(C3CCC3)C2)=O)C1C(=O)O 12657,N12CC(C(n3ccnn3)C1)C2=O.CC1C(NC(=O)CSc2cccnc2)C1(F)F 12658,C1(NC(c2n(C(C)C)ncn2)C)CCN(c2nc(-c3ccccc3)co2)CC1 12659,C(C(O)CC(=O)NCC(=O)NC1CC1)NC(c1c(COC)cc[nH]1)=O 12660,O=C1CCC(C(=O)NCCOC2CN(C(c3ccccc3C(F)F)=O)C2)CN1 12661,c1(C(=O)NC(CC)CN(C(=O)C(CSC)OC)C)cn(C)nc1-c1nccs1 12662,Cc1cc(F)sc1C(=O)NC(C1CCN(C(C2CC2(C)C)=O)C1)C 12663,N1(c2ccc(CC)nc2OC)CCN(C(C)=O)CC(C)(C)C1 12664,c1(C(N(C2CN(C(c3cnc(C(C)O)s3)=O)CC2O)C)=O)nccc2ccsc12 12665,Cc1cc(Cl)c(NC(c2cc(F)c(Cl)cc2O)=O)cc1O 12666,CC(C)(C#CC(=O)NCC(C)(O)C1CC1)CNC(=O)CN1CCOC1=O 12667,C1(C(=O)NCc2cn(CC(=O)NC3(C(=O)OCC)CC3)nn2)CCCCC1F 12668,CC1COc2ccc(C(N3CC4CN(C(=O)CC5=CCCC5)CC4(C)C3)=O)cc21 12669,N#Cc1cn[nH]c1C(=O)NCCC1CCN(C(C2C(Cl)(Cl)C23CC3)=O)C1 12670,C(=O)(CCCCCC(C)O)N(CCOCCCNC(C(C)OC(C)=O)=O)C 12671,Cc1cc(Cl)c(Cl)cc1C(=O)OCc1ncoc1C(C)C 12672,C(N=c1[nH]c(NC2CCCn3ncnc32)nc2ccccc12)c1cc(C)ncn1 12673,S(=O)(=O)(c1cnccc1COCC(C)C#N)N(CCOC)Cc1ccc(Cl)cc1 12674,c1(CNC(=O)C(c2sncc2Br)N2CCCC2C2CC2)ccccc1 12675,N1(C(CCCCCN(C)C(c2cncnc2)=O)=O)CC2CCC1C(CO)C2 12676,c1(C(=O)NC2(CC=C)CCN(C(=O)CC(C)OC)C2)cc(C)cc(Br)c1 12677,C1(C(N(C)CC2(O)CN(C(=O)C=Cc3cc[nH]n3)C2)=O)COCCN1C 12678,c1(C(N(CC(CC)NC(=O)CCC2CC=C(C)CC2)CC)=O)cccc(C)c1F 12679,N1(C(C(c2ccn(C)c2)C)=O)CC2CCCC(N(C(=O)CN(C)CCO)C)C2C1 12680,c1(NC(C)=O)c[nH]c(C)c1C(=O)NCC=C1CCN(C(=O)C=C2CC2)CC1 12681,CN1CCCC2CCN(C(=O)NCC3CCCC4(CCCC4)O3)CC12 12682,CCN=c1[nH]cc(C(=O)NCC(Cn2cc(CC3CCCC3)nn2)OC)s1 12683,N1(C(CCn2ccc(C)n2)=O)CCC(C)N(C(=O)CC2COCC2O)CC1 12684,N1(C(C(C)(C)SC)=O)CCN(C(c2n[nH]c3c2CCC3)=O)C(C2CCC2)C1 12685,c1(CNC(C(C)NC(=O)CCCc2cnn[nH]2)=O)c(O)cccc1F 12686,c1(C(=O)NC(C)CN(C)C(c2ccc(N)cc2)=O)cc2ccc(O)nc2s1 12687,N1(C(c2cccc(N)c2Br)=O)CCOCC(F)(CNC(c2cnc[nH]2)=O)C1 12688,CCC(CN=c1cc(NCCN2CCCCC2C)nc[nH]1)OC 12689,CC#CCCC(=O)NCC(C1CCOC1)NC(=O)Cc1cnn(C)c1C(F)F 12690,C1(C(=O)NC2COCCC2O)COC2(C1)CN(C(=O)CC1CC1C1CC1)C2 12691,c1(C(N2CC(OC)C(CNC(=O)C(C)CC3CCCC3)C2)=O)cc2n(n1)CCO2 12692,CC(C)CCC(C(=O)NCC(C)(O)CO)NC(c1cn(C)cn1)=O 12693,c1(NC(CC)=O)ccc(C)c(C(=O)NCc2ncc(Br)cc2N)c1 12694,C1(NC(=O)C=CC2CCOC2)CCCC12CCN(C(C13CC(C1)C3)=O)CC2 12695,c1(CCC(=O)NCC(C)(CO)NC(C2(OC(C)=O)CC2)=O)nnc(S)n1C 12696,N1(C(c2ccc(OC)c(O)c2)=O)CCC2(C1)CN(C(c1ncsc1C1CC1)=O)C2 12697,c1(C(N2CCN(C(C3CC(=C)C3)=O)C(C)C2)=O)cc2ccccc2nc1O 12698,c1(NC2CC(CNC(CCC(=O)N(CC)CC)=O)C2)ncn(C)c(=O)c1Br 12699,Cc1cnn2ccc(C(N3CCC(C(C)NC(=O)CP(C)(C)=O)C3)=O)nc12 12700,C1(CC)CN(C(c2cc(C)ccc2Cl)C(=O)NC(C)C)C2(CCC2)C1 12701,N1(C(C(CC)O)=O)CCC(C2(NC(=O)Cn3cccn3)CCC2)CC1 12702,C(=O)(C(O)P(C)(C)=O)NCC(CN(C)C(c1cncc(C(C)(C)C)c1)=O)(C)C 12703,N1(C(C2CCN(CC)C2)=O)CC(CO)C2(C1)CN(C(C1(C#N)CCSCC1)=O)C2 12704,C(=O)(C(CNC(=O)CC(F)(F)F)C(C)(C)C)NCCc1cn(CC)nn1 12705,CC(C)S(=O)(=O)c1ccccc1C(=O)NC1CCN(C(C2CC(F)C2)=O)C1 12706,c1(C(=O)NC23CC(CNC(CC4CCCN(C)C4)=O)(C2)C3)ccc(F)cc1Cl 12707,C(=O)(C(F)(CNC(C1CCC(C)O1)=O)C(C)C)NCc1onc(COC)n1 12708,Cn1cc(-c2n[nH]cc2C(=O)Nc2nc(C3CC3)cs2)cn1 12709,C(CCCCC(C(=O)NC(C)(C)C)N1CCn2nc(C)c(I)c2C1)OC 12710,O=S(=O)(c1ccccc1C(F)(F)F)N1C2CN(Cc3cncc(Br)c3)CC12 12711,C(=O)(CCCC(F)(F)F)NCCOCCN(C)C(c1nccnc1-n1ccnc1)=O 12712,C1(CC)CN(C(C2CC(C(C)(C)C)C2)=O)CCN1C(=O)Cn1nc(O)ccc1=O 12713,c1(C(N(CC(C)CNC(=O)C(O)C2CCC2)C)=O)cccc(S(=O)(=O)CF)c1 12714,C12(C(=O)NC3CCCCN(C(c4c(Cl)cc(C)s4)=O)C3)CC1Cc1c[nH]nc12 12715,C(N=c1[nH]c(=NC)[nH]c(=NCC2C=CCCC2)[nH]1)c1ccc(N(CC)CC)cc1 12716,c1(N(C)CCOC(F)F)nc(=NCc2cc(Br)ccc2C)[nH]c2c1CSC2 12717,Cn1cc(C=CC(=O)NCCC2(C(=O)NCC3CC3C3CC3)CCC2)nn1 12718,C1(C(C)NC(C(CC)NC(N)=O)=O)CCN(C(=O)CCCC2CC2)CC1 12719,C1(COC)(CNC(=O)CCC2CCOCC2)CCN(C(C2CC(=O)N(C)C2)=O)C1 12720,C#CCC(C)(C)C(=O)NC(CNC(=O)C(C)n1ccnc1)CCOC 12721,C1(NC(c2[nH]c(=N)sc2)=O)CN(C(=O)C(F)C2CCC2)CC12CCS(=O)(=O)CC2 12722,C=C(F)CN=C(NCc1cccc(CC)c1)NC1CC(=O)N(c2ccccc2)C1 12723,N1(C(C(C2(O)CN(C(C(C)OC(C)=O)=O)C2)F)=O)CCc2ncn(C)c2C1 12724,c1(C(=O)OCC)c(NC(=O)CCCc2ccsc2)sc2c1CCC(C)C2 12725,C(=O)(C(C(F)(F)F)C(F)(F)F)NCC(N1CC(C)(C)c2c1cccc2)=O 12726,C(=O)(C(C)(C)C(O)C(C)C)NCC1(F)CC(CNC(Cc2n[nH]c(=NC)s2)=O)C1 12727,S(=O)(=O)(c1ccncc1)NC(c1c(N(c2ccco2)C(C)=O)cccc1)=O 12728,C1(NC(c2cnoc2C2CC2)=O)COCCC1NC(C1CC1C(F)(F)F)=O 12729,CCC(C(=O)NC(CNC(c1cc(C2CC2)ns1)=O)Cc1ccccc1)NC(N)=O 12730,C1(C2CN(C(=O)C(Br)=C(C)C)C2)(NC(CC2ON=C(CC)C2)=O)CC1 12731,c1(C(N2C(C3CCN(C(c4cc(CC)ncc4)=O)C3)CCC2)=O)ncc(N)cc1C 12732,c1(C(N(C(c2ccccc2)CNC(=O)C(F)=C2CCC2)C)=O)cccnc1O 12733,c1(C(C(=O)NC(C)C(=O)OC)N(C)Cc2scc(CC)c2)nc(C2CC2)n(C)n1 12734,C1(OC)CCC12CC(C(=O)NCCC1(NC(c3coc(C#N)c3)=O)CCC1)C2 12735,C(CC(=O)N=c1cc[nH]c(C(=O)N(C)C)c1)C1N(c2cc(OC)ncn2)CCC1 12736,C1(CCNC(c2cnn(CCC)c2C)=O)CCN(C(=O)CN(C)CCO)C(C)C1 12737,C1(C(N2C(C)CC(NC(C3CC3C3CC3)=O)CC2)=O)CCCCC1N=[N+]=[N-] 12738,CCCC(C)(C)CC(=O)N1CC2CCC2(CC(=O)NCc2cc(C)ncn2)C1 12739,c1(C(=O)NC(CNC(C(F)=CC)=O)CC(F)(F)F)cc(=O)n2nccc2[nH]1 12740,CN=c1ncc(-c2nc(C(N3CC4CCC(C3)O4)=O)cs2)c[nH]1 12741,C1(NC(c2cnn(-c3nccs3)c2)=O)CN(C(c2ccsc2)=O)CCC1CO 12742,N1(C(Cc2scc(C)c2)=O)CCC(C)(NC(c2coc(C(F)(F)F)c2)=O)C1 12743,C1(NC(CCCN(C(C)C)C)=O)CCC(CNC(C2CC(CN(C)C)C2)=O)CC1 12744,N1(C(C2OCC(CN)C2)=O)CCc2cc(C(C)C)ccc2C1 12745,C(=O)(CC(O)CC(C)C)NCC(CCC)C(=O)NC1C=CC(C(=O)OC)C1 12746,C(=O)(C1c2c[nH]nc2CN1C(=O)CCCn1ccnc1)NCC(N1CCCC1)C 12747,c1(C(=O)NCCOCCC(=O)NCC=C)ccc(CC)o1 12748,c1(NC(C)=O)ccc(Cl)c(C(=O)NCC(C)NC(=O)C(c2ccccc2Cl)O)c1 12749,c1(C(=O)NC2CC(C)(NC(c3ccnc(C)n3)=O)C2)cc(N)c2ncccc2c1 12750,c1(C(N2CCCCC2C(=O)Nc2csc(Br)c2)=O)cc(F)cc(Br)c1Cl 12751,C(=O)(C1=CCC(NC(=O)CCC2(C#N)CCC2)C1)NCC(=O)NCCC 12752,C1(C(=O)NCCNCC2CCC(C(=O)OC)C2)CCCC(C)(C)CC1 12753,N1(C(C(CCC)O)=O)CCC(C(F)(F)F)CC1CNC(c1nn(C)cc1SC)=O 12754,Cn1ccn2ncc(C(N3CC4C(NC(=O)C=Cc5cc[nH]c5)C4C3)=O)c12 12755,C1(NC(C(CSC)O)=O)CC2CC1CC2C(=O)NC(CCO)C(C)(C)C 12756,C=CC(CC)CC(=O)Nc1c[nH]c(=N)c(C)c1.C12CN(CC1C=C)C2=O 12757,c1(C(N2C(C)CC(CNC(=O)C=Cc3cc[nH]c3)C2)=O)cnc2n1CCS2 12758,Cc1nn(C)c2ncc(C(=O)NCCCC(C)NC(c3nc(=O)n(C)[nH]3)=O)cc12 12759,C(=O)(C1Cc2ccc(Cl)cc21)NC(CCCC)CNC(c1cc(C2CC2)[nH]n1)=O 12760,C(=O)(C(C)(C)N(C)C)NCCC(C)N(C)C(c1ccc(Br)o1)=O 12761,c1(C(N2C(C)(CNC(c3ccsc3C(F)F)=O)CCC2)=O)ccc2nonc2c1 12762,c1(CCC(=O)NC(C)CNC(C2(CC3CCC3)CC2)=O)ccc(Br)s1 12763,C(=O)(C1=CCCC1P(C)(C)=O)N1CC(C)C(CNC(=O)C(C)(C)CN(C)C)C1 12764,c1(NC(=O)NCCN2CC(F)C(F)(c3ccccc3)C2)ccc([N+](=O)[O-])cc1O 12765,C(=O)(C(CNC(=O)CC1CCOC1)N(C)C)N1CC(OC)C1 12766,N1(C(C2(CC)COC2)=O)CCC2(CC1)CC2C(=O)NOCC(O)CO 12767,c1(C(=O)NCC2CCC(NC(c3c(CC)non3)=O)C2)nccc2c1NCCC2 12768,N1(C(c2cc(Br)cs2)=O)CCOC(CNS(=O)(=O)CCBr)C1 12769,C(=O)(C1=Cc2ccccc2C1O)N1CC(O)(CNC(c2cncc(CC)c2)=O)C1 12770,CC1(C(=O)NCCN(C(=O)CSC2CC2)Cc2ccccc2Cl)COCCO1 12771,C(=O)(C(C)C(F)(F)F)N(CC=CC(=O)N(C)Cc1c(CC)noc1)C 12772,CC1(C)NC(=O)N(CC(N2CCCC(O)(CNC(=O)C(=O)NC3CC3)C2)=O)C1=O 12773,CCC(CC)CC(=O)N1CC(CNc2nccc(-n3ccnc3)n2)C1 12774,C#Cc1ccc(C(=O)NC(CCN(C)C)C(=O)NCCc2nnc(C)n2C)cc1 12775,C=C(Br)CC(=O)NC(C(CO)N(C)C(=O)C1CC1)c1ccccc1 12776,c1(OC)cscc1C(=O)NC(CN(C)C)C(=O)NCc1cncnc1 12777,CCCC(CCCNC(C1CC1(F)F)=O)NC(=O)CCCCc1ccccc1 12778,c1(C(=O)NC2CCC(N(C(CCSCCCC)=O)C)C2)nccnc1CC 12779,C1(F)(C(=O)NCC2(F)CC(CNC(CC3(C)OCCO3)=O)C2)CCCCC1 12780,CCCC(CC)CCC(=O)N(C(C)C(=O)NC1CCCCC1OC)C1CC1 12781,CC1=CCC(C)(C(=O)NCC23CCC(C2)N(C(c2csc(C)c2N)=O)C3)CC1 12782,N1(C(CN(CCC)C)=O)CCC(CNC(=O)C(O)Cc2cnc[nH]2)(OC)C1 12783,C1(NC(c2nc(CC)oc2C)=O)COC2(CNC(=O)C(C(C)C)SC)CC1C2 12784,C1(CN(C(=O)C(O)Cn2cncn2)C)CCCCN1C(=O)CCC#N 12785,c1(C(=O)NCCN2CCCN(C(C3C(OC)C3)=O)CC2)cccc2c1ncn2C 12786,Cc1cccnc1CN1CCC1C(=O)NCc1ccc(C(F)(F)F)s1 12787,c1(OC)ccc(C(=O)NCc2cc(C(F)(F)F)nn2C)c2cccnc12 12788,C1(O)(CNC(c2cc(OCC)n[nH]2)=O)CCN(C(=O)CC2CCCC2O)C1 12789,C1(C(=O)NCc2ncc(C)nc2)CC12CCN(C(=O)CCc1cncn1C)CC2 12790,C1(NC(c2ccc(Cl)o2)=O)CN(C(=O)C(F)C2CCC2)CC1CO 12791,CCC(CC(=O)NC1CCN(C(C2CC23CCCCC3)=O)C1(C)C)CC(F)(F)F 12792,c1(C(=O)NC(C)C(C)NC(c2c(F)cncc2Cl)=O)cc(F)cc2cc[nH]c12 12793,C1(N(C(COCC(=C)C)=O)C)C2CN(C(C3(C(C)C)CNC(=O)C3)=O)CC12 12794,N1(CC)CCN(CC(=O)NCC(CO)NC(=O)Cc2ccco2)CC1 12795,N1(C(CCN(C(CCOCCC)=O)C)=O)CCC2CC2C1 12796,c1(C(N(CC(CC)NC(=O)C(C)Cn2cccn2)C)=O)cnc(C)cc1C 12797,C(=O)(C(C)CCC(C)(C)C)N1CCC(NC(c2ccc(C)cc2)=O)(CF)C1 12798,c1(N(C)Cc2c(C)ccnc2)nc(N(C)CC2CC(F)C2)nc2ncn(C)c12 12799,c1(C(=O)NC2(C)CC2)cn2c(n1)CCN(C(=O)Cn1cc(S(C)(=O)=O)cn1)CC2 12800,C(=O)(C1=CS(=O)(=O)CCC1)NCC(C)(O)CNC(c1ccncc1C(F)(F)F)=O 12801,C1(C(C)(C)CNC(=O)CNC(N)=O)CCCCN1C(=O)C=Cc1ccco1 12802,C(=O)(CCC(=O)NC1CCCC1CNC(=O)C=CS(C)=O)NC(C)=O 12803,Cc1cnc(C)c(C(=O)NCC(C)CN(C)C(c2sc(F)cc2Cl)=O)c1 12804,C(=O)(C1=CC2CCC1C2)N1CCCC(N(C)C(c2cccc(Cl)c2)=O)C1 12805,c1(NC(C2N(C(c3nc(CC)oc3)=O)CCC2)=O)c(C)ccc(I)c1C 12806,c1(N2CCC(C(C)(C)NC(C3CCCC(CF)C3)=O)CC2)nccnc1C#N 12807,C1(NC(=O)CN2CCSCC2)CCCC(NC(c2cccc(C(F)F)c2)=O)CC1 12808,C1(NC(CCn2c(C)ccc2C)=O)CCN(C(c2ccncc2N)=O)C12CCC2 12809,c1(N(C)Cc2nccs2)nc2cc[nH]c2c(=NCC2CCc3cccnc32)[nH]1 12810,O=C(C1=C(Cl)CCCC1)N(CC(=O)NCC12CCCCC1C2)C1CC1 12811,C(C)(CCCCNC(=O)CCC1CCC1)NC(CSCCC)=O 12812,C1(NC(Cc2c(C)noc2Cl)=O)CC1C1CCN(C(c2cncc(O)c2)=O)CC1 12813,C1(O)(CNC(C2(N(C)C)CC2)=O)CCN(C(c2cc(Cl)ccc2F)=O)CC1 12814,c1(C(=O)NC2(CNC(C=C(CC)C)=O)CCOCC2)cccc2oc(C)cc12 12815,CCC(C)(CNC(c1cccn1C(C)C)=O)C(=O)NCC1OCCCC1(C)C 12816,CC(CNC(=O)CC=CCNC(=O)CCn1ccnc1)CN1CCCC1 12817,C(=O)(C(C)(C)C(F)(F)F)NC1CC(NC(c2cccc(SCCCC)c2)=O)C1 12818,CCS(=O)(=O)CCNC(C1(CNC(C2CC2(F)Cl)=O)CC(=C)C1)=O 12819,c1(C(N2CC(CCNC(CS(=O)(=O)NC)=O)OCC2)=O)nn(C)c(Cl)c1Cl 12820,c1(CNC(C(CCOC)NC(=O)CSC(F)F)=O)cccc(F)c1F 12821,C1(NC(CC2(NC(C)=O)CCCCC2)=O)CC(F)CN(C(=O)CCS(C)(=O)=O)C1 12822,c1(CNC(=O)Cc2ccc(CC3(F)CCNCC3)cc2)ncnc2ccccc12 12823,N1(C(C(N2CCOCC2)C)=O)CC2CC(NC(=O)C=Cc3cccnc3)CC1C2 12824,c1(C(=O)NCCCN(C(=O)Cn2nnc(=O)[nH]2)C)ccc(CNC(=O)NC)o1 12825,C1(C(N(C)Cc2snc(C)n2)=O)CN(C)CCN1C(c1cccc(O)c1)=O 12826,C1(O)(COC(c2nc(C)n(-c3ncccn3)n2)=O)CCCC(C)(C)CC1 12827,c1(C(=O)NCCN(CCOC)C(C2CCC(C)S2)=O)cc(Cl)cc2c1OCC2 12828,O=C(C(F)CC1CCCC1)NC1(NC(=O)CC2CS(=O)(=O)C2)CC1 12829,N1(C(CN(CCOC)C)=O)CC2CN(C(c3[nH]c(C)cc3C)=O)CCC2(CO)C1 12830,N1(C(C(C)(C)C#N)=O)CCC2CCCN(C(c3ccc(C(F)F)cc3)=O)C2C1 12831,C1(C)(C(N(CCS(C)(=O)=O)C)=O)CCN(C(c2ccc(C(=O)O)o2)=O)CC1 12832,C(C(C)N=c1nc(NCc2cc(F)ccc2F)c2sccc2[nH]1)c1ccc(C)s1 12833,N1(C(CCCC(C)NC(CCOC)=O)=O)CCCC12CCOC2=O 12834,N1(C(CSCC)=O)CC(NC(=O)COCc2nnc(C)s2)CC(F)C1 12835,CC1CCCCC1(CNC(c1ccc(=O)n(C)n1)=O)NC(=O)CCNC(=O)CO 12836,C(CN=C(NC1CCS(=O)(=O)C1)N1CCCC(C(=O)N(C)C)C1)OC(CC)(C)C 12837,N1(C(CS(CC)=O)=O)CC2CCC1(CNC(=O)C#CC(C)(C)C)CC2 12838,N1(C(c2cc(CCOC)on2)=O)CC(C)CN(C(=O)CC2CCSC2)CC1C 12839,C1(C(=O)OC)(OC)CCN(C(=O)C(CN)Oc2ccccc2)C1 12840,C(=O)(C#CC1(C)CCCO1)N(CCCCN(C)C(C1(C)CC1Br)=O)C 12841,c1(C(N(C)CC2CCN(C(Cc3c(C)ccs3)=O)CC2)=O)csc2ccncc12 12842,N1(C(c2cc(CC)oc2C)=O)CC2CCC1CN2C(=O)CCC1CCN(C)C1 12843,Cc1nnc2n1C(C(=O)NCCCC(C)NC(c1sccc1Cl)=O)CC2 12844,Cn1cc(Cl)c(C(=O)NCC(C)(O)CNC(c2ccc(OCC(F)F)cn2)=O)n1 12845,CC1(C)CC(C(=O)NC2CC3CCCC3C2)CN(C(=O)CN2CCSCC2)C1 12846,C1(NC(=O)CCCn2cccn2)CS(=O)(=O)CC1NC(C12CCCN1CCC2)=O 12847,N1(C(C(CCSC)NC(C2CN(C)CC(C)O2)=O)=O)CCn2nccc2C1 12848,C(=O)(C(F)CCC(C)(C)C)NCc1c(C(=O)Nc2c(C)csc2)nco1 12849,CC1ON=C(C(=O)NC(C2CCCN2C(c2csnn2)=O)(C)C)C1C 12850,CCCCCC(O)CC(=O)NC1CCCC1NC(C1(C(N)=O)CC1)=O 12851,C1(C)(CNC(C(CC)Sc2nc(=N)[nH][nH]2)=O)CCN(C(=O)OC(C)(C)C)CC1 12852,CCC(CC)CCCC(=O)N1CC(C)CCC1CNC(=O)CCSCC(N)=O 12853,c1(C(=O)NCC2C(Nc3nccc(C)n3)CCCC2)ccc(C)c2c1CCC2 12854,N1(C(c2c(OCC)scc2)=O)CCN(C(C2CCC(CN(C)C)C2)=O)C(CC)C1 12855,c1(OC)ccc(CCC(=O)NCC(C)NC(=O)C(O)Cc2nnc(C)n2C)cc1 12856,C1(O)(COC)CN(C(C2CCC2CNC(=O)C(C)c2ccco2)=O)C1 12857,CCC(C(=O)NC(c1ccc(-c2cc(NC)sc2)s1)=O)c1ccccc1 12858,Cn1nc(CC(=O)Nc2cc(-c3ccccc3Br)on2)c2ccccc2c1=O 12859,C1(CN(C(CCOC)=O)C)CCCCN1C(c1sccc1OC)=O 12860,C(C1CCCCCC1)=CC(=O)NCC1(F)CN(C(CCC(=C)Cl)=O)C1 12861,C=CC1CN(C(c2cnc(C)c(CC(C)C)c2)=O)CC1NC(=O)C#CC1CC1 12862,CC(C)CC(CNC(C1CC(C)(C)CN1C)=O)C(=O)Nc1ccc(F)cc1CO 12863,CC1CCCCN1CC(=O)NC1C2CCN(C(c3ccc(SC4CC4)cc3)=O)C12 12864,c1(C(=O)NCC2N(C(CC(c3scc(C)c3)O)=O)CCC2)c(C)coc1C 12865,C(=O)(C1=NOC(CNC(=O)CCOCC)C1)NCC(=C)F 12866,N1(C(C)C(=O)NCCC2CC(NC(C3(C4CC4)CC3)=O)C2)CCCCC1=O 12867,c1(C(C)C)ccoc1C(=O)NC12CC(NC(=O)C(F)C3CCCC3)(C1)C2 12868,c1(C(C)C)ccc(CNC(=O)N(C)CC2CCCN2Cc2cccnc2)cc1 12869,c1(CC)nc(Cl)c(F)c(=NCCCCNC(=O)C(Cc2ccccc2C)CC)[nH]1 12870,c1(C(N(CCCCNC(=O)CC2CC(C)(C)CO2)C)=O)ccc2oc(=N)[nH]c2c1 12871,N1(C(C(C2CC(C)(C)C2)OC)=O)CCC2(CCC(NC(=O)CC(F)(F)F)C2)C1 12872,C=CCCC(CC(C)C)C(=O)N(CC(C)NC(C1CCOC(C)C1)=O)C 12873,c1(C(=O)NC(CCCC=C)c2ccccc2)[nH]cc2c1CCCC2 12874,N1(C(COC2CC(NC(c3c(OC)nccc3)=O)C2)=O)Cc2ccc(O)cc2C1 12875,c1(C(N2C(CN(C(CN(C)CCO)=O)C)COCC2)=O)cc(O)c2ccoc2c1 12876,C(=O)(C#CC1(C)CC1)NC(CCOC)CNC(=O)C(C(C)O)NC(C)=O 12877,c1(C(=O)NC2CC3CCC2(NC(c2ccon2)=O)C3)cc2ccccn2c1 12878,c1(C(=O)NCCCNC(CSCC(=O)OC)=O)ccc2c[nH]nc2n1 12879,C1(S(C)(=O)=O)(N(C)Cc2conc2C(F)(F)F)CC1C(F)(F)F 12880,CC(C)(C)CCCC(=O)NCC1CCN(C(=O)CC2CCOC(C(C)(C)C)C2)C1 12881,C1(C(N(CC)CC)=O)CC2CC2N1C(=O)CCOC1CC1 12882,N1(CCOC)CCC(N=c2[nH]c(N3CCSC(C(F)(F)F)C3)nc3c2COC3)C1 12883,c1(COC)nn[nH]c1C(=O)NC(C)C(C)NC(=O)CN(C)CCO 12884,c1(SC)cccnc1C(=O)NCC1CC2CC2N1C(=O)CCc1cscn1 12885,C1(NC(C#CC(C)(C)C)=O)CC(N=c2ccnc(Cl)[nH]2)C1(C)C 12886,c1(CNC(C2N(CC)CC2)=O)nnc2n1CCN(C(C1Cc3nccn3C1)=O)C2 12887,N1(C(CCCN(C(C)C)C)=O)CCN(C(C2COC(=O)N2C)=O)C(C)C1 12888,N1(C(C(C)OCC(C)C)=O)CCC(C2CCN(C(C3CCCCN3C)=O)CC2)C1 12889,C1(c2cn(CCCC(=O)OC)nn2)CCCN(C(=O)CCC(C)SC)C1 12890,N1(C(c2n(CC)nnc2)=O)C2CCC1CC(N(C(=O)CN(C1CCSC1)C)C)C2 12891,c1(C(CNC(C2CCCO2)=O)NC(c2cc(C(F)F)[nH]n2)=O)ccc(F)cc1 12892,c1(C(N2CC(C)C(CNC(=O)C(c3ccnn3C)O)C2)=O)cncc2nc[nH]c12 12893,c1(OCC(=O)NCC(CC)NC(=O)C(F)C2CCC2)ccc(Cl)cc1C 12894,N1(C(C(C)OCCCC)=O)CCCC2(CCCCC2NC(=O)C=C(C)CCC)C1 12895,C1(C(=O)NCC2(CNC(c3ncsc3C(F)(F)F)=O)CC2)CCCC2(CCC2)C1 12896,C1(NC(c2cc(OC)n(C)n2)=O)CCCN(C(C2CN(S(C)(=O)=O)C2)=O)CC1F 12897,CC1C(=O)CC1C(=O)NC(C)(CNC(=O)CCC1(C)CC1(F)F)CO 12898,C(C(C(C)(C)C)NC(=O)CCCN1CCCC1)NC(C1CC(OC)C1)=O 12899,N1(C(C2(C)COCCO2)=O)C2CCC1CN(C(c1ccc(C(F)F)nc1)=O)C2 12900,Cc1cc2[nH]c(C(=O)NCC3(O)CN(C(C4CC5CCC4O5)=O)C3)cc2o1 12901,C1(C(=O)NCC2C3CN(C(COCCCC#C)=O)CC32)CCC(S(N)(=O)=O)CC1 12902,C1(NC(C(C)(CO)NC(C(OCC)OCC)=O)=O)CCOC12CCCC2 12903,N1(C(C(CCCC)NC(=O)CCN(C)C)=O)CCC12CCCCC2 12904,C(=O)(C(CC)CC=C)NC(CCCCNC(c1cc(CCCCC)[nH]n1)=O)C 12905,N1(C(C2C(NC(Cc3cc(C)[nH]n3)=O)CCC2)=O)CCOC(CO)C1 12906,Cc1cc(C(N2CC(NC(=O)CC(C)CF)C2)=O)cc(N)c1 12907,Cc1cc2ccccc2nc1C(=O)NC1CC(C)(NC(=O)C2=CCS(=O)(=O)C2)C1 12908,c1(CN2C(C)CCC(C(=O)OC)C2)cccc(C#N)c1OC 12909,C1(C(N2CCCC(C(=O)Nc3cnn(C(F)F)c3)C2)=O)CCCC2(CC2)C1 12910,N1(C(Cc2c(C)nsc2)=O)CCC(F)C(NC(c2ccnc(C(F)(F)F)n2)=O)C1 12911,C#CC1CN(C(=O)C(=Cc2cnc[nH]2)C)CCN1C(C1Cc2nc(C)cn2C1)=O 12912,N1(C(C(Br)=C(C)C)=O)CC2CN(C(c3cccc4cncn34)=O)CC2C1 12913,C1(NC(CCC(=O)OC)=O)CC(O)CN(C(c2cc(Br)c(C)o2)=O)C1 12914,N1(C(c2ccn(CC(F)(F)F)n2)C(=O)NCCSC)CC(CO)C(CO)C1 12915,c1(C(=O)NCC(C2CCCN(C(c3ccc(Cl)cn3)=O)C2)(C)O)cccc(Cl)c1 12916,C1(C(C(=O)OCCCCCC)CC)CCN(c2ccccc2)CC1 12917,Cn1nc(C(N2CC3CC2C3C(N2CCC(C)(CO)C2)=O)=O)cc1O 12918,N1(C(c2cncc(C#C)c2)=O)CCC2CCCC12CNC(=O)C(C)(C(C)C)OC 12919,CCCC(C)(CC)C(=O)NCC1CC(C(=O)Nc2cnn(C(F)F)c2)=NO1 12920,C1(CC)CN(C(c2ccncc2OC)=O)CC1NC(=O)C1=CCCS1 12921,CCC(CC(=O)NCC(C)CC(=O)N1CC(C(C)(C)C)C1)C1CC1 12922,c1(C(=O)NC2CN(C(C(C(C)C)NC=O)=O)C2)cc2c([nH]1)CCC2 12923,C1(CCCCCC)CCCC1(c1nnnn1CC)NCC(c1ccccc1)(C)C 12924,CC12CN(C(=O)C(=O)NCCCC(F)F)CC1(CO)C2 12925,c1(OCC)ccc(CNC(=O)NC2CCN(C(=O)C(F)n3cccn3)CC2)cc1 12926,CC(CCCCNC(c1cc(Cl)cnn1)=O)NC(=O)C(C1CCCCCC1)O 12927,c1(NC(CCC)CC(F)F)ncccc1S(=O)(=O)NC(CC1CC1)CC 12928,C(CC(C(C)(C)C)NC(c1ccc(F)c(F)c1)=O)N(C(C1(C)CC(C)C1)=O)C 12929,O=C(C1=CCCN(CCn2ccc3ccccc23)C1)NCCCc1ccncc1 12930,C1(NC(C2CCN(CC)C2)=O)CCC2(CC1)CCN(C(=O)C1=NOCC1)C2 12931,C(=O)(C(O)CC(N)=O)N(C)CC1(O)CN(C(C2(OC)CCC(C)C2)=O)C1 12932,C#Cc1ccc(CCC(N2CC3(NC(=O)COCC=C)CCC2C3)=O)cc1 12933,CC(C)CC(O)C(=O)N1CC(O)CC1CNC(C1C2(CC2)C12CC2)=O 12934,C(=O)(C(CO)C(C)(C)C)N1CC(C(=O)NCCOC2CCC2)(CC)C1 12935,CC(C)CC(CNC(c1cccc(=O)o1)=O)C(=O)N(C)CC1CC1 12936,C1(CNC(CCc2c(OC)cccc2)=O)CCC(C)N(C(c2cc(C)co2)=O)C1 12937,C(C(=O)NCCc1scnc1C)(C(C)(C)C)NC(c1c(CC)ocn1)=O 12938,CC1=C(C(=O)NC2CN(C(c3nn(C)c(Cl)c3Cl)=O)CC2F)SCCO1 12939,C1(CC(N2CCC(CN(C)C(c3ncn(C)n3)=O)C2)=O)CCC(=O)C1C 12940,N1(C(c2ccc(C)c(F)c2)=O)CCN(C(=O)C(C)S(C)(=O)=O)CC(CO)C1 12941,CCC(O)C(F)(F)C(=O)N1CCOCC(CNC(=O)C(C)(C)O)C1 12942,N1(C(C=C(C)c2cccs2)=O)CCC2CCC12CNC(c1ccc(O)c(F)c1)=O 12943,c1(C(=O)NC2CCCN(C(c3cc(CC)ncn3)=O)C2C)cc2c(s1)CCSC2 12944,C1(NC(CC2N(C(C=C(C)C3CC3)=O)C3C2CCC3)=O)CCc2n[nH]cc2C1 12945,c1(NC(C2CCCN2S(=O)(=O)c2ccccc2)=O)cc(Cl)cc2nc(O)oc12 12946,C1(Br)(C(=O)NCC(CN(C(=O)C2=CC(C)(C)C2)CC)(C)C)C(C)(C)C1(C)C 12947,C(CN=[N+]=[N-])(C(=O)N1CC(OC)C1)NC(C1CCN(CC)C1)=O 12948,C1(C(=O)NCC(O)CC2CCCC2)CC2CC2N1C(C1CCCCO1)=O 12949,Cn1nc2c(c1C(N1CC(NC(=O)CSC(C)(C)C)C3(CC3)C1)=O)COCC2 12950,C(=O)(CC(C)(C)C(F)F)N1CCC(C(C)C(N2CC(CO)C(O)C2)=O)C1 12951,c1(C(N(CCCNC(C2CC2Cl)=O)CC)=O)cc2cc(C)ccc2o1 12952,C1(CNC(C(=Cc2cccs2)C)=O)C2CCC(C2)N1C(=O)CNS(N)(=O)=O 12953,C12(NC(C(CC)C)=O)CCC(n3cc(C=CC(C)C)nn3)(CC1)C2 12954,N1(C(C(C)NC(COC)=O)=O)CCC(CO)(NC(=O)CN2CC=CC2)CC1 12955,n1(CCC(=O)NCCN(CCOC)C(c2cc(C(N)=O)no2)=O)cc(Cl)cn1 12956,Cc1[nH]nc(C(N2CCC(n3cc(-c4ccc(CCO)cc4)nn3)CC2)=O)c1O 12957,C#CCC(C(=O)NCC(O)CN(C)C)NC(=O)COC(CC)CC 12958,c1(C(=O)NCC(C)(CO)NC(=O)CSC2CC2)cccc(OC(F)F)c1 12959,N1(C(C2(NC(c3ccc(C)n3C)=O)CCCC2)=O)CCOC(C)(C)CC1 12960,Cc1cc(=NCc2cnoc2)[nH]cc1S(=O)(=O)NCC1CC(n2ccnc2)C1 12961,c1(C(N2CCN(C(c3ccccc3)=O)C(CC3CC3)C2)=O)cc([N+](=O)[O-])n[nH]1 12962,c1(NC(=O)NC2C(C)(C)C2)cccc(CN2CCOCC2)c1 12963,C(C)(CCC(=O)NCC1(CCNC(=O)Cc2cc[nH]n2)CC1)OC 12964,c1(C(N2CCN(C(c3c(CC)onc3)=O)C(CCO)C2)=O)ccc2ccoc2c1 12965,C1(NC(C(=O)OC)c2csnn2)CCCC1(C)C 12966,C1(NC(=O)NCC(C2CCOCC2)(C)C)CC2(C1)CC(F)(F)C2 12967,c1(C(=O)NC(C=CC(=O)NC2(C)CC(=C)C2)C)cc(C)ccc1O 12968,C1(C(=O)NC2(c3onc(C)n3)CC2)CNC(=O)CN1C(C1CC(C)(C)CN1C)=O 12969,Cc1cc(NCCC(C)NC(C2(O)CCCC(C)(C)C2)=O)n2ncc(C)c2n1 12970,C#Cc1c[nH]nc1C(=O)NCCN(C)C(C1CCC(NC(C)=O)CC1)=O 12971,C(CCC#N)(C(N)=O)NC(=O)NC1CC(CC)OCC1 12972,C1(C(N(C)CC2CCCN(C(c3cc(CO)on3)=O)C2)=O)CC2(CCCC2)CO1 12973,C1(CC)CC(CC(=O)NC2(C)CN(C(c3ccncc3C(F)(F)F)=O)C2)CCO1 12974,c1(C(N2CCC2)C)cn(CC2CCCN2C(c2cc(-c3ccns3)on2)=O)nn1 12975,N1(C(C(CCCC)C)=O)CCCC2CN(C(=O)COC)CC12 12976,c1(NC2C(CC)CN(C(=O)CCC(=O)N(C)C)CC2)ncnc2sc(C)nc12 12977,C=CC1(C(=O)NCC2CC2CNC(c2coc(C(F)F)n2)=O)CCOCC1 12978,c1(C(N(C(C(=O)NCCn2ncc(C)c2)C2CC2)C)=O)cn(C)nc1C 12979,CCCCC(F)(F)C(=O)NC(CN(C(=O)C1=NOC(C)C1C)C)CC 12980,c1(C(=O)NC2CC(C)(C)N(C(C3COC(=O)O3)=O)C2)cccc([N+](=O)[O-])c1 12981,c1(NC(C(C2CCN(C(c3sccc3Cl)=O)C2)C)=O)ccc2c(c1)OCC2 12982,N1(C(C(CCCNC(C2CCC3CC2CO3)=O)O)=O)CC=CC12CCCCC2 12983,N1(C(C2CC3(C2)C(=O)N3)=O)CCN(C(CC=C)=O)CC(C)(F)C1.C(C)(C)(C)SC 12984,N1(C(C(C)=C2CC2)=O)CC2CCCC2(NC(=O)C(C)NS(=O)(=O)c2cccs2)C1 12985,C(C(CC(C)C)NC(=O)C(C)O)NC(CCCN(CCC)CCC)=O 12986,N1(C(C2C(C)(C(C)C)C2)=O)CC(C)CN(C(C2CCSC(C)C2)=O)CC1C 12987,C(=O)(C1CC(NC(N2CCOCC3(CC3)C2)=O)c2ccccc21)OC 12988,c1(C(=O)NC2CCCN(C(C(C)OCC(C)C)=O)C2)cccc2c1NCC(C)C2 12989,c1(C(=O)NC2C3CN(C(C(C)n4cccc4)=O)C(C3)C2)nccc2occc12 12990,c1(C(N(CCCNC(C2CCC(C(F)(F)F)CC2)=O)C)=O)ncn2c1COCC2 12991,C12(C(=O)NCc3c(Cn4cc(CNC=O)nn4)nco3)CCN(CC1)C2 12992,c1(NC(=O)NC2CCCN(C(C)(C)C)C2=O)cc(O)nc(Cl)c1C#N 12993,c1(C(N2CCC(Nc3ccc(C)cc3)C2)=O)ccc(C)c2cccnc12 12994,N1(C(C2C(C)(C)C2)=O)CCC(COC2CCN(C(=O)CN3CC4CC4C3)C2)CC1 12995,Cc1cnc(NC(C)CC(C)C)c(S(=O)(=O)N2CC(N(C)C)C3(CC3)C2)c1 12996,c1(SC)cc(N2CC(CN(C(=O)CC3SC(=N)NC3=O)C)C2)nc(SC)n1 12997,N(C)(C1CCCc2ccccc21)Cc1c(OC)cccc1Br 12998,C1(NC(c2cnc(CC)[nH]2)=O)(CNC(c2nc(C)oc2C)=O)CC2CCC1C2 12999,C1(CNC(c2nc(OCC)sn2)=O)CCCCC1N(C(=O)C=Cc1ccco1)C1CC1 13000,c1(C(=O)NC(CNC(COCCCCC)=O)(C)C)cc(N)c(C)cc1Cl 13001,N1(C(CC2(CC(=O)OC)CC2)=O)CC(NC(c2ccc(SC)s2)=O)CC(C)C1 13002,N1(C(c2cc(CCCC)c(Cl)cc2)=O)CCCN(C(=O)NC2CCCC2)CC1C 13003,c12cc(Cl)ccc1NC(C)C(=O)N1CCC(C1)N(C)C(=O)C21CC1.CCOC 13004,c1(C(C)(C)C)nnc2n1CC(NC(=O)C(=O)N(c1ccc(O)cc1)CCO)CC2 13005,Cc1cc(C)c(C(=O)NC2CC3(C2)CN(C(=O)CC2CCCC2C)C3)c(S)n1 13006,C#Cc1ccc(NC(C2(F)CCCN(C(C3CCCN3C3CC3)=O)C2)=O)cc1 13007,c1(CS(C)(=O)=O)nc(Cl)cc(=NCCNC(C2CCCC3C2C3(F)F)=O)[nH]1 13008,N1(C(C2(OC)CCCCC2)=O)CCC(C)C(NC(c2cc(F)ccc2Cl)=O)C1 13009,C1(C(=O)NCCCSCC)C(NC(c2cc(C(F)F)[nH]n2)=O)C1(C)C 13010,N=c1[nH]c2ccc(C(N3CC(NC(c4cc(CO)on4)=O)CC(F)C3)=O)cc2o1 13011,N1(C(CCc2cnc(C)s2)=O)CC2CCC(CNC(c3ccc(=O)oc3)=O)(C2)C1 13012,C(=O)(C(F)C(=O)NC1(C)CC(NC(=O)CC2CC2(C)C)C1)OCC 13013,c1(N(C(=O)CSCOC(C)C(F)(F)F)CCOC)sc2ccccc2c1Cl 13014,CC1CCCCC1(C)C(N1CCC(c2cn(Cc3cnn(C)c3)nn2)C1)=O 13015,N1(C(c2cc(CO)on2)=O)CCC2CCN(C(C3CC4(C3)CC4(F)F)=O)CC2C1 13016,N#Cc1cn[nH]c1C(N1CCC(N(C)C(C2CCCCO2)=O)CC1)=O 13017,C1(NC(Cc2cccc(C)n2)=O)CN(Cc2cnc3ncccn23)CC(F)(F)C1 13018,c1(C(=O)NCC2(CNC(c3ccc(Cl)nc3)=O)CC2)cnc(O)c2ncccc12 13019,Cc1ccc2nc(N3CCCC(C(C)NC(c4cn(CCO)nn4)=O)C3)sc2n1 13020,c1(C(N2CCC(NC(c3cc(C)c(F)cc3)=O)CC2C)=O)cc(C)c(=O)n(C)c1 13021,N1(C(c2c(OCC)scc2)=O)CC2(C)CN(C(=O)C(CC)NC(C)=O)CC2(C)C1 13022,Cc1csc(=O)n1CC(N1CCN(CC(C)(C)F)CC1)=O 13023,C1(CC(=O)NC2CN(C(=O)C=Cc3ccccn3)CC2C)(COC)CCOCC1 13024,C1(SCC)COC2(CCN(C(c3cnn4ccccc34)=O)C2)C1.C12(CC1)C(=O)N2 13025,c1(COCC(=O)NCC(C2CC2)NC(C2(CC3CC3)CC=CC2)=O)ccccc1 13026,Cc1ncc(C=CC(=O)NCCCCCNC(c2ccc(C(N)=O)o2)=O)c(O)n1 13027,C(c1cccnc1)=CC(=O)NCc1ccc(C(=O)NC2CC(O)C2)nc1 13028,c1(CN2CC(C)(CC(=O)NCc3cccnc3)C2)cc(C(=O)O)ccc1F 13029,CCC(O)C(F)(F)C(=O)N1CCCC(CCC(=O)NC2C(O)CC2O)C1 13030,CCCCC(O)C(C)C(=O)N(CC(N1CCOC(C)CC1)=O)C1CCC1 13031,C1(CNC(C2(CC#C)CCOC2)=O)CN(C(c2cnc(=N)[nH]c2)=O)CCC1(F)F 13032,c1(OC)cc(CC(N2CC(CNC(c3cnc(C#N)s3)=O)CC2C)=O)ccn1 13033,c1(C(N2CCCC(CS(N)(=O)=O)C2)C(=O)NC2CCOC2)cc(Cl)ccc1Cl 13034,c1(OC)ccc(Br)c(CN=C(NCC2(CC(N)=O)CC2)NC(C)C)c1 13035,Cc1nc(-c2ccccc2)ncc1C(=O)NC1CN(C(C2CCCC(O)C2)=O)C1 13036,c1(C(=O)NCCCN(C(=O)CC2CC2(C)C)Cc2ccccc2)snc(O)c1Cl 13037,C(C(=O)N1CC2C(C(=O)NC(C)(CO)C3CCC3)C2C1)(C(C)(C)C)OC 13038,Cc1cnc(C(C)NC(=O)C=CC(C)(C)NC(=O)CCCNC(=O)OC)s1 13039,c1(CC)n[nH]c(=NC2CC3CN(C(=O)Cc4cc(C(F)(F)F)co4)CC23)o1 13040,N(C1CCOc2ccc(F)cc21)C(=O)NCc1ccc(N)c([N+](=O)[O-])c1 13041,C(=O)(CC(C)CC(C)C)N1CCC(C(N(CCN(CC)CC)C)=O)(CO)C1 13042,C1(NC(c2c(Cl)cn(CCC)n2)=O)CCC12CN(C(=O)C(C1CCCCC1)O)C2 13043,C(C(O)CCNC(=O)C(CO)NC(c1ncsc1NC)=O)OC 13044,N1(C(C2CC(=C)C2)=O)CCN(C(C)CNCCCC(=O)Nc2nccs2)CC1 13045,N1(C(CSCC(C)C)=O)CCC2(C1)CN(C(=O)C(N1CCC(C)C1)=O)CCO2 13046,N1(C(c2cc(CCOC)on2)=O)CCC2(CCCN2C(=O)CP(C)(C)=O)C1 13047,N(C1CCc2cccnc21)C(N(C)Cc1ncc(Br)cc1Cl)=O 13048,c1(C(=O)NC(CCNC(CCn2ccc(C)n2)=O)C)cnn2cc(C#N)cnc12 13049,C1(CNC(c2ccc(C3CC3)s2)=O)CCC(NC(C2(CO)CCC2)=O)CC1 13050,C12(CNC(C(C)NC(COC)=O)=O)CC1CN(C(C1(F)CCCCC1)=O)C2 13051,N1(C(c2cc(C(CC)C)no2)=O)CC(F)(F)CC1CCNC(=O)CCSC 13052,c1(COC)ccccc1NC(C1(COC)CCN(C(=O)C(C)n2cnnn2)C1)=O 13053,N1(C(C2CCCN(C)C2)=O)CCC(CNC(C2CC(=O)N(C)C2)=O)C12CC2 13054,C1(CN(C(CN(C)CC)=O)C)COCCN1C(=O)CCCc1csc(C)n1 13055,c1(NCC(CCCCC)O)ncccc1S(=O)(=O)N(C(C)CCSC)C 13056,C1(NC(c2cnc(C)[nH]2)=O)COCCN(C(c2cn(CC3CC3)nn2)=O)C1 13057,N1(C(C=CC(C)NC(C2CCCS2)=O)=O)CC2(CCNC(=O)O2)C1 13058,c1(OCC)ncc(NC(C2CCCC(NC(=O)CCc3nc(=N)[nH][nH]3)C2)=O)cn1 13059,C(CNC(=O)CCOC1CCC1)(C(=O)NCCCn1cccn1)OC 13060,C#Cc1ccc(C(N2CC3CC(CO)C(C3)C2)=O)c(C)c1.C12CC(C1)C(=O)N2 13061,c1(NC(C=CCNC(c2c(CC)nn(C)c2)=O)=O)ccc2occc2c1 13062,c1(C(CNC(C2CNC(=O)C2)=O)NC(C2CC(=C)C2)=O)ccccc1OC 13063,C(=O)(C(C)(C)CC(F)F)N1CC2C(NC(Cc3c(C)n[nH]c3)=O)(CC2)C1 13064,C(=O)(C1COc2ccc(F)cc21)N1C(CCNC(C(F)OC)=O)CCC1 13065,CCCCC(CC)C(=O)NCC1CCC(N(C(=O)C(C)=CC2CC2)C)CC1 13066,c1(C(=O)NC2CCC(NC(C3(C)CCC(=O)N3)=O)C2)cccc2c(C#N)c[nH]c12 13067,c1(OC)nnc(Cl)cc1NC(=O)Cc1ccccc1NC(c1sccc1C)=O 13068,CCC(C)CCC(O)CC(=O)NCCC1CCN(C(=O)CS(=O)(=O)C2CCCC2)C1 13069,C=C(C)C(C)(C)C(=O)NC1CC1NC(C1CCN(Cc2cccnc2)CC1)=O 13070,N(C(=NCCc1ncc(Br)s1)NC1CCOCC1)CCN1CC(=O)NCC1 13071,N1(C(=O)CSc2cccs2)CCCC2CN(c3nc4ccccc4o3)CCC12 13072,c1(C(=O)NC2CN(C(C(CCOC)OC)=O)CC2O)cc2cc(C)ccc2[nH]1 13073,C(C)(CCC(=O)N1CC(C(F)Cn2cc(CC3CCCC3)nn2)C1)OCC 13074,c1(C(N2C(CO)CC(NC(C(CC)SC)=O)C2)=O)n[nH]c2cc(C)ccc12 13075,N1(C(c2cnc(C)[nH]2)=O)CCC(C2CCCN(C(c3nc(C)c(C)s3)=O)C2)C1 13076,N1(C(CNC(CC)=O)=O)CCN(C(c2cc(C(N)=O)n(C)n2)=O)C2CC12 13077,C(=O)(C(C(C)O)N(C)C)N(CCNC(C(CC1CC1)OC)=O)C(C)C 13078,C1(O)(CCC)CCN(C(=O)C(C)(C)CNC(=O)C(C)OCCOC)CC1 13079,c1(C(=O)NCC2CC(NC(C3CC3F)=O)C2)cccc(Br)c1 13080,N1(C(COCCOCCOC)=O)CCC(O)(Cn2cc(CC(O)COC)nn2)C1 13081,Cc1cc(=NCc2nnc(C(C)(C)C)s2)[nH]c(N2CC(=O)NC(=O)C2)n1 13082,C=C(F)C1(CC(=O)NC(C)(C)C(C)NC(C2CC2(C(C)C)CC)=O)CCC1 13083,C1(N(C(CC)=O)C)CCCCN(C(C23CC(c4ccc(OC)cc4)(C2)C3)=O)C1 13084,N1(C(C2CN(C)C(=O)C2)=O)CCCOC(CCNC(c2c[nH]cc2C2CC2)=O)C1 13085,c1(OC)ccc(C(N2CC3CC(NC(C4CCC(=O)N4C)=O)C3C2)=O)c(C)c1 13086,c1(C(C)=O)ccc(OC(C)C(N2CC(NC(C3(CO)CC3)=O)C(O)C2)=O)cc1 13087,c1(CN(C(=O)CC2CC(F)C2)CCNC(=O)C=CBr)ccccc1 13088,C1(CC(N2CCC(N(C(=O)C=CCOC(C)(C)C)CC)C2)=O)CC(C2CC2)C1 13089,N1(Cc2ccc(C#N)c(Cl)c2)CCC2(CCN(c3ncc4[nH]ccc4n3)C2)C1 13090,C1(O)(CNC(C(C)(C)C2CCOC2)=O)CCCN(C(=O)CCCN2CCCC2)C1 13091,C12(OC)CCC(C(N3CCC(CCNC(=O)CC4C=CCC4)C3)=O)(CC1)C(=O)C2 13092,C1(NC(c2n(C)ccn2)=O)CCCC(NC(c2cn(CCCF)nn2)=O)C1 13093,N1(C(C(C)C(=O)OC(C)(C)C)=O)CCN(C(=O)CC2CN(C3CCC3)C2)CC1 13094,C1(C(N2CC(NC(CS(CC)=O)=O)(CO)C2)=O)CCc2nn(C)cc2C1 13095,C=CC(CC)CC(=O)N1CCN(CC(N2CCOCC2CN(C)C)=O)CC1 13096,c1(OC)ccc(SCC(=O)NC(=O)CN(C)C2CC2)cc1 13097,c1(N2CCC(COC)C2)ccccc1CSc1nnc(C2CC2)n1-c1ccccc1 13098,C1(C(=O)NC23CC(NC(C(CC=CCC)C)=O)(C2)C3)CN2CCN1CC2 13099,C1(CNC(C)=O)C(C)CCN1C(=O)Cc1cc(C(F)(F)F)n[nH]1.C1CC(=O)N1 13100,c1(C(=O)NCC(CNC(CC(=C)Br)=O)(C)O)cc(C(N)=O)cn1C 13101,N1(C(c2occ(C(N)=O)c2)=O)CCC(O)(CCNC(C2(C(F)F)CCCO2)=O)C1 13102,c1(OC)ccc2c(C(=O)NCC3CC3NC(=O)CCn3ccnc3)cnn2c1 13103,n1(CC)c(=N)[nH]c2cc(C(N3CCC(CNC(C4CCN(C)C4)=O)C3)=O)ccc12 13104,c1(CC)cc(C(=O)NCC(CC(C)C)NC(C2(NC(N)=O)CC2)=O)ccc1O 13105,C(=O)(C(CC(C)C)NC1CCCC1)NC(c1cccc(OC)n1)CC 13106,C(=O)(C1CCc2ccccc21)N(CCC(N1CCCC1CCO)=O)C 13107,c1(C(=O)OCC)ncn(-c2ccccc2F)c1NC(=O)CC1(C)CCCN1 13108,C(=O)(C(F)CC1CN(C(c2cc(C(C)C)on2)=O)C1)NC(C(=O)N(C)CC)C 13109,c1(C(=O)O)ccc(NCC2CCC(C(F)F)CC2)n2ncnc12 13110,C1(C#N)(C(N2CC3C(CN(C(Cc4nnc(C)s4)=O)C)C3C2)=O)CC12CCCC2 13111,c1(OC)ccc(C(=O)NC(C)C(C)NC(=O)CCOC(C)C)c2[nH]ncc12 13112,N1(C(C2(c3cc[nH]n3)CCC2)=O)CCCCC1C(C)(C)CNC(=O)CSCC#N 13113,c1(C(N2C3CC(CC(NC(C(C)C(F)F)=O)C3)C2)=O)cc(F)cc2ccncc12 13114,c1(C(N2CCCC(CNC(c3c(C)ncnc3)=O)C2)=O)ccc(F)c(C(F)F)n1 13115,C1(C(=O)NC2CC(OCC(=O)N(CCCC(O)CO)C)C2)CC2(CCO1)CC2 13116,c1(CC(N2CCC3(NC(CNC(N)=O)=O)C(C2)C3)=O)c[nH]c2ccc(Cl)cc12 13117,O=C(C#CC1CCCO1)NCC1(CNC(=O)C(CO)c2ccccc2)CC1 13118,C1(CC(=O)NCC2(C)CC(NC(Cc3c(C)n(C)nc3)=O)C2)CCCCC(=O)N1 13119,C(=O)(CC1=NN(C)C(=O)C1)N(CCCNC(c1cccc2ncsc12)=O)C(C)C 13120,C1(CC(C)C)(C(=O)N(CC(C)CNC(=O)C(F)=CC2CC2)C)CCCC1 13121,c1(C(=O)NCC2(NC(c3ccc4cccnn34)=O)CC2)ccc2ncccc2c1 13122,O(NC(=O)CC(C)(C)C1CCCCC1)C(C1CC=CCC1C)C(=O)N(C)CC1CC1 13123,N1(C(c2cccc(OCc3cccnc3)c2)C(=O)OCC)CCNC(=O)CC1 13124,c1(C(N2C(CNC(C3CCC(C(F)F)O3)=O)CC2)=O)ccc(-c2ccco2)nc1 13125,C(CC(=O)NCC(CO)NC=O)(OCC)OCCC1CCCN1CC 13126,C1(C(C(=O)NC(C)=O)N(C2CC(F)(F)C2)C(CC)C)CCC(CCC(C)C)CC1 13127,C1(C(N2C(C=C)CC2)=O)(NC(=O)C#CC(C)C)CCC(C)(C)C1 13128,CC1CC=C(C(=O)NC2CCC(CNC(c3cnc4n3CCOC4)=O)CC2)CC1 13129,C1(C(N(CCN(C)C(C2CC(CC3CC3)C2)=O)C)=O)CCOC2(CCCC2)C1 13130,CC(C)CC(C(=O)N(CCCNC(C1CNC(=O)C1)=O)C)NC(=O)OC(C)(C)C 13131,N1(CC)CCN(C(C2(CC)C=CCN2C(c2cnc(O)c(F)c2)=O)=O)CC1C 13132,c1(C(N2C(CNC(c3c(C)cc(C)nc3)=O)CCC2)=O)cc2cccnc2cn1 13133,C1(CCCCC2C(C(=O)OC(CC)(C)C)C2)CCCN(C(=O)C(F)(F)COC)C1 13134,n1(CC(=O)N(C2CC3N(C(CCC#C)=O)C(CC3)C2)C)nc2n(c1=O)CCOC2 13135,C#Cc1ccc(CC(=O)NCCC(C)(CC)NC(C2C=CCCC2)=O)cc1 13136,CC1(C)CCC(CC(=O)NC(C)(CO)C(=O)NC2(c3ccsc3)CC2)O1 13137,C1(C(=O)NCCC(C)NC(=O)C(F)(F)c2nccn2C)CCCC2C1C2(F)F 13138,c1(C(C)(C)C)ccc2c(c1)OCC2C(=O)Nc1nccn1CC1CC1 13139,Nc1sc2c(c1C(=O)NCCC1CN(C(=O)CN(C3CCCC3)C)C1)CCC2 13140,c1(C(=O)NC2(CCC(=O)NC(C)C(C)n3cccn3)CCC2)coc2c1COC2 13141,Cn1cc(C=CC(=O)NC2C3CCC4C(C3)C24C(=O)O)c2ccccc12 13142,N1(C(c2ccc(NC(C)=O)o2)=O)CCC(NC(=O)C(C)S(C)(=O)=O)C2(CCC2)C1 13143,[N-]=[N+]=NCCCCCC(=O)N1CC(C(=O)NCCC2CCC3CC23)CC12CCC2 13144,C(=O)(C1=CCC(C)CC1)NC1CCN(C(CCn2c(C)nc(C)n2)=O)C1C1CC1 13145,C1(n2cccn2)(C(=O)NC(COCC)C)CCN(C(C2CCC2OC)=O)CC1 13146,CC(=O)CCCC(=O)N1CCCC(NC(=O)C(c2ccc(Cl)cc2F)O)C1 13147,c1(C(=O)NC2CCCC(NC(C3CC4CC4C3)=O)C2)ccc2nn[nH]c2n1 13148,C1(NC(c2ncc(C)nc2)=O)C(C)CCN(C(c2cnc3scc(C)n23)=O)C1C 13149,c1(C(C(=O)NCCOC)N(C2CCC2)CC)ccc(OC(F)F)cc1.OCF 13150,C1(CC)CN(C(=O)CCn2cnccc2=O)CCC1NC(=O)C(CC)C(C)O 13151,C12(CCCC1)C(=O)NC2.C(=O)(CCOCC1CCCC1)NC1(CC=C)CC1 13152,N1(CC(=O)NC2CC(C)(NC(=O)CC3CC4CC4C3)C2)CCC(=O)NC1=O 13153,N1(C(C(CC#C)C)=O)CCC(NC(c2cn(C)nc2-c2ccco2)=O)C(CO)C1 13154,N1(C(C(C(C)C)(C)O)=O)CC(NC(c2ccc(F)s2)=O)CC(C)(C)C1 13155,N1(CCNC(NCC(C)C)=NCCC2CCS(=O)(=O)C2)CCc2ccccc21 13156,c1(-c2c(F)ccc(OCCC)c2)ccc2c(c1)CN(C(C1(C#N)CCC1)=O)CC2 13157,C#CC(CNC(=O)CC1(CNC(C2CCO2)=O)CC1)CC1CC1 13158,N1(C(C2C(CC)C2)=O)CC2(C1)CC1(C)CC(OC)C(C(=O)OC)(C1)C2 13159,NS(=O)(=O)c1ccc(NNC(=O)Cc2ccc3sccc3c2)nc1 13160,N1(C(CCCCC#C)=O)CC2(C1)CN(C(C1CC13CCCCC3)=O)CC2CO 13161,C1(NC(CCCSC)=O)CCOC(CNC(=O)C(C)N=[N+]=[N-])C1 13162,CN1CC=C(CNC(=O)C(C2(O)CCC2)NC(C2CC(C)(C)CO2)=O)CC1 13163,c1(C(N(C(C)CNC(c2ccn(C(F)F)n2)=O)C)=O)ccc(CO)cc1F 13164,N1(C(C(F)=CC)=O)CCC(C(C)NC(C2(c3oncc3C)CC2)=O)C1 13165,Cc1nccc(C(=O)NC2CN(C(C3CC3C)=O)CC2CC(C)(C)C)c1N 13166,n1(-c2ccc(OC)cc2)ccc(=NC(=O)C(C)N2CC(Cc3nn[nH]n3)C2)[nH]1 13167,N1(C(c2ccn(CC)n2)=O)CC(NC(C2CN3CCC2(C)CC3)=O)CC12CCC2 13168,S(=O)(=O)(c1ccccc1Cc1ccccc1)N1CCOCC(C(C)C)C1 13169,S(=O)(=O)(CC(=O)N(C)CC1CCCCN1C(c1cnn(COC)c1C)=O)NCC 13170,c1(OC)ccc(C(=O)NCCCC(C)NC(c2cnc(C3CC3)o2)=O)c(F)n1 13171,C(=O)(C(CC(N)=O)NC(C1CC(C(C)C)=NO1)=O)NC(CC=C)CO 13172,Nc1ccc(OCC(N2CCC(CNC(c3scnc3C(F)(F)F)=O)C2)=O)cc1 13173,CCCCCC(=O)NC1(CCOC)CCN(C(c2cn(CCC(C)C)nn2)=O)C1 13174,C1(C(=O)NC23C(CN(C(C4N(C(C)=O)CSC4)=O)C2)C3)CC2CSCC(C1)C2 13175,C1(C(=O)NCC2(C)CC3(CC3)C2)(CNC(CC)=O)CC12CCC2 13176,N1(C(C2C(C(N)=O)CCCC2)=O)CC2CC(C1)N(c1cc(F)ncn1)C2 13177,CON(C)C1CN(C(=O)CC2CCCCN2C(=O)COCCCF)C1 13178,C1(CNC(CC2(COC)CC2)=O)CN(C(c2cc[nH]c(=N)c2)=O)C2CC12 13179,c1(OC)cccc(CC(N2CCCC2C(C)NC(=O)C=Cc2ccco2)=O)n1 13180,C(=O)(C1=NOC2(CCC2)C1)NC1CC(C(=O)NC2CN(C)C(=O)CC2)C12CCC2 13181,c1(NCC2(OC)CNC2)cnc2n1CCOC2 13182,N(C1c2ccccc2CC1NC(=O)C=C1CCC1)C(C1N(N=O)CCCC1)=O 13183,CC1(C)CC(C(=O)NCCNC(=O)C(c2ccc(Cl)cc2Cl)O)CC(C)(C)O1 13184,c1(C(C)=O)cccc(OCC(N2CC(NC(=O)CCC3(C)CC3)C3CC23)=O)c1 13185,n1(CC(C)CO)cc(C2CCCN2C(=O)C=CI)nn1 13186,Cc1nccc(C(=O)NCc2cncc(C(=O)NC3CCN(C(C)C)C3)c2)c1N 13187,c1(CNC(c2c(OC)ccs2)=O)ccc(CNC(C2CCC(=O)N2C)=O)c(F)c1 13188,N1(C(c2ccc(OC)nc2)=O)CCN(c2cccc(Cl)c2)C(C)C1 13189,C1(CNC(c2cc[nH]c2)=O)C2CCC1CN(C(=O)CC(O)c1ccccc1)C2 13190,N1(C(C(=Cc2ccccc2)C)=O)CCCC(C)(C(=O)NCC(C)(C)O)C1 13191,C(CC(C(=O)NCC(C)(C)C(C)O)NC(=O)CC1CCCC(=O)C1)OCC 13192,C1(C(=O)NC(CNC(C(CCSC)O)=O)(C)C)Cc2ccc(Br)cc2C1 13193,C1(COC)CN(C(c2ccc(F)s2)=O)CCN1C(C1CC(=O)N(CC(C)C)C1)=O 13194,C(C(C(=O)N1CCCC1CCNC(=O)C(C)Oc1ccccc1)OC)OC 13195,C1(C(N2CC(c3ccc(OC)cc3)OCC2)c2ccccc2)CCC(F)(F)CC1 13196,N1(C(C#CCNC(N)=O)=O)CCC2CCN(C(=O)C3Cc4ccccc43)CC2C1 13197,c1(C(N2CC(C3(NC(C(CC)CN(C)C)=O)CC3)C2)=O)cc2cccnn2c1 13198,c1(C(=O)NCC(C)(C2CC2)NC(C2CCC2(F)F)=O)cc2c(nn1)CCOC2 13199,C1(C(N2C(CNC(C3CCC(C)(C)CO3)=O)CCC2)=O)CCCN(S(N)(=O)=O)C1 13200,C(CN=c1ccnc(N2CCN3CC(O)CC3C2)[nH]1)(C1CCCCC1)OC 13201,CCC(C)(CO)C(=O)N1CC(CNC(c2ccnnc2)=O)C(F)(F)C1 13202,CC1CC(C)(C(=O)NCC2CN(C(=O)CCCOc3ccccc3F)C2)CCO1 13203,c1(CC)cc(C(=O)NCC(C)(F)CNC(C2CCCCC2O)=O)ccc1C 13204,CC(CNC(=O)CNC(=O)CN(C)C)C(F)C(=O)NCC1CC1(F)F 13205,C(=O)(C(C)CS(C)(=O)=O)NC1CC(C)(NC(CC2N(C(C)=O)CCC2)=O)C1 13206,c1(OCCO)cccc(NC(=O)CC2CCN(c3ncc(Cl)cn3)C2)c1 13207,c1(OCC)ncccc1C(=O)NCC1(CNC(=O)CCN2CCC2)CC1(F)F 13208,CC1CN(C(c2ccc(C(F)(F)F)cc2Br)=O)CCN1C(c1ccnnc1)=O 13209,c1(C(N(CCC(=O)NC(C(C)SC)C)C2CC2)=O)ccnc(C)n1 13210,N1(C(CSCCCC)=O)CC2(C1)C(NC(C1CCC3CC3CC1)=O)CCS2(=O)=O 13211,Cc1cc(C(N2CCC2CNC(c2cc(-c3ccco3)no2)=O)=O)cn1C 13212,c1(C(=O)NCC(c2ccc(OC)cc2)NC(CC=CCC)=O)cc(C)c(F)cn1 13213,c1(C(=O)NCCC2CCCN(C(C3C(=C)CC3)=O)C2)cc(F)c(CC)cc1F 13214,c1(CN2C(CCC(=O)NCCCCCC)CCC2)ccc([N+](=O)[O-])cc1OC 13215,C1(C(C)C)CN(C(=O)CN2CCNC(=O)C2)CCN1C(=O)CC1CCCCC1O 13216,c1(C(N(C2CCN(C(C3CCCS3)=O)CC2)CC)=O)n[nH]c2c(C)cccc12 13217,c1(C(=O)NCC(C(C(C)C)C)NC(c2nsnc2O)=O)cc(F)c(F)c(F)c1F 13218,c1(CC(=O)NC2CCC(CNC(C(C)(F)F)=O)C2)cccc2cnccc12 13219,C(=O)(C1=NOC2(CCC2)C1)NC(C)(C)CCCNC(C1(C)CCC(=O)NC1)=O 13220,C1(C(N2CC(NC(=O)NC)C2)=O)C2CC(O)C1N(C(=O)C(c1ccnn1C)C)C2 13221,C(=O)(C(CC)(CC)CC)N1C2C(NC(C3N(CC)CC3)=O)CC(C2)C1 13222,C=CCC(C)(C)CC(=O)NC1CC(NC(c2ncccc2Cl)=O)C1 13223,c1(C(=O)NCCC2CC(C(=O)Nc3ccsn3)C2)c[nH]nc1-n1cnnn1 13224,C1(N(C(c2cn(C)nn2)=O)C)CCCCC1O.C1(C(=O)NC)(CN)CC1 13225,C1(NC(C2C=CCC2)=O)C=CCN(C(=O)CC(c2ccccc2)c2ncc[nH]2)C1 13226,CC1(C)CCC(O)(NC(=O)CCCC2(NC(=O)CN3CCOCC3)CCC2)C1 13227,c1(CN2CCC(N3CCN(c4cc(CC)ncn4)CC3)C2)cccn2nccc12 13228,CC1CN(C(c2ncn3c2CCCC3)=O)CC(C)C1NC(c1ccc[nH]1)=O 13229,CS(=O)(=O)CC(=O)NCC1(C(=O)Nc2cccc(CCO)c2)CC12CCC2 13230,C1(F)(CNC(C(c2c(C)cccc2)C)=O)COCCN(C(=O)CSC(F)F)C1 13231,c1(CN2CCC(N(C)C(c3ccsn3)=O)C2)cccc(C=O)c1Br 13232,C(CC(=O)NC1CCN(C2CCN(C)C2=O)CC1)(C(F)(F)F)NC 13233,N1(C(c2ccc(C)cc2F)=O)CCC2CN(C(=O)CC3CCCCO3)C2C1 13234,c1(COCC)noc(C2CC2C(=O)NCCC(C)NC(=O)Cc2ccccc2)n1 13235,c1(NC)ccnc(C(N2CCC(CNC(=O)CCC(C)c3ccccc3)C2)=O)c1 13236,C(=O)(CCCC(=O)NCCCC(C)(C)NC(C1CC2CCC1C2)=O)NCC 13237,N1(C(C2(CC#C)CCCO2)=O)CCC(N=c2cc(C)nc([N+](=O)[O-])[nH]2)C(CC)C1 13238,N1(CC(=O)NC(C)CCNC(=O)Cn2nnc(C3CC3)n2)CCC(N(C)C)CC1 13239,c1(COC2CCN(C(C3(C(=O)O)CCC3)=O)C2)c(C2CC2)cccc1F.CCO 13240,c1(C(N(C(C)CCNC(c2ncn(C)n2)=O)C)=O)ccnc(C(C)(C)C)c1 13241,Cc1cccc(CCN(CC(C)C)C(C)Cc2ccc(OC(F)F)cc2)c1C 13242,N1(C(C2CCC(C)(CC)O2)=O)CC=C(CC(=O)NCc2ccc(F)c(O)c2)CC1 13243,N1(c2c(OC)c(C3CCN4CCCC3C4)ncn2)CCCC(C)(C)CC1 13244,C1(CNC(c2nn(CC)nc2C)=O)(NC(C2CC(O)C2)=O)CCCCC1C 13245,c1(C(=O)NC2COCCN(C(C(CCSC)O)=O)C2)cc2ncccc2s1 13246,c1(C(=O)NC(C2CCN(C(C=CCC)=O)C2)C)c(C)cnn1C 13247,c1(CC(N2C(CCNC(=O)Cc3ccno3)CCC2)=O)ccc2ncsc2c1 13248,C(CC(C)C)(C(=O)NC1(CNC(C2CCOC2)=O)CC1)OC 13249,C1(C(=O)NCC(CNC(=O)C2CC2)OC)CC2CCC(C1)N2S(C)(=O)=O 13250,C(C(C)C(=O)N(C1CCC1)C)N(C(CCNC(C)=O)=O)C 13251,C1(NC(C(CC=CC)C)=O)C2CCC(C2)C1C(=O)NCC1CCC(C)C1 13252,c1(C(N2CC(CNC(C(C=C)(C)O)=O)C(COC)C2)=O)ccc(SC)c(Br)c1 13253,C1(C(=O)NCC(C)(C)C(F)F)CN(C(=O)CC2CC(C3CC3)C2)C2(CCC2)C1 13254,N1(C(c2cncc(SC)c2)=O)CC(NC(=O)CC2CNC(=O)C2)CC(C)(C)C1 13255,C(=O)(C1CCc2c[nH]nc21)N1CCCN(C(C(CCC)(C)O)=O)CC1 13256,c1(C(=O)NCC(C)N(C(c2cnc[nH]c2=N)=O)CC)ccc(F)cc1OC 13257,C1(C(C)OC)CCN(C(=O)C=CC(C)NC(=O)C(C)C2CCCC2)CC1 13258,N1(C(C=CCC)=O)C2CCC1C(NC(c1cccn1C1CCCC1)=O)C2 13259,C1(CCC)CN(C(=O)C(C)(C)n2cccn2)CC1NC(C1C=CCC1)=O 13260,N1(C(CC(CN(C)C)O)=O)CC(C(=O)NCC(C)(C)CCCO)C(F)(F)C1 13261,N1(C(CCC(C)N(C)C)=O)CCCN(C(C2(n3cncn3)CC2)=O)CC1 13262,Cc1cccn2ncc(C(N3CC4(CCN(C(=O)CN5CCOCC5)C4)C3)=O)c12 13263,CN1CCN(C(=O)Cc2cc(C3CC3)on2)C(CNC(c2n[nH]cc2Cl)=O)C1 13264,c1(CN2C(C(=O)NCc3ncc(Br)s3)CC(O)C2)c(Cl)ccnc1Cl 13265,C1(=O)CC(C)(C)C(CC)CNC2C(CNCc3ccc(C(=O)NC)o3)CCN12 13266,N1(C(c2cc(C(N)=O)c(O)cc2)=O)C(CNC(=O)CCC(F)F)CC2COCC12 13267,c1(-c2ccc(Sc3ccc(CC)cc3)cc2)n[nH]c(=NC(=O)Nn2cncn2)s1 13268,C(N=c1[nH]cc2c(c1C#N)CCCC2)c1ncc(C)o1 13269,C(CCCC(=O)O)n1cc(SCCNC(C(c2ccnn2C)C)=O)nn1 13270,Cc1c(CC(N2CCOC(C(=O)N(C3CCCC3(F)F)C)C2)=O)cnn1C 13271,C(CS(=O)(=O)C1=CCCCC1)Nc1c(F)ccc(C(N)=O)c1 13272,C12(C(=O)NCC(CCNC(C3(CCN(C)C)CC3)=O)O)CCC(C1)C2(C)C 13273,CC(C)CC(O)CC(=O)N1CCC(C(C)(C)CNC(C2CCOC2)=O)CC1 13274,C#Cc1cc(NC(c2ccoc2CNC(=O)CC2CSC2)=O)cc(F)c1 13275,N1(C(CCCC)=O)CCC(NC(c2csc(-c3ccsc3)n2)=O)C(CC)C1 13276,c1(C(=O)NC2CC3(CN(C(C(C)CN(C)C)=O)C3)C2)nnc(O)c2ccccc12 13277,N1(C(C2CC=CC(NC(C3(CO)CCCCO3)=O)C2)=O)CC2C=CCC(C2)C1 13278,c1(C(=O)N)cn2ccnc2cn1.C1(C2CCC2)CCCN1C(C1CC1F)=O 13279,C1(C(N(C(C)C(=O)NC2CCOC2)CCC)=O)CCCC(C#N)C1 13280,Nc1ccc(C(N2CC(NC(=O)C(F)C(F)(F)F)C2)=O)nc1C(F)(F)F 13281,C(C(CC(C)C)NC(C1CCCO1)=O)NC(CSC(C)C)=O 13282,C1(NC(C=CC(C)NC(c2c(CC)[nH]cc2)=O)=O)(CO)CCCCC1C 13283,C12CN(CC1F)C2=O.C1(NC(CNC(=O)NC)=O)CCCOC1 13284,CC1CC(=O)NCC1C(N1CCC(C)(CNC(=O)CC2(O)CC2)CC1)=O 13285,c1(OC)ccc(OCCNC2COC3CC2C3)cc1 13286,c1(CC2(NC(c3cncc(OCC)c3)=O)COC2)ncnc2cc(Br)ccc12 13287,C(=O)(C1CCCc2sccc21)NCC1(NC(C2CCN(C)C2)=O)CC1 13288,Cc1cccc(CN(C(=O)C(CCC2CC2)NC(=O)C(C)c2cc[nH]n2)C)n1 13289,N1(C(C(CC(C)C)CNC(c2ccon2)=O)=O)CC2CCOC(=O)C2C1 13290,c1(OC)cc2nn[nH]c2cc1C(=O)NCCCCNC(c1cnn(C)n1)=O 13291,C1(Cc2onc(C3N(C(c4cnc(COC)s4)=O)CCC3)n2)CCN(C)CC1 13292,c1(C(N(C)CC2(CNC(C3C(CC)C3)=O)CC2)=O)ccnn1CC 13293,c1(CC(N2C(C)CC(NC(c3cc(C(C)=O)[nH]n3)=O)C2)=O)ccc2nonc2c1 13294,C1(C(=O)NC(C23CCC(CC2)C3)C)(NC(C2CCO2)=O)CCCCC1 13295,c1(C(N2CC3CC3(C(=O)NCc3cncs3)C2)=O)cc(Cl)c(O)cc1F 13296,C#CC1(C(=O)NCC(C)(C)C2(O)CCC2)CCN(C(=O)CCC2CC2)CC1 13297,CC(C)C(F)(CNC(C1(CCN(C)C)CC1)=O)C(=O)NCC(C)(O)C1(C)CC1 13298,n1(CCC(N2C(C)CN(C(C3(CO)CCCO3)=O)CC2)=O)ccc2ccccc12 13299,C1(NC(C2(NC(CC(=O)OCC)=O)CCSC2)=O)CC(C2CCCC2)C1 13300,C(=O)(C1CCCn2cnnc21)NCC1(NC(=O)COc2cccnc2)CC1 13301,c1(N(CCC(N)=O)C)ncnc(N2CCC(OCc3ccccc3)C2)c1[N+](=O)[O-] 13302,c1(C(=O)OCC)nnn(C)c1CNCc1cscc1Cl 13303,C1(CNC(C2(C3N(C(CCSC)=O)CCC3)CC2)=O)CNC(=O)CO1 13304,n1(CC)ccc(CNC(=O)CC2(OC)CN(C(=O)CC(O)c3ccccc3)C2)n1 13305,C1(C(N2CCN(c3nc(C)cc(C)n3)C(C)C2)=O)CCCC2CCCCC12 13306,Cc1ncccc1NC(c1c[nH]nc1CCCNC(=O)CC1CCCC(C)O1)=O 13307,c1(C(=O)NCC(CC)NC(C2NC(=O)CC2C)=O)ccc(N)cc1O 13308,C1(C(=O)NCCOCCC(=O)NC(CC)C2CC2)CCC1C#N 13309,c1(OC)cc(F)c(F)cc1CN1CC(C(=O)Nc2cnc(Br)nc2Cl)CC(F)C1 13310,N1(C(C2N(C(C3C(C(C)C)CCO3)=O)CCC2)=O)CC2(CCC2)CC1CO 13311,C1(CC#C)(C(=O)NC(CC(N)=O)C2CC2)CCN(C(c2ccnn2C)=O)C1 13312,c1(OC)cc(C)nc(NC2CC(NC(c3nsc(OC(C)=O)n3)=O)C23CCC3)n1 13313,O=C1NCCCCC1C(=O)NCC12CC(CN1C(c1ncccc1Br)=O)C2 13314,N1(C(c2ccc(OCC)nn2)C(=O)NCCC)CCS(=O)(=O)C2(CCC2)C1 13315,N1(C(C(CC#C)C)=O)CCOC2CN(C(=O)Cc3cccc(OC)c3Cl)CC12 13316,C1(NC(C2CC(O)(c3ccncc3)C2)=O)CCC(NC(C2CCOCC2)=O)C1 13317,Cc1ncc([N+](=O)[O-])cc1NC(=O)CC1CCN(Cc2cc(F)c(F)c(F)c2)C1 13318,O=CN1CCCN(C(=O)CC(CC2CC2)NC(=O)COC2CCOC2)CC1 13319,c1(C(=O)NC2CCN(C(CNC(=O)OC)=O)C(C)C2)coc2cc(C)ccc12 13320,C(CC)(CCCO)NC(C1(CC=C)CCCN1C(=O)C(C#N)CC)=O 13321,c1(OC)ccc2[nH]ccc2c1C(N1CCC(C)(NC(=O)C(CC(C)C)OC)C1)=O 13322,C(=O)(C(C)(C(C)C)OC)NC(CC=C)CNC(c1n[nH]c(C)n1)=O 13323,c1(C(=O)NC2C(C)CN(C(=O)CCC3(C)CC3)C2)ccc(N)cc1Cl 13324,C=CCC(C)(C)C(=O)N1CCC(C(C)NC(=O)C=Cc2cnn(C)c2)C1 13325,Cc1ccc(O)cc1C(N1CC(C)CC1C(=O)N(C1CC2CC2C1)C)=O 13326,c1(CC)nn(C)cc1C(=O)NCCCN(CCO)C(C1CC(C)(F)C1)=O 13327,CC1(C)C(NCC(F)(F)C(F)(F)F)C2CCCN(C(C3CC34CCCC4)=O)C12 13328,Cc1ccc2ccc(C(=O)NC3(CNC(C4CCCSC4C)=O)CCC3)nc2c1 13329,CC1CCN(C(C2CCCCO2)=O)CCN1C(c1ccn2ccccc12)=O 13330,C(CN=c1[nH]c(=N)[nH]c(=NCCC(C)CC(C)(C)C)[nH]1)C1OCC(C)C1 13331,CC(CO)(C(=O)NC(C1CCCCC1)CO)NC(=O)CCC1CCOCC1 13332,N1(C(CC2(C)OCCO2)=O)CCOC(CC(N2CCC(O)(CO)C2)=O)C1 13333,c1(CC)cnc(C(=O)NCCCCNC(c2cc(Cl)n(C)n2)=O)nc1 13334,CC1CN(C(=O)CS(N)(=O)=O)CCC1N(C)C(c1cnc(C(F)F)nc1)=O 13335,C1(CC(=O)N(CC(C)NC(=O)CCCCCn2cnnn2)C)CCS(=O)(=O)CC1 13336,CCC(CC)C(=O)NC1CC(CO)N(C(=O)CNS(C)(=O)=O)C1 13337,CC1CC2CN(C(C3CC3(Cl)Cl)=O)CC2N1C(=O)C(O)CC(N)=O 13338,C1(OCC(N2CC(Oc3ccsc3)C2)=O)CCN(C(C23C=CC(CC2)C3)=O)CC1 13339,C1(C(=O)NC(c2ccnc(F)c2)C)CCCCCN1C(c1ccc(C(N)=O)o1)=O 13340,CCC(C(=O)N(CC(C)O)CCNC(=O)CC1CCCO1)NC(c1ccco1)=O 13341,C1(C(N2CCCC2CNC(C23CC(F)(C2)C3)=O)=O)CCN(CCO)C(=O)C1 13342,C1(NC(C(C)OCC)=O)CN(C(c2c(Cl)csc2Cl)=O)CC1(C)C 13343,N1(C(CN(C)C)=O)CCC(C(N2CCC2c2ccccc2O)=O)CC1 13344,CCCCCC(C)CC(=O)NCCC1(C(N2CC3CC2CS3=O)=O)CCC1 13345,C1(C(=O)NC2CCC(CNC(=O)CSC3CC3)C2)CC2(CCOC2)C1 13346,C(=O)(CC(C)(C)NC(=O)C(C)C)NCCN(C(=O)C(C)(C)COC(C)C)CC 13347,CN(C)S(=O)(=O)N(C)CC(=O)NCCC1CCC(NC(=O)CC2CC(F)C2)C1 13348,c1(OC)cc2c(cn1)NC2=O.N1(C(c2csc(C(N)=O)n2)=O)CCCC(OC)C1 13349,c1(C(=O)NCC2(F)CC(NC(C3C(OC)CCC3)=O)C2)oc(CO)nc1C 13350,C1(NC(c2ccnc(C)n2)=O)C2CC1CN(C(=O)CSc1ccccc1Cl)C2 13351,CC1CCC(CNC(=O)C(O)C(F)(F)F)CN1C(c1cnc[nH]1)=O 13352,CC(C#N)CCC(=O)N1CC(CNC(c2cc(-c3cnn(C)c3)on2)=O)C(O)C1 13353,C1(C)(C(=O)NCC2(CC3CCC3)CN(C(C(CC)NC(N)=O)=O)C2)C=CCCC1 13354,C1(N(CC#C)C)CCN(C(C2CC2C(=O)OCC2CC(=O)N(C3CC3)C2)=O)CC1 13355,c1(C(=O)OCC)cnc(N2CCC(OCCNC(=O)C(O)Cc3cnc[nH]3)C2)s1 13356,C1(C(=O)NCC(C(C)C)O)CN(C(C2CCC2C)=O)CC1(C)C 13357,c1(C(N2CC(CCO)(NC(CSC(C)C)=O)C2)=O)nncc2ccccc12 13358,C(=O)(C(CO)C(C)C)NCC(C)N(C(Cc1cccc(C(C)C)c1)=O)C 13359,c1(OC)ccc(C(=O)NCCNC(=O)CC2CCCC(C)C2)nc1Br 13360,N1(C(CC(CC)C(C)C)=O)CCCC2(CCN(C(=O)C(C)(C)C(O)CF)CC2)C1 13361,C1(NC(c2c(C)cns2)=O)CCC(CNC(c2csc(Br)n2)=O)CC1 13362,C1(C(=O)N=c2ccnc(-c3ccccc3)[nH]2)CC(c2cccnc2)=NO1 13363,CC(C)C(CNC(=O)C=C(C1CC1)C1CC1)C(=O)N1CCC(O)(C(N)=O)C1 13364,Cc1c(CC(=O)NCCCCN(C)C(c2ccnn2C)=O)ncn1C 13365,N1(C(C(C)OCC(F)(F)F)=O)CC2(C1)SCCC2NC(=O)CCCC(N)=O 13366,CC1CN(C(c2cccc(F)c2)=O)CCC1NC(c1ccccc1SCC#N)=O 13367,C1(C(N(CC(CCC)O)C)=O)(CNC(c2c(C)cnn2C)=O)CC12CCC2 13368,C1(C(N2CCN(c3cncc4nccn34)CC2)=O)CC2(C1)CC21CCC1 13369,c1(OC)cc(NC2CCN(CC(N)=O)CC(F)(F)C2)c([N+](=O)[O-])c(F)c1 13370,N1(C(CC2(N(C(c3ccc(C)o3)=O)C)CC2)=O)CC(C)C(C)(CO)C1 13371,N1(C(C(CC)N(C(N)=O)CC)=O)CC2CCC1C(NC(=O)C(c1cccnc1)O)C2 13372,C12(C(=O)NCCCC(=O)OC)CC1CN(C(c1c[nH]c(=N)s1)=O)C2 13373,C1(C(N(CCN(C(=O)C(O)CC(N)=O)C)C)=O)CSc2ccccc2O1 13374,c1(OC)ccc(F)cc1CCC(=O)N1CC(NS(=O)(=O)CC2C(C)(C)C2(F)F)C1 13375,C(C)(CCC(=O)OCCOCC)NCc1cccc(CN(C(=O)N(C)C)CC(C)=O)c1 13376,c1(CC(=O)NCCCC(C)NC(c2ccoc2)=O)cccc(OC(F)(F)F)c1 13377,N1(CC(=O)NC2CCC2NC(C2(CC(F)F)CC2)=O)Cc2ccccc2C1 13378,Cc1nc(O)nc(O)c1CC(=O)NC12CCCC1N(C(=O)C(F)(F)C(C)O)CC2 13379,N1(C(CC(CC)(C)C)=O)CCCN(C(c2ccc(OC3CCC3)cc2)=O)CC1C 13380,CC1CCC(CNC(=O)C(Cn2cccn2)NC(=O)CC23CCC(CC2)C3)N1C 13381,C1(C(c2ccccc2)C(=O)NCCN(CCC(C)C)CCOC)CCCCCC1 13382,c1(C(=O)NCC(CC)NC(c2ccn(-c3cccc(F)c3)n2)=O)cccnc1C 13383,C12(C(=O)NCCCN(C(=O)CN3CCCS3(=O)=O)CC)CCCCC1C2(F)F 13384,c1(COC)nc(NCCCS(C)=O)cc(=NCC2(CS(C)(=O)=O)CCC2)[nH]1 13385,N1(C(COCCCC)=O)CCC(C(C)(C)CNC(=O)CC2NC(=O)NC2=O)CC1 13386,CC1CC(NC(=O)CC2CC3(CC3)C2)CCN1C(=O)CCN1CCCCC1=O 13387,CC(C)CC(C)(CNC(=O)Cc1c[nH]nc1O)NC(C1CC(=O)NC(=O)N1)=O 13388,C1(C(=O)NCCN(C(=O)CCc2cncs2)CC)CCC(=O)N1CCC(F)(F)F 13389,C1(OCC(=O)NC2CC(NC(Cn3ncc(C(=O)OC)c3)=O)C2)CCCCC1C 13390,C1(NC(C2=C(C)CC2)=O)CN(C(c2csc(CO)n2)=O)CC(F)(F)C1 13391,CCC(CC(=O)NCC1(O)CCN(C(=O)COC2(C)CCCC2)C1)CC(C)C 13392,C(=O)(CC(C(=O)N1C(C)C1)NC(C)=O)OC.C(=O)(CCCC(C)=O)NCCS.O 13393,N1(C(=O)OC(C)(C)C)CCC(C(N2CC3CC3(C(=O)O)C2)=O)C(C)(C)C1 13394,Cc1cc(C)c(C(=O)NCCC2CN(C(C3CNC(=O)N3C)=O)CCO2)c(C)n1 13395,CCN=c1[nH]c(C)c(C(=O)NC(C2(CNC(=O)Cn3nc(C)oc3=O)CC2)C)s1 13396,c1(C(N2CC(C(=O)NC(CN(CC)CC)C)C(OC)C2)=O)ccc(C#N)n1C 13397,c1(C(N2CCC(NC(C(CC)CO)=O)C(F)C2)=O)cc2nc(C)ccc2o1 13398,c1(C(=O)NCC2CC(NC(C3CC34CC4)=O)CCO2)cc2ccc(F)cc2o1 13399,c1(C(=O)NCCCCCN(C(C(C)OCC2CC2)=O)C)ccc(Br)cc1O 13400,C1(CC)CN(C(C2CN(C)CCN2C)=O)CCC1NC(c1cnc(C(C)=O)s1)=O 13401,N1(C(C(C)NC(C2CN(C)C2)=O)=O)CC(=O)NC(=O)C1C 13402,c1(OC(C)C)ccc(CCC(C)NC(=O)CC2CSCCS2)cc1 13403,CC1(C)OC(=O)NC1C(=O)NC1COCCC1NC(C1CC(F)(CF)C1)=O 13404,c1(SC(C)C)ccccc1C(=O)NCC(C)(C)CNC(c1cc(O)ccn1)=O 13405,c1(C(=O)NCC=CCC(=O)NC(COC)(C)C2CC2)ccn(C)n1 13406,N1(C(CC2N(C(c3cccc(OC)n3)=O)CCCC2)=O)CCC2(CC=CCO2)C1 13407,C1(F)(C(N(C)CC2COCCN2C(=O)C=Cc2cccs2)=O)C(C)(C)C1(C)C 13408,C(C(CC(C)C)NC(C1CC(=O)N(C)C1)=O)NC(C=CC=CC)=O 13409,c1(C(C)C)onc(C2CCCO2)c1C(=O)NC(C)CCNC(=O)C=C(Cl)Cl 13410,c1(N(C)C)ccc(C(CNC(C2(C)CCOC2)=O)NC(=O)CCNC(N)=O)cc1 13411,C1(C(=O)NCC(C)S(C)(=O)=O)CCCCS1(=O)=O 13412,c1(CNC(=O)COCCCCCC)cccc(-n2cc(-c3ccncc3)nn2)c1 13413,N1(C(c2c(C)oc(Cl)n2)=O)CC(NC(C2CN3CCN2CC3C)=O)CC(F)(F)C1 13414,N1(CCC)CCCC(C(=O)NC(C)(C)CNC(c2c[nH]c(=N)o2)=O)C1 13415,N1(C(C(C)N2CCC2)=O)CC(CNC(=O)Cc2ccc(F)nc2)CC1(C)C 13416,C1(Br)(C(=O)NCC(C)N(C(c2cc(CC)on2)=O)C)CC12CCC2 13417,c1(C(=O)OC(C)(C)C)cn(C)nc1CN(C(C(C)C)=O)CCCN(C)C 13418,Cc1ncn(CCNC(c2conc2C(C)NC(=O)CCC2CC2(F)F)=O)c1C 13419,C1(C(N(C2CC(NC(C(SC)SC)=O)C2)C)=O)CCCC2(CC2)C1 13420,c1(N2CC(CNC(=O)C(F)CC3CCCC3)OCCC2)nc2ccc(F)cc2o1 13421,c1(CC(=O)N(CCC(C)NC(COCC(=C)C)=O)C)ccc(S(=O)C2CC2)cc1 13422,C#CCC(C)(C)C(=O)N1CCOC(CCNC(=O)Cn2ccc(C)c2)C1 13423,CC(O)C(C(=O)NCC1CCCCN1C(c1coc(C(F)F)c1)=O)N(C)C 13424,c1(C(N2CCC(C(C(C)C)NC(CCC=CC)=O)CC2)=O)cc(S(C)(=O)=O)cs1 13425,N1(C(CCCCSC)=O)C2CC1CN(C(=O)CCP(C)(C)=O)C2 13426,c1(CCC(=O)NCC(C)(C2CC2)NC(C2(F)CCCCC2)=O)nc2ccccc2[nH]1 13427,N1(C(c2ccc(CC)[nH]2)=O)CC2CC2(CNC(=O)CC2CCC(=O)N2C)C1 13428,c1(C(=O)OC)ccc(OC)nc1NC(c1nc(NC(=O)CC2CCC2)cn1C)=O 13429,Cc1ccc2[nH]c(C(=O)NC3CN(C(=O)C(C)Oc4cccnc4)C3)cc2c1F 13430,Cc1nc(C(C)(F)F)ccc1C(N1CC(NC(C23CCCC2C3)=O)C(C)(C)C1)=O 13431,C(=O)(CCCCC(F)(F)F)NC1CC(NC(c2cc(C3CCC3)[nH]n2)=O)CC1O 13432,c1(OC)ccc2c(c1)C(C(=O)NCCCNC(c1cnc(C(N)=O)cn1)=O)CC2 13433,C(=O)(CC(C1CC1)NC(=O)C=Cc1ccco1)N(C1CCOC1)CC 13434,N1(Cc2nnc(CC)s2)CCCOC(CNC(c2occ3c2CCC3)=O)C1 13435,CC1CCN(C(C23CC(C)(C2)C3)=O)CCN1C(=O)C(Cc1ccccc1)N(C)C 13436,C1(NC(c2c(COC)noc2)=O)CC(CO)N(C(=O)CSCc2ccncc2)C1 13437,Cc1cc(NC(C2(C)CC(O)CN2C)=O)ccc1NC(c1sccc1CO)=O 13438,C=CCCCCCC(=O)NCC(CCCC)NC(=O)CN1CCCCC1=O 13439,N1(c2n(CCC=C)c(C(n3cncn3)C)nn2)CCCC(n2ccnn2)CC1 13440,C1(CNC(C(C)(F)C(F)(F)F)=O)CCCC2CN(C(=O)C(Cl)=CCl)CC12 13441,C#CC1(C(=O)NCc2ccncn2)CCN(C(=O)C(=O)C2CCCC2)C1 13442,Cc1noc(C(C(C)C)NC(=O)CC2CCN(C(=O)C(C)CN(C)C)C2)n1 13443,c1(C(=O)NC(C2CCN(C(CNC(C(C)(C)C)=O)=O)C2)(C)C)c[nH]c(=N)nc1O 13444,C1(N(C(CCOCC#C)=O)C)CCN(C(=O)C=C(CCC)CCC)CC1C 13445,C(=O)(C(CCNC(=O)CCCCC1CC1)OC)N(C1CCN(C)C1)CCC 13446,C1(=O)C(C)NCC(C)NC(=O)C=CCN1C.C(=O)(C1CC1)OC.OC 13447,C1(CC(=O)OC)(CNC(=O)C(C2CCCC2)NC(c2coc(O)n2)=O)CCCC1 13448,c1(C2(C(=O)NCCOCCNC(CC(C)F)=O)CCC2)ccc([N+](=O)[O-])cc1 13449,NS(=O)(=O)CCCC(=O)NCCC1CCCCN1C(=O)CCN1CCCCC1 13450,N1(C(C(C)N(C)C(C2C3CCCCC23)=O)=O)CCC12CC(CO)C2 13451,C12C3CCC(C3)C1NC(=O)N2.N1(C(C2CC2)=O)CCN(CCF)CC1 13452,C(=O)(C1=CS(=O)CCC1)N1CCC(NC(CS(CC)=O)=O)(COC)C1 13453,c1(C(=O)NCC2(F)CCN(C(CN3C(C)CCC3)=O)C2)nc2ncccn2n1 13454,c1(CC(=O)O)nc2ccccc2o1.C12(CC1)C(=O)N(C1CC1)CC2.C1CC1 13455,C1(SC)CN(C(=O)CCc2cncs2)CC1NC(=O)CN1CCCCCC1 13456,C(C)(C)(CC(=O)NCC1(NC(=O)Cc2cncnc2O)CCCC1)SC 13457,c1(C(N(C(C)CN(C(=O)CCCCc2cnc[nH]2)C)C)=O)cnc2ncccn12 13458,c1(CCC(=O)N(C)CC2CCN(C(=O)CCSC(F)(F)F)C2)cccc(O)n1 13459,C#Cc1cc(F)c(C(N2CCC(C(C)NC(=O)Cc3ccoc3C)C2)=O)c(F)c1 13460,C#CCCCC(=O)NC1CCC(CNC(C2CCCOC2)=O)C1 13461,c1(C(N2CC(O)(CNC(c3cnn(C(F)F)c3)=O)C2)=O)ccc2cc[nH]c2c1Br 13462,c1(C(=O)NCCN(C(=O)CCC2CCCCC2)CC)nn(C)cc1SC 13463,C1(CN2CCN(C(C)=O)CC2)CCN(N2CCC(c3cccc(Cl)c3)C2)CC1 13464,CC(C(C(=O)NC1CCOC1)N(C1CCC1C)C)C(C)(C)C 13465,C1(F)(C(N2CC(OC)C(OC)C2)=O)CCN(C(c2ccc(O)nn2)=O)C1 13466,c1(N2CC3CC(NCCSc4cn(C)nc4)C3C2)nc(Cl)nc2ccccc12 13467,C=CCCCC(=O)NCCS(=O)(=O)Cc1cn(CCN2CCNC2=O)nn1 13468,c1(C(N(C)CC2CCN(C(C3CCC(F)(F)C3)=O)C2)=O)cc2ccncc2s1 13469,c1(CC(=O)NC2CN(C(C3(CCC=C)CC3)=O)CC2C)cc(C)ccc1OCC 13470,C(N=c1[nH]c(=NCC2(C)CS(=O)(=O)C2)c2[nH]ccc2[nH]1)c1c(C)cc(F)cc1 13471,C(=O)(C(F)(F)C1=CCOCC1)NCC#CCNC(=O)COCC1CCOC1 13472,C(=O)(CC(C(F)F)NC(C1(n2cccc2)CC1)=O)N1CC(O)(CCC)C1 13473,c1(N(C)C)cccc(NC(=O)Nc2ccccc2OCCCn2ccnc2)c1 13474,c1(C(N(C(C)CN(C)C(C2(CF)CC2)=O)C)=O)nccc(Br)c1O 13475,c1(C(N(CCCCN(C(=O)Cc2ccn(C)c2)C)C)=O)csc(C(C)(C)C)n1 13476,C1(CC)(OCCC(=O)NCCNC(C2CCN(C)C2)=O)CC(C)(C)C1 13477,C(C(CC(C)C)C(=O)NCC(C)CNC(c1nccn2cnnc12)=O)OC 13478,C1(C)(C(=O)NCC2CN(C(CS(=O)(=O)NCC)=O)CC2C)CCC2CC2C1 13479,N(C(=NCC1CCCO1)NC1CC(c2ccc(F)cc2)C1)CC1(C)CCC1 13480,c1(OC)ccc(C(=O)Nc2cccc(CNC(=O)C(F)(F)C(F)F)c2)c(C)n1 13481,CC(C)C(C#N)C(=O)N1CCC(NC(c2cnc(-c3cnccn3)s2)=O)C12CC2 13482,c1(C(=O)NC23CC(C(N(C4(C#C)CC4)C)=O)(C2)C3)cccc(O)c1 13483,CC#Cc1ccc(C(N2CCN(C3CC3)C(C#N)C2)C(=O)NC2CC2)cc1 13484,C(CC1=CCN(C(C2(C)CC2C(F)(F)F)=O)CC1)NC(CC(CCC)O)=O 13485,N1(C(c2cnc(C)c(Cl)c2)=O)CC2CC1CCN2C(C1CCCN1N=O)=O 13486,c1(C(N2CCC(N(C)C(c3ccccn3)=O)C2)=O)ccc(C(C)(F)F)nc1 13487,N1(C(CCN(C)CC)=O)CCC(C)N(C(=O)CCCCC(N)=O)CC1 13488,O=C(C1=CCCSC1)NCCCCCCNC(C1COCCC1c1ccccc1)=O 13489,C1(C(=O)NCCN(C(C)=O)CC)CCCCN1C(C1(C2CCC2)CC1)=O 13490,c1(C(N(C)CCOCCNC(C2CCC23CCC3)=O)=O)cc2cccnc2cn1 13491,C1(C(=O)NCc2nc(CC)[nH]n2)C=CCN(C(C2CCCC(=O)C2)=O)C1 13492,N1(C(C(C=C)C)=O)CCN2CCN(C(c3cc(Cl)c[nH]3)=O)CC2C1 13493,C(=O)(CC(C)(C)C(F)F)N1CC2C(C(=O)NCCCC(C)N(C)C)(C2)C1 13494,C1(CCNC(Cc2c(C)n[nH]c2C)=O)CN(C(c2nn(C)cc2Cl)=O)CC(C)O1 13495,C1(N(C)C(C2CC2(C)C)=O)CN(C(=O)Cc2ccc(Cl)cn2)CC1(C)C 13496,c1(C(=O)NC2CCN(C(CC=CCC)=O)C2C(C)(C)C)ncnc2c1CCC2 13497,c1(C(=O)NCC2N(C(C(C)(F)F)=O)CC(O)C2)ccc2nc(Br)nn2c1 13498,c1(C(C)NC(CS(CC)(=O)=O)=O)ccc2c(c1)CN(C(=O)C(C)C(F)F)C2 13499,N1(C(Cc2n(C)nnc2)=O)CCC=CC1C(N1CCOC(CC(N)=O)C1)=O 13500,N1(C(N(c2ccc(C)c(C)c2)C)=O)CCCc2ccc(Br)cc2C1 13501,CN1CC=C(C(=O)NCCC(c2ccccc2)N(C)C(C2CC3(CSC3)C2)=O)C1 13502,c1(C(N2CC(C(N)=O)(CNC(C(C)n3cncn3)=O)C2)=O)ccnc2[nH]ncc12 13503,c1(OC)ccc(-c2cncc(C(=O)N(C)CCN(C)C(C3CC3Cl)=O)c2)c(C)c1 13504,Cc1[nH]nc(Cl)c1C(=O)NCC1CC(NC(=O)CCc2cn(C)nn2)CCO1 13505,N1(C(C(CC)(C)OC)=O)CCOC2(CCCN(C(=O)C=CC3CCCC3)C2)C1 13506,c1(C(C)=O)ccc(C2CCN(C(N3CCCCC3C3CCOCC3)=O)CC2)cc1 13507,c1(C(=O)NCCCN(C(CCC=C)=O)C2CC2CC(C)C)ccc(N(C)C)cc1 13508,Cc1cc([N+](=O)[O-])ccc1C(=O)NC(C)C(C(C)C)NC(c1sc(C)cc1Cl)=O 13509,c1(C(=O)NC2CC(CNC(C3=CCCC3C)=O)C2)n[nH]c2c1CCSC2 13510,C1(C(=O)NCC2(C)CC(NC(CC3(OC)CC3)=O)C2)CC(c2ccccc2)=NO1 13511,c1(C(N2C(CNC(CN(CC)CC)=O)COCC2)=O)cc2ccccc2s1 13512,N1(C(C2CCSCC2)C(=O)NC(C(=O)OC)C)C2CCC1CC(CO)C2 13513,C1(NC(C(N2CCC(C)(CCO)C2)c2ccc(CF)cc2)=O)CCC(F)(F)CC1 13514,CC(C)(O)C(C)(C)C(=O)N1CCCC1CNC(C1OCC2CCCC12)=O 13515,C1(C)(OCC(=O)NCC2(CN(C(=O)CCCc3nncn3C)C)CC2)CCCC1 13516,C(=O)(CC(CC(C)C)NC(c1csc(C)c1)=O)NC(C#CCC)(C)C 13517,c1(C(=O)NCC(C)NC(CC(C)C(F)F)=O)cc2ccc(Br)cc2s1 13518,C(=O)(C#Cc1ccccc1)N1CC2C(C(=O)Nc3cc(OC)ncc3Br)C2C1 13519,C1(CNC(CCN(C(C2(C(C)C)CCCC2)=O)CC)=O)CC(C)CC(C)C1 13520,CC#CCC(C)NC(C1(CCNC(=O)CC(Cl)Cl)CC1)=O 13521,c1(C(=O)NC2CC(CNC(C3C(C)CC(=O)N3)=O)C2)cc(O)ccc1[N+](=O)[O-] 13522,c1(C(N2CC(NC(=O)C(F)C3CCC3)(CO)C2)=O)cncc([N+](=O)[O-])c1 13523,C1(C(F)(F)F)(C(N2CCC(C)(CNC(c3cncs3)=O)C2)=O)CC2CCC1CC2 13524,C1(C(=O)NC2CC(NC(C=CCC)=O)C2)C(F)(F)C12CCC2 13525,c1(C(=O)NC2CC3CC(NC(C(C)(C)N(C)C)=O)C2C3)ccc2nccnc2c1 13526,C(C1=CCCOC1)NC(C(c1cccs1)NC(c1cc(CO)on1)=O)=O 13527,N1(C(C=C(C)C)=O)C2CCC1C(CNC(=O)C(F)F)C2 13528,Cn1ccc(C(=O)NC(C2CCOC2)CNC(c2ccsc2)=O)c1C1CCC1 13529,C(C)(C)(CC(=O)N1CC(CCNC(=O)CNc2ccccn2)C1)SC 13530,c1(C(=O)NC2CC(F)(CNC(C(C)C3CCOC3)=O)C2)[nH]nc([N+](=O)[O-])c1Cl 13531,CC1C(NC(=O)CN2C(=O)CCC2=O)CCN1C(=O)Cc1ccccc1Cl 13532,N1(C(C(CC)OC)=O)CCSCC1C(=O)N(C1CCC1(C)C)C 13533,C#CC1(NC(C2CN(C(C3CCC3(OC)OC)=O)CCO2)=O)CC2CCCC12 13534,C12(CNC(C(C)=C3CCC3)=O)CC1CN(C(=O)Cc1cc(-c3ccco3)on1)C2 13535,C(=O)(C(CC(C)C)N(C)C)N(C(C(=O)NCc1c(C)c[nH]n1)C1CC1)C 13536,N1(C(c2c(CC)n[nH]c2)=O)CC2CC2(CNC(=O)C(O)CC2CC2)C1 13537,n1(CC(=O)OC)cc(S(=O)(=O)NCC(O)CC(C)(C)C)c(C)n1 13538,N1(C(Cc2c(C)nc[nH]2)=O)CC2CCCC1C2CNC(c1cn[nH]c1)=O 13539,N1(C(C(CC)O)=O)CCCC(N(C)C(c2ccnc(OC)c2)=O)C1 13540,CCCCCC(C)CC(=O)N(C1CC(NC(C2C=CCS2)=O)C1)C 13541,C(=O)(CC(C)(C)O)N1CC(C(C(N2CC(N(CC(C)C)C)C2)=O)O)C1 13542,Cc1cc(CNC(=O)C(CC2CCOCC2)NC(c2scnc2Cl)=O)n[nH]1 13543,C1(=O)C(CC(C)C)O1.C1(O)(C(C(=O)NCC)(F)F)CCCCC1 13544,C1(C(=O)NCC2N(C(C=CCCC)=O)CCN(C)C2)CCc2cnnn2C1 13545,C(=O)(CC(CC)C(C)C)N(CCCCC(=O)OCC)C(=S)NCC1CC(OCC)C1 13546,c1(C(N2CCC(O)(C(C)NC(c3cc(C(N)=O)no3)=O)C2)=O)ccc(Cl)nc1Cl 13547,C(=O)(CCC(=O)N1CCC(C(C)(O)CNC(=O)C(C)C2CCC2)CC1)NC 13548,C1(CCNC(C2CSCCS2)=O)CCCN(c2nc(C3CCCC3)ns2)C1 13549,C1(C)(C(=O)NCC(N2CCCCC2)C)CN(C(=O)C=CCN2CCC2)C(C)(C)C1 13550,C1(N)(C(=O)Nc2cc(COC)c(OC)cc2)CCC(C)(C)CC1 13551,CC1CCC(NC(c2nn[nH]c2Cl)=O)CN1C(=O)CCCCc1ccccc1 13552,c1(OC)ccc(C(=O)NCCC2CCCN(C(=O)CCC(C)N(C)C)C2)c(N)c1 13553,CN1CCN(C(=O)C(CC(F)F)NC(C2CC3CCCC3C2)=O)CC1=O 13554,N1(C(C(CC(=C)C)C)=O)C2CCC1CC(N(C)C(c1ccc(Br)s1)=O)C2 13555,Nc1ccc(C(=O)NCCC2(O)CCN(C(C3(CO)CCCO3)=O)CC2)cc1F 13556,c1(C(=O)NC2C(C(=O)NCC3CCC3)CCCC2)cc(Br)cc([N+](=O)[O-])c1Cl 13557,CCC(CC(=O)NC1(CNC(C2CCCSS2)=O)CCC1)c1ccccc1 13558,c1(C(N2CCC(NC(=O)C=Cc3cocn3)CC2)=O)ccc(Br)cc1[N+](=O)[O-] 13559,C1(C(=O)NC(C2CCN(C(Cc3c(C)nc(C)s3)=O)C2)C)CCCCC12CCC2 13560,C(=O)(C1CCCc2ncccc21)N(CCCNC(C1CC2(CC2)C1)=O)C 13561,c1(NC(C2CCN(Cc3cccc(-c4nn[nH]n4)c3)C2)=O)cc(Br)ccc1Br 13562,C1(NC(c2cc(Cl)cnn2)=O)C2CCC1N(C(=O)Cc1cccc(F)c1O)C2 13563,N1(C(CSCC=C)=O)CCN(C(c2cnn(C)c2C(F)F)=O)CC1CC(F)F 13564,N1(C(CC2(CSC)CC2)=O)CC(NC(=O)C(C)C(C)O)CC12CCCC2 13565,c1(C(C)(C)C)cccc(C(=O)NC2CCC(CNC(=O)CCc3cscn3)C2)n1 13566,C1(NC(C(CCC)C)=O)COC2(CCN(C(c3ccc(CC(C)C)cc3)=O)C2)C1 13567,N1(C(=O)OCC)CCC(c2ccccc2)S(=O)(=O)CC1.c12conc1C(=O)N2 13568,C1(NC(C(CC)(C)OC)=O)CCCCN(C(c2ccc(C)nc2N)=O)C1 13569,CONC(=O)C(=O)N1CC(F)CC1CN(C(=O)CSCC(N)=O)C 13570,N1(C(C2C(C(C)C)OCC2)=O)CC2CC(NC(=O)Cc3ccc(F)cc3)C1C2 13571,N1(C(c2cn(C)nc2)=O)CCC(CNC(c2ccc3n[nH]cc3n2)=O)C12CCC2 13572,N1(C(C(CO)N(C)C)=O)CCn2nc(C(=O)NCC(O)CO)cc2C1 13573,N1(C(C(CC=C)C)=O)CCC(CNC(=O)Cc2ncc(C)[nH]2)C(F)(F)C1 13574,CC(CF)CC(=O)NCC1CC1CNC(c1cc(-c2ccncc2)ccn1)=O 13575,N1(C(c2ncccc2F)=O)CCN(C(C2(C(F)F)CCOCC2)=O)CC1C(F)F 13576,c1(C(=O)OCC)cnn2c1C(C)N(C(c1sc3nnc(C)c(C)c3c1N)=O)CC2 13577,c1(C(N2CCC(N(C(C3C(C)(C)CC3)=O)CCO)C2)=O)cc[n+]([O-])cc1 13578,c1(C(=O)NCC2C=CCN2C(=O)CC2CCCOCC2)ccc(F)cc1Br 13579,C(N=c1[nH]cnc2ccc(O)cc12)C1C(NC(c2n(CC)ccn2)=O)CCCC1 13580,n1(C(C)C)ccc(C(=O)NC(C)(C)C(=O)NC(C2CCC2)C)n1 13581,CC12COCC1CN(C(N1CCCC1c1ccco1)=O)C2 13582,c1(CC(=O)NCC2N(C(CC(=O)NCC#C)=O)CCC2)cccc(C)c1Br 13583,N1(C(c2n(CC)ncc2Cl)=O)CCN(C(=O)CCc2ccoc2)C(C)CC1C 13584,C1(CC)CCCC(N=c2[nH]c(=NCCc3ocnc3CO)[nH]c3c2CCCC3)C1 13585,c1(C(=O)NC(CC)CN(C(=O)CSCc2cccnc2)C)cn(C)nc1C(C)C 13586,C1(OC)CN(Cc2ccc(C(=O)OC)cn2)CCC1O 13587,Cc1nn(C)c(Cl)c1C(=O)NC1CC1CNC(=O)C(n1ccc(C(F)(F)F)n1)C 13588,Cn1nc(CNC(C2CCCCC2)=O)cc1NCCC(O)C(F)F 13589,C1(N2CC(C(=O)NCC3C(NC(=O)COCCF)CC3)C2)CCCCC1 13590,N1(C(c2n(COC)ncc2)=O)CCC(C)C(CNC(c2nc(Cl)cs2)=O)C1 13591,N1(C(c2c(C)ccnn2)=O)CC2(CC(NC(C34CC3COC4(C)C)=O)C2)C1 13592,c1(C(N2CCC(N(C(c3nn(CC)cc3Cl)=O)CC)C2)=O)cc2n(n1)CCC2 13593,Cc1cccc(C(N2CC(O)(CNC(c3ncccc3N)=O)C2)=O)c1C 13594,c1(OC)[nH]c(=NC2CCCCCN(C(=O)C(=O)NC(C)C)C2)sc1C 13595,C1(CNC(C2N(CC)CCCC2)=O)CN(C(C23CC(C)(CO2)C3)=O)CC12CCC2 13596,N1(C(C2(CC#C)CCCO2)=O)CC2CCCN(C(=O)C(C(C)C)NC(=O)OC)C2C1 13597,CC(CCCC(=O)NCC1(CN(C)C)CC1)NC(c1ccnc(CO)c1)=O 13598,C1(C)(C(=O)NCC2CC(NC(C3CC(C(=O)OC)C3)=O)C2)CCCNS1(=O)=O 13599,c1(N(C(=O)OC(C)(C)C)C2CC2)cnn(C)c1.C1(=O)CCN(C)CC1=O 13600,c1(CC)[nH]ccc1C(=O)N(CC(=O)NCC1CC1Cl)C1CC1 13601,c1(CC(N2C(CNC(c3cc(I)on3)=O)CC2)=O)ccc(CO)cc1 13602,Cc1csc(=O)n1CCC(=O)NCCOCCN(C(=O)C=CC(N)=O)C 13603,C1(C(=O)NCC2OCCN(C(c3nc(CC)[nH]n3)C)C2)Cc2ccccc2O1 13604,N1(C(C2C3CCCC23)=O)CC2C(Cc3cn(CC(F)(F)F)nn3)C2C1 13605,C1(N(C(C2CSC2)=O)CC)CCCN(C(c2ccc(O)c(Cl)c2)=O)CC1 13606,c1(CC)ncc(C(=O)NC(CNC(C2CC3C=CC2O3)=O)CCOC)c(O)n1 13607,C1(C(N2CCCCC2)=O)CCCN(C(=O)CN(C2CC2C(F)(F)F)CC2CCC2)C1 13608,C1(OC(C)=O)CCCN(C(=O)NC(CO)C(C)OC(C)(C)C)C1 13609,Cc1cc(N(C)C2CC2)ccn1.C12CCN(CC1)C(=O)CCC1CC1CNC2 13610,C1(N(C(=O)C=CC2CCCO2)C)CCCN(C(C2CCOCC2)=O)CC1 13611,C1(OC)CCC12CC(C(=O)NC1CC(CNC(=O)C3=CCCSC3)C1)C2 13612,c1(C(N2CCC(C(C)C(=O)NCC(C)CC3CCC3)CC2)=O)ccc(C#N)cn1 13613,c1(C(=O)NCC2CC(NC(C3C(OCC)C3C)=O)C2)cnc2c(c1)nnn2C 13614,n1(CC(=O)NC2(C(=O)N)CC2)nc(C(=O)NCCOCCCC(C)C)cc1C.CC 13615,Cc1coc(C)c1CNC(=O)C(C)N(C(c1ccccc1)=O)C1CC1 13616,N1(CC(=O)N(CCNC(=O)C(F)=CC2CC2)CC)CC2CC2C1 13617,c1(OC)cnc(Br)cc1C(N1CCN(Cc2cnn(C)c2)CC1CC#N)=O 13618,C1(C(=O)NCC2CN(C(C=Cc3cc(C)[nH]c3)=O)C2)C2C(=O)OCC12Br 13619,c1(CC(=O)NC2CC(NC(=O)C(F)=CC3CC3)C2)noc2ccccc12 13620,Cc1cc(C(=O)NC2CCCC(NC(C3C4CCCOC34)=O)C2)cc2ccsc12 13621,C(c1ccccc1)=C(C)C(N1CC2CC2(C(=O)NC(C)(C)C(F)(F)F)C1)=O 13622,C1(CC(=O)NC2CN(C(c3cn(CCO)nn3)=O)C2)CC(=O)c2ccccc2C1 13623,C#Cc1ccc(NC(C2CC(F)(F)CN2c2nccc(C)n2)=O)cc1Cl 13624,C1(CC(C)O)CCN(C(=O)CCC2CCC(NC(=O)COC3CC3)C2)CC1 13625,CN1CCC(CCC(=O)NCCC2CCCN2C(c2cc(C3CC3)on2)=O)CC1 13626,N1(C(c2cn(CC)nn2)=O)CC2CC(NC(c3ccc(C)cc3C)=O)CC2C1 13627,C1(CN(CC(C)C)C(c2cn(CCOCC)nc2)=O)CCCC12CC2 13628,C1(NC(Cn2ncn(C)c2=O)=O)CCN(c2cc(C(F)F)ncn2)CC1O 13629,C(=O)(C(C)(CC)C(N)=O)N(CCCNC(=O)CCOc1cc(F)ccc1F)CC 13630,n1(CCC)cc(C(=O)N(CC(O)CCNC(=O)CSCC(N)=O)CC)c(C)n1 13631,C(=O)(CCC(C)(C)F)NC1C(C)CN(C(c2ccc(N3CCC(O)C3)cc2)=O)C1 13632,C=CC1CN(C(=O)C=CCC2(NC(=O)CNC(N)=O)CCC2)CCO1 13633,C1(C(=O)NC(c2ncc(C)o2)C)CCC2(CC2)N1C(c1nn(C)cc1C)=O 13634,N1(C(C(C)CC2CC2)=O)CCCC(C(=O)NC(C)(C)C(F)(F)F)CC1 13635,C1(C)(CC)NC(=O)N(CC(=O)NC2CCCN(c3snc(Cl)c3C#N)C2)C1=O 13636,c1(NC(=O)C(F)OC(F)(F)F)cn(CC(=O)NOCC2CCNCC2)nn1 13637,CCC(CC(C)C)C(=O)NC1CN(C(c2ccc(C#N)nc2O)=O)CC1(C)C 13638,CC1CCC(C(=O)NCc2nnnn2C)N1C(c1ccn(C)n1)=O 13639,N1(C(c2ncn(C)n2)=O)CC(NC(=O)CSC(C)(C)C)C(C)(C)C1 13640,C=CCCCC(C)NC(=O)C(C)CNC(=O)CN(C)C(=O)OC 13641,Cc1ncc(C(=O)NC2CN(C(c3c(C)noc3C3CC3)=O)CC2C)cc1C#N 13642,CCCC(C(=O)N1CC(N(C)C(C2(C3CCCO3)CCOCC2)=O)C1)OCC 13643,c1(C(=O)NCc2cccc3c2OCO3)c(F)ccc(CN2CCCCC2)c1F 13644,N1(C(C2(C(=O)NC)CC2)=O)CCCC(O)(CNC(=O)C(C)CN(C)C)CC1 13645,Cc1cc(NC(c2ccc(CNC(c3cnns3)=O)s2)=O)c(O)cc1F 13646,c1(CC)ccnc(CNC(=O)CC2CC(NC(c3cc(OC)ccn3)=O)C2)c1 13647,C12(CNC(C3(CO)CCC3)=O)CC1CN(C(=O)COC1CCC1)C2 13648,N1(C(CCC(C)C)=O)CCCC2C1CCCCN2C(=O)CCc1cccn1C 13649,C(=O)(C(F)C(F)(F)F)N(C1CC(NC(c2cc(N3CCCCC3)ncn2)=O)C1)C 13650,N1(S(=O)(=O)CCn2cncn2)CCCC2C1CCN2Cc1cc2ccncc2[nH]1 13651,C12(CNC(C=CC(C)(C)C)=O)CCC(CC1)CN2C(C1CC12CCC2)=O 13652,N1(C(CC(=O)OC)=O)CC(C(=O)Nc2c(CO)noc2C)CC12CCC2 13653,C1(CC)C(NC(=O)C(C)SC(F)(F)F)CCN1C(c1ccncc1SC1CC1)=O 13654,CC1=C(C(=O)N2CC(CNC(=O)CN3CCSCC3)CC(C)C2)CCCO1 13655,CCC(CC(=O)N1CC2CN(C(c3c[nH]c(=NC)o3)=O)CC2C1)C(C)C 13656,N1(C(=O)CC2CCC3CC3C2)CC23CCCC2(C1)CN(C(C1CCC=CO1)=O)C3 13657,C1(CNC(Cc2nccc(C)c2)=O)C(C)CCCN1C(c1ccc(C)cc1F)=O 13658,C(C(C)(C(C)C)C(C)C)NC(CC1C(C)CN(C(c2sccc2Cl)=O)C1)=O 13659,c1(C(=O)NC2CN(C(CCc3ccn(C)c3)=O)C3C2C3)ccc2cc[nH]c2n1 13660,c1(OC)cc(C(=O)NC2CCC(NC(=O)Cn3cc(Cl)cn3)CC2)ccc1[N+](=O)[O-] 13661,c1(C(N(CCNC(C(N)=O)=O)C2CC2)=O)cc2c(O)ncnc2cn1 13662,c1(CC)nccnc1C(N1CCCCC1CCN(C)C(C1(C)CCC(=O)N1)=O)=O 13663,C(C(C)(C)C(=O)N1CCC1CNC(C1(C)CCC(C)C1)=O)OC(C)C 13664,c1(C(N(C(CNC(C2CN(C(C)=O)C2)=O)C)C2CC2)=O)ccc(C)c(Br)c1 13665,Cc1ccc(C#N)cc1C(N1CC2CC1CCC2NC(=O)C(F)(F)C(F)F)=O 13666,C1(NC(CC2C(C)CCO2)=O)CCN(C(c2cccc(C(C)(F)F)c2)=O)C(C)C1 13667,Cc1conc1CC(=O)N(CC(=O)NCCCc1cccnc1)C1CC1 13668,N1(C(CC2CC(OC)C2)=O)CC(CC(N2CCCC(CO)C2)=O)CC1C 13669,c1(C(N(C(C)CCNC(C2SC3C=CC2CC3)=O)C)=O)cc2ccc(Cl)cc2s1 13670,c1(CC)cc(C(=O)NC2CCCCC2NC(=O)CC2C(C)(C)C2(C)C)cc(O)n1 13671,c1(C(C)=O)ccccc1OCCC(=O)NCC1CCCCN1C(=O)C(C)CCO 13672,c1(SC)cccc(C(=O)NCCN(C(c2cnc(S)[nH]2)=O)C2CC2)c1 13673,c1(C(CNC(=O)CCn2cccn2)NC(CNS(NC)(=O)=O)=O)ccccc1Cl 13674,Fc1ccc(F)c(NCC2CCCC(C(F)(F)F)C2)c1F 13675,C(=O)(C(C)(C)C(N)=O)NCCC1C(C)CN(C(=O)COCc2cccnc2)C1 13676,c1(NC(C2C(C(=O)OC)C2)=O)ccc(C(=O)Nc2cnc(O)cc2C)cc1C 13677,Cc1cc(C(=O)N(C2CCCN(C(C3CNC(=O)C3)=O)C2)C)cc([N+](=O)[O-])c1O 13678,c1(OC)ccc(CC(=O)NC2CC(C)(NC(=O)CCc3ccccn3)C2)cn1 13679,C(=O)(C1=CCCOCC1)NCC(C)(C(C)C)NC(c1c(C)oc(Br)c1)=O 13680,C1(CC(=O)NC(CNC(c2scc(C)c2)=O)CO)CCCN(C(C)C)C1 13681,C(=O)(C(C)(C)Cc1ccccc1)NCCCC(C)NC(=O)CSc1nccn1C 13682,n1(CC(C)NCCCC(C)(C)CO)cnc2c(cnn2C)c1=O 13683,N1(C(c2c(CC)c[nH]c2)=O)CCC2C(C(=O)NCC(C)(O)CSC)C2C1 13684,CN1C(=O)Cc2ccc(C(=O)NC3CC3CNC(=O)C=Cc3cccn3C)cc21 13685,CCCCCCCC(=O)N1CCC(NCc2cccc(C(C)C(=O)OC)c2)C1 13686,C(=O)(C(C)CCCC)N1CC(CC(=O)NCC=CC)OCC1 13687,CCCC(O)(CNC(c1cnn(-c2cccc(C)c2)n1)=O)CCC 13688,N1(C(Cc2c(C)non2)=O)CC(NC(=O)CCC2CCCC2)CCC1C 13689,C=CC(F)(F)C(=O)NCC(O)CC(=O)N(C)Cc1cc(C)nn1C 13690,c1(C(=O)NCC(C)NC(c2cnn(CC)c2Br)=O)ccc2[nH]c(=N)sc2c1 13691,C1(CNC(c2[nH]n(C)c(=O)n2)=O)COCCN(C(c2csc(C#N)c2)=O)C1 13692,c1(OC(COC2CN(C(COCCC=C)=O)C2)=O)ccc(OC)cc1Br 13693,C1(CC(=O)N(C2CC2)CC2N(C(C(C)Cn3ccnc3)=O)CCC2)CC2(CCC2)C1 13694,N1(C(C2C(CNC(c3c(Cl)cn(C)n3)=O)CCO2)=O)CCOCC(C)(F)C1 13695,Cc1nc(-c2nn[nH]n2)c(NC2CCCN(C(=O)C(=O)NC3CC3)C2)o1 13696,C1(CC#C)(C(=O)NCC(c2cccc(Br)c2)C)CCCNC1 13697,N1(C(C(C)C2CC2)=O)CC(C(=O)NCc2ccnc(F)c2F)C2(CCC2)C1 13698,N1(C(c2ccc(C)o2)=O)CCc2nc(CNC(=O)C(C)(C)c3cnc[nH]3)sc2C1 13699,c1(C(=O)NCC2(C(=O)NC(CC)C(=O)N(C)C)CC(=C)C2)cnc(C)n1C 13700,Cc1cc(C)c(C(N2CCN(C(c3ccns3)=O)CC2C(C)C)=O)cc1N 13701,Cc1cc(CC(=O)NC(CNC(=O)Cc2[nH]cnc2C)C(C)(C)C)n(C)n1 13702,C1(C2CCCC2)(C(=O)NCC(CNC(c2c(OC)cc(C)s2)=O)F)CCNC1=O 13703,C1(CNC(C(C=C)C)=O)CN(C(=O)Cc2cc(C)cs2)CC12CC2 13704,O=C1CCC(S(=O)(=O)NCC2CCCC2OC(=O)C2=COCCC2)CC1 13705,Cc1ncnc(O)c1C(=O)NC1CC(C)(NC(=O)CCc2cc(F)cc(F)c2)C1 13706,C1(CC)CC(C(N2CCCC2(CNC(C2CCOCC2)=O)COC)=O)CC(=O)N1 13707,Cc1cc(C(=O)NCC2(O)CCCN(C(c3cc(C(F)F)cs3)=O)C2)cnc1O 13708,C12(CNC(CC3C(CC)C3)=O)CC(NC(c3scnc3Br)=O)(C1)C2 13709,C(c1cccc([N+](=O)[O-])c1)=CC(=O)NC1(C)CCN(C(C2(O)CCOC2)=O)C1 13710,c1(CC(C(=O)NC2CC(Cn3cc(C(C(=O)OC)(C)C)nn3)C2)O)cccc(Cl)c1 13711,c1(OC)sccc1C(=O)NOC(C)C(=O)NC(C)C(CO)OC 13712,C1(CC(=O)NCCc2cc(C(N(C)Cc3c(C)cco3)=O)no2)CC(O)C1(C)C 13713,N1(C(CCCc2onc(C(C)C)n2)=O)CCN(C(C2CCC(O)C2)=O)C(C)C1 13714,C1(CNC(C2(C#C)CCCC2)=O)CN(C)CCN1C(c1cc(CF)on1)=O 13715,C(C(CC(=O)N(C1CCCCN(C(=O)Cn2nccn2)C1)C)C(F)(F)F)N(C)C 13716,Cc1cc(Cl)cnc1S(=O)(=O)N1CCSC(c2cnn(C(C)C)c2)C1 13717,c1(N2CCC(N(C)C(C3CCC(C)CC3)=O)C2)ccnc(C(F)(F)F)n1 13718,CCC(CC(=O)NCC1(NC(c2cc(=N)[nH]c(Cl)n2)=O)CC(F)(F)C1)CC(C)C 13719,N1(C(C(CC)C#N)=O)CC(CC(=O)N(CCCO)CCO)C2(CC2)C1 13720,Cc1cc(C(N2CCC(CCNC(C3(C)CC3Br)=O)CC2)=O)nc(O)c1 13721,N1(C(c2ncc(C)s2)C(=O)NCCCSC)CCC(C(C)(F)F)CC1 13722,N1(C(CCN(C(C)C)C(C2CCCCC2(C)C)=O)=O)CC2OCC(N(C)C)C2C1 13723,N12CCC(CNC(C3(CF)CCC3)=O)(C1)CC2=O.c1(C2CCCO2)ncccn1 13724,O=C(CCCNC(C1(CNC(=O)Cn2cccn2)CC2(CC2)C1)=O)NO 13725,c1(CC(N2CC(CCC)N(C(=O)C(O)C(C)C)CC2)=O)coc2cc(O)ccc12 13726,c1(C(N(C)CC2CCN(C(CSCC)=O)C2)=O)cc(C(F)(F)F)cc(Cl)c1 13727,C1(CC(=O)NC2CNC3CC2C3)CC2OCCC2O1 13728,Cc1cc(=NC(C(C)NC(=O)Cc2ccc3ncsc3c2)C(C)C)[nH]c(Cl)n1 13729,CC1(C(N2CCC3(CCC3)C2)=O)CCN(Cc2cnc(Br)c(F)c2)CC1 13730,C(C(C(C)C(C)C)NC(=O)Cc1cc(C)[nH]n1)NC(CCc1cccc(C)c1)=O 13731,CN1CC(C(=O)NCCN(C(=O)CCN2CCCC2=O)C)C(C(F)(F)F)C1 13732,C1(C(N2CC(C=C)(CC(=O)NC(C#C)(CC)CC)C2)=O)CCC(C#N)CC1 13733,CC(F)(F)C(F)C(=O)N1CCC(N(C(C2CCCCC2)=O)CC2CC2)C1 13734,C1(CNC(CCCOCCC)=O)CC2CCC1N2C(=O)C(N)=O 13735,CN1CCn2cc(C(N3CCCC4(C3)CN(C(C3(C)CCC3)=O)C4)=O)nc2C1=O 13736,C(=O)(C(C)S(=O)(=O)C(C)C)NC(CCCNC(c1c(C)onc1Br)=O)C 13737,N1(C(c2c(CC)c(C(N)=O)c(C)[nH]2)=O)CC2CC(NC(C34CC3C4)=O)CC2C1 13738,CC1CC(NC(=O)Cc2sc(O)nc2O)CN(C(=O)C(C2CCOCC2)O)C1 13739,C1(NC(=O)Nc2cc(COC)ncn2)C2Cc3cc(F)ccc3C12 13740,N1(C(C2(CC(=O)OC)CC2)=O)CCCCC(N(C)C(C2OCCC2(C)C)=O)C1.C1(C)CC1 13741,CCCCCCCCOCC(N1CCCC1CN(C(C1CCC(C)C1)=O)CC)=O 13742,C1(NC(c2c(OC)ccs2)=O)CC2CCC1CN(C(=O)CNC(C1CC1C)=O)C2 13743,c1(C(=O)Nc2c(OC(C)C)ccc(C#N)c2)ccc2c(c1)NCCC(=O)N2 13744,C1(C(=O)NC(c2ncc(-c3ccc(Br)cc3)o2)C)(C(C)C)CNC(=O)C1 13745,C(=O)(CCCCOC)NC(C1CCCC1)CNC(c1c(NC)scc1)=O 13746,C1(NC(c2ncc[nH]c2=O)=O)CC12CCN(C(c1ccc3ncccn13)=O)CC2 13747,c1(CNC(=O)C(=O)NCC(C)C)ccnc(Oc2ccccc2)c1 13748,C(=O)(C(CO)NC(=O)CC1CCOC1C)NC(C=C)(C)C 13749,c1(C(=O)Nc2c(F)ccc(NC(CC)=O)c2)c2c(nn1C)CCNC2 13750,c1(C(N(CC#N)CC#N)=O)ccnc2ccc(O)cc12.C12CC1C(=O)N2 13751,c1(C(=O)NC(C(C)NC(c2cnc(Cl)s2)=O)C)ccc2c(c1)NS(=O)(=O)C2 13752,C(=O)(C#CC1CCCCO1)NCC(c1ccccc1)CNC(C1(CC=C)CC1)=O 13753,C1(CNC(=O)Cc2cc[nH]c2)(NC(C2CC2c2ccccc2)=O)CCOC1 13754,c1(CNC(N2C(N3CCCC3)(CC)CCC2)=O)sccc1S(C)(=O)=O 13755,c1(C(=O)NC2CCN(Cc3ccc(C)[nH]3)CC2F)n[nH]c2c1CS(=O)(=O)C2 13756,N1(C(C(C)C(C)O)=O)CCCC2(CC(NC(=O)COC(F)F)C2)C1 13757,c1(NC(C2C3CN(C(c4ncccn4)=O)CC23)=O)cc(F)ccc1I 13758,c1(N2CCCC(OC)C2)ccc(Br)c(S(=O)(=O)NCC2(Br)CC2(F)F)n1 13759,C(=O)(C#CC1(C)CCCO1)N(CCN(C(C1CC(C)(CC(F)(F)F)C1)=O)CC)CC 13760,C1(NC(C(C)OC)=O)CCCN(C(C2CCC(C)C2)=O)C1C 13761,C1(C(=O)NCC2(C(=O)NC(CC(=O)NCC)C)CC23CCC3)CC2CCCC2C1 13762,C=CCCCCC(=O)NCC(CC1CC1)C(=O)NC(c1cn(C)nc1C)C 13763,Cn1nc(C(=O)NC(CNC(=O)C(F)C2CCC2)C(C)(C)C)cc1C(F)F 13764,CCCCCC(C(=O)N1CC2CC(Nc3nc4cc(Br)cnc4s3)C2C1)C(C)C 13765,N1(CC2C(n3cc(-c4c(C)cccc4Cl)nn3)CCC2)CCOCC12CCOC2 13766,C12(C(N3C(C)(CNC(CC=C)=O)CCC3)=O)CCC(C)(CC1)OC2(C)C 13767,C(=O)(CC1NC(=O)c2ccccc21)NC1C(C)CN(C(C2CCC(F)CC2)=O)C1 13768,c1(N(CC(CN(C(c2cc(C)n(C(C)(C)C)n2)=O)C)O)C)ncnc2c1SCCC2 13769,C1(NC(=O)NCC2CN(S(CC)(=O)=O)C2)CCCN(CCOC(C)C)C1 13770,c1(C(C)C(=O)NCC(C)N(C)C(c2cc(-c3ccco3)no2)=O)cccc(Cl)c1 13771,N1(C(CC(CC)(C)C)=O)CCC(NC(c2ccc(Cl)nc2C)=O)C12CCC2 13772,C1(NC(C(C)OC2CCOC2)=O)CCCC(NC(c2c(Cl)cnn2C)=O)C1 13773,C1(C2CCCN(C(=O)CN3CCCCCC3=O)C2)(NC(C(C)CC#N)=O)CC1 13774,C1(C(N(CC(CCC)O)C)=O)CCCN1NC(=O)c1c[nH]c2cccnc12 13775,C1(CCOC)CCN(N2CC3(CCOCC(=O)N3)C2)CC1 13776,Cc1cc(C(N2CCC(O)C(NC(c3ccc(C)n3C)=O)C2)=O)c(S(N)(=O)=O)s1 13777,N1(C(C2CCC(CC#C)CC2)=O)CC(C#C)(C(N2CC(O)(CC(C)C)C2)=O)C1 13778,C1(CNC(c2cc(C)sc2C)=O)(NC(c2cc(O)nn2C)=O)CCCCC1C 13779,c1(N2CCCC(CN(C)C)C2)nc2ccccc2nc1NCC1CCC1(F)F 13780,c1(NC(C=Cc2c(Nc3cc(OC)cc(F)c3)cccc2)=O)ncc2cn[nH]c2n1 13781,c1(N2CCCC(=C)C2)nc(=NCCC2CCCN2C)[nH]c2c1CC(C)CC2 13782,C=C=CCC(=O)NC(C(=O)NCc1cnn(CC)c1)C1(C)CC1 13783,c1(OC)cc(NCc2ncccc2Cl)ncn1 13784,C1(CN(C2CCN(CC3CC3)C2)C(=O)CC2CC3CC3C2)CCCNC1=O 13785,Cc1c(Cl)ccnc1C(=O)NC1CCC(F)(CNC(=O)C=C2CCC2)C1 13786,c1(C(=O)NC2C(C)CN(C(=O)CC3CCOCC3)CC2)c(F)ccc2occc12 13787,N12C(=O)NC(C1=O)Cc1ccc(o1)C2.C1(OC)CCCC(C)C1 13788,N1(C(CC2(C)CCC2)=O)C2CCC1C(CNC(C1(c3ccccc3)CC1)=O)C2 13789,C1(C(=O)NCCC2CCN(C(C(C)(C)n3ccnn3)=O)C2)CCc2nccn2C1 13790,N1(C(c2ccc(NS(C)(=O)=O)cc2)=O)CC2CC1CCN2C(=O)CCS(C)=O 13791,C(N=c1nc2sccc2c(NCC2C=CCC2)[nH]1)C1(OCC)CCCSC1 13792,Cc1noc2nc(C(N3CC(NC(=O)Cc4nnc(O)s4)CCC3C)=O)ccc12 13793,C=Cc1cc(C(N2CCC(NC(=O)CCSCCCC)C2CC)=O)cc(F)c1 13794,c1(NC)ccc(C(=O)NC(CC2CCC2)C(N2CCC(C(C)O)CC2)=O)cc1 13795,c1(CC(=O)NCC(CN(C)C(C2CCCCC2O)=O)(C)C)cccc(C2CC2)c1 13796,C#CCC(CC(=O)Nn1cnn(C)c1=S)NC(c1cnc(O)o1)=O 13797,c1(NC(CC2N(C(C(CC)OCC)=O)CCC2)=O)ccc2nonc2c1 13798,C1(CCNC(C=C(C)C(F)F)=O)(NC(=O)OC(C)(C)C)CC1(C)C 13799,C1(NC(CCC=CC(C)C)=O)CCCC(N(C)C(c2csc(C(N)=O)n2)=O)C1 13800,c1(NC(=O)NCC(CNC(=O)Cc2nnc(O)s2)OC)ccccc1C 13801,c1(CNC(=O)C(N2CCC3CC23)=O)ccc(I)cc1 13802,Cn1c(C(=O)NC2CCCC(NC(c3ccc(N)c(O)c3)=O)C2)cc2sccc12 13803,C1(CC(=O)NC(C(=O)NC(CC)C2CCC2)Cc2cc[nH]n2)CCCC12CC2 13804,C1(NC(C2(C)CC(=C)C2)=O)CCCC(NC(c2cccc(C(=O)NC)n2)=O)CC1 13805,CC1(CNC(C2CCC(=O)N2)=O)CCN(C(C2CCCN2N=O)=O)C1 13806,C1(C)(NC(CCSCC)=O)CCN(C(C2CCCC2(C)C)=O)CC1 13807,CC1CN(C(=O)Cc2cnns2)CCC1CNC(=O)C(C)SCc1ccccc1 13808,c1(C(C)CNC(C2CCCCC2)C(=O)OCC)ccc(Br)cc1.C(C)(C)(C)O 13809,N1(C(CCOC)=O)CCC(C(C)(C)NC(=O)C(c2cnn(C(C)(C)C)c2)=O)C1 13810,C1(CNC(COCc2n(C)ccn2)=O)CN(C(=O)CC2(O)CCC2)CCC1(C)C 13811,Cc1nnc2n1CC(C(=O)NC1CC(CNC(c3ccncc3Cl)=O)C1)CC2 13812,C(CCSC)(C(=O)NCC1(C(=O)OC)CN(C(c2scc(C)c2C)=O)C1)OC 13813,CCC(C)C(C(=O)NC(C)CCNC(=O)C=Cc1cncc(C)c1)NC(=O)OC 13814,CC1CCC(F)(C(N2CC(OCCC(=O)NCCCCCCC3CC3)C2)=O)CC1 13815,c1(-c2nc(C3C(CCC)CCC3)n(CC(F)F)n2)cc(F)c(N)c(F)c1 13816,C(=O)(C(CO)C(C)C)NC(CCCC)CNC(=O)CN(C)C(=O)C1CC1 13817,C(=O)(CCCCc1cnn[nH]1)NCCCC1N(C(C(C)n2ccnn2)=O)CCC1 13818,C(C(CN=c1[nH]c(N(C)CC2CCCOC2)nc2c1CCCCC2)OC)OC 13819,CC1C2CC(C2NC(c2cc[nH]n2)=O)N1C(c1nc[nH]c1C(C)(C)C)=O 13820,N1(C(c2cnn(C)n2)=O)CCC2C(NC(C34CCCC3(C(N)=O)C4)=O)CC12 13821,N1(C(Cc2ccn(C)n2)=O)CC2CC(C(=O)Nc3ccccc3C(C)(F)F)C1C2 13822,N(C1CCCn2ncnc21)C(C(C)NC(C1CN(C2COC2)C1)=O)=O 13823,N1(C(c2cc(I)ccc2F)C(=O)NC)CCCC2CC(C)CCC12 13824,C(CC1=CCN(C(c2nc3cnccc3s2)=O)CC1)NC(CCN(C)CC)=O 13825,Cc1nc(NCc2ccc3sccc3c2)cc(=NCc2nccn2C2CC2)[nH]1 13826,C1(C(=O)NC2CCCC2CNC(=O)COC(F)F)CCCN1c1ncccn1 13827,c1(NC2CC(NC(C3CCCCCC3)=O)C2)nc2ccc([N+](=O)[O-])cc2[nH]1 13828,N1(C(c2occ(C)c2)=O)CCCC(C2(NC(=O)C(O)Cc3[nH]cnc3C)CC2)C1 13829,n1(CC)ncc(C(=O)NC2CN(C(C3CC3(F)F)=O)CC2F)c1C 13830,C1(CCNC(C2(C(=O)OCC)CC2)=O)CCN(C(=O)Cn2cccn2)C(C)C1 13831,CC(O)C(C)(C)C(=O)NCC(C)(C(C)C)NC(c1cc(C2CC2)cc(F)c1)=O 13832,c1(CCCNCC(C)SC)[nH]nnc1C 13833,C(C)(CCC(=O)NC(CNC(=O)CS)(CC)CC)OCC.C1CN1CC 13834,c1(C(=O)NC2CC(C(N3CC4CCC3CC4)=O)C2)cc(I)c(O)c(I)c1 13835,N1(C(C2(COC)COC2)=O)CCC(C)(NC(=O)CCc2cccc(N(C)C)c2)C1 13836,N1(C(COCc2ccc(OC)nc2)=O)CCC(NC(=O)CCC(C)O)C1(C)C 13837,CCC(O)CC(=O)N(CC(=O)NC(c1cnc(C)s1)C)C1CCC1 13838,C(=O)(CCCCC(=O)N1CC(C(C)NC(C2CN(C)CCN(C)C2)=O)C1)NC 13839,Cc1cccc2cc(C(N3CC(N(C(=O)CCF)C)C3)=O)oc12 13840,C(C(O)CC(F)(F)F)NC(C(CCNC(=O)CSC(C)(C)C)OC)=O 13841,Cc1[nH]c2ccc(Cl)cc2c1C(=O)NC1CC1NC(=O)C(C(C)(C)C)N(C)C 13842,C1(CNC(c2c(C)cc(C)nc2)=O)CC(C(C)(C)C)=NO1 13843,N1(CCC)CCCCC1C(=O)NCCC(C(C)C)NC(=O)Cc1cc(C)[nH]n1 13844,C1(C)(C(=O)NCC(CNC(c2c(C)cc(CC)o2)=O)(C)C)CCC(C)=C(C)C1 13845,c1(C(=O)NC(CNC(c2cc(SCC)ncc2)=O)CC)ncnc2ccsc12 13846,c1(OC)cc(C(=O)Nc2cccc(CN(C)C)c2)cnc1-c1sccc1CO 13847,c1(C(=O)NCC(CO)NC(c2ccn(C)c2)=O)cccc(S(C)(=O)=O)c1 13848,C1(C(=O)NCC2=CCCN(C(=O)Cc3ccccc3)C2)(CC)CCC(F)(F)CC1 13849,CC1CCN(C(=O)CSC2CC2)CCN1C(C12CC(CO)(C1)OC2(C)C)=O 13850,CC12CC(C(N3CCC(NC(c4cc(C(F)(F)F)c(Cl)cn4)=O)C3)=O)(CCO1)C2 13851,N1(C(CS(CC)=O)=O)CCC2(CCCC2NC(=O)CCSc2n[nH]c(C)n2)CC1 13852,c1(C(N2CCC(c3c[nH]cc3C(F)(F)F)C2)=O)cc(Cl)nc(C2CCCO2)n1 13853,N1(C(COCC(=C)C)=O)CCC(CNC(C2CCS(=O)(=O)C2)=O)C12CC2 13854,N1(C(COC(C)=O)=O)CCC(C2(CNC(C3CC3F)=O)CCOCC2)CC1 13855,c1(CC)nc(C)c(CC(=O)NC2CC3(C2)CC(NC(C2CC2F)=O)C3)c(C)n1 13856,N1(C(C=C(COC)C)=O)CC(NC(=O)C(F)CC2CCCC2)C(C)(C)C1 13857,N1(C(c2cc(C)sn2)=O)CCC(O)(CCNC(C2(CO)CCOC2)=O)C1 13858,N(C(=NCCCOC)Nc1ccc(OC(F)F)cc1C)CC1(SC)CCC1 13859,C1(C(N2CC(C)C(NC(c3cncc(N)n3)=O)C2)=O)CCC2CC(C)CN2C1 13860,c1(CC(=O)NCCN(C(=O)CC2CCNC2=O)C)cc(Cl)sc1Cl 13861,N1(C(CC2CC(CC)C2)=O)CCCC(CCNC(C2CC(OC)C2)=O)CC1 13862,C(=O)(C(C)CS(C)(=O)=O)N(CCNC(C(C1CCC(C)CC1)CC)=O)CC 13863,C1(NC(N2CC3C(CC#N)CC(C3)C2)=O)CCCC12CCOCC2 13864,C#Cc1cc(NC(C2CC(=O)C2C2CCC2)=O)ccc1C 13865,N1(C(C)=O)CCC(C)(C(=O)N(C)CC2CCCCN2C(c2cncn2C)=O)C1 13866,C1(NC(c2cc(CCOCC)on2)=O)CC(F)CN(C(=O)COCCOC)C1 13867,CCCCC(C(=O)NCC1CCC1NC(=O)C(C)(C)c1ccsc1)C(C)C 13868,N1(CCC(C)NC(=O)C=CC(F)F)CCCC(C)C1 13869,N1(CC(N2C(C(C)(C)CNC(c3cnsc3)=O)CCC2)=O)CCP(C)(=O)CC1 13870,c1(C(=O)NC2CC(C)N(C(C3C(C)(C)OC3(C)C)=O)C2)ncsc1S(N)(=O)=O 13871,N1(C(C23CCCC2C3)=O)CCC(c2ncc(C(F)(F)F)[nH]2)C1 13872,C1(C2(O)CCN(C)CC2)(C(=O)NC(CCCNC(CC=C)=O)(C)C)CC1 13873,C(C)(C)(C(O)C(F)F)NC(CC1(NC(Cc2c(C)nn(C)c2)=O)CC1)=O 13874,Cc1nc2[nH]c(C(=O)NCCCCN(C)C(C3(C)CC4CC4C3)=O)cc2s1 13875,c1(C(=O)NCCN2CCCN(C(C3CCSC3)=O)CC2)noc2c1CC(F)(F)CC2 13876,C12(CNC(C3C(CC)CCC3)=O)CCC(CNC(c3cc[nH]n3)=O)(CC1)CO2 13877,Cc1cc(C(N2CCN(C(=O)C(c3cnn(C)c3)C)C(C(C)C)C2)=O)cc(O)n1 13878,N1(C(=O)COC(CF)C(F)(F)F)CCC(F)(c2cn(C3CC4CCC3O4)nn2)C1 13879,c1(CC)noc(CN(CCNC(=O)CCc2nc(C)no2)C2CC2)n1 13880,c1(-c2nc(C3C(C)(C)C3)nn2CCN(C)C)cncc2c(Cl)cccc12 13881,c1(C(N2CCCC(C(C)NC(C(C)=C3CC3)=O)C2)=O)cc2cc(C)c(C)cc2o1 13882,N#CC12CCC(C(=O)Nc3ncn4ccccc34)(CC1)CC2 13883,c1(-n2ccc(C)n2)cccc(C(=O)NCCC2(O)CCOC2)c1 13884,C1(C(N(CCC(C)O)C)=O)CN(C(c2cccc(O)c2F)=O)C(C)(C)C1 13885,N1(C(c2nncc(C)c2)=O)CCC(C)C(NC(c2cc(C)sc2C)=O)C1 13886,CC1C(C(=O)N(C)CC2CCCC2)CCN1C(=O)Cc1ccnn1C 13887,N1(C(C2CSC2)=O)CCCC2C(CCCN2C(c2cccc3[nH]ccc23)=O)C1 13888,Cc1nn(C)c(C)c1C(=O)NCC(CC(C)C)NC(c1cccc(Cl)c1F)=O 13889,c1(CC(=O)NC2CCC(C)(CNC(C3(COC)CC3)=O)C2)c(Cl)ccc(O)c1Cl 13890,N1(C(c2n(C(CC)C)ncc2)=O)CC(NC(c2cnc(O)c(F)c2)=O)C2(CC2)C1 13891,N1(C(C(C)N(CC)CC)=O)CCC(C=CC(N2CCC(C)C2C)=O)CC1 13892,c1(OC)cc(C(=O)N(C(CNC(=O)C(C)=C(C)C)C2CC2)C)[nH]n1 13893,c1(C(N2CC3C(NC(CN(C4CC4)CC)=O)(C3)C2)=O)cc2cn[nH]c2cn1 13894,C(=O)(CC1=NN(C)C(=O)C1)N(CC(CC)OC)C.C1(=O)C(O)CN1 13895,C(=O)(CC(F)(F)C(C)C)NC1CCC(C)(NC(C(CCCOC)C)=O)CC1 13896,N1(C(c2cnc3[nH]nnc3c2)=O)CC(C2CCCN(C(C3CCOC3)=O)C2)C1 13897,Cc1noc2nc(C(=O)NCCCCNC(=O)CCCNC(N)=O)ccc12 13898,C(=O)(C(F)CCC(C)C)NCC1C(NC(C(CC)(F)F)=O)CCCC1 13899,c1(C(=O)NCC(C)N(C(=O)CC(C)CF)CC)ccc(CO)c(F)c1 13900,c1(C(=O)NCCN(C(C(C(C)(C)C)SC)=O)C2CC2)ccc2c(c1)OCCC2 13901,N1(C(C(CCCC)(F)F)=O)CC2CN(C(c3cccc[n+]3[O-])=O)CC(C1)O2 13902,C1(NC(C(C#C)(C)C)=O)CN(C(C2CC3(CC3)CO2)=O)CC1C=C 13903,C1(C(=O)NCC2C(NC(CN3CCN(CC)CC3)=O)C2)CC2(CCCC2)CO1 13904,c1(C(C)(C)C)ccc(S(=O)(=O)N2CC3CC2CC3N2CCC(Cl)C2)cc1 13905,C1(C(=O)NC2C(CNC(CC(C)(C)OC)=O)CCCC2)CCC2(CC1)CC2(F)F 13906,C(=O)(NNC(=O)C(C)(C)CCCCNC(=O)C(C)=CC)C1(CC=C)CCOCC1 13907,C(CC1=CCCCC1)NC(c1c(CNC(C2(Cl)C(C(C)=O)C2)=O)ccs1)=O 13908,c1(C(N2CCN(C(C3CCSCC3)=O)C3CC23)=O)cc(Cl)c(F)cc1Cl 13909,C1(N(C(c2c(C)nn(CCO)c2)=O)C)CCN(C(C2(C)SCCCS2)=O)CC1C 13910,C1(C)(CC(N2CCC(C(C)NC(c3cc(Cl)c[nH]3)=O)C2)=O)Oc2ccccc2O1 13911,CC1CCc2[nH]c3ccc(C(N4CCN(C(=O)CCN(C)C)CC4)=O)cc3c2C1 13912,Cc1cc2ncn(CC(=O)NC(C)(C)C(C)NC(C3CC3C3CC3)=O)c2cc1C 13913,c1(C(=O)NC2C(NC(CCc3cc(C)on3)=O)CC2)cn(C)nc1C(F)(F)F 13914,C1(C)(NC(c2c(CC)nccn2)=O)CCN(C(c2nccc(N)c2Cl)=O)CC1 13915,C1(C)(C(=O)NCC2(CN(C(=O)COC3CC=CC3)C)CC2)CCC(=O)NC1 13916,N1(C(c2c(=N)[nH]cnc2)=O)CC2CCN(C(=O)CSCC(N)=O)CC12 13917,N1(C(c2ccc(C(C)=O)o2)=O)CC=CC(C(=O)N(CC(C)C(C)C)C)C1 13918,N1(C(C2N(C(C)=O)CCC2)=O)CCC(C)C(CNC(=O)C(c2cscn2)N(C)C)C1 13919,C(=O)(CC1=NN(C)C(=O)C1)N1CCC(C(=O)NC(CC#C)(C)C)C1C(C)C 13920,c1(OC)cc(O)c(CN2CC3(CC(CC(=O)NCCCC(=O)OC)C3)C2)cc1Cl 13921,c1(C(N2CC(C)(CNC(C3CC=CC3)=O)OCC2)=O)ccc(S(N)(=O)=O)cc1 13922,c1(COC)cnc(OC)c(C(=O)NCC#CCNC(c2coc(Cl)n2)=O)c1 13923,C1(c2n(CC=C)nnn2)(NCC(C)Sc2ccccc2)CC(C)SC(C)C1 13924,C1(CNC(C2CC(SC)C2)=O)C=CCN1C(c1ncn(C)n1)=O 13925,N1(C(C23N(C(c4c(OC)ccs4)=O)CC(CO)(C2)C3)=O)CCCC12CCOC2 13926,c1(-n2cc(CN3C(CCCO)CCC3)nn2)cc(Br)ncc1Br 13927,N(C(=NCC(C)OC)NCC1CCCCC1)Cc1ccc(CC)cc1 13928,c1(CCC(=O)NCC2C3CN(C(=O)CC4CCCO4)CC23)cc(Cl)ccc1Br 13929,CC1(C)CC(CC(=O)NCC(C)(CO)NC(c2cccnn2)=O)C1 13930,c1(C(=O)OC)cc(F)cc2c1CCN(C(C1CCC(C(=O)N(C)C)O1)=O)C2 13931,C1(OC)CCN(CC(=O)NC2CCC(N(C)C(C3CC3(F)F)=O)C2)C1 13932,Cc1cnc(C=CC(=O)NCCC2COCCN2C(=O)Cc2cc(Cl)cs2)[nH]1 13933,N1(C(C=CC(=O)NC2CC2)=O)CCCCCC(NC(C2(C3CCC3)CC2)=O)C1 13934,C#CCCCC(C)C(=O)N(CCN(C(=O)CCc1cocn1)CC)CC 13935,C(c1ccccn1)=C(C(=O)N(CCOC)CCNC(C1CCOC1C)=O)C 13936,Cc1cc(C(=O)NCCC2C(C)CCCN2C(=O)C(F)=CC2CC2)cc(F)c1C 13937,O=C1CC2C(C(=O)NCc3csc(CNC(=O)Cn4nccn4)n3)C2C1 13938,C(=O)(C(C)C(C)(C)C)NC(C(C)C)CN(C(=O)CC1CS(=O)(=O)C1)C(C)C 13939,N1(C(c2snnc2C)C(=O)NCC2(C(=O)OCC)CC2)CC2(CC2)CC1C 13940,CC1CC(C)(C(=O)NC2CCC2NC(c2cc(F)n(C)n2)=O)CCO1 13941,n1(CC(=O)N(C(CN(C(c2cnc(C(C)=O)s2)=O)C)C)C)nc(C)cc1C(F)F 13942,Cc1cc(=NCC2CN(C(c3cc(C(C)(C)C)on3)=O)CC2(C)C)c(C#N)c[nH]1 13943,c1(OCC)cncc(C(=O)N(CCCCCNC(c2cncc(OC)n2)=O)C)c1 13944,CCC(C)CCCC(=O)NC1CCN(C(=O)CS(C)(=O)=O)CC(O)C1 13945,N1(C(CCC#C)=O)CC(NC(=O)CCc2cccnc2C)CC12CCCCC2 13946,C(CC(CC)C(=O)NC1CCCCC1C(=O)N(C(C)CC)CCO)=CC 13947,c1(C(=O)NC2C(NC(c3ncc(OC)nc3)=O)CCOC2)cc([N+](=O)[O-])nn1C 13948,C1(NC(C(c2cn(C)nc2)(F)F)=O)CCN(C(=O)CCOCC(F)(F)F)C1(C)C 13949,c1(CC)nc(C)c(C(=O)NC(C)C(CO)NC(c2nc(C)sc2C)=O)o1 13950,CN1CCC(C(N2CC3CC(C(=O)NC4CCN(CC5CC5)C4)(C3)C2)=O)CC1=O 13951,CCC(C)C(O)C(C)C(=O)N(CCC(=O)NCC1CC1)CCCO 13952,c1(C(=O)NCC2CC(NC(C3CCS(=O)(=O)C3)=O)C2)cc2c(nn1)CCC2 13953,N1(C(C2CCC(N=[N+]=[N-])C2)=O)CCC2(CC1)CN(C(=O)CCCCO)CCO2 13954,Nc1nccn2ncc(C(=O)NC3CCC(CNC(=O)Cc4ncc(Cl)s4)C3)c12 13955,C1(C(=O)OCCOCC(C)(F)F)CCCCN1O 13956,CC1(C)CC(C(N2CCCC(CCNC(C3CCC(=O)C3)=O)C2)=O)CC(C)(C)S1 13957,CC1CCCCC1C(=O)NCC1(CNC(=O)C(F)(F)c2ccncc2)CC1 13958,c1(C(=O)NC2CCC2NC(=O)C(O)c2cnc[nH]2)ccc2c(c1)CCCS2(=O)=O 13959,C1(CNC(c2csc(C)c2C)=O)CN(C(=O)CCC#N)CCC1C 13960,C1(C(N(CCN(C(C)C)C(c2ccc(CCO)cc2)=O)C)=O)C2CC2C2CC12 13961,C1(CNC(c2ccn(CCN(C)C)n2)=O)COC(C)(C)CN1C(c1cn[nH]c1)=O 13962,c1(-c2c(CC)nco2)nc(C2CCCC2)nn1C1CCSC1 13963,C(=O)(C1=C(C(C)=O)N(CCF)C(=O)NC1c1cc(Cl)c(F)cc1F)OCC 13964,N1(C(Cc2c(C)ccs2)=O)CCC(C)(NC(=O)Cc2nnn(C(C)(C)C)n2)C1 13965,c1(C(N2CCCC(NC(c3ccc(CO)nc3)=O)CC2)=O)cn2ccnc2cn1 13966,c1(CNC(CC2CCN(C(CCCCOCC)=O)C2)=O)ccc2cc[nH]c2c1 13967,C#Cc1cc(C(=O)N(C)CCN(C(=O)C(c2ccc(F)cc2)F)C)cc(F)c1 13968,CC#CCCCC(=O)NCC1CCCCC1NC(c1oc(Br)cc1C)=O 13969,c1(C(N(CC(C)C)CCC)=O)occc1CNC(c1nccn1CC)=O 13970,C(=O)(C(CN(C)C)N(C)C)NCCN(CCOC)Cc1cn(C(C)(C)C)nn1 13971,C(=O)(C1CCCc2nncn21)NCC(C)CNC(c1ncn2c1CCCC2)=O 13972,c1(C(=O)NCC2CCC(NC(C(c3cnn(C)c3)OC)=O)C2)ccc(O)nc1Cl 13973,Cn1c(C(=O)NCC(C2CCOC2)NC(c2cnc3n2CCS3)=O)cccc1=O 13974,CCCCC(C)CCC(=O)N1CCC(F)C(NC(c2ncoc2C2CC2)=O)C1 13975,c1(C(=O)NC(c2cnn(C)c2)C(=O)NC(c2ccccc2)C)n[nH]c2c1CCC2 13976,C1(CNC(C=Cc2n(CC)ncc2)=O)CCN(C(=O)C(C)(C)SC)CC1C 13977,Cc1cc(C(N2CCCC2CNC(C2(c3cccnc3Cl)CC2)=O)=O)cc(F)c1C 13978,C(=O)(CC(C)C(C)(C)NC(C1CNC(=O)N1)=O)N(CC(C(C)C)OC)C 13979,CC(C)C(CNC(C1C2CCCCCC12)=O)C(=O)NC(C1(O)CCC1)C 13980,c1(C(C)C(=O)NCCNC(=O)Cc2csc(NC=O)n2)ccc(OC(F)F)cc1 13981,c1(OCC(N2CCC(N3CCCC3=O)CC2)=O)ccc(Br)cc1OCC(F)(F)F 13982,C1(C(=O)NC(c2ccc(C)cc2)CNC(C2CC(=C)C2)=O)CCC2(CC1)CC2 13983,Cc1cnc(C)c(C(N2CC(NC(c3c[nH]nc3C(C)C)=O)CCC2C)=O)c1 13984,N1(C(C=C(COC)C)=O)CCCC(NC(=O)CN(C2CCC2)C)CCC1 13985,C1(C(C)C)CC(CC(N(C2CCCC2)CC(=O)NCC(=O)N)=O)C1.C(CN(C)C)S 13986,CCCC(C(=O)NC1CCCC(CNC(=O)CSCc2ccncc2)C1)C(C)C 13987,c1(NC(c2ccc(Br)s2)C)[nH]c(=NCC(C)Oc2ccccc2)nc2scnc12 13988,CCCCCCC(C)C(=O)NC1CC(C(=O)NCc2nnn(C)n2)=CC1O 13989,Cc1c[nH]nc1CC(=O)NCC(C(C)C)NC(C1CN(S(=O)(=O)C(F)F)C1)=O 13990,N1(C(c2c(C)nn(CC)c2C)=O)CC2CCCC2(NC(=O)Cn2cncc2C)C1 13991,CC1(C)C(c2ccc(Br)cc2)CCN1C(C1CCN(C(=O)CN)CC1)=O 13992,c1(C(=O)NC2(C(=O)NCC(C)Cn3cccn3)CC2C)cc([N+](=O)[O-])n[nH]1 13993,C1(CCNC(C2CCN(CC)C2)=O)CSCCN1C(=O)CC(C)n1cccn1 13994,N1(C(C(C)C(C)(C)C)=O)CCC2(CCCCN(C(=O)Cc3ccsc3)C2)C1 13995,c1(CN2CCN(c3ncc(C)s3)CC2)ccc(S(=O)(=O)C(F)F)cc1 13996,c1(C(=O)NC(CNC(CCCCC#C)=O)C2CC2)cc(Cl)cc(Cl)c1O 13997,n1(CC)nc(C(C)C)cc1C(C)C.c12ccc(nc1)C(=O)ON1CC2(O)C1 13998,c1(C(=O)NC2CC(F)(CNC(C(CC)C(C)C)=O)C2)c(F)cc(Cl)cc1F 13999,C1(C(N(C)CC2CCN(C)C2)=O)CC2(CCC2)CN1C(c1ccc(C#N)s1)=O 14000,CCC(C)CCC(=O)NCc1nc(C)c(C(=O)NCC2(CC)CCCC2)o1 14001,C(=O)(C1=NOC2(CCN(c3nccc(Br)n3)C2)C1)Nc1cc(C)c(C)c(C)c1 14002,C1(C(=O)NCC(C(C)C)NC(c2csc(C(F)F)n2)=O)CC(=O)N(C)C1 14003,c1(ONC(C2OCCN(C(C(C)C)=O)C2)=O)ccc2sccc2c1 14004,N1(C(c2ccc(CC)s2)=O)CCC(F)CC1C(N1CCN(C)CC1C1CC1)=O 14005,C(CC1=CCCCC1)NC(C1C=CCN(C(c2ccsc2Cl)=O)C1)=O 14006,C(=O)(C(C)(C)CF)N(C1CCN(C(=O)CC2CCN(C)C2=O)CC1)C 14007,c1(C(=O)NC2CC(CCNC(Cc3n(C)nnc3)=O)C2)ccc(N)cc1O 14008,c1(C(N2CC(CNC(CC3(OC)CC3)=O)C(O)C2)=O)cc(C)c(Cl)cc1F 14009,Cn1c(CN(C=O)Cc2ccc(N3CC=CC3)cc2)nnc1-c1ccccc1 14010,c1(NC2CN(C(C)=O)C2)[nH]c(=NC(C)c2cnc[nH]2)nc2sccc12 14011,N1(C(=O)Cn2cnnc2)CC2CC(N=c3ccnc(CO)[nH]3)CC1C2 14012,C(=O)(CC(C1CCC1)NC(C1CCN(C2CCOCC2)C1)=O)OCC 14013,N1(C(CC(CC)c2ccc(C)cc2)=O)CCC2(CC1)CN(C(=O)CCC(C)=O)C2 14014,C(c1ccc(Cl)s1)=CC(N1CCCC(NC(=O)C(F)(F)C2CCCCC2)C1)=O 14015,C(=O)(C(CCC1CCC1)NC(=O)C1=CCCC1)NC(c1ccc(O)cn1)C 14016,C1(C2(NC(C34CC3CN(C(=O)CCc3cnc(C)o3)C4)=O)CC2)(OC)CCC1 14017,C1(C(N2CC(CCNC(C(CC)NC(C)=O)=O)C2)=O)CC2(CCC2O)C1 14018,C12(C(N(C3CCN(C(C(C)OCC)=O)C3)C)=O)CCC(OC)(CC1)CC2 14019,S(=O)(=O)(CCC(=O)NCC1COCCN1C(c1ncnn1C(C)C)=O)NC 14020,N1(C(CCSCC)=O)CCC(NC(c2ccc3cc(C)cn3c2)=O)C2(CCC2)C1 14021,N1(C(CCCCSC)=O)C2CCC1C(C(=O)NOCC(C)(C)C)C2 14022,c1(C(=O)NCCC2CCC(NC(c3ccc(Cl)o3)=O)C2)cccc2cc[nH]c12 14023,Cc1c(Cl)cc(C(=O)NCC(C)NC(=O)C(N2CCCC(C)C2)=O)cc1Br 14024,c1(C(N2CCN(C(c3nc(CC)oc3)=O)CC2CC)=O)c(C)cc(Br)cc1C 14025,c1(CC)cc(C(=O)NC2CC(C(=O)NC3C=CCC3)C2)ccn1 14026,c1(C(=O)NCC23CC(NC(CN(CCC)C)=O)(C2)C3)ccc2cccnc2c1 14027,C1(CC)(NC(C2CCC(c3ccccc3)C2)=O)CCN(C(=O)CC(C)(F)F)CC1 14028,N1(C(c2c[nH]c(=NC)s2)=O)CCCC12CCCN(C(=O)C(C)CSC)C2 14029,c1(C(=O)NCC(CNC(C2C(OC)CC2)=O)(C)C)cccc(SC)c1[N+](=O)[O-] 14030,C(CCCCN(C(=O)CC(C)n1cc(Br)cn1)C)NC(C=C(C)C1CC1)=O 14031,n1(CCC)cc(Cl)c(C(=O)NC(C)CN(C(c2cccc(F)c2)=O)CC)n1 14032,c1(OC)cc(C)c(C(=O)NCC2CCC3(CN(C(=O)CC(C)SC)C3)O2)c(C)c1 14033,C1(NC(C(CC=C)NC(=O)C=CCOC)=O)CC(C)(C)OC1(C)C 14034,C1(N(C(c2cc(CC)on2)=O)C)CCCC(N(C(=O)CCCN2CCCC2)C)C1 14035,CCC(N)C(C)(C)C(=O)N(C1(CO)CCN(Cc2ccccc2)CC1)C 14036,N1(C(CC(C(C)OC)NC(c2c(CC)oc(C)c2)=O)=O)CC=C(C(C)(C)C)CC1 14037,C(c1ccc(OCC)c(Cl)c1)=CC(N1CC(NC(COCC)=O)C(C)C1)=O 14038,C12(NC(CC3CC(OC)C3)=O)CC3CC(C1)CC(NC(C1CCC(C)O1)=O)(C3)C2 14039,C1(C(N(CC(=C)C)CC(=C)C)=O)CCCC(NC(c2ccc(C3CC3)nc2)=O)C1 14040,N1(C(c2n(C)ncc2Cl)=O)CC(O)CCC1C(=O)NCC1CC2(CC2)C1 14041,c1(OC)ccccc1CC1CCCN1C(=O)C(C)(C)NC(c1ccc(C)cn1)=O 14042,N1(C(C(CC=CC)C)=O)C(C(N2CCCC2C(O)CC)=O)CCC12CC2 14043,C1(C(=O)NCC2(SC)CCC2)CC(F)CN(C(=O)C(c2cccn2C)=O)C1 14044,Cc1cccc(C(=O)NCCC23CCC2CN(C(c2nocc2Br)=O)C3)c1O 14045,c1(CNC(C2COCCN2CC)=O)coc2cc(N)c(-c3ccc(CO)s3)cc12 14046,CC1=C(C(=O)OCC(F)(F)F)C(c2cc(C(C)C)cc(C)c2)NC(=O)N1C 14047,c1(C(=O)NC2CC(NC(=O)COCCOCCO)C2)ccc(F)c(O)c1F 14048,C(=O)(CCN=c1cc(NCC2CC(C3CC3)C2)nc[nH]1)N(C)C 14049,c1(SCC(=O)NCC2(F)CC(NC(C3C4CC4C4CC34)=O)C2)cccc[n+]1[O-] 14050,N1(C(C(C=CC)O)=O)CCC2CC12C(=O)N(C)CCN1CCCC1=O 14051,N1(C(=O)CSc2n[nH]c(O)n2)CCN2CCNCC2C1 14052,C1(C(=O)NC2C(NC(C3(C)CCCC3)=O)CS(=O)(=O)C2)CCC(C2CC2)CC1 14053,N1(CC(=O)NC(CNC(CC=C)=O)C(C)C)C(=O)NC(C)(COC)C1=O 14054,c1(CC(=O)NCC(CNC(Cc2cnc(C)[nH]2)=O)F)ccc(Br)cc1 14055,c1(C(=O)NCCCC2N(C(C(C#N)C3CC3)=O)CCCC2)cc2c[nH]nc2s1 14056,c1(OC)ccc(S(=O)(=O)N2CCCC(C)(C(=O)Nc3c[nH]nc3C#N)C2)cc1Br 14057,C(=O)(CCCC(F)(F)F)NCCCN1CCC(NC(C(NOC)=O)=O)C1 14058,C1(NC(CNC(=O)NC)=O)(CNC(=O)Cc2cnc[nH]2)CCCCCC1 14059,c1(OC)ccc(CN2CCCC(C(=O)N(C)CC3CCCCC3)CC2)c(Cl)n1 14060,C(CN=C(NCC(=O)N(C)C)NCC1CCOC1)(c1ccc(F)cc1)OC 14061,CCCC(C)(CC)C(=O)NC1CC(CCNC(=O)C(C)(CC)CC)C1 14062,C1(NC(C(CC)N(CC)CC)=O)C2CN(C(c3cccnn3)=O)CC12 14063,N1(C(C(CCCC)=O)=O)CCOC2(CCN(C(=O)C=Cc3cccs3)C2)C1 14064,CC1(NC(C2Cc3nccn3C2)=O)CCN(C(c2cc(Cl)cs2)=O)CC1 14065,Cc1cc(CC(=O)NCCN(C(C23CCCCC2C3)=O)CC2CC2)n(C)n1 14066,CCCCC(O)C(C)C(=O)N1CCN(C(=O)Cc2cc(C)[nH]n2)CC1CCC 14067,c1(C(=O)NC2C(NC(C3CN(C)C(=O)N3)=O)CCCC2)cccc(C(N)=O)c1F 14068,c1(NCC2C(C)CC=CC2)ccc2c(c1)COCC2 14069,c1(C(=O)NCC(C)NC(=O)C(=O)N(C)C)ccc(NC(=O)Cn2cnnc2O)cc1 14070,c1(C(c2n(CCOCC)nnn2)NCCC2CC=CC2)cc(C)nn1C 14071,c1(C(N2CCC(NC(CNS(CC)(=O)=O)=O)C(C)C2)=O)ccc2nc[nH]c2c1F 14072,N1(C(c2c(CNC(C=CCOC)=O)ccs2)=O)CC(C)(C)C1C1CC1 14073,Cc1cccc(C)c1C(O)C(=O)NCC(C)CN(C(=O)CCc1nccs1)C 14074,C1(C(c2ccccc2)NC(=O)C(=O)NCC(=C2CCSCC2)F)CCCC(=O)N1 14075,c1(OC)c(F)ccc(CN(C(=O)CNc2ccc(C(F)(F)F)cc2)C)c1F 14076,c1(-c2nc(CC)nn2-c2cccc(NC(C)=O)c2)onc2ccccc12 14077,c1(NC(c2n(CCCC(=O)OCC)nnn2)(C)CC)ccc2c(c1)CCCS2 14078,c1(C(N(C2CC(NC(=O)CC3CCC3)C2)C)=O)ccc(OCC(F)(F)F)c(Cl)c1 14079,c1(C(=O)NC2CC3CN(C(C4(CCN(C)C)CC4)=O)CC32)ccc(S(C)=O)cc1 14080,C1(NC(CCCCOC)=O)C2CC3C1C3C2C(=O)NCCN1CCOCC1C 14081,Cc1nc(CC(=O)NCCn2cc(C3(CCO)CC3)nn2)c(Br)s1 14082,c1(C(N)=O)ccccc1OCC(=O)NCCC1(O)CN(C(C2CCNC2=O)=O)C1 14083,N#Cc1cnn(CC(N2CC3CC2CN3C(c2cnnc(O)c2)=O)=O)c1N 14084,c1(N(C)C)ncc(C(=O)NC(CC(N)=O)c2cn(CC3CCCO3)nn2)cn1 14085,C(c1cccc(O)c1)=CC(=O)NCC(C)(F)CNC(C1CCCN1C1CC1)=O 14086,N1(C(C2(OC)CCOCC2)=O)CC2CCN(C(C3COCC(C)(C)O3)=O)CC2C1 14087,CCCCC(C(=O)NC1CC2(C1)CN(C(c1cc(CC)[nH]n1)=O)C2)NC(N)=O 14088,C(=O)(CCCCCCC=C)NC(CC#C)C(=O)NCCCc1cccs1 14089,C1(NC(c2ccc(C#C)o2)=O)(CO)CCCN(C(=O)CCCc2ccccn2)C1 14090,c1(C(=O)NC2CCCN(C(CC(COC)C)=O)C2C)ccc2c(c1)C(=O)NC2=O 14091,c1(C(N2CC(NC(C3C(C)C3c3ccccc3)=O)C2)=O)nccnc1Cl 14092,C1(CNC(C2(C)CCCS2)=O)CCC(F)(CNC(=O)CN2CCSCC2)C1 14093,N1(C(C(CC=C)OC)=O)CCCC(O)(CCNC(C2(O)CCCCCC2)=O)C1 14094,C(=O)(C(C)(C)C(N)=O)NCCCC(C)NC(=O)C(C)c1ccco1 14095,C1(CC)(NC(c2ccc(Cl)c(OC)c2)=O)CCCN(C(=O)CCc2cn[nH]c2)C1 14096,CC1CN(C(=O)CC(C)(C)O)CC2(CCN(C(c3ccc(=O)n(C)n3)=O)C2)O1 14097,c1(SC)cccc(C(=O)N(CCCNC(C2C3CN(C)CC23)=O)C)c1 14098,c1(C(=O)NC(C2CCCN2C(=O)CN=S(C)(C)=O)(C)C)ncc2c(F)cccn12 14099,CC(C)C(C(=O)NCCNC(c1cccnc1-c1ccc(F)cc1)=O)C1CCC1 14100,C1(CNC(=O)Cc2ccccc2CO)CN(C(c2cccc[n+]2[O-])=O)CC12CC2 14101,C12(NC(CCCC3C(C)C3)=O)CCC(C(=O)NC34CC=CC(C3)OC4)(CC1)C2 14102,C1(NC(c2c(CC)noc2)=O)CN(C(c2cccc(N)n2)=O)CC(C)(C)C1 14103,C1(C2(O)CN(C(c3cccc(OC)c3)=O)C2)(CNC(C(COCC)C)=O)CC1 14104,C(=O)(CCCCNC(=O)Cc1cncc(C)c1)NCC#CC 14105,CCCCC(C)(F)C(=O)N1CC2(CCN(C(c3cocc3Br)=O)C2)C1 14106,c1(CC)ccccc1-c1ccc(N2CCNCC2)nc1.c1(C=O)ncnn1C 14107,C1(C(C)C)CN(C(c2ccc(Cl)nc2)=O)CCN1C(c1cn(C(C)C)nn1)=O 14108,c1(C(=O)NCC2C(C(=O)NCC(CCOC)O)CC2)cccc(C)n1 14109,N1(C(Cc2scc(C)n2)=O)CCCCC2(CCCCC2)C1 14110,C1(CNC(CC=C)=O)CN(C(=O)CN(CCC)C(=O)OC(C)(C)C)CCC1(F)F 14111,C12(C(=O)NC3C(NC(CCc4cn(C)nc4)=O)CC3)CCC(CC1)C(C)(C)O2 14112,c1(C2C(C)C2)ccc(C=CC(N2CC(CNC(=O)CC3CC4CC4C3)C(C)C2)=O)o1 14113,CC1CCCCCCN1C(=O)C(C)N(C(=O)CCN1CCOC1=O)C1CC1 14114,Cc1c(N(CC(c2ccc(Br)cc2)O)C)nc(Cl)nc1C(F)(F)F 14115,N1(C(c2c(C)nns2)=O)CCC(N2CCN(C(c3cccnc3Cl)=O)CC2)CC1 14116,CN1CCC(C(=O)NOCC(O)C(=O)O)(NC(=O)CC2CCCC2O)C1 14117,c1(C(N2CCC(N)(COC)C2)=O)cc(Br)c(O)nc1C 14118,N1(C(c2cnc(SC)n2C)=O)CC(C)CCC1CNC(=O)COC(F)(F)F 14119,c1(NC(C(CC)NC(C)=O)=O)ccc(-n2ccnc2)cn1.C123CC(C1)(C2)NC3=O 14120,N1(C(c2n[nH]c(CC)c2C)=O)CCCCC(C(=O)NCC(c2cnn(C)c2)C)C1 14121,C#Cc1ccc(CC(=O)NCCN(C)C(C2(C)CCC(=O)C2)=O)c(F)c1 14122,c1(CC)ccc(C(=O)NCC2CCC(NC(C3CCN(C(C)=O)C3)=O)C2)nc1 14123,N1(C(C(C(C)O)(F)F)=O)CC2(C1)CN(C(C1(c3ccno3)CC1)=O)CCO2 14124,c1(C(C(=O)NCC(C)N(C)C(c2cnccn2)=O)(C)F)ccccc1F 14125,CS(=O)CCC(O)C(=O)NC1CC(CNC(c2cncc(F)c2Cl)=O)C1 14126,C1(C2(O)CN(C(c3ccncc3N(C)C)=O)C2)(CNC(C(C)(C)CO)=O)CC1 14127,C(=O)(C(C)(C)C(O)C(C)C)NCC1(F)CCN(C(c2n(CC=C)ccc2)=O)C1 14128,CC1CN(C(=O)C=CC2CCCC2)CC(C)N1C(C1CCC(C2CC2)C1)=O 14129,c1(N(CCNCc2cccc(C)n2)C)ncnc(NC2C=CCN2C)c1C 14130,CCCCC(C(=O)NCC1C(C)(C)C1(F)F)NC(c1cc(C2CC2)[nH]n1)=O 14131,Cc1nn(C)cc1C(=O)NC(Cc1cnc[nH]1)C(=O)NCC1CC(C2CC2)C1 14132,C(=O)(C(CC(=C)C)NC(c1c[nH]nc1OC)=O)NCCCCCC=C 14133,C1(C(=O)Nc2cn(CC#C)nc2)CN(C(C2(NC(C)=O)CC2)=O)CCO1 14134,C1(O)(C(C)CNC(c2cnsn2)=O)CCN(C(c2cnc(S)nc2)=O)C1 14135,C=CCC(CC)C(=O)N(C1CN(C(c2ccnn2C)=O)CC1(C)C)C 14136,C1(C(c2occ(C(N3CCC(OC(C)=O)C3)=O)c2)=O)CCN(C(=O)C(C)C)CC1 14137,C1(C(=O)OC)CC12CCC(NC(=O)Nc1ccc(F)cc1Cl)CC2 14138,CC(C)(C)C#CC(=O)NCC1CN(C(=O)C=Cc2ccsc2)CC1(F)F 14139,N1(C(C2N(C(Cc3cc(C)[nH]n3)=O)CC2C)=O)CCC2(COC(=O)N2)C1 14140,N1(C(C(C)NC=O)=O)CC(O)(CCNC(=O)Cc2ccsc2)C1 14141,C1(N(C(CCC=C)=O)CCO)CCCN(C(C2(C)CC=CC2)=O)C1 14142,C(=O)(C(S(C)(=O)=O)C1CC1)NCCC(C)NC(C(n1ccc(C)n1)(C)C)=O 14143,C1(C)(C(=O)NC(CC)(C)CNC(=O)CC2(CSC)CC2)CC(C)(C)C1 14144,N1(C(C(C=CC)O)=O)CCC(CC(=O)NCCCOC(=N)O)CC1 14145,N1(C(c2cc(C)ns2)=O)CCC2CC2(C(=O)NCc2ncccc2F)CC1 14146,Cc1nsc(CNC(=O)CC(C)NC(=O)C(c2cncnc2)C)n1 14147,N1(Cc2c(OCC)cccc2)CCCC(=O)C1C 14148,c1(OC)cc(NC(C2CC(NC(C3CC(OC)C3)=O)C2)=O)cc(F)c1 14149,c1(C(=O)NC(CC)CNC(C2CCN2C2CCCC2)=O)ccc2ncccc2c1 14150,c1(OCC)cc(C(=O)NC(C)CN(C(=O)Cc2c[nH]ccc2=O)CC)ccn1 14151,c1(C(=O)NCC(N(C)C(C2(C(F)(F)F)CCCC2)=O)C2CC2)ccnc(OC)c1 14152,N1(C(CSC(C)(C)C)=O)CCC(NC(c2ccn(C(C)(C)C)n2)=O)C1 14153,c1(CN(C(=O)CCOC2CN(C(c3ccco3)=O)C2)CC)cnn[nH]1 14154,N1(C(C(C)NC(C)=O)=O)CC2CC(N(C(=O)C(C)CN3CCOCC3)C)C1C2 14155,C1(S(=O)(=O)C(N2CCSCC2CCO)=O)(C(C)C)CC1 14156,N12CC3CC(CC1C3)NC(=O)C2=O.Cc1cc(OC(C)C)ccc1-n1cnnn1 14157,C#Cc1ccc(NCc2ccnc(CO)c2)cc1C#N 14158,CC(C)C(O)C(=O)N1CC2CC1(CNC(=O)CC1CC3(CC3)C1)C2 14159,c1(-c2ccc(-c3n(-c4ccn(CC)n4)ccn3)s2)cccc(S(C)(=O)=O)c1 14160,C1(NC(c2c(OC)oc(C)n2)=O)CN(C(=O)CC2CCC(=O)NC2)CC1C1CC1 14161,C1(NC(=O)Nc2cnc(O)c(C(F)(F)F)c2)CN(c2ncncc2Cl)CC2(CC2)C1 14162,c1(NC(C)=O)ncc(S(=O)(=O)NC2CCC(C(=O)Nc3cc(Br)ncc3F)C2)s1 14163,c1(OCC(CN2C(CNC(c3c(COC)ncs3)=O)CCC2)O)cccc(C)c1 14164,N1(C(c2cc(OC)c(OCC(O)CN(C)C)cc2)C)CCC(C2CCOC2)C1 14165,CC1(C)CC(NC(=O)Cn2cncn2)CCN(C(=O)CCOC2CCC2)C1 14166,CC(O)C(C(=O)NCC(C1CCN(C(c2ncoc2C(C)C)=O)CC1)C)N(C)C 14167,C1(CC(=O)NC2CCCC(CNC(c3cccc[n+]3[O-])=O)C2)CCS(=O)(=O)CC1 14168,N1(CCCC(C)NC(=O)Nc2ccnn2C)C(=O)c2ccccc2C1=O 14169,N1(C(C2(C)C(C)(C)C2)=O)CCC(CC(=O)NCC2CC3C=CC2O3)CC1 14170,N#CC1(C(N2CCC(NC(c3cnccn3)=O)C(F)C2)=O)CC12CCC2 14171,Cc1cccnc1C(C)NC(c1ccc(-n2cc(-c3ccn(C)n3)nn2)nc1)=O 14172,c1(C(N2CC(CCC=C)(C(N3CCCCCCC3)=O)C2)=O)ccc2[nH]ccc2n1 14173,Cc1ccc2c(-c3ncn4c3CN(C(=O)C(C)n3ccnc3)CC4)cccc2n1 14174,C1(C(=O)NCCCc2onc(C)n2)CN(C(=O)CCCNC(=O)C2CC2)CCO1 14175,N1(C(C2N(C(C)=O)CCC2)=O)CCOCC(CNC(C2C=CCC2)=O)C1 14176,c1(CC)cc(CC(N2CCCC2C(C)NC(c2cn(C(C)(C)C)cn2)=O)=O)on1 14177,n1(CC(=O)NCC(CNC(CC)=O)F)cnc(-c2ccccc2)n1 14178,N1(C(CN(CC)CC)=O)CCC(CNC(c2ccc(O)cc2F)=O)C(CC)C1 14179,Cn1cc(C#N)cc1C(=O)NCC#CCNC(c1coc(-c2cccnc2)n1)=O 14180,CCCC(CCCNC(C12CC(NC(c3cc(CC)cc(C)c3)=O)(C1)C2)=O)OC 14181,C1(NC(c2cn(CCOC)nn2)=O)CC12CCN(C(C1CCC3CC1CO3)=O)C2 14182,C(=O)(C1=CC(C)(CC)C1)N1C(C(=O)NCC(CC=C)(C)C)C=CC1 14183,C=CCC(F)(F)C(=O)NCC(C1(O)CCN(C(c2coc(C(N)=O)c2)=O)C1)C 14184,CC(CCNC(C1CN(C(c2cc(O)ccc2F)=O)C(C)(C)C1)=O)CC(C)(C)C 14185,CCCN(Cc1ccc(O)cc1)N1Cc2ccc(C(C)=O)cc2C1 14186,N1(C(C(C)Cn2ccnc2)=O)CC(NC(=O)CCN(C)CCO)CC2(CC2)C1 14187,N1(C(CC(c2ccc(OC)cc2)C)=O)C2CCC(C(=O)O)C1CC2 14188,CCCC(C)(O)C(=O)N1CC(C(C)NC(c2ccc(=O)n(O)c2)=O)C1 14189,c1(C(N2CC(CCCCNC(C=COCC)=O)C2)=O)cc(C)c(C)nc1C 14190,C1(NC(COCC=C)=O)CC1C1CCN(C(C2CCc3nn[nH]c3C2)=O)CC1 14191,N1(C(CSCC=C)=O)CC2CCCN(C(=O)C(C)Oc3cccc(C)c3)C2C1 14192,c1(CC(=O)NCC=CC(N2CCCC(N(C)C)C2)=O)coc2ccccc12 14193,N1(C(CCC(=O)OC)=O)CCN(C(c2ccc(C)cc2Cl)=O)C(C2CCCC2)C1 14194,N1(C(C2N(C(c3ccc(C#N)cc3)=O)CCCCC2)=O)CCC2(COC(=O)N2)C1 14195,C1(O)(CC)CCN(C(c2cc(C(N)=O)co2)C(=O)NC(C)CC)C1 14196,c1(CN2CC3(CCC(C(N4CCn5cnnc5C4)=O)O3)C2)c(F)ccc(Br)c1F 14197,c1(NC(C23CCCCC2C3)=O)ccc(NC(c2nccs2)=O)c(F)c1 14198,c1(C(=O)NCC(=C2CN(C(CC3CCC(OC)C3)=O)C2)F)cc(C)ncc1C 14199,N1(C(C(CC)O)=O)CC2C(CNC(c3cnn(-c4ncc(Cl)cn4)c3)=O)C2C1 14200,c1(C(=O)NCC(C2CCCC2)C)cc(C(F)F)nc2ccc(Cl)cc12 14201,c1(C(=O)NCC2(O)CN(C(CC3CC(OC)C3(C)C)=O)C2)ccc(Cl)c(N)c1 14202,N1(C(C)=O)C=Cc2ccccc2C1CC(=O)NC1CC(n2cc(C(C)(O)CC)nn2)C1 14203,c1(CC)ccc(C(=O)NC(C)CNC(=O)CS(=O)(=O)C2CC2)cc1[N+](=O)[O-] 14204,C1(C)(CC)CCN(C(c2csc(Cl)c2)C(=O)NC2CC(F)(F)C2)C1 14205,CCCC(O)(CCC)CC(=O)NC(C)CN(C)C(C1CCn2nccc2C1)=O 14206,N1(C(C(C)=C(C)C)=O)C2CCC1C(F)C(NC(C1(N(C)C)CCN(C)CC1)=O)C2 14207,CC1CCCc2ncc(C(N3CCC(CO)(NC(=O)Cc4ccon4)C3)=O)n21 14208,C(CNC(C1(O)CCCC1)=O)(CC(C)C)NC(Cc1cnc(C)s1)=O 14209,C12(F)CN(CC1c1ccccc1)C2.C(=O)(N=c1[nH]nco1)C1CC1OC.O=CO 14210,c1(C(N2CC3(CC(NC(C(CC(C)C)F)=O)C3)C2)=O)coc2cc(F)cc(F)c12 14211,c1(OC)ccc(C(N2CCC2CNC(=O)Cn2c(C)c(C)sc2=O)=O)c(N)c1F 14212,C1(C(=O)NCCCNC(COCCCC)=O)CCCCC1F 14213,Cc1ccc2sc(N3CCC(C4CC4)C3CNC(c3ncccn3)=O)nc2c1 14214,C1(NC(C(C)(C)CO)=O)CN(C(c2n[nH]c3ccccc23)=O)C2(CCCCC2)C1 14215,N1(C(c2ccc(CSC)cc2)=O)CC2CC(C)N(C(C3CCC3CF)=O)C2C1 14216,N1(C(c2ccc(OC)c(Br)c2)=O)CCC2(CCN(Cc3ccc(O)c(O)c3)C2)C1 14217,O=C(C1CCc2cccnc21)NC1CN(C(c2cccc(CO)c2)=O)CC1O 14218,C1(C(CC)C)CCN(C(=O)C(C2(O)CCC2)NC(c2cccs2)=O)CC1 14219,C(=O)(C#CC1CC1)N(CC)CC1(C(N2CCOCC2)=O)CC1.C1(=O)C=CCO1.CN 14220,c1(CC)nc(C(C)C)ccc1C(=O)NCC(CC(C)C)NC(=O)COCC1CC1 14221,C(=O)(C(C(C)NC(C1CCC(=O)CC1)=O)C(C)C)N1CC(CC)(CC)C1 14222,C(C(C)(C)CNC(c1cc(C)ns1)=O)NC(CCOCC)=O 14223,C#CCCCC(=O)NC1(CO)CN(C(c2ccc(Cl)[nH]2)=O)C1 14224,Cc1cc(C(=O)NCC2CCN2C(=O)NC2CC23CCOCC3)ccc1[N+](=O)[O-] 14225,CON1CCC(CC(=O)NCCNC(C2CC(F)(F)C2(C)C)=O)CC1 14226,c1(OC)ccc(C(=O)NCC2CC2NC(C2(CN(C)C)CCOCC2)=O)cc1 14227,N1(C(C(CC2CC2)OC)=O)CCCN(C(=O)CN2CCCCCC2)C(C)C1 14228,c1(CNC(C=CCOC)=O)nocc1C(=O)NC1(c2nc[nH]n2)CCC1 14229,C#CCCCCCC(=O)NCC(CC=C)NC(c1cc(C)nn1C(C)(C)C)=O 14230,N1(C(c2cc(C(C)C)[nH]n2)C(=O)NCCC(=O)OCC)CC2CC=CC1C2 14231,CC(C)CC(O)C(=O)NCC1CCCN1C(=O)C1=CCCCC1 14232,C1(C)(OCC(=O)NC(CC)C2CC2)CN(C(=O)COCCSC)C1 14233,c1(OC)cccc(CCC(=O)NC2CCCCN(C(=O)C(C)(C)C)C2)c1F 14234,c1(SCC(=O)NCC(C)NC(=O)C=CCN2CCCC2=O)nccn1C 14235,C1(C(=O)NC2C(NC(COCCOCC)=O)COC2)CC2CCCC2C1 14236,N1(c2ccnc(OC)n2)CCOC2CN(C(c3ccn(C)c3)=O)CC12 14237,CC1CC=CCC1C(N1CC(NC(c2ccccc2C(C)(F)F)=O)C(F)C1)=O 14238,c1(OC)ccc(CCC(=O)N2CCC2CNC(=O)CS(N)(=O)=O)cn1 14239,c1(CC)cc(OC)ccc1N.c12ccc(cc1)N(CC)C(=O)C2N 14240,N1(C(C=CC(=O)OCC)=O)CCC2C(NC(=O)CC3CN(C)CCO3)CC12 14241,c1(OC)cscc1C(N1CCC(CCNC(C2CC2F)=O)C1)=O 14242,C1(C(=O)NCC2(C(C)NC(C3CC=CC3)=O)CC2)C=CCCC1 14243,c1(C(C)C)conc1CC(=O)NC(CNC(=O)C(C)CC1CC1)C(C)C 14244,c1(OC)cccc(-n2nc(-c3ccsc3)nc2-c2scnc2Cl)c1 14245,C=CCCCCCCCC(=O)N(CC)CC1CC(O)C1(C)C 14246,C1(CCNC(CCN(C(C)=O)C)=O)(NC(c2nnn(C)c2N)=O)CCOCC1 14247,N1(C(CCCOCC=C)=O)CC(C(N2CCC(N3CC(O)C3)C2)=O)CCC1(C)C 14248,c1(OC)ccc(C(=O)NC2CCN(C(c3cncn3C)=O)CC2C)cc1N 14249,N1(C(COCCOCC)=O)CCC(NC(=O)COCc2cccc(C)c2)CC1 14250,c1(C(=O)OCC(c2noc(-c3ccccc3)n2)=O)cc2ccc(O)cc2[nH]1 14251,C=CCC(C)C(=O)NC1(CF)CCN(C(=O)C(C)NC(c2ccc(Cl)nc2)=O)C1 14252,C(=O)(CC(C(F)(F)F)P(C)(C)=O)NCCC1CC(NC(c2c(C)[nH][nH]c2=N)=O)C1 14253,CCCCCCC(CC)NC(=O)C(C1CCCN(C(=O)CC(C)(F)F)C1)C 14254,C#Cc1ncc(F)cc1NC(c1ccc(Cl)s1)c1nnnn1CC1CCCO1 14255,c1(OC(c2nc(C(=O)OCC)n(C)n2)=O)cc([N+](=O)[O-])ccc1SCC 14256,c1(OC)c(Cl)ccc(C(=O)NC(C)C(C)NC(=O)CN2C(=O)CN(C)C2=O)c1F 14257,C(c1nc2ccccc2o1)=CC(=O)NCC1(F)CCN(C(C(C)OCC)=O)CC1 14258,N1(C(C(CC)c2ccccc2)=O)CC2(CC(NC(c3c(C)ncn3O)=O)CO2)C1 14259,Cc1[nH]c(=N)sc1C(=O)NC1CCCC1(O)C(F)(F)F 14260,CC1CN(C(=O)CC2(C)CCCO2)CC1CNC(c1nn(C)cc1Cl)=O 14261,C1(CCNC(c2n(CC(=C)C)nnn2)c2cnoc2)CCCC(C)C1 14262,C(=O)(C1=NNC(C(F)(F)F)C1)NCCc1c(CNC(C(C)CF)=O)nco1 14263,c1(CC(=O)NC2C=CCN(C(c3c(C(=O)OC)cco3)=O)C2)cc(F)ccc1Cl 14264,N1(C(CC(CCC)C)=O)CCC2(CCCN(C(=O)C(C)(C)C(C)O)C2)CC1 14265,c1(CC(N2CCC(N(C(=O)CS(=O)(=O)CC)CC)CC2)=O)nc2ncccn2n1 14266,c1(N2C3(CNC(=O)C4=NOCC4)CCC2CC3)ncnc2sc3ccccc3c12 14267,N1(C(CC)C)CCN(C(=O)CCC2(C(=O)O)CCCC2)CC1 14268,C(C#Cc1nccc(N2CCC(O)C(C3CC3)C2)n1)OCC1(N=[N+]=[N-])OC(NC(=N)N)C1 14269,C1(C(C)C)CC(CNC(N2CC(NC(C)(C)C)C2)=O)CCO1 14270,N1(C(C2C(C(=O)OC)C2(F)F)=O)CCOC(C)(CNC(=O)COC2CC2)C1 14271,Cc1cc(=NC(=O)C2CCc3c(sc(C(C)=O)c3C#N)C2)cc(C)[nH]1 14272,c1(OCC(N2C(C(C)NC(c3cc(Br)co3)=O)CCC2)=O)ccccc1O 14273,N1(C(c2c(C)nn[nH]2)=O)CCC(F)C(NC(c2cc(Br)ncc2Br)=O)C1 14274,c1(C(=O)NCC(c2c(OC)cccc2)O)csc2ccccc12 14275,c1(C(N(C2CCN(Cc3cnn(C)c3)C2)CCC)=O)ncoc1C 14276,c1(OC(CC)=O)ccc(OCC)cc1C(N1CCCCC1CCO)=O.C1C(=O)N1 14277,N1(C(c2c(CC)nn(C)c2)=O)CCCC(F)(C(N2CCCC2(C)CO)=O)C1 14278,c1(C(=O)NC2CC(NC(C(C(C)C)N(CC)CC)=O)C(O)C2)cc(F)cnc1O 14279,C1(NC(C2CCN(C)C2)=O)C2CN(Cc3ncc(Br)s3)CC12 14280,c1(CC(N2CCC(C)(NC(C=Cc3ccc(C)o3)=O)C2)=O)cccc([N+](=O)[O-])c1 14281,c1(NC(C2CCN(C(=O)CCc3ccnn3C)C2)C)ncc([N+](=O)[O-])c(=N)[nH]1 14282,N1(C(Cn2cnc(=N)[nH]2)=O)CCC2CCN(C(=O)CC=C(Cl)Cl)CC2C1 14283,O=C(C1CCCc2c[nH]nc21)NC1CN(C(c2cc(F)c(F)cc2O)=O)CC1F 14284,Cc1cnc(Cl)c(C(=O)NC(C2CCN(C(c3ccco3)=O)C2)C)c1 14285,c1(C(=O)NCC2(CNC(CC(COC)C)=O)CCCCC2)cnn2ncccc12 14286,C1(C(=O)NCCC2CN(C(=O)CC3CC3)C2)CCC(CC(F)(F)F)CC1 14287,C1(C(=O)NC2CC(CNC(c3nc(C)oc3C)=O)CC2O)CC2OC1C1CC21 14288,c1(C(N(C(C)CNC(=O)Cc2cc(C3CC3)on2)C)=O)ncc(C#N)cc1F 14289,C1(CNC(c2csc(Br)n2)=O)CCCCN1C(C1(C2CC2)CC1)=O 14290,n1(CC=C)cc(C(=O)NC2(C)CN(C(C3(OC(C)=O)CCC3)=O)C2)cn1 14291,C1(N2CCC(NC(C3C(C)(C)C3(C)C)c3n(C)nnn3)C2)CC(F)(F)C(=O)N1 14292,N1(C(CC(CC2CC2)NC(=O)CCc2ccsc2)=O)CC2CCCC(O)C2C1 14293,C(=O)(CC(C)CC(C)C)NCC(C(=O)N(C(CC)CO)CC)C(C)C 14294,N1(C(c2ccnc(C)c2N)=O)CCCC(C)(C)C1C(=O)NCCC(C)C(F)F 14295,O(S(=O)(=O)c1cccc2c1OC(C)C2)c1c(CC)nn(C)c1CC 14296,CC1(C)OCC2CC12C(=O)NCCC1COCCN1C(=O)C=Cc1ccccn1 14297,Cc1n[nH]c(C)c1C1CC1C(=O)N(C1CCCN(C(=O)CC2CCC2)C1)CCF 14298,CCCC(=O)NCC(=O)NCC(F)CNC(=O)Cn1cccn1 14299,C1(CNC(c2cccc(SC)c2)=O)CN(C(c2cnns2)=O)CCC1C(F)(F)F 14300,N1(C(CCCC)=O)CCC2(CCC(C(=O)NC3CC3CC(C)(C)C)C2)C1 14301,N1(C(C(C(C)C)NC(C)=O)=O)CCC2CCC(NC(=O)CC3(C)CC3)C1C2 14302,c1(C(=O)NC(CCCNC(C(C)OC)=O)C)cccc(SC)c1[N+](=O)[O-] 14303,C#Cc1cncc(C(N2CCCC2(C(=O)Nc2ccc(O)cc2CC)CC)=O)c1 14304,N1(C(c2c(C)sc(O)n2)=O)CCC2(CC1)CC(NC(c1ccc(O)nn1)=O)C2 14305,N1(C(CSc2n(C)cnn2)=O)CCC(C)(C)C(NC(=O)CSC(F)(F)F)C1 14306,C1(NC(C2CCCC2)=O)COCCN(C(=O)CC(O)Cc2ccccc2)C1 14307,C1(CC(N2CC(CNC(c3ccn(C4CC4)n3)=O)C(O)C2)=O)CCC2(CCC2)O1 14308,c1(C(N(CCNC(c2ns[nH]c2=O)=O)CC)=O)cc(S(=O)(=O)CC)ccc1OC 14309,CC1CC(c2cn(CCN3CCNC3=O)nn2)CCN1C(C1CS(=O)(=O)C1)=O 14310,N1(C(CCC#C)=O)CCN(c2ncc(-c3ccc(C(C)N)cc3)cn2)CC1 14311,Cc1n[nH]c(C)c1C(C)C(=O)NC1CC(C(C)NC(c2coc(N(C)C)n2)=O)C1 14312,c1(C(N(C)CC2COCCN2C(=O)CC2(C)CCCC2)=O)cccc(S(C)=O)c1 14313,N(C1c2ccccc2CC1NC(=O)C(O)P(C)(C)=O)C(C(OC)OC)=O 14314,c1(OC)c(C(=O)NC2CC(C)CN(C(c3cnc(C)c(N)c3)=O)C2)cccc1Cl 14315,C1(CN(C2CCCN(C(c3c(C)nc(CC)o3)=O)C2)C)CC12CCCCC2 14316,N1(C(CCC=CC(C)C)=O)CCN(C(C2CCCN2C2CCOCC2)=O)CC1C 14317,N1(C(C(C)CC(F)(F)F)=O)CCC2C(CCN2C(=O)C(c2ccccc2)C)C1 14318,C(S(=O)CC(=O)N1CCC(C(=O)NCC(C)C)CC1)c1ccc(COC)o1 14319,C1(NC(CC(=C)C)=O)CN(C(=O)C(C)Oc2cc(C)ccc2Cl)CC(F)(F)C1 14320,Cc1c(C(=O)NC2CC(C)CN(C(C3CCC(C)CC3)=O)C2)cccc1F 14321,C1(NC(c2occ(C(=O)OC)c2)=O)C2CC(CN(C(c3csnn3)=O)C2)C1CO 14322,CCCC(C(=O)NCC(C(C)C)NC(c1cn(CC(=O)N(C)C)nn1)=O)N(C)C 14323,N1(C(CC2OCC(C)(C)OC2)=O)CC2=C(C1)CN(C(=O)COCC1CCC1)C2 14324,N1(C(c2ccc(CC)o2)=O)CCN(C(CNC(C2CC2C)=O)C(F)F)CC1 14325,Cc1ncc(C#N)cc1NC(=O)C(O)CCNC(C1C2CCCCCC12)=O 14326,N1(C(C2CCCCN(C(c3cc(COC)no3)=O)C2)=O)CCC(O)C(C)(C)C1 14327,CC1(C)CC(NC(C2CN(C(c3ccccc3)=O)CCS2)=O)CC(C)(C)O1 14328,C1(C(N(CCC(=O)NC(c2nn(C)cc2O)C)C2CC2)=O)CC2CC(=O)C1C2 14329,C#CCCCC(C)C(=O)N(CCNC(C1CCCSC1C)=O)CC 14330,Cc1cc(F)c(CC(=O)N(C)CCN(C(C2CCCC3CC23)=O)C(C)C)cc1F 14331,C1(C#N)(C(=O)NCC(CNC(c2c(OCC)cccn2)=O)OC)CCCCC1 14332,c1(C(N(CC(C)N(C)C(C2CC3CC3C2)=O)C)=O)ccncc1I 14333,C1(C2CCC2)(C(=O)NCc2cnc(N)s2)CCC1.n1(CC)cc(C(=O)OC)cn1 14334,c1(CN2CC3N(C(c4c(OC)ccc(F)c4)=O)C(C3)C2)cccc(F)c1C#N 14335,C1(CNC(CCOC(C)C)=O)CC(F)(F)CN1C(=O)C(c1ccn(C)n1)C 14336,c1(OC(C)C)cccc(-c2ccc(C(=O)Nc3ccsc3C(N)=O)nc2C)c1F 14337,N1(C(C(C)=C(C)C)=O)CC2CC3CC2C1C3NC(=O)Cc1ccoc1 14338,Cc1ccccc1COC1CC1NC(=O)Cn1cnnn1.N12CCC(C1)C2=O 14339,C1(N(CCCC)C(c2ccc(CO)o2)=O)CCN(C(=O)CNS(=O)(=O)NC)CC1 14340,C1(CNC(C(COC)O)=O)CC2(CO1)CN(C(=O)CSSC)C2 14341,c1(-c2cn(CCC(N3CCN(C4CCSC4)CC3)C)nn2)cc(C)nc(C)c1 14342,c1(C(=O)NCC(C)N(C(=O)Cc2cn(C)nn2)C)ccc2ncnn2n1 14343,Cc1nnc2n1CC(C(=O)NC(CNC(c1nccn3cnnc13)=O)C(C)C)C2 14344,C1(C(N(C2CN(C(Cc3c(C)noc3)=O)CC23CC3)C)=O)CC(=O)N(C)C(=O)N1 14345,C#Cc1cccc(CN2CCOC(C)(NCc3ccccc3I)C2)c1 14346,c1(C(=O)NCC(C)CN(C(=O)C2=CCCC2C)C)cc2c([N+](=O)[O-])cccc2[nH]1 14347,C=C(C)C(CC(=O)NCc1csc(NC(C2CC(OC)C(OC)C2)=O)c1)OCC 14348,C1(NC(c2ncc(OC)cn2)=O)CC(N=c2[nH]nc(C3CCCC3)s2)C1(C)C 14349,C12(CNC(C34CC(CC(C)O3)C4)=O)CN(C(C3SCCCS3)=O)CC1CCO2 14350,O(S(=O)(=O)c1ccc(C#N)cc1)c1ccc(F)cc1F.C(=O)(CON)N(C(C)=O)CC 14351,C(=O)(C1=CC2(CCN(C(=O)CC3COC(=O)C3)C2)C1)NC(CC#C)CC#C 14352,C1(C(N2CC(COC)(CNC(=O)Cc3cnoc3)C2)=O)CCC(C)(C)O1 14353,C12(Nc3snc(C)c3C#N)CCCC1CN(C(=O)C(N1CCCC(C)C1)=O)C2 14354,c1(CNC(N2CCC(C)C2)=O)nc2cc(Cl)c(Cl)cc2[nH]1 14355,O=C(CCCNC(c1ccnnc1)=O)NC1CC1.C1(Cc2ccoc2)C(=O)N1 14356,C(c1cccc(Cl)c1)=CC(=O)NC(c1sc(C(=O)OCC)c(C)n1)C 14357,c1(C(N2CCC(O)(C(C)NC(c3nnc(C)s3)=O)C2)=O)csc2cccnc12 14358,c1(C(=O)NCC2CC(O)(CNC(=O)C(F)C3CC3)C2)cc(F)cc(Cl)c1 14359,CCCC(C(=O)NCCCN(c1ncnc(=N)[nH]1)CC)S(N)(=O)=O 14360,c1(C(=O)NC2CC3CC(NC(c4cncc(C)c4)=O)C2C3)nc2ccccc2[nH]1 14361,c1(C(N2CC(N(C)C)C(C)(C)C2)=O)coc2c1CN(C(C1CCCC(O)C1)=O)C2 14362,C1(C)(C(N2CC(C)C(O)C2)=O)Cc2ccccc2N1.c1(CC)ccc(CC)s1 14363,C1(NC(CCCC(C)=O)=O)CCN(C)C12CCCN(C(C1CCC(=O)N1)=O)C2 14364,Cc1cc(C(N2CCC(O)(CNC(=O)C(F)(F)C(C)O)C2)=O)ncc1C#N 14365,CCC(O)C(F)(F)C(=O)N1CCN(C(=O)CN2CCNC(=O)C2)C(CC(F)F)C1 14366,C1(NC(c2c(OC)c(F)ncc2)=O)CC2(CCN(C(c3sc(C)nc3C)=O)C2)C1 14367,N1(C(C(C)O)=O)C2CCC1CN(C(C1CCN(CC(F)(F)F)CC1)=O)CC2 14368,N1(C(c2cc(N)cc(OC)c2C(=O)OC)=O)CC2CCCC(NC(=O)C(C)Br)C2C1 14369,C(C(=O)NC1C=CC(CNC(=O)Cc2c[nH]nc2O)C1)(C(C)C)OCC(C)C 14370,C1(NC(CC(C(=C)C)OCC)=O)C2CCCN(C(=O)CC3CCSC3)C2C1(C)C 14371,c1(OC)ccc(Br)c(CN2CCCC(C(=O)NCC3CN(C)CCO3)CC2)n1 14372,Cn1nnc2cc(-c3nc(Cc4ccnc(Cl)c4O)no3)cnc12 14373,Cc1cc(N)n2ncc(C(=O)NCC=CCNC(=O)COc3ccccc3)c2n1 14374,CC(C)CC(C)(O)C(=O)NC1CCCC(C(=O)NCC(O)C(F)(F)F)C1 14375,c1(C(N2C3C(NC(c4cnc(COC)s4)=O)CC(C3)C2)=O)cc(F)cc(N)c1F 14376,C1(NC(c2cc(C)no2)=O)CC(Nc2nccc(CO)n2)C1(C)C 14377,O=C(C(O)C(F)(F)F)N1CCOCCC1C(=O)NOCCCC(F)(F)F 14378,CCC(C#N)C(=O)NC(C(=O)NCc1ncc(C)s1)C1CCC1 14379,c1(C(=O)NCC(CC)(C)N2CCOCC2)cc(S(N)(=O)=O)c(Cl)o1 14380,c1(CC(=O)NC2CCCN(C(C34CC(C)C3C4)=O)C2)c(F)cccc1Cl 14381,C=C(CNC(=O)C(c1ccnn1C)NC(c1cc(CO)c(C)o1)=O)C1CCOCC1 14382,C1(N(C(c2cnc(O)o2)=O)CC)CCCN(C(c2cnccc2C(F)F)=O)CC1 14383,c1(NC(=O)NCCc2ccc(C)o2)cccc(N=c2cc[nH]cc2)c1 14384,N1(C(c2c(C)cc(SC)o2)=O)CC2CC(NC(C3CCCC3(C)C)=O)C2C1 14385,C1(CCNC(CSC)=O)CCN(C(c2noc3cc(Cl)ccc23)=O)CCC1(F)F 14386,C1(NC(C(C)NS(CCCC)(=O)=O)=O)CCN(C(=O)CCCC)CC1O 14387,N1(C(CC(C)N(C(C(CCCC)O)=O)C)=O)CC2(CCCCCC2)C1 14388,O=C(C(O)C1CN(C(=O)CC2CSC2)C1)N(CC(O)CO)CCO 14389,C1(C(=O)NCCC2N(C(CSCCCC)=O)CCOC2)CCC(C)=C(C)C1 14390,N1(C(c2n(C(C)C)ncc2)=O)CCCC2(CCC(NC(c3cccnc3)=O)C2)C1 14391,C(=O)(C1=NOC2(CCC2)C1)NC(CNC(C1C(c2n(C)c(S)nn2)C1)=O)(C)C 14392,CC1=CCC(N=c2ccc(Br)c(S(=O)(=O)NC3CCC4(CC4)C3)[nH]2)CC1 14393,C(c1cc(Cl)c2c(c1)OCO2)=CC(=O)NCC(CO)NC(C1(C)CC1(F)F)=O 14394,S(=O)(=O)(c1ccc(Cl)cc1)N(CC(=O)Nc1cnn(C2CCOCC2)c1)C 14395,c1(OC)cc(C(N2CC(C(=O)NC3CCC(C(C)O)CC3)C(C)C2)=O)nn1C 14396,c1(C(=O)NCC2C3CN(C(C(C(C)C)OC)=O)C2C3)cc(Cl)cc2cccnc12 14397,C12(NC(c3cc(C)[nH]n3)=O)CC(CNC(=O)C(C)C(C)C)(C1)OC21CCOCC1 14398,C(=O)(CC(C(F)(F)F)NC(=O)C(n1ccc(C)n1)C)NCCC1ON=C(C)C1 14399,Cn1ncc2cccc(C(N3CCC4CN(C(=O)C#CC5CCC5)CC34)=O)c12 14400,CC1CCN(C(=O)C(C)Cc2cnn(C)c2)CCN1C(=O)C=C1CCN(C)C1 14401,S(=O)(=O)(c1cc(C(F)(F)F)ccc1NCCCC(C)O)N(CC(C(C)C)O)C 14402,c1(C(N2CC=CC(NC(c3cc(CC)ncc3)=O)C2)=O)oc2ccccc2c1Cl 14403,c1(CC)cccc(F)c1C(=O)NCCOCCCNC(C1C(F)(F)C12CC2)=O 14404,C#CCCCCC(=O)NC(Cn1cccn1)C(=O)N(C1CCC1(C)C)C 14405,c1(C(=O)NCc2ccc(C(C)NC(CS(CC)=O)=O)cc2)cnc(O)cc1C 14406,Cc1cc(=O)n(CCC(N2CCC(NC(c3cnns3)=O)C2C(C)(C)C)=O)cn1 14407,C=CCC(CO)NC(=O)CC1(NC(C2CCC(=O)C2)=O)CC1 14408,C1(CN(C)C(C23CSCC2C3)=O)CCN(C(C2CC23CCC3)=O)CC1 14409,C1(C(C)CNC(=O)C(=O)NCC2CC2)CCCN(C(=O)C=CC2CC2)C1 14410,C1(CNC(CCCC#C)=O)COC(C)(C)CN1C(C1CCC(F)(F)C1)=O 14411,C=CC(CCC)CC(=O)NCCC1CCCN(C(C2(C(C)C)CCC2)=O)C1 14412,c1(C(=O)NCCNC(c2c(C)c3c(s2)ccs3)=O)cc2c(s1)CC(C)CC2C 14413,c1(N2C(CNC(c3c(C)cc(C)o3)=O)CCC2)nc2ccccc2s1 14414,n1(CCC)c(CN2CCCC(NC(c3cc(C(C)C)nn3C)=O)C2)nnc1C 14415,N1(CC(C)NC(c2c(C(C)C)c[nH]n2)=O)CCN(C(=O)C(C)(O)C2CCC2)CC1 14416,c1(C(N2CC(NC(CCSCC)=O)C(C)CC2)=O)nn2c(c1C)OCCC2 14417,CCC(CC)(CC)C(=O)N1CCC(N(C)C(c2csc(C3CCCC3)n2)=O)C1 14418,C#Cc1ccc(C(=O)N(C2CCCN(C(c3ccn(C4CCC4)n3)=O)C2)C)nc1 14419,C(CNC(c1c(F)cccc1Cl)=O)(CC(F)(F)F)NC(CC(C=C)C)=O 14420,c1(CNC(=O)C#CC2CCC2)nc2c(s1)CN(C(=O)C=Cc1ccc(Cl)s1)CC2 14421,c1(OC)ccc(S(=O)(=O)NCC2CC(CN(C)C)C2)c2ccccc12 14422,C(CCC(N)=O)(C(=O)NCc1cc(C2CC2)n[nH]1)n1cc(CCN(C)CC)nn1 14423,N(C1CCCn2ncnc21)C(CC(C(F)(F)F)NC(=O)Cc1ccc(O)cn1)=O 14424,CN1N=CC(CC(=O)NC2CC(CCC(N3CCOCC3CO)=O)C2)C1=O 14425,CC1(C=CC(=O)NCC2CCC(NC(=O)CCc3cncs3)C2)CCOCC1 14426,c1(C(=O)NC2CCCN(C(CC(=O)NCC)=O)C2)nc(OC)ccc1F 14427,N1(C(CCC(=C)C)=O)CCC(NC(c2ccc(OC(F)F)cn2)=O)CC1C1CC1 14428,C(c1ccc(Br)cc1)=CC(=O)NC(C)CCCNC(=O)CP(C)(C)=O 14429,N1(C(COCc2cc(C)no2)=O)CCCC1(C)CNC(c1nccs1)=O 14430,c1(SC)nc(N2CCC=C(C(=O)Nc3ccc(C(N)=O)nc3C)C2)c(Br)c(C)n1 14431,C(=O)(C(O)(C(C)C)C(F)(F)F)NCC1(CNC(c2cc(OC)ns2)=O)CC1 14432,CC1CC(NC(c2cccc(Br)c2)=O)CCN1C(=O)CC1CCCCN1C 14433,C#CC1CCC(C(=O)NCCN(C(=O)C(C)N2CC(C)C2)CCOC)CC1 14434,C12(C(N3C4C(CNC(=O)CSc5ccc(O)cc5)C(C4)C3)=O)CCCC1OCC2 14435,C1(O)(CN(C(COCCC)=O)C)CCN(C(C2COC(C)(C)CO2)=O)CC1 14436,C(CC(C(=O)NCC1CC1(C)C)NC(C1CC(CC2CC2)C1)=O)OC 14437,C1(NC(C(CSC)C)=O)CCCN(C(c2ccccc2OC2CCC2)=O)CCC1 14438,Cn1[nH]nnc1=NCCCC(C)(C)NC(C1(c2cccc(F)c2)CC1)=O 14439,c1(C(=O)NCCC(C)N(C(=O)C=C2CCCCC2)C)ccc2c(c1N)CCCC2 14440,c1(CCC)ncc(C(C(=O)NCCC2CC2)N(CCCNC(=O)C(C)C)CC)s1 14441,N1(C(c2ccc(Cl)cc2)C(=O)NCCC#N)CCCN2CCCCC12 14442,c1(C(N2CCC(N(C(CSC)=O)CCO)C2)=O)cc2c(nn1)CCCC2 14443,Cc1nn(C)c(C(=O)NCC(CO)NC(C2CCO2)=O)c1I 14444,c1(C(=O)OC)cc(C)c(-c2nc(CCOC(C)(C)C)nn2C2CCC(C)(C)C2)o1 14445,C(=O)(C(C)(CC)CC)NCc1ccc(C(N(CC=C)CC)=O)o1 14446,C1(NC(=O)CCNc2ccccn2)CCN(C(c2cncc(C(F)F)c2)=O)CC1 14447,N1(C(C2(CC(C)C)CC2)=O)CCN(C(=O)CNC(=O)Cc2cc(C)nn2C)CC1 14448,C1(N(C)CC)(C(=O)NC2CC(CCNC(=O)C(C)OCCF)C2)CCC1 14449,c1(C(=O)NCC(C)(C2CC2)NC(C(CC#C)C)=O)cc(C)ccc1N 14450,c1(OC)cc(C(=O)NC2CC(CCNC(c3cn(C)c(O)n3)=O)C2)nn1C 14451,N1(C(C2C(C)CCC2)=O)CCCCC(Cn2cc(CCc3ccccc3)nn2)C1 14452,O=S(=O)(c1ccc2nc(N3CCC(O)C(F)C3)ccc2c1)N1CCSCC1 14453,c1(CC(=O)NC(C2CCN(C(c3cncnc3)=O)CC2)C)ccccc1S(C)=O 14454,C1(n2c(-c3nnn(-c4ccccc4)c3C)nc(C(C3CC3)OC)n2)C(C)CCCC1C 14455,N1(C(c2c(OC)nc(C)nc2)=O)CCCN(C(c2ccc(F)cc2C)=O)CC1C 14456,c1(NC(CCC)C)cc(=NCCc2cnc3ncccn23)[nH]c(COC)n1 14457,CCCC(CCC)CC(=O)N1CCOCC1CNC(=O)C(C)(CC)CO 14458,CONC(=O)CNC(=O)CCC1CC(NC(c2coc(C(N)=O)c2)=O)C1 14459,C12(NC(C(C)SCCCC)=O)CCCC1N(C(=O)Cc1ccccc1SC)CC2 14460,C1(NC(c2cc(C3CC3)cs2)=O)CCN(C(C2CCCCS2(=O)=O)=O)CC(O)C1 14461,N1(C(=O)COCCCF)CCN(C(=O)CCCSC(C)(C)C)C2CC12 14462,C1CCN(N2CCN(C)CC2)C1.c1(CN(C)C(c2ccsc2)=O)cncn1C 14463,CC(CC#N)N=c1[nH]c(=NCCNC(c2ccccc2Cl)=O)c2sccc2[nH]1 14464,N1(C(c2ccc(Cn3cc(CNC=O)nn3)o2)=O)C(CO)CCC12CCC2 14465,c1(C(=O)NC2CCC(CCNC(C3(CCCC)CC3)=O)C2)cc(C)c(O)c(C)c1 14466,c1(C(=O)OC)cccnc1C(=O)N(CCCCNC(=O)C(c1cccnc1)O)C 14467,c1(C(=O)NCC2(O)CN(C(c3c(C)oc(CO)c3)=O)C2)cnn2c1OCC(C)C2 14468,C(=O)(C(C)CC(C)C)NC1C(C(=O)NC(C(=O)OC)(C)C)CCC1 14469,c1(NCCN(C(C)(C)C)C(C2C(NC(=O)OC(C)(C)C)C2)=O)cc(Br)cc(F)n1 14470,N1(C(C(C)n2cncn2)=O)CC2C(N(C(=O)CCCN(C)C)C)C2C1 14471,c1(CC(=O)NCC2C3CN(C(c4n(CC)ccc4)=O)CC32)nsc2ccccc12 14472,N(C(=S)N1CCC1c1cccc(F)c1)CC.c12cccc(c1)NC2=O 14473,Cn1cc(C(=O)NCC23CC2CN(C(c2ccnn2CC2CCC2)=O)C3)c(Cl)n1 14474,CCC(C)(COC)CNC(=O)CONC(=O)C=Cc1cncs1 14475,C(C)(C)(CC(=O)NC(C)CC(C)NC(=O)CCCCc1cnc[nH]1)OC 14476,C1(C(N2CC(N(C(C(CC)(C)O)=O)C)C2)=O)CC(c2cccnc2)=NO1 14477,C1(OC)CN(C(c2ccn(-c3ccc(Nc4cnn(C)c4)cc3)n2)=O)CC1O 14478,c1(OC)cc(F)c(C(N2CCC(NC(c3cnn4ccn(C)c34)=O)C2)=O)cc1N 14479,C1(CC)C(C(=O)NCc2cccc(OC)c2)CCN1C(c1cnn(C)c1Cl)=O 14480,N1(C(C(F)(F)C2(OC)CCC2)=O)CCC(NC(=O)C2=CCCCC2)CC(C)(C)C1 14481,N1(C(C(C)OC2CCCCC2)=O)CCC(C)C(NC(=O)C(C)(C)CO)C1 14482,CCC(CC)C(=O)N(C)CC1CN(C(c2ncn(C(C)(C)C)n2)=O)CCO1 14483,c1(C(=O)OCC)cnn2c1CN(C(C1CC1NC(=O)CN(C)C)=O)CC2 14484,N1(C(CC(=C)C)=O)CCC2CCN(C(C3CC(C)(C)CN3C)=O)CC12 14485,c1(SC(C)C(=O)N(C2CCN(C(c3coc(C(F)F)c3)=O)C2)C)ccccn1 14486,C#Cc1cccc(C(=O)NC2CCN(C(C3COC3)=O)C(C3CC3)C2)c1Cl 14487,c1(N2CCC(C(CC)CC)CC2)nc2c(c(=NC3CCSC3)[nH]1)CCCCC2 14488,C(C(CO)(CO)NC(c1cncnc1)=O)N(C(C1C(OC)C1)=O)C 14489,c1(C(=O)Nc2ccc(OCC(=O)NCC)cc2)c(C#N)cnn1C 14490,C1(NC(C(CC(=O)OC)C)=O)CC2CCC1CC2NC(=O)CC1(CS(C)(=O)=O)CC1 14491,c1(C(=O)NC23C(CN(C(CC4C(C)(C)CC4)=O)C2)C3)cccc2c1OCCO2 14492,C1(C(N2CC(CNC(c3cc(OC)no3)=O)(COC)C2)=O)CCCCN1C(C)C 14493,C(CC(C)(C)C(=O)N1CCCC(N(C(=O)Cc2csc(Br)n2)C)C1)OC 14494,C1(C(=O)NCCCCC)CCCCCC1NC(C1CCC(F)CC1)=O 14495,N1(C(CN(c2ccccc2)C)=O)CCCC(C(=O)NCC2CC3(CCO2)CC3)CC1 14496,N1(C(c2c(C)coc2)=O)CCCN(C(=O)C(CO)N(C)C)CC1c1ccccc1 14497,N=c1cc[nH]cc1C(=O)NCC(O)CNC(c1ccnc(OCC(F)(F)F)c1)=O 14498,C1(O)(CNC(Cc2cncc(C)c2)=O)CCCN(C(c2nn(C)c(C)c2Cl)=O)C1 14499,c1(CC(=O)NCCN2CCN(C(CSCCCC)=O)CC2)c(C)nc(O)nc1C 14500,Cc1nc(CNC(C2CC2c2ccco2)C)sc1C(=O)O 14501,Cc1c[nH]cc1C(=O)N(C)CCOCCNC(C1CC1CF)=O 14502,C12(CNC(C=CC)=O)CC(NC(=O)CC(CC)SC)(C1)C(C)(C)O2 14503,C1(N)(CC)CCCN(C(=O)C(N2CCCC(N3CCC3)C2)=O)C1 14504,CCCC(CC)CCC(=O)NC12CC(C(N3CC(O)(CO)C3)=O)(C1)C2 14505,CCCCS(=O)(=O)NCC(=O)NC1CC1CNC(c1ccc(C(F)(F)F)cn1)=O 14506,C(=O)(C(CC(N)=O)NC(c1cc(C)n(C)c1)=O)NCCCOCCCC 14507,c1(C(CC)C)nc(-c2coc(C)n2)n(C(C)C(C)(C)C)n1 14508,N1(C(CSCC=C)=O)CCCN(C(C2(C3CC3)CC2)=O)CC1c1ccccc1 14509,N1(C(CN2C(C)CCC2)=O)CC=CC(NC(=O)Cc2ccn(C)n2)C1 14510,N1(C(C(CC(C)C)(F)F)=O)CCOC2(CCC(NC(=O)C(C)(C)CF)CC2)C1 14511,C1(NC(c2c(C(C)O)cccc2)=O)CCN(C(C2CC(O)C2)=O)C(C)C1 14512,C1(C2CCCOC2)(NC(C(CC2CCCC2)NC(C(C=C)OC)=O)=O)CC1 14513,CCC(C)(C)CCCC(=O)NC1CCN(C(c2cc(C)cc(F)c2)=O)C12CC2 14514,c1(OCCCOC)ccc(C(=O)N(CC(O)CNC(=O)C#CC2CC2)C)c(Cl)c1 14515,C1(C(=O)NC2(CO)CCN(C(c3cc(CC)no3)=O)CC2)CCCC1S(C)(=O)=O 14516,c1(C(N(C(=O)CC2CC=CCC2)C(C)=O)=O)cncc2nc[nH]c12 14517,C=Cc1ccccc1NC(=O)CC(=C)C 14518,Cc1c(C(=O)NC2CC2NC(=O)CCC2CCCC2)cc(-c2ccccc2)n1C 14519,N1(C(CC2(OC)CCC2)=O)CCN(C(c2cccc(F)c2O)=O)C2(CC2)C1 14520,N1(CC(=O)N(C)C)CCC2CCN(Cc3nc(-c4ccccc4)n[nH]3)CC12 14521,C1(O)(C(C)NC(COCCNC(c2c(C)scc2)=O)=O)CCCCC1 14522,C1(C(=O)NCCN(C(=O)CO)CCC)CCC(C(F)(F)F)O1 14523,CC1CN(C(C2CC3COCC3C2)=O)CCC1CO.c12nocc1C(=O)NC2 14524,c1(CC(N2CC3(CC(CNC(C(C)(O)C4CC4)=O)C3)C2)=O)csc2ccccc12 14525,Cc1cc(NC(=O)NCc2ccc(C(N3CCOCC3)C)c(Br)c2)cc(C)c1I 14526,N1(C(C(C2CC2)SC)=O)CC2(C(=O)N(CC3=CCSC3)C)CC1CO2 14527,N(C1CC2(CN(C(=O)C=C3CC3)C2)n2ccnc21)C(C1C(=O)NCC1)=O 14528,C1(NC(=O)OCc2nc(CN(C(C)(C)C)C3CC3)co2)CCc2nnc(O)n2C1 14529,Cc1cccc(OCC(=O)NCCC(C)N(C(=O)CCCC#N)C)c1 14530,CCCCC(C(=O)N1CCN(C(c2cc(C(C)(C)C)oc2C)=O)CC1CC)N(C)C 14531,c1(C(C(C)C)Nc2c(O)ccc(C#C)c2)ccc2ccccc2c1 14532,C(=O)(C(C)S(N)(=O)=O)N1CCC(C)(CNC(c2c(C)n(C3CCOC3)nn2)=O)C1 14533,C(=O)(CC1C(=O)Nc2ccccc21)NCC1N(C(CC(C)(C)CC(F)F)=O)CC1 14534,C1(C2CCNCC2)(C(=O)NC(c2ccccc2)C)CCC1 14535,C(=O)(C(C)CC(C)(F)F)N(C(CCNC(CC(C=C)(C)C)=O)C)C 14536,C1(NC(C(=O)N(C)Cc2cccnc2Br)=O)CCCN2CCCCC12 14537,C(=O)(CCCCC(N)=O)N1CCC(CNC(CN2CCCC(N(C)C)C2)=O)CC1 14538,CC1OC2(C(=O)N(CCNC(C3CC(C(F)F)C3)=O)C3CC3)CCC1C2 14539,c1(C(C)(C)C)nc(N2CC=CC(NC(c3ccccc3CO)=O)C2)[nH]c(=N)n1 14540,CCC(C)(C)C(C)CC(=O)NC1CC2CCC1(NC(=O)CN(CC(C)(C)C)C)C2 14541,c1(C(=O)NC(CNC(=O)CNC(N2CCCC2)=O)C2CC2)cc[n+]([O-])cc1 14542,c1(C(C(F)(F)F)N(C(c2ccc(C)o2)C)C(N2CC(F)(F)C2)=O)ccc(O)cc1 14543,C1(NC(C2CC3CCC3C2)=O)CC2(CCN(C(=O)CN3CCCOC3=O)CC2)C1 14544,C1(C(N)=O)CCC(CCC(=O)NCC2CCN2C(c2ccsc2Cl)=O)O1 14545,c1(N(C)C)ccncc1C(=O)NC1COCCC1NC(c1csc(C(N)=O)n1)=O 14546,c1(C(N2CC3(CCN3C(c3cc(Cl)sc3Cl)=O)C2)=O)cc2n(c1)CCOC2 14547,N1(C(CC=CCC)=O)CCCC(OC(N2CCC2C)=O)C1 14548,c1(C(=O)NCC2C=CCN2C(c2cnc(O)s2)=O)coc2c(Cl)cccc12 14549,C1(N(C(CC(=O)NCC#C)=O)C)CCC(Nc2ncncc2I)CC1 14550,c1(CNC(c2c(C)n[nH]c2)=O)ccc(CNC(c2c[nH]c(C(F)(F)F)c2)=O)cc1 14551,C1(C(=O)NCc2c(CNC(c3n[nH]c(C)c3O)=O)cccc2)CC12CCCCC2 14552,C(=O)(C(CCC=C)NC(c1cnn(C)c1)=O)NC(C#C)C 14553,C1(CNC(=O)C=Cc2cn[nH]c2)(NC(C2SCCCS2)=O)CC2CCC1C2 14554,c1(CC)ccc(C(=O)OCC(=O)CC(C)(C)C2CC2)cc1[N+](=O)[O-] 14555,O(NC(=O)C(CCC1CC1)NC(=O)C(C)CC)CC(=O)OCC 14556,CCC(CC(=O)NC1CC(N(C)C(c2cccc(F)c2)=O)C1)SC 14557,c1(CNC(C2(CC)CCN(C(C3C4COCC34)=O)C2)=O)cc(C)nc(O)c1 14558,C1(NC(c2c(C)ncs2)=O)CCCOC12CCN(C(=O)CC1CC=CCC1)CC2 14559,N1(C(CC#N)=O)CCN(C(=O)Cc2noc3ccccc23)CC(CO)C1 14560,C1(NC(C2C(C(C)C)C2)=O)C=CCCC1C(=O)NCc1cn(C(C)C)nn1 14561,CC1CN(C(=O)CCCC2CN(C(=O)CN(C)C)C2)CC1NC(=O)OC(C)(C)C 14562,C1(CNC(C(COC)(F)F)=O)CN(C(=O)C(C)NC(C)=O)C2(CCC2)C1 14563,C(=O)(C(C)(C)CC(C)C)N1CCN(CCCNC(C(CSC)C)=O)CC1 14564,N1(C(CCOC)=O)CCCC1C(C)(C)CNC(C1C(C)C1(F)F)=O 14565,C(=O)(C(C)(C)C(F)F)NC1CC2(C(NC(c3cc(COC)cn3C)=O)C2)C1 14566,c1(CC)ccccc1N(C(=O)C#CCNC(=O)C(C)O)C 14567,C1(NC(C2CC(N(C)CC)C2)=O)CCCC(NC(c2cncc(F)c2)=O)CC1 14568,C12(C(N3CCC(CNC(C4(CC5CC5)CC4)=O)C3)=O)CCCCC1OCC2 14569,C1(CNC(N2C3(C(N)=O)CC(C2)C3)=O)CN2CCC1CC2 14570,c1(C(=O)NCC2N(C(C(C)(C)OC(C)=O)=O)CCC2)cccn2nccc12 14571,CSC1=C(C(=O)NCC2CCCC2NC(c2ccc(C)cc2C)=O)CCCC1 14572,Cc1c(C(=O)NCc2ccsc2C(=O)NCC2CCN2C(C)(C)C)cccc1F 14573,c1(C(N(C)CCNC(c2ccc(N)c(Cl)c2)=O)=O)nsc2ccccc12 14574,c1(N(CCCNC(=O)CC(C)OC)CC)cccc(C)n1 14575,O=C(CCC(CF)CF)N1CCC(CO)C(NC(C2(c3ccno3)CC2)=O)C1 14576,C(CNC(C1CCC1(C)C)=O)(C(C)(C)C)NC(C(C)OC1COC1)=O 14577,N1(C(c2ccc(C)n2C)=O)CCCC2C1CCCN2C(=O)C(F)F 14578,c1(C(=O)NCC2COCCN(C(C(CC(=O)OC)C)=O)C2)cnn2ccncc12 14579,c1(C(N2CC(CNC(CSCCOC)=O)C2)=O)nc(N(C)C)nc(=N)[nH]1 14580,C1(NC(C(C)NC(=O)CC(F)(F)F)=O)CC(O)CN(C(=O)OC(C)(C)C)C1 14581,Cc1ccc(C)c(C(N2CCN(C)C(C(N3CCC(OC4CC4)C3)=O)C2)=O)n1 14582,c1(CC(N2CC(O)(C(=O)NC)C2)=O)ccc(CN(C(CC2CC(=C)C2)=O)C)cc1 14583,c1(OCC(N2CCC(NC(=O)C=CSc3nc[nH]n3)C2)=O)cccc(Cl)c1 14584,CCCN=C(NCCN1CC(C)CC(C)C1)N1CCC(CC2CC2)C1 14585,c1(C(=O)NCC(C(N2CC(C#C)C2)=O)OC)cc(C)n(C)c1C 14586,C1(C)(CC)CC(C(N2CC(N(C(=O)CCc3cc[nH]n3)C)C2)=O)C1 14587,c1(C(=O)NCCN(C(C2CC(OC)C2)=O)C)cccc(C#CC2CC2)c1 14588,C1(O)(CCNC(C2CCCN(C(C)C)C2)=O)CCCN(C(=O)COCCF)C1 14589,c1(C(=O)NC(C)CN(C(=O)CC2CC(=O)NC(=O)C2)C)ccc2cccnc2n1 14590,CC(C)CC(C)(CNC(C1(CF)CC1(F)F)=O)NC(c1cc(CCO)on1)=O 14591,C1(C(=O)NCC(C#C)CC)(CNC(C2CCCN2C(C)C)=O)CC2(CC2)C1 14592,N1(C(CCCCC)=O)CC2CCC(C1)N2C(=O)CC1(O)CCOCC1 14593,C(=O)(C1SCCc2sccc21)N1C2CC(CNC(Cc3c(C)non3)=O)(OC2)C1 14594,N1(C(CCCOCC)=O)CCN(C(C2(CN(C)C)CCCC2)=O)CC1C1CC1 14595,c1(C(=O)NC2CN(C(C3CCCCO3)=O)C2)cc([N+](=O)[O-])c2nsnc2c1 14596,c1(OC)cc(NC(=O)N(C2CNC(=O)C2)C)c(Br)nc1Br 14597,CC(C)CCCCCC(=O)N1CCC(O)(C(C)CNC(=O)C2=CC3C=CC2C3)C1 14598,c1(C(=O)NCCC(C)NC(C2CCC(N=[N+]=[N-])CC2)=O)c[nH]c2cc(O)ccc12 14599,Cc1cc(Br)cnc1C(N1CCCC1CC1CC1)C(=O)NCCC#N 14600,C(=O)(C(C)C(=O)NC(C)(C)CCNC(c1cc(-n2ccnc2C)ccn1)=O)OC 14601,c1(CCC)ccc(C=CC(=O)N(CCC(C(C)C)NC(=O)C(O)CCC)C)cc1 14602,Cc1ccc(F)c(CNC(C2CCC(NC(c3cnc(Cl)c(Cl)c3)=O)C2)=O)c1F 14603,C(=O)(C(F)C(F)(F)F)NCCC1N(C(c2cc(C(C)(C)O)ncc2)=O)CCCC1 14604,CCC(CCCO)NC(c1sccc1CNC(=O)CC(C)SC)=O 14605,N1(C(COC)=O)CC(C)(C)CCC1CNC(=O)CS(=O)(=O)CC1CCCO1 14606,Cc1cnccc1C(C(=O)NCC(C)C)N(CC(N1CCCCC1)C)C 14607,N1(C(c2nc(C)oc2)=O)CC(NC(c2cc(C)c(Br)o2)=O)CCC(O)C1 14608,c1(C(N2CC(C)(C(=O)NCC(CC)(C)Cl)C2)=O)ccc(F)cn1 14609,N1(C(C(CCCC)N(C(N)=O)CC)=O)C(C(N2CCC(O)C2)=O)C2CC(F)C1C2 14610,C1(N(C(C(F)=CCC)=O)C)CCC(NC(=O)CCCC2CCCC2)C1 14611,n1(CC)nc(C(N2CCN(C(C3ON=C(C)C3C)=O)CC2COC)=O)ccc1=O 14612,N1(C(c2cncc(OC)n2)=O)CCCN(C(=O)C2=CCC2)CC1c1ccccc1 14613,N1(C(c2c(OC)cncn2)=O)CC2(CC(NC(=O)CSC(C)C)c3nccn32)C1 14614,C(=O)(CCC(F)(F)F)N1CC(NC(CN2CC(C)(C)C2)=O)C(CC2CC2)C1 14615,N1(C(c2cn(CC)nc2)=O)CCC(C=CC(=O)NCC2(C)CCCS2)CC1 14616,CC1CCC2(CN1C(=O)NCCCn1ccccc1=O)OCc1ccccc12 14617,C=CCCN=C(NCCC(=O)OCC1CCOC1)NCC1(F)CCC1 14618,C1(N(C)C(c2coc(C(F)F)n2)=O)CCN(C(c2cc(Br)n(C)c2)=O)CC1 14619,N1(C(c2c(C(=O)OC)scc2)=O)CCN(C(=O)C=CC(C)C)CC1 14620,CC(C)(C(=O)NCC=CCNC(c1csc(O)n1)=O)C1CCCC1 14621,C(=O)(C(CC(F)F)NC(=O)C=NOC)N(CCSC)CC 14622,c1(C(N2C3C(NC(CCOCC)=O)CC(C3)C2)=O)c[nH]c2cc(OC)ccc12 14623,c1(C(=O)NCCN(C(c2ccc(C(C)C)o2)=O)CC)n[nH]cc1I 14624,C=C1CC2CC1CN2C(=O)CC1CC(C)N(C(c2cnn(C)c2C=C)=O)C1 14625,n1(CC)nc(C)c(CC(=O)NC2C(Cn3cc(C4CC(=O)C4)nn3)C2(F)F)c1C 14626,c1(CN2CCC(O)C(O)C2)ccc2nn[nH]c2c1 14627,C=C(C)C1CCC(C)(O)C(NCCc2ccc3c(c2)CCO3)C1 14628,N(C(=NCC(C)C)N1CCCCC(C)(F)C1)CC1(OCC)CCOC1 14629,C1(NC(C2C(N)CCC2)=O)CCCC(F)(F)C1 14630,c1(C(=O)NCC2CCN(C(C(C)SC)=O)C2)sc2ccccc2c1Br 14631,CC(C)CC(C)(C(N)=O)NC(c1ccc(CNC(C2CCC(=O)N2C)=O)nc1)=O 14632,Cc1cc(=O)oc(C)c1C(=O)NCCCCCN(C)C(c1c(C)cnnc1O)=O 14633,C1(NC(C2(OC)CC2)=O)CCC2CCN(C(c3c(C(F)F)cccc3N)=O)C1C2 14634,C12(CNC(C=COCC)=O)CCCCC1CN(C(c1ccc(SC)o1)=O)C2 14635,CC1CCC(NC(=O)NCc2ncoc2-c2ccccc2)C1 14636,C1(C#N)(C(N2CC(C(C)NC(c3cc(C4CC4)on3)=O)OCC2)=O)CCOCC1 14637,Cc1ccnc(N2CCC(CNC(c3ccc(F)cc3C)=O)C2)c1[N+](=O)[O-] 14638,Cc1cnc2n1CCN(C(=O)C(C)(C1CC1)N(C(=O)CCc1cn(C)nn1)C)C2 14639,C(=O)(C1=CC2CCCC12)NCC1C(C)CCN1C(=O)Nc1cc(F)ccc1Cl 14640,c1(OC)ccc(CCN2CCOC(Cn3ccnn3)C2)cc1 14641,C(c1cncc(O)c1)=CC(=O)NCC(CNC(c1cc(OC)ncn1)=O)O 14642,CCC(CC(=O)NCCC(C)(C)OC)N(C)C(C1CCCC(CF)C1)=O 14643,CC(C)C(F)(F)CC(=O)NC(C)(CNC(c1ccc2n[nH]cc2c1)=O)C1CC1 14644,CC1(C)C(C(=O)NOCC2CCOC2)C1CNC(=O)CCc1nc(O)n[nH]1 14645,Cn1nccc1C(=O)NCC(O)CNC(c1cc(-c2ccncc2)[nH]n1)=O 14646,CC1CC2(CC(NC(C3CC(C)N3C(c3ccc(O)c(F)c3)=O)=O)C2)C1 14647,C=CCCC(C)(C)C(=O)N(C)CCOCCNC(c1nn[nH]c1C(C)C)=O 14648,N1(C(c2nc(CC)oc2)=O)CCCC(C2CCN(c3cc(OC)ncn3)CC2)C1 14649,c1(C(=O)NCCCOCC)cc(Cl)cnc1NC(C)=O.C1(C)C(=O)NCCO1 14650,c1(C(c2nnnn2-c2ccccc2)(C)NCc2cc(Br)co2)ccc[n+]([O-])c1 14651,N1(C(C(CC)n2cncn2)=O)CC(NC(=O)CC2CCN(CCF)CC2)C(O)C1 14652,C(=O)(CCC(=O)N(C)C(C)C)NC(CNC(COc1cc(C)on1)=O)C.COC 14653,C(C)(C(=O)NCC1(CCN(C)C(C2(NC(=O)NC(C)(C)C)CC2)=O)CC1)CC 14654,c1(CC(=O)NC2CC(NC(=O)Cc3cnn(C(F)F)c3)C2)ccc([N+](=O)[O-])cc1 14655,C1(C(N2CC3C(CN(C(Cc4cc(C)on4)=O)C)C3C2)=O)CC2OC(=O)OC2C1 14656,C12(C(N3C(CC(NOCC(N)=O)=O)CCC3)=O)CCCC1C2(F)F 14657,Cc1ccc2nc(C(N3CC(O)CC3CNC(C3(C)CC=CCC3)=O)=O)cn2c1 14658,C(=O)(CC(CC)C(C)(C)C)N(CC=CC(=O)NC(C=C)C)C 14659,N1(C(c2cn(CCC)nn2)=O)CC2=C(C1)CN(C(c1ccc[nH]1)=O)C2 14660,C(CNC(C1CC2(CSC2)C1)=O)(CC(F)(F)F)NC(C=NOC)=O 14661,CC(C)(C)C(CO)C(=O)N1CCCC1CCNC(=O)CC1C=CCC1 14662,C12(C(N(CC(C)N(C(COCCCOC)=O)C)C)=O)CCC(F)(CC1)C2 14663,n1(CC(=O)NC2C3CC(NC(C4CC4[N+](=O)[O-])=O)CC23)ncccc1=O 14664,C(C)(C(=O)NCCC1(OC)CN(C(=O)Cc2ccccc2SC)C1)(C(C)C)OC 14665,C1(CNC(c2ncn(CC)c2)=O)CCCCN1C(=O)CCn1ccnn1 14666,N1(C(c2ccc(C#C)cn2)=O)C2CCC1CN(C(c1ncc(C)cc1OC)=O)C2 14667,C12(COC)CC(CNC(C3C=CCC3)=O)(CN1C(c1ccccc1CC#N)=O)C2 14668,C1(NC(c2scc(COC)c2)=O)CN(C(=O)CC(C)F)C2(CCCC2)C1 14669,C1(OC)CCCCC1NC(=O)C(C1CCN(C(C2CCNC2=O)=O)CC1)C 14670,O=S(CC(F)(F)F)N1CCCC(CNS(=O)(=O)Cc2ccccc2)C1 14671,CN1CCCC(C)(C(=O)N(C)CCNC(=O)C=CCN2CCCC2)C1 14672,C1(NC(C(CCSC)OC)=O)CCCN(C(=O)C(C)C(C)c2ccccc2)CC1 14673,N1(CCC(=O)NC2CC(CNC(CN3CC(C)(C)C3)=O)C2)CCC(O)CC1 14674,c1(C(N2CCN(C(c3c(C)nc(CO)o3)=O)CC2C)=O)cc2cc(Cl)ccc2[nH]1 14675,C#CCCCCCC(=O)NCC(CCOC)NC(=O)CC1C(=O)NN=C1C 14676,C#Cc1cc(C(N2CCCCC2CCN(C(=O)C(O)CC2CC2)C)=O)ccc1Cl 14677,C1(CC(=O)NCCN(C)CC)CN(C(c2cn3c(n2)CCC3)=O)CCC1C 14678,C1(C(N2CCCC2C(F)(F)F)=O)CCCN(Cc2ncccc2Br)C1 14679,c1(NC2(CNC(CC(c3ccc(C)cc3)C)=O)CC2)ccc([N+](=O)[O-])cn1 14680,c1(C(=O)NCC(C)CNC(C2CCN(C3CC3)C2=O)=O)c(F)cncc1Br 14681,c1(C(=O)NCCC2(C(=O)NCC(CC)(C)OC)CCC2)cc(C#N)c[nH]1 14682,C#Cc1cccc(NC(C2(NC(=O)COC(C)CC)CC2C)=O)c1 14683,c1(CC)ccc(C(N2CC(NC(c3cccc(O)n3)=O)C(SC)C2)=O)c(Cl)c1 14684,CCC(C)(CC)C(=O)NCC(C)(CO)NC(c1cnc(C(C)OC)s1)=O 14685,S(=O)(=O)(c1cccc(=NCC2CC(C)C2)[nH]1)NC1C(CCCC)CCC1 14686,c1(OC)ccncc1C(=O)NCC1(CNC(c2cc(F)cs2)=O)CC1 14687,C1(OC)CC(C)CN(C(=O)CC(C)CNC(C2(F)CCC2)=O)C1 14688,c1(CC)ccoc1C(=O)NCC1CCCC1NC(=O)CNC(=O)NC 14689,CC1CN(C(c2ccnnc2O)=O)CC1NC(C1(Cl)CC1(F)F)=O 14690,C#Cc1cnn(C)c1C1(C(N2CC=CC(O)C2)=O)N(C(=O)NC)CC1 14691,C1(C(=O)NCC(CC(C)C)NC(=O)COC2CCOC2)CCc2nnn(C)c2C1 14692,N1(C(C(CC)CCOC)=O)CC2(C=C(C(=O)N3CCC(O)CC(C)(C)C3)CO2)C1 14693,c12cc(ccc1Cl)OC2=O.C(C(=O)OC)(C(C)C)N(C)CC 14694,c1(C(=O)NCC2(CNC(CC#N)=O)CCC2)ccc(Oc2cccc(F)c2)nc1 14695,C1(C(N(CCC(C)NC(c2coc(Br)n2)=O)C)=O)C2COCC12 14696,N1(C(C(C=C)OC)=O)CCCC1(C)C(=O)NC(c1ccccn1)C 14697,C1(NC2(C(=O)Nc3cn(CC#C)nc3)CC2)CC1C1CC1C 14698,c1(C(=O)NCC(C2CC2)NC(=O)C=CBr)cc(Cl)ccc1F 14699,CC(C(=O)N1CCN(C(=O)CCC2CC2)CC1CCO)C(C)(C)C 14700,C1(CNC(CC(c2cccc(F)c2)C)=O)CCCCC1NC(C1(Cl)CC1)=O 14701,c1(C(C)C)cccc(C(=O)NC2CC(N(C)C(c3ccc(C(C)C)o3)=O)C2)c1O 14702,c1(C(N2CCCC(C(C)=O)C2)=O)cc(F)ncc1NS(C)(=O)=O 14703,c1(C(=O)NCCC2(OC)CN(C(c3c(CC)csc3)=O)C2)cc(C)ncc1C 14704,C12(CNC(C(CC)N(C)C)=O)CCC(CC1)N2C(c1nncn1CC)=O 14705,Cc1sc2ncnc(NC3CCCC4(CCOC4)O3)c2c1C.c12csc(n1)CNC2 14706,N1(C(CN(C(=O)OCC)C)=O)CCN(C(c2sc(C)cc2Cl)=O)CC1C(C)C 14707,c1(C(N(C(CC)CC(=O)NCCc2ncon2)C)=O)ccc([N+](=O)[O-])[nH]1 14708,S(=O)(=O)(c1cnc(NCc2ccsc2)c(Cl)c1)N1CCCC(C(F)(F)F)(OC)C1 14709,C(=O)(C(CC(C)(C)C)NC(c1cscc1C)=O)NCC(CC(=O)OC)O 14710,N1(C(C=CC)=O)CCN(C(C2C3CN(CC(F)(F)F)CC23)=O)CC1CCO 14711,CCC(C)CCC(O)CC(=O)NCCC(C(C)C)NC(=O)C(C)(C#N)CC 14712,C(C1CCCN1C(=O)CC1CCC1)=CC(=O)NCCCc1cccs1 14713,N1(c2cncc(-c3c(F)ccc(N)c3)n2)CCCC2(CC=CCO2)C1 14714,N1(C(c2cnc(C)o2)=O)CCCN(C(=O)C=Cc2cn[nH]c2)CC1C 14715,c1(C(N(CCC(C)NC(C2CC(N(C)C)C2)=O)C)=O)cc(CO)[nH]n1 14716,CC1(CNC(=O)C(O)c2ccsc2)COCCN(C(c2cc(C#N)c[nH]2)=O)C1 14717,c1(C(N2CCOCC(NC(=O)CC3CCCC4CC34)C2)=O)cnc2occc2c1 14718,C#CCC(C)(C(=O)N1CC=CC(O)C1)NC(C1(C#N)CCCCC1)=O 14719,c1(CC(=O)NCCCCCNC(C2CC2C(F)(F)F)=O)cc(O)cc(Br)c1 14720,Cc1nn(C)c(C)c1CC(N1CCC(O)(C(C)NC(c2c(Cl)nsc2Cl)=O)C1)=O 14721,C(C1CN(C(C2OCCC2C)=O)CC1C(=O)N(C)Cc1cscn1)=CC 14722,C(C(C(F)(F)F)OC)NC(c1scc(CNC(C(C)OCCCC)=O)c1)=O 14723,C1(C(=O)NCC(C)NC(C2(c3cncn3C)CC2)=O)C2C3CCC(C3)C12 14724,C(=O)(C1=CCC(C)(C)CC1)N1CCC(C(N2CC(F)(CC)C2)=O)(CC)C1 14725,C(=O)(C(C)C(O)C(C)C)NC(CNC(CN(C1CC1)CC)=O)Cc1ccccc1 14726,c1(OC)cc(C(=O)N(CCC(C(C)C)NC(C2CCO2)=O)C)c2c(c1)CCCC2 14727,c1(CCC(=O)NCCN(C(=O)CSCc2ncccn2)CC)ccc(Cl)cc1 14728,C(C)(C)(CC(=O)NCc1ccc(C(C)(C)CNC(c2occc2C)=O)cc1)OC 14729,Cc1c(C(N2CCC2CNC(=O)CCSc2ccccc2)=O)c(C(F)F)nn1C 14730,C1(C)(C(=O)NC(C)CC2CN(C(=O)Cn3cnc(=N)[nH]3)C2)CCC(C)(C)CC1 14731,N1(C(c2cccc(F)c2)=O)CCC2(CCN(C(=O)OCc3ccccc3)CC2)C1 14732,C#CC1(C(=O)N(C(CCO)C(F)F)C)CCN(C(c2c[nH]cc2C)=O)C1 14733,CC1=C(C(=O)NCC(C2CCCC2)NC(C2CCC(C)NC2=O)=O)CCO1 14734,C1(NC(C2(C)C(C(=O)OC)C2)=O)CC(NC(=O)CC2CCOC2(C)C)C(O)C1 14735,C(c1ccc(C2CC2)cc1)=CC(=O)NC1CCCCC1NC(C1(CCF)CC1)=O 14736,c1(C(=O)NC2C(OC)CN(C(C(F)OC)=O)C2)ccn2cncc2c1 14737,CC1=C(CC(=O)N(C)C(c2ccccc2)C2CCOCC2)c2ccccc2C1 14738,C(=O)(CCCC(C)(C)C)N1CC(C)(CNC(c2c(C)n(C3CC3)nc2)=O)C(C)C1 14739,CC1(C)CC(NC(c2cccc(C(N)=O)n2)=O)CN1C(c1ccc(Cl)cn1)=O 14740,C(=O)(CC(C)(C)C(=O)NCC1C2CN(C(=O)C(C)OCC(C)C)CC12)OC 14741,N1(C(COC(C)(C)CNC(=O)CCC2CCCC2)=O)CCOC(C#N)C1 14742,C1(NC(CC2N(C)CCC2)=O)CC2(C1)CC2NC(=O)CCC1CCCCCC1 14743,CC(C)(C)CC(O)C(=O)NCCCCCNC(C1CCCCC1C(C)(C)C)=O 14744,c1(OC)nccc(C(=O)N(C)CCNC(C2CCCN2C)=O)c1Br 14745,C(=O)(CCCC(CC)NC(C1CCCO1)=O)NC(CC=C)(C)C(F)F 14746,N1(C(CNC(CC)=O)=O)CC(CNC(=O)Cc2ncccc2C)CC1(C)C 14747,Cc1cc(C(N2CCOC(C(C)NC(C3(C#N)CC3C(F)(F)F)=O)C2)=O)nn1C 14748,C(=O)(C(F)(F)C(C)(C)O)N1CCC(O)(CN(C(=O)CC2(O)CCCOC2)C)CC1 14749,N1(C(CC(CC(C)(C)C)O)=O)CCc2sccc2C1CNC(C1CC(F)(F)C1)=O 14750,c1(C(=O)NC2(C)CCN(C(CCc3ccc(C)s3)=O)C2)ccc2c(c1)C(C)CO2 14751,C(CCN=c1[nH]ccc(=NC2CC3(C2)CC(C)(C)C3)[nH]1)OCC=C 14752,C(c1ccccc1)=CCOCC(=O)OCCO.N1(N(C23CC(C)(C2)C3)C)CCC(C=O)C1 14753,N1(C(C(C(C)C)NC(C)=O)=O)CCC(C)C(NC(c2snc(Cl)c2Cl)=O)C1 14754,C1(C(=O)Nc2c(-n3cccc3)ccc(OC)c2)CC2CCC(C1)C2O 14755,CC(O)(CC(=O)N1CCCCC1CNC(c1cc(Br)sn1)=O)C(F)(F)F 14756,C1(CNC(c2n(C(C)C)ncc2)=O)CN(C(=O)CN2C(=O)CCC2=O)C2CC12 14757,c1(CC(N2C(CCC(=O)Nc3ncc(Br)cc3I)CCC2)=O)cc(F)ccc1Br 14758,S(=O)(=O)(c1ccc(C)cc1)NCC(=O)NCC(CCCC)NC(=O)C=CSC 14759,c1(NC(N2CCOC(C(F)F)C2)=O)ccc(-c2cnco2)cc1 14760,N1(C(C2C(=O)NCC2)=O)CC2CN(C(=O)C=CC(F)(F)F)CC(C1)O2 14761,c1(C(=O)NC(C(C)NC(c2ccc(F)cn2)=O)(C)C)cn2cc(Cl)cc(Cl)c2n1 14762,Cc1cc(N2CCCC(CCF)C2)ncc1S(=O)(=O)N1CCOCCC1C(C)C 14763,c1(OC)cncc(CCC(=O)NCc2ncoc2CCNC(=O)C(CC)OC)c1 14764,N1(C(c2c(C)ccs2)=O)CCC2(NC(=O)C(c3ccc(Cl)s3)=O)CC2C1 14765,C1(C(=O)NC2CCCC(CC(=O)N(CCCCCO)C)C2)(CC)CCNC1=O 14766,C#Cc1ccc(NC(C2CCCN(C(=O)Nc3cc(F)ccc3C)CC2)=O)cc1 14767,CC(C)C(F)C(=O)NC1CCC(C(=O)NCCC2CCCN2C)C1 14768,c1(C(=O)NC(C(C)NC(c2nc(C(C)OCC)sc2)=O)C)cnn(C)c1C 14769,C(CC(=O)NCc1cccc(F)c1F)(C(F)F)NC(CC(C=C)C)=O 14770,C1(CCC(=O)NC23C(CN(C(C(C=C)(F)F)=O)C2)C3)CCc2ccccc2C1 14771,C1(S(N)(=O)=O)(C(=O)NC(CCCC)CNC(=O)CNC(=O)C2CC2)CCCC1 14772,N1(C(C2C(C)OCCC2)=O)CCOC2(CCN(C(=O)Cc3cnccc3Cl)C2)C1 14773,N1(C(c2c(C)nc(CNC(C3CC(C)CO3)=O)o2)=O)CCN(C)CC1C1CC1 14774,N1(C(=O)CCc2ncccn2)CCC(O)CC1C(N1CCC(N2CC=CC2)C1)=O 14775,C#CCC(C)(C(=O)N1CCC(C(=O)NC)C1)NC(c1cc(CO)c(C)o1)=O 14776,c1(C(=O)NC(CC=C)CNC(=O)CNC(c2cccs2)=O)cc([N+](=O)[O-])oc1C 14777,c1(OC)ccc2c(C)c(C(N3CC(C(C)NC(=O)CCCC(N)=O)C3)=O)[nH]c2c1 14778,O=C(C1CCCc2scnc21)NC1CCN(C(C23CCCCN2CCC3)=O)CC1 14779,CC(C)(C)C(CNC(c1ccc2nccn2c1)=O)C(=O)NC1(CO)CC(F)(F)C1 14780,CC(CCCC(=O)NCC1(C#N)CCC1)NC(c1ccc(F)c(O)c1)=O 14781,Cc1nccc(C(=O)NC2(C(=O)NCc3ccc(Cl)cc3)CCN(C)C2)n1 14782,C=CCCCC(=O)NC1(CNC(=O)CCN2CCCC(C(N)=O)C2)CCOC1 14783,Cc1ccc(C)c(C(=O)NC(C)CNC(c2nccc(Cl)c2F)=O)c1 14784,N1(c2nnc(CCC)s2)CCCC(C2CC2NC(=O)CCNC(=O)CC(C)C)C1 14785,Cc1ccc(CN2CCC(O)(CC(=O)NCCC(C)CO)CC2)c(F)c1F 14786,Cc1ccc(CNC(=NCc2cccs2)NC(c2ccn(C)c2)C)nn1 14787,C=CCC(C)(CC)C(=O)NCC1(O)CCCN(C(c2oc(CC)cc2C)=O)CC1 14788,c1(NCc2cc(C)ncn2)nc(N2CCCC(CO)C2)nc2c1ncn2C(C)C 14789,c1(-c2n(-c3ccn(C)n3)nc(-c3ccc(Br)cc3)n2)cccc(C#CC2CC2)c1 14790,CC(C(=O)NCC1CC(NC(c2cc(CCCO)on2)=O)C1)C(C)(C)C 14791,C1(C(=O)NC(C(C)C)CNC(c2occc2CN(C)C)=O)COC(=O)N1C 14792,CSC1=C(C(=O)NCC2CC3CN(C(=O)C(C)(O)CC(C)C)CC23)CCCC1 14793,c1(C(N2CC(CCCCNC(C3C(OC)CCC3)=O)C2)=O)c(O)ncnc1O 14794,c1(C(=O)NC2CCC(NC(c3ccncn3)=O)C2)cccc2nscc12 14795,N1(C(C(C(C)C)SC)=O)CCN(C(=O)CCn2ccnc2)C(CF)C1 14796,N1(C(COC)=O)CCOC2CCN(C(c3cccc(C4(F)CC4(F)F)c3)=O)CC12 14797,C(=O)(CCC(=O)NCC1(NC(C2SCC=C2C)=O)CCCCC1)OC 14798,c1(C(CC)=O)ccc(C(C)(C)NC(=O)CC2CCCN2C(C2CC(C)(O)C2)=O)cc1.C 14799,CCCCN=C(NCc1c(SC)cccc1F)NCC1(C)CC2CC2C1 14800,c1(C(N(CCNC(C(C(=O)OCC)(C)C)=O)C)=O)cc2n(n1)CCN(C)S2(=O)=O 14801,c1(OC(C(=O)NCCC(C)(C)NC(C(=Cc2cnc[nH]2)C)=O)C)ccc(F)cc1 14802,n1(CC(=O)NC2CCC2NC(=O)CC2(CO)CCCCC2)nc(O)ccc1=O 14803,c1(OC)cn(C)c(C(=O)NCCN(C(=O)CCCCC2CCCCC2)C)cc1=O 14804,N1(C(c2c(CC)c(C)sc2)=O)CCN(C(=O)C(C)(C)CC)CC1CS(C)(=O)=O 14805,C1(C(=O)NCC2CCN(C(=O)C(c3cccc(C)c3)C)C2)(CC)CCCCC1 14806,N1(C(c2ccc(C)cc2N)=O)CCCC(O)(CNC(c2cnncc2C)=O)CC1 14807,C1(C(=O)NCC2(OC)CN(C(C3(F)CCOC3C)=O)C2)C2CCC1(C)C2(C)C 14808,c1(C(=O)NCCC(C)N(C(CCCC(=O)OC)=O)C)cccc2c1CCO2 14809,CC1=C(C(=O)N(CCCNC(=O)C(F)n2ccnc2)C(C)C)C(=O)OC1(C)C 14810,C1(CN=[N+]=[N-])CCCCN1CC1CCCN1 14811,C1(C(=O)NCc2cc(C(=O)NCC(COCC)O)ncc2)C2C3CCC(C3)C12 14812,N1(C(C=CCOC)=O)CC(NC(=O)CC(C)C(C)(C)CC)C2(CCOCC2)C1 14813,C1(F)(CNC(c2cc(CC)no2)=O)CCCN(C(C2CCCCCCC2)=O)CC1 14814,C(CC(C)(C)C(=O)NCCC(C(C)C)NC(C12CCC(CC1=O)C2)=O)OC 14815,c1(C(C)NC(=O)NCC2CC(=C3CCC3)C2)cc(Br)ncc1F 14816,CCCCCC(=O)NC1CC1CNC(=O)CN(c1ccc(Br)cn1)C 14817,O=C1CC(CCCN2CC3CC2C2CC32)C12CCC2 14818,C1(NC(CC2CCC(=O)N2)=O)CCN(C(=O)CCc2cccnc2F)CC1C(=O)O 14819,Cc1ccc(F)cc1C(=O)NC1C2CC3C(C2)C13C(=O)NC1CN2CCC1CC2 14820,C1(C(N(CC(CC)NC(=O)CN(c2ccncc2)C)C)=O)C(C)(C)C1(F)F 14821,N1(C(CC2CCCN(C(c3cccc(SC)c3)=O)C2)=O)CCC2CCC(C1)N2C 14822,N1(C(CCCC(=O)NCCC)=O)CCC2(CCN(c3cc(C)ncc3C#N)C2)C1 14823,C1(C(=O)NCCNC(COCCC)=O)CCCC(C)(C)C1 14824,C(CCN=c1[nH]c(=N)[nH]c(=NCc2csc(C(=O)N(C)C)c2)[nH]1)(C(C)C)OC 14825,c1(C(=O)NC2CN(C(Cn3c(C)csc3=O)=O)CC2C)cnc2ccc(F)cn12 14826,N1(C(c2ccc(OCCO)cc2)C(=O)NC(CC)(C)C)CCOC2(CCCCC2)C1 14827,N1(C(c2c(CC)oc(C)c2)=O)CCC(NC(=O)C(F)C2CCC2)C12CCCC2 14828,C1(CN(C(=O)CC(C)(C)O)C)CC(F)CN1c1nnc(CO)s1 14829,C1(C(=O)NCC(C)NC(c2ccn(CCC(F)(F)F)n2)=O)CS(=O)(=O)CCO1 14830,C1(C(=O)NC2(CC)CC(C)(C)C2)CN(C(=O)C=Cc2ccncc2)CC1C1CC1 14831,c1(-c2scc(C(=O)NC3CNCCC3(F)F)n2)cc(F)c(F)c(F)c1 14832,C1(S(C)(=O)=O)(C(N2CCCC(CN=c3nc(CC)[nH]s3)C2)=O)CCCC1 14833,C12(C(N3CCC(N(C)C(C4CC=CCC4)=O)C3)=O)CC(C#N)(C1)C2 14834,c1(OC)nccc(C(=O)NC2COCC2C(=O)N(C(C)(C)C(=O)OC)C)n1 14835,C1(C(N2CCC(N(C(Cc3c(C)non3)=O)C)C2)=O)CCCC(=O)N1C 14836,CC1CCN(S(=O)(=O)CC(=O)NC(C)(C)CCCNC(C2(O)CCCC2)=O)CC1 14837,C(C)(CNC(c1nc[nH]c1C(C)(C)C)=O)(CNC(=O)C(C)=C(C)C)OC 14838,c1(NC(CC(C)SC)=O)cccc(NC(=O)C(=O)NC(C2CCCC2)C2CC2)c1 14839,Cc1cccc(CS(=O)(=O)NCCN(C)CCNC(=O)C#CC(C)C)c1 14840,C(=O)(C(C)CN(C)C(C1CCC1C)=O)N1CC(CSC)C1 14841,c1(NC2CCN(C(C(C(C)(C)C)NC(C)=O)=O)CC2)nc(C)c([N+](=O)[O-])cc1Cl 14842,N1(C(C2CN(C)C(=O)N2)=O)CC2CCC(C(=O)NCC(C)(C)CO)(C2)C1 14843,C1(CNC(CCC)=O)CC2(CCOCC2)CN1C(c1cc2cc(Br)sc2[nH]1)=O 14844,C(CC(=O)N(C1CN(C)C1)C)(C(F)(F)F)NC(C(CC(C)C)O)=O 14845,C1(CCOC)(NC(c2ccsc2Cl)=O)CCN(C(C2OCCC2C)=O)C1 14846,N1(C(C(C=C=C)C)=O)CCC2(CC1)CN(C(c1cnc3c(c1)COC3)=O)C2 14847,C1(CNC(CCOCCC)=O)CN(C(c2c(N)cc(C)cc2F)=O)CC(C)(C)O1 14848,N1(C(CCCN(CCC)CCC)=O)CC(CNC(=O)CCC(C)(C)F)CCC1C 14849,C1(C(=O)NC2CC(c3ccccc3)(NC(C=CC=CCC)=O)C2)C2CCCOC12 14850,C(=O)(C1=NOC(CC2(O)COC2)C1)N(CC(C)O)CCNC(=O)CC(F)(F)F 14851,c1(C(=O)NC2CCN(C(CC(C)(C)C#N)=O)CC2O)cc(Cl)ccc1[N+](=O)[O-] 14852,C(=O)(C(CCC(N)=O)n1cc(CO)nn1)ONC(=O)OC(C)(C)C.C(CCC(C)CO)NC 14853,c1(CC)nn(C)c(CC)c1C(=O)NC1CN(C(=O)CC2CC3CC3C2)CC1C 14854,C1(NC(CC(C=C)C)=O)CN(C(=O)CC23CCCN2CCC3)CCC1F 14855,c1(OC)ccc(C(N2CC(CCNC(C3CCSC3)=O)C2)=O)c(OC(F)F)c1 14856,c1(C(N2CCC(CC#C)(C(=O)NC(C)CF)C2)=O)cccc2c1CCC2 14857,Cc1cc(C(=O)NCC2CCN2C(=O)C(F)CC2CC2)sn1 14858,Cc1c(CC(N2CC(NC(=O)Cn3cncn3)CC2C)=O)sc2ccccc12 14859,c1(OC)ccc(Br)c(C(N2C3CCC2C(C(=O)NC24CC(F)(C2)C4)C3)=O)c1 14860,c1(NC)cnncc1C(=O)NCC(C)NC(c1cncn1-c1ccc(Cl)cc1)=O 14861,C1(CC(=O)NC23CC2CN(C(=O)C(C)(C2CC2)OC)C3)(OC)CCCCC1 14862,C(c1cccc(F)c1)=CC(=O)N(CCCNC(C1(C)CC2CC2C1)=O)C 14863,c1(C(=O)NC(C(C)C)CNC(=O)C=CCF)cc2cc(Cl)cnc2[nH]1 14864,CC1CCC(C)(C)N1C(=O)CNC(=O)C(C)(C)C.c12cnc(nc1)-n1cc-2nn1 14865,N1(C(CNC(CCCCC)=O)=O)CC(NC(=O)Cc2ccc(C)nc2)C2CC2C1 14866,Cc1ncn(C)c1C(=O)NOCc1cn(CC2CC(F)(F)CO2)nn1 14867,N1(C(C(CCC)C)=O)CC(NC(c2cnc(N(C)C)c(Cl)c2)=O)CC2(CCC2)C1 14868,CC1(C)CC=C(c2ccc(NC(C3(O)CC3)=O)cc2F)CC1 14869,CCC(CC)C(C)C(=O)N(CC(=O)N(C1CC(O)C1(C)C)C)C 14870,c1(CNC(C(N2CCC(C)C2C)c2c(CC)cco2)=O)ccccc1C 14871,c1(C(=O)NC(C)CCN(C(=O)CCC2CCCCO2)C)ccnc2ccsc12 14872,C=C(C)C1OCCC1C(=O)NCCCN(C(=O)COCCCF)C(C)C 14873,c1(C(N(CC(C)NC(C2CSCCS2)=O)CC)=O)cnn(CCN(C)C)c1C 14874,CC(C)(CCC(=O)N1CC(NC(C2CCC(CN(C)C)O2)=O)C2(CC2)C1)[N+](=O)[O-] 14875,Cc1ccnc(O)c1C(=O)N(C)CC1CCN(C(=O)CCc2cnn(C)c2)C1 14876,c1(C(=O)NCC2CC(NC(CCC(C)(F)F)=O)C2)ccc2c(c1)CCCS2 14877,C(=O)(CC1OCCc2sccc21)N1CC(C)(NC(c2cc3sc(Cl)cc3[nH]2)=O)C1 14878,CC1OCCC1N=c1[nH]c(N2CCOCC2)nc(=NCC2CC(O)C2)[nH]1 14879,C1(NC(=O)CC2CSCCS2)CCCC(CNC(c2cc(Cl)c[nH]2)=O)C1 14880,c1(C2N(C(c3cc(C4CC4)no3)C(=O)NCCOC)CCC2)cccc(Cl)c1 14881,c1(C2C(NC(=O)CC3CCN(C(=O)NC4(C(F)(F)F)CC4)C3)C2)ccncc1Cl 14882,Cc1cnc(NC(C(C)C)C2CCC2)c(S(=O)(=O)NCCCCS(C)=O)c1 14883,c1(OC)ccncc1C(N1CC(O)(C(F)C(=O)NCc2nccnc2C)C1)=O 14884,c1(OC)ccc(C(N2CCN(C(=O)C=CC(C)(C)C)C(CCOC)C2)=O)nc1Cl 14885,C1(C=O)CC2(CC2)CN1C.N1(C(C(C)NCCC)=O)CCC(C(C)(C)O)C1 14886,c1(OC)ccc(OC)c(CNC(c2cccnc2N(C)CCO)=O)c1.N12CC(C1)C2 14887,CC1(C(=O)Nc2ccc(NC(=O)C3CC3)cc2)Cc2ccccc2NC1=O 14888,c1(C(=O)NCCC2(C)CCCC2)ccc(I)c(F)c1 14889,O(C1CCCc2ccccc21)CCNC(CCC1(C#N)CCOCC1)=O 14890,C1(C(N2CC(O)(C(C(=O)NC3CC(N(C)C)C3)F)C2)=O)CCOC(=O)CC1 14891,CC#CCC(C(=O)NCCC(O)CCC)NC(=O)CN(C)C(C)C 14892,CCC(C)C(O)C(=O)NCCCCCN(C(=O)C(C)SC(C)C)C 14893,CCC(C)C(=O)C(=O)N(CCCNC(=O)C(N1CCCCC1)C)C 14894,C1(NC(C2(CC=C)CC=CC2)=O)CC2CC1CN(C(=O)C(C)(C)C(C)(C)C)C2 14895,c1(C(N2CC(C)C(NC(=O)CC3(C)CC3)C2)=O)ncnc2c1c(Br)cn2C 14896,C1(NC(c2c(Cl)cc(C)s2)=O)CCOC12CCN(C(=O)C=Cc1ccsc1)CC2 14897,C1(CNC(C(C)=C2CCC2)=O)CCCCN(C(=O)CC(C)N(C)C)C1 14898,C(=O)(CCCCCC#N)N1CCC(NC(C(C)(O)c2ccccc2)=O)C(O)C1 14899,C1(C(N2C(CNC(c3c(C)n(C)nn3)=O)C=CC2)=O)CC12CCS(=O)(=O)CC2 14900,Cc1cccc(CNC(c2c[nH]nc2CCNC(=O)Cn2cc(C)cn2)=O)n1 14901,c1(C(=O)NCC=CC(=O)NC(C#C)C2CC2)c[nH]nc1[N+](=O)[O-] 14902,Cc1ccc(C(N2CCC(C)C2C(N2CC3CC2(C(N)=O)C3)=O)=O)cc1C#N 14903,c1(C(c2n(CC(=C)C)nnn2)NC(C)Cn2ccnc2C)cc(Br)ncc1F 14904,c1(CC)nc(N2CCCC(NC(c3cc(C)ccc3C)=O)C2)cc(C)n1 14905,C(N=c1[nH]c(N2CCCN3CCCC3C2)nc2c1SCC2)C1CCC(C)(C)CO1 14906,C1(NC(CCC(C)O)=O)CC2CCCC(C1)N2C(=O)Cn1cnc(=N)[nH]1 14907,c1(C(=O)NCC2(O)CN(C(CCCCSC)=O)C2)ccc2nn(C)cc2c1 14908,C1(CC(=O)NC2CN(c3cc(CC)ncn3)C(C)C2)CCC(C)(C)CC1 14909,c1(CNC(C)(CCOCCOCCO)c2nnnn2C2CCC2)cccnc1Cl 14910,C(=O)(CCCC#Cc1ccccc1)NC1C(C)N(C(=O)C2=COCCO2)CCC1 14911,c1(C(N(CC(C)NC(c2c(CC)nn(C)c2)=O)C)=O)ccc(COC)c(F)c1 14912,CC(CC(N)=O)C(=O)NCC1=CCN(C(=O)C(C(C)(C)C)C2CCCCC2)CC1 14913,C#CC1(NC(=O)C(C)(C)CCNC(c2n[nH]c(=N)[nH]2)=O)CCC(C)CC1 14914,c1(C(C)=O)cc(C(N2CCOCC2CCNC(=O)C=C2CCC(C)C2)=O)oc1C 14915,C(=O)(C(C(C)C)NC(=O)OC(C)C)NC(CC)CNC(c1csc(COC)n1)=O 14916,C1(N(CCC)C(C2CCC2C)=O)CCN(C(c2ccnn2CC(F)F)=O)C1 14917,Cc1ccc(C(=O)NCCOCC(=O)NCCN2CCCC(C)C2)cn1 14918,C(=O)(C(COC(C)(C)C)CC(C)C)N1CC2CN(C(CCCNC(C)=O)=O)C2C1 14919,C1(OC)CN(C(=O)C(=O)NCCNc2ccc3c(c2)CCO3)C2(CCC2)C1 14920,Cc1ccc(C(N2CC(C(C)NC(=O)CCCn3cccn3)C2)=O)c(N)c1Br 14921,N12CC=C(CN1C)CC2.c1(OC2(C=O)CC2)ccc(F)cc1.C1(CO)CC1C=O 14922,C1(NC(CNC(CNC(C2C(C)OCCO2)=O)=O)=O)CC2(C1)CC(O)C2 14923,N1(C(CC2CC(N(C)C)C2)=O)CCC(C(=O)NC2CCOC(C)(C)C2)CC1(C)C 14924,O=C(C1CCCc2cncn21)NC1CCN(C(C2(F)CCC(=O)CC2)=O)C1 14925,S(=O)(=O)(CCC(=O)NCC1(CNC(c2cncn2C)=O)CCCCC1)N(C)C 14926,C(=O)(CC1OCc2ncccc21)NCC1C(C)(C)CCCN1C(=O)C1=CCCC1 14927,N1(C(c2c(NC)cnnc2)=O)C(C(N2CCC(O)CC2C2CC2)=O)CCC12CC2 14928,N1(C(C(C)NC(C)=O)=O)CC=C(CNC(C2(c3ccnc(Cl)c3)CCC2)=O)CC1 14929,C1(OC)CC(CO)(NC(=O)CCc2cn(C(C3CCCCC3)C)nn2)C1 14930,CC1CC(CNC(=O)CCc2cc[nH]n2)CN1C(=O)Cc1cccc(Br)c1 14931,N1(C(Cc2cc(C)[nH]n2)=O)C2CCC1C(C)C(NC(=O)Cc1cncnc1)C2 14932,c1(C(c2n(CC=C)nnn2)NCCC(C)F)cccc2nn(C)cc12 14933,c1(CC(=O)N(C)CC2OCCN(C(C(C=C)(C)O)=O)C2)cc(F)c(C)cc1F 14934,Cc1c(NC(c2cc(I)cs2)c2nnnn2C2(C)CC2)cccc1Cl 14935,C1(NC(=O)NCCc2ccc(F)c(Cl)c2)CCOC2(CCS(=O)(=O)C2)C1 14936,C1(c2cn(C(CC=C)OCN3CCC(O)CC3)nn2)CCC2(CCCC2)C1 14937,C(=O)(C#CC1CCC1)NC1(C)CC(NC(=O)CCC2CC2(Cl)Cl)C1 14938,C(=O)(C1=C(Cl)CCCC1)N(CC(=O)N(C)Cc1cnnn1C)C(C)C 14939,N1(C(C2CC(OC)C2)=O)CCOC2(CCN(C(=O)Cc3ccccc3Br)C2)C1 14940,c1(C(=O)NC2CCCC(NC(C(CCC)(C)C)=O)C2)ccc2nccc(C)c2c1 14941,C(=O)(CC(O)CC(C)(C)C)N1CC(CN(C(CCC=C)=O)C)OCC1 14942,C(C(F)C)NCC=CCOCCNC(C)=O.C12CC(C1)N2.S(C)(=O)(=O)NC 14943,C1(C2(O)CN(C(=O)C(=O)NCCNC(C)=O)C2)(CNC(C(CC)(C)F)=O)CC1 14944,CCC(C)CC(C(=O)OC)NC(c1ccnc(O)c1F)=O 14945,Cc1ccc(=N)[nH]c1C(N1CCCC(NC(c2nc(Br)c[nH]2)=O)CC1)=O 14946,CC(CS(C)(=O)=O)C(=O)N1CC2(CC(NC(=O)Cn3ncn(C)c3=O)CO2)C1 14947,N1(C(c2n(CC)ncc2)=O)CCC(C(C)C(=O)NC(C)C(C)CC)CC1 14948,N1(C(C(C)Br)=O)CCCn2nc(C(N3CCC(O)C(F)C3)=O)cc2C1 14949,CC(CC(=O)NC1C=CCC(C(=O)NC(C)(CO)C2CCCC2)C1)CC(C)(C)C 14950,C1(NC(CN(C)C(N)=O)=O)CCC(NC(c2ccc(NC(N)=O)s2)=O)CC1 14951,C1(c2nnnn2C2CCCC2)(NCCC(C=C)(C)C)CCOC(CC(=O)OC)C1 14952,CC1CC(CCNC(=O)C=CC2CCC2)CCN1C(=O)C(=O)NCC(F)(F)F 14953,c1(CCC)cc(C(=O)N(C2CCCN(C(C3(F)CCCC3)=O)C2)CC)c(C)o1 14954,c1(OC)cc(C(=O)N(C2CCCC(N(C(=O)C3=C(C)OCC3)C)C2)C)c(Cl)cn1 14955,c1(C(=O)OC)cc(C#N)cnc1NCC1CC(C)N(C(=O)C=Cc2ncc[nH]2)C1 14956,N1(C(CC(CC)C)=O)CCCC2C1CCN2C(=O)Cc1scnc1-c1cccs1 14957,CC(C)(F)CCC(=O)N1CCC(CCCCCNC(=O)Cc2csc(=N)[nH]2)CC1 14958,Cc1ccc(NC(=O)C(=O)NC(C)CC2CN(C(c3csc(C)c3)=O)C2)cc1 14959,S(=O)(=O)(c1cccc(F)c1)NCCNC(c1cc(CC)oc1C)=O 14960,NC(=O)CS(=O)(=O)c1ccc(C(=O)NCC(O)CNC(=O)Cc2cscn2)cc1 14961,C(=O)(CS(=O)(=O)C(C)C)NCCN1CCN(c2c(OC)ncnc2Cl)CC1 14962,C1(COC)CN(C(=O)CCOc2ccc(Cl)c(Cl)c2)CC12CCC2 14963,N1(C(Cn2nc(C)c([N+](=O)[O-])c2)=O)CCCC2C(NC(=O)C3CC3)C(C)(C)C12 14964,c1(CN(C(C)=O)C)ccc(C(=O)N(C)CC23CCC(CO2)C3)cc1 14965,N1(C(CCC#CC)=O)CCCCC(CNC(c2cccnc2OCC(C)C)=O)C1 14966,C(C(CNC(C1CCCOC1)=O)C(F)(F)F)NC(CCn1c(C)ncc1)=O 14967,N1(C(CCOCC#C)=O)CCCC1(C)CNC(c1ccc(Cl)cn1)=O 14968,c1(CCCC(=O)NC2CCN(C(CC3(NC(C)=O)CC3)=O)C2)ccc(O)c(F)c1 14969,C(=O)(C1=CC2CCCC12)N1CC(CNC(=O)C2=CCCO2)OCCC1 14970,C1(CC(=O)N(C)CCO)CN(C(c2cnc(S)nc2)=O)CC12CC2 14971,Cc1ccc([N+](=O)[O-])cc1C(N1CCN(C(=O)C(O)C2CC2)CC1C)=O 14972,c1(C2CN(C(=O)NCC(=O)Nc3ccccc3)C2)ncccn1 14973,C(=O)(C1=CC2CCCC12)NC(C)CC1CCN(C(C2C(C)(C)C2(C)C)=O)CC1 14974,C1(CC(N2C(CNC(c3cnc(C)s3)=O)C=CC2)=O)CC2(CCC2)CO1 14975,Cn1ncc(NC(=O)CCC(N)=O)c1-c1cn(CC2CCCO2)nn1 14976,CN1CC2CCN(Cc3cccc4c3COC4)C2C1 14977,c1(CCC(=O)NC2C(NC(CCc3c[nH]c(=N)[nH]3)=O)C2)ccc(C2CC2)cc1 14978,c1(C(=O)NC)cccc(C(=O)NC2CC(CCNC(C3CCOC3C)=O)C2)c1 14979,C1(NC(c2ocnc2C(F)(F)F)=O)CCC(c2ccccc2)CC1 14980,c1(C(=O)NCC(CC)NC(C2CC(C3CCC3)C2)=O)c(F)ccc(OC)c1N 14981,c1(N2CCC(C(C)NC(CC(CC)CC)=O)C2)nc(C)nc2n[nH]cc12 14982,C1(C(=O)NCC(=O)NCCC)CC2(CCC2)CN1C(=O)CNC(C1CC1C)=O 14983,Cc1ccc2ncc(CN3CCCCC(C(N4CCOC5CC45)=O)C3)n2c1 14984,c1(NCC2(CC)CCCCCC2)cc(=NCC2CC3(CC3)CO2)[nH]c(C)n1 14985,CCCCCC(O)C(=O)N(CCC(C)(C)NC(=O)Cn1cncc1C(=O)OC)C 14986,C#Cc1ccc(C2CC2C(=O)N(CC(C)N(C)C(CCCC)=O)C)cc1 14987,C1(C)(OC)CCCN(C(=O)C(C)(C)CCCNC(C2CC(C)(C)CCO2)=O)CC1 14988,C(=O)(CCc1ccco1)N(C(C)C(=O)OC)C1CC(n2cccn2)C1 14989,c1(C(N2CCCCC(N(C(CCCC(C)C)=O)C)C2)=O)nccc2c1NCCC2 14990,c1(C(=O)NCCC2CN(C(C3(C)CC(C)OCC3)=O)C2)cnc2c(ccn2C)c1 14991,C1(CNC(c2ccc(CC)c(CC)c2)=O)CC2(CCC2)CN1C(=O)CC(C)(F)F 14992,CCCC(CCC)C(=O)NCC1CCCN(C(C2CCC(OC(F)F)CC2)=O)C1 14993,c1(CC)ccccc1-n1nnnc1C1(NCC2CC2(C)C)CCOC1C 14994,c1(C(=O)NCC(C)CNC(C2(C)CC(F)C2)=O)cccc2c1nc(O)n2C 14995,N1(Cc2ccc(OC)c(Br)c2)CC2CCC1CN2C(c1cocn1)=O 14996,O=C1C=COC2(CCN(C(c3cc(Br)c(Br)o3)=O)CC2)C1 14997,C1(N(C(c2c(CC)n(CC)nn2)=O)C)CCN(C(C2(F)CC=CC2)=O)CC1C 14998,C=CCCCC(=O)N1CC(O)(C2CCCN2C(=O)C=CCCC=C(C)C)C1 14999,c1(OC)ccc(Cl)c(CN2CCCCC2CNC(=O)CC2CCC2)c1 15000,Cc1nc(C)c(C(N2CC(O)(CNC(c3scnc3C3CC3)=O)C2)=O)s1 15001,N1(C(C(C(C)C)=O)=O)CCC2(CCCN2C(=O)CC2NC(=O)NC2=O)C1 15002,c1(C(=O)NC(CCOCC)C(=O)NC(CC2CC2)C(=O)OC)cncc(C#N)c1 15003,N1(CC)CCOCC1CC(=O)NCC1(F)CC(NC(c2cccc(CO)n2)=O)C1 15004,CN1CCN(C)CC(C(N2CC(C3CN(C(c4cccc(O)n4)=O)C3)C2)=O)C1 15005,C1(CSCC)CCN(C(c2ccc(C(F)(F)F)n2C)=O)CC1 15006,CC1CCCN(C(c2ccc(F)c(F)c2)=O)C1CNC(C1CC(F)(CO)C1)=O 15007,N1(C(CC2C(CNC(C=CC)=O)C2)=O)CC(C2=NOC(C)C2)C1 15008,N1(C(C(C2CCN(C(c3cccc(CO)n3)=O)C2)F)=O)CCC2(CC1)N=N2 15009,C1(C(N(CCC(C)NC(=O)CNC=O)C)=O)OCCC1C(N)=O 15010,c1(N2C(CCCNC(c3cn(CC)nn3)=O)CCC2)cc(C)nc(COC)n1 15011,c1(C(N(CC(O)CO)C(C)C)=O)cccc(CNC(=O)CC2CC(=O)NC2=O)n1 15012,C1(C(N(CCCNC(=O)CCCN2CCCC2)C)=O)CCc2nncn2C1 15013,C(CCC(N)=O)(C(=O)NC1CCN(C(=O)COCC(C)(C)C)CC1O)NC(C)=O 15014,N1(C(c2c(CC)n(C)nn2)=O)CCOC(C)(CNC(=O)CC2CCOC2(C)C)C1 15015,C1(NC(C2C(OCC)C2)=O)CN(C(=O)CCn2cc(Br)cn2)CC2(CC2)C1 15016,N1(C(c2ccc(C#C)nc2)=O)CC(NC(=O)C(O)CN(C)C)CC2(CC2)C1 15017,c1(NC(c2n(C(CC)C)nnn2)CCCSC)cc(Br)c(F)cc1OC 15018,c1(-c2nc(C3C(F)(F)C3)on2)scc2c1OCCO2 15019,N1(C(C(C(CC)C)O)=O)CC2CCCC1C2CNC(=O)C1=CCOCC1 15020,C(CCNC(c1nnnn1C(C)C)CCc1ccccc1)(C(C)C)OCCOC 15021,N1(C(c2cccc(OC)n2)=O)CC(C(=O)NC(c2ccc(F)cc2)C)CC(F)C1 15022,C1(CN(C(=O)C=Cc2cc[nH]n2)C)CCCN(C(C2CCOC(=O)N2)=O)C1 15023,c1(CNC(C(CC)N(C)C(c2ccnnc2O)=O)=O)cc(O)ccc1F 15024,C12(C(=O)NC3(C)C(C)CCC3)CC(CN(C(c3cccc(O)c3)=O)C1)C2 15025,c1(OC)ccc(F)c(C(N2C3CN(Cc4cccc(C#N)c4Cl)CC23)=O)c1F 15026,C(CN=c1cc(C)[nH]c(=NCC23CCC(CO)(CC2)CO3)[nH]1)=CCCC 15027,c1(C(=O)NC2(C)CCCN(C(C3CCC(O)C3)=O)C2)cncc2c1CCC2 15028,C#CC(C)CN=C(NCc1cnc(C)o1)NC(C)COC 15029,Cc1cnc(-c2noc(C(C3(C)CC3)F)n2)nc1 15030,c1(OC)ccc(N(C)C(=O)Nc2cc(N3CCOC3=O)ccc2F)cc1F 15031,Cc1nn(C(C)(C)C)c(C)c1C(N1CC=CC(NC(C2(F)CC=CCC2)=O)C1)=O 15032,Cc1cc(F)ccc1NC(=O)C(c1cccc(C(N)=O)c1)N(c1ccsc1)C 15033,C1(C(N(C)CC2N(C(CC(C)F)=O)CCC2)=O)CN(C)CCN1C 15034,C(=O)(N=c1ccc(S(C)(=O)=O)n[nH]1)Nc1cc(C)cc(C)c1 15035,Cc1cccc2cc(C(N3CC4(C3)CN(C(=O)C3CC3)CCO4)=O)nn12 15036,C1(CN(C(CC(=O)N(C)C)=O)C)CN(C(=O)C(O)c2ccsc2)CC12CC2 15037,C1(COC)(NC(c2cnc(C3CCOC3)s2)=O)CCN(C(=O)COCCCF)C1 15038,C1(NC(C2(F)C(C)OCC2)=O)CC2(CCN(C(=O)C=Cc3ccccc3)C2)C1 15039,C1(NC(C=C(C)C(F)F)=O)CCC(N(C(=O)C(c2cnn(C)c2)C)C)CC1 15040,C(=O)(C1=NNC(C(F)(F)F)C1)N1CC(CC(C)NC(=O)CCC(C)(C)F)C1 15041,c1(OC)ccc(NC(=O)C(c2cc(C)ccn2)N2CCC(F)(COC)C2)cc1 15042,C1(C)(CNC(CCOCCOCC)=O)CCN(C(c2cc3occc3[nH]2)=O)CC1 15043,C=CC1CN(C(C)=O)CC1NC(C1CCCCN1C(c1ccnnc1)=O)=O 15044,c1(CC)n[nH]cc1C(=O)N(CC(C)NC(c1cnns1)=O)C 15045,N1(C(CCc2n(C)c(S)nn2)=O)CC(NC(C2C3(CC3)C23CC3)=O)C2(CCC2)C1 15046,c1(C(=O)N(CCCN(C(=O)C(C)C2CC2)CC)C(C)C)cc(C)ccc1C(C)C 15047,C1(C(N2CCN(CC)C(=O)C2)=O)CC2(CCN(C(=O)Cc3cccn3C)C2)C1 15048,N1(C(C(CC(=C)C)C)=O)CCC(C2CC2NC(C2(O)CCC(C)(C)CC2)=O)CC1 15049,C1(C)(C(N2CCC3C(NC(C(C)=CC)=O)C32)=O)CC(c2ccccc2)=NO1 15050,N1(c2nc(N(C)Cc3ncc(CC)s3)nc(C)c2)CCCc2ccccc2CC1 15051,C1(CC)(NC(C2CCC(=O)C(C)C2)=O)CCN(C(C2CCC(=O)N2CC)=O)CC1 15052,c1(C(=O)NCCCNC(c2ccnnc2O)=O)ccccc1OCCF 15053,c1(C(=O)NC(CN(C(c2cc(=O)n(C)o2)=O)CC)C)csc2ccccc12 15054,c1(C(=O)NC2C3(CCN(C(C=CC)=O)CC3)C2)c[nH]c2ccc(OC)cc12 15055,N1(C(=O)Cn2cnnn2)CCC2CC12C(=O)NC(c1ncc[nH]1)CO 15056,c1(C(=O)NCC(CC=C)NC(c2csc(Br)n2)=O)cc2c[nH]nc2s1 15057,C1(CCNC(C(C)n2ccnc2)=O)CC(F)(F)CN1C(c1cc(Cl)cnn1)=O 15058,c1(C(C)C)nc(C(=O)NCC(O)CCNC(=O)Cc2ccc(Cl)s2)co1 15059,Cc1nn(CC(N2CCC(CO)C(NC(=O)CCOCC(F)F)C2)=O)c(C)c1Cl 15060,N1(C2CCN(C(C(CSC)OC)=O)C2)CCN(C(=O)CC2CCOCC2)CC1 15061,n1(CC(=O)NC(C2(O)CN(C(C3CSCN3C)=O)C2)C)cc(N)cn1 15062,c1(C(N(C(CNC(C(C)NS(C)(=O)=O)=O)C2CC2)C)=O)sc(F)cc1Cl 15063,S(=O)(=O)(CCC(=O)NCC(C1CCOC1)NC(=O)C(F)(F)c1cscn1)NC 15064,CC1(C)CCCC2(CN(S(=O)(=O)CC3COCCO3)C2)O1 15065,C(=O)(C(C)CC(F)(F)F)NCC1N(C(c2n(CC)ncc2)=O)CC(OC)C1 15066,C(C(C)CN=c1c(C#N)c[nH]c2c(C)cccc12)NC(Cc1cc(C)nn1C)=O 15067,c1(C(=O)NC23CC(C(=O)NCC4CCC(C)CO4)(C2)C3)coc2ccccc12 15068,CN1CCCC(C(c2scc(CC(=O)NC(c3cccs3)=O)n2)=O)C1=O 15069,c1(OC)cc(N)c(C(=O)NC(C2CCCCC2)CNC(=O)COC(F)F)c(F)c1 15070,C(CO)(C(=O)NCC1C=CC(NC(C2CCCS2)=O)C1)NC(=O)C1CC1 15071,c1(CNC(=O)NC2(c3cccnc3)CCC2)ccc(CN2CCOCC2)cc1 15072,C1(C(=O)NC2(CNC(=O)CC(=O)N(C)C)C(C)C2)CCOC(C)(C)C1 15073,C(=O)(C1CCCc2nc[nH]c21)NC1(C)CN(C(=O)CC2CSC2)C1 15074,c1(C(=O)NC2C(C)CCN(C(C3CCS(=O)(=O)C3)=O)C2)cnc2cc[nH]c2c1 15075,C1(C(N2CC(C)C(NC(c3ccc4ncnn4c3)=O)C2)=O)CCCC(F)(F)CC1 15076,CC#CCCC(=O)NC1CN(C(c2cnn(-c3ccncc3)c2)=O)CC1OC 15077,c1(CCC)nc(C)c(C(=O)NCC(C2CCN(C(C3(C)COC3)=O)CC2)F)o1 15078,c1(C(=O)NCC(CC(C)C)NC(c2ccc(CO)c(F)c2)=O)ccc(N)c(Cl)n1 15079,C1(C(=O)O)CN(CCC(F)(F)F)C2(CCC2)CO1 15080,C1(C(N2CCN(C(CC(C)(C)O)=O)C(CCO)C2)=O)CC2CCC(C1)S2(=O)=O 15081,c1(C(N2CCC(OC3CC3)CC2)C(=O)NC)cnc2sc(Br)cn12 15082,c1(C(=O)NC23CCN(C(c4c(CC)noc4)=O)CC2C3)ccc2c(c1)SCCN2 15083,c1(C(N2CCOCC2)C(=O)NCCCNC(=O)C(F)F)ccccc1 15084,C1(C(N(CCC)CCNC(=O)C(CC)(CC)CO)=O)Cc2cccc(C)c2O1 15085,C(N=c1[nH]cnc(Cl)c1CO)C1C(C)CN(C(=O)Cc2cc(C3CC3)on2)CC1 15086,CCCC(C)(C)C(=O)N1CC(CCNC(C2CCC2C(F)(F)F)=O)C(C)C1 15087,N1(C(c2nn(C)c(Cl)c2Cl)=O)CCN(C(C2CCNC2=O)=O)CC12CC2 15088,C(C)(C)(C(C)(C)CO)NC(CCC1CCCN(C(CNC(=O)OC)=O)C1)=O 15089,c1(CC)nc2c(C)csc2c(=NC(C)CC(C)NC(C2CCCN2C2CC2)=O)[nH]1 15090,CCS(=O)(=O)CC(=O)NC1CC1NC1(CO)CCCN(Cc2ccccc2)C1 15091,N1(C(C(CC2CC(C(=O)OC)C2)OC)=O)CCCCCC1OC(C)=O.C(C)(C)(C)O 15092,C1(NC(=O)CCCF)CCCCN(C(C2CCS(=O)(=O)C2)=O)C1 15093,C1(C(=O)NC2CC(CNC(CCCNC(C(C)(C)C)=O)=O)C2)C(Cl)(Cl)C12CC2 15094,N1(C(C2(C#C)CCC2)=O)CC(F)CC1CC(=O)NCCN1CC2CC2C1 15095,c1(COCC(=O)O)cn(Cc2ccc(C(=O)NCc3cc(CC4CC4)no3)o2)nn1 15096,CC(CS(C)(=O)=O)C(=O)NCC1(F)CCN(C(c2ccc3ncnn3n2)=O)CC1 15097,C1(NC(CSCC=C)=O)COC2(CCCN(C(c3ccc(N(C)C)cc3)=O)C2)C1 15098,C1(C(N(C2CCN(C(C)C)C2)C)=O)CCN(C(=O)Cn2cnc(=N)[nH]2)C1(C)C 15099,S(=O)(=O)(c1c(Cl)cc(Br)cc1Cl)N1C2CN(C(c3c(F)cncc3F)=O)CC21 15100,N=c1[nH]nc(Cl)cc1C(=O)NCC1(CO)CCN(C(=O)CCc2cnc[nH]2)CC1 15101,C1(CN(C(CCCOCC)=O)C)CN(C(=O)CC2(O)CCCOC2)CCO1 15102,N1(C(CCSCCC)=O)CCN(CCNC(=O)C(C)C(C)O)CC1 15103,c1(C(=O)NCC(c2ccccc2)NC(C(CSC)OC)=O)ccc(N)c(Cl)c1 15104,N1(C(CN(C(=O)OC)C)=O)CCC(C)(C)C(C(=O)NCc2nc(C3CC3)no2)C1 15105,C(=O)(C1=C(Cl)CCOC1)N1CCC2(C(C(N(C(C(C)C)C)C3CC3)=O)C2)C1 15106,C1(C(=O)NC(CC(=O)NC)C)(NC(C2C(C(=O)OC)C2(C)C)=O)CCCC1C 15107,CC1CCC(NC(=O)CCOCC(F)F)CN1C(=O)Cc1ccc(O)c(O)c1 15108,c1(C(N2CCCC(NC(c3n[nH]c4c3CCOC4)=O)C2)=O)cnc2nccn2c1 15109,C12(OC)CCC(C(=O)NC3(C)CN(C(=O)C(F)(F)C(F)(F)F)C3)(CC1)CC2 15110,N1(C(C2C(C)OCCC2)=O)CC2(CC2)CC1CNC(=O)C1=NNC(C(F)(F)F)C1 15111,c1(CC(=O)N(C)CCN(C(=O)C(F)(F)C2CC2)C)cncc(Br)c1 15112,N1(C(Cc2cccc(C#C)c2)=O)CC2CC(NC(=O)CCC3CC3(Cl)Cl)CC1C2 15113,N1(C(CCCC(=C)C)=O)CCOC2(C1)CN(C(C1CC(=O)N(CCOC)C1)=O)C2 15114,C1(N(C)C(c2ccc(F)o2)=O)CCCN(C(=O)CC(c2cccc(F)c2)O)C1 15115,N1(C(c2c(CC)noc2)=O)CC2(CNC(c3ccn(C)n3)=O)CC(F)(C1)C2 15116,c1(OC)cccc2c(N3CC(CO)(NC(=O)Cc4cc[nH]c4)C3)ncnc12 15117,C1(C(N(C(C)CO)Cc2ccccc2)=O)CN(C(C2CCC=CO2)=O)CCO1 15118,N1(C(C(CC)C)=O)C2CCC1CC(F)(CNC(=O)C=CC(F)(F)F)C2 15119,N1(C(C2COCCN(C(C3CN(C(C)C)C3)=O)C2)=O)CCC12CCCOCC2 15120,C(C1=CCN(C(=O)Cc2csc(C(F)(F)F)n2)CC1)NC(C1(C)CC(F)(F)C1)=O 15121,N1(Cc2ccc(C(=O)OC)cc2)CCSC(C)CC1.C12CCN(CC1)C2=O 15122,C1(CC=C)(C(=O)NCc2n[nH]c(C)n2)CCCN1C(=O)CCc1cn[nH]c1 15123,CC1(C)COCC(C(=O)NCC(Cc2ccccc2)NC(C2(C(N)=O)CC2)=O)O1 15124,c1(C(C(=O)NCCOCC)N(CC(F)(F)Cl)C)cc(NC(C)=O)cn1C 15125,N1(C(CC2C(C)C(=O)CC2)=O)C2CC1CN(C(c1ccc(CCF)cc1)=O)C2 15126,c1(C(=O)OCc2nn(C)c(Cl)c2)nc(Cl)c(=O)[nH]c1N 15127,C=C(F)C1(CC(N2CCC(N(C(=O)CC(CC)OC(C)=O)C)CC2)=O)CCC1 15128,CS(=O)(=O)c1ccccc1-c1ccc2c(C(=O)N=c3cc(CO)[nH][nH]3)nsc2c1 15129,N1(C(C(C)OCC)=O)CC(F)(F)CC1CNC(=O)C(C)Sc1ccccc1 15130,C1(C)(C(=O)NCC(C2CC2)NC(C2(C(=O)OC)C=CCC2)=O)C(C)(C)C1(C)C 15131,N1(C(C2C(C(C)C)CCC2)=O)C2CCC1C(F)C(NC(c1cc(Cl)cs1)=O)C2 15132,c1(C(CNC(=O)C(C)(C)CO)NC(C=CC)=O)ccccc1CC 15133,C1(NC(c2ccncn2)=O)CCN(C(C2CC(CF)C2)=O)CC1CO 15134,c1(C(N2CCCC(C(=O)OCC)C2)=O)cc2ccc(-c3cccc(F)n3)nc2[nH]1 15135,C(=O)(C(C)(C)CC(C)(C)C)NC1(COC)CN(C(c2ccnnc2C)=O)C1 15136,C1(CNC(C(C)NC(COC)=O)=O)CC2CC2N1C(c1ccc(C(C)=O)o1)=O 15137,c1(C(=O)NCCOCCN(C)C(c2cnc(O)o2)=O)cc(Cl)ns1 15138,c1(Cn2cc(CS(CC)(=O)=O)nn2)ccccc1CNC(=O)CC12CCCC1C2 15139,Cc1cc(C(N2CC(O)(CCNC(c3conc3C(C)C)=O)C2)=O)c(O)c(C)c1 15140,C1(C(=O)Oc2ccc(CO)cn2)CCC2(CC1)CN(C(=O)OC(C)(C)C)CCO2 15141,c1(C(=O)NCC2(COC)CCCN2C(C2CC2(C)C)=O)cncc(N=[N+]=[N-])c1 15142,c1(N2CCC(C)C(F)(F)C2)nc2cc[nH]c2c(=NCC(C)(C)c2ccccc2)[nH]1 15143,C1(N(C)C)CCC(c2ccccc2)(NC(=O)NCC2(S(C)=O)CC2)CC1 15144,c1(N2CC3C(C)C3C2)nc2ccccc2nc1N(C)Cc1ccc(S(C)=O)cc1 15145,C1(NC(COC(C)=O)=O)CCN(CCNC(=O)CNC(=O)CC(C)(C)C)CC1 15146,C#Cc1cnn(C)c1C(=O)NCCC1CSCCN1C(C1CCCNC1=O)=O 15147,CCC(C(=O)N1CC(NC(=O)CCC2CCCO2)C1)N1CCCC1=O 15148,CC(O)C(C(=O)NCCCCCCC1CC1)NC(c1ccc(O)cc1)=O 15149,c1(N2CC3CN(C(=O)OC(C)(C)C)CC3C2)cc(Cl)c2cnn(C)c2n1 15150,c1(NCC(=O)N(CC(C)N(C)C(C2COCCO2)=O)C)cnn(C)c1 15151,C1(CC(=O)N(CC(C(C)C)C)C)CC(NC(=O)C=CC(=O)NC2CC2)C1(C)C 15152,N1(C(=O)C=CC2CCCC2)CCC(CCNC(C23CCC2CC3)=O)CC1 15153,C1(NC(C2(CC)CC2(F)F)=O)C2CN(C(C)=O)CC12 15154,CC1(C)CN(C(c2csc(S(N)(=O)=O)c2)=O)C(CNC(=O)C(C)(C)C(F)F)CO1 15155,c1(SCC(=O)NC2CC(NC(C3COCCC3(F)F)=O)C2)ccc(F)c(F)c1 15156,S(=O)(=O)(c1cccnc1N(C)CC1CCCS(=O)(=O)C1)NCCN(C(C)C)C 15157,Cc1ccc(CN2CCC3CN(CCO)CC3CC2)c2ccccc12 15158,C(=O)(C(c1cccs1)=Cc1cccs1)NC(C(C)NC(C1(Cl)CC1)=O)C 15159,N1(CC)CCN(CCNC(N2CCCC(COc3cccc(SC)c3)C2)=O)CC1 15160,CC(CCNC(=O)CC1CCC1)CCNC(C1COCCO1)=O 15161,N1(C(C(CCC)(C)O)=O)CC(C2CCCN(C(c3cnc4cccnn34)=O)C2)C1 15162,C1(NC(C(C2CCC2)OCC)=O)CCC(F)(CNC(c2cc(C3CC3)[nH]n2)=O)C1 15163,C1(F)(CNC(c2c(C)snc2)=O)CCCN(C(c2cnnn2C2CC2)=O)C1 15164,CCCCC(C(=O)Nc1ccccc1CC)NC(c1ccc(C)nc1C)=O 15165,CC1CN(C(C2CN(C(c3ccc(C#N)o3)=O)CC2(C)C)=O)CCS1=O 15166,N1(C(CS(CC)=O)=O)CCCN(C(c2cnc(C)nc2C)=O)CC1C(C)C 15167,c1(C(=O)NC(C)CC(C)NC(=O)C(C)CSC(F)(F)F)csc(=NC2CC2)[nH]1 15168,Cc1ccccc1Oc1ccc(C(N2CCC(N(C(=O)CC#N)C)CC2)=O)cc1 15169,c1(CC)ncc(C(=O)NCc2ocnc2C(=O)NCC2(O)CCOC2)cn1 15170,CC1CN(C(=O)C=Cc2ccco2)CC(CCNC(=O)CCC2CC2)O1 15171,c1(SC)nc(C(N2CC(NC(=O)C(C(C)O)N(C)C)C(C)C2)=O)c2ccccn12 15172,c1(C(=O)NC(CC)CN(C(=O)CC2(CSC)CC2)CC)cncc(OCCO)c1 15173,c1(C(C(C)SC)C)ccc(NC2(C)CC(NC(=O)OC(C)(C)C)C2)cc1 15174,c1(NC(C2(F)CN(S(C3(CC=C)CC3)(=O)=O)C2)=O)cc(O)c2ccccc2n1 15175,C1(NC(C=CC(C)C)=O)CCN(C(=O)CCc2cc(Cl)no2)CC1C(C)C 15176,Cc1ncc(CNC(=O)C(CN(C)C)NC(=O)Cc2cnnn2C)s1 15177,C(C)(C)(C(=O)NCCC1CC(NC(=O)Cn2cnc(-c3nc(C)no3)c2)C1)OC 15178,C1(NC(C(CCCOC)C)=O)CCCCN(C(=O)Cc2cccc(C)c2)CC1 15179,Cc1cccc(C(N2CCCC(C)C2CNC(c2c[nH]ccc2=O)=O)=O)c1O 15180,c1(-c2nc(NC(c3ccc(I)c(Cl)n3)=O)sc2)cccc2[nH]ncc12 15181,N1(C(c2cc(C)ncc2C)=O)CCCC(O)(CNC(=O)CCSCC(N)=O)CC1 15182,N1(C(Cn2c(=O)sc(C)c2C)=O)CC2ON=C(CNC(c3ccn(C)n3)=O)C2C1 15183,N1(C(c2c(C)nc(CC(C)C)o2)=O)CCC2(CC1)CC2NC(=O)CSCC(N)=O 15184,N1(C(CCOCc2nnc(C)s2)=O)CCCC(N(C)C(c2ccccn2)=O)C1 15185,N1(C(C=CCC)=O)CCC(=CCNC(C2CC=CC(O)C2)=O)CC1 15186,C1(OC)CN(C(=O)C(C)=CC2CC2)CC1NC(c1ccc(F)s1)=O 15187,c1(CCCC(=O)NCCN(C)C(c2ccc(F)c(N)c2)=O)c[nH]c2ccccc12 15188,N1(C(C(Cc2ccc(OC)cc2)N)=O)CC2CC(C1)c1cccc(=O)n1C2 15189,Cc1cc(C(=O)NC2CCN(C(C3(C)CC3)=O)CC2C)c(C)n1-c1cnn(C)c1 15190,C1(C(N(C2CCCCCC2)CCNC(c2c(C)cno2)=O)=O)CCCCS1(=O)=O 15191,C12(NC(=O)CCCc3cccnc3)CC(C1)N(C(c1cc[nH]c1)=O)C2 15192,C1(CNC(CSCC#C)=O)CC2COCC2N1C(C1(CC#C)CCOCC1)=O 15193,C(C)(C(=O)NNC(=O)c1ccoc1C)c1nnc(-c2c(C)cccc2)o1 15194,C(CCC(CO)NC(c1coc(C2CC2)n1)=O)NC(=O)CCCF 15195,c1(OC)cc(OC)[nH]c(=NCC2(C)CCN(C(=O)C=C3CCSCC3)C2)n1 15196,Cc1cccc(O)c1C(=O)NC1CC(CCC(=O)NCc2cn(C3CC3)cn2)C1 15197,N1(C(C(CC)OC2CCCC2)=O)CCCC(CC#N)C1 15198,c1(OC)cnc(CNC(C2(C)CCCN2C(=O)CN2CCCC2)=O)cn1 15199,C1(C(=O)NC(CSC)(C)C(=O)N2CCOC(C(C)C)C2)CC2(CC(=O)C2)C1 15200,C(C(CC(C)C)C(=O)Nc1cnncc1C(F)(F)F)OC 15201,C1(CNC(c2cc(CC)n(C)n2)=O)CC12CCN(C(c1cnccn1)=O)CC2 15202,CCCCCS(=O)(=O)NC(=O)CC(F)(F)c1cccnc1Br 15203,Cc1c(C(=O)N(C2CN(C(C3CCCC3C)=O)C2)C)cnn1-c1ccncc1 15204,N(C1C(=O)Nc2cccc(C)c21)C(CCn1cc(-c2ccc(C)cn2)nn1)=O 15205,N1(C(c2ncn(C)n2)=O)CC2CC2C1CNC(c1cncc(O)c1)=O 15206,c1(N(CCS(C)(=O)=O)C(=O)C(=O)NN2CCCCC2)ccc(Cl)c(C(F)(F)F)c1 15207,N1(C(c2cc(Cl)c(C)cc2Br)C(=O)NCCOC)C(C)C2CCCCC2C1C 15208,CC1(C(=O)NCC2(CNC(c3ccc(F)c(Cl)c3)=O)CCC2)CCCCNC1=O 15209,c1(OC)ccc(Cl)c(C)c1C(N1CCC2(NC(c3cc(CO)[nH]n3)=O)CC2C1)=O 15210,CCCC(O)CC(=O)NC(C)(C)CN(C(=O)C(c1ccc(Br)cc1)CC)C 15211,c1(C(=O)NC2CC(NC(C(CC=C)C)=O)CC2O)ncc(F)c(OC)n1 15212,c1(C(N(CCNC(C2CCCSS2)=O)CC)C)ccc2ccccc2c1 15213,c1(C(=O)NC2CC(NC(=O)CC3COCCO3)C2)c(Br)ccc2cccnc12 15214,Cc1ccc(-c2cc(CN3C(C)C(=O)NCC3)on2)cc1.C(N)(=O)NC 15215,c1(CC(C(N2CCC(N(CCO)CC3(C=C)CCC3)C2)=O)C)ccc(C#N)cc1 15216,C(=O)(C=CS(C)=O)NC(C1(O)CN(C(=O)C(F)(F)c2cscn2)C1)C 15217,CC1(C)CCCc2c1n[nH]c2C(N1CC(NC(c2occc2F)=O)C1)=O 15218,c1(CC(=O)NC2(C)CC(C(N(CC(=O)OCC)CC)=O)C2)cccc(F)c1 15219,N1(C(C(C)CC2CCC2)=O)CCC(CO)(CNC(c2c[nH]cc2C2CC2)=O)CC1 15220,C1(NC(CC(C)C)c2nnnn2C2CC2C2(C)CCOCC2)CC2CCC(C1)S2 15221,Nc1cc(C(N2CCCC3(NC(C4CC=CC4)=O)CC3C2)=O)cc(F)c1O 15222,C1(c2cccnc2)(C(=O)NCC(CNC(C(F)=CCC)=O)F)CCCC1 15223,C1(NC(C2(CC#C)CCCC2)=O)CCC(C)N(C(c2ccc(Cl)cc2N)=O)C1 15224,c1(CNC(C2CSCCN2C(c2cc(F)c[nH]2)=O)=O)ccccc1F 15225,c1(C(N2CC(COC)(CNC(=O)CC=C(C)C)C2)=O)ccc2cc[nH]c2c1 15226,C12(NC(C#CC(C)C)=O)CCN(C(c3cccnc3C(F)(F)F)=O)CCC1C2 15227,C1(NC(C=CC(=O)NCCC(C)N(CC(F)F)C)=O)CCCCCO1 15228,CC(c1cnn(C)c1)=CC(=O)NC1(CNC(C2CCNC(=O)C2)=O)CCOC1 15229,C#CCCC(O)C(=O)N1CCN(C(=O)COCCCC)CC1C(F)F 15230,c1(C(=O)NC2CC(C)(NC(C(CC)NC(N)=O)=O)C2)cnn(C)c1Br 15231,C1(C(=O)N(C(c2sccc2Cl)=O)CC)CCCN(C(=O)CSC2CCCCO2)C1 15232,C1(CNC(C=C(C)Cl)=O)CC2CCC1N2C(=O)Cc1cccc(F)c1 15233,N1(C(COCC(=O)NC)=O)CC(CNC(=O)C(C2CCOCC2)C)CC1(C)C 15234,N1(C(C2C(C(=O)OC)C=C2)=O)C(C(=O)N(CC(C)(C)O)C2CC2)CC1C 15235,N1(C(CC(=C)C)=O)CCN(CCNC(=O)CC(F)(F)Cl)C(c2ccccc2)C1 15236,CC1(CCNC(c2csnn2)=O)CCN(C(C2OCCC2C(F)(F)F)=O)C1 15237,C(=O)(NNC(=O)C(C)(O)CNC(=O)OC(C)(C)C)c1c(Cl)ccc(NCC(C)C)c1 15238,C(=O)(C(Cn1ccnn1)NC(C1CC=CCO1)=O)NCCNC(CC)=O 15239,Cn1ccc(=NC(=O)C(CCc2cc[nH]n2)NC(c2c[nH]c(=O)cn2)=O)[nH]1 15240,C(C(C)(C)C(=O)N1CC(CCNC(c2cc(-c3ccncc3)on2)=O)C1)OC 15241,N1(C(C)=O)CCC(O)(C(N2CCNC(=O)C2)=O)CC1.C12CC(C1)C(=O)N2 15242,C1(C)(CNC(C(C)(F)F)=O)CC(F)(F)CN1C(c1cccn2cnnc12)=O 15243,N1(C(c2cc(C)[nH]n2)=O)CCC(C(C)CNC(=O)CCCF)CC1 15244,C=CC(C)(C)C(=O)NC(C1CCN(C(=O)CC2(NC(C)=O)CC2)CC1)C 15245,N1(CCOCCOC)CCC(CC(CC2CCCO2)C(=O)OC)C1 15246,C1(CC)CCOC1C(=O)NC1CC(CN(C(c2nnn(C)n2)=O)C2CC2)C1 15247,C1(NC(C(CC)(C)C)=O)CCC2CCN(C(=O)CCc3ccccc3[N+](=O)[O-])C12 15248,c1(N2CC=CC(NC(c3nn(CC)nc3C)=O)C2)ncc([N+](=O)[O-])cc1CO 15249,C1(CC(=O)NC(c2sccc2Cl)C)CCN(C(C2(c3ccncc3)CC2)=O)C1 15250,C(=O)(C(CCCC)C(C)C)NC1C(NC(CCCCOCCC=C)=O)C1 15251,C1(CNC(C=CCCC)=O)(OC)CCN(C(=O)C(c2cccnc2)C)CC1 15252,c1(C(=O)NC2CC(CNC(C3N(CC)CC3)=O)C2)c(N)cc(F)cc1Cl 15253,C1(C(=O)NC2(CNC(C3CC(SC)C3)=O)CCOCC2)Cc2ccccc2N1 15254,C1(OC)CN(C)C(C)(C(=O)NC2CC3CN(C(c4ccc(C(F)F)o4)=O)CC23)C1 15255,CC(O)(CC(=O)N1CC=CC(NC(c2ccc(Br)s2)=O)C1)C1CC1 15256,c1(SCC(N2CCN(C(C34CCCC3C4)=O)CC2)=O)nc2ccccc2[nH]1 15257,c1(C(N(C)CC2N(C(C(CCC)O)=O)CCC2)=O)ccc(Br)c2cn[nH]c12 15258,c1(C(=O)NC2CCC(NC(C3N(C(C)=O)CCCC3)=O)CC2)ccc(F)nc1C 15259,N1(C(Cc2n(C)cnc2)=O)CCC2(CCCCN(C(c3cnn(C)c3F)=O)C2)C1 15260,c1(C(=O)NC2CCC(CNC(CC(=C)Br)=O)C2)nnc(O)cc1O 15261,c1(C(N2CCCC(N(C(c3ccns3)=O)CC)C2)=O)c(OC)cccc1O 15262,CC1CN(C(=O)Cc2csc(=N)[nH]2)CC1C(=O)NCCC(=O)Nc1ccccc1 15263,c1(C(N2C3CC(NC(C4(CC(C)C)CC4)=O)C2CC3)=O)cnn2c1CC(F)(F)C2 15264,c1(CC)nc(-c2cn(C)nc2OC)n(C2CCS(=O)(=O)C2)n1 15265,c1(C(N2CCn3nccc32)=O)cc2n(c1)CCC2 15266,C1(C(N(CC(C)N(C(C(C)CO)=O)C)C)=O)CCC2(CC1)NC(=O)NC2=O 15267,CCCC(C)(C)C(=O)NC1CC(CCNC(=O)C(F)OC)C1 15268,Cc1cc(C(=O)NC(C)CCN(C)C(c2cc(C(C)C)no2)=O)n(C2CC2)n1 15269,C(=O)(C(O)CC(C)(C)C)NCC1ON=C(C(=O)NCC(C)C)C1 15270,c1(SC)cccnc1C(=O)NCC(C)NC(=O)C(c1cccc(O)c1)(C)C 15271,N1(C(C2OCC(C)C2)=O)CCC2(CCCN(CCc3ccccc3)C2)C1 15272,C1(O)(Cc2nc(O)n[nH]2)CN(CC(F)F)C1.C12CN(C1)NC2=O 15273,C(=O)(C1=NOC2(CCC2)C1)N(CC(CO)(CO)NC(Cc1c(C)con1)=O)C 15274,N1(C(C2(OCC)CCC2)=O)CC2(CCN(Cc3ccc(C)cc3)CC2)C1 15275,Cc1cnc(C(=O)NC2CCCCC2CNC(=O)C(C)Cn2ccnc2)c(C)c1 15276,Cc1cc(C)c(C=CC(=O)NCC2CC(NC(C3CCOC3=O)=O)C2)cc1C 15277,Nc1nc(C(N2CCC(NC(=O)CC3(CO)CC3)C(O)C2)=O)ccc1[N+](=O)[O-] 15278,C(=O)(CC(C)CC(C)C)N1CCC(C(N2CC(O)(CC)C2)=O)(CCOC)CC1 15279,C(=O)(C#CC1CCOC1)NCCC(CNC(c1c(C)n(C)nn1)=O)O 15280,c1(OC(C)C(=O)NCC2(O)CC(NC(C3OCCO3)=O)C2)ccc(F)nc1 15281,c1(C(=O)NCC2N(C(c3scc(COC)c3)=O)CC(F)C2)cccc2c1CCC2 15282,C(=O)(CCCCCN=[N+]=[N-])N(CC(N(C)OCC(F)(F)F)=O)C1CCCCC1C 15283,C12(CC(=O)N(C)CCNC(c3cnn(C(F)F)c3)=O)CCC(CC1)C2 15284,c1(C(=O)NCC(C(C)(C)C)NC(C2CCC(=O)O2)=O)cnc2[nH]ccc2n1 15285,Cc1ccc2oc(C(=O)NC3CC4CC3N(C(c3cnc(C)nc3)=O)C4)cc2n1 15286,c1(OC)ccc(CN2CCC2C(=O)NCC2CCCN(C)C2)c(OC(C)C)c1 15287,C1(NC(Cc2ccc(C)nc2Cl)=O)CC2CCCC(C1)N2C(=O)CC(C)C1CC1 15288,CC1(C)CN(C(c2cnc(Br)s2)C(=O)NC2CC(F)(F)C2)CCS1=O 15289,C(=O)(C1=NOC(C(=O)NC2CCCN(C(=O)CC(C)(C)O)C2)C1)OC(C)(C)C 15290,C1(O)(C(C(=O)OCC)(F)F)CN(N2CCC3(CC2)C(O)CC3O)C1 15291,N1(C(C)CCc2nccs2)C(=O)NC(c2ccsc2)C1=O 15292,C1(O)(C(C)CNC(C2CCCS2)=O)CCN(C(c2cnn(CC(F)F)c2)=O)C1 15293,CCC(CN(C)C)CC(=O)NCC1CC1CNC(c1csnc1C)=O 15294,N1(C(C(C)(CO)NC(CC2(N(C)C)CCC2)=O)=O)CC23CCC2(COC3)C1 15295,C1(NC(C(C)C)=O)CCCCC1CNC(=O)C(O)COCc1ccccc1 15296,CC1(C)CC(NC(C2CC(C)(C)OC2(C)C)=O)CN(C(c2c[nH]ccc2=O)=O)C1 15297,c1(C(=O)NCC(CO)NC(c2csc(CO)n2)=O)cc(C(F)F)ccc1Cl 15298,CCCC(CNC(=O)CC1CCC(C)(C)O1)C(=O)NCC1OCCC1(C)C 15299,c1(C(N2CCC(C(CNC(C3C4CCCC34)=O)F)CC2)=O)cccc2cncn12 15300,C1(NC(=O)CSCCC(F)(F)F)(CO)CCCN(C(c2csc3nccn23)=O)C1 15301,C1(NC(CS(CC)=O)=O)CC2CC1CN(C(c1c(C)ccc(Cl)c1F)=O)C2 15302,CC1CC=CCC1C(N1CCCC(CC(=O)NC2CCNC(=O)C2)C1)=O 15303,C1(C(CC(=O)OCC)NCc2ccn(C)c2)CCC(F)(F)CC1 15304,c1(C(N(CCCNC(C2(C)CC(C)C2)=O)C2CC2)=O)n[nH]c2cc(Cl)ccc12 15305,C(=O)(CC(C)(O)C(F)(F)F)NC(C1CCCN1C(=O)C=Cc1cccc(O)c1)C 15306,C(=O)(C(S(C)(=O)=O)C1CC1)NC(C)CC1CN(C(C2(CCO)CC2)=O)CCO1 15307,C1(C2CC2)(C(=O)NC2(CN(C(C3CN(S(CC)(=O)=O)C3)=O)C)CC2)CCC1 15308,Cc1noc2nc(C(=O)NC(C)CCCCNC(c3cnc(Cl)s3)=O)ccc12 15309,C1(CC(=O)NCC(CC)(C)NC(=O)CC(C)COC)CCC=CCC1 15310,CC1CN(C(c2nc(C(C)(C)C)no2)=O)CCC1NC(c1ccnc(O)c1)=O 15311,N(C(=NCc1ccc(C#N)cn1)N1CCC2=C(CCCC2)C1)C1C(C)C1 15312,C(CCOCCO)(C(=O)NCC1CC12CC2)NC(c1cnc(C)s1)=O 15313,C1(CC)C(NC(c2cn(CCC(C)C)nn2)=O)CCCN1C(=O)C=C(C)C 15314,O=C1CN(C(C2CN(C(=O)CC3CCCSC3)CC2F)=O)CCN1 15315,N1(C(CN2CCN(C)CC2)=O)CC2(CC(NC(=O)C(O)C(F)F)CO2)C1 15316,C12(NC(CCC3C(C#N)C3)=O)CC(CNC(C34CSCC3C4)=O)(C1)C2 15317,C1(C(=O)NC(c2c(C)cccn2)C)CN(S(=O)(=O)Cc2ncccn2)CCN1C 15318,c1(N(CC(c2cccc(I)c2)O)C)ccc(C#N)nn1 15319,c1(C(=O)NCC2(O)COC2)ccc2nc(-c3cccc4ccncc34)cn2c1 15320,c1(C(=O)NCCC(C(C)C)NC(c2c(CC)nn[nH]2)=O)cncc(Cl)c1C 15321,c1(C(N2CCCC(C)(C(N3CCC(CC)C3)=O)C2)=O)cnc2cc(Cl)ccn12 15322,CCC(C(=O)N1CC(O)CC1CNC(C1(c2ccccc2)CCC1)=O)C(C)C 15323,c1(OC)c(Br)ccc(CN2CC(NC(=O)Cc3cccc(O)c3)C(F)C2)c1F 15324,C(=O)(C(C(C)CC(C)(C)C)N1CC2OCCOC2C1)NCC=C 15325,N1(C(C2=CCCC2C)=O)CC23CCCC2(C1)CN(C(C1(C(C)(C)O)CC1)=O)C3 15326,c1(CC)c(C(N2CCOC(CC(=O)NC3CCC(O)C3)C2)=O)cnn1C 15327,c1(CC(=O)N(C(C)CNC(=O)CC2OCCOC2(C)C)C)coc2ccccc12 15328,C1(NC(c2cc(C)[nH]c2C)=O)CC2CCC1C(NC(=O)CSc1ccccc1)C2 15329,CC(CNC(=O)COCCc1cccs1)(CO)NC(c1cnoc1-c1ccoc1)=O 15330,c1(CCC(=O)NC2CCCC2CNC(=O)COC2COC2)ccc(C(F)F)cc1 15331,C(C1=NOC2CN(C(c3csc(-c4cnc[nH]4)n3)=O)CC12)NC(c1cnsc1)=O 15332,c1(OC)ccc(Cl)cc1CC(=O)NC1CN(C(C2CC(C(C)C)C2)=O)CC1(C)C 15333,S(=O)(=O)(c1nc(N2CCN(C3CCCC3)CC2)ccc1Br)N1C2CN(C)C(C2)C1 15334,C1(CNC(c2c(C)nn(C)n2)=O)CN(C(=O)Cc2ccc(O)nc2)C2CCN1C2 15335,c1(C(=O)NCC(C)NC(c2ccc(C(C)C)cc2F)=O)n[nH]c2c1CC1CC21 15336,N1(C(c2ccc(CNC(C(C)c3ccsc3)=O)s2)=O)CCCC12CCOCC2 15337,CC1(NC(=O)CC2CCC3CC23)CCCN(C(c2ccccc2C(F)F)=O)C1 15338,c1(C(N(CC(C)NC(=O)C(C)(C)N2CCCCC2)CC)=O)c[nH]cc(C)c1=O 15339,C(=O)(CS(=O)(=O)C1CCCC1)N(C1C2CN(C(=O)CN3CCOCC3=O)CC12)C 15340,c1(CC)cccc(CNC(C2CCCCN2C(C2(C)CC=CC2)=O)=O)c1 15341,C1(OC)C(OC)CN(C(c2ccon2)=O)C1CNC(C1(C)CC2CC2C1)=O 15342,c1(N(C(CCNC(c2cc(CCC)[nH]n2)=O)C)C)ccc(S(C)(=O)=O)cn1 15343,c1(C(N2CC3N(C(c4ccc(OC)o4)=O)C(CC3)C2)=O)cn2cccc(Cl)c2n1 15344,c1(C(=O)NCCC(C)NCC2(C)CCC(=O)C2)ccnc2c1cnn2C 15345,C1(N(CC#C)C(c2cc(CCO)on2)=O)CCN(C(=O)COC2CCC2)CC1 15346,C(=O)(C1(Cl)CCCC1)NC1C(NC(c2ccc3c(c2)CC3)=O)CCC1 15347,C1(NC(C2(C)CC(=C)C2)=O)CN(C(c2cncc(CC)c2)=O)CC1C(F)(F)F 15348,c1(NC(C2(NC(C3CCC(N=[N+]=[N-])C3)=O)CCCCC2)=O)cc[nH]c2nccc1-2 15349,CN1CCN(C(=O)CC2CN(C(=O)CCC(C)(C)F)CCO2)CCC1=O 15350,C1(NC(C2C(C)CCO2)=O)CCSC12CN(C(C1CCCCC1N=[N+]=[N-])=O)C2 15351,C1(C(C)NC(C(C2CCCC2)NC(C)=O)=O)CCN(C(C2(O)CCOC2)=O)C1 15352,c1(OC)cc(O)ncc1C(=O)NCC1CCN(C(=O)CC2CC2(C)C)C(C)C1 15353,C1(C(N2CCC(C(C)(C)NC(CCC#C)=O)CC2)=O)CC2CCCCCC12 15354,C1(CCC)CN(C(c2cn(C)nc2C2CCC2)=O)CCN1C(=O)CCF 15355,c1(SC)ncc(C(=O)NCCC2CCN(C(c3cnn(C)c3N)=O)C2)c(O)n1 15356,Cc1cc(O)nc(C)c1C(N1CC2(CO)CC1(CNC(=O)C#CC(C)(C)C)C2)=O 15357,C1(CCC)CN(C(c2sccc2F)=O)CCN1C(C1CC(=O)NC(COC)C1)=O 15358,c1(CC)cc(C)ccc1C(=O)NC(C1CCCCC1)CNC(=O)C(C)(O)C(C)C 15359,C1(C(=O)NCC(n2cc(-c3cc(OC)c(Cl)cc3)nn2)C)Cc2ccccc2O1 15360,N1(C(C=COCC)=O)CC2C3CCC(C2C1)N(C(c1coc(C(F)(F)F)c1)=O)C3 15361,N1(C(C=C(C)C(F)F)=O)CCCCC1c1n[nH]cc1C(=O)N(CC(N)=O)C 15362,C1(C(N2CCC(F)(CNC(=O)C(Cl)=CCl)C2)=O)Cc2ccccc2O1 15363,S(=O)(=O)(C1CCCN(C(=O)C2CC2)C1)N(C1CC1c1ccc(C#N)cc1)C 15364,c1(N(C)CC)ncnc2c1ncn2CC.N12CCC(C1)SCC2=O 15365,N(C(=NCCC(C)F)NC1CC1C1CC1C)C(C)C1CC1 15366,Cc1ccc(C(=O)NC2CCN(C3CC3)C2)cc1Cl 15367,C(=O)(CS(=O)(=O)CC)N(C)OC(c1cnn(CCCC)c1CC)=O.n12cc(nn1)C2 15368,N1(C(CN(CCOC)C)=O)C(CNC(c2nc(Cl)ccc2F)=O)CC2COCC12 15369,c1(C(=O)NCC2C(NC(c3cn(CC=C)nn3)=O)C2)cc(OC)cc(Br)c1 15370,c1(N2CCC(=C)C2)nc(=Nc2cccnc2C)[nH]c2c1ncn2C 15371,C=C(C(=O)N1CCC(C(=O)OC)C1)C1CCN(C(=O)OC(C)(C)C)CC1 15372,N1(C(Cc2nc(CC)sc2)=O)CCC(NC(C2CC=CCC2)=O)C1(C)C 15373,N1(C(c2ccc(F)cn2)=O)CCCCCC1C(N1CCCC1C(=O)NC1CC1)=O 15374,c1(C(=O)NC(CNC(C(C(C)C)C)=O)CO)cc(N)cc2ccccc12 15375,c1(C(=O)NCCC(C)NC(C2CC23CC(O)C3)=O)cnc(C(F)F)nc1 15376,C#CCCN=C(NCCC(C)F)N1CCC(C2CC2)C1 15377,C#Cc1ccc(C(=O)NC2CN(C(C3CC(C(=O)OC)=NO3)=O)CC2(C)C)nc1 15378,N1(C(C2(C)CC=CC2)=O)CCCC(CCNC(c2ncsc2C2CC2)=O)CC1 15379,N1(C(c2ccc(CC)s2)=O)CCC(C(=O)NCCCN2CCCC2C)CC1 15380,c1(C(N2CC(O)(CC(=O)NC(C3(C)CC3)CO)C2)=O)ccncc1O 15381,C(C)(CNC(c1coc(C(C)OC)n1)=O)(C(C)C)NC(Cc1cn(CC)nn1)=O 15382,c1(OC)ccc(NC(c2sccc2Cl)=O)c(OC(F)F)c1 15383,Cc1cccn2c(C(N3CCCC(NC(c4cccn4C)=O)CCC3)=O)cnc12 15384,C(=O)(CC(C)(C)CNC(C1CC=CCC1)=O)NCC1CCCC(C)O1 15385,N1(C(c2c(C)cn(C(C)C)c2)=O)CCN(C)C(CNC(c2n[nH]c(C)c2C)=O)C1 15386,C1(CNC(C(C(C)C)SC)=O)CN(C(=O)CC(C)(C)C)CC1(C)C 15387,c1(C(N2CCC(OCCNC(c3ncc(C)nc3)=O)C2)=O)cn2nc(C)sc2n1 15388,c1(OC)ccc(N2CCC(C(c3ccccc3Cl)OC)CC2)nn1 15389,C1(C(=O)NCCNC(c2c(C(C)C)n(CC3CC3)nc2)=O)CN(C)C(=O)CCO1 15390,C1(NC(C2CC(NC(C3CCSCC3)=O)C2)=O)C=CCCCC1 15391,C#CCC(C)(C(=O)NCC1CCCSC1)NC(=O)CCc1cncn1C 15392,C1(C)(C(=O)NCC(CNC(C(CC)C2CCC(=O)N2)=O)O)CC(C)(C)C1 15393,C(CCC(C)(C)C(=O)N1CCCC1C(N1CC(O)(CCO)C1)=O)OC 15394,N1(C(c2n(C(C)C)cnc2)=O)CC2C(CNC(=O)Cc3ccncc3Cl)C2C1 15395,c1(NC(C)C)ccccc1N(CC(=O)OC)C(=O)NC1CCC1C 15396,c1(C(=O)NCCCCCN(C(C2C(OCC)C2)=O)C)ccc(Cl)c(Cl)c1 15397,C1(CNC(C(C)OCCCC)=O)CN(C(=O)CC(C)(F)F)CCC1(F)F 15398,c1(C(N2CC(C)C(NC(=O)C(C)(C)CN(C)C)C2)=O)nc(Cl)ccc1F 15399,c1(C(=O)NC2(C)CN(C(c3c(C)ccc(OC)c3)=O)C2)cccc2nc(O)oc12 15400,c1(C(=O)NC2CCN(C(c3c(CC)nccn3)=O)C2)c(Br)sc(C)c1C 15401,n1(CC)ccc(C(=O)NCC2(C(N3CC(CO)CC3C)=O)CC(C)(C)C2)c1C 15402,c1(N2CC(NC(C3CC4(CCC4)CO3)=O)CC(C)(C)C2)nc2cccc(F)c2s1 15403,C1(CNC(C(CNC(c2ccnc(O)c2)=O)OC)=O)CC2(CC2)C(=O)O1 15404,Cc1ccc2c(CC(=O)N(C)CCOCCNC(C3(C)CCCC3)=O)c[nH]c2c1 15405,N1(C(C2CC=C(C)CC2)=O)CC2CC1CCC2NC(=O)CCc1cn(C)nn1 15406,Cc1ccc(C(=O)NCC2CC2NC(C23CC(F)(C2)C3)=O)cc1C#N 15407,n1(CCC(=O)N(c2ccccc2)CC)nnnc1C(C(C)(C)C)NCc1cnoc1 15408,C1(C(=O)NCc2cc(OC)no2)CCC2(CN(Cc3ccc(C#N)cc3Cl)C2)O1 15409,N1(C(C)=O)CCN(C(=O)NCC2COCOC2)C(C)C1 15410,N1(C(C=C(CCC)C)=O)CCCC2CN(C(=O)CCCOCCOCC)CCC12 15411,c1(CNC(C(=Cc2ccco2)C)=O)nnn(C)c1C(N1CCC(C)(CO)C1)=O 15412,C=CCC(C)(CNC(C1CCCC1CNC(c1coc(COC)n1)=O)=O)CO 15413,N1(C(C)C(=O)NC(C)(C)C)CCN(C(=O)CCCCC2CC2)CC1 15414,C1(NC(C2CS(=O)(=O)C2)=O)C2CC3CN(C(=O)COc4ccc(O)cc4)C1C3C2 15415,CC1(CNC(c2cnc(Cl)s2)=O)CCCN(C(c2c[nH]ccc2=O)=O)C1 15416,C12(N(C)C(C3CCCC3O)=O)CCC(CN(C(=O)COc3cccnc3)C1)C2 15417,C12(C(=O)NCC(CNC(C(C)Cc3ccco3)=O)F)CC(C1)C(C(F)(F)F)O2 15418,c1(C(=O)Nc2ccnc(C(C)(C)C)n2)cn(CCO)c(=O)nc1O 15419,C1(C)(OC)CCN(C(C2CC3C=CC2CC3)=O)CC1 15420,C1(C#N)(C(=O)NC(CC(C)NC(C(C)OC)=O)C)CC1(C)C 15421,C#CCC(C)(CC)C(=O)NCc1csc(C(=O)N(CCCC(=O)NC)C)c1 15422,N1(C(c2cnc(C)s2)=O)CCC(C)C(NC(C2CC(n3cnnc3)C2)=O)C1 15423,N1(C(C(CC)=CC)=O)CCC(C)C1C(=O)NCC(F)Cl 15424,C(C(=O)NC1CC(C)(NC(c2ccon2)=O)C1)(C(C)C)n1ncc(C)c1 15425,C1(C(=O)NCCOCCOC)CCOC1C(N(CCC(=O)NC)CCO)=O 15426,O=C(CC(CNC(C1CCC2CC12)=O)C1CCC1)NCC1(Cl)CC1(F)F 15427,C1(CNC(=O)COCC2CCOC2)CC(F)(F)CN1C(=O)CC12COCC(C1)C2 15428,c1(CC(=O)N(CCNC(=O)C(C2CCC(=O)N2)C)CC)cn2cccc(C)c2n1 15429,C(=O)(C(C(C)C)NC(=O)C(C)C)N(CCN(C(C(C)OCC)=O)C)CC 15430,c1(OC)ccnc(-n2cc(-c3ccnc(CNc4cc(C(=O)O)c[nH]4)c3)nn2)n1 15431,Nc1c(C(=O)NCC(C2CC2)NC(C2(c3cccs3)CC2)=O)cccc1Cl 15432,Cc1cncc(C(=O)NCCC(C)CCNC(c2coc(CC3CC3)n2)=O)n1 15433,c1(C(=O)NCCC2(NC(C(C3CC3)SC)=O)CC2)ccc(Cl)o1 15434,Cn1nc(C(=O)NC2CCOCC2C(=O)NCCc2cocn2)cc1F 15435,N1(C(C)=O)CCOC2(CCN(C(=O)C(c3cccc(Br)c3)O)C2)C1 15436,c1(C(C)C)nc(C(=O)NCC(C2CC2)N(C(=O)C(c2cscn2)N(C)C)C)co1 15437,N1(C(Cc2nccc(OC)n2)=O)CC(NC(C23CCC(C2)OC3)=O)CCC1C 15438,C(CC(C)C)(C(=O)N1CCCC(N(C)C(c2[nH]ccc2C)=O)CC1)NC(=O)OC 15439,c1(CC(N2CC(CCn3cc(CC(C)(C)C)nn3)C2)=O)c[nH]ccc1=O 15440,c1(CN(CCNC(c2n[nH]cc2Br)=O)C(C2CC2C(F)F)=O)ccccc1 15441,c1(NC(c2c(-c3c(C)csc3)cncn2)c2ccccc2)ccc2cc[nH]c2n1 15442,CC(C)(C)C(CCO)NC(C1(CNC(=O)C2=COCCC2)CC=CC1)=O 15443,Cc1ccc(CCCCC(=O)NCCCC(C)NC(C2COCCN2C)=O)cc1 15444,C1(CNC(CCCOCC)=O)CC2CCC1N(C(C1(C)CCCS1(=O)=O)=O)C2 15445,C1(NC(c2c(C)ocn2)=O)CN(C(c2cc(Cl)cn2C)=O)CC1C 15446,c1(C(=O)NC2CN(C(C3N(C)CCOC3)=O)CC2F)cccc2nn[nH]c12 15447,C(=O)(CCOCCOCCNC(C1(CC(C)C)CCC1)=O)N(CC=C)C1CC1 15448,c1(OC)cccc(OC)c1NC(C1CSCCN1Cc1cccc(O)n1)=O 15449,c1(C(=O)NC23CCN(C(CCCCCC)=O)CC2C3)cn(CC)c2ccccc12 15450,C1(CC(=O)NC2CCN(C(CCCC)=O)C2CC)NC(=O)CN(C)C1=O 15451,CC(C)CC(CNC(c1cnn2ccccc12)=O)C(=O)NC1COCCC1(F)F 15452,c1(-c2ccc(C)c(C)c2)ccc2c(c1)CNC2.c1(C=O)cc(Br)cc(Cl)c1O 15453,C12(C(=O)NC3CC4C(NC(c5c(OC)cncn5)=O)C4C3)CC=CCN1CCC2 15454,N1(C(c2nc(CC)oc2C)=O)CCC(C)(C)C(NC(c2cc(C)nc(O)n2)=O)C1 15455,C1(NC(c2cnc(Br)s2)=O)C2CN(C(c3cnoc3C3CCC3)=O)CC12 15456,c1(C(=O)NC(CC)CNC(C2CCCC2(C)C)=O)cccc2c[nH]nc12 15457,c1(C(=O)NCC=CC(=O)NC(CN(CCCC)C)C)cccc(C)c1N 15458,N1(C(C(C)C2CCOC2)=O)CC(NC(=O)C(C2(O)CCCC2)F)CC(C)(C)C1 15459,CCC(CC)(C(=O)N1CCN(C(c2cc(COC)on2)=O)CC(C)C1)C(C)C 15460,N1(C(CC(=C)C)=O)CCC(O)(CNC(c2ccnc(OC3CCCCC3)c2)=O)C1 15461,C1(CC)(CC)SCCNC1C(=O)NCc1ccc(N2CCCCC2C)cc1C 15462,Cc1nc(C(N2CCC(C3CCCCN3C(=O)Cc3cnc[nH]3)C2)=O)c(C)s1 15463,C12(C(=O)NC3(CO)CN(C(C4C(C)(C)C(=O)C4)=O)C3)CC=CC(C1)OC2 15464,O=C1CC(CC(=O)NCC2(NC(C3CC3OCc3ccccc3)=O)CC2)CN1 15465,CCCCC(CN(C)C(c1cc(CNC(C2(C#N)CC2(C)C)=O)ccn1)=O)CC 15466,Cc1cc2c(cc1NC(=O)CN1CC3CC1CN3C(N)=O)OCO2 15467,n1(CC(=O)N(CCOCCNC(CC(CCC)C)=O)C)nc2ccccn2c1=O 15468,c1(CC(CC)C)nc(C2CCC2(F)F)n(-c2cccc(F)c2)n1 15469,Cc1cc(S(=O)(=O)N2CC3CCCCC23C)c(C)cc1-c1cc(F)cc(F)c1 15470,C1(NC(C(C)(O)C2CCC2)=O)CN(C(c2cnc(C(F)(F)F)nc2)=O)CCC1F 15471,c1(C(=O)NC2(CC)CCOC2)nc(C)ccc1F 15472,CC1(C)CN(CC(=O)NC2COCC2CNC(=O)CNC(=O)C(C)(C)C)C1 15473,CS(=O)c1ccccc1CC(N1CCC(N2CCNC(=O)C2)CC1)=O 15474,C(=O)(CCCC(=O)NCC1CC1CNC(c1c(C)nn(C)c1C(F)(F)F)=O)OC 15475,C1(C(=O)NC2C(NC(c3occ(C)c3)=O)COC2)CC2CCCC(C1)C2 15476,N1(C(=O)C(Cl)(Cl)Cl)CCC2(CC1)CN(S(=O)(=O)Cc1ccccc1Br)C2 15477,C1(F)(CNC(CC2N(CC)CCOC2)=O)CCN(C(=O)CN(C)S(N)(=O)=O)CC1 15478,c1(C(=O)NCC(C(C)C)NC(=O)C(c2ccc(Cl)s2)=O)ccnc(O)c1 15479,C(=O)(C(CC)C(=O)NC(CN=[N+]=[N-])C(=O)NC(c1ccc(C)cc1)C)OCC 15480,Cc1ccc(C(=O)NC2C=CC(CNC(c3csc(Cl)n3)=O)C2)c(N)c1F 15481,c1(Nc2cccc(C(=O)NC(C)CCNC(=O)CO)c2)ccc2[nH]ccc2n1 15482,C(=O)(C1CCC(=O)c2cccn21)NC1(CNC(CC(C)P(C)(C)=O)=O)CCCC1 15483,c1(NC(C(=O)NC(C)C(C)(C)NC(c2ccccc2CO)=O)=O)ccc(Cl)nc1 15484,c1(OC)ccc(C(=O)NC2CC(NC(=O)C(F)C(C)C)C(O)C2)cc1Cl 15485,N12CC(C(Cc3ccccc3)C1)NC(=O)C1(CC2=O)CC1.c1(C)occc1F 15486,c1(C(=O)N(C)C)ccccc1SC(C)Cn1cc(C(c2cccc(Cl)c2)OC)nn1 15487,C1(CNC(C2C(C(N)=O)C2)=O)CCC2(CCC2)CN1C(C1(C(F)(F)F)CC1)=O 15488,c1(C(=O)NC(C2CN(C(=O)C(C)(F)C(F)(F)F)CCO2)C)cc2n(c1)CCCC2 15489,C12(NC(=O)CSc3nc[nH]n3)CC1CN(C(C1CC1C(F)(F)F)=O)C2 15490,N1(C(C(C)Cn2cccn2)=O)CCN(C(=O)C(c2ccc(Cl)cc2)O)CC12CC2 15491,C1(O)(CCC)CN(C(C2(CNC(=O)C(C)CC3CCCC3)CCC2)=O)C1 15492,c1(C(=O)NCC(C2(O)CN(C(C=CSC)=O)C2)(C)C)ccnc(O)c1 15493,C1(C(=O)NCC(CC)NC(=O)CCN(C)CC)CCc2nc(C)ncc2C1 15494,Cc1nnc(NC2CC(C(F)F)C2)nc1C.n12ccc(n1)CCNC(=O)C2C 15495,c1(SC)ccc(O)c(C(=O)NCC2(O)CCCN(C(C3CC3C)=O)C2)c1 15496,C(CCN=C(NCC1CCSC1(C)C)N1CCN(CC2CCCO2)CC1)OC 15497,N1(C(c2ccc(CC)cc2)C(=O)NCCCOC)CCC(F)(F)C(C)C1 15498,CN=c1[nH]cc(C(=O)N(CCCN(C(=O)CCOCc2ccccc2)C)C)o1 15499,CCCCCCCCCC(C)CC(c1nnnn1C(C)C)NCCC1(C)COC1 15500,CN1CCC(O)(CC(N2CC(C)(NC(c3ccc[nH]3)=O)C2)=O)CC1 15501,Cc1cc(C(N2CCN(C(=O)CSC(C)C)CC2C(C)C)=O)n2nccc2n1 15502,c1(OC)ccccc1C(O)C(=O)NCC(CNC(c1c[nH]nc1OC)=O)OC 15503,CCCC(C(=O)NCCCN(C(c1ccn2cccc2c1)=O)CC)C(C)C 15504,c1(C(=O)NCC(C)C)cc(CNC2CCN(C3CCOCC3)C2=O)oc1C 15505,CC1CN(C2CC3CC2CN3C(C2CCCCC2(F)F)=O)CCCC1(C)O 15506,Cc1cnc(C)c(C(=O)NC(C2CCCN2C(=O)C(C2CCCCCC2)C)C)c1 15507,c1(C(=O)NCCn2cc(C(N(CC(C)O)CC)=O)nn2)cc(C)n(C)c1 15508,C(=O)(C(CN=[N+]=[N-])NC(=O)C(O)C1CCC1)N(C)Cc1ccccc1 15509,C(CCOCCO)(C(=O)NCC1(Cl)CC1(F)F)NC(C(N1CCNC1=O)C)=O 15510,N1(C(c2cc(OC)no2)=O)CC(C2CN(C(c3ccc(CC(C)C)cc3)=O)C2)C1 15511,N1(C(c2ncn(CC)c2)=O)CCC(CNC(c2cccc(CC(C)C)c2)=O)CC1 15512,Cc1c(F)ccc(C(=O)NCC2CCN(C(C3(C)CC3(F)F)=O)CC2O)c1F 15513,C(=O)(C(O)CC(F)(F)F)N(C)CC1CCCN1C(c1cc2n(n1)CCO2)=O 15514,c1(C(=O)NCC2(COC)CN(C(=O)C(O)C(F)(F)F)C2)ccc2oc(C)nc2c1 15515,N1(C(C2C(NC(c3cn(C(C)C)nc3)=O)COC2)=O)CCC(O)C(F)C1 15516,c1(C(=O)NC(C(=O)NC(CCC=C)C)COC)cc(O)nc(O)n1 15517,C#CC12CCC(C(N3C4CCCC3CN(C(=O)C(C)OCC)C4)=O)(CC1)CC2 15518,c1(OC)ccc(C)cc1C(=O)N(CCCNC(c1nnn2c1CCC2)=O)C 15519,C1(NC(CCOc2c(CC)cccc2)=O)CC(F)CN(C(=O)C(F)C2CCC2)C1 15520,S(=O)(=O)(c1ccncc1)NC1CCC(CC(=O)NC2CCC(F)(F)C2)CC1 15521,c1(CC)sc(C(=O)NCC#CCNC(=O)Cc2ccc(Cl)cn2)cc1C 15522,N1(C(CCCC(=O)OCC)=O)CC2CC3CC2C1C3NC(c1coc(C)c1)=O 15523,c1(C(N(CCCCNC(C2(Cl)CC2(C)C)=O)C)=O)ccn2c1CCCC2 15524,C(CC(C)(C)COC)C(c1ccoc1C1CC1)=O.c12cc(cs1)CNC2=O 15525,c1(C(=O)Nc2n(CC)nc(C(C)(C)C)c2)ncnc2c1ncn2C 15526,Cn1nc(C(N2CC=CC(NC(C3CN4CCC3CC4)=O)C2)=O)c2c1CCOC2 15527,c1(OCC)ccccc1CC(=O)N(C1CCN(C(=O)CCOCC2CC2)CC1)C 15528,C1(CNC(CCC2CCC(C)O2)=O)(Nc2nnnn2C)CCOCC1 15529,N1(C(CCC)=O)CCN(C(=O)C(c2cnn(C)c2)C)C(c2cccc(F)c2)C1 15530,C(=O)(C1=NOC2(CCOC2)C1)NC1C2CCN(C(C=C(C)C3CC3)=O)C21 15531,c1(C(N2C(C(=O)O)(CC)CC(OC)C2)=O)cc2scc(Cl)c2[nH]1 15532,N1(C(COCCOCCOC)=O)CC2(CC2)CC1CNC(=O)C(C)CC(N)=O 15533,CC(CNC(=O)CC(O)C1CCCC1)C(F)C(=O)NCCc1ccccc1 15534,C1(C(=O)NCCC(CCNC(C=NOC)=O)C)CN2CCCN1CC2 15535,C1(C(N2CCC(CCNC(C3CC(O)(c4cccnc4)C3)=O)C2)=O)CC2CC1C2 15536,c1(C(=O)NCC(CN(C(=O)Cn2ncn(C)c2=O)C)O)ccccc1C1(C)CC1 15537,N1(CCNC(c2ccsc2)=O)CCOc2ccc(-c3nn[nH]n3)cc21 15538,c1(C(=O)NC(CC)CNC(=O)CC2(O)CCCC2)ccc(Cl)cc1O 15539,C12(NC(C3CCN(C(C45CC(OCC)(C4)C5)=O)C3)=O)CCC(CC1)CC2 15540,Cc1oc(C)c(C(=O)NCC(O)CCNC(c2cn[nH]c2)=O)c1Br 15541,C(=O)(C1CCc2cccc(Cl)c21)N1CCC(NC(c2ccccc2F)=O)C(F)C1 15542,C1(C)(CO)CCCCO1.C1(C)(C(NOCCCC(=O)OC)=O)CC2CC2C1 15543,N1(C(C2CN(c3ncc(OC)cn3)CC(F)C2)=O)CC2COCC(C1)C(=O)N2 15544,C1(C)(C(N2C(C(=O)NCC(C)S(N)(=O)=O)CC2)=O)CCC(=O)NC1 15545,N1(C(Cc2cc(C)on2)=O)CC=CC(NC(=O)C(C)(C)CN2CCN(C)CC2)C1 15546,C1(NC(=O)CC2C=CCC2)CC(F)(CNC(c2cc(C(F)(F)F)cs2)=O)C1 15547,C(=O)(C1=CCC2(COC2)OC1)NC(CC)CN(C)C(c1nc(Cl)cs1)=O 15548,C(=O)(CCS(C)(=O)=O)N(C(C)C)CCN(C)C(C1CCCCC1O)=O 15549,CC(c1cnn(C)c1)=CC(=O)N(C1CCCC1)CCNC(=O)CC1CC(CF)C1 15550,C(c1ccccc1Cl)=CC(=O)NCCC1CCCN(C(C(C)(C)OC(C)=O)=O)C1 15551,c1(C(=O)NCC2(O)CN(C(CC3CCCC(OC)C3)=O)C2)ccc2nsnc2c1 15552,CC1(C)CCC(C)(NC(C2CC(=O)CN2C(=O)Cc2cccnc2O)=O)C1 15553,C1(NC(=O)NC(CC=CC)Cc2ccccc2)CC2CCC(C1)N2C 15554,CC1CCC=C1C(=O)NCC=CCC(=O)NOC1CCCC1 15555,C(=O)(CCC(=O)N(C(C)CNC(=O)CCCn1ccnn1)C)N(C)C(C)=O 15556,N1(Cc2ccc(C#C)s2)CCC2(CC(C(=O)NC3CCN(S(C)(=O)=O)C3)C2)C1 15557,C(c1ccncn1)=CC(=O)NC(C)C(C)NC(c1cc(C2CCC2)no1)=O 15558,C(C(=O)NC1CCN(C(C2(F)CC=CC2)=O)C1)(C(C)C)OC 15559,c1(-c2ccc(CNC(C)(C)C(F)(F)F)cc2)ccc2oc(O)nc2c1 15560,C(=O)(C(C)(O)C(C)(O)C(=O)OC)N1CC(c2ccc(COC)cc2)C1 15561,c1(CC(=O)NCC#Cc2cn(C(C)C)nn2)nc2ccc(Br)cc2o1 15562,Cc1ccc(C(=O)N(C2CCN(C(c3cnc(O)o3)=O)C2)CCO)nc1O 15563,n1(CC)cnc(C(N2CSCC2C(=O)N(C)CCc2ccccc2)=O)n1 15564,C#Cc1cc(C(N2CCC(NC(C3CC4CC4C3)=O)C2)=O)ccc1Cl 15565,C(CCN(C(=O)C(C)n1ccnc1)C)(C(C)(C)C)NC(CCOC(C)C)=O 15566,C(=O)(C(F)(F)CNC(C1CC(CNC(=O)CCN(C)CCO)C1)=O)OC 15567,N1(C(C2(C(C)NC(c3ccc(O)nn3)=O)CC2)=O)CCCN(C)CC1 15568,c1(COC)cc(CNC(c2ccoc2CNC(C2(C(C)C)CC2)=O)=O)no1 15569,c1(C(=O)NC2C(CNC(Cc3cc(C)sc3)=O)CCCC2)ccc2nccn2n1 15570,CC1(CNC(=O)CCC2CCCC2)CCCN(C(=O)Cc2ccnc(O)c2)C1 15571,C1(CC(C(=O)C(C)(C)n2ccnn2)=O)C(NC(c2ccoc2)C)CC1O.CCO 15572,N1(C(C2C3CCCC23)C(=O)NCCC)CCCC(c2ccc(Cl)cc2)C1 15573,CC1(O)CCCN(C(C2(NC(c3cc(Cl)c[nH]3)=O)CCOCC2)=O)C1 15574,C#Cc1ccc(C(=O)OCC(=O)NC(CO)(C(F)(F)F)c2ccc[nH]2)cc1Br 15575,c1(NC2CC(C(=O)OC)CN(C(=O)NCCO)C2)cc(Br)c(OC)cc1C 15576,c1(-c2cccc(-c3c(C)cccc3)c2)ccncc1S(=O)(=O)NC(CO)C(C)C 15577,N1(C(C(C=CCCC)O)=O)CCN(CCNC(=O)C(C#N)CC)CC1 15578,c1(C(=O)NCCOCCNC(=O)CCCC2CCCOC2)ccc(C2CC2)cn1 15579,C1(C(=O)O)CCC2(CCC2)N1C(C1CC(c2cccc(Br)c2)C1)=O 15580,CC1(C)CCN(C(=O)C2=CCCSC2)C1CC(N1CCOCC1)=O 15581,C12(CNC(C(CC)O)=O)COC(CNC(=O)Cc3ccc(OC(F)F)cc3)(C1)C2 15582,C1(C(=O)NC2C=C(C)CCC2)CN(C(=O)CN2CCNC(=O)C2)C2(CCC2)C1 15583,CCCC(C(O)C(=O)N1CCCC(C(C)(C)C)C1)NC(C1CCOC1C1CC1)=O 15584,N1(C(C2CC(NC(=O)Cn3ccnn3)C23CCC3)=O)CCC(F)(F)C(F)C1 15585,c1(NCC2(N(C)C)CCOCC2)ccc(S(=O)(=O)N2C3C=CCC2CC3)cc1Br 15586,O=C(C1=CCCOC1)NCc1ccn(C2CN(C(C3CC34CCC4)=O)C2)c1 15587,CCC(C)CC(CO)NC(=O)CSCCNC(c1ccncc1CC)=O 15588,C(=O)(C(CC1CCOCC1)C(F)(F)F)NCC(N(C(=O)CS(N)(=O)=O)C)C1CC1 15589,CC(N)CCCC(=O)N1CCC(CC(=O)NCc2ccc(F)cc2F)CC1 15590,Cc1cc(-c2cn(C(C)C(=O)NCC3CC4(CNC(=O)N4)C3)nn2)c(C)cc1Cl 15591,c1(C(=O)NC2C(CNC(C(CCC)F)=O)CCCC2)c(C)cccc1C 15592,N1(C(C(C)NC(C)=O)=O)CC2CN(C(=O)CCc3ccnc(C)c3)CC12 15593,CC(C)C(C#N)C(=O)NC1(C(=O)NCCC2CC=CC2)CSC1 15594,C1(O)(NC(N2CCN(C(c3ccc(Cl)c(F)c3)=O)C3C2C3)=O)CN2CCC1CC2 15595,c1(C(=O)NC(CNC(CSCCOC)=O)CC(C)C)ccc(F)c(Cl)c1 15596,N1(C(CSCC(N)=O)=O)CCC2C(C1)CN2C(=O)C(=Cc1c[nH]cn1)F 15597,CCC(O)C(C)(C)C(=O)NCCNC(C1CN(C(=O)CCCC2CCCO2)C1)=O 15598,Cc1cnc(C(=O)NCC(C)(C)CN(C(=O)CC2COCC(C)O2)C)cc1C 15599,C1(C(=O)NCc2cccc(C)n2)(COC)C=CCN1C(c1sccc1CO)=O 15600,c1(N2CCC(CCNC(=O)C(c3ccc(F)cc3)F)C2)ncnc(O)c1Br 15601,C12(C(N3CCC(O)(c4cn(CCCCCO)nn4)CC3)=O)CCCC(F)(C1)OC2 15602,CC1OC(=O)NC1C(=O)NCC(C)(C)CCNC(=O)Cn1ncnn1 15603,C=CC(C)C(C)C(=O)NCC(C)(C)CNC(=O)CC1(CC(=O)OC)CCCC1 15604,C=C(F)C1(CC(=O)NC2CCCC(NC(C3(C(F)F)CCCO3)=O)C2)CCC1 15605,N1(C(C2CCCC(C)C2)=O)CC2(CNC(c3coc(N(C)C)n3)=O)CCC1CC2 15606,c1(CC(=O)NCC2(F)CCC(NC(=O)CC3CC3)C2)ccc(O)c(Cl)c1 15607,c1(C(N(C)CC2(CF)CCC2)=O)ccc(CCC(N)=O)cc1.C12(CC1)C(=O)NC2 15608,O(N1CCC(NC2CCCN(c3nnc(C)s3)CC2)CC1)CC 15609,N1(C(C2N(CC)CCOC2)=O)CCCCC(N(C(=O)C(F)=CCCF)C)C1 15610,c1(C(=O)NC(CC(C)NC(CCOC)=O)C)ccc(C(C)=O)c(F)c1 15611,C#Cc1cncc(NC(C2CNC(=O)CN2C(=O)C2=COCC2)=O)c1 15612,C1(CNC(CNS(C)(=O)=O)=O)CCC2(CN(C(c3cc(N)c(N)cc3F)=O)C2)O1 15613,S(=O)(=O)(c1ccc(C(F)(F)F)c(C#N)c1)N(C1(C)CCOC1)C 15614,c1(NC(C2C(NC(C3(COCC)CC3)=O)C2)=O)c(O)cccc1C#N 15615,C1(C)(C(N(CCCNC(c2c[nH]nc2C2CC2)=O)CC)=O)CCC(C)C1 15616,C1(CC(=O)NCC23CC(NC(C(N(C)C)C4CC4)=O)(C2)C3)CC(O)C12CCC2 15617,c1(C(=O)NC2CC(CNC(C(C3CCOC3)OCC)=O)C2)scc2c1OCCO2 15618,C1(NC(C2C(OC)CCC2)=O)CN(C(=O)CN2CCC(F)CC2)CC(C)(C)C1 15619,c1(C(N(CC(O)CN(C)C(C2(C)CCCC2(F)F)=O)C)=O)noc2c1CCCC2 15620,N1(C(c2c(N)csn2)=O)CCCC(C2CC2NC(C2CC23CCC3)=O)C1 15621,CCC(C)(C)C(O)C(=O)NCC1CC(C)CN(C(=O)C(F)(F)CO)C1 15622,c1(CC(=O)NC2C3CC(NC(C4C(CC)C4)=O)CC32)ccc2nc(C)[nH]c2c1 15623,c12ccc(cc1)CN(C)C(=O)C2.C1(NC(C2(OCC)CC2)=O)CNC(=O)N1 15624,N1(C(c2c(C)ocn2)=O)CCCC(NC(c2cc(=O)c(Br)c[nH]2)=O)CC1 15625,C1(C(=O)NCc2cc(C(=O)NCC3(Cl)CCC3)on2)(CC)CCCO1 15626,CCCC(C)(C)NC(=O)NC(Cc1ccccc1)C(=O)Nc1cccs1 15627,C#CCCCC(=O)NCC1C=CC(NC(c2ncsc2-c2ccccn2)=O)C1 15628,CCCC(F)C(=O)NCc1cccc(CNC(=O)C(F)CC)c1 15629,c1(CC(N2CC(Nc3ncnc(CC)c3F)C(C)C2)=O)noc2ccccc12 15630,CC1CCCC(O)(C(=O)NCCCCN(C(=O)COc2cnc(Cl)cn2)C)CC1 15631,CCCCC(O)C(C)C(=O)NC1CCOC(C(=O)NCc2occc2C)C1 15632,C(=O)(CCCCC(C)(C)OC)N1C(C(C)(C)NC(CCC=CCC=C)=O)CCC1 15633,Cc1cc(C(=O)NCCC(C)(C)NC(=O)C(=O)N(C)C)nn1CC(F)(F)F 15634,CC1CCCCC1N1CCCC(C(N2CCSCC2)=O)C1 15635,c1(N2CCN(CC(=O)NCc3ccc(C)cn3)C(=O)C2)ccnc2cc(Br)nn12 15636,CCCC(CCCNC(=O)CCC(C)OC)NC(c1cc(F)ccc1N)=O 15637,c1(C(=O)NCC(CNC(C=CC(=O)N(C)C)=O)F)n[nH]c2c1CCCCC2 15638,C1(CC(=O)NCCCC(C)NC(c2c(C)nsc2C)=O)CCCNC(=O)C1 15639,C1(C(=O)NCC2CCCCN2C(c2ccc(F)c(Cl)c2)=O)CC2(CCC2)CCO1 15640,O=S(=O)(c1c[nH]c2cc(Cl)ccc12)N1CC(O)(c2cscc2Br)C1 15641,C=C(C)CCC(C)(c1nnnn1Cc1ccccc1)NC(c1ccc(Br)cc1)C 15642,N1(C(C2CC(=O)NC2)=O)CC2CCC1C(C(N1CCCCC1CCO)=O)C2 15643,Cn1cc(C#N)cc1C(N1CC(NC(=O)CCNC(=O)C=CCl)C(C)(C)C1)=O 15644,C1(C(C)C)CCC(N=c2[nH]c(=NC3CCc4c[nH]nc4C3)[nH]c3ccc(Cl)cc23)C1 15645,N1(C(c2nccc(C)c2)=O)CC(CNC(=O)CCc2cnc(C)o2)CC1(C)C 15646,C1(N(CCC(CC)C)C2CC2)CNCC(F)C1 15647,CC1CCCCCC1Nc1cc(NCCCN2CCCC2)ncn1 15648,CC1CN(C(=O)C(C)C2CCOC2)CC(C)N(C(c2cc(O)cnc2N)=O)C1 15649,C1(CC=C)(NC(=O)CN2CCCCC2C)CCN(C(c2cnn(CCF)c2)=O)C1 15650,C=C1CCN(C(c2ccco2)=O)C(C(=O)NOCCOCCF)C1 15651,N1(C(C(C2CC2)OC)=O)CCC2(C)CN(C(=O)C(O)C(C)(C)C)CC12 15652,CCCCC(C(=O)NCC(C)(C)C#CC(=O)NC1CC(CCF)C1)C(C)C 15653,C1(C(N2CCCC2C2(C(=O)NOCC3CCC3)CC2)=O)COCCO1 15654,C1(C(=O)NC2C(C)(CNC(CSCC=C)=O)CCC2)CCc2nn[nH]c2C1 15655,C(=O)(C(O)CCC(F)(F)F)N1CCN(C(c2c(CC)nns2)=O)C2C1C2 15656,CC(C)C(C(=O)NCCC1(C(=O)NC2CCOC2(C)C)CCC1)N(C)C 15657,c1(OC)cc(C(=O)NCC(C)(C)CN(C)C(C2CC3CC3C2)=O)cc(OC)n1 15658,C#CCC(C(=O)N(C(CO)CC(C)C)C)NC(c1cnc(CC)nc1)=O 15659,c1(NC(C2CCCN(C(=O)C(c3ccccc3)F)C2)=O)nccc(C(F)F)c1F 15660,C#Cc1ccc(C(=O)N(CC(=O)NC(C)Cc2ccco2)C(C)C)o1 15661,C=C(F)C1(CC(=O)N(CC(C)NC(=O)CCCC(=O)OCC)C)CCOCC1 15662,n1(CC(=O)NC2CC(N(C(C)=O)C)C2)cc(C(F)(F)F)cn1 15663,C=CCC(CC(=O)NCC(N1CCC=CC1)=O)NC(=O)Cn1nc(C)oc1=O 15664,C1(CNC(C(C)(C)OC(C)=O)=O)CN(C(=O)CN2CCS(=O)(=O)CC2)CCCO1 15665,c1(C(N2C(C(=O)Nc3ccc(F)cc3Cl)CC3(CC3)C2)=O)c(Cl)cc(F)cc1Cl 15666,c1(CN2C(C(=O)NC(CCC)C)CC3(CC3)C2)c(F)cc(Br)cc1Br 15667,C1(C)(C(=O)NCCN(C(c2cc(CC)c(C)s2)=O)C2CC2)CCC(=O)N(C)C1 15668,CC(C)C(CCO)N=c1ccnc(NC2CNC(=O)OC2)[nH]1 15669,C1(CC(=O)NCC2(C(=O)OC)CCC2)CCN(C(=O)C(C)O)CC1 15670,C(CCCCC(=O)N1CCC(CNC(c2cccc(Cl)c2O)=O)C(O)C1)SC 15671,C1(C(=O)NCC(C)(C)OCCNC(CCC(=O)OCC)=O)CC12CCCOC2 15672,N1(C(CC=CC=C)=O)CC(NC(=O)Cc2cc(=O)n(CC(C)C)[nH]2)C(O)C1 15673,c1(CC)cc(=NC(=O)C(C)(C2CC2)N(C(=O)CC2C=CCC2)C)[nH]n1C 15674,N1(C(C(CC)COC)=O)CCCC12CCN(C(c1cnc(O)n(C)c1=O)=O)C2 15675,c1(C(N)=O)ccc(NCC2CCN(C(C3CCOCC3(C)C)=O)C2)c([N+](=O)[O-])c1 15676,CC(CNC(=O)CCCN(C)C)C(F)C(=O)NCCc1cc[nH]n1 15677,C(=O)(C(CCCCCN)C(C)C)N(C12CC3CC(C1)CC(F)(C3)C2)CC 15678,C1(C(=O)OC)CC(OC)CN1Cc1cccc(C2COC2)c1 15679,N1(C(C2(F)CCN(C(C3C4(CC4)C34CC4)=O)C2)=O)CCC(F)(F)C(O)C1 15680,c1(C(=O)NC2C(C(=O)NCCC)COCC2)cc2cnccc2[nH]1 15681,C(=O)(CCC1=NNC(=O)CC1)NC1(CN(C(c2c(SC)cn(C)n2)=O)C)CC1 15682,C(CC(F)F)(C(=O)NC1C(O)CC1O)N(C)C(C1CCC1)=O 15683,CCC(CNC(C1CC(=O)CN1C(=O)CSCC(N)=O)=O)(CC)CO 15684,C1(C)(C(N(CC(CNC(C(C=C)O)=O)(C)C)C)=O)CCC2CC2C1 15685,C12(C(N3CC4C(NC(c5c(CC)scc5)=O)C4C3)=O)CCC(CC1)C(C)O2 15686,Cc1cc(=NCc2csc(Br)n2)[nH]c(=NCc2nc(C(C)(C)C)n[nH]2)[nH]1 15687,Cc1ccc(CC(=O)NC2CN(C(=O)CCc3cccn3C)CC2C)c(Cl)c1 15688,c1(C(N2CCC(CNC(c3cc(CC)cc(Cl)c3)=O)C2)=O)cccc2c[nH]nc12 15689,Cc1ncsc1C=CC(=O)N(CCC(C)NC(=O)CS(=O)(=O)NC1CC1)C 15690,C1(CNC(C(CC)N(CC)CC)=O)CCN(C(=O)Cc2cncc(OC)c2)CC1 15691,c1(C(=O)NC2C(OC)CN(C(c3cnn(C(F)F)c3)=O)C2)ccc2cc[nH]c2n1 15692,C1(C(=O)NC2CC2NC(=O)Cc2ccn(C)n2)(COC)CCCO1 15693,C1(c2ccc(CC)o2)COCCN1CC(=O)NC(c1ccccc1)CSC 15694,c1(CN2C(CNC(c3c(OCC)nccc3)=O)CCC2)c(F)ccc(F)c1O 15695,C1(NC(C2(OC)CC2)=O)C2CN(C(C3CCCN3Cc3ccccc3)=O)CC12 15696,c1(OC)c[nH]c(C(=O)NC(C)CCCCNC(=O)C(F)n2cccn2)cc1=O 15697,N1(C(C(C(C)NC(C2CC(F)(F)C2(C)C)=O)(C)C)=O)CCOc2ccccc21 15698,N1(C(Cc2nc(C)sc2)=O)CC(NC(c2cc(CC(C)C)c[nH]2)=O)C2CC2C1 15699,C1(CC(=O)NCC(C23CCC(CC2)C3)NC(C2CC(F)C2)=O)CC2C=CC1CC2 15700,C1(NC(=O)CCc2ccc[nH]2)CCC(NC(C2(C(F)(F)F)CCC2)=O)C1 15701,N1(C(C=C(C)C)=O)CC2CC(NC(c3ccc4ncoc4c3)=O)CC2C1 15702,Cc1ccc2ncc(C(=O)NCC(CO)NC(C3(C4CC4)CCC3)=O)cc2c1 15703,c1(C(N2CC(C)(NC(c3cncc(CC)c3)=O)C2)=O)c(C)cc(F)cc1Br 15704,CC1CN(C(C2CCC(n3cc(CN4CC5CC5C4)nn3)C2)=O)CCC1O 15705,N1(C(C(C2(O)CN(C(c3cccnc3O)=O)C2)F)=O)CC2C(C1)C2(F)F 15706,N1(C(C2(C)CC2)=O)CC(C)CN(C(c2ccc(C3CC3)cn2)=O)C(C)C1 15707,N1(C(C2CC(CC)C2)=O)C(C(=O)NOC(C)(C)C)CCC1C1CC1 15708,C#CCC(O)C(=O)NC(C(=O)NC1CC(CCF)C1)C1CCOC1 15709,C1(NC(C(F)=CC)=O)CC2CCC1CN(C(c1cc(C(F)(F)F)ccc1C)=O)C2 15710,c1(C(=O)NC2C(C)(CNC(C3C(=C)C3)=O)CCC2)c(S(C)(=O)=O)cnn1C 15711,CS(=O)(=O)CC(=O)NC(C(=O)N1CC(CC(F)F)C1)C1CC1 15712,CC(CCCCCO)NC(c1nnnn1CCC1CC1)C1(C)CCCC1 15713,c1(NC(C2CC(CCNC(C3C(OC)CC3)=O)C2)=O)cnn(CC2CC2)c1 15714,Cc1cnccc1C(=O)N(C(CNC(=O)C(C)NC(c1cccs1)=O)C1CC1)C 15715,Cc1cnccc1C(C)C(=O)NCC(C)(C)CN(C)C(c1[nH]nnc1C1CC1)=O 15716,C1(NC(C2COCCO2)=O)CN(C(c2ccc(-n3ccnn3)cc2)=O)CC1(F)F 15717,N1(C(=O)O)CC(NC(=S)Nc2cccc(Cl)c2)C(C)(C)C1.CC(C)(C)NCCC#N 15718,CN1CC=C(CNC(=O)CONC(C2(C)C(C)(C)C2(C)C)=O)CC1 15719,C(=O)(CCCCC(=O)OC)NCC1CCC(N(C(C(CCOC)OC)=O)C)CC1 15720,CCCCC(COC)NC(C1(CF)CCN(C(=O)C=CC(F)(F)F)C1)=O 15721,C1(C(=O)NCc2cn(CC#C)nc2)COCCN(C(=O)Cc2scnc2C)C1 15722,c1(C(=O)NCC2N(C(=O)C3=CCCS3)CCC(C)C2)cnc2ccoc2c1 15723,C1(C(=O)NCCN(CC)CC)CCCC1OC(C1CCOC1C(C)C)=O 15724,N1(C(=O)CCCc2cnn[nH]2)CCN(C(C2CC3(CCC3)C2)=O)C(CO)C1 15725,N1(C(C2(OC)CCCOC2)=O)CCC=C(CNC(=O)C(C)C(C)C)C1 15726,C1(CN(C(c2cc(CNC(CCCC)=O)on2)=O)C)CCCCCC1 15727,C1(CC)CN(C(c2cc(CC(C)C)c[nH]2)=O)CCN1C(=O)C=C1CCN(C)C1 15728,Cc1nnc2n1CCCC2C(=O)NC1CN(C(=O)C(c2ccnn2C)C)C1 15729,c1(C(=O)NCC(CNC(C2=CCC(C)CC2)=O)F)ccc2c(c1)CCCS2(=O)=O 15730,c1(CC(N2C(CCNC(Cn3c(C)ccn3)=O)CCC2)=O)cnn2ccccc12 15731,C(=O)(C(C)(C)C)OCC(=O)NCC(n1cc(C2CCCC2O)nn1)C 15732,Cc1cc(C(=O)NCc2ncc(C(=O)NC3CC4CCC3C4)cn2)cnn1 15733,Cc1cn(C)c(CN(C)C(c2csc(C(=O)O)n2)=O)n1 15734,C(=O)(CCC(CF)CF)N1CC2C(NC(c3n[nH]c(C)c3O)=O)(CC2)C1 15735,c1(CCC)nc(C)c(C(=O)Nc2ncc(C(=O)OCCS)cn2)s1.NC 15736,c1(CC(N2CC(CC(C)(C)C)C(NC(C3CC34CC4)=O)C2)=O)ccc(Cl)cc1F 15737,c1(C2(C(=O)[N+](CCOC3CN(C(C(C)CO)=O)C3)(C3CC3)[O-])CC2)cccc(C#N)c1 15738,C(CCN=c1[nH]c(=NCC(C)C2CCC2)[nH]c2c(F)cccc12)N(CCOC)C 15739,C(CCCC1(NC(C2CC2Br)=O)CC1)NC(CC1(COC)CC1)=O 15740,CC1CC(NC(=O)CN2CCN(CCO)CC2)CN(C(C2CCCC2(F)F)=O)C1 15741,c1(C(=O)NCCCC(C)NC(C2CC(CC)C2)=O)cnc(C)nc1COC 15742,N1(C(CCC2C(C)(C)C2)=O)CC2CCCC2(CNC(=O)COC(=O)CO)C1 15743,c1(C(C(=O)NCC(CNC(=O)C=Cc2cnc[nH]2)F)O)ccc([N+](=O)[O-])cc1 15744,C12(NC(C3CCC3)NC(=O)CC3CCCCC3)COC(CF)(C1)C2 15745,C1(C(=O)NCC(C)N(C(c2cn[nH]c2)=O)CC)COCCC1(F)F 15746,c1(C(N(C(C)CNC(c2c[nH]c(C#N)c2)=O)C)=O)ccc([N+](=O)[O-])s1 15747,C(=O)(C(O)C(F)F)N1CCC(N(C(COCCOCC#C)=O)CCC)C1 15748,c1(C(=O)NC2C(CNC(c3ccn(CC)n3)=O)CC2)cc(Cl)cc2c1NCCC2 15749,N1(C(N2CC(O)(CCN(C)C)C2)=O)CC(F)(F)CCC1C(=O)OC(C)(C)C 15750,N1(C(c2ccc(C(=O)OC)s2)=O)CCC2(CCCN(C(=O)C(O)P(C)(C)=O)C2)C1 15751,N1(C(Cn2c(C)ncc2)=O)CC2(CC(CC(=O)Nc3c(O)cccc3Br)C2)C1 15752,C1(C(N2C(C)(CNC(CSCCC)=O)CCC2)=O)COCC(C)(C)O1 15753,c1(C(=O)NC(C(CC)CC)C)n[nH]c2c1CN(C(C1(F)CC=CCC1)=O)C2 15754,N1(C(c2cnc(CNC(C3(C)CCCC3)=O)nc2)=O)CC2CCCC(O)C2C1 15755,Cc1cnc(Br)cc1NC(C1(F)CCN(C(=O)CCc2cccc(C#N)c2)C1)=O 15756,N1(C(C2(SCC)CC2)=O)CC(NC(=O)C=C(C)c2ccsc2)C(O)C1 15757,C12(c3nc(-c4ccc(Cl)cc4)nn3C3CCCSC3)CCCN(CC1)C2 15758,C1(NC(C(CCOC)C)=O)CC2CCC(C1C)N2C(c1cc(CN(C)C)on1)=O 15759,C1(O)(CNC(C2C(c3ccn(C)n3)C2)=O)CCN(C(c2cnsc2)=O)CC1 15760,N1(C(CCC(=C)Cl)=O)CC(NC(C2(c3ccncc3)CC2)=O)CCC1C 15761,c1(NCc2cn(C)[nH]c2=N)[nH]c(=NCC2OCCc3sccc32)nc2sccc12 15762,c1(OC)cccnc1C(=O)NCC1CCC1NC(=O)CC(C)CF 15763,N1(S(C2CC(OC)C2)(=O)=O)c2ccccc2C(C)(C)C1C 15764,C(C(C)(C)NC(=O)CCC1CCC1)N(C(=O)C(C)SC1CCCO1)CC 15765,N1(C(c2n(C)nnc2)=O)CCOC(C(=O)NC2COC3(CCC3)C2)CC1 15766,N1(C(C2C(CCC)C2)=O)CCC2(C(=O)NCC(N3CCOCC3)C)CCCC12 15767,c1(C(=O)NC2(CNC(C3CC(C)(CC)C3)=O)CCOC2)cncc2c1CCC2 15768,c1(CC)cccc(C(N2C(C)C3CC2C3NC(c2ncn(CC)n2)=O)=O)c1C 15769,CC1CCCC1(C(=O)Nc1ccccc1)NC(=O)C(c1cncnc1)C 15770,CCC(CC)(CCNC(C1(F)CCOC1)=O)NC(c1ccc(C)c(Cl)c1)=O 15771,C1(C(=O)NC(C2CCCO2)(C)C)COCCN1C(=O)C=CC1CCOCC1 15772,Cc1[nH]nc2c1CCC(C(N1CCC(C)(CNC(c3c(Cl)n[nH]c3C)=O)C1)=O)C2 15773,Cc1cc(F)c(F)cc1C(=O)NC1CN(Cc2ccc(F)c(O)c2)CC1F 15774,Cc1cc(=N)[nH]cc1C(=O)NCC1(CCNC(=O)C(O)CC(N)=O)CC1 15775,C1(NC(CN2CCCC(CC)C2)=O)CCN(C(=O)CC2CCC(C)CC2)C(C)C1 15776,CCCCCCCCC(=O)NCC(C)(CC(C)C)NC(=O)CC1CC1(Cl)Cl 15777,N1(C(C(C2CC2)SC)=O)CCN(C(c2cccc(F)c2O)=O)CC(O)C1 15778,c1(C(=O)NCC(CO)NC(=O)C(C2CCCC2)C2CCC2)ccc2c[nH]nc2c1 15779,C1(NC(Cc2c(C)noc2)=O)CCN(C(c2ccc(C3CC3)cc2)=O)CC1 15780,N1(C(CCn2ncn(C)c2=O)=O)CCN(C(C2COC(C)(C)CO2)=O)CC(O)C1 15781,c1(Nc2cncc(CNC(C3C=CC(CC)C3)=O)c2)ccc(C)c(C(F)(F)F)c1 15782,c1(C(=O)NCC2(NC(c3c(C#C)c[nH]n3)=O)CCCCC2)cc(C)ccc1O 15783,CCC(CC(=O)NC(C)(C)CNC(=O)CCCNC(c1ccccc1)=O)C(F)F 15784,Nc1cnc(C(F)(F)F)cc1C(N1CCC(F)(CNC(C2CC(F)C2)=O)C1)=O 15785,S(=O)(=O)(c1cncc(Br)c1)N(CC)Cc1cccc(C2CC2)c1F 15786,C1(O)(CCNC(c2cn(C3CCOCC3)nn2)=O)CCN(C(=O)C=C2CCC2)C1 15787,C1(C(=O)NCC(C)C#N)CC(N=[N+]=[N-])CN1C(=O)CC(C)(C)C#N 15788,c1(C(=O)NC(CO)C(O)C2CCCCC2)cnn2ncccc12 15789,c1(OC)cc(CCC(=O)NC23CC(NC(C4CCCO4)=O)(C2)C3)ccc1O 15790,c1(OCC)cccc(C(=O)NC2CCC(CCNC(C3(OC)CC3)=O)C2)c1 15791,CC(C)C(C)C(C)CC(=O)N1CC2(CC2)CC1CNC(c1cccc(F)n1)=O 15792,C12(NC(c3ccc(C)cc3C)=O)CCC(CN(C(=O)CCC3CC3)C1)C2 15793,C1(c2cn(CCOCCNC(c3ncccn3)=O)nn2)CCCCCC1.CCO 15794,C(=O)(C1CCCc2ncnn21)NC(C(C)CSc1ccc(S(N)(=O)=O)cc1)=O 15795,N1(CCC)CC(C(=O)NCCC2(C)CCN(C(c3cncnc3C)=O)C2)CC1=O 15796,CC(C)CC(C)(O)C(=O)NCC12CCC(CC1)N(C(C1CCSCC1)=O)C2 15797,C(CC(F)=C(F)F)NC(C12CC(NC(=O)C=Cc3cc[nH]c3)(C1)C2)=O 15798,c1(C(=O)NCCC(C(C)C)C)cccc2c(Cl)cccc12 15799,c1(OC)cc(C)c(CN(CC([Si](C)(C)C)c2ccccc2)CCO)cc1OC 15800,C1(CC=C)(NC(c2cnccc2C)=O)CCCN(C(C2CC(OC)C2)=O)C1 15801,N1(C(c2ccn(CCC)n2)=O)CC2CN(C(=O)Cc3cc(O)nnc3O)CCC12 15802,N1(C(CC(=O)OC)=O)CCCCC1C1CCCN1C(c1cnn(C)c1)=O 15803,c1(NC(N2CCN3CC(F)CC3C2)=O)cc2c(cc1Br)OCCO2 15804,Cc1ccc(C(C)CC(=O)NC23CC(NC(c4cncc(N)n4)=O)(C2)C3)cc1 15805,C1(C(=O)NC2C(NC(c3c(C)nn[nH]3)=O)CC2)CCCC2(CC2)C1 15806,C1(C(=O)NCC2(NC(C3CC(CC)C3)=O)CCOC2)CC2CC1CC2O 15807,c1(C(=O)Nc2cccc(NC(C3CSCCS3)=O)c2)c[nH]c2cc(F)c(F)cc12 15808,c1(C(C)(C)C)ccc(C(=O)NC2CC2CNC(=O)C=Cc2cncs2)nc1 15809,c1(NC(C(C)NCc2ccccc2Cl)=O)ncc(-c2cncc(O)c2)cc1O 15810,c1(NC(=O)NC2C(O)CCC(C)C2)ccc([N+](=O)[O-])cc1I 15811,c1(NC(C2C3CN(C(C(C)Cc4ccccn4)=O)C2C3)=O)cc(Cl)nnc1Cl 15812,C1(C(=O)NC(C(C)C)(C)CNC(c2ccn(C3CCC3)n2)=O)CCCCCCC1 15813,C(=O)(C1=CNS(=O)(=O)N=C1C)NC1CN(C(C2CCN(C(CC)=O)C2)=O)CC1C 15814,c1(NCC2C(C(C)C)C2)ccc(S(=O)(=O)NCCC2OCCC2C)cc1Cl 15815,N1(C(C2OCC(C)C2)=O)CCOCC(CNC(=O)CC2NC(=O)NC2=O)C1 15816,C(=O)(C1=CNC2=NCCC2=C1)N1CC(O)(CNC(=O)CC2CCCCCO2)C1 15817,C1(NC(c2c(OCC)nc(Cl)cc2)=O)CC2CN(C(=O)C(C)(C)O)CC2C1 15818,CC(c1ccccc1)=CC(=O)NCC1CN(C(C2(CO)CC2)=O)CCN1C 15819,c1(CC)cnc(CNC(=O)C(c2cnn(C)c2)NC(c2cc(C)c[nH]2)=O)[nH]1 15820,CC(C)CC(C(=O)NCC(C)(C)CCNC(=O)CC1CCCN1C)C(C)C 15821,C1(CC(=O)NCC=CCNC(C2CC3OC(=O)OC3C2)=O)CCc2sccc2C1=O 15822,C(CCS(=O)(=O)c1ccccc1)C(CC)CC(C)(O)CC.N 15823,c1(C(N(C2CC(NC(CN(CC)CC)=O)C2)C)=O)cnn2c1CCCC2 15824,N1(C(C(C)=CC)=O)CCC(NC(=O)CC(O)c2ccccc2)C1(C)C 15825,c1(C(=O)NCCCCN(C)C(c2cc(C3CC3)ccc2Cl)=O)cc([N+](=O)[O-])n[nH]1 15826,N1(C(C2(C(F)F)CC(F)(F)C2)=O)CC2ON=C(CNC(C3(C4CC4)CC3)=O)C2C1 15827,N1(C(CCCN(C)C)=O)CCN(C(=O)CCCC2CCOCC2)C(C2CC2)C1 15828,n1(CC)nc(C2CCOCC2)cc1C(=O)NC1CN(C(=O)OC)CC1NC(C)=O 15829,C1(S(N)(=O)=O)(C(=O)NCCNC(C(c2ccc(Cl)cc2)(C)N(C)C)=O)CCCC1 15830,C1(C(N(C2CN(C(c3n[nH]c(C)c3O)=O)CC23CC3)C)=O)CCc2cnnn2C1 15831,CC1(Cc2cn[nH]c2)CCCN1C(=O)NC(c1ccncc1)C1CCCC1 15832,C=CCC(C(=O)NC(C)CN(C)CCOC1CCCCCC1)C(C)C 15833,c1(CC(=O)NC2CC(C)(NC(c3cnc[nH]3)=O)C2)ccc(-n2cnnc2)cc1 15834,C(=O)(C1COc2ccc(F)cc21)N1CCC(NC(C2(C(F)(F)F)CC(=C)C2)=O)C1 15835,c1(CC(N2CC(c3ccccc3)(NC(C3CCC3)=O)C2)=O)cnn2c1OCCC2 15836,c1(C(=O)NCC#C)ccc2nc(C(F)(F)F)sc2c1.C12(CC1)C(=O)OC2 15837,c1(CSCC)ccc(C(=O)NC(C)CC2CN(C(=O)C(F)CC)C2)cc1 15838,c1(C(N2CC3CC2CO3)=O)cc2n(n1)CCCN(Cc1cc(F)c(Cl)c(F)c1)C2 15839,N1(C(C2(C=C)CC2)=O)CCC(C2(CNC(C3CCC(=O)N3)=O)CCOCC2)CC1 15840,c1(CN2CCN(CC(=O)Nc3ccc(F)nc3)C(=O)C2)cc(F)c(O)cc1F 15841,C=C(C)C1OCCC1C(N1CCCCC1CNCc1cc(OC)cc(OC)c1)=O 15842,c1(OC)ccc(OC)c(CCC(=O)NCC(C2CCC2)NC(=O)CC=C(C)C)c1 15843,c1(OC)cccc(C(=O)NCC2(F)CC(NC(c3c[nH]nc3C(F)(F)F)=O)C2)c1 15844,CC(C)C(CNC(c1cn(CC2CC(=O)C2)nn1)=O)NC(C1CC12CCC2)=O 15845,c1(C(N2C(CN(C)C(C3CCC(C)(C)O3)=O)CCCC2)=O)ccc2ncsc2c1 15846,C1(c2n(-c3cccc(C)c3)nc(Sc3ccc(N)c(F)c3)n2)CCS(=O)(=O)N1C 15847,N(C(=NCCSC)N1CCC(Cc2cnn(C)c2)C1)CC1CCN(C(=O)OC)C1 15848,N1(CCNC(c2c(OC)nsc2)=O)CCC(NC(=O)C#CC(=O)N(C)C)CC1 15849,C1(NC(c2c(OCC)cccc2)=O)CCN(C(=O)CCC2CC2(F)F)C(C)C1 15850,c1(C(N2CCC(C(CNC(C(CC)NC(C)=O)=O)O)CC2)=O)c[nH]c(=N)cc1C 15851,C(c1nc(C)co1)=CC(N1CC(CNC(C(c2ccccc2F)OC)=O)C1)=O 15852,C12(CNC(c3n(C)ccc3)=O)CCCC1CCN2C(c1csc(CO)n1)=O 15853,CC(CN=c1nc(N2CCc3ncncc3C2)c2c([nH]1)COC2)c1nccs1 15854,c1(OC)cc(C)cnc1C(N1CC(CNC(c2cc(C)co2)=O)C(C)(C)C1)=O 15855,C1(NC(C(CN(C)C)O)=O)C2CCN(C(=O)CCSc3nnnn3C)C12 15856,CCC(C(=O)N1CCCC1CC(=O)NC(C)(C)C#CC)NC(C)=O 15857,C(c1ccoc1)=CCN(C(=O)CC1CCN1C(=O)COCC1CCOC1)C 15858,N1(C(CN2C(C)CCC2)=O)CC2CC1CCC2NC(c1ccc(F)c(CO)c1)=O 15859,Cc1cccc(OCCC(N2CC(NC(=O)Cc3occc3C)C(C)C2)=O)c1C 15860,c1(C(=O)NC2C(NC(C(CC)N(C)C)=O)CCOC2)cccc2[nH]cc(C#N)c12 15861,C1(C(N(CCNC(C)=O)C)=O)CC2CC1CC2NC(c1cncc(O)c1)=O 15862,Cc1ncc(-c2cn(CCOc3sccc3-n3ccnn3)nn2)o1 15863,N1(C(C2CCC(=O)N2)=O)CCCCC1CNC(C1CCC(O)CC1)=O 15864,c1(C(=O)NC(CC(C)C)C(=O)N2CCC(N3CC=CC3)C2)ccn2ccccc12 15865,C#CCCCC(C)C(=O)N1C(CNC(c2sccc2C#N)=O)CC2CCCC12 15866,C(=O)(C(C)CNC(C1CCSCC1)=O)NC(c1ncco1)C 15867,C#CC1(c2ccccc2)COCCN1C(=O)NCCc1cn(C(C)C)cn1 15868,C=CCC(C)(C)C(=O)N1CCN(C(C2CC23CC(OCC)C3)=O)C(CF)C1 15869,N1(C(c2cnc(CCC)s2)=O)CC(C)(CNC(=O)CCCC(C)(C)C)CC1(C)C 15870,N1(Cc2ccc(C#N)cc2)CCC2CN(C(c3csc(Br)c3)=O)CC2C1 15871,c1(OC)cc(Br)ccc1C(C)NC(C1C(CO)C1(C)C)=O 15872,c1(OCC(N2C(C(N(CC(=C)C)C)=O)CC(O)C2)=O)ccc(C)c(C)c1 15873,N1(c2nnc(C)o2)CCC2(CCC(NC(c3cc4c[nH]nc4cc3C)=O)CC2)C1 15874,CC1CC2CCC(C1)N2C(=O)CC1C(NC(=O)C(C#N)C(C)C)CC1O 15875,C=C(C)CN=c1[nH]c(=NCC2(CS(C)(=O)=O)CC2)c2ccccc2[nH]1 15876,N1(Cc2n(CCCC)nnn2)CCCC2CN(C)CCC12 15877,c1(C(=O)NCC2N(C(C(C(C)C)NC(C)=O)=O)CC2)cnc2cc(C)nn2c1 15878,CCCCCCC(=O)N1CCCC(CCNC(C2CCCNC2=O)=O)C1 15879,Cc1ccc(C)c(C(=O)NC2C=CC(CC(N3CCC4CC34C)=O)C2)n1 15880,N1(C(CC(CC)OC)=O)CCc2nc[nH]c2C12CCN(C(=O)C=CI)C2 15881,c1(C(=O)NC2C(CNC(COC)=O)C2)cc2ccccc2nc1C(F)(F)F 15882,N1(C(C2C(n3nc(C)c(-c4ccc(CO)cc4)c3)C2)=O)CCC2(CCCC2)CC1 15883,c1(C(N2CC3C(C(=O)NC(C)CN=[N+]=[N-])(C3)C2)=O)c(O)cccc1F 15884,C1(N(C)C)(CNC(C2OCCC2NC(C2C=CCC2)=O)=O)CCOCC1 15885,C1(C(=O)NCCN2CCC(C)(C)C2)CCC(C)(C)N(C(=O)C=C2CC2)C1 15886,C1(N(C(CN(c2ccccc2)CC)=O)C)CCN(C(C2(C)C=CCCC2)=O)CC1 15887,C1(NC(C2CN(C(C=C(CCN(C)C)Cl)=O)CC2CO)=O)CC2CCCCN2C1 15888,C1(NC(c2[nH]c(=N)sc2)=O)(CNC(=O)COc2cccc(F)n2)CC2CCC1C2 15889,c1(OCC)cc(C(=O)NC(C)CC2CN(C(=O)CSSC)C2)[nH]n1 15890,C(=O)(CC(O)CCCCC)NC(CC(N1CC(C#C)N(C)CC1)=O)C(F)(F)F 15891,N1(C(CCC2CCN(C(CC(COC)C)=O)CC2)=O)CC2(C1)CN(C)C2 15892,c1(OCC)ccccc1C(=O)NC1CCN(C(=O)CCCn2c(O)nnc2O)C1 15893,C1(C(N2CCC(CNC(CCN(c3ccncc3)C)=O)C2)=O)CCC2(CC2)C1 15894,CC(C)CC(CNC(C1(C)CCCCO1)=O)C(=O)NCc1ccc(O)nn1 15895,C(C1CC1)(C1CC1)=CC(=O)NC1CC(NC(C2CSCC2c2ccccc2)=O)C1 15896,C(=O)(CS(=O)(=O)C(C)(C)C)NCC1N(C(CC2(C=C)CCOCC2)=O)CCCC1 15897,N1(C(C2(CC)CCOCC2)=O)CC2CCC1CC2NC(=O)C(C1CCOCC1)C 15898,c1(N2C(CCNC(C(C(COC)C)C)=O)CSCC2)ncc2c(Br)cccc2n1 15899,C(=O)(C(C)C(F)(F)F)N(C(C)C)CCNC(=O)C(O)Cc1ccc(Cl)cc1 15900,C(=O)(C(F)(CNC(=O)CCc1cnco1)C(C)C)N(C(c1cccs1)C)C 15901,c1(C(=O)NC(CC2CCN(C(COCCSC)=O)CC2)C)nccc2n[nH]cc12 15902,C(CCCC(=O)NCC1CCC(NC(=O)CC2CCCN2C)CC1)N(C(C)C)C 15903,C1(c2cccc(F)c2)(NC(CCOCC#C)=O)CCN(C(=O)C=NOC)C1 15904,C(c1cccc(O)c1)=CC(=O)NCC1CN(C(c2cccc(C)n2)=O)CC1C 15905,C1(NC(C(c2cn(C)nn2)N(C(C(C)n2cccn2)=O)C2CC2)=O)CCC12CCCC2 15906,O=C1CCC(CC(N2CCC(O)(C(=O)O)C2)=O)CN1 15907,N1(C(c2noc(CC)c2C)=O)CC(C)CN(C(=O)C2=NNC(C(F)(F)F)C2)C(C)C1 15908,C1(C(=O)NC2(CC(=O)NCc3ccccc3Cl)CCC2)CCC(F)(F)CC1 15909,c1(C(N2CCC(C(N(CCCC)CCCC)=O)C23CC3)=O)cc2ccncc2[nH]1 15910,N1(C(CCNC(C)=O)=O)CC(=O)NCC1C(=O)NC1(CN(C)C)CC1 15911,C1(NC(=O)NCC(=C2CCSCC2)F)CC2(CCCCC2)C1 15912,C#CCC(C)(CC)C(=O)N1CCCC1CNC(C1CC12CC(F)(F)C2)=O 15913,C(CCCCC(=O)NC1(C2CCCCN2C(=O)C(C)n2cccn2)CC1)OCC 15914,Cc1cnccc1CN(C)C(c1cc(C2CC2)nn1C(C)(C)C)=O 15915,C1(NC(=O)C=Cc2cn[nH]c2)CC2CC1N(C(C1(c3ccc(F)cc3)CC1)=O)C2 15916,C1(CN(C(=O)Cc2conc2C)CC)CCCN1C(c1coc(Cl)c1)=O 15917,N1(c2n(CC=C)c(C(c3ccc(Cl)cc3)CC)nn2)CCCc2ccccc2C1 15918,C1(C2(O)CN(C(C3(Cl)CC3(F)F)=O)C2)(CNC(C(F)=C(C)C)=O)CC1 15919,c1(NC(C)=O)cccc(NC(=O)COC(c2cccnc2C(F)F)=O)c1C 15920,C(C)(CCCCN=c1nc2c(cnn2C)c(NCC(C(C)C)C(C)C)[nH]1)OC 15921,Cc1csc2ncnc(N3CCCCC(CNC(=O)CCc4cscn4)C3)c12 15922,c1(C(=O)OCC)n[nH]c(=NCCCNC(c2coc(C(N)=O)c2)=O)s1 15923,c1(C(=O)OCC)ccc2c(c1)CCN(c1nccc(N3CCCC3)n1)C2 15924,c1(N2CC(CN(C)C(c3cn(CCCF)nn3)=O)OCC2)ncnc(Cl)c1C#N 15925,O=C(C1=NOC(CNC(C2(O)CCSC2)=O)C1)NCCC12CC(CO1)C2 15926,c1(CC(N2CC(CCNC(C)=O)C2)=O)c(N)nc(C)nc1O 15927,C(C(C)CC(F)(F)F)OCC.c12cccc(c1)N2C(=O)OC(C)(C)C 15928,Cc1csc2ncc(C(=O)NC3(C)CN(C(C4CC5(C4)CC(O)C5)=O)C3)n12 15929,N1(C(c2cscn2)=O)CC2CC(C1)N(C(C1CC(F)(F)C1)=O)C2 15930,C1(n2cc(CCNC(C3(C)C(C)C3)=O)nn2)CCCC=C1Br 15931,C1(NC(=O)Oc2ccccc2)CCN(C(c2ncccn2)=O)C(C2CC2)C1 15932,c1(C(=O)NC2(CCCNC(C=Cc3cc(C)no3)=O)CC2)ccccc1S(C)(=O)=O 15933,C1(NC(c2n(CC)ncc2)=O)CC2CCC(C1)N2C(c1nocc1Br)=O 15934,N1(C(C(=CC2CCCC2)C)=O)CCCC(NC(=O)C(C)(C)CC2CCC2)C1 15935,Cc1cc(=NC(=O)C=CC(C)(C)NC(c2cnn3c2CCC3)=O)[nH]n1C1CC1 15936,N1(C(c2n(CC#C)ccc2)=O)CCC(CN(C(C2CSC(C)=N2)=O)CC)CC1 15937,Cc1cc(NC(C2CN(Cc3cccc(C#N)c3)CCO2)=O)cnc1F 15938,Cc1cc(C(=O)N(C(C(=O)NCC2(C)NC(=O)NC2=O)C2CC2)C)nc(O)n1 15939,C1(C2CCN(C(C(=C(C)C3CC3)F)=O)C2)CCCCN1C(=O)CC1CCCOC1 15940,CC1CC(C)N(C(=O)CC2CC2)CCN1C(=O)Cc1nc2cc(Cl)ccc2s1 15941,c1(NCc2cc(C)cc(F)c2)ccc2c(c1)CCC2NC(=O)OCC(C)(C)C 15942,c1(C(N2CC3CCN(C(COCCC#C)=O)C3C2)=O)cnc2c(c1)CCOC2 15943,C1(NC(c2c(CC)cno2)=O)CN(C(=O)Cc2cscn2)CCC1O 15944,C12(C(N3C(CNC(c4nccc(C(C)(F)F)c4)=O)CCC3)=O)CCC(CC1)OC2 15945,C1(N(C)C(c2ccn(C)n2)=O)CC2CC1N(C(=O)C(CC1CC1)CC1CC1)C2 15946,n1(CCC)nc(CC2CCC2)nc1-c1nc(-c2ccncc2)ns1 15947,C1(NC(C(C2CCC(=O)N2)C)=O)CCN(C(=O)CCc2nc(=N)[nH][nH]2)CC1(C)C 15948,Cc1csnc1C(=O)NC(Cc1ccoc1)C(=O)NC(C)CCC1CC1 15949,c1(C(N2C(CNC(c3cc(Br)c[nH]3)=O)CC2)=O)ccc2cnoc2c1 15950,C(=O)(C(F)CCCC)NC(C1CCN(C(CCC=CC)=O)CC1)CO 15951,C1(NC(C(n2ccc(C)n2)(C)C)=O)CN(C(c2cnc(O)c(C)c2)=O)CCC1O 15952,c1(OC(C)C)ccc(NC(c2nnn(C)c2C(F)F)=O)c(Cl)c1 15953,Cn1ncc2c1CCN(C(=O)CC1(C)CCN(C(=O)C(O)CC3CCCC3)C1)C2 15954,c1(NC(N(C2COCC2n2cc(COC(C)=O)nn2)CC)=O)cc(C)c[nH]1 15955,C1(CNC(=O)NCc2cnc(Br)s2)CC(O)CN1C(=O)C(Cl)(Cl)Cl 15956,C(N=c1[nH]c(N2CCC(CCF)C2)nc2c1CCC2)C1(C)CC1.NC 15957,c1(OCC)nc(Cl)ccc1C(=O)NCC(CO)NC(C12CCC1C2)=O 15958,N1(C(C2C(C#N)CC2)=O)CCC(C(=O)NCC2CC23CC3(F)F)(CO)CC1 15959,N1(C(c2n(C)ccc2)=O)CCCC2(CNC(=O)CCS(C)=O)CCCC12 15960,c1(OCC2C(C)CCC2)ccc([N+](=O)[O-])c2c(C#N)c[nH]c12 15961,C(C(CC(=O)NCCN1CCOCC1)C1CC1)NC(CN(C(C)=O)C)=O 15962,Cc1ccc(SC(C)C(=O)NC2CCC(NC(C3CCC(CO)CC3)=O)C2)cc1 15963,C12(NC(C(C)N(C)C(c3c[nH]c(C#N)c3)=O)=O)CC1COC21CCC1 15964,N1(C(c2c(CCC)occ2)=O)CCC(C2CCN(C(=O)CCCCO)C2)C1 15965,C(=O)(C(CCC)S(N)(=O)=O)NC(CCC)CCCNC(=O)Cn1nc(C)nc1C 15966,C1(F)(C(=O)NCC(CNC(C2(CC3CCC3)CC2)=O)CO)CCCOC1 15967,Cc1ccc(SC(C)C(=O)NC2CN(C(=O)C#CC(C)C)CCC2F)c(C)c1 15968,Cc1nc(C(N2CC(NC(=O)COc3cccc(F)c3F)CC2C)=O)cc(O)n1 15969,C=CCC(C)(C(=O)N1CC(CO)C1)OC.c1(C(=O)NCC)occc1CC 15970,N1(C(c2c[nH]ccc2=O)=O)CCC2(CC1)CN(C(C1CCCC1)=O)CCO2 15971,C1(NC(c2ccnc(C)n2)=O)COC2(C1)CN(C(c1cc(C(F)F)ncn1)=O)C2 15972,c1(NC(c2c(CCC)[nH]cc2)=O)ccc(NC(C2CC2[N+](=O)[O-])=O)c(C)c1 15973,N1(CC(=O)NC(C)CCNC(=O)CCc2nc[nH]n2)CCCOC1=O 15974,c1(CN2CCCC(NC(c3nc(SC)nc(O)c3)=O)C2)ccc(F)c(C#N)c1 15975,Cc1cc(C(=O)NC2CC(NC(C3CCCN(CC(C)C)C3)=O)C2)ncc1C#N 15976,C1(C2(O)CN(C(=O)C=C3CCCCC3)C2)(CNC(C2(CC=C)COC2)=O)CC1 15977,c1(C(=O)NC(CC)CNC(C2(CO)CC2)=O)ccc2c(n1)NC(=O)CO2 15978,c1(C(=O)NC2CN(C(=O)CC3CCC(F)(F)C3)C2)cnc2cccnc2c1 15979,c1(C(=O)NCC(C)NC(=O)CN2CCCC2CO)ncnn1C1CCOCC1 15980,C#CCC(C)(C(=O)NC1(CC)CCOC1)NC(c1nc(C)ccc1C)=O 15981,N1(C(c2cn(CCCOC)nc2)=O)CCC(C)C(CNC(C23CC(CO2)C3)=O)C1 15982,C1(NC(C=CC(=O)OCC)=O)CCCC12CN(C(C1CN(S(N)(=O)=O)C1)=O)C2 15983,CON1CCC(CC(=O)NCC2(O)CCN(C(=O)C(C)n3cnnn3)C2)CC1 15984,c1(NC(=O)NCCc2nc(C(F)(F)F)cs2)cccc(Oc2ccc(Cl)cc2)c1 15985,C1(C(=O)NC(c2ccco2)COC)CN(C(=O)Cn2nc(C)nc2C)CC1C 15986,C1(N(C)C(c2ccc(-n3cnnc3)cc2)=O)CN(C(=O)C(C)(F)F)CCC1O 15987,c1(C(=O)NCC(CC)NC(C2CCC(C)(C)CC2)=O)csc2cncn12 15988,CCCCCCC(C(=O)OC)N1CCN(C(=O)C(CCC)C(C)C)CC1 15989,CC(CC(=O)N1CC(CC(F)C(C2CC3CCC2C3)=O)C1)C(F)(F)F 15990,CC1(F)CN(C(=O)COC(F)(F)F)CCN(C(=O)CN2CCC(F)(F)CC2)C1 15991,CN1CCCCC1C(=O)NC(CNC(c1ccc(OC2CC2)cc1)=O)CO 15992,C1(C(=O)NCCC(=C)CNC(C2C3CC4C(C3)C24)=O)CC2(CC(OC)C2)C1 15993,N1(C(C2C(CC(C)C)C2)=O)CC(NC(=O)C(=O)N(C)C)C2(CCOCC2)C1 15994,Cc1cc2c(C(N3CC4CC(NC(C5CCC(C)CC5)=O)C3C4)=O)nccn2n1 15995,C(CC1=CCCCC1)N(CC(CO)C1CC1)C(=O)Cc1ccc(Cl)cc1 15996,O=C1C=C(c2nc3c(s2)CC(C(=O)NC(CO)CO)CC3)CCC1 15997,C1(C)(NC(C2C3CN(C(C(CCCC)C)=O)CC32)=O)CCCC(C)(C)C1 15998,C1(C(N(C2CCCC(NC(=O)COCCCF)C2)C)=O)Cc2cccnc2C1 15999,C12(C(=O)NCC(C(=O)OC)Cc3ccccc3OC)CCCC(C1)C(=O)NC2 16000,C1(NC(=O)NC2CN(C(CCC)C)C(=O)C2)CCOCC1(C)C 16001,Cc1nc2cc(F)ccc2cc1C(=O)NC(C)CNC(c1ccnn1C)=O 16002,S(=O)(=O)(c1ccc(NCCCC2CC2(Cl)Cl)cc1Br)NCc1cncc(OC)n1 16003,c1(C(N2C(C(N)=O)CCOCC2)C(=O)NCC2CC2)c[nH]c2ccc(Cl)cc12 16004,C1(C(N(CC(=O)N(C2CCCC2)CCO)C)=O)CCC(=O)O1 16005,CC1(C)CC(C(=O)NC(c2cscn2)CO)CN(C(c2cnc(=N)[nH]c2)=O)C1 16006,C1(NC(CCOCCOC)=O)C(C)(C)C(NC(c2cc(F)n[nH]2)=O)C1(C)C 16007,N1(C(C2N(C)C(=O)CC2)=O)CC2(CC2)CC1CNC(=O)CCC(F)(F)F 16008,C(C#CC(F)(F)F)NC(C1CCCN1C(=O)CNC(=O)NC1CCCC1)=O 16009,N1(C(C2CCC(C)C2)=O)CCC2(CCN(C(C3(O)CCOCC3)=O)CC2)C1 16010,C1(C(=O)OCC)CC(NC(=O)NCc2ccnn2CC(F)F)CCO1 16011,C(CCCCC(=O)N1CCOC(CNC(c2cc(C)cnc2C)=O)C1)OC 16012,Cc1cc(F)cc2[nH]c(C(=O)NCCNC(=O)C(c3ccc(Br)cc3)O)cc12 16013,C(=O)(C1=CCN(C(C2CC(=O)N(OC)C2)=O)C1)NC(CC)CCCO 16014,c1(C(=O)NC(C(=O)NC(C#C)Cc2ccco2)C2CC2)cc([N+](=O)[O-])c[nH]1 16015,C1(C(N2CCC(CC)C2CNC(C2CC(C)C2)=O)=O)CCC2(CC1)CC2 16016,c1(CCC(=O)N(C)CCNC(c2ccc(Cl)[nH]2)=O)n[nH]c2ccccc12 16017,c1(C(=O)NCCC2CC(NC(CC=C)=O)C2)cn(-c2ccn(C)n2)cn1 16018,S(=O)(=O)(c1ccccc1)N(CC(N1C(CCCNC(C(C)SC)=O)CCC1)=O)C 16019,C1(C(=O)NC2C(NC(Cc3nc(C)c(C)o3)=O)CC2)C2CCC3C(C2)CC13 16020,C(=O)(C(CC(C)C)N(C)C(C1CNC(=O)O1)=O)N(C(CC)C1CC1)C 16021,N1(C(CC(C=C)(C)O)=O)CC2CCC(C1)C(NC(c1cnc(OC)c(C)n1)=O)C2 16022,C1(O)(C(C)C)CCCN(C(=O)NC(c2n(C(=O)OC(C)(C)C)nnn2)C2COC2)C1 16023,N=c1nc2c(c[nH]1)CCN(N1CCC(c3nc4ccccc4s3)CC1)C2 16024,N1(C(c2c(C(C)C)con2)=O)CCCCCC(NC(c2ccc(F)cc2F)=O)C1 16025,C1(C(=O)NCC2(NC(=O)C=CC=C(Cl)Cl)CCCC2)CC12CCOC2 16026,CC(O)C(C)C(=O)NCC1CCCN1CC=C(Cl)Cl 16027,C1(OC)CCNCC1c1cccc(-c2ccccc2OC)c1 16028,C(=O)(CC(C)(O)C(F)(F)F)NCC(C)NC(CCC(=C)Cl)=O 16029,C1(OC)CC(CCNC(=O)CCC=C(C)C)N(C(=O)CC(C)n2ccnc2)C1 16030,C1(NC(C(C=C)(C)CC)=O)CCN(C(c2ccc(OCOC)cc2)=O)CC1(C)C 16031,N1(C(c2cc(C)nc(C)n2)C(=O)NC(CC)C)CCc2ccc(F)c(Br)c2C1 16032,c1(C(N2CCCC(CC(N3CCOCC3)=O)C2)=O)noc2c1CC(F)(F)CC2 16033,N1(C(c2cnc(C(C)=O)s2)=O)CCCC(C)(NC(C2C(F)(F)C23CCC3)=O)C1 16034,c12ccc(cc1)S(=O)(=O)CC1COCCN1C2=O.Cc1ccc(CN)c(Cl)c1 16035,c1(C(N2CCC(NC(c3n(C)ccn3)=O)C2)=O)cc(-n2cnnc2)ccn1 16036,N1(C(C2N(C(C(C)C)=O)CCC2)=O)CCCCC(NC(=O)CCC(=O)N(C)C)C1 16037,c1(C(=O)NC2CC(NC(CC(=O)OC)=O)C(O)C2)ccc2ncncc2c1 16038,n1(C(C)(C)C)ccc(=NC(=O)C2=CCCN(C(c3cc(CO)[nH]n3)=O)C2)[nH]1 16039,N=c1cc[nH]cc1CNc1cncc(C(N)=O)c1.c12ccccc1C(=O)N2 16040,c1(C(CCC(=O)N2CC(NC(C(CCCC)C)=O)C2)=O)ccc2c(c1)CCCC2 16041,C(CC(C(=O)NCCN1CCNC1=O)NC(c1cn(CCF)nc1C)=O)=CC 16042,CCCC(C)(O)C(=O)NCC1CCCCC1C(=O)NC1CN(C)CCC1O 16043,c1(C(=O)NCC2(COC)CCN(C(C3CCC3C)=O)C2)cc2ccccn2n1 16044,S(=O)(=O)(c1cccc(NC(N2CC(F)(CO)C2)=O)c1)N1CC(C)OC(C)C1 16045,C(=O)(CS(N)(=O)=O)N(CCCCCNC(C1(C)CC1Br)=O)C 16046,c1(C(N2CC(C)CC(NC(CC3(OC)CC3)=O)C2)=O)cc2n(n1)CCCO2 16047,C1(NC(c2cn(CC3CC3CC3CCOC3)nn2)=O)CCC(F)(C(=O)O)C1 16048,C1(C(N2CC(CNC(c3ccn(CCF)n3)=O)C2)=O)(CC)CCOC1 16049,CN1CC(C(=O)NC2CC(F)(CNC(=O)Cn3cnc(=N)[nH]3)C2)C(C(F)(F)F)C1 16050,C12(CNC(C(=O)N(C3CC(OC)C3(C)C)C)=O)CCC(O)C1CC2 16051,C1(CN(C(=O)CC2CCOC2)C)CN(C(=O)CCc2ccc[nH]2)CC12CC2 16052,CC1CCC(NC(=O)CCCC(C)N)C(=O)N1 16053,C(c1cccc(F)c1)=CC(=O)NCC(C)(F)CNC(=O)CC12CCCC1C2 16054,C1(c2cccc(OC)c2)CCN(Cc2ccccc2N(C)C)C1(C)C 16055,CC(C)(C)C(C(=O)N1CCC(O)CC1C1CC1)Sc1cc(O)ccc1Cl 16056,N1(C(CC(CC)OC)=O)CC(C)(C)C(NC(c2cnc(Cl)s2)=O)C(C)(C)C1 16057,Cc1cccc(C(=O)NCCCCCNC(C2(C3CCCCO3)CC2)=O)c1O 16058,N(C(=NCc1c(Br)cncc1Br)N1CC(O)C(C)(C)C1)C(CC)C 16059,C1(C(=O)Nc2c[nH]c(-c3ccncc3)n2)CCCN(C2CC2)C1=O 16060,C1(CC)CCCN1C(=O)C(=O)NC1CCC1NC(C1(n2ccnc2)CCCC1)=O 16061,C(=O)(C(C)CC(F)F)N(C1CCN(C(c2ccc(CO)nc2)=O)CC1)CCC 16062,N1(C(CCc2n(C)ccn2)=O)CCC2(CC2C(=O)NCC2CC3C=CC2O3)C1 16063,Cc1cc(C(=O)NC(C2(C(=O)NCC3C4CCCCC34)CC2)C)sc1C 16064,CC1CC(NC(=O)C(C)C(=O)OC(C)(C)C)CCN1C(=O)CN1CCS(=O)CC1 16065,c1(C(=O)NC(CC(C)NC(C(CN(CC)CC)F)=O)C)cc(S(N)(=O)=O)sc1C 16066,N1(C(C(C(=O)OCC)CC)=O)CC2(CCN(C)CC2)C1 16067,C(CCC(=O)NCCC(C)NC(=O)C(C)OCCC(C)C)=CCC=C 16068,C1(NC(C(C)(C)n2cc(Cn3cncn3)nn2)=O)CC2CCCN2C1 16069,CC(C)C(C(=O)NC(C)CCN(C)C)NC(C1(CO)CC(C)(C)C1)=O 16070,CC1C(NC(c2c[nH]nc2C(F)F)=O)CCCN1C(=O)Cc1cnccc1Cl 16071,c1(C(=O)NCC2CCN(C(C3CCCS3)=O)CC2)cccc2ncccc12 16072,C1(CNC(c2cnn(-c3ccncc3)c2)=O)C2CN(C(=O)CSC3CC3)CC12 16073,[N-]=[N+]=NC1CN(C(C2C3CC4C(C3)C24)=O)CC1NC(C1(C(=O)NC2CC2)CC1)=O 16074,N1(c2ncc(N3C(=O)CCC3)cn2)CCC(S(=O)(=O)NC2CC2)C1 16075,C1(CNC(CS(CC)(=O)=O)=O)CN(C(=O)CC2(CSC)CC2)C2COCC2O1 16076,Cn1c(CCNC(c2ccnc3[nH]nc(N)c23)=O)nc2cc(F)ccc12 16077,c1(OC)ccc(CC(N2CC(CNC(=O)Cc3cnc(C)nc3O)C2)=O)c(Cl)c1 16078,N1(C(CCS(C)(=O)=O)=O)CCC2(CC1)CC(NC(C1CCCO1)=O)CO2 16079,c1(C(C)=O)nc(C(=O)NC2CCCC2NC(=O)CC2(C)CCCC2)cs1 16080,CN1CCN(C(=O)C2=NOC(CNC(=O)CN3CC(C)(C)C3)C2)CCC1=O 16081,C(=O)(C1=NOC(C)(C)C1)NCCC(C)CCNC(=O)CCCC1CCCCC1 16082,CN1CC(O)CC1C(=O)NCCNC(=O)CCCc1ccsc1 16083,CC1(C)CCC(CNC(C2CCCC2CNC(c2ccc(F)cn2)=O)=O)CC1 16084,C=C=CC(C)C(=O)NCc1c[nH]nc1C(=O)NCCCCCN(C)CC 16085,Cc1cc(C(=O)NCC2(O)CN(C(=O)C(C)NC(C3CCC3)=O)C2)cc(C)c1F 16086,c1(CNC(C2C3CN(Cc4ccc(OCC)cc4)C2C3)=O)cc(C)cc(C)c1 16087,c1(C(=O)NCC(CNC(c2c(C)n(CCO)nc2)=O)C)cc(S(N)(=O)=O)cn1C 16088,c1(C(=O)NC2CCCC(N(C(C=CC=CCC)=O)C)C2)c(F)cc(OC)cc1Cl 16089,C1(NC(CCN(CCC)C)=O)CC(O)CN(C(c2cnc(CC)s2)=O)C1 16090,C(=O)(C1CCc2c(Cl)cccc21)NC1CCN(C(CCNC(=O)CO)=O)CC1 16091,C(=O)(CC(=O)NC1CCC1NC(c1nnc(C(C)C)s1)=O)OC 16092,c1(C(N2C(C)CCC(NC(c3ccc(C(N)=O)o3)=O)C2)=O)ncn2ccccc12 16093,C1(NC(CC(=O)N(C)C)=O)CC2CCC(C1)N2C(=O)Cc1cccc(F)c1Cl 16094,C1(C(N2CC(NC(=O)OC)C2)=O)CN(C(=O)C(C)(C)N(C)C)CC1F 16095,C12(NC(=O)NC(CCO)C3CCC3)CC(CCO1)N(C(c1ccc[nH]1)=O)C2 16096,CC(CC(N)=O)C(=O)N1CC(CNC(c2ccnn2C(C)(C)C)=O)C2(CC2)C1 16097,c1(C(N(CCn2cc(COCC(OCC)OCC)nn2)C)=O)cc(C)sc1C 16098,c1(C(=O)NC(C(=O)NCC(O)CC2CCCC2)C2CCCO2)ncoc1C1CC1 16099,Cc1cccc(F)c1CC(=O)NC1CC(NC(C2C3CCC(F)(F)C23)=O)C(O)C1 16100,N1(C(C=C2CCN(C)CC2)=O)CCC(NC(=O)CC2CCC3CC23)CC(C)(C)C1 16101,CC1=C(C(=O)NC2CCN(C(=O)C=C(C3CC3)C3CC3)C(C3CC3)C2)CCC1 16102,C1(F)(CNC(C2C(=O)NCC2)=O)CCN(C(c2cccc(OC(F)(F)F)c2)=O)C1 16103,C1(NC(CCC)=O)CCN(C(c2cc(N3CCCC3)nc(Cl)c2)=O)CC1C 16104,c1(CC)cccc(-n2nc(C(CC)OC)nc2-c2coc(C3CC3)n2)c1 16105,CCCCS(=O)(=O)NC(C)C(=O)NC1CC(CNC(=O)C(C)(C)NC(C)=O)C1 16106,CC1=C(C(=O)N(C)CCOCCNC(=O)CCc2cncc(Br)c2)CCC1 16107,N1(C(c2c(CC)cno2)=O)C2CCC1CC(C(=O)Nc1cnc(C)nc1C)C2 16108,CC1(C(=O)NCC#CCNC(C2CC(=O)N(C3CCCC3)C2)=O)CCC(=O)N1 16109,C(CNC(=O)CN(C(=O)CCn1ccnc1C)C1CCC1)(CC(C)C)OC 16110,O=C(CC(O)CNC(C1CCC(O)C1)=O)N1CC(Cn2ccnn2)C1 16111,c1(CC(N2C(CNC(=O)C=CCF)CCC(C)C2)=O)csc2ccccc12 16112,C1(NC(C2CCC(C)C2)=O)CCOC2(CCN(C(C3(O)CCSC3)=O)CC2)C1 16113,O(C1CCCc2ccccc21)CC(N1CCN(C(CCSC)=O)CC1C(F)F)=O 16114,C1(NC(c2cc(F)cc3nn[nH]c23)=O)CN(c2ncns2)C2CCCCC12 16115,C12(C(=O)NC(C(CO)NC(c3c(COC)cccn3)=O)C)CC1COC21CCC1 16116,Cc1cc(CNC(c2nc3ccccc3n2C(F)F)C)n2nc(C)cc2n1 16117,C(=O)(C(F)(F)C(C)O)NCC(C1CCCCC1)NC(C(CCC)O)=O 16118,C1(NC(c2cc(C)c(C)[nH]2)=O)CN(C(c2ccc(O)cn2)=O)C2CCCC12 16119,CS(=O)(=O)C1CC(C(=O)NC23CC2CN(C(c2ccccc2SC(F)F)=O)C3)C1 16120,CCCCCC(O)CC(=O)N(C)CCN(C)C(c1cc(Cl)c[nH]1)=O 16121,c1(CNC(C2C(C)CN(C(=O)C(C3CC3)C3CC3)CC2)=O)ccc2c(c1)CCC2 16122,C1(NC(c2c(C)[nH]cc2)=O)CCOC(C(=O)N(C2CC(C)(C)C2)C)C1 16123,C(Cc1cn[nH]c1)(C(=O)NOCCn1cccn1)NC(C1CCCOC1)=O 16124,C(=O)(C(CCOC)OC)NCCC1(NC(Cc2nc(CC)sc2)=O)CC1 16125,N1(C(CCNC(=O)NC)=O)CCC(O)(C(C)CNC(=O)CNC(=O)CC(C)(C)C)C1 16126,N1(C(COCCCOC)=O)CC2CC(O)C1C2NC(C1CCCCNC1=O)=O 16127,C(=O)(C1=NNC(=O)CC1)NCCC1CC(NC(C(C(C)(C)C)N(C)C)=O)C1 16128,c1(C(=O)NCC2(C(=O)NCc3ncc(C)nc3)CC2)cccc(O)c1C 16129,CC(C)CCC(=O)C(=O)N1CCC(C(=O)NC(C2CCCC2O)C)CC1(C)C 16130,c1(C(N2CC(NC(COCCC#C)=O)C(C)(C)CC2)=O)cc(S(N)(=O)=O)c(C)s1 16131,C1(NC(c2nc(COC)[nH]n2)=O)CCN(C(C2CCC3CC3CC2)=O)C(C)C1 16132,Cc1ccc(C(F)(F)C(=O)NC(C2CCCN(C(=O)CSCC(N)=O)C2)C)cc1 16133,c1(C(=O)NC(CNC(CSCCN(C)C)=O)CO)cc(N)c(Cl)c(O)n1 16134,CCC(CC)CCC(=O)NCC1CCN(C(=O)Cn2cnc(C(F)(F)F)c2)C1 16135,C1(C(=O)NCC2CN(C(C=CCOC)=O)C2)(OC)CCCC(C)C1 16136,C1(C(N2CCC(N(C(C3CC(=C4CCC4)C3)=O)CC3CC3)C2)=O)COCC1C(N)=O 16137,C1(C(NOCC)=O)CCN(C(c2cnn[nH]2)=O)CC1O 16138,CCCCCCCCNC(=O)C(=O)NC(C)CNC(=O)CC1CC(SC)C1 16139,c1(C(=O)NC(c2cn(C)nc2)C(F)(F)F)nc2c(o1)CCSC2 16140,C1(C(=O)NCC=CCNC(=O)CC2CCCC2(F)F)CCn2ccnc2C1 16141,c1(C(C(=O)NCc2ccnn2C)N(C)C)ccccc1F 16142,C1(NC(C(C(C)C)SCC)=O)CC2CCC(C1)N2C(c1ccc(C(C)(C)C)[nH]1)=O 16143,N1(C(C(C=C)OC)=O)CCC(C)CC1C(=O)NC(COC)CCCC 16144,C(C1c2ccccc2CN1C(C1CC2(CC2)C1)=O)NC(C(C)CS(C)(=O)=O)=O 16145,C123CCOC(C1)(C2)CNC3=O.c1(NC(C2C(=C)CC2)=O)nn(CC)cc1Br 16146,Cc1ccc(C(=O)NC(C)C(CO)NC(C2CC(S(C)(=O)=O)C2)=O)cc1C 16147,C1(C(CC)O)CCCN1C(=O)C#CCNC(c1ccoc1Cl)=O 16148,c1(C(C)NC(C(C)N(C(=O)COC2CCCC2)CC)=O)ccc(C)cn1 16149,Cn1ccc2c(C(N3CCN(C4CCCCC4O)CC3)=O)cccc12 16150,C1(CC)CN(C(C2(F)CCOC2)=O)CCN1C(=O)CCCCc1ccc(Cl)cc1 16151,n1(CC)cc(CC(=O)NCCCN(C(=O)CC23CC(CC)(C2)C3)C)cn1 16152,C1(NC(=O)CC2(CO)CC2)CN(C(C2CC(=O)N(C3CC3)C2)=O)CC1F 16153,C12(C(=O)NC3CC4(C(C(N(C)Cc5c(C)n[nH]c5)=O)C4)C3)CC(C)(CCO1)C2 16154,N1(C(Cn2c(C)ccc2C)=O)CCN(C(=O)COC2CC2)C(C2CCCC2)C1 16155,c1(OC)cc(C(N2CC(N(C(=O)C(O)c3ccsc3)C)C2)=O)nnc1C1CC1 16156,C(=O)(C(C)(C)C(=O)NCC1(O)CCN(C(=O)CC2CC(C)(C)CO2)C1)NC 16157,C(c1ccc(F)c2ccccc12)=CC(=O)NCC1CC(NC(C2(O)CCC2)=O)C1 16158,C12(CC(C(CCCCN)=O)=O)CCCN1CCC2.C1(=O)C(=O)NCCN1.C1(C)CC1 16159,C(CC(C(C)C)NC(=O)C(F)C(=O)OC)N(C(C(C)(C)OCCC)=O)C 16160,c1(C(=O)NC(C2CCN(C(Cc3ncc(CC)[nH]3)=O)C2)C)cc(F)cc(F)c1N 16161,CS(=O)CCC(=O)N(CCNC(=O)CNC(=O)C1CC1)Cc1ccc(Cl)nc1 16162,CC(C)CC(O)CC(=O)N1CCC(N(C(=O)CC(C)C2CCCC2)C)C1 16163,C(=O)(CCS(N)(=O)=O)N1CC(=C(CNC(c2ncc(CC)nc2)=O)F)C1 16164,c1(NC(C(C2CN(C(c3cc(CCC)[nH]n3)=O)C2)O)=O)ccc(C)c(C)c1 16165,c1(C(=O)NC(C)CNC(c2cnsc2)=O)cccc(-c2nc(=O)o[nH]2)c1 16166,C1(C(=O)NCCCn2ncc(C)c2)(CNC(c2scc(C)c2C)=O)CCCCC1 16167,CC1CC(C(=O)N2CCC2CNC(c2cncc(-c3cccc(F)c3)c2)=O)=NO1 16168,CC(C)(C)C(C(=O)NCCc1nc[nH]n1)NC(c1ccnnc1)=O 16169,c1(CC(N2C(CN(C(c3cnc(C)s3)=O)C)CCC2)=O)ccc2[nH]ccc2c1 16170,CC1CCCN1CC(=O)NCC1CCC1C(N1CCC(N2CCC2)C1)=O 16171,n1(CC(=O)NCC(CNC(CC(n2ccc(C)n2)C)=O)O)cc2ccccc2n1 16172,C#CCCC(O)C(=O)Nc1cccc(NC(=O)C(c2ccc(F)cc2)OC)c1 16173,n1(CCC)nc(C)cc1C(=O)NC(CN(C(=O)C(C)CC)C)CC 16174,N1(C(CSCC)=O)CCC2(CCN(C(c3ccc(OC)nc3)=O)C2)C1 16175,Cn1cc(C(=O)NC2CCCCC2NC(c2nccs2)=O)c2ccccc12 16176,c1(COC)ccc(NC(C2(CNC(=O)CC3COC(=O)N3)CC2)=O)cc1 16177,c1(C(N2CCCC(N(C)C(C3CCS(=O)(=O)N3)=O)CC2)=O)ccc2nc[nH]c2n1 16178,CC1(C)CN(C(c2csc(=N)[nH]2)=O)CC1C(=O)NCCC1OCCC1(C)C 16179,C1(NC(c2ccc(C)cn2)=O)CCCC12CN(C(=O)CCC1CCCCC1)C2 16180,C#CCC(C(=O)N1CCCC1(CC=C)C(N1CC(F)C(F)C1)=O)C1CC1 16181,c1(C(=O)NC(CC)CNC(C2CC2(F)F)=O)ccncc1C(F)(F)F 16182,C1(CNC(C2C(C)C2)=O)CCC2(CCN(C(c3cccc(N)c3F)=O)CC2)O1 16183,CC(C)CC(C(=O)Nc1ccc(F)cc1F)NC(C1CCC12CCCO2)=O 16184,c1(NC(CNC(C2CC(C)(C)C2)=O)CO)ncnc2cccc([N+](=O)[O-])c12 16185,CC(C(=O)NC(CN(C)C(c1cn(C2CCOC2)cn1)=O)(CO)CO)C(C)(C)C 16186,C(CC(F)(F)CO)NC(C1(n2cc(-c3ccccc3F)nn2)CCOCC1)=O 16187,C1(Cc2ncn(Cc3scc(C(=O)NC(CCCC)C)n3)c2)CCCCCC1 16188,c1(C(=O)NC(CNC(=O)CC2(O)CCOC2)C2CC2)cccn2ccnc12 16189,N1(CC)CCCCC1C(N1CC(C(=O)NCC2CSC2)C(C(C)C)C1)=O 16190,CC(O)C(=O)N1CC(C(=O)NCC2(CO)COC2)C1 16191,c1(C(N2CCCC(C(N(C)Cc3c(C)occ3)=O)C2)=O)cc2ncccc2[nH]1 16192,n1(C(C(=O)OCC)C)nnnc1C(c1nncn1CC)NC1CC(C(=O)OC)C1 16193,C(=O)(CC(C)C(=O)N(CC(=O)NCC1CC(C)C1)C1CC1)OC 16194,c1(-c2cc(CN(CC(C3CCCC3)OC)C)no2)ccc(Cl)cc1Cl 16195,N(C(=NCCC(C)C)N1CCc2ocnc2C1)CC(c1c(C)noc1C)C 16196,C1(C)(C(=O)NC(CCCNC(c2c(CC)n(C)nn2)=O)C)CC2(C1)CC2(F)F 16197,c1(CNC(c2c(OC)ccs2)=O)ccc(NC(=O)C(C)OCC2CCCO2)cc1 16198,c1(C(=O)NCC23OCC(NC(C4C(C=C)CC4)=O)(C2)C3)cc([N+](=O)[O-])ccc1Cl 16199,C(=O)(CC1OCCc2ccccc21)NC12CCCN(c3c(OC)cncn3)CC1C2 16200,N1(C(CN(C)C(C2CCC(C3CC3)C2)=O)=O)CCCCCCCC1 16201,C1(C(=O)NCCCN(C(C(C)NC(COC)=O)=O)C)COCC(C)(C)O1 16202,C1(NC(C2CC3(CC3)C2)=O)CN(C(=O)CCC2CCCC2)C2(CCCC2)C1 16203,C(=O)(C#CC1CCCOC1)N1CCOCC(C)(CNC(C=CCCC)=O)C1 16204,N1(C(C2CC(=C)C2)=O)CC2C3CCC(C2C1)N(C(=O)COc1ccc(Cl)cc1)C3 16205,N1(C(C(C(CC)C)NC(C)=O)=O)CCC2(CCC2)C(NC(C2CCC(=O)N2)=O)C1 16206,C1(NC(C2(OC)CC2)=O)COCCC1NC(c1scc(C)c1C(=O)OC)=O 16207,n1(-c2ccc(C(=O)OCC)cc2)c(C)cc(CNN(CC(F)F)C(C)CO)c1C 16208,C(=O)(C1=NOC(C)(C)C1)N1C(C(C)C)(C(=O)NCCC2CCCN2C)CCC1 16209,N1(C(C(C)OCCCC)=O)CC2(NC(=O)CCn3c(C)csc3=O)CCC1C2 16210,C(=O)(C1=NOC(C)(C)C1)N1CCN(C(c2c(C)nn(C)c2C)=O)C(C2CC2)C1 16211,N1(C(c2c(CC)ccs2)=O)CC2CCC2(CCNC(=O)CCC=C(C)C)C1 16212,c1(C(=O)NC2CCCN(C(=O)C=Cc3cnccn3)C2)cccc2nc(Cl)sc12 16213,c1(C(CC(=O)N2CC(NC(C3C(CCC)C3)=O)C2)C)ccc(F)c(F)c1 16214,C1(C2CCCN(C(c3c(C4CCC4)cnn3C)=O)C2)(NC(CC(C)C)=O)CC1 16215,N1(C(c2snc(C(=O)OCC)c2Br)C)CCC(=O)N(C)CC1 16216,Cc1noc(NC(C2CCCN(C(C3CC(=O)N3)=O)C2)=O)c1Br 16217,N1(C(C(CCC)OC)=O)C2CCC1CC(CNC(=O)C(C#N)=CC1CC1)C2 16218,O=c1c(Cn2cc(OC3COC(c4ccccc4)C3)cn2)c[nH]cc1Cl 16219,CC1CCN(C(c2cc(CNC(=O)C=Cc3cc[nH]c3)ccn2)=O)C1CO 16220,CCC(CC)CCC(=O)N1CCN(C(=O)CC(O)CC(C)C)CCC1C 16221,C1(N(C(c2ccc(C)cc2)C(=O)NCCC#N)CCC)CCN(C)C1(C)C 16222,C(=O)(C1CCc2nccn21)NC(C(=O)NC1(CC)CCCC1)CC1CC1 16223,C1(C)C(=O)NN2CCN(CC2)c2cccc(c2)S1.S(=O)(=O)(c1cn(C)nc1C)NC 16224,N1(C(C(CCC)F)=O)CCN(C(=O)Cn2cc(C3CC3)cn2)CC1C1CCC1 16225,Cc1cnc(C(=O)NC2CCC(N(C)C(c3c(N)cnn3C)=O)CC2)c(C)c1 16226,C1(NC(CCc2n(C)c(S)nn2)=O)CCN(C(=O)C2=CCOC2)C12CC2 16227,N1(C(C(N)=O)=O)CCCOC(CNC(=O)CC(O)C2CCCC2)C1 16228,C1(NC(CCCN(CCC)CCC)=O)CCN(C(=O)CCC(=O)OC)C1CC 16229,C=CCC(C)(C)C(=O)N1CCCC(F)(C(=O)NCc2nnc(O)o2)C1 16230,N1(C(=O)NCc2noc(C(F)(F)F)n2)CC2C(Cc3cccc(Cl)c3)C2C1 16231,C1(CN(C(C(c2ccc(CC)s2)=O)=O)C)CCCCN1C(=O)CCSC 16232,C1(C(N2C(CC)CC(C)C2)=O)CCC2(CC2)N1C(c1c[nH]c(C)c1)=O 16233,c1(CN2CC3(C(C(=O)NC(C4CCOCC4)C)C3)C2)ccc(N(C)C)cc1Cl 16234,C12(OC)CCC3(C1)N(C2)C(=O)NOC(C)C(=O)N3.C(C)(C)(C)NC(C)=O 16235,C1(C)(CNC(C=C=C(C)C)=O)CN(C(=O)CC2CCC(=O)N2C)CCO1 16236,N1(C(C(C=C)O)=O)CC(NC(=O)CC2CCCCCC2)CC2(CCC2)C1 16237,c1(CCC)cccc(OC(=O)Cc2csc(Cl)c2)c1 16238,N1(C(C(CN(C)C)O)=O)CCC2C(CCCN2C(C2CCCCN2C)=O)C1 16239,C1(CC)CCC(NC(=O)CC2(N(C)C(C3CCCN3C3CC3)=O)CC2)C1 16240,N1(C(CC2(C)CCOC2)=O)CCC2(CC1)CC2C(N1CC2CC2C2CC12)=O 16241,C12(CNC(C3C(C)(C)C3)=O)CCC(C1)N(C(=O)CCCN1CCCC1)C2 16242,Cc1ncc(C(N2CC=C(CNC(C3CCC4C3C4(F)F)=O)CC2)=O)cc1C#N 16243,c1(OC)cccc(N2CCN(C(c3cccnc3O)=O)CC(C)(F)C2)c1[N+](=O)[O-] 16244,N1(CC(=O)N(C(=O)C(F)F)NC(C)C)CCN(CCc2cccs2)CC1 16245,c1(COC(C(=O)NCC(C)CN(C)C)C)ccccc1 16246,C1(NC(C#CC(C)C)=O)CN(C(C2(C#N)CCCO2)=O)CC12CCOCC2 16247,C(CC(C)C(=O)N1CC(C)(NC(=O)C(C)NC(=O)OC2CCCC2)C1)OC 16248,C=CC1(C(=O)NC(c2ccccc2F)C)CCN(C(c2ccsn2)=O)C1 16249,N(C1CCCc2occc21)C(C(CC(C)C)NC(C1CCC(=O)O1)=O)=O 16250,c1(OC)cc(CCC(=O)NC(C)CCNC(=O)CC(C)OC)ccc1F 16251,Cc1cc(C)n(C(C)C(=O)NC2CC(NC(C3CCC(F)(F)C3)=O)C2)n1 16252,c1(C(N2CCN(C(c3n(C=C)nnc3)=O)C(CCO)C2)=O)cc(F)cc(N)c1F 16253,N1(C(CCn2ccc(C)n2)=O)CCN(C(=O)CN2CC(=O)NC2=O)C(C(C)C)C1 16254,Cc1ccc(C(=O)NCC23CC(NC(=O)C(C)NS(C)(=O)=O)(CO2)C3)cc1F 16255,Cc1cc(N2CCC3NC(=O)CCC3C2)nc(=NCC(F)(F)Br)[nH]1 16256,c1(C(=O)NC2C(C)CN(C(c3ccnc(S)c3)=O)CC2)cc2c(F)cccc2[nH]1 16257,c1(OC)cc(O)c(C(=O)NCC(C)N(C)C(C2CC(OC)C2)=O)cc1OC1CC1 16258,N1(C(CC2CCN(C(C(C)=CC=C)=O)C2)=O)CCC(C)(C)C(CO)C1 16259,c1(COCC(=O)NCC=C(C(=O)OCC)C)ccc(F)nc1 16260,C12(NC(CCC(=O)NC)=O)CCCC1N(C(C1CC1C1CCCCC1)=O)CCC2 16261,c1(CC)cccc(C(=O)NCC2(C(C)NC(c3cnc(C)o3)=O)CC2)c1 16262,C1(C(C)NC(COCC(=C)C)=O)CCCN1C(=O)C=C(C)C(F)F 16263,CC1CCN(C(c2cn(C)nc2C(C)(F)F)=O)CCN1C(C1CNC(=O)C1)=O 16264,CC1CC(CNC(c2cn(C3CC3)nn2)=O)CN1C(c1cn(C)c(O)n1)=O 16265,Cc1nn(C)cc1CCC(=O)NC(C1CCCN1C(c1ccccc1)=O)C 16266,N1(C(C2CC(CCC)C2)=O)CCC(F)(C(=O)NCc2nc(C)cs2)CC1 16267,c1(C(=O)NC2CCN(C(C3N(C(=O)OCC)CSC3)=O)C2)c[nH]nc1[N+](=O)[O-] 16268,c1(C(N(CCC(C)NC(C2CC(OC)C(OC)C2)=O)C)=O)c(F)cc(F)cc1F 16269,C1(NC(C(C)c2cccs2)=O)CN(Cc2ccccc2CCBr)CC1C#N 16270,c1(C(=O)NCC2(C)C(C)CN(C(C(C)C(F)F)=O)C2)cnc2cc[nH]c2c1 16271,N1(C(=O)NCCc2ccc3c(c2)COC3)CCCc2cc(Br)cc(F)c21 16272,C1(NC(COC)=O)CCN(C(=O)Nc2ccc(Oc3ccccc3)cc2)C1C 16273,C#Cc1ccc(C(=O)NCC2CCN2C(c2nocc2C2CC2)=O)o1 16274,c1(C(=O)NCC2(NC(c3cnc(CC(C)C)[nH]3)=O)CCCC2)cc(O)cc(=O)o1 16275,C1(C(=O)NCCN(C(=O)CC(C)(C)c2ccccc2)CCC)CC(O)C1(C)C 16276,CC1(C)CCN(C(=O)CCOCC(F)F)CC1C(N1CCCCC1CF)=O 16277,CCCCCC(C(=O)NCC1CC1NC(=O)CCN=c1[nH]ccs1)C(C)C 16278,N1(C(C2CN(C(C(CCC)=CCC)=O)CC(C)C2)=O)CCC(=O)N(C)CC1 16279,C(C(CC(C)C)C(=O)N1Cc2cncnc2C1)NC(C1(COC)CCCC1)=O 16280,c1(C(=O)OC)cc(=NC(=O)C2(c3ccc(-c4ccc(Br)cn4)cc3)CCC2)[nH][nH]1 16281,c1(C(=O)NC23CC(CNC(CCOC)=O)(C2)OC3C)snc2ccccc12 16282,C1(NC(c2c(C)ncnc2)=O)CC2CC1N(C(c1ccc(F)cc1Br)=O)C2 16283,c1(CNC(C(C)N(CCC)C(C2CC2(C)C(F)F)=O)=O)cccc(F)c1C 16284,C=Cc1cccc(-c2ccc(COc3ccccc3OCC)s2)c1 16285,C1(CC(C)(C)C)CN(C(c2ncccc2O)=O)CC1NC(C1COCC1(C)C)=O 16286,c1(N2CCC(N(C(c3ccc(F)cn3)=O)CC)C2)nc(C2CCC2)nc(Cl)c1C 16287,C1(C(N2CC(CNC(C3CCCN(CC)C3)=O)C2)=O)CCCC1C1CC1 16288,C(=O)(C(C)CC(F)(F)F)N(C1CN(C(c2cc(C)cc(N)c2)=O)CC1(C)C)C 16289,CCS(=O)CC(=O)N1CC(CNC(C2(CO)CCC2)=O)C1 16290,N(C)(C1CS(=O)(=O)c2ccccc21)C(c1ncc(SC)[nH]1)C(=O)NCCOC 16291,N1(C(CCOCCC)=O)CCC2CCN(C(=O)CCNS(C)(=O)=O)CC12 16292,c1(NC(C2N(C(C3(CC(=O)OC)CC3)=O)C(C)C2)=O)ccc(Cl)cc1C 16293,c1(C(=O)NS(CCOCC)(=O)=O)cnc(N)c(Cl)c1 16294,C1(NCn2cc(C3CCN(C)C3)nn2)CCC=CCCC1.N12CCC(CC1)C2=O 16295,C(CCC(=O)NNC(=O)c1ccc(F)cc1Br)OC 16296,c1(C(N2CC(N(C(c3c(CC)nc[nH]3)=O)C)C(F)C2)=O)cnc(OC)cc1OC 16297,c1(N2C(C)CC(NC(C3CC(C)(F)C3)=O)C2)ncnc2sc3c(c12)CCC(C)C3 16298,Cn1nncc1CC(=O)NCC=CC(=O)NC1(C)CC(NC(C)(C)C)C1 16299,N1(C(C(CSC)O)=O)CC=CC(C(=O)N(C)CCOCCO)C1 16300,c1(C(C2(O)CN(C(=O)C(O)C3CC3)C2)C)cccc2[nH]cc(CC(=O)NCOC)c12 16301,C1(C(=O)NC2(CF)CCN(C(c3c(C)nsc3N)=O)C2)CCc2ncncc2C1 16302,C1(NC(c2c(C)cc(Br)o2)=O)CN(C(C2CC2F)=O)CC1S(C)(=O)=O 16303,C1(CN)CCC(c2ccccc2)=NO1.c12nc(ccc1Cl)NC2=O 16304,C1(C2CN(C(C3CC3Cl)=O)C2)(NC(c2ccc(CN(C(C)C)C)cc2)=O)CC1 16305,c1(C(=O)NC(CNC(=O)Cc2cnccc2Cl)CO)cc(Cl)c([N+](=O)[O-])[nH]1 16306,N1(C(C(C)(C)OC(C)C)=O)CCN(C(=O)CC(C)Sc2ccccc2)C(CO)C1 16307,C1(C(=O)NC(CNC(C(C)OCC=C)=O)C2CC2)CCC(C)(C)O1 16308,CC(=Cn1ccnn1)C(=O)N(C1CCCC(NC(c2ncsc2C(C)C)=O)C1)C 16309,N1(CC(=O)NC(C(=O)OC)Cc2cn(CCCOCCSC)nn2)CCNC(=O)C1 16310,C1(NC(C2CCCCC2)=O)CC12CCN(c1nnc(C3(O)CCSC3)n1C)CC2 16311,N1(C(c2c(CC)c(C)sc2)=O)CCC2(CC1)CC2NC(C1COCCO1)=O 16312,c1(C(=O)NC(C(C)NC(COCCC)=O)C)nc(C)oc1C 16313,C(=O)(CC(C)C(F)(F)F)N(C(C(=O)N(CC(C)C)CCO)C)C1CC1 16314,c1(CC(=O)NCC2N(C(C(C)NC(COC)=O)=O)CC2)cc(N)c(O)c(F)c1 16315,Cc1cnc(C(N2CCC(C(C)(C)NC(c3cnc(N)c(Cl)c3)=O)C2)=O)cc1Cl 16316,C1(C2CC2)(NC(CCCC)=O)CCN(C(c2ccc(-n3ccnc3O)cc2)=O)C1 16317,c1(C(=O)NCC2(F)CCN(C(CC(C)N(C)C)=O)C2)cnc2[nH]nc(O)c2c1 16318,N1(C(c2c(OC)cncc2)=O)CC2=C(C1)CN(C(=O)C(c1cnccn1)C)C2 16319,O=C(CC(F)(F)C(F)(F)F)NC1CCC2(CC1)CN(c1ccccc1[N+](=O)[O-])C2 16320,C1(C(=O)NCCc2csnn2)CC(F)CN1C(=O)CC1CC=CC1 16321,C(=O)(CCC(=O)NC1CCCCC1NC(=O)C(F)=CCOCCO)N(CC)CC 16322,c1(C(N2C(CCC(=O)NCC(CNC(N)=O)O)CCC2)=O)ccc2c(c1)CC2 16323,C1(C(=O)NC2(C#N)CN(CC)C2)CCCN(CC(=O)NC)C1C 16324,C1(CNC(C(CC)=CCCC)=O)CC(C)CN(C(=O)CS(=O)(=O)NC2CC2)C1 16325,CC1=C(C(=O)NC2CCCC(NC(c3c(N)sc(C)c3C)=O)CC2)CCCC1 16326,C1(C(N(CC(CNC(c2c(C)n[nH]c2)=O)C)C)=O)Cc2ccccc2N1 16327,C1(C(N(CCCNC(c2ccc(CO)nc2)=O)CCC)=O)CC2(C1)CC1(CC1)C2 16328,C1(C(=O)NCC(C)(C)NC(CN(C)C(c2ccsc2)=O)=O)CCc2[nH]nc(O)c2C1 16329,c1(NC(C2CCN(C(C3C(=C)C3)=O)C(CC)C2)=O)cccc2cnccc12 16330,c1(C(CNC(C(CC)CC2CC2)=O)(F)F)ccc(F)cc1F 16331,C(=O)(CCCC1CCC1)NC(C1CCCN1C(c1cnccn1)=O)C 16332,C1(C)(CNC(C2C(C)C2)=O)CN(C(c2ccc(CO)c(Cl)c2)=O)C(C)(C)C1 16333,C1(C(N(C(CC)CC)C)=O)CC2(CCN(C(=O)CCC3CCCCO3)C2)C1 16334,C(C)(CNC(=O)C(C)(C)CF)(C(C)C)NC(CC(n1ccc(C)n1)C)=O 16335,C(=O)(C(F)C(C)(F)F)N1CC(C(=O)NC2CCC3(CC3)C2)(SC)C1 16336,c1(OC)ccc(C)c(C(N2CCCCC2c2cn(CCC(F)(F)Cl)nn2)=O)n1 16337,Cc1[nH]nc(Br)c1C(=O)NC(C)CC(C)NC(=O)CSC1CC1 16338,CC(=O)CCCCC(=O)N1CCC(NC(=O)CCCN2CCCC2)CC(O)C1 16339,N1(C(C=C2C(C)(C)CCCC2)=O)CCC2CC1CN(C(=O)C(O)c1ccsc1)C2 16340,S(=O)(=O)(c1cccc(C(N2CC(=O)NCC2C)=O)c1)NCC(C)O 16341,c1(C(N2C(CNC(C3CC4CC4C3)=O)CC(C)(C)C2)=O)cc2ccnc(Cl)c2[nH]1 16342,c1(OC)ccc(C2=CCN(C(C3(C(F)(F)F)CCCC3)=O)CC2)cc1 16343,c12ccccc1C=CC(=O)N1CC(C(C)(C)O)(C1)C2.CC(C)N(C(C)C)C(C)C 16344,C1(CNC(C(C)(C)C)=O)Cc2ccccc2CN1C(C1CC(S(C)(=O)=O)C1)=O 16345,C1(C(=O)NCC(CNC(COC(CC)(C)C)=O)(C)OC)OC(C)(C)OC1(C)C 16346,N1(CC(=O)NCC(CC)OC)CCN(C(=O)C(C)CCN(C)C)CC1 16347,Cc1cc2ccc(C(=O)NCC3CN(C(c4cocc4C)=O)C3)cn2c1 16348,C=C=C(C)CC(=O)NC1(CN(C)C(C2CCN2C2CCCC2)=O)CC1 16349,N1(C(C(CC(CC)C)=O)=O)CC2OCCN(C(=O)CCCC(F)(F)F)C2C1 16350,C(=O)(C(F)(F)C(O)C(C)C)N1CC2(C(NC(c3cccc(C)c3F)=O)CCC2)C1 16351,C12CC(C)(C1)C(=O)N2.C1(CC(=O)NC)(C(=O)NCCOCCCF)CC1.COC 16352,c1(C(N2CCN(C(C)C(=O)NCC(F)(F)F)CC2)=O)nccn2nccc12 16353,c1(C(N(C)CCn2ccnc2)=O)cccc(CNC(C2OC3CCC2C3)=O)n1 16354,Cc1c(Cl)ccc(C(N2CCOC(C)(CNC(=O)C(C)OCC(C)C)C2)=O)c1O 16355,c1(C(N2CC(C)C(NC(=O)C#CC3(C)COC3)CC2)=O)cccc2c1OCCC2 16356,N1(CCCCCCC)CCC2C(CCCN2C(=O)CC2(C)CC2)C1 16357,C1(OC)CCCCC1(c1nnnn1CCC1CC1)Nc1cn[nH]c1 16358,C1(C(=O)Nc2ccns2)CC2(CCN(Cc3cc(O)cc(Cl)c3)CC2)C1 16359,C1(O)(C(=O)NCc2ccc(OC)cc2)CCN(C(c2cnns2)=O)CC1 16360,c1(OCC)ccnc(N2CCC(N(C(=O)C(C3CCC3)OCC)C)C2)n1 16361,N1(CC(=O)NCC2N(C(Cc3nc(C)[nH]n3)=O)CC=C2)CCCCS1(=O)=O 16362,N1(C(COCCC)=O)CC2COCCC2(NC(c2cc3sccc3[nH]2)=O)C1 16363,C(=O)(NN1CCCC(C(=O)CCN2CC3CC3C2)C1)c1cnc(C)[nH]1 16364,n1(CC)cc(Cl)c(C(N2CC(CNC(=O)CC(C)(F)F)CC2C)=O)n1 16365,C1(C(N2C3(CNC(C4(CN(C)C)CC4)=O)CC(C2)C3)=O)CC12CCC(=O)CC2 16366,C1(C(C)C(=O)NCC(F)Br)CCN(C(C2CC(=O)C2)=O)C1 16367,C(CCCCS(=O)(=O)CCCCCO)NC(=O)NCC(c1cccs1)O 16368,N1(C(=O)C2=CCCC2)CC2(CO)CC1(C(=O)NCC1CC(O)CCO1)C2 16369,N1(C(c2cnn(CC)c2C)=O)CCC(NC(=O)CCn2ccccc2=O)C(C)C1 16370,N1(C(=O)CCC2CC2)CC2(CCN(C(c3cc(C4CCOC4)[nH]n3)=O)C2)C1 16371,C1(C(=O)NC(CC(=O)OCC)C)CCN(C(c2c(C)cnn2C)=O)CC1(C)C 16372,Cc1cc(Cl)ncc1CC(=O)NC1CC(C)(NC(c2nc(Cl)oc2C)=O)C1 16373,C=C(C)CC(C)C(=O)N1CC2CC2(CNC(=O)CCC=Cc2ccccc2)C1 16374,c1(C(N2C(CN(C(c3nc(Cl)oc3C)=O)CC)CCC2)=O)cnn2ccsc12 16375,N1(C(CCC2N(C)CCCC2)=O)CCN(C(=O)CCCF)C(CC2CC2)C1 16376,c1(OC)ccc2cc(C(=O)NC3CC3NC(=O)C(C)S(C)(=O)=O)n(C)c2c1 16377,N1(C(C2(F)C(C)C2)=O)CCC(NC(=O)COc2cccnc2Cl)CC1 16378,Clc1ccc2ccc(=NCCc3noc(-c4ccccn4)n3)[nH]c2n1 16379,C1(NC(C2CC3CCCC23)=O)CCCNC12CC2 16380,c1(NC(c2ccc(NCC3CC3)nc2)=O)cc(Cl)nc2ncnn12 16381,c1(NCC(CCC)OCC)ccc(S(=O)(=O)NCC(CO)C(C)(C)C)cc1Cl 16382,c1(-c2cn(CC(C)NC(C3C(CC)OCC3)=O)nn2)ccc(Cl)cc1Cl 16383,c1(C(=O)NCCOCCNC(C2(C)CNC(=O)C2)=O)cc(Cl)cc(F)c1F 16384,N1(C(CC)=O)CCC(C)C(CCOc2cc(OC(C)(C)C)cc(COC)c2)C1 16385,c1(C(C)C)ncc(C(=O)NC2CC(CNC(c3cn(CCO)nn3)=O)C2)s1 16386,C1(CNC(=O)OC(C)(C)C)CN(C(=O)Cc2cn[nH]c2)CC1O 16387,C1(NC(C2(SC)CC(O)C2)=O)CN(C(=O)CSc2cccc(Cl)c2)CC1(C)C 16388,C(N=c1[nH]cnc2c(Br)nn(C)c12)C1CN(C(C=NOC)=O)C(C)C1 16389,c1(CC)cc(C(=O)NCC2CCC2NC(C2(C#N)CCC=CC2)=O)cc(F)c1 16390,N1(C(C2CC(OC)C2)=O)CC(CNC(c2cc(CO)[nH]n2)=O)C(C)C1 16391,CCCCCCCCC(F)C(=O)NC(C)CNC(c1cnc2ccnn2c1N)=O 16392,c1(C(=O)OC)ccc(NC2C3CN(c4ccccc4)CC23)c(F)c1 16393,C12(CNC(C=CSC)=O)CCC(CC1)N(C(c1cc[nH]c1)=O)C2 16394,c1(C(=O)NC2(COC)CCN(C(C(CCC)OC)=O)C2)cncc2ccsc12 16395,c1(C(=O)NCC(CC=C)NC(=O)CCc2cncs2)n[nH]c2c1CC(C)OC2C 16396,c1(C(N(CC(CNC(C(c2cccc(C)c2)F)=O)C)C)=O)cccc(C)c1O 16397,C(=O)(CC(C)CNC(c1ccccc1CC#N)=O)NCC(=C)Cl 16398,c1(CCCC(=O)NCCCNC(CSCCC(C)C)=O)cc2ccccc2o1 16399,c1(C(=O)NC(CCCC)CNC(c2cncc(C(F)F)c2)=O)c(C)ccnc1C 16400,c1(C(N2CC(CNC(C(CC)CO)=O)C(C)CC2)=O)cn2cnnc2cn1 16401,C1(NC(=O)CN2CC(C(F)(F)F)CCC2=O)CCCCN(C(C2CCC2)=O)CC1 16402,C1(C(=O)NC2(CC=C)CCC2)C2CCC(C2)N1C(=O)Nc1cc(NC)ccc1Cl 16403,N1(C(CSC)=O)CC(CCNC(C23CCC(CC2)OC3)=O)OC(C)C1 16404,c1(NC2C(C)CN(C(c3c[nH]ccc3=O)=O)C2)nc2c(cc1Cl)C(=O)OC2 16405,c1(OC)ccnc(OC)c1C(=O)NCC1(NC(C2COC(=O)N2C)=O)CCOC1 16406,Cc1ccc(F)cc1N(C)C(C1C2CN(C(c3cncnc3)=O)CC12)=O 16407,C1(N(C(=O)CC2CCCCC2)C)CC2CC1N(C(c1c[nH]cc1C(F)(F)F)=O)C2 16408,C1(CC#C)(C(=O)N(C(C)CNC(=O)Cc2ccnn2C(C)C)C)CCCCO1 16409,N1(C(CNC(CN(C)C)=O)=O)CC(NC(C23CCCC2C3(F)F)=O)C(C)(C)C1 16410,c1(C(=O)NC2CCN(C(C3CC(C(F)F)C3)=O)C2)ccc(CO)c(Cl)c1 16411,C(N=c1[nH]c(=NCCC(F)(F)Cl)[nH]c2c1SCC2)c1cc(CO)ncc1 16412,c1(SC)ncc(C(=O)NCCC2(O)CN(C(c3csc(F)c3)=O)C2)n1C 16413,c1(C(N2CCC(NC(CC(CCC)O)=O)CC(O)C2)=O)cnc2c(cnn2C)c1 16414,C#CCCCCC(=O)N1CCN(C(C2(C)CCOC2)=O)CC1C(F)F 16415,N1(C(c2n(CCC)nc(C)c2)=O)CCCCC(CNC(=O)CC2CC(SC)C2)C1 16416,N1(C(c2cc(N3CCOCC3)ncn2)=O)CCC(C2CC2(F)F)C1 16417,CCC(F)(F)C(=O)NCc1ccccc1N1CCN(C(C2(C#N)CC2C)=O)CC1 16418,c1(C(=O)NCC(O)CCNC(C2CCCCCCC2)=O)cncc2c1CCCC2 16419,C1(N(C(C=C(C)C(F)F)=O)C)CCC2CN(C(=O)Cc3ccsc3C)CC12 16420,N1(C(CCCC(C)(C)NC(C2CC2(F)Cl)=O)=O)CCCC2(CCOC2)C1 16421,C1(CNC(C(CCOC)(C)C)=O)CC2COCC2N1C(=O)Cn1ncn(C)c1=O 16422,N#Cc1ncn(CC(=O)NCC2CCC(NC(=O)Cc3ccn(C(F)F)n3)C2)n1 16423,C(CNC(c1cccc(-n2cccn2)c1)=O)(CC(C)C)NC(c1c(C)con1)=O 16424,c1(-c2ccccc2)ncc(OCCn2cc(C3CCCO3)nn2)cn1 16425,N1(C(CC2(NC(C)=O)CC2)=O)CCCN(C(C2CCS(=O)(=O)N2)=O)C(CO)C1 16426,C(C(=O)N(CC)OC)NC(C(C)N(C(=O)Cc1cnccc1C)CCC)=O 16427,c1(C(N2C(C)CCC(NC(c3c(CC)cno3)=O)C2)=O)ccc2cnncc2c1 16428,c1(C(=O)NC2CC(CCNC(c3cncc(C#C)c3)=O)C2)cc(S(C)(=O)=O)cs1 16429,N1(C(c2cn(CC=C)nn2)=O)CCC2(CCC2)C(CNC(=O)Cn2cnnc2)C1 16430,C(=O)(C#CC(C)(C)CNC(c1c[nH]c(C)c1)=O)NC1CCCN(CC)C1 16431,C(=O)(C(C)CC(C)C(C)=O)N1C(C)(CC(=O)NCC=CCSC)CC1 16432,Cc1cc(C(=O)NCC2CCC(CNC(C34CCCCC3C4)=O)CC2)ccc1F 16433,C1(C(N2CCC(N(C(=O)CCSCC)CCC)C2)=O)CC(F)CN1C 16434,C(=O)(CCCC(C)(F)F)NCCN(C(CCNC(CC(C)C)=O)=O)CC(C)O 16435,C1(CNC(c2c(C)onc2Cl)=O)CN(C(C2CCC(=O)C2)=O)CCC1(F)F 16436,C1(CCC(=O)NC(C)(CNC(c2cccs2)=O)C2CC2)CCCCO1 16437,c1(C(=O)NC(C)CCCCNC(=O)C(C)(O)C2CCC2)cn(C)c(=O)nc1O 16438,Cc1cc(F)c(C(N2CCN(C(=O)CC(C)(C)C)CC2C(C)C)=O)cc1F 16439,N1(C(CC2CC(C)(C)OC2)=O)CCC2CN(C(c3ccncc3)=O)CC2C1 16440,n1(CCCC)nccc1C(N1CCC(C(C)NC(c2nnsc2C)=O)C1)=O 16441,N1(C(CN2CCC(N(C)C)CC2)=O)Cc2ccccc2C(C(=O)NC2CC2)C1 16442,Cc1cc(CC(=O)NC2(CF)CCN(C(C3CCS(=O)(=O)CC3)=O)C2)cc(F)c1 16443,c1(CS(C)(=O)=O)ccc(C(=O)NCC2CN(C(c3scnc3C(F)F)=O)C2)cc1 16444,Cc1cc(C)c(C(=O)NC2CC(NC(=O)C(O)CC(F)(F)F)C2)c(O)n1 16445,C(C(=O)NOCC(=O)N(CC(C)O)C)(C(C)(C)C)OC 16446,CC(=O)C(C)CC(C)C(=O)NCC1CCC1NC(c1c(C)cc(C)oc1=O)=O 16447,C1(C)(CNC(CCc2c(C)ncs2)=O)COCCN(C(=O)C(C)C(F)F)C1 16448,N1(C(=O)NC)CC2CCC2(OCCCSC)C1 16449,CC1CCN(C(=O)CC23CC(C2)C3)C1CNC(c1ccsc1)=O 16450,c1(C(N)=O)nc(NC2CS(=O)(=O)CC2CC2CC2)cc(C2CC2)n1 16451,Cc1ncc(C(N2CC3(CCN3C(=O)CS(C)(=O)=O)C2)=O)c(Br)c1Cl 16452,C(=O)(C#CC1(C)CCCO1)N(C)CC1CCCN1C(c1cc(F)cnc1Cl)=O 16453,C12(C(N3CCC(COCC)C3)=O)CC(CO)(CN1C(=O)CCNC(C)=O)C2 16454,c1(CC(=O)NCC2CN(C(c3ccc(CO)s3)=O)CCCO2)cn2ccsc2n1 16455,C1(NC(C(COCC)NC(=O)CN2C(C)CCC2C)=O)C(C)CCC1C 16456,Cc1ccc2cccc(C(N3CC(O)(CNC(c4c(C)nsc4C)=O)C3)=O)c2n1 16457,C1(OC)CCCC(C(=O)NCC23CC2CN(C(=O)C(CCSC)OC)C3)C1 16458,CC1CN(C(c2cc(F)c[nH]2)=O)CC(C)N(C(c2cc(Cl)c(F)cc2O)=O)C1 16459,c1(CC(=O)NCC2C(NC(C(C)OC)=O)C2)cc(C)nn1C 16460,C#CCC(O)C(=O)NCC1C=CC(NC(C2(C(c3ccccc3)=O)CC2)=O)C1 16461,N1(C(c2c(OCC)cccn2)=O)CC2CC(NC(=O)C(=O)N(C)C)C2C1 16462,C(=O)(NNc1cc(F)ccc1C(F)(F)F)c1c(Cl)ccc(NC(CC(C)C)=O)c1 16463,C1(NC(c2cc(C3CC3)ccn2)=O)CN(C(=O)C(F)(F)Cl)CC1(F)F 16464,c1(OCC=C)ccc(S(N)(=O)=O)cc1C(N1CCC1CNC(=O)C(O)C1CC1)=O 16465,c1(C(COC)N(CC(C)C(=O)OC(C)(C)C)C(=O)C(C)(C)C)cccc(Cl)c1.C1(=O)CC1=O.O 16466,C(=O)(CC(C)(CN(C)C)C(F)(F)F)NC1(C)CN(C(C2C(CC)C2)=O)C1 16467,c1(CN(C)C)ccc(-c2ccc(C3(CNN4CCN(C)CC4)CCC3)cn2)cc1 16468,Cc1ccc(C(c2nnnn2C)NCC2(C(F)F)CCCO2)cc1 16469,C(Cc1ccccc1)(C(=O)N1CC(O)(CNC(=O)Cc2nc(=N)[nH][nH]2)C1)N(C)C 16470,c1(C(=O)NC2C3CN(C(CCCSC)=O)C2CC3)nc(C)c(N)cc1C 16471,C(CC(C(=O)N1CCC(C)(CN(C)C)C1)NC(=O)COC)=CC 16472,C1(NC(c2ccc(CSC)cc2)=O)CC2CN(C(C3(C)CCCC3)=O)CC12 16473,C1(CNC(COC(CC)CC)=O)CCCN(C(c2nnsc2C)=O)CC1 16474,N12CCC(CC1)C2=O.C1(c2cn(CCC3CC(OC)C3)nn2)CC2C=CC1C2 16475,Cc1ccc(I)cc1CNC(=O)C(=O)NC1CC(CCN(C)C)C1 16476,N1(C(C=CC)=O)CCCC2(C1)CN(C(C1C3Sc4ccccc4C13)=O)CCO2 16477,c1(C(=O)NCCN(CCC)C(c2cc(O)cc(Cl)c2)=O)cnn2cccc2c1 16478,Cn1c(C(N2CC(NC(=O)C3=CCCC3(C)C)C(O)C2)=O)c2n(c1=O)CCCC2 16479,CCCC(C)CC(C)(c1nnnn1C(C)C)Nc1ccc(C(=O)N(C)C)c(C)c1 16480,C12(NC(CCCCC(N)=O)=O)CN(C(=O)CCN3CCCC3)CC1CS(=O)(=O)C2 16481,CC(CC(=O)NC1CCCN(C(c2ccc(C3CC3)cn2)=O)CC1)C(F)F 16482,CC1CCN(C(=O)CCc2nncs2)CC1NC(C1CCN(C(=O)N(C)C)CC1)=O 16483,CCCC(CC)CC(=O)N1CC(COC)(NC(c2csc(COC)n2)=O)C1 16484,N1(C(c2[nH]nc(OC)c2Cl)=O)CCC2(NC(=O)Cc3cscn3)CCCCCC12 16485,c1(C(N2C(C(N)=O)COCC2)=O)cc2c(OC(F)(F)F)cccc2[nH]1 16486,C(=O)(C(C)P(C)(C)=O)NCCC1(NC(c2cncc(C(=O)OC)c2)=O)CC1 16487,Cc1cc(Cl)c(C(=O)NCC(C(C)C)NC(c2onc(C)c2C(F)(F)F)=O)s1 16488,CCCC(COC(=O)C(CC)OC)CCO 16489,S(=O)(=O)(c1ccc(NCC2CCCC3(CCOC3)O2)c(Cl)c1)NCCCCCC 16490,c1(OC)ccc(C(N2CCCC(C)(CNC(C3(N(C)C)CCC3)=O)C2)=O)cc1Cl 16491,CC1CC(C(N2CCCC2CN(C)C(c2cncs2)=O)=O)CC(C)C1 16492,c1(CNC(CN(C)C)=O)cccc2c1CN(C(c1cc3c(ccn3C)[nH]1)=O)C2 16493,c1(C(=O)NCC2CCC(NC(CN3CCC(C)C3)=O)C2)ccc2nc(O)[nH]c2c1 16494,N1(C(c2ccc(C(C)F)cc2)=O)CCCC(CNC(=O)CN(C)C2CC2)CC1 16495,Cc1nc(C)c(F)c(=NCCN(C(=O)C(C)(O)C(C)c2ccccc2)C)[nH]1 16496,CC(CC(C)(C)C)NC(=O)C(c1cccs1)NC(=O)CC1NC(=O)NC1=O 16497,C(=O)(CCCCC(C)CC)N1CCC(C)(CCNC(c2c(CC)noc2C)=O)C1 16498,c1(OC)ccnc(CC(=O)N(CC(C)(C)CNC(C2CC2c2ccco2)=O)C)n1 16499,N1(C(C(C)(C)C#N)=O)CCN(C(c2ccc(F)nc2F)=O)C(CCO)C1 16500,C=C1CCN(C(=O)CSCCC)C(C(=O)N(CCn2ccnn2)C2CC2)C1 16501,C1(CC(=O)NCC2COCCN2C(=O)CC2CCCCC2)CCC(F)(F)CC1 16502,N1(C(C(C(C)C)C)=O)CC(CNC(c2cc3ccccc3o2)=O)OC(C)(C)C1 16503,N1(C(c2n(C)ncc2Br)=O)CC2CCC2(CC(=O)O)C1.C1(N)CCC1 16504,C1(C(=O)NC(CCCNC(CSCCN(CC)CC)=O)C)Cc2ccncc2C1 16505,c1(CC(=O)OC)cn(CCCC(=O)OC)nn1 16506,C1(CNC(c2c(C)scn2)=O)CC2CCC1N2C(C1(C)CC(F)C1)=O 16507,CC(CC1CC1)C(=O)NCC(C)(C)NC(=O)C(C)n1ccnc1 16508,C1(C(=O)N2CCC(N3CCC3)C2)(C(CC)=O)CCCc2ccccc21 16509,CS(C)(=O)=NC(=O)C(=O)NC1CC(c2ccccc2)(NC(=O)COC(F)(F)F)C1 16510,C1(CNC(C(COC)N(C)C)=O)CN(C(=O)CC2CN(C(C)=O)C2)CCN1C 16511,O=C1NCC2(CCN(C(C3(NC(C4CC4c4ccco4)=O)CCC3)=O)C2)N1 16512,C(=O)(CC(C)NC(=O)CC1(C)OCCO1)NC(CC#C)C 16513,N1(C(C=CC=CC)=O)Cc2nccn2CC(NC(=O)CNC=O)C1 16514,C(c1cccc(CO)c1)=CC(=O)NCC(C)NC(c1ccnc(C(F)F)c1)=O 16515,c1(OC)ccc(C(=O)NC2CCCCC2NC(c2ncc(N)nc2C)=O)c(Cl)c1 16516,Cc1cc(C(=O)NC(C)(CNC(=O)CCC=CC(C)C)CO)n[nH]1 16517,CCC(CC(=O)N1CCC1CNC(c1ccc(CSCC)o1)=O)c1ccccc1 16518,N1(C(c2c(C)noc2C)=O)CC2(C1)SCCC2NC(=O)C(O)C1CCCC1 16519,CC(Cc1cccs1)N=c1ccnc(N2CCOCC(C)(F)C2)[nH]1 16520,c1(OC)cc(Br)cnc1C(=O)NCCC1(NC(c2cnn(C)c2)=O)CCC1 16521,c1(C(=O)NC(C(C)NC(=O)C=Cc2cc[nH]c2)C)cc2cc(Cl)cc(Cl)c2[nH]1 16522,c1(CCC(=O)NCC(CNC(c2ccn(CC)c2C)=O)CO)ccc(C)cc1C 16523,C1(NC(CCCN(C)C(c2cccnc2O)=O)=O)CCOC12CCOC2 16524,N1(C(C=CC(C)C)=O)CC(NC(c2ccc(-n3ccnc3)nn2)=O)CC2(CC2)C1 16525,CC(=O)CCCC(=O)NC(C)(CNC(c1nccc(Cl)c1Cl)=O)C1CC1 16526,n1(CCNC(C(C)C2CCCO2)=O)ccc(C(=O)NCC2(C(C)(F)F)CC2)c1 16527,CC1CN(CCCN2CCCNC2=O)CC1C(=O)O 16528,CCCCCC(C1CC1)NC(C1CCC(C2CC2)N1C(c1cnccn1)=O)=O 16529,C(=O)(CCCCCCNC(c1cccnc1)=O)N1CC(CC(C#C)C)C1 16530,C(C)(C)(CCN=c1[nH]cnc(C)c1Br)NC(c1c(C)occc1=O)=O 16531,CC(C)(C(=O)NCC(CC1CCCC1)C(=O)NCCCP(C)(C)=O)C(F)(F)F 16532,C#CCN(OC)C(=O)C1(CF)CCN(C(c2cn(C)c(C)n2)=O)C1 16533,CC(CCC(F)(F)F)NC(=O)CC(C)(C)NC(=O)Cc1ccsn1 16534,C(=O)(C1=CCCCCC1)NCc1ocnc1CNC(=O)CC1NC(=O)NC1=O 16535,c1(C(C)C(=O)NCC2(O)CN(C(=O)CSCc3cc(Cl)no3)C2)ccc(F)cc1 16536,Cn1cc(CN2CCC(NC(c3cncc(-n4cccn4)n3)=O)C2)c(Cl)n1 16537,CCC(CC(F)F)C(=O)N1CCC(CN(C(=O)C(C)c2ccco2)C)C1 16538,c1(SC)nc(C)c(CCC(=O)NCC23CCCC2CCN3C(=O)C(C)C)c(O)n1 16539,C1CC(=O)NNc2ccccc2-c2nc1n(CC)ccccc2 16540,C1(NCCS(C)(=O)=O)CC(NC(=O)Cn2cncn2)C12CCC2 16541,C(=O)(CC1=CCCCC1)Nc1ccc(OC)c(O)c1.C123CCC1CN(C2)C(=O)C3 16542,c1(C(N2C3C(NC(C=CC)=O)C(CC3)C2)=O)sc2ccccc2c1CS(C)=O 16543,Nc1nc(C(N2CCC3(NC(=O)COC(F)F)CC3C2)=O)ccc1O 16544,C1(c2nc(C)[nH]n2)CCC(CNC(N2CCOCC2c2ncnn2C)=O)CC1 16545,c1(C(N2CCC(N(C(C=CC=CCC)=O)CC)C2)=O)csc(=NC2CC2)[nH]1 16546,N1(C(c2cn(CC)nn2)=O)CCC(NC(=O)CCc2cccc(C)c2)C(CO)C1 16547,C(C1=CCN(C(=O)OC(C)(C)C)C1)C(C)=O.c12coc(n1)NC2=O 16548,CCC(C)(C)C(=O)N1CCC(N(CCO)C(C2CCC(C)(C)O2)=O)C1 16549,c1(C(C(=O)NCc2cccs2)N(CC)CC2CC(C)=NO2)cc(Cl)ccc1C 16550,C12(C3CCCN(C3)C(=O)N1)CC2.C1(C)(CC(=O)OC)CC(OC(C)(C)C)C1(F)F 16551,CN1CCCC2(CCN(C(CC3CCC4CC34)C(=O)NC(C)(C)C)C2)C1 16552,N1(C(c2c(C)c[nH]n2)=O)CCN(C(=O)CC2CC(O)C2(C)C)C(CCO)C1 16553,N1(C(C(C)CN(C)C)=O)CCn2ncc(C(c3cc(Br)ccc3F)=O)c2C1 16554,N1(C(c2onc(CC)n2)=O)CCC(C)C(CNC(=O)CCCCF)C1 16555,c1(C(N2CCCC(CN(C)C(C3CC(=O)NC3(C)C)=O)C2)=O)cccc(O)c1Cl 16556,N1(C(CCSCCC)=O)CCOC(CN(C(=O)CN2CC(C)(OC)C2)C)C1 16557,Cc1ccc(C(N2CCC(F)(C(=O)NCCCC(O)CO)CC2)=O)nc1C 16558,C1(CCC)CN(C(C2OCCC2C)=O)CC1C(=O)N(C)Cc1ccn(CC)n1 16559,CCC(C)(CNC(=O)COC1CC(NC(=O)CC2CCCCO2)C1)CC 16560,C1(O)(C(=O)NCC2CC(NC(Cc3ccn(CC)n3)=O)C2)CCCC(C)(C)CC1 16561,Cc1ocnc1CC(N1CSCC1C(=O)NOC(c1ccccn1)C)=O 16562,N1(C(C)=O)CCCC1CC(N1CC(O)(CCNC(=O)C(C)(C)c2ccno2)C1)=O 16563,C(=O)(C1=NOC(C)C1C)NCC1(NC(c2cc(F)cc(Cl)c2N)=O)CC(OC)C1 16564,CN1CC(N=c2nc3sccc3c(NCC(=O)NC3CC3)[nH]2)CC12CCC2 16565,c1(NC(=O)NC2CCCC(O)C2)nc2ccc(F)cc2o1 16566,C(=O)(C1=Cc2cc(Cl)ccc2OC1)NC1C2CN(C(Cc3cc(C)[nH]n3)=O)C1C2 16567,CC(C)(CC(F)C(=O)NCCC1CCSC1)NC(C1CC12CC2)=O 16568,c1(C(N2CC(NC(C3(CO)CC3)=O)CC(O)C2)=O)ccc2ncccc2n1 16569,c1(C(N2CCC(C)(CC(=O)N(CCCCC)C)C2)=O)cn2c(n1)CCC2 16570,C(=O)(CCCN=[N+]=[N-])N(CCOCCCNC(C1(OC)CCCC1)=O)C 16571,C1(CNC(c2coc3c2COC3)=O)CN(C(=O)C=CBr)C2CCN1C2 16572,c1(C(N2CC(c3n(C)cnn3)OCC2)=O)ccc(OC(F)F)c(F)c1 16573,c1(C(C(=O)NC(=O)OC(C)(C)C)N(C2COCC2CC)CC2CCC2)ccnc(O)c1 16574,C1(C(=O)NCC2(F)CC(NC(C3(CC(C)C)CC3)=O)C2)CCC2C(C1)C2(F)F 16575,C1(NC(c2c(C)cc(CO)o2)=O)CN(C(C2(C)CCCCO2)=O)CC1(C)C 16576,C1(NC(C2(C(=O)OC)CC2)=O)CC2CCC1CC2NC(c1cc(Cl)ncc1OC)=O 16577,N1(C(CCC#C)=O)CCC2CC(C(N3CCC(F)(CN)CC3)=O)C2C1 16578,C(C)(C)(C(C)CC(=O)N(C1CCCN(CC(F)(F)F)C1=O)C)NC 16579,N1(C(C=CC(C)(C)C)=O)CC2(C1)SCCC2NC(=O)COC1COC1 16580,C1(N(C(C=CC(CC)=CC)=O)C)CN(C(=O)Cn2ncc(Cl)c2C)CC1(C)C 16581,Cc1nnccc1C(=O)N(C)CC1CCN(C(c2ccc(C(C)(C)C)cn2)=O)C1 16582,N1(C(C2C(=C)C2)=O)CCC2CN(C(=O)CCCc3nncn3C)CC12 16583,C1(C(=O)NCC2(C)OCCO2)(NC(c2ccccc2)=O)CCCCC1 16584,Cc1nn(C)c(N)c1C(N1CCOC(CC(N2CC(C)C2(C)C)=O)C1)=O 16585,CC1(C)C(C(=O)NCC2CN(C(=O)C(C)(C)c3sccc3Cl)CCO2)C1(C)C 16586,NC(CC(=O)N1CCCCC1Cc1ccccc1F)C(=O)O 16587,c1(OC)c(Br)cc(CN(C(C)CC2CCC2)C)cc1Br 16588,Cc1cnc2n1CCC(NC1CCS(=O)(=O)CC1)C2 16589,c1(OC)ccc(C(=O)NCC(C(C)(C)C)NC(=O)Cc2cc[nH]n2)c(F)n1 16590,S(=O)(=O)(c1cc(C(=O)NC(C)CNC(=O)C(C#N)C(C)C)ccc1F)NCC=C 16591,N1(c2snc(C)c2C#N)CC2CCC1C1CN(C(=O)CSc3ncccn3)CC21 16592,C(C(C)(O)CC(=O)NC1CC(NC(c2nc(C)n(C)c2C)=O)C1)OC 16593,c1(CC)[nH]nc(C(=O)NC(CNC(c2ccnc(C(C)C)n2)=O)C(C)(C)C)c1Cl 16594,c1(C(=O)NC2CC(NC(c3c(C)ccc(F)c3)=O)C(O)C2)cccc2c1NCC2 16595,O=C1CN(C(=O)CCC2CCN(C(=O)Cc3ncccc3F)CC2)C2(CC2)CN1 16596,C(=O)(CCC(C)NC(C1CC(O)C(F)C1)=O)NC1(C(=O)OC)CC(C)C1 16597,c1(C(N2CC(C)C(NC(=O)C#CC3CCC3)C2)=O)cc2c(F)ccc(F)c2[nH]1 16598,c1(C(=O)NCC(C(C)(C)C)NC(c2cnc(S)[nH]2)=O)cc(O)ccc1Br 16599,C1(C(N(C2(C(N3C(C(=O)OCC)CC(O)C3)=O)CC2)C)=O)CCCCN1N=O 16600,N1(C(=O)CC2(CO)CC2)CC2CN(C(C3(c4cccs4)COC3)=O)CC2C1 16601,C(=O)(C(CC(C)C)C(C)C)NS(CCCOC1CN(S(C)(=O)=O)C1)(=O)=O 16602,N1(C(C2(CC=C)CCOCC2)=O)CC(NC(c2cccc(F)c2C)=O)C(C)(C)C1 16603,C(=O)(C1=NOC(C)C1)NCC(C(C)C)NC(C=CC(C)C)=O 16604,NS(=O)(=O)c1cccc(NCCCCc2nc(-c3ccccn3)cs2)c1 16605,C(=O)(C1=CCC2CCC1N2C(=O)C(C#N)C(C)(C)C)NCC=CC=CC 16606,C1(OCC)CC2(C1)CC2C(=O)NC1CCC(NC(C2CCCS2)=O)CC1 16607,C1(C(N2CC(CNC(COCc3ncc(C)o3)=O)C2)=O)CC2(CCC2O)C1 16608,N1(C(C2(C(CC)=O)CC2)=O)CC(C(N2CCOC(CCF)C2)=O)C(F)C1 16609,CN=c1[nH]c(C(N2CC(C(C)NC(C3CCN(CC(F)F)CC3)=O)C2)=O)cs1 16610,c1(OC)ccc(C(C(=O)O)NC(C2CCCCC2(F)F)=O)cc1Cl 16611,C(=O)(C(CNC(c1cc(C(N)=O)[nH]n1)=O)OC)NCC(=C)Cl 16612,C1(O)(C(CNC(C(C)N(C)C)=O)C)CCN(C(=O)Cc2sccc2Cl)C1 16613,N1(C(C#CC(C)(C)C)=O)CCCC(NC(=O)C=C2CCCCC2(C)C)C(F)C1 16614,Cc1ncccc1C(=O)NC1CC(O)(CNC(C2CC3(CSC3)C2)=O)C1 16615,C(=O)(C(C)CCCOC)N1CCC(OCCCNC(C(C)OCCC=C)=O)CC1 16616,c1(SCC(=O)NC(C2CCN(C(C(CC)F)=O)C2)=O)ccc(Br)cc1C 16617,c1(C(N2CC(NC(C3CN(OC)C(=O)C3)=O)C(C)C2)=O)nccn2cc(C)nc12 16618,C1(NC(c2ccc(OCC(F)(F)F)cc2)=O)CC(F)CN(C(C2CCCO2)=O)C1 16619,N1(C(C=C2CCC(C)C2)=O)CCC2CN(C(c3ccc([N+](=O)[O-])[nH]3)=O)CC12 16620,S(=O)(=O)(c1ccc(C#N)c(N2Cc3ccc(C)cc3C2)c1)NC1CC(=C)C1 16621,Cc1c(NCCCCN2CCC2)nc[nH]c1=NCCNC(N1CCOCC1)=O 16622,N1(C(c2cc(CC)nn2C)=O)CCCCC(C(=O)N(C)CCOC(F)F)C1 16623,c1(C(=O)NC2C3CN(C(c4ccc(NC)c(F)c4)=O)C2C3)cc2n(n1)CCCO2 16624,N1(CC(COC)O)CCC(N(C(=O)CC2CCN(c3ccccc3)C2)C)CC1 16625,C1(C(N2C(C(F)F)(CNC(=O)CSc3cccs3)CCC2)=O)CCOC(=O)CC1 16626,C#CC1CCN(C(=O)C(CNC(=O)CCCOC(C)C)N(C)C)CC1 16627,c1(C(=O)NCC2COCCN2C(C2CCS(=O)(=O)C2)=O)cc2nc[nH]c2cn1 16628,N1(C(C2CCN(C(C3(CO)CCC3)=O)C2)=O)CCCC2(CCC2)C1 16629,C12(CNC(C(C)(C3(C)CC3)OC)=O)CN(C(=O)CC3C=CCC3)CC(F)(C1)C2 16630,CC1(C)CC(NC(c2ccc(C3CC3)cn2)=O)CN(C(c2cccnc2S)=O)C1 16631,N1(C(C(CC=C)CNC(C2C3(CC3)C23CC3)=O)=O)CCc2ccc(F)cc21 16632,N1(C(CC(C(N)=O)NC(C)=O)=O)CC(CCO)OCC1(C)C 16633,c1(C(N2CC(COC)(CNC(C3CC3C)=O)C2)=O)noc2ccc(Cl)cc12 16634,N1(C(c2c(C)oc(CNC(=O)Cc3cc[nH]n3)n2)=O)CCc2nc(O)[nH]c2C1 16635,S(=O)(=O)(c1cc(Cl)sc1Cl)N(C(C(C(=O)OC)C)=O)Cc1ccccc1 16636,c1(OCCC(=O)NCCN(C(c2cnccc2C)=O)CC)cc(C)cc(C)c1 16637,CC1CN(C(c2cccc(C#N)n2)=O)CCC1NC(c1cc(=O)cc[nH]1)=O 16638,C1(OC)CCC2(C(=O)NCCCN(C(c3cnns3)=O)C(C)C)CCC12 16639,C(C(C)(C(=O)N1CC(C)(CO)C1)NC(=O)Cc1ccc(C)nc1)SC 16640,c1(NC(C2(CC)CCCC2)=O)cccc(CNC(c2ccoc2Br)=O)c1 16641,C1(NC(CSCCC)=O)CCCN(C(c2c[nH]cc2C(C)(C)C)=O)CC1 16642,C1(C2(O)CCN(C(C3CC3(C)Br)=O)CC2)(NC(C=C(C)c2ccco2)=O)CC1 16643,C1(C)(C(=O)ON(CCSC)CC)CN(CCCO)CCO1.c1(C)ccccc1 16644,Cc1ccc(Cl)c(CN2CCOC(CNC(c3c(O)cccc3Cl)=O)C2)c1F 16645,n1(C(C)(C)C)cc(Cl)c(=NC(=O)NCC(F)(F)F)[nH]1 16646,N1(C(C=CC(CC)=CC)=O)CCOCC(C)(CNC(c2cnncc2C)=O)C1 16647,Cc1c(C(=O)NCC(C2CCC2)NC(c2cc(-c3ccco3)no2)=O)nnn1C 16648,N1(CC)CC(C(N2CC=C(CNC(=O)CCc3ccnn3C)CC2)=O)CCC1=O 16649,c1(NC(CC(C)(C)N(C(C(N2C(C)CCCC2)C)=O)C)=O)cccc2c1CCO2 16650,C1(CC(=O)OC)(NC(C2CN(Cc3ccc(C)o3)CCS2)=O)CCCCC1 16651,C1(NC(C2N(C)CCCC2)=O)C2CC3C(C2)C13C(=O)N(CC1CC1)CC1CC1 16652,c1(C(N2C3CC(C(=O)NC(CC#C)C(=O)NC)C2CC3)=O)ccn2ccccc12 16653,C1(NC(C2ON=C(C)C2)=O)CCOCC1NC(c1nocc1C1CC1)=O 16654,c1(CC(=O)NCC(C2CC2)NC(C(C2CCC2)OCC)=O)sc(O)nc1O 16655,C1(C(=O)NCCNC(CC2(C=C)CCC2)=O)CCN(C(=O)NC2CCCC2)CC1 16656,N1(C(CC2C(C)CCN(C(C(C)(C)OC)=O)C2)=O)CCCc2ccccc21 16657,C1(N(C)C)CCCN(CC(=O)NCCNC(=O)Cc2ccc(CO)cc2)C1 16658,CCCCN=C(NCCc1ncc(C)cn1)NCC1CC1CC 16659,CC1OCCC1(F)C(=O)NCC1(CCNC(c2ccncn2)=O)CC1 16660,c1(C(=O)NCC2CCN(C(=O)Cc3cn[nH]c3)C2)cc2n(n1)CCO2 16661,C1(NC(c2nc(C(C)C)sc2)=O)CCN(C(=O)C(C)CF)C1C(C)(C)C 16662,C1(C(N2CCOCC(CNC(CC(C)C)=O)C2)=O)CCCN2CCCCC12 16663,CCCCCC(C(=O)N1CCC(NC(c2ccn(COC)n2)=O)C1)C(C)C 16664,C1(C(=O)NCC2(NC(C(CC)F)=O)CCCC2)CCCCN1S(C)(=O)=O 16665,N1(C(C2(C#C)CN(C(c3cc(C)ccc3O)=O)C2)=O)CCC(C2CCC2)C1 16666,CC(C)(F)CC(=O)NCC1COC(CNC(c2ncsc2Br)=O)C1 16667,C(=O)(C1=NN(CCO)C(=O)CC1)N1C(CC)CN(C(c2cnc[nH]2)=O)CC1 16668,CS(=O)CCC(O)C(=O)NC12CC(NC(=O)C=Cc3ccco3)(C1)C2 16669,CCCCCC(O)C(C)C(=O)N1CC(CNC(C2Cc3nccn3C2)=O)C(O)C1 16670,c1(CC(C)NC(=O)C(Cn2cncn2)NC(c2cncs2)=O)ccccn1 16671,C=CC1CN(C(C2(N(C)C)CCCC2)=O)CC1NC(=O)CC(C)C1CCCCC1 16672,N1(C(C2C(C(=O)OC)C=C2)=O)CCCC(C(=O)NC(C2CCCCC2)C)(CC)C1 16673,c1(NCC2C(C)C2C)nccc(=NC2CC(c3ccccc3)C2)[nH]1 16674,C1(C(C)C(=O)NCCc2ccccc2)CCCN(C(C2CC(F)(F)C2)=O)C1 16675,C1(CNC(CC=C)=O)CCCCC1NC(c1cnn(C2CC2(F)F)c1)=O 16676,Cc1oc(C)c(C(=O)NC2CCCC(NC(=O)CC3CC(=O)C3)C2)c1C 16677,C1(C(N2C(C)(CCC(=O)NCCC#CCO)CCC2)=O)CCCC12CCC2 16678,C1(CNC(C(C=C)(C)O)=O)CN(C(=O)CS(N)(=O)=O)CCCO1 16679,N1(C(C(C)C2CCOC2)=O)CCCCC1CN(C)C(c1ccno1)=O 16680,C1(C(=O)NC(C(N2CC(C(N)=O)OCC2)=O)c2ccco2)CC2CCCC2C1 16681,Cc1cc(=NC(C)CCNC(C2(F)CCC2)=O)c([N+](=O)[O-])c(C)[nH]1 16682,c1(CC(CO)NC(C2CCN2C(c2c[nH]c(C(=O)O)c2)=O)=O)ccccc1 16683,C#CCC(C)(CNC(C1C=CCN(C(=O)CC(C)n2cccc2)C1)=O)CO 16684,N1(C(C(C)Oc2cccc(F)c2)=O)CCCC(C)(NC(C2CC(F)C2)=O)C1 16685,c1(OC)ncc(CN2CC(NC(c3cc(O)n[nH]3)=O)C(F)(F)C2)c(OC)n1 16686,Cc1c(C(=O)NC(C2CCOC2)CNC(=O)C2=CCCCO2)nc2sccn12 16687,C1(CNC(C2C(C(C)(C)C)CC2)=O)CN(C(C2CC(CC3CC3)C2)=O)CCC1C 16688,C=CCC(C(=O)N1CCCC1CN(C(=O)Cn1ccnn1)C1CC1)C(C)(C)C 16689,c1(CC(N2CC(C)C(NCc3cc(Cl)c(F)cc3F)C2)=O)cn2ccccc2n1 16690,CCCC(C(=O)N1CC(O)CC1CC(N1CC2(CC(OC)C2)C1)=O)C(C)C 16691,CC1CN(C(c2cc(=O)cc[nH]2)=O)CC1CNC(=O)CC1(O)CC1 16692,C1(NC(COCC#C)=O)CS(=O)(=O)CC1NC(c1sccc1SC(F)F)=O 16693,S(=O)(=O)(c1ccc(Cl)cc1)NCC(=O)NC(CNC(CCC(=C)Cl)=O)C(C)C 16694,CCCC(CCCNC(c1ccc(CC)nc1)=O)NC(=O)CN(C)C(C)=O 16695,C1(CNC(C(C(CC)C)O)=O)C(C2CC2)CCN1C(c1ccsc1C)=O 16696,c1(NC(C23CC(C(=O)Nc4cncc(Br)n4)(C2)C3)=O)cc(O)cc(O)c1 16697,C1(C(N2CC(NC(c3c(CC)ncs3)=O)C(F)C2)=O)CCC2(CCC2)CC1 16698,C1(C(=O)NCCc2cccnc2)CN(Cc2ccncc2)CCN1 16699,CC(C)(C)C#CC(=O)NCCC1CCCN(C(C2CCC(N(C)C)CC2)=O)C1 16700,c1(C(=O)NCCC2CN(C(C3(CC#C)CC=CCC3)=O)C2)cnc(C)cc1C 16701,N1(CC(=O)NCC2(CN(C(=O)Cc3cccs3)C)CC2)CC(C)(C)C1 16702,Cc1ccccc1C1(C(=O)NC2CCCC2NC(c2ccnc(S)c2)=O)CCC1 16703,c1(-c2c(C(=O)NC(C(C)NC(C=NOC)=O)C)c[nH]n2)cccc(F)c1 16704,C1(NC(C(CSC)OC)=O)CCC(NC(=O)CC2(O)CCCCC2)CC1 16705,C(=O)(C1CCCc2nn[nH]c21)NC1CN(C(CCCCN(C)C)=O)CC(F)C1 16706,CC1CCCN1CC(=O)N(CC(=O)NC(c1cnn(C)c1)CO)CC(C)O 16707,C1(CNC(c2n(CC#N)ncc2)=O)CC2CC2N1C(c1ccncc1Br)=O 16708,N1(C(C(C2CCCC2)NC(c2n(C)ccc2)=O)=O)CCC(O)CC1 16709,c1(CN2CCCC(CC(=O)NCCC(=O)OC(C)(C)C)C2)cnc2[nH]ccc2c1 16710,Cc1nc(C)c2c(n1)OC(COC(C1CCCC(C(N)=O)CC1)=O)C2 16711,CC(C)C(C)(O)C(=O)NCCC1CN(C(c2c[nH]nc2C2CCC2)=O)CCCO1 16712,c1(C(=O)NCC(C)N(C(C(C)OCC#C)=O)C)ccc(-c2cccs2)cc1F 16713,C(=O)(CCC(C)NC(=O)CC1(NC(C)=O)CC1)NC1(CC=C)CCCC1 16714,C12(CC(N3CC(SC)C3)=O)CCC1CN(C(C1CCC=CCC1)=O)C2 16715,c1(CCC(=O)NC2CC(NC(C(C)C(C)(F)F)=O)C2)n[nH]c2c1CCCC2 16716,C1(F)(CNC(c2c(CC)cns2)=O)CCN(C(c2c(C)nsc2N)=O)C1 16717,c1(CN(C(C)CN2CCOCC2)CC(=O)N(C)C)cccc(F)c1C(F)(F)F 16718,N1(C(c2c(C)csc2)=O)CCCC2C1CCCN2C(=O)Cn1nc(C)c(C)c1C 16719,Cc1cc(F)c(I)cc1C(=O)NC1CC2CC1CN2C(C1CCCC1C)=O 16720,CCCC(C(F)(F)F)c1nc(-c2cc(OC(C)C)ccn2)nn1CCOC 16721,c1(OC)ccc(C(=O)N(CC(C)NC(=O)COCCc2ccccc2)C)cn1 16722,C1(NC(C(=O)NC(C)C)=O)CCS(=O)(=O)C2(C1)CC(CNC(=O)CC(C)C)C2 16723,CC1(F)COCCN(C(C2CN(C(=O)CC3=CCCC3)CC2(F)F)=O)C1 16724,C1(C)(NC(CC(=O)NCC)=O)CCCN(C(=O)CCC23CCC(CC2)C3)C1 16725,c1(C(N2CC(CCCCNC(C(C)CC(F)F)=O)C2)=O)c(O)cc(Cl)cc1F 16726,N1(C(C2CC3(C(OC)CC3)C2)=O)CCC(NC(=O)C(=O)N(C)C)C12CCC2 16727,C1(NC(CS(CC)=O)=O)CC1C1CCCN(C(=O)C(CO)NC(=O)C(C)C)C1 16728,c12cccc(F)c1C(=O)N2.c1(NC(N(CCC)CCC)=O)[nH]nnc1N(C)C 16729,C(=O)(C1=CCCOCC1)NC1(CC=C)CCN(C(c2n[nH]c3c2CCSC3)=O)C1 16730,c1(OC)cc(Cl)c(CN2CCC3CN(c4ncncc4Br)CC23)cc1OC 16731,C1(C(N2CC(CC=CC)N(C)CC2)=O)(NC(=O)OC(C)(C)C)CCS(=O)(=O)C1 16732,c1(OC)nc(Cl)ccc1C(N1CCC(CNC(c2ccc(Cl)cn2)=O)(OC)C1)=O 16733,c1(C(=O)NC2CC(CNC(C=CC(=O)N(C)C)=O)C2)cc(=O)n2ccccc2n1 16734,C(=O)(CCC(=O)NN(C)C)N(CCCNC(C(CCC)NC(N)=O)=O)C 16735,C(=O)(CCS(=O)(=O)CC(C)C)NCCN(C(c1c(CCC)occ1)=O)C 16736,C1(O)(C(N2CCCC(CCNC(c3c(C)n[nH]c3)=O)C2)=O)CCCC(C)CC1 16737,CCC(CNC(C)=O)CC(=O)N(CCCCCC(=O)N(C1CCOC1C)C)C 16738,CCC(CC)(CC)C(=O)NCC1CN(C(C2CCC(C)(C)O2)=O)C(C)(C)C1 16739,c1(OCC(=O)NC(c2nc(C(=O)O)cs2)C)ccc(N2CCCC2=O)cc1 16740,C1(CC)CN(C(C2CC3CCC2O3)=O)CCN1C(c1ccc(NC(N)=O)cc1)=O 16741,c1(C(=O)NC2CCN(C(C(C)OC)=O)CC2F)n[nH]c2c1CCC2C 16742,C(=O)(C(CCF)NC(c1ncccc1C)=O)NC(CCC=C)C 16743,C(CCC(=O)N(C)CCNC(C1CCCC1CC)=O)N(CCC)CCC 16744,N1(C(C=CCOCCOC)=O)CCCC(N(C(=O)C(N2C(=O)CCC2=O)C)C)C1 16745,N1(C(C(CC(N)=O)O)=O)CCC(C2CCCN(C(c3cnns3)=O)CC2)CC1 16746,c1(CNC(C2C(C)(C)C2(C)C)C)ccc(Cl)cc1F 16747,CC1(C)CCC(=CC(N2CCCCC2CNC(c2n[nH]cc2[N+](=O)[O-])=O)=O)CC1 16748,c1(CCC(=O)N(C2CCN(C(C3CN(C(C)C)C3)=O)C2)CC)n[nH]c(=N)s1 16749,C12(C(=O)NCCC(C)NC(Cc3cc(C)ns3)=O)CC(C)(C1)OC2(C)C 16750,c1(OC)cc(C(=O)NC(Cc2cnn(C)c2O)C(=O)N2CC(C(C)C)C2)n(C)n1 16751,C1(OC)C2CC3CN(C(c4sncc4Br)C(=O)NC4CCOC4)C1C3C2 16752,C1(N(C(CC(=O)NC)=O)C)CN(C(=O)C(C)C=Cc2ccccc2)CC1O 16753,c1(CCC(N2C(C3(NC(C(CSC)C)=O)CC3)CCC2)=O)csc2ccccc12 16754,C(=O)(C(CCC)NC(=O)C(C)(C)O)NCc1cn(CC#C)nc1 16755,Cc1cc(F)cc(C(=O)N(CC(C)NC(c2nc(C)n(C)c2C)=O)C)c1N 16756,CC(C)C1=NOC(C)(C(=O)NC(CNC(C2CCN(C)CC2)=O)C(C)C)C1 16757,n1(CC)nnnc1C(c1nc(C(F)(F)F)cs1)NCC1(C)CCCC1 16758,CCC(C)CCC(=O)N(CCC(C)NC(c1cnn(CCN(C)C)c1)=O)C 16759,c1(NC)ccc(C(N2CC3CC(NC(c4cc(C)c(C)o4)=O)C2C3)=O)cc1F 16760,N1(C(C(C)OCCCC)=O)CCN(C(=O)C=C(CC)CC)CC(CO)C1 16761,c1(CNC(C2CCC3(CCC3)CC2)=O)nc2cccnc2[nH]1 16762,C12(C(=O)NCCOCCNC(C3CCS(=O)(=O)N3)=O)CCN(CC1)CC2 16763,c1(C(N2C3CC(CNC(C(COC)COC)=O)(OC3)C2)=O)nccn2nccc12 16764,c1(NC(C(C)OC(C(CCSC)OC)=O)=O)ccc(CN)cc1F 16765,C1(CNC(=O)Cc2cc[nH]n2)CCCC12CCN(C(c1cccnc1Cl)=O)CC2 16766,c1(C(N2CC3C(C(=O)NC4CCCCC4(F)F)C3C2)=O)cc(F)cc(F)c1F 16767,Cc1cnc(C(N2CC(C(=O)NC3(C)CC=CCC3)C(C(C)C)C2)=O)cn1 16768,C1(C(N2CCCC(NC(=O)CCc3ccncc3)CC2)=O)CCC2(CCC2)CO1 16769,N1(C(c2c(C)nc(CCC)o2)=O)CCC(NC(C2CCC(O)CN2C)=O)C(F)C1 16770,N1(C(c2c(C)cc(C)s2)C(=O)NCc2ccco2)CCSCC1(C)C 16771,c1(C(=O)OCC)cncn1CCN(C(c1ccc(C(C)(C)C)o1)C(=O)NCC)C 16772,CCCCC(O)CC(=O)N1CCC(C(=O)N(C)Cc2cccc(C)n2)C(C)C1 16773,C1(C(=O)NC(C2CN(C(=O)CC3NC(=O)NC3=O)CCO2)C)C2C3CCC(C3)C12 16774,c1(C(=O)NCC2C(NC(C3CC(C)(C)C3)=O)CCC2)c[nH]c(=O)cn1 16775,n1(CC#C)cccc1C(=O)NCC1(F)CC(NC(=O)CC(C)N2CCCC2=O)C1 16776,c1(C(N(CCCOCCNC(C2C(C=C)C2)=O)C)=O)ccc(C)nc1N 16777,c1(CC)nc(C(=O)NC(C)C(C(C)C)NC(c2ccnn2CC(F)F)=O)c(C)o1 16778,C1(NC(c2c(SCC)nccn2)=O)COC2CN(C(c3cc(OC)cs3)=O)CC12 16779,C(=O)(C(CCOCCO)NC(=O)CCC1(C)N=N1)N(CC(COCC)O)C 16780,C(C1CCCN1C(=O)COCCC)=CC(N1C(C#C)CC1)=O 16781,c1(C(=O)NC(CNC(C(CCC)C(C)C)=O)(C)C)cc(O)nc2cnccc12 16782,C(CO)(C(=O)NCC1CCCN1C(C1(CC(=O)OC(C)(C)C)CC1)=O)N(C)C 16783,c1(C(=O)NCC2(F)CCCN(Cc3c(C)ccc(C)c3)C2)c(Br)ccc(C)c1F 16784,C1(C(N(C(CNC(Cn2ccc(C)n2)=O)C)C)=O)COC2(CO)CC1C2 16785,C1(C(=O)NCC2C=CCN2C(c2cnc(C3CC3)s2)=O)C(Cl)(Cl)C12CC2 16786,c1(C(N2CCOC(CCO)C2)C(=O)NCCC#N)cncc(C2CC2)c1 16787,N1(C(C=Cc2c(C)nccc2)=O)CCCC12CCN(C(C1CN(C3COC3)C1)=O)C2 16788,S(=O)(=O)(c1ccc(NC2CCCCCC2CO)c(F)c1)NC(CC)CSC 16789,C1(NC(C(C=C)(C)CC)=O)CC2(CCN(C(C3(C#N)CCCC3)=O)CC2)C1 16790,N1(C(C(CNC(c2cnn(C=C)c2N)=O)CC2CC2)=O)CCC2(COC(=O)N2)C1 16791,CC1=C(c2ccco2)CN(C(=O)NCC2CC3CC4CC(C3)CC2C4)CC1 16792,CN1CCC(NC(=O)Nc2ccccc2OCC2CCCCO2)CC1=O 16793,n1(C(C)C)cc(C(=O)NC(C)C(C)NC(c2cc(N)c(Cl)cn2)=O)c(O)nc1=O 16794,c1(CC(=O)NC(C)(C)CCNC(C2CCCC2(C)C)=O)cc(Cl)cc2c1OCC2 16795,CC1CC2(CC(NC(c3ccnc(OCc4ccccc4)c3)=O)C2)C1 16796,C1(NC(c2cc(CC(C)C)n[nH]2)=O)COCCC1NC(=O)C(C)c1ncco1 16797,Cc1nc2cccc(C(N3CC(CNC(c4ccc(=N)[nH]c4)=O)CC3C)=O)c2[nH]1 16798,N1(C(=O)Cc2nc(Cl)cs2)CCN(Cc2ccc(Br)c(F)c2)C2CC12 16799,N1(C(c2snnc2C)C(=O)NCCOCC)CCC(CCN(C)C)CC1 16800,c1(C(=O)NC2CC(NC(C(COC(C)C)(C)C)=O)C2)ncn2c1CCC2 16801,C1(CC(=O)NCCC2CCCN2C(=O)CN2CSCC2=O)CCCCO1 16802,c1(NC(C2N(Cc3cnn(C)c3Cl)C3CCC2C3)=O)cccc(Br)c1[N+](=O)[O-] 16803,C1(C(N2CCN(C(c3n[nH]c(C)c3F)=O)CC2)=O)CCC2CCCCN12 16804,N1(C(COCCCC)=O)CC2CCN(C(C3(CCCF)CC3)=O)CCC2C1 16805,N1(C(CCC(C)C)=O)CCCCC(CNC(=O)C(c2cncnc2)C)CC1 16806,c1(CCC(=O)NCC2(F)CN(C(C3C4CC5C(C4)C35)=O)C2)ccc(F)cc1Cl 16807,N1(c2nnc(CC)o2)CCCC2(CN(C(=O)CC(C)O)CCO2)C1 16808,N1(C(C(C)CN(C)C)=O)CC2CC(NC(=O)CCC3CCC3)CC1C2 16809,N1(Cc2nnc(C(C)(C)C)o2)CCC2(CCN(C(c3c(F)cccc3Cl)=O)C2)C1 16810,N1(C(c2nc(OC)c(C)s2)=O)CCN(C(C2CC3CCC2O3)=O)CC(CO)C1 16811,C(=O)(C(CO)C(C)(C)C)NC(C(=O)NCC(C(=O)OC)C)C 16812,N1(C(c2c(C)snn2)=O)CCCC(O)(CCNC(=O)C(O)C(F)(F)F)C1 16813,C=CC(C)(C)CC(=O)NCC1(C)CCC(NC(c2ccoc2Cl)=O)C1 16814,C(CNC(C1(S(C)(=O)=O)CCC1)=O)(C(C)C(C)C)NC(c1nc(CC)oc1)=O 16815,c1(CC(=O)NC2CC(CNC(c3cc(F)cs3)=O)C2)nnc(O)s1 16816,C1(C(=O)Nc2c(OC(CC)C)cc(C(N)=O)cc2)CCc2nnc(C(F)F)n2C1 16817,c1(C(N2CC(CNC(C(C)CC3CCCC3)=O)OCC2)=O)cncc(N=[N+]=[N-])c1 16818,C1(NC(C2C(OC)CCC2)=O)CCN(Cc2ncc(C)o2)CC(C)(C)C1 16819,N1(C(=O)CN(CCO)CCO)CC2CN(Cc3c(Br)ccnc3Br)C2C1 16820,C1(C(=O)NC2(CNC(c3c(C)[nH]cc3)=O)CCOCC2)CC12CCOCC2 16821,c1(N(C)C)cc(C(=O)NCCNC(C2CC(N3CCCC3)C2)=O)cc(Cl)n1 16822,c1(CC)ccc(C(=O)N(C)CCNC(c2ccccc2CS(C)(=O)=O)=O)cn1 16823,c1(C(c2nnnn2CCSC)Nc2cnn(CCC)c2C)cc(Br)cc(F)c1O 16824,c1(C(=O)NC2CC(O)CN(C(=O)CCc3ccnc(Cl)c3)C2)cnc2nccn2c1 16825,N(C(=NCCCC(C)(C)C)NC1CCC1)CC1C(C)COCC1 16826,C1(NC(C(=Cc2cccs2)C)=O)CC2(CCN(C(=O)Cc3ccsc3Cl)C2)C1 16827,C1(NC(c2cnn[nH]2)=O)CCN(C(c2nnc(O)cc2O)=O)C(C2CC2)C1 16828,C1(C(=O)NCC(C2CC2)NC(CCN(S(C)(=O)=O)C)=O)CCCCN(C)C1=O 16829,c1(C(N2CCN(C(c3c(SC)ccs3)=O)C(CO)C2)=O)cccn2nncc12 16830,C(CCCCC(=O)N(CC)CC1CCC1)NC(c1c(-c2cn(CC)nc2)n[nH]c1)=O 16831,O=C(N=c1[nH]ccnc1Br)c1csc(=NCc2cc(F)ccc2I)[nH]1 16832,C(=O)(C1=NOC2(CCNC2)C1)N1CC(C)N(C(=O)Cc2ccc(F)cc2)CC1 16833,C1(C(N2C(CNC(=O)CCc3cccc(Cl)c3)CC2)=O)CCc2cncn2C1 16834,N1(C(c2nn(CC)c(C)c2)=O)CC2CN(Cc3ccc(C)cc3C)C2C1 16835,N1(C(CCCC)=O)CCN(C(=O)C(CC)CC)C(c2cc(F)ccc2F)C1 16836,C1(CC(NOCCCC)=O)CCN(C(c2ncoc2C2CC2)=O)CC1 16837,C(=O)(CC(F)(F)Cl)NCCOC1CCN(C(C2CC(CC(C)(C)C)C2)=O)C1 16838,CC1CC(CNc2cn(C3CCCCC3(F)F)nn2)CC(C)C1 16839,CC(CC(=O)NC1C(C)(C)CN(C(=O)C2=CCCSC2)CC1(C)C)CC(C)(C)C 16840,Cc1ccc(CNC(C2(CO)CCCCO2)=O)cc1C1CC1 16841,CN1CCOC(C(=O)NCC(C2CCCC2)NC(c2cnc(N(C)C)s2)=O)C1 16842,C#Cc1ccc(C(=O)NC(CC2CC2)C(=O)NCc2nncn2C2CC2)c(C)c1 16843,C(=O)(CCC(C(C)C)NC(=O)CCOCC1CCC1)NC(C(=O)OC)CO 16844,c12c(C)sc(C)c1NC(=O)Cn1cc-2nn1.C1(C)(C(=O)OC)CCC1(C)C(=O)O 16845,N1(C(c2ccc(OC)cn2)=O)CCC(N2CCC(CCCO)CC2)C2(CC2)C1 16846,N1(C(=O)C=C2CC2)CCC(C2CCCN(C(c3cc(C(F)(F)F)ccn3)=O)C2)C1 16847,N1(C(C(C)=CC)=O)CC2CC(C1)C(CO)C2NC(=O)C(O)(CC)c1ccccc1 16848,c1(C(CC)=O)ccc(C(=O)NC2CC(NC(=O)C(C(C)C)n3cncn3)C2)cc1 16849,C=Cc1cnn(C)c1C(=O)NC(C)CC1CN(C(=O)C(C)(C)C(=O)OCC)C1 16850,c1(C(=O)NCCNC(C2(n3cnnn3)CCOCC2)=O)cc2n(n1)CC(F)C2 16851,CC1CCN(C(=O)CCN2CCN(C)CC2)CCN1C(C1CC2(CCC2)CO1)=O 16852,CC(F)(C(=O)NC(CNC(=O)CNC(C1CCCCC1)=O)C1CC1)C(F)(F)F 16853,c1(NC)ccc(C(=O)NC(C)(C)CN(C)C(C2(C(F)F)CC2(F)F)=O)cn1 16854,c1(C(=O)NC(CC(C)NC(=O)C=C(Cl)Cl)C)nccc2c1[nH]c1ccccc21 16855,C1(NC(c2scc(C)c2)=O)CCN(CCNC(C2CCS(=O)(=O)C2)=O)CC1 16856,N(C1c2ccccc2C2CC12)C(N1CCC12CCOCC2)=O 16857,C(=O)(C1=CS(=O)CCC1)NCCN(CCC)C(c1cn(C(F)F)c(C)n1)=O 16858,c1(C(=O)NC2(C)CCN(C(c3c(C)[nH]nc3Br)=O)C2)ccc(Cl)c(F)c1 16859,N1(C(c2nccc(C)n2)=O)CC(N(C)C(c2oc(C)cc2C)=O)C2(CC2)C1 16860,c1(OC)cc(C(=O)NCC(O)CN(C(=O)C=C2CCOCC2)C)c(OC)cc1Cl 16861,Cc1ccc(N)c(C(N2CCC(C(C)NC(C3C(C)C3C)=O)C2)=O)c1 16862,c1(NC(N2CCN(CCc3cccs3)CC2)=O)cn2ccc(Cl)cc2n1 16863,N1(C(c2cc(C)n(Cc3ccccc3)c2C)=O)CCc2cc(C(C)(C)C)ccc21 16864,C1(C)(CC)C=C(C(=O)N2CC(C(=O)NC3CN(C(C)C)CC3C)(CC)C2)C1 16865,C1(C(=O)NC(CCNC(CCOC(CC(C)C)C)=O)C)CCC2C(C1)C2(F)F 16866,c1(NC(CCC)c2ccco2)cc(C(N2CCCC2CS(C)(=O)=O)=O)ncn1 16867,Cc1cc(C(F)(F)F)ccc1S(=O)(=O)NC(=O)C1CCc2scnc21 16868,N1(C(CCC)=O)CCCC1(C)C(=O)NCCNC(C1CCCC1)=O 16869,C1(COC)(NC(=O)CCNC(C)=O)CCN(C(=O)CC2CCNC2=O)C1 16870,C(=O)(C1CCCc2cncn21)NCC(C)(C)NC(C(c1ccc(F)cc1)C)=O 16871,c1(C(N2CC(NC(c3cnc(C)[nH]3)=O)C(F)C2)=O)c(F)cc(C(F)(F)F)cc1F 16872,C1(C(N(CCOC)Cc2ccc(F)cc2)=O)CC2CC2N1C(c1cnc(Cl)s1)=O 16873,c1(C(=O)NCC(C)NC(c2nc(C(C)=O)sc2)=O)cc2c(s1)CCOC2 16874,C(=O)(C(F)CC(C)(C)NC(=O)C(C)=C1CC1)N1CC(OC(=O)NC)C1 16875,c1(CCC(=O)NC2CN(C(C(COC)O)=O)CC2C(F)F)ccc2c(c1)CCO2 16876,N1(C(c2ncc(OC)nc2)=O)CC2CCN(C(C34CCC(OC)C3C4)=O)C2C1 16877,O(NC(=O)C(C)(C1CC1)N(C)C(c1ccc(SC)o1)=O)CCCOC 16878,c1(COC)nc(N(CCCCO)C)cc(N2CCCC(c3ccccn3)C2)n1 16879,N1(C(C(C)OCC)=O)CCN(C(c2c([N+](=O)[O-])c(C)nn2C)=O)CC(C)(F)C1 16880,CC1CC(O)CCN(C(C2CC(CNC(=O)C(O)CC(F)(F)F)C2)=O)C1 16881,c1(CC(=O)NCC2(O)COC2)ccc(CC(F)(F)F)cc1 16882,C(=O)(CCCN(C(=O)C(Cc1cc[nH]n1)NC(=O)CSCC(F)F)C)OC 16883,S(=O)(=O)(c1ccc(N2CCC(O)C(F)C2)c(C#N)c1)NC(c1cccs1)(C)C 16884,c1(OCC)ccc(C(N2CC(CO)(NC(c3ccc(F)o3)=O)C2)=O)c(F)c1F 16885,N1(C(c2n(CC)cnn2)=O)CC(NC(c2nc(Cl)cs2)=O)CC(C)C1 16886,C(=O)(CCCCCO)NC12CC(C(N3CCCC3c3ccc(Br)cc3)=O)(C1)C2 16887,C1(N(C)C)CCCN(C(C2CC23CC(NC(c2ccc(Cl)cn2)=O)C3)=O)C1 16888,C(=O)(C(O)C(C)(C)C)N1C(C(=O)NC(C2(CC(F)F)CCC2)C)CCC1 16889,CC1CCC(O)C(C2CCCN2CCC2CC23CC3)C1 16890,CC1CCc2nc(C(=O)NC3CCCC3NC(=O)CC3CC=CC3)cn2C1 16891,CC1(C)C(C(=O)NC2(CNC(c3cscc3Br)=O)CCOC2)C1(C)C 16892,c1(C(=O)Nc2c(C#N)scc2)ccc(F)c2c1CCC2 16893,c1(C(=O)NCC(CC)NC(=O)C(c2cn(C)nc2C)C)cncc(NC)c1 16894,c1(NC(C2CCN(C(C3C(CC)CCO3)=O)C2C)=O)cc(OC)cc(O)c1 16895,CCC(CCCC(=O)NC1CN(C)CC(F)(F)C1)NC(c1nnc(O)nc1O)=O 16896,c1(CC)ccc(OCCC(=O)NCC2CCN2C(=O)CC(CC)C2CCC2)cc1 16897,c1(CCC(=O)NC2C(NC(CCCCCC=C)=O)C2)cccc2ccccc12 16898,C1(C(N2CC(SC)C2)=O)CCN(C(C2C3CCCC23)=O)C(C)C1 16899,c1(C(N2CC3C(C2)N3C(=O)Cc2cccc(Cl)c2)=O)cc(F)nc(F)c1 16900,c1(CNC(Cc2cnn(C)c2O)=O)c(Cl)ccnc1Br 16901,C1(C(=O)NCCC=C=C)CN(C(=O)Cc2ccccn2)CCN1C 16902,C(=O)(C(CC(C)C)OC)NC(C(N1C(CC)(CC)CC1)=O)CC1CCCC1 16903,c1(-n2c(Cc3cnc(C)o3)nc(C(F)F)n2)ccc(F)c(C)c1 16904,C1(C(=O)NC(CC#C)CO)C2CC3C(C2NC(C2CCCC(CF)C2)=O)C13 16905,c1(C(=O)NC2CCC(NC(c3nocc3C3CC3)=O)C2)cc2ccc(F)cc2o1 16906,Cc1[nH]nc2c(C(N3CC4(CNC(=O)Cc5cc[nH]n5)CCC3C4)=O)cccc12 16907,c1(-n2cc(C(C)N(C)C(c3nn(C)nc3Br)=O)nn2)cc(F)cc(F)c1 16908,n1(CC(=O)NC(C2CCCC2)CNC(=O)C2=CCC2)nc2n(c1=O)CCCCC2 16909,C(C)(C(C)(C)C(=O)NC1COC(C(C)C)C1)NC(c1cccc(CC)n1)=O 16910,N1(C(CCC=CCC=C)=O)CC2CC(C)N(Cc3ncc[nH]c3=O)C2C1 16911,c1(OCC=C)ccccc1C(=O)NCC(=C)CCNC(=O)Cc1sc(C)nc1C 16912,C#CC1(OCC(=O)NCC(=O)NCCc2noc(CC)n2)COC1 16913,n1(CCC)cc(C(=O)NC2C3CC2N(C(=O)Cn2nnnc2C(C)C)C3)c(C)n1 16914,CCC(C)CCC(=O)N1CC(C2CC2C(N2CCC(COC)C2C)=O)C1 16915,N1(C(C2(c3ccc(C)cc3)CCC2)=O)CCCCCC(NC(c2cc[nH]c2)=O)C1 16916,N1(C(CC(=C)C)=O)CCC2(CC1)CC(NC(=O)Cc1cnn(C)c1)CO2 16917,C#CCC(CC(F)F)C(=O)NC(C)CCNC(=O)C=CCN(CC)CC 16918,Cc1oc(C(=O)OCC2CCC3(C2)CC3(F)F)cc1S(=O)(=O)Nc1ccccc1 16919,C123COC(C1)(C2)C(=O)NCC=CCNC3=O.c1(COC)ccc(C)nc1 16920,C(=O)(C(C)C(O)CC(C)C)N1C2(C(=O)NCCn3c(CC)ncc3)CC(C1)C2 16921,C1(C(C(=O)NCCCOC2CCC2)NC(C(=O)NCC)=O)CC=CCC1 16922,c1(C(=O)NCC2CC(F)(F)C2(F)F)ccc2nc(O)[nH]c2c1F 16923,C1(C(=O)NCC2CN(C(C(C)(C)c3nccs3)=O)C2)CCCC2C1C2(F)F 16924,C(=O)(CCC(=O)N1CCN(C2CCC2)CC1)NCC(CC)CC 16925,N1(C(C(C2CCC2)OC)=O)CCC(C=CC(=O)NC2CCCC(O)C2O)CC1 16926,c1(C(N(CC(C)OC)C(C)C)=O)conc1C(C)NC(=O)C(C)NC=O 16927,C=CCC(C)(N)C(=O)NC1CC(C)CCC1C 16928,c1(CCC(=O)NC(CC)CN(C(=O)CNC(C)=O)C)cccc2c1OCC2 16929,c1(C(N2CC(CN(C(CN(C3CC3)CC)=O)C)C2)=O)cnn(CC)n1 16930,CC1(C)CCC(C)(C(=O)NC2CC(O)CN(C(=O)Cn3cnccc3=O)C2)CC1 16931,C1(NC(C(N2CCCC(NC)CC2)=O)=O)CCC(F)(F)CC1F 16932,C1(OC)CCCC(C(=O)NCC2CC2NC(=O)C(C)=C2CCC2)C1 16933,N1(C(c2c(CCC)nco2)=O)CCCC(CN(C(=O)CC(C)C2CC2)CC)C1 16934,C1(NC(C2CCCC(C)(C)CC2)=O)CCC2(CCN(C(=O)C3=CCCS3)CC2)C1 16935,C1(OC)CN2CCCC2(C(=O)NCC(C(C)C)NC(=O)Cc2nc(C)sc2C)C1 16936,C12(C(=O)NC(CC)CNC(C3CC(C)(C)C3)=O)CC1COC2(C)C 16937,C1(CNC(=O)CCn2cccn2)CC2CCCCC2N1C(=O)Cc1ccccc1 16938,C1(F)(C(=O)NCC=CCNC(C2CN(CC)C(=O)C2)=O)CC2(CCC2)C1 16939,C1(CNC(CSC)=O)CCC2(CCC2)C1NC(=O)CCc1ccc(C)cn1 16940,c1(C(=O)NC2CC(CNC(c3c(COC)noc3)=O)C2)ccc(C(N)=O)c(Cl)c1 16941,c1(OC)cccc(C2=NOC(C(=O)NC3CCCC(C4CC4)C3)C2)c1 16942,c1(NC(CCN(C(CCCOCC=C)=O)C)C(C)C)ncc(C)c(S(C)(=O)=O)n1 16943,C(=O)(NNc1cc(Br)ccc1Cl)C1CC(n2cc(C3CCN(C)C3)nn2)C1 16944,C1(COC)(CNC(=O)CSC2CC2)CCCN1C(N1CCC(C)C1)=O 16945,CC1(CO)CCN(C(C2(NC(C3(C)CC=CCC3)=O)CSC2)=O)C1 16946,CC(O)CC(C)(C)CNC(c1ccccc1)c1csc(-c2cnn(C)c2)n1 16947,CC(C(=O)NCC1CCC(NC(C2C=CC=CC=C2)=O)CC1)C(F)F 16948,N1(C(C(C(C)C)SC)=O)CC2CCCC(NC(c3cn(CCCF)nn3)=O)(C2)C1 16949,C(=O)(CC=C(Cl)Cl)N(C1CCN(C(=O)COCC=Cc2ccccc2)C1)C 16950,c1(C(=O)NCC#CCNC(C2C(C)(C)COCC2)=O)c(N)cc(F)cc1Cl 16951,C12(NC(c3cnccn3)=O)CCOCC1CN(C(c1ccc(Cl)c(Cl)c1O)=O)C2 16952,N1(C(COCCC)=O)CCN(C(C2CC3C=CC2O3)=O)C(CCO)C1 16953,N1(C(c2cnc(C)[nH]2)=O)CCC2(NC(c3nccc(Cl)c3F)=O)CCCCCC12 16954,Cc1ccc(C(C)N(C2CCCN(C(c3cccc(C4CCC4)c3)=O)C2)C)cc1 16955,C1(CNC(=O)CCc2cncnc2)CC(F)CN1C(C1OCCCO1)=O 16956,c1(NC(C(=O)NC2C3CC(N)CC2C3)=O)ccc2c(c1)CCC(=O)N2CC(F)F 16957,c1(CC)onc(C)c1CNC(=O)CCN(CCO)C(C12CCCCC1C2)=O 16958,C1(OC(C)(C)C)CC(NC(c2sc(Br)cc2I)=O)C1(C)C 16959,N1(C(c2sc(C)c(O)n2)=O)CCCC(C2CCN(C(C3(Cl)CC3)=O)CC2)C1 16960,C(CC)(C(=O)NC1COCC1n1cc(NC(=O)OC(C)(C)C)nn1)=CC 16961,c1(SCC)ccc(NC(=O)CN(CCCOC)CCCO)cc1 16962,C(=O)(C1=NN2CCCN=C2N1)N1CCN(C(C=CC)=O)CC1CC(F)(F)F 16963,c1(C(=O)NCCCNC(CC2(OC)CC2)=O)cc(=O)n(-c2ccccc2)[nH]1 16964,c1(COC(C2(CCCC)CCC2)=O)ccccc1SC.C1(NC(C)=O)CCN(C)C1=O 16965,C(=O)(C(F)CCC(C)C)NC(C(C(=O)NCC1CC(CC)C1)(C)C)C 16966,C1(NC(C(C)CSC(F)(F)F)=O)CCCN(C(c2ccnc(Cl)c2)=O)C1C 16967,c1(OCC)cc(CN2CCCC(C)(C(F)F)C2)ccc1OC 16968,c1(C(=O)NC2C(CNC(C(N3CCC(C)CC3)=O)=O)CC2)cccc(F)c1Cl 16969,O=C(CC(C(F)F)n1ccnc1)NCCCNC(=O)C=Cc1nc[nH]n1 16970,c1(CCC)cc(C(=O)NC(C)(C)CNC(=O)C=C(C)C(C)C)ccc1Cl 16971,c1(C(=O)NCC2C(NC(c3c(CC)nccc3)=O)C2)cc2nc[nH]c2cn1 16972,c1(C(=O)NC2CCN(C(C(COC)C)=O)CC2F)nc2ccccn2c1F 16973,CS(=O)(=O)c1ccc(Cl)c(C(N2CC3CN(C(c4ccnc(Cl)c4)=O)CC23)=O)c1 16974,C1(NC(CCN2CCC(C(N)=O)CC2)=O)CCC2CN(C(C3CCC3)=O)CC2C1 16975,C1(C)(C(N(C2(C(=O)NCC(C(C)O)O)CCC2)C2CC2)=O)CCN(C)CC1 16976,C(=O)(C1CCCc2nc[nH]c21)N(C(CNC(C1CC2CCC(C1)O2)=O)C1CC1)C 16977,C1(C(=O)NCC2COCCN2C(c2cnn(C3CC3)c2)=O)Cc2ccccc2O1 16978,Cc1c(C(=O)N(C2CCN(C(C34CC(C(C)C)(CO3)C4)=O)C2)C)cccc1Cl 16979,N1(C(c2nn(CC)c(O)c2)=O)CC2CCC(NC(=O)CC3CCCC3)CC2C1 16980,c1(C(=O)NC(CC)CN(C(=O)COCC(C)C)C)cc(C)nn1C1CC1 16981,c1(C(=O)NC2C(NC(C3(C#C)CC3)=O)CCC2)c(C)cc[nH]c1=N 16982,c1(C(N2CCC(C(CNC(C(C)SC)=O)C)CC2)=O)ncc(Cl)cc1F 16983,C1(CCC=C)(C(=O)NCCCC2CCOC2=O)CN(C(c2csc(O)n2)=O)C1 16984,c1(C(=O)NC2C(N(C(CC(C)C3CC3)=O)C)CCCC2)ncc2cc(Cl)ccn12 16985,N#Cc1ccccc1Oc1ccc(CNC(=O)CC2CC(F)CN2)cc1 16986,C(=O)(C#CC(C)(C)CNC(=O)Cc1cn(C)cn1)NC(C(=O)OC)CCF 16987,c1(C(N2CC(NC(C3CC(OC)C3)=O)C2)=O)cnoc1C1CC1 16988,C(=O)(C(C)(C)C(C)NC(=O)NCCNC(C(C1CC1)OC)C)OC(C)(C)C 16989,c1(C(=O)NCCNC(N2CCCC2c2ccncc2)=O)ccccc1Cl 16990,N1(Cc2cc(CC)cc(C)c2)CCn2cccc2C12CCNC2 16991,C(N=c1[nH]c(-c2ccccn2)ccc1OC)C1(c2c(OC)cccc2)CCCC1 16992,C1(CN(C)C(c2csc(O)n2)=O)COCCN1C(c1cc(C2CCCC2)[nH]n1)=O 16993,N1(CC)C(=O)CCC1C(=O)NCCC1(NC(c2ccn(CCOC)n2)=O)CCC1 16994,C1(NC(=O)Cc2ccc(Cl)cc2Cl)CC2CC(C1)N(C(=O)C(O)C1CC1)C2 16995,c1(C(=O)NCC2N(C(CNC=O)=O)C3CCC2C3)cc2c(F)cc(Cl)cc2[nH]1 16996,C1(C(CO)NC(C(CC)OCC)=O)CCN(C(C2CCC(O)C2)=O)CC1 16997,c1(C(N2C(C(=O)Nc3cc(Cl)cnc3Cl)CC(C)C2)=O)ccc(F)c([N+](=O)[O-])c1 16998,C#CCCCCCC(=O)NCCCCC(C)(C)NC(C1CC2CC(=O)C1C2)=O 16999,c1(NC)ccc(F)cc1C(N1CCCCC1CCNC(c1cnc[nH]c1=N)=O)=O 17000,c1(NC(=O)Nc2cccc(NCCOC)c2)ccc(-c2ccccc2)c(F)c1 17001,N1(C(c2c(C)[nH]nc2CO)=O)CC2(C1)CN(C(C1COCCN1C=O)=O)C2 17002,C(=O)(CCC1=NNC(=O)CC1)N1CCN(C(C(C)n2cccn2)=O)CC1C(F)F 17003,C1(CC(=O)NCCN(C(C)C)C(c2n[nH]cc2Cl)=O)CCC2(CCOCC2)CO1 17004,c1(OCC(=O)N(CC(O)CNC(C23CCCC2C3)=O)CC)ccc(C(C)O)cc1 17005,C1(C(=O)NC2CC3CNCC23)CC2(CCCCC2)CN1 17006,c1(NCC2(NC(C3CCNC3=O)=O)C(C)CCCC2)ncc2c(n1)CCOC2 17007,c1(C(=O)NCC2CC(C)N(C(=O)CC3CCCCC3)C2)sc2nccnc2c1N 17008,CC(C)(C)C(C)(C)C(=O)N1CCOC(CC(N2Cc3c[nH]nc3C2)=O)C1 17009,N1(C(C2CC(SC)C2)=O)CC(C)CCC1CNC(c1[nH]cnc1C)=O 17010,C1(NC(c2ccc(C)c(C(F)(F)F)c2)=O)CC2CCC(C1)N2C(C1CC1(C)C)=O 17011,C(CC1CCC1)(C(=O)NC1CCCC1NC(=O)C(C)Cc1ccncc1)OC 17012,c1(C(=O)NC2CC(C)N(C(=O)CC#N)C2)cc2c(Br)cccc2c(=O)o1 17013,c1(NC(C(C)(C2CCC2)NC(=O)C(C2CCOCC2)F)=O)ccc(F)cc1 17014,C1(NC(=O)C=CC2CC2)CCC1C(=O)NCCc1cnc[nH]1 17015,c1(OCCC(=O)NCC2COCCN2C(c2cccc(F)n2)=O)cccc(F)c1 17016,Cc1ccc(S(=O)(=O)N(C2CCNCC23CC3)Cc2ccsc2)cc1[N+](=O)[O-] 17017,c12ccc(cn1)c(=O)[nH]2.C(C(=O)NCCOC(C)(C)C)OCCOCC 17018,C1(CNC(c2ccc(F)cn2)=O)CCCC2(CN(C(=O)CCC(F)(F)F)C2)O1 17019,C1(C(=O)NC(C2CN(C(CC3CC(C)C3)=O)C2)C)NC(=O)OC1C 17020,C(=O)(CC(C)CC(C)C)NCC(=O)NCC(=O)NC(CCCCC)C 17021,C(=O)(C(CCC1CCC1)NC(=O)NCc1cnsc1)NC 17022,Cc1ncccc1CC(N1CCC(NC(=O)CN(CC(C)(C)C)C)CC1)=O 17023,c1(C(C(=O)NCC(CNC(C2CCC(C)C2)=O)O)(F)F)ccc(F)cc1 17024,C1(C)(NC(COC(CNC(CC2CC(=C)C2)=O)(C)C)=O)CCOCC1 17025,C12(CNC(c3cn(C)nn3)=O)CCC(CN(C(C34CCC(CC3)CC4)=O)C1)C2 17026,C12(CNC(=O)Cn3cnc(C(N)=O)n3)CC1CN(C(C1(C3CC3)CCCO1)=O)C2 17027,Cc1coc(C2CN(C(=O)Nn3cc(C(=O)OC(C)(C)C)nn3)C2)c1C(C)(C)C 17028,c1(C(N2CCC(NC(CS(C)(=O)=O)=O)CC2)=O)c(Cl)ccc(F)c1F 17029,C1(SC)CC(C(=O)NCCN(C(=O)Cc2ccsc2)C(C)C)C1 17030,c1(C(=O)NCC2N(C(C3COC(=O)O3)=O)CCC2)cn(C(F)F)nc1C(F)F 17031,C1(NC(COCCN(C)C)=O)CCCC12CCN(C(c1ccc([N+](=O)[O-])o1)=O)C2 17032,C1(CN(CC(=O)NC(c2ccccc2)CC)C)(OC)CCOCC1 17033,C1(NC(C(C)(C)C)=O)CN(C(C2CN(CC(F)(F)F)C2)=O)CCC12CCOCC2 17034,CC(C)C(N=[N+]=[N-])C(=O)N1C(C(=O)NCCOCCC2CC2)CCC1C1CC1 17035,C(=O)(C#CC1(C)COC1)N1C(C2(C(N3C(C)C(=O)NCC3)=O)CC2)CCC1 17036,c1(C(=O)NC(C(C)C)C(=O)NCC2CC(C)(C)CCO2)cncc(C#N)c1 17037,C1(CCNC(COC)=O)CN(C(c2cc(C(F)F)n(C)n2)=O)CC1C 17038,CCCC(O)CC(=O)NC(C)(C)CNC(=O)CCc1ccc(C(C)C)cc1 17039,Cc1nc(=N)[nH]cc1C(N1CCOCC(CNC(=O)Cc2ccc(F)cc2)C1)=O 17040,C#CCC(C)(C(=O)Nc1ccc(CO)c(F)c1)NC(=O)C(CC1CC1)SC 17041,N1(C(=O)C=Cc2ccsc2)CC2CN(c3ncncc3F)CC2C1 17042,c1(OC)cccc(C)c1NC(=O)CCCCCNC(C1NC(=O)OC1C)=O 17043,N1(C(Cc2ccn(CC)n2)=O)CCN(C(c2cc(C)ccc2O)=O)C2CCC12 17044,N1(C(c2c(C)ocn2)=O)CCC2(CC1)COC(CNC(C1(C(N)=O)CCC1)=O)C2 17045,c1(C(=O)NC(C(C)NC(=O)Cn2cnnn2)C)cncc(Br)c1 17046,CC1N(C(C2CCCN(C(c3n[nH]c(C(F)(F)F)n3)=O)CC2)=O)CCC1(C)C 17047,N1(C(=O)CN2CCOCC2)CCN(C(c2ccncc2Cl)=O)C2CC12 17048,C1(CNC(c2c(CC)cc[nH]2)=O)CN(C(=O)CC2CC2)CCC1C 17049,N1(C(c2cccc(CC)c2)=O)CC(C)CCC1C(N1CCCC(CCO)CC1)=O 17050,C(=O)(CCC(=O)NC(C)(C)CC(=O)NC(c1csnn1)C)NCC 17051,C12(C(N3C(CNC(C4CC5CCC4C5)=O)CCC3)=O)CC3CC(CC(C3)C1)C2 17052,N1(C(C)=O)CCC2OC(=O)OC2C1.C12(CN(CC)C1)n1cc(nn1)COC2=O 17053,c1(C(N(C2CCN(C(c3n[nH]c(C)c3C)=O)C2)CC)=O)cncc2ccccc12 17054,c1(OC)cc(C(=O)NCC2CC2NC(C2(C)CC=CC2)=O)on1 17055,C1(CC)CCN(C(C23CCC(NC(C4CCCC4O)=O)(CC2)C3)=O)CCO1 17056,N1(C(c2c(CC)con2)=O)CCC(NC(C2(Br)CC23CCC3)=O)CC1C 17057,c1(OCC)cc(C)c(NC(C2CC(O)CN2c2ncncc2I)=O)cc1Br 17058,c1(C(N2CC(O)(CC)C2)=O)nc2nc(C(=O)O)ccn2n1 17059,C(=O)(C(C)(C)C(=O)NCC1(F)CCCN(C(=O)CC2CC(C)(C)CCO2)C1)NC 17060,c1(C(=O)NCCCC2N(C(C(F)=CCC)=O)CCC2)nn(C)c2c1CCC2 17061,C1(C(=O)NCCC(O)CNC(c2cnccc2C)=O)(COC)CCCCC1 17062,N1(C(c2cc(CCC)oc2C)=O)CCN(C)CC1CNC(=O)CCC(C)O 17063,C(c1ccc(Cl)c(Cl)c1)=CC(N1CC2C(NC(=O)CC3CCCC3(F)F)(C2)C1)=O 17064,C1(C(=O)NC2(C(=O)NCCCc3cc(C)no3)CC(F)C2)CC(C)CCO1 17065,C=CC(C)CC(=O)NCCn1cc(CNC(c2cncs2)=O)nn1 17066,C1(C(=O)NC2CC(CCNC(c3cccc(C(F)F)c3)=O)C2)CC2CCCC2C1 17067,c1(CNC(c2cccc(Cl)c2)CO)cc(Cl)cc2c1CCC2 17068,N1(C(C(CC=C)C)=O)CCN(C(C2(C(C)(C)C)CCC2)=O)CC1C 17069,N1(CC(F)F)CC(N=c2nc3scnc3c(NCc3ccc(Cl)s3)[nH]2)C1 17070,CC(O)C(C(=O)NCCCC(C)NC(=O)COC(C)(C)C)NC(=O)OCC(N)=O 17071,CC(C(=O)NC(C)(C)C(C)NC(c1sccc1Br)=O)C(=O)N1CCOCC1 17072,c1(C(=O)NCC(C)C(=O)NC2CC2)cc(=O)n(C)cn1 17073,c1(C(N2CC3(CCN(C(C(C(=C)C)(C)O)=O)C3)C2)=O)cc([N+](=O)[O-])c(C)cc1C 17074,C1(CC)CCCC(C(=O)OC)C1.N12CCC1C(=O)N1CC(C1)C2=O 17075,C(=O)(C(C(C)(C)C)[N+]1([O-])CCCC1=O)NC1C(NC(CS(=O)(=O)NC)=O)CC1 17076,C(=O)(C(C)CC(C)(C)C)NC1CC(CNC(C2C(C)OCC2)=O)C1 17077,N1(C(C(CC)CC)=O)CCN(C(=O)CSc2ccncc2)C(CO)C1 17078,C1(N(CCC(=C)C)C(C)C)CCCSC1 17079,C(=O)(C(O)CC(F)F)NCC(CN(C(CCCc1scc(C)n1)=O)C)C 17080,N1(C(C(CCC)F)=O)CCN(C(c2cc(Cl)cn2C)=O)C(C(C)(C)C)C1 17081,c1(C(N2CC(C)(NC(=O)CN3CCOCC3)C2)=O)ccnc(C(C)(C)O)c1 17082,C1(NC(C2C(=C)C2)=O)CC2(C1)CC(NC(=O)C(C)Sc1ccccc1)C2 17083,c1(N2C(C)CC(CNC(C3(C)C(CC)CCC3)=O)C2)ccc(C#N)nn1 17084,c1(C(=O)NCCC(CCNC(C2CC(=C)C2)=O)C)cc(Br)ccc1OC(C)C 17085,N1(C(c2cc(C(C)=O)c(C)o2)=O)CCN(C(c2cscc2C)=O)CC1C1CCC1 17086,c1(-c2cn(CC3N(C(c4ccc(N(F)F)nc4)=O)CC3)nn2)c(F)cccc1Cl 17087,c1(C(=O)Nc2n(C)nc(-c3ccc(Cl)cc3)n2)cc(Cl)ccc1Cl 17088,C#CCC(O)C(=O)N(C)CC1CN(C(=O)CC2CCCCC2)CCO1 17089,Cn1nc2c(c1C(N1CCC(NC(C3CCCOCC3)=O)C(F)C1)=O)COCC2 17090,C1(NC(c2c(OC)cc(C)cn2)=O)CCC2(CCN(C(=O)CC3(SC)CC3)C2)C1 17091,S(=O)(=O)(c1cnc(NC2CC3CC(CO)CC23)c(Cl)c1)NCCCCC 17092,C1(C(=O)NCC(C)NC(=O)C(C)(C)n2cc(Cl)cn2)(OC)CCCCC1 17093,N1(C(c2c(C)nc[nH]2)=O)CCN(C(c2ccc(Cl)nc2F)=O)C(C#N)C1 17094,C(=O)(N=c1cc(Cl)nc(C)[nH]1)C1N(C(c2noc(CC)c2C)=O)CCSC1 17095,N1(C(c2c(O)nc(CC)c(C)c2)=O)CCC2(CCCN(CCC3CCOC3)C2)C1 17096,C1(C(=O)N(CC(C)C#N)CC)(NC(COCCCC#C)=O)CCCC1 17097,c1(N2CC(CC)OCC2)ncc2c(ccn2Cn2nnnc2OC)n1 17098,N1(C(C(C)=CC2CC2)=O)CC(CNC(=O)C(F)OC(F)(F)F)C2(CC2)C1 17099,C1(NC(C2CCC2)=O)CC2CC1CN(C(c1cccn3nccc13)=O)C2 17100,Cc1nc(NC2CCCN(C(=O)Cn3nnnc3C(C)C)C2)cc(Cl)n1 17101,c1(C(=O)NCC(C(C)C)NC(c2c(CC)c[nH]c2)=O)ccc2c(c1)COC2 17102,c1(C(C(=O)NC(CC2CN(C(c3cc(C)c(C)s3)=O)C2)C)C)ccc(F)cc1F 17103,C(=O)(C1=C(Cl)CCC1)NC1C(NC(c2ccn(C(CC)CC)n2)=O)CC1 17104,CC(C)C(CCc1ccccc1)C(=O)N1CC2(CCCC2NC(=O)C=CCO)C1 17105,c1(N(Cc2nc(CC)sc2)CC2CC2)ncnc2ncn(C3CC3)c12 17106,C(=O)(CC(F)(F)F)NC(C(=O)Nc1c(OC)c[nH]n1)C.C12CCC1C(=O)N2 17107,CC1=C(C(=O)N2CCC(F)C(NC(c3cnc(C)[nH]c3=N)=O)C2)S(=O)(=O)CCO1 17108,N1(C(C2C(CC)CCC2)=O)CCN(C(C)CNC(=O)Cn2cccn2)CC1 17109,C1(CC)CCN(C(C2CC(=O)N(C)C2)=O)C(C(=O)NCc2ccc(OC)cn2)C1 17110,Cc1cc(F)ccc1C(F)(F)C(=O)OC(C)Cc1cn(C)nc1C(F)(F)F 17111,C=CCC(CC(=O)NC(c1nc[nH]n1)(C)C)NC(C1CC2CC2C1)=O 17112,N1(C(CCCSC)=O)CCN(C(=O)Cc2ccc(C3CCC3)cc2)C(CCO)C1 17113,Cn1cnc(C=CC(=O)NCC2CC(=O)N(c3ccccc3)C2)c1 17114,N1(C(c2ccc(C)c(C#N)c2)=O)CC2(CCN(C(c3ccc(Cl)nc3)=O)CC2)C1 17115,Cc1ccc(CC(=O)NC2CCC(CNC(=O)C(C)Sc3csc(C)n3)C2)cc1 17116,c1(C(=O)NCCN(C(C2(CC)CCNC2=O)=O)C2CC2)nccc2ccn(C)c12 17117,N1(C(c2scc(CC)c2)C(=O)NCC2CCCO2)CCN(C)C(=O)C1C 17118,C#CCC(C)C(=O)NC(CN(C(=O)COc1ccsn1)C)CC 17119,c1(C(=O)NCC2CCCN(C(=O)NCC3C4COCC34)C2)ncc(F)cc1F 17120,C1(CNC(C(C2CCOCC2)C)=O)CCN(C(C2CC3(CCC3)C2)=O)CC1O 17121,C(=O)(CC(CN(C)C)CC(C)C)NC(C1(O)CN(c2cc(OCC)ncn2)C1)C 17122,C1(NC(=O)CCCCCn2cc(C3CCOC3)nn2)CCNCC12CCC2 17123,C1(CNC(C(C)(C)SC)=O)C2CCC1CN(C(c1ccnc(C)c1)=O)C2 17124,C1(C(C)C)CN(C(=O)CC2CCCCC2)CCN1C(C1CCCC(C)(C)O1)=O 17125,c1(C(N2CCCC(NC(C3C(C)C3)=O)C2)=O)cc(S(N)(=O)=O)cc(Cl)c1Cl 17126,C1(C(N2CCC(OC3CC3)C2)=O)COCCN(C(C2(O)CCCCCC2)=O)C1 17127,N1(C(C(C)CN(C)C(C2(CO)CCCC2)=O)=O)CCC(N=[N+]=[N-])C1 17128,C(=O)(CCNC1CCCC1)NCC1(C(N(CC#CC)CC#C)=O)CC1 17129,c1(CC(N2CCC(COC)(NC(=O)CCC(C)SC)C2)=O)ccc(C)c(F)c1F 17130,c1(C(N2CCC(C3N(C(c4[nH]c(=NC)sc4)=O)CCC3)C2)=O)ccc(F)cc1Cl 17131,CC(C)(C)CC(C(=O)NCc1cccnn1)NC(=O)CCCC#N 17132,CCCC(C(=O)NC)NC(=O)C(CNC(c1ncsc1C)=O)N(C)C 17133,Cc1oc2ccccc2c1C(N1CCCC(C(C)NC(C2SCCS2)=O)C1)=O 17134,N1(C(C(C)=C2CCCC2)=O)CCC(C)(C)C1C(=O)N(CCCCCO)C 17135,c1(OC)ccc(NC(=O)CC2CN(C(c3ccc(C)[nH]3)=O)CCC2C)c(C)c1 17136,c1(NC(=O)CC2(NC(=O)C(F)CC3CCCC3)CC2)ccc(F)c(CO)c1 17137,C(c1cccc(F)c1F)=CC(=O)N(C(C)CN(C)C(C1COCC(C)(C)O1)=O)C 17138,c1(C(CC)(C)NC(c2cn(C3CCOC3)nn2)=O)ccc(Cl)cc1 17139,N1(c2nc(CC(CCOC)(C)C)on2)CCS(=O)(=O)C2COCCC12 17140,C1(CC(=O)NCC2CN(C(c3nc(COC)sc3)=O)C2)CCCCC1C 17141,c1(COCC(=O)NCC2C=CCN2C(=O)CCC2CCCO2)ccccc1Cl 17142,c1(C(C)(C)NC(=O)NCC23CC(CO2)C3)ccc(O)cc1F 17143,CCCCCCCCCC(=O)N1CCC(O)(CNC(c2csc3nccn23)=O)C1 17144,c1(NCCc2c(C)ncs2)cc(N(C)Cc2cccc(F)c2)ncn1 17145,c1(OC)cccc(CC(N)C(=O)N2CCC2(C)c2ccccc2)c1 17146,N1(C(CN(C(COC)=O)C)=O)CC=C(CC(=O)NC(C)C(C)(C)C)CC1 17147,C1(CNC(C2CN(C)C(=O)C2)=O)CN(C(c2cnn(C3CC3)c2)=O)CCCO1 17148,c1(C(=O)NC2C(CNC(=O)CCc3ncccn3)C2)ccc2occc2c1 17149,N1(C(C(C)CC(F)(F)F)=O)CC(CNC(=O)CS(C)(=O)=O)CC12CCOCC2 17150,CC1(C)CC(NC(C2CCC(OC(F)(F)F)C2)=O)CN1C(C1(O)CCC1)=O 17151,C1(C(N(C2CCN(C(=O)CCC(C)NC(N)=O)C2)CC#C)=O)CCC=CCCC1 17152,C=C(C)CCCC(=O)NCCC(O)C(=O)N(CCCN(C)C)CCC 17153,Cc1ccc(C(F)(F)C(=O)N(CC(C)CNC(=O)CN(C2CCCC2)C)C)cc1 17154,c1(OC)ccc(C=CC(=O)NCC2COCCN2CC)cc1OC 17155,CC(CCS(=O)(=O)c1ccc(Cl)c(Cl)c1)NC(=O)N(C)C(c1ccccn1)C 17156,CC1CN(C(c2csc3nccn23)=O)CC1(C)CNC(C1CC1C#N)=O 17157,Cc1cc(C(=O)NCC(C)N(C)C(C2CCN(C)C2=O)=O)cnc1C(F)F 17158,Cc1nn(C)c(OCC2CC2c2ccc(C(=O)N(C)C)cc2)c1OCC1CC1 17159,C#Cc1ccc(C(=O)N(C(CNC(c2cnn(C(C)C)n2)=O)CC)C)c(C)c1 17160,C1(CNC(C(=CC2CCCC2)C)=O)CCN(C(=O)CCS(C)=O)CC1C1CC1 17161,CC1CCN(C(C2CCCC(O)C2)=O)C1CNC(=O)CC(O)c1ccccc1 17162,C1(CNC(CS(CC)=O)=O)CCC2(CN(C(=O)Cc3ncc(C)o3)C2)O1 17163,C1(CNC(c2cn(C)nc2)=O)CCc2cc(N)ccc2O1 17164,Cc1sc(C(=O)NC2CC(CNC(C3CC4CCC4C3)=O)C2)cc1[N+](=O)[O-] 17165,C1(NC(CC(C)(C)N(C(CCCC=C)=O)C)=O)CCOC12CCOC2 17166,c1(SCCNCCC)cc(O)nc(C)n1 17167,C1(C(=O)OC)COCC2(CCN(C3CN(S(C)(=O)=O)CCC34CCC4)C2)O1 17168,c1(C(=O)NC(C)(C)CCNC(c2cc(C3CC3)ccn2)=O)cc(Cl)cnc1O 17169,c1(OC)cccc(Cl)c1C(N1CC(NC(C2CC23CCC3)=O)CC(F)C1)=O 17170,c1(OC)nc(N2CCC(F)(C(=O)Nc3cccc(-c4nnco4)c3)C2)ncc1Br 17171,C1(NC(C2(SCC)CC2)=O)CN(C(=O)C(C)(C)Nc2ccccc2)CCC1CO 17172,CCC(C(=O)NCCC1(O)CCCN(C(C2CC(F)(CO)C2)=O)C1)C(C)(F)F 17173,CC1CC(NC(c2cc(CO)on2)=O)CN1C(c1cnc(-c2ccccc2)s1)=O 17174,CC(C)(C)C(CNC(=O)CC(=O)C(C)(C)C)C(=O)NCC(C)(O)CO 17175,C1(NC(c2n(CC)nnc2)=O)CN(C(=O)C(c2cccnc2)C)CC2(CC2)C1 17176,N1(C(c2oc(CC)c(C)c2)=O)CCCC(C)C1CNC(=O)C=Cc1ccncn1 17177,C(c1c(C)noc1C)=CC(N1C(C)CCC1)=O.CC(c1cccs1)=CC(=O)NC 17178,c1(OCC)cc(N2CCC(N(C)C(C3CCCC4CC34)=O)CC2)ccc1[N+](=O)[O-] 17179,CCCCCC(O)CC(=O)N1CCN(C)C(CNC(=O)Cc2ncccc2C)C1 17180,CC(C)CC(C(=O)N(CC(C)C(=O)Nc1csc(Cl)c1)C)N(C)C 17181,c1(C(N2CC(NC(C(C)=C(C)C)=O)C3(C2)CC3)=O)nc2cccnn2c1Br 17182,N1(CC(=O)NCCN(CC=C)C)CCN(C(=O)C(COC)COC)CC1 17183,c1(C(=O)NCC(CCNC(C2CCCC(O)C2)=O)OC)c(C)ccc(N)c1C 17184,C1(CNC(C(COC)OC)=O)CN(C(c2cc(OC)ccn2)=O)CC1(C)C 17185,C1(NC(c2ccc(Cl)s2)=O)CN(C(C2CC(C3CC3)=NO2)=O)C2CCCC12 17186,C1(F)(CNC(=O)COC2CCCC2)CC(NC(c2occc2C2CC2)=O)C1 17187,C(=O)(CC(CC)CC)NC(CSCC)C(=O)NCc1cnnn1C 17188,CCC(CC)CC(F)C(=O)NC1(C(N2CCCN(C)CC2)=O)CC1 17189,c1(C(N2C(C(N(C)CCC3CCCC3)=O)C=CC2)=O)ccncc1F 17190,C1(C(N2CC(CC(C)(C)CNC(C3CCSC3)=O)C2)=O)CC(F)C(=O)N1 17191,N1(CC(C)(C)NC(=O)NC(c2sccc2C)CC)CCC(NC(C)=O)CC1 17192,c1(OCC(N2C(C)CSCC2)=O)c(Cl)cc(Cl)cc1Cl 17193,C#CCCCCCCC(=O)NCc1ccc(C(=O)NC2(C3CC3)CCOC2)n1C 17194,N1(C(C(C)OCC2CC2)=O)CC2CCCC(NC(=O)C=C(Cl)Cl)(C2)C1 17195,c1(C(=O)NCC(CC=C)NC(=O)CCC(N)=O)cccc2occc12 17196,c1(C(N2CC3N(C(CCC(C)C)=O)C(CC3)C2)=O)cccc2c1OCC2C 17197,C(C(C)(C)CCNC(c1ccnc(O)c1)=O)NC(c1cn(CC=C)nc1)=O 17198,C(=O)(C(F)(F)C(F)(F)C(F)F)N1CCC(NC(C2OCC(C)(C)C2)=O)(CF)C1 17199,C(c1cn(CC(=O)Nc2ccccc2)cn1)=CC(=O)OC(C)C(=O)N(C)C 17200,S(=O)(=O)(c1cccnc1N1CC2(CC(C)CO2)C1)NCC(c1ccsc1)OC 17201,C1(C(N2CC(C)CS(=O)(=O)C2)=O)=CC=CC=CC=C2N(C=C1)C2=O 17202,N1(C(CSC)=O)CC2CCCC(CNC(C3CC34CCCCC4)=O)C2C1 17203,CN1CCN(C(c2cc(CF)on2)=O)C(CNC(c2cnn(CC(F)F)c2)=O)C1 17204,c1(NC(C2C3CN(C(CCCOC)=O)CC32)=O)ccc2ncnn2c1 17205,c1(CC(=O)NCC(C)(O)CNC(=O)CC2CCC2)ccccc1O 17206,c1(C(C(=O)NC(C)C)N(C)Cc2nc(CO)n[nH]2)cc(C#N)cs1 17207,N1(c2cc(C)nc(CO)n2)CCC(C2CC2)C1CNC(=O)CCc1nccn1C 17208,c1(OC)ccccc1C(O)C(=O)NC1CCC1NC(=O)Cc1ccc(Cl)cn1 17209,C12(C(=O)NCC(CNC(C=CCN(CC)CC)=O)O)CC=CCN1CCC2 17210,c1(C(N(C(CNC(CC2ON=C(C)C2)=O)C)C)=O)cc2ccoc2cc1F 17211,N1(C(C2(COC)CCCO2)=O)CCCC(NC(=O)CCNC(=O)OC)C1 17212,N1(C(c2c(SC)cnn2C)=O)CC2=C(C1)CN(C(=O)C1=CCCCO1)C2 17213,C(C)(C)(CC(=O)NCc1ncccc1C(N1CCCC1)=O)OC 17214,c1(C(=O)NC(C)CN(C(=O)C=CSc2nc[nH]n2)C)cccc2nc(CO)[nH]c12 17215,n1(C(C)(C)C)cnc(C(=O)NCC2(O)CC(CNC(=O)C(Cl)=CCl)C2)n1 17216,C(=O)(CCCC(F)(F)CO)N(C)CC1(NC(C(CCCC)N(C)C)=O)CC1 17217,C1(NC(c2c(OC)scc2)=O)CCN(C(=O)CCn2cc(Cl)cn2)CC1O 17218,S(=O)(=O)(c1cccc(F)c1)N1CC(N(C(C(c2ccccc2)C)=O)C)C1 17219,N1(C(C)C)CCCC(CN(C)Cc2ccnc(OC(C)CC(=O)O)c2)C1 17220,n1(CCOC)ncc(C(=O)NCC(C)CNC(C2C3CCN2CC3)=O)c1C 17221,C1(COC)CN(C(=O)CC2(C)CC(F)(F)C2)CCN1C(C1CC(C)(C)CO1)=O 17222,S(=O)(=O)(c1ccc(F)c(F)c1)N1C2CCN(C(c3cc(Cl)ncn3)=O)C2CC1 17223,N1(C(=O)Cc2cnn(C(F)F)c2)CCC2C(CCCN2C(C2COCCO2)=O)C1 17224,c1(C(N2C(C(=O)NC(CC=C)C(=O)OCC)C(O)CC2)=O)cnc(F)c(C)c1 17225,c1(NC(C)=O)cccc(C(=O)NC2CCCN(C(=O)C(C)(C)C3CC3)C2)c1C 17226,C1(NC(C2(CC)CC2)=O)CCC(CNC(=O)COCC2CCCOC2)C1 17227,c12ccccc1S2.C1(CC)CC(NC(=O)NC(C)(CO)SC)C1 17228,Cn1nc(O)cc1C(N1CC(O)CC1CNC(c1ccoc1C(F)(F)F)=O)=O 17229,C(N=c1cc(NCCOc2cccc(Cl)c2)nc(C)[nH]1)c1ccc(OCC)cc1 17230,c1(CC(=O)NC(C2(O)CN(C(Cn3nc(C)oc3=O)=O)C2)C)c(Cl)cccc1Cl 17231,CC(C)CC(O)C(C)C(=O)N1C(C(=O)NCC(C)(O)CCO)CC2CC12 17232,N1(C(C(C(C)(C)C)=O)=O)CCC=C(C(=O)Nc2cnn3cccnc23)C1 17233,Cc1c(Cl)c(C(N2CCOCC(NC(=O)CCCC(F)F)C2)=O)nn1C 17234,C(C)(C)(CC(F)C(=O)N1CC2CC2C2CC12)NC(C1C(C(=O)OC)C1)=O 17235,CCCC(C)(C)CC(=O)NC1COC2(C1)CN(C(c1ccn(C)c(=O)c1O)=O)C2 17236,N1(C(c2nc(C)c(C)[nH]2)=O)CCC(C2CCNC2)C1 17237,C1(NC(C(C)N(C(=O)C2=CCCC2)CC)=O)CCCC2(CCC2)C1 17238,N1(C(C2N(C(C)(C)C)CC2)=O)CC=CC(C(=O)NCC2CNC(=O)CO2)C1 17239,CC1CC(NC(=O)C(c2ccccn2)O)CN1C(c1cc(C(N)=O)cs1)=O 17240,c1(C2CN(C(c3cc(C(=O)OC)on3)=O)C2)ccc(-c2nn[nH]n2)cc1 17241,n1(CCCC)ncc(NC(=O)C=C2CCC2)c1CC1CCCS1 17242,C(=O)(Nn1c(C)nc2sccc2c1=O)c1cc(OC)c(OC)cc1[N+](=O)[O-] 17243,c1(N2CCCC(CCC)C2)nc(NCCc2nccnc2C)c2ncsc2n1 17244,Cc1ncccc1CC(=O)NC(C(=O)NC(C)CO)C1CCCO1 17245,N1(C(c2cnc(C)nc2)=O)CC2CCN(C(C3CCC(N(C)C)CC3)=O)CC2C1 17246,C(C(=O)NCC(C)(C)CCNC(c1ccc(C(C)(F)F)cc1)=O)(C(C)C)OC 17247,c1(OC)ccc(S(C)(=O)=O)cc1C(N1CCC(NCc2nc(Br)cs2)C1)=O 17248,CC(C(=O)NCC(=O)NCCCc1cn[nH]c1)N(C)C(C1CC1)C1CC1 17249,CCCC(C)(CC)C(=O)NC1CC2(C1)CN(C(=O)C(C(C)C)n1cnc(C)c1)C2 17250,c1(C(N2CC3C(C(=O)OC(C)(C)C)C3C2)C(=O)NC)ccc(C#N)cn1 17251,c1(C(C)C(=O)NCC2CC(F)(CNC(C3CC3F)=O)C2)ccc(F)cc1F 17252,CC(C)(O)C(C(=O)NCCCc1ccsc1)NC(=O)COCCCF 17253,N#Cc1cccc(NC(c2nnnn2CC(F)F)C2CC=CC2)c1 17254,c1(NC(C2C3CN(S(c4c(C)onc4)(=O)=O)CC32)=O)ccc2c(c1)C(=O)N(C)C2=O 17255,N1(CCOCC=C)CCN(C2CCN(C(C3CC34CC4)=O)C2)CC1 17256,N1(C(=O)COCCF)CC2CCN(C(c3cnc4c(c3)COC4)=O)C2C1 17257,c1(CC)ccc(F)c(C(N2CCC(NC(c3ccnc(Cl)c3N)=O)C(C)C2)=O)c1 17258,C1(COC)(NC(=O)C(O)C(C)C)CCN(C(=O)COC2CCOCC2)C1 17259,C(C)(C(C(=O)NCCCC1CC(C)C1)C(C)C)NC(C(C)=C(CC)C)=O 17260,C(=O)(C(C(CC)CC)OC)NC(CC=CC)C(=O)N(C)CCO 17261,c1(C(=O)NCC2N(C(C=CCC)=O)CCOC2)ccc(C)c2c1CCC2 17262,N=c1cc(C(N2CCN(CCC(N3CCNCC3)=O)CC2)=O)cc[nH]1 17263,Nc1cc(C(=O)NCC2(CNC(=O)C(C3CCOCC3)F)CCC2)ccc1Cl 17264,C1(C)(CC)CCC(C(=O)N(C)CCOCCCN(C(=O)CCc2cnoc2)C)O1 17265,c1(C(=O)NCC(CCCC)NC(c2cccs2)=O)n[nH]c2c1COCC2 17266,C(=O)(CCS(C)(=O)=O)NC(CCOC)C(=O)N1CCCC(O)C1 17267,c1(CC)nc(N2CC(NC(c3cc(=O)c(OC)c[nH]3)=O)C(C)(C)C2)cc(C#N)n1 17268,c1(C(=O)OCC(CC)F)cnc2sc(C)nc2c1 17269,C=CCCCC(c1nn[nH]n1)NC(C=CCC1(C(=O)OC)CCC1)=O 17270,N1(C(c2ccnn2CCF)C(=O)NC2CCC2)CCc2c(cccc2[N+](=O)[O-])C1 17271,c1(CC)[nH]nc(-c2nc(CCCO)nn2Cc2ccc(Cl)cc2)c1Br 17272,C(CC(F)F)(C(=O)NCCCc1cccs1)NC(C1OCCN(C)C1)=O 17273,C1(c2ncc(C(=O)OCC)s2)CCCN(C(c2nc(Cl)c(CC)[nH]2)=O)C1 17274,C#Cc1ccnc(C(N2CCC(N(C)C(c3cccc(N)c3F)=O)C2)=O)c1 17275,N1(C(C2(NC(=O)CC3CCCSC3)CC2)=O)CCc2cncnc2C1 17276,C(=O)(C(C)CCCC(C)C)N1C(C(=O)NC(CCC)C2CC2)(COC)C=CC1 17277,CN1CC(=O)N(CC(=O)NC2CC(CO)N(C(c3nccc(Cl)c3F)=O)C2)C1=O 17278,C(=O)(CC(CC(N)=O)CC(C)C)NC(CN(C(c1c(C)nco1)=O)C)(C)C 17279,C(=O)(CCCCCC(C)C)NC(CCCCNC(C(C)=CC)=O)C 17280,N1(C(C(=C(C)C2CC2)F)=O)CC(CNC(=O)CN2CCS(=O)CC2)C(C)(C)C1 17281,C(=O)(C1=C(c2ccccc2)SCCO1)NC1CN(C(CC(C)(C)C#N)=O)C2C1C2 17282,c1(C(N2CC(NC(COCC(=C)C)=O)C(N=[N+]=[N-])C2)=O)cn2cccc(C)c2n1 17283,CC1CC(C(=O)N2CCN(C(=O)CNC(c3cccnc3)=O)CC2CCO)=NO1 17284,c1(CNC(=O)NC2C(F)(F)C23CC3)ccc(F)c(N2CCCC(C(F)F)C2)c1 17285,N(C(=NCC(C(C)C)C(C)C)NC1CC1c1ccco1)C(CC)CC 17286,C1(O)(Cn2cc(C(CC)(C)C)nn2)CCN(C(=O)CCc2ccc(C)cc2)CC1 17287,Cc1ccc(C)c(C(=O)NCC2CC(NC(=O)C=Cc3cccs3)C23CCC3)n1 17288,c1(OCC)ccc(CNC(=O)C(C)NC2CCC(NC(=O)CCC(C)=O)C2)cc1 17289,C(=O)(C(C(C)C1CCCC1)N1CCC(C(=O)NS(C)(=O)=O)CC1)NC(CC)C 17290,Cc1nc(C2CC2)nc(C)c1C(=O)NC(C)CC(C)NC(C1CC1CN(C)C)=O 17291,CCCCCC(C)(CC)C(=O)NC1CCC(NC(=O)CCc2ccn(C)c2)CC1 17292,C12(C(N(CCCCN(C)C(C3CC(=O)CS3)=O)C)=O)CC3CC(CC1C3)C2 17293,C(C)(C)(CC(F)C(=O)Nc1ccc(Cl)c(O)c1)NC(c1cc(C)nnc1)=O 17294,Cn1c(O)nc2ccc(C(=O)NCCC3CCC(NC(=O)CNC=O)C3)cc12 17295,C=Cc1cnn(C)c1C(=O)NCC(CCCC)NC(c1scnc1CC)=O 17296,c1(CC)cnn2ccc(C(=O)NC(C)CCCNC(=O)CN(C)CC)nc12 17297,C1(CC=C)(NC(C2CC(C)(NC(=O)C=CCO)C2)=O)CCCC1 17298,C1(NC(c2c(CC)c[nH]n2)=O)C(C)CN(C(=O)C=CC(=O)NC2CC2)CC1C 17299,C(CCN(C)C(C1CC2(C1)CC(F)C2)=O)(C(C)(C)C)NC(CC(=O)OCC)=O 17300,c1(-c2cc(C)c(NC(c3cc(F)c(C)cc3F)=O)nc2)c[nH]c2ccccc12 17301,CC1=C(C)CC(CC(=O)NCC2CN(C(C3CN(C4CCCCC4)C3)=O)C2)CC1 17302,CC(C)(CCC(=O)N1CC2CC1CS2=O)NC(c1cc[nH]c(=N)n1)=O 17303,C1(=CC(=O)Nc2cnn(C)c2C(F)F)C2CC3CC(C2)CC1C3 17304,Cc1sc(=O)n(CCC(N2CC(N(C(=O)CCCCCF)C)C(F)C2)=O)c1C 17305,c1(C(=O)NCc2nnc(CC)s2)ccc(CNC(c2oc(C)cc2C)=O)nc1 17306,N1(C(C2CC(C)OC2)=O)CCC(NC(=O)CCc2ccn(C)n2)C12CCCC2 17307,c1(NC(N(CCOC)C2CC2)=O)nc2ccccc2n1-c1ccc(Cl)cc1 17308,CCC(CC)CC(F)C(=O)N1CCCC1C(C)(C)CNC(c1n[nH]cc1C)=O 17309,CC(C)C(C(=O)NC(C1CCCC1)CNC(=O)C(c1ccccc1)F)NC(N)=O 17310,c1(C(c2onc(C)n2)N(C)C)nc(-c2nc[nH]n2)nn1C(C1CCOCC1)C 17311,CCC(C)C(C(=O)NCC1(CNC(=O)C(C2CC(F)(F)C2)O)CC12CCC2)OC 17312,N1(C(CC2CC(C)(C)OC2)=O)CC2CCC(C1)N2C(c1cncc(O)c1Cl)=O 17313,C1(CNC(C(CC)(C)CO)=O)N(C(c2nc(C)ccc2F)=O)CCCC1(C)C 17314,CC(F)(F)C(C)(C)CC(=O)N1CCCCCC(S(C)(=O)=O)C1.c12nccc(n1)C2 17315,C=CCC(C)(C)CC(=O)NCC(=C1CN(C(=O)C(CCC)c2ccccc2)C1)F 17316,C1(C)(C(=O)NCc2cccc(NC(CCCCCOC)=O)c2)CC(C)OC(C)C1 17317,CC(C)C(C)CC(=O)N1CC=CCC1.C1(=O)CN1 17318,C(=O)(C(C#N)C(C)(C)C)N1CC(OCCC(=O)NCc2ccc(C)cc2F)C1 17319,C12(CCNC(C(CC)(F)F)=O)CCC1CN(C(c1cncc(C)n1)=O)C2 17320,C1(C2CC2)(CNC(=O)CCc2cnoc2)CCN(C(c2cccnn2)=O)C1 17321,c1(C(=O)NC2CC2)cn(CC(=O)N(CCN(C(CC2CC(OCC)C2)=O)C)C)nn1 17322,CC(C)(C)CCCC(=O)N1CCCC(CNC(C2COC(=O)C2)=O)C1 17323,CCC(COC)(CC)C(=O)Nc1ccc(NC(=O)C(C)COC)cc1C 17324,c1(C(C)NC(c2c(CNC(CCCOCC=C)=O)noc2)=O)cccnc1F 17325,C(=O)(C(CCOCCCN(C)C)NC(=O)CC1CC2(CC2)C1)N(CC)CC 17326,c1(C(=O)NCCN(C(CCC(=O)NC)=O)CCC2CC2)ccc(OC)nc1Cl 17327,C1(CNC(=O)CC2(O)CCOCC2)CCC2(CN(C(=O)C(O)C3CC3)C2)O1 17328,C1(CCCC)CCC(C(=O)NCC2CC(NC(c3cccc(CO)c3)=O)C2)CC1 17329,c1(SCC=C)cc(=NCCOC)[nH]c(N2CCCC2)n1 17330,c1(C(N(CCNC(=O)C(c2sccc2C)=O)CC)=O)ccc(F)c(F)c1F 17331,C(=O)(C1=NN(C)C(=O)CC1)NCC(CCOC)NC(c1c(C)cccc1Cl)=O 17332,c1(N(CC(CN(C)C(C2(F)CCCCC2)=O)O)C)nc2c(cc1C#N)CCOC2 17333,Cc1cc(C(N2CC(CNC(C3(CO)CCC3)=O)C(O)C2)=O)cc(Br)c1C 17334,n1(C(C)C)ncc(C(=O)NC(CNC(=O)Cn2cccn2)C(C)C)c1F 17335,C1(C(=O)NCC2(C3CC3)CCC2)(OC)CCN(C(=O)Cc2ccoc2C)C1 17336,C(=O)(C1=CC2CCC(C1)C2)N1CC2C(CN(c3ccccc3)C(C)C)(CC2)C1 17337,N1(C(C2CC(OC)CN2C(=O)CC2CCN(C)CC2)=O)CCC2(CNC(=O)O2)C1 17338,c1(C(=O)NCC(=C)CCNC(=O)CN(C)C)cnc(OC)cc1C 17339,C1(NC(C(C)OCCCCCC)=O)CCC(OC(=O)C2=NOCC2)CC1 17340,C12(C(=O)NCC3CC(O)(CNC(C(C)n4cccn4)=O)C3)C(=O)C3CC1C2C3 17341,c1(C(=O)NCCCC(CCC)NC(=O)CC(C)O)cc(S(=O)(=O)N(C)C)oc1C 17342,c1(C(CC(=O)OC)NC(=O)NC2(C(C)(C)O)CCC2)ccc(C2CC2)cc1 17343,N1(C(C(C)Cc2cccnc2)=O)CCCN(C(C2(NC(N)=O)CCC2)=O)CC1 17344,C=Cc1cncc(C(N2CCC3CC23C(=O)NCCc2cc(C)no2)=O)c1 17345,C1(CNC(COCC)=O)CCN(c2ccnc(NC3CCCCC3C)n2)CC1 17346,C(=O)(CC(C)(C)COC)NC1(CC=C)CCN(C(c2cc(Br)n[nH]2)=O)C1 17347,c1(C(N2CCCC(N(C(=O)CCN3CCOCC3)C)C2)=O)ccc2c(n1)COCC2 17348,C1(C(=O)OC)CC(NC(=O)C(C)Cc2cccc(C)c2)CCN1 17349,C1(NC(C2(C)CCN(C(C)=O)C2)=O)CCN(C(C2CCS(=O)(=O)CC2)=O)C(C)C1 17350,c1(NC(C23OC(C)C(C2)C3)=O)cc2c(cc1Br)CN(C=O)CC2 17351,C1(NC(C(CSC)(C)C)=O)CN(C(c2cc(Cl)c(Br)[nH]2)=O)CCC1C 17352,C1(CC(=O)NC(C=C)(C)CC)CCN(C(C)=O)C1(C)C 17353,N1(C(CCOCCOCC)=O)CCC(C(C)CNC(C2(C)CC=CCC2)=O)CC1 17354,C1(NCC(c2cccs2)N(C)C)CP(C)(=O)CC1O 17355,N1(C(CCC)=O)CC(NC(c2ccc(Br)c(C)c2F)=O)C2(CCC2)C1 17356,c1(C(=O)NCc2c(CCNC(c3c[nH]nc3F)=O)ocn2)c(Cl)cccc1Cl 17357,N1(C(Cn2nc(C)oc2=O)=O)CCC(NC(C2(CC(F)F)CCC2)=O)C(O)C1 17358,c1(N2CC(CNC(c3c(CC)nco3)=O)N(C)CC2)ccc([N+](=O)[O-])cn1 17359,CC(C)(C)CC(C)(C)C(=O)NCC(F)CNC(c1nccnc1N)=O 17360,c1(C(=O)NC(CNC(c2nc(C)[nH]n2)=O)C)coc(=O)c2ccccc12 17361,c1(C(=O)NCC2CCC(NC(C3CC(N4CC(O)C4)C3)=O)C2)sc(F)cc1Cl 17362,c1(SC)cc(C(=O)NCC2CC2NC(=O)CS(=O)(=O)NC(C)(C)C)c(C)o1 17363,c1(OC)cc(Br)ccc1C(=O)CN(C1CCCCC1NC(=O)OC(C)(C)C)C 17364,C1(NS(=O)(=O)Cc2cc(F)ccc2F)CC2CCC(C1)S2(=O)=O 17365,n1(CC=C)cc(C(=O)NC2(C)CC(C(N3CCC3(C)C(=O)NC)=O)C2)cn1 17366,N1(C(c2cccc(-c3cn[nH]c3)c2)C(=O)NCC=C)CCC(C)C(C)(C)C1 17367,c1(C(=O)NCC(C)CN(C(=O)C2=NOC(C(C)(C)C)C2)C)ccc(O)nc1Cl 17368,C1(CNC(=O)C(C2CCCCC2)O)CN(C(c2cc(C3CC3)[nH]n2)=O)CCCO1 17369,C1(NC(c2nc(CC)oc2)=O)(COC)CCN(C(C2(N3CCOC3=O)CC2)=O)C1 17370,CCCCCCCC(=O)N1CC(NC(c2cc(F)ccc2C)=O)C(O)C1 17371,c1(CC)cccnc1C(=O)N(C(CC)C(=O)NC1CCN(CCF)C1)C 17372,c1(C(=O)NC(CNC(c2cnc(OCC)s2)=O)(C)C(C)C)cnn2c1CCC2 17373,Cc1sc(Cl)c(C(=O)NCCOCCCNC(=O)CCC2CCN(C)CC2)c1C 17374,CC#CCCCC(=O)N1CCCC1CCCNC(=O)COc1cccc(C)c1 17375,N1(C(C(COCC)C)=O)CCC2C1CCCN2C(c1cccc2ncnn12)=O 17376,C1(C(=O)NCC2CN(C(=O)Cc3ccsc3Cl)C2)COCCC1(F)F 17377,C1(C(N2CCN(C(=O)OC)CC2)=O)CC12CCN(C(c1ccc(I)c(O)c1)=O)C2 17378,C1(C(N(C)Cc2c(C)cco2)=O)CC(NC(=O)Cc2cncn2C)C1(C)C 17379,N1(C(c2cnn(C)c2Cl)C(=O)NCCSC)CCc2ccc(Cl)nc2C1 17380,c1(OC)ccc(C(=O)NC2CN(C(=O)CN3CC4CC4C3)CC23CC3)cc1OC 17381,CC1CCCC(C(=O)N(CCCNC(=O)Cc2csc(C(C)(C)C)n2)C2CC2)CC1 17382,N1(Cc2c(C(=O)OCC)ccs2)CCN(C(=O)C(O)CC(C)C)C2CC12 17383,C1(NC(CCn2ncn(C)c2=O)=O)CC(NC(C2(S(C)(=O)=O)CC2)=O)C12CCC2 17384,N1(C(C(C(C)NC(C)=O)C(C)C)=O)CCC2=C(CCCC2)C1.N1CC(CC=O)C1 17385,C#CCCCCC(=O)Nc1ncoc1C1CNC1.N12CCC(C1)C1CCCN1CC2 17386,c1(C(N2CCN(C3CN(C(C4ON=C(C)C4)=O)C3)CC2)=O)ccc(O)nc1C 17387,C1(C(=O)NC(C(C)NC(c2cc3occc3s2)=O)(C)C)CCc2nncn2C1 17388,c1(C(N(C(COC(C)=O)=O)CCOC(C2CCC(F)C2)=O)=O)cc(O)ccc1N 17389,C=CCC(C)(C)CC(=O)NC1CN(C(c2cnc(CC)s2)=O)CCC1CO 17390,c1(C(N2CCC(NC(c3c(CC)ocn3)=O)C2C2CC2)=O)c(F)cc(F)cc1Cl 17391,N(C1CCc2c(Br)cccc21)CCCn1c(C(C(CC)CC)N)nnn1.OCC 17392,CCCC(CCC)C(=O)NCCC(C)NC(C1CCS1(=O)=O)=O 17393,C1(C(N2CCC(OCCNC(c3ccc(SC)cc3)=O)C2)=O)CCCCN1N=O 17394,c1(C(=O)NCC2(CCNC(CN(C3CC3)CC)=O)CC2)cc(C(N)=O)co1 17395,C=C(C)CCCNC(=O)C(=O)NCC(C)(C)OC(CSCC)=O.C(C)(C)(C)O 17396,O=C(C1=C(F)CN(C(C2(F)CCOC2)=O)CC1)NCc1nn[nH]n1 17397,c1(C(N(C(C(N2CCC(NC(=O)NC)C2)=O)C)C)=O)nn(C)cc1C 17398,N1(C(CNC=O)=O)CCOCC1CCNC(=O)COC1CCOC1 17399,O=C1COc2ccc(C(=O)NC34CC3CN(C(c3cnc(Cl)[nH]3)=O)C4)cc2N1 17400,c1(C(=O)NCC(C)(C)NC(=O)Cc2ccc3c(c2)CCC3)cc(Cl)c([N+](=O)[O-])[nH]1 17401,N1(C(CCS(C)=O)=O)CCC(NC(=O)Cc2ccc(F)c(Cl)c2)C12CC2 17402,c1(C(N(CC(CNC(Cc2scc(C)n2)=O)C)C)=O)cccc(C2CC2)n1 17403,CCCC(O)(CCC)CC(=O)N1CCCC(Cc2cn(CC3(CO)CC3)nn2)C1 17404,C(c1cnn(C)c1C)=CC(N1CC(NC(c2cc(CC)ncn2)=O)C(OC)C1)=O 17405,c1(NC(C2(NC(=O)OC(C)(C)C)CC23CCC3)=O)cnnc2ccccc12 17406,c1(COC)ccc(C(=O)NC2(CNC(=O)CC3(O)CCC3)CC2)s1 17407,C(=O)(C1CCCc2nncn21)N(CCN(C(=O)C=Cc1ccco1)C)C 17408,S(=O)(=O)(c1ccc(C(N2CCC(C)(CNC(c3ccoc3)=O)C2)=O)cc1)NCC 17409,c1(C(=O)NCC(CC=C)NC(c2nn(C)nc2Br)=O)cnc(C)n1C 17410,N1(C(c2cc(CCC)on2)=O)CCCC(CC(=O)NC2CC3CCC2O3)C1 17411,CC1CN(C(=O)C=C(Cl)Cl)CC2(CCN(C(c3ccc(S(N)(=O)=O)o3)=O)C2)O1 17412,c1(CSC)c(C(=O)NC(C2CN(C(c3csc(=N)[nH]3)=O)C2)C)oc2ccccc12 17413,C1(NCc2c(F)ccc(CC(=O)O)c2)C2C3CC4C5CC(C1C35)C24 17414,C1(C)(NC(c2ncn(C(C)C)n2)=O)CCN(C(c2cc3n(n2)CCO3)=O)CC1 17415,c1(C(=O)NCC23OCC(NC(C(C)O)=O)(C2)C3)cc2c(F)ccc(Br)c2[nH]1 17416,N1(C(c2c(C)csc2C)=O)CCCN(C(=O)C=CCCc2ccccc2)CC1 17417,S(=O)(=O)(c1csc(C(N2CC(CNC(=O)C(C)(C)F)C3CC23)=O)c1)NC 17418,c1(C(N(CC(C)NC(c2c(C(C)C)con2)=O)C)=O)cn(C)nc1C(F)F 17419,c1(C(N2CC3C(CNC(c4n(CC)cnn4)=O)(C3)C2)=O)ccc2c(n1)CCCC2 17420,CC(O)CC(C)CNC(=O)Nc1cccc(OCC(F)F)n1 17421,CN1C(=O)Cc2ccc(-c3nc(-c4cccc(N(C)C)n4)nn3CC(N)=O)cc21 17422,N#Cc1cc(N2CCC(NC(=O)CSc3n[nH]c(O)n3)C2)nc(C2CC2)n1 17423,C1(NC(c2c(CC)occ2C)=O)CN(C(c2oncc2C)=O)CCC1F 17424,CC1CCCN(C(c2cnsc2)=O)C1CNC(C1OCCN(C)C1=O)=O 17425,C1(C(=O)NCC(C2CCC2)OC)CN(C(c2cn(C)cc2C)=O)CC1(F)F 17426,c1(NCC=CCNC(CC2C(OC)COCC2)=O)ncn(C)c(=O)c1Br 17427,c1(C(=O)NCCCCCN(C(C)C)C(C2CSCCS2)=O)ccc(O)c(F)c1F 17428,N(C(=NCCC(=O)N(C)C)N1CCC2(CCN(C)C2)C1)Cc1ccc(C)c(C)c1 17429,c1(C(C2CC2)NC(=O)NC(CC)CCCO)cc(Cl)ccc1Cl 17430,CC1(C)CC(NC(C2CC2c2ccc(Cl)cc2)=O)CN1C(c1ccc(F)cn1)=O 17431,C(CCCC(=O)NC(C)(C)C(=O)N1CCC1C(C)C)OC 17432,C1(NC(Cc2cc(CC)no2)=O)CC2CCC1C1CN(C(C3CCOC3)=O)CC21 17433,C1(C(=O)NCCCCNC(c2c(C)cc(C)nc2)=O)CCc2nnc(O)cc2C1 17434,c1(C(N2CCN(Cc3ccc(C(F)(F)F)nc3)C3CC23)=O)cn2ncccc2n1 17435,N(C1CC(F)(F)c2ccccc21)C(C1CCSCC1)=O 17436,Cc1nc2cc(C(=O)NCC3(F)CCN(C(c4cnc[nH]c4=N)=O)C3)[nH]c2s1 17437,CCC(CCCC(=O)NCCOC(C)C)NC(c1[nH]ccc1COC)=O 17438,C1(CC(N2CCC(COC)(NC(=O)C3=COCC3)CC2)=O)CC(C)CC(C)(C)C1 17439,c1(CC)cc(C(N2CCOC(c3cn[nH]c3)C2)C(=O)NC(C)(C)C)n(C)n1 17440,c1(C(=O)NC2CC(C(N(CCCC(C)O)C)=O)C23CCC3)cccc2[nH]ncc12 17441,Cc1cccc(CNC(C2CCCN2C(=O)C=CC2CCOCC2)=O)c1 17442,CCC(CC)C(C)C(=O)N1CCN(C(=O)CC(F)(F)CC)C(c2ccccc2)C1 17443,c1(C(=O)NCC(C)CNC(=O)CCN(C)CCO)ncnc(O)c1Cl 17444,CC1CCC(CCC(=O)N(C(Cc2ccco2)CO)CCN)O1 17445,c1(CN2CCCC(CN(C)C(c3cccnc3S)=O)C2)cccc2ncccc12 17446,C(=O)(CCCC(C)(C)C(=O)OC)NC(CN(C(C(C(C)OC)N(C)C)=O)C)C 17447,Cc1ccc(CNC(C2C3CC3CN2C(=O)CCC2CC2C)=O)nn1 17448,N1(C(C(C=C)CC)=O)CC2(C1)CN(C(=O)C=Cc1ccco1)CC2CO 17449,c1(C(N(C2CCCCCC2)CCNC(C2CCC2(F)F)=O)=O)nnn2c1CCCC2 17450,c1(C(N2CC(NC(CS(=O)(=O)NC)=O)C(F)CC2)=O)ccc2c(c1)OCCCO2 17451,N1(c2ncc(C#C)cn2)CCN(C(c2cc(F)c(Cl)cc2F)=O)C(C#N)C1 17452,Cc1cc(C(=O)NCC(C(C)C)NC(=O)CCCC2CC2)c([N+](=O)[O-])c(O)n1 17453,C1(NC(c2cnn(CC)n2)=O)CC2(C(=O)NCC3CC(=O)N(C)C3=O)COC1C2 17454,c1(C(N(C2CN(C(=O)CN3CCC(O)CC3)CC2O)C)=O)cc2occc2n1C 17455,C(=O)(C(C)C(C)C1CN(C(=O)CCn2cc(-c3c(C)ncn3C)nn2)C1)OC 17456,N1(C(CCC=C(C)C)=O)CC2CCN(C(c3scc(C)c3Cl)=O)C2C1 17457,Cn1cnc2c(C(N3CCOC(CNC(=O)CC4(C)CCCO4)C3)=O)ccnc12 17458,Cc1cc(C(N2CC(C)C(C)(CNC(=O)CN(C)C3CC3)C2)=O)nnc1C 17459,CCCCCC(CC)C(=O)NC1CCC1CNC(c1cnnc(C)c1)=O 17460,C(c1ccc(F)c(F)c1)=C(CCC(=O)N(c1ccc(F)cc1C)CC)C 17461,c1(C(=O)NCC2(CNC(C3C(C=C)OCC3)=O)CCCC2)cc(Cl)c(Cl)n1C 17462,Cc1cc(C)c(S(=O)(=O)N2CCC(O)(CC(=O)N(CC(O)CO)C)CC2)c(C)c1 17463,O=C1Cc2cnc(N3CCC(C(=O)Nc4c(Cl)ccnc4Br)C3)nc2N1 17464,N1(C(c2cc(CC)on2)=O)CCCC(CC(=O)NCC2(CC3CC3)CCC2)C1 17465,C1(C)(NC(C=C(C)c2ccco2)=O)CCN(C(=O)C(C)c2ncco2)CC1 17466,C1(C(=O)OC)CC12CCCC2.O(NC(=O)CN1CC1)CCC=C 17467,C(=O)(C(C)(C)CC(F)F)NC(C)CC(C)NC(C1CCN1C(C)(C)C)=O 17468,CCC(C(=O)N1CCC(CCNC(C2CCC(N(C)C)CC2)=O)C1)C(C)C 17469,Cc1sc(O)nc1C(N1CC(C(N)=O)(CNC(=O)Cn2cnnc2)C1)=O 17470,CC1OCC2(CCN(C(c3sccc3NCc3nccnc3Cl)=O)CC2)C1N 17471,CC1C(C)CCN1C(c1c[nH]nc1CCNC(=O)CCC(=O)N(C)C)=O 17472,N1(C(c2cn(CCNC(C(C)SC)=O)nn2)=O)CCN(C)C(C2CC2)C1 17473,c1(OC)ccccc1NC(=O)N(C1CCCC1)Cc1cscn1 17474,C(CCNC(C1CCCN1C(N)=O)=O)(C(=O)NCC(O)(COC)CO)OC 17475,CC1CN(C(=O)CC2COC(=O)C2)CCC1NC(=O)CC(C)(O)C1CC1 17476,CC(C)(C)CCCCC(=O)NC1CN(C(c2ccn(C(F)F)n2)=O)CC(C)(C)C1 17477,C(C)(CCC(=O)NCC1CCCC1NC(=O)CSC(F)(F)F)OC 17478,c1(NC(=O)CCCNC(C2(C3OCCO3)CCCOC2)=O)cc(Cl)c(Cl)cc1Cl 17479,C1(NC(c2sc(CC)c(C)c2)=O)CN(C(C2(CCOC)CCC2)=O)CC1(C)C 17480,CC1CC(CNC(=O)CC(C)(C)c2ccc(F)cc2)CN1c1nnc(C2CC2)o1 17481,c1(CC)ccc(C(=O)NCC2CCCN(c3ncccn3)CC2)cc1CC 17482,C1(NCCC2N(C(CCC(=O)NC3(C)CC3)=O)CCSC2)CCCC(F)(F)CC1 17483,N1(C(CCC#C)=O)CCC(N(C)C(c2cc(SC)oc2C)=O)CC1 17484,C12(C(=O)NC3(CNC(c4ccc(C)cc4Cl)=O)CCOC3)CCCC(C)(C1)OC2 17485,c1(COC)cncc(C(=O)NCCOCCCNC(=O)CC(C)n2cccc2)c1 17486,C1(CNC(c2cc(C)ns2)=O)CC(F)(F)CN1C(c1ccc(N)c(Cl)n1)=O 17487,N1(C(c2occ(C(C)=O)c2)=O)CC(NC(=O)Cn2ccc(Br)n2)C(C)C1 17488,N1(C(c2ncn(CC)c2)=O)CCCC2CN(C(c3cc(O)ncn3)=O)CCC12 17489,N1(C(CSS(C)(=O)=O)=O)C2CCC1CC(NC(c1cc(Cl)no1)=O)C2 17490,c1(NC(CCC(C)NC(=O)CC2CC(N(C)C)C2)=O)cccn2ncnc12 17491,CC1(C)CCC=C1C(=O)NCC12CN(C(C3SCCCS3)=O)CC1(C(F)(F)F)C2 17492,CN=c1cc(C(=O)NCC(c2cn(C(C)C)nn2)(C)C)c(Br)c[nH]1 17493,C1(CNC(C(C)SC(F)(F)F)=O)CN(C(=O)COCc2ccnn2C)CCN1C 17494,C(c1ccc([N+](=O)[O-])cc1)=CC(=O)NCCNC(c1cc(F)c(OC)c(F)c1)=O 17495,c1(CN2CCC(N(C(c3cccc(CC)n3)=O)C)C2)ccc2c(c1)OCCO2 17496,C1(CNC(C2(NC(=O)NC)CCCC2)=O)CCC(NC(C2CC2CF)=O)CC1 17497,C=CCCC(O)CN(C)C(C1CC(C)CN1C(=O)C=C1CCCCC1)=O 17498,C1(N(C(Cn2c(C)cnc2)=O)C)CC2CC1N(C(=O)CNC(C1CCC1)=O)C2 17499,c1(C(C(=O)NCCCCC)N(c2ccccc2)CC)ncc(COC)cn1 17500,c1(C(=O)Nc2ccc(CC)nc2)c(NC(=O)CS(C)(=O)=O)sc2c1CCC2 17501,c1(CCC(=O)NCC2(NC(C3CCC(C)S3)=O)CC2)cccc([N+](=O)[O-])c1 17502,c1(C(N2C(CN(C)C(C3CC3(Cl)Cl)=O)CCC2)=O)cn2c(n1)COCC2 17503,CC1(C(=O)NCCCNC(=O)Cc2ccc(Cl)cn2)CS(=O)(=O)C1 17504,Cc1ccc(CC(=O)NC(C)(C)CCNC(C2(C)CC2F)=O)o1 17505,C12(CN3CCN(CC(N4CCCC4)=O)C(C)C3)COCC(C3CC3)(C1)C2 17506,CC1CCC(CCC(=O)N(C)CC2CN(C(=O)CCCC3CC3)C2)O1 17507,c1(C(N2CC(CC)N(C(c3cccc(=O)o3)=O)CC2)=O)ccc2c(c1)COCC2 17508,N1(C(Cc2cc(C)on2)=O)CCOC2CN(C(=O)C(C)(O)C(F)(F)F)CC12 17509,C12(NC(=O)CCC3CC3(F)F)CCCN(C(=O)COc3ccccc3O)CC1C2 17510,N1(C(C(CO)NC(N)=O)=O)CCCC(CNC(C2(S(N)(=O)=O)CC2)=O)CC1 17511,C1(NC(C(CCC)NC(N)=O)=O)CCN(C(=O)CS(=O)(=O)CC)CCC1CO 17512,C(=O)(C1=CS(=O)CCC1)NC1CCN(C(c2c(C)c(Br)ccn2)=O)C1(C)C 17513,c1(CC(N2CCC(N(C(=O)C(F)C(C)C)CC)C2)=O)cc(F)cc([N+](=O)[O-])c1 17514,c1(C(=O)NCCCCCNC(C2(C)CC2(Cl)Cl)=O)cc2c(nn1)CCC2 17515,Cc1cc(F)c(C(=O)NCC(C)(C(C)C)NC(c2ncsc2C)=O)c(Cl)c1 17516,CC1CCN(S(=O)(=O)CCn2cncn2)CCC1N1CCC(F)C1 17517,c1(OC)ccc(-c2noc(C3CCCC3N)n2)c(Cl)c1 17518,N1(C(C2C(=O)NCC2)=O)CCC2CC1CN(C(c1ccc3c[nH]nc3c1)=O)C2 17519,c1(C(=O)NCC2N(C(C3(SC)CCC3)=O)CCCC2)noc2cc(Cl)ccc12 17520,Cn1cc(C(Cc2cn(CC(=O)O)nn2)NCC2COC(=O)C2)cn1 17521,N1(C(C(C(C)NC(CSCCOC)=O)(C)C)=O)CC2CCCC(O)C2C1 17522,CC1(CC(=O)NCC(C2CC2)NC(=O)C(F)=C2CCC2)CC1(F)Cl 17523,N1(C(CCc2nnc(C(C)C)o2)=O)CCN(C(=O)C=CCF)CC12CCC2 17524,c1(C(N2C3C(C(=O)Nc4cncc(OCC)c4)C(C3)C2)=O)ccnc([N+](=O)[O-])c1 17525,N1(C(C(C)C2(O)CCC2)=O)C(C(=O)NCCN(C)CCF)CCC1C 17526,C1(O)(CC(C)C)CCN(C(=O)CC2(N(C)C(c3ccnnc3)=O)CC2)C1 17527,CC1(CNC(C2(F)CC=CCC2)=O)COCCN(C(c2ccc(Cl)c(O)c2)=O)C1 17528,c1(NC(CC2(OC)CN(C(C3CCCC3OC)=O)C2)=O)cccc(F)c1 17529,C#CCC(CC#C)C(=O)NCC(C)N(C(=O)CCc1cccc(OCC)c1)C 17530,c1(CC(C(=O)NCC23N(C(CC(C)O)=O)CC(C2)C3)F)ccc([N+](=O)[O-])cc1 17531,c1(NC(C(CSC)C)=O)cccc(NC(=O)CCc2nncn2C)c1 17532,C1(NC(c2c(SC)n(C)nc2)=O)CN(C(=O)CN2CCCCC2)CC(C)(C)C1 17533,N1(C(=O)C=Cc2cscn2)CCCN(C(=O)CC2CCC3(CCC3)O2)CCC1 17534,N1(C(c2cc(C(C)(F)F)on2)=O)CC2CCN(C(C3(c4cc[nH]n4)CC3)=O)C2C1 17535,C12(NC(c3cc(C(F)F)ccn3)=O)CCC1CN(C(=O)CC1CCCCC1O)C2 17536,c1(NC(C2C(CNC(=O)NCC3CC(n4cncn4)C3)CC2)=O)ccccc1Cl 17537,CC(C(=O)NCC(C)(C)CNC(c1csc(C(=O)NC2CCC2)n1)=O)C(F)F 17538,c1(OC)ccc(Cl)c(F)c1-c1cn(CCCCCNC(C2(C#N)CC2C)=O)nn1 17539,c1(C(C)C)ccc(C(=O)NCCn2cc(-c3cccs3)nn2)cc1F 17540,c1(CNC(CN(C(C(=O)NCC)=O)CC)=O)nccn1CC 17541,c1(C(=O)NC2C=CC(CC(=O)NC(CCCC)C)C2)ccnc2cc[nH]c12 17542,c1(C(=O)NCCC)ccc(C(=O)NC(C)(C)CNC(=O)Cc2ccccc2)nc1 17543,C1(C(N(C(C)C(=O)NCC(C(C)(C)C)OC)CC)=O)CCN(C)C(=O)C1 17544,c1(CC(=O)OC)ccnc(NCC2(CCNC(c3occc3Br)=O)CC2)n1 17545,C(CCCCCNC(c1nocc1Br)=O)N(C(=O)COC1CC(F)(F)C1)C 17546,C12(CNC(c3c(C)nc(N(C)C)s3)=O)CCC(CC1)N2C(c1cocn1)=O 17547,N1(C(C(CC=CCC)C)=O)CC(C(=O)NCC(F)Cl)CC12CCC2 17548,C1(C)(C(=O)NCC(C)CN(C)C(c2cnn(C(F)(F)F)c2)=O)CCNC1 17549,C1(C(N2CCCC(CCC(=O)NC3(C)CCC3)C2)=O)CC2CCCC2C1 17550,C1(NC(C(C(CC)O)C)=O)CCN(C(=O)C(C)(O)c2ccccn2)CC12CCC2 17551,c1(C(C(=O)NC2CC(NC(c3c(CC)occ3)=O)C2)(F)F)ccc(Br)cn1 17552,c1(C(N2CCCC2C2CCOC2)C(=O)NC(CC)C)ccc(C(=O)OC)cc1 17553,C(=O)(C(C)(C)C(=O)NCCC(COC(c1cc(Cl)ncc1OC)=O)OC)OC 17554,CC1(C)CCCC(C(=O)NC2CN(C(c3cccnn3)=O)CC2(C)C)C1 17555,N(C(=NCCc1ncccc1C)NCc1nn(C)cc1Br)C(COC)C 17556,N1(C(C(C)C2CCCC2)=O)CCN2CCN(C(=O)C(C)C3CCC3)CC2C1 17557,N1(C(C(C)=CC2CC2)=O)C2CCCC1CN(C(C1CC3CCC1O3)=O)C2 17558,CCC(CC)C(C)C(=O)N(CC(=O)NC1(COC)CC(C)(C)C1)CCOC 17559,c1(CC)occc1C(=O)NC1CC1CNC(=O)CCc1cn[nH]c1 17560,c1(C(=O)NC2C(CC)CN(C(=O)CCNC(N)=O)CC2)cc(C)cc(C)c1N 17561,C12(NC(C(C)(C)O)=O)CN(C(c3[nH]nnc3C3CC3)=O)CC1CS(=O)(=O)C2 17562,CC1CCCN(C(c2cnn(C(F)(F)F)c2)=O)C1CCNC(c1cnccn1)=O 17563,c1(NCC(CCC)C)ncccc1S(=O)(=O)NC1(c2cc(F)cc(F)c2)CC1 17564,C1(CNC(=O)COCC2CCOC2)CC2CCC(C1)N2C(=O)C=Cc1cnc[nH]1 17565,c1(C(=O)NCC(C2CCN(C(CC(C)SC)=O)CC2)(C)C)c(O)cccc1F 17566,CCCCC(F)C(=O)NC1CC(OCC(N2CCC(C(F)(F)F)C2)=O)C1 17567,c1(OC)cccc(C(=O)NC2CCC(CNC(=O)CC3(OCC)CCCC3)C2)n1 17568,CCC(CC(=O)N(CC(=O)NC(C)Cn1cnnc1)C1CC1)CC(C)C 17569,C1(F)(CNC(C=CCCC)=O)CCN(C(=O)CSCCOC)C1 17570,C(=O)(C(O)CC(C)(C)C)NCC1(F)CCN(C(C(CC)C#N)=O)CC1 17571,C(=O)(C1=C(Cl)CCC(C)C1)NCC1(CNC(C(C)S(N)(=O)=O)=O)CCC1 17572,C1(Nc2n(C)c(=O)nc(O)c2)CC2(CCCCN2C(=O)CCN2CCC(F)C2)C1 17573,N1(C(CCC)=O)CCCC(CCNC(=O)C(c2cc(Cl)cc(Cl)c2)(C)C)CC1 17574,Cc1ccc(CSc2ccc(C(=O)NC3(C4CCCCO4)CC3)o2)cc1 17575,c1(C(C)(C)C)cc(C(c2nnnn2C2(C)CC2)NCC(CO)C2CC2)on1 17576,CN1CC(=O)N(CC(=O)NCC2CN(C(c3cnsc3)=O)C2)C1=O 17577,c1(N(CCCSC)C)cc(C)c(S(=O)(=O)N2CCSC2c2ccco2)cn1 17578,C(C(=O)NOCC1CCS(=O)(=O)C1)(c1ccccc1)NC(CC=C(C)C)=O 17579,C=CCC(C(=O)NCCC1(SC)CN(C(=O)C(C2CCCCC2)O)C1)NC(C)=O 17580,N1(C(C2CN(C(C)=O)C2)=O)CC(N(C)C)C(CNC(=O)Cc2csc(C)n2)C1 17581,N1(C(c2nn(CC)c(C)c2)=O)CCC2(CCCN2C(=O)C(O)C2CC2)CC1 17582,Cc1nn2cc(C(=O)NCCN(C(C3CC(C)(C)O3)=O)C3CC3)nc2s1 17583,C1(C)(C(=O)NC2CCN(C(COCC#C)=O)C2C2CC2)CCS(=O)(=O)CC1 17584,CON(CCC(=O)N(C)C(c1ncccn1)C)C(=O)C1(C#N)CCOC1 17585,N1(C(CCNC(=O)NCC)=O)CC(OC)CC(NC(c2ccc(O)nc2Cl)=O)C1 17586,CC(C)CC(C)(C)CNC(C1(NC(=O)CSC(C)(C)C)CC(F)(F)C1)=O 17587,C1(C(=O)NC(CC(=O)NC)C)COCCN(C(=O)CCC2CCCOC2)C1 17588,C1(NC(CCOCC)=O)CN(C(C2Cc3nccnc3C2)=O)C2(CCOCC2)C1 17589,c1(NC(C2COCCN2C(C2CC(O)C2)=O)=O)c(F)c(F)nc(F)c1F 17590,c1(C(=O)NC)cc(C)[nH]c(=NCC2CCCC2NC(c2nn(C)cc2Cl)=O)n1 17591,C1(C)(CNC(c2n(CCCC)nnn2)c2ccnn2COC)CCC(=O)N1 17592,CC1(C)C(NC(C2(n3cncn3)CC2)=O)CCN1C(c1ccnc(C(N)=O)c1)=O 17593,c1(C(=O)NC2CCN(C(c3c(C)c(F)ccc3N)=O)C2)c(F)cccc1[N+](=O)[O-] 17594,CS(C)(=O)=NCC(=O)NC1CCOCC1NC(=O)C=Cc1ccccn1 17595,C#CCC(CC#C)C(=O)NCC12CC1CN(C(C1(COC)CCCC1)=O)C2 17596,C12(NC(C=CS(C)=O)=O)CCOCC1CN(C(c1ncnc3ccsc13)=O)C2 17597,C1(NC(NCCCN(c2ccc(Cl)c(Cl)c2)C)=N)CC2(CCOCC2)C1 17598,c1(C(=O)Nc2c(OCC)cccc2)ccc2[nH]nc(-c3c(C)nn(C)c3C)c2c1 17599,N1(C(C(C)CC2CCCC2)=O)CCC(CO)(CNC(c2cccc[n+]2[O-])=O)C1 17600,c1(C(=O)NC2C(CNC(c3c(CC)[nH]cc3)=O)CCCC2)nn(C)c(N)c1C 17601,Cc1nc(SCC(=O)NCCCN(C(=O)C(C)N2CCCC2)C2CC2)n[nH]1 17602,Cc1ccc(-c2ccnn2C)cc1NC(N1CCC(c2ncc(Br)cn2)C1)=O 17603,N1(C(c2cc(C)nnc2)=O)CC2CCC2(CCNC(c2cc(F)ccc2O)=O)C1 17604,C1(NC(=O)NC2(CO)CCN(C3CCC3)C2)CCCN(c2ncc[nH]c2=O)C1 17605,N1(C(c2cc(C)c(Br)s2)C(=O)NCCSC)CCC12CCN(C)C2 17606,c1(C(=O)NC(CN(C(=O)C2=CCCC2(C)C)C)(C)C)cc(F)cc(N)c1F 17607,C(=O)(CCS(C)(=O)=O)NCC(CC)(CC)NC(C1CC2C=CC1O2)=O 17608,Cc1cc(Cl)ccc1C(N1CC(CNC(=O)CSCc2cccs2)C1)=O 17609,C1(NC(=O)CCC2CCC2)CC2CC1CN(C(=O)CC1CNC(=O)C1)C2 17610,C1(OC)CN(C(c2cocn2)=O)CCC1NC(c1cc(Cl)cnc1Br)=O 17611,Cn1cc2c(n1)CCC(C(N1CCC(NC(=O)C=Cc3ccc(Cl)cc3)C1)=O)C2 17612,Nc1ncc(C(=O)NCC2CN(C(=O)Cc3cncs3)CC2(F)CO)cc1Cl 17613,C1(C(=O)N(C)CCNC(C2CC2C(F)(F)F)=O)(NC(C)=O)CC1 17614,N1(C(C(c2nc(C(C)(C)C)no2)C)=O)CCCCCC1CO 17615,CC1CN(C(c2coc(C3CCC3)n2)=O)CCN1C(c1cc(Cl)c[nH]1)=O 17616,c1(NC2CN(C(Cc3cc(C)cc(C)c3)=O)CC(F)C2)ncnc2occc12 17617,CC(C)C(C)CC(=O)NC(CC1CCC1)C(=O)N1CC(c2cnsc2)C1 17618,CC(C)(C)C(CNC(C1CC2CCC1CC2)=O)C(=O)N1CCC(CCO)CC1 17619,C1(CNC(c2ccc(C=C)cc2)=O)CN(C(=O)CO)C2(CCC2)C1 17620,C(=O)(C1=CCC(C)CC1)NCC(CC)(CC)NC(=O)Cn1nnc(=N)[nH]1 17621,C1(C(N2C(CNC(c3c(CC)noc3)=O)CCCC2)=O)Cc2cccc(C)c2O1 17622,N1(C(CCCCCC)=O)CC(C)CN(C(=O)CCC=CC(C)C)CC1C 17623,c1(C(=O)NC(CNC(C2N(C(C)C)CCCC2)=O)C)ccc(N)c(O)c1 17624,c1(C(N(CC(C)N(C)C(C2CCC(=O)N2)=O)C)=O)coc2c(F)c(Cl)ccc12 17625,CC1CCOC(C(=O)NCCCN(C(=O)Cc2cccs2)C2CC2)C1 17626,c1(C(=O)NC2C(CNC(C3C(CC)CCO3)=O)CCC2)ccc(C2CC2)cc1C 17627,CC1(C)C(C)(C(=O)NC2CN(C(c3sccc3C(F)F)=O)CCC2CO)C1(C)C 17628,c1(CCC)ccc(NCc2ccc(C(C)(F)F)nc2)cc1 17629,C1(C(=O)NC(C2CN(C(c3cnncc3O)=O)CCO2)C)CC12CCSCC2 17630,N1(C(=O)Nc2c(CC)cccc2)CC2CC1CN2C(=O)OC(C)(C)C 17631,C1(C(N2CCC(CCNC(c3ccccc3Cl)=O)C2)=O)CCC2(CC1)CC2(F)F 17632,N1(C(c2nc(OC)c(C)s2)=O)CC(CNC(=O)C(C)(F)C(C)(C)F)CC(C)(C)C1 17633,N1(C(c2c(C#N)ccs2)=O)CC2CC(C1)C2NC(c1ccnc(OCCO)c1)=O 17634,CC1CCN(C(=O)OC(C)(C)C)CC1NC(C1C2CCCC12)=O.C12CC(C1)N2 17635,N1(C(=O)CCc2ccsc2)CCC(CNC(C2(F)CCOC2)=O)C1 17636,C1(NC(=O)CC2CC(n3cnnc3)C2)(CF)CCN(C(=O)CC2CC2(Cl)Cl)C1 17637,C1(C(=O)NCc2ccc(CNC(=O)COC3CCCC3)cc2)CC2(CCO1)CC2 17638,C1(N(C)C(C2CCC(O)CC2)=O)CCCN(C(=O)CN2CSCC2=O)CC1 17639,c1(CC)nc(C)oc1C(=O)NC(CO)C(=O)NCC1CCCSC1 17640,C(=O)(C1=CC2CCCC12)NCC=CCNC(c1cc(C)c(Cl)s1)=O 17641,N1(C(C(CC)(F)F)=O)CCC2C(CCCN2C(c2coc(C(F)(F)F)n2)=O)C1 17642,N1(C(N2CCC(C)CC2)=O)CCc2c1ccc(F)c2F 17643,C1(CC(=O)NCCc2n(C)c(=O)on2)CN(C(=O)C2=COCC2)CC12CC2 17644,c1(C(NOC(c2ccccc2)C)=O)cc(O)c(F)cn1 17645,C1(CNC(c2n(CC)ncc2Br)=O)CC2CCC1N(C(C1(OC)CC1)=O)C2 17646,C=CCCCCCCCC(=O)N1CC2(C1)CN(C(c1cnc(C)s1)=O)CCO2 17647,C(CS(=O)(=O)CC(=O)NCc1ccc(C(=O)NC(CO)C2CC2)o1)OC 17648,C(=O)(C#CC1CCCCO1)NC1C(OC)CN(C(c2cc3n(n2)CCCC3)=O)C1 17649,C=CC(CC)CC(=O)NCCOC1CCN(C(=O)C(Cc2cnc[nH]2)N(C)C)C1 17650,C1(C2CCCN(C(=O)C3=C(Cl)CCC3)C2)(NC(C2(C)ON=C(C)C2)=O)CC1 17651,c1(CC)ccc(OCC(=O)NC2CCN(C(C3(C)COC(=O)C3)=O)C2)cc1 17652,c1(OC)n[nH]cc1C(=O)NC(CN(C)C)C(=O)N1CCC(OC2CCC2)C1 17653,C1(CCC(=O)N(C(CCSC)C)C)CCC(NC(c2nccn2C(C)C)=O)C1 17654,c1(C(=O)NCC2N(C(Cc3cnn(C)n3)=O)CC2)cc(=O)oc2ccc(O)cc12 17655,c1(OC)cc2c(cn1)NC2.c1(C(N2CCC(N3CCCC3)C2)=O)nccnc1Cl 17656,C(C)(CO)(C(=O)NCCCN(C(c1cnc(N)cn1)=O)C1CC1)OC 17657,C(=O)(C(C(C)CC)CNC(C)=O)NC1CCN(C(C2(C(=O)OCC)CCC2)=O)C1 17658,N1(Cc2ccc(C(=O)NCc3ccc(CC)cc3)cc2)CCC(C#N)(OC)C1 17659,C(CC(=O)NC1CCCC1NC(c1c(C)nn(C)c1Cl)=O)(C1=CCCC1)OCC 17660,Cc1nc2ccc(C(N3CC(N(C)C(C4CC4(C)C)=O)C4(CC4)C3)=O)cc2s1 17661,c1(CC)cc(C(=O)N(C2CCC(NC(c3cnc(C)n3C)=O)CC2)C)n(C)n1 17662,C(=O)(C(C)C(O)C(C)C)N1CCC2C(C(=O)NCC(CSC)OC)C2C1 17663,N1(C(CNS(N)(=O)=O)=O)CC2CCCN(C(c3cc4n(n3)CC(F)C4)=O)C2C1 17664,Cc1ccc(O)c(NC(c2cc(CNC(C3(COC)CCOC3)=O)cs2)=O)c1 17665,C1(CC)CCCC1C(=O)NC12CC(C(=O)NCC(c3cnn(C)c3)C)(C1)C2 17666,N1(C(C=CC)=O)CCC2(CCCC2C(=O)Nc2cccc(Cl)c2F)C1 17667,CC1(F)CCC(C(=O)NC2(CF)CCN(C(=O)CC3CC(=O)NC3=O)C2)CC1 17668,Cc1cc(C(=O)NCC2CC(F)(CNC(C3NC(=O)OC3C)=O)C2)nn1C(F)F 17669,CC(C)P(=O)(CC(=O)NCC(O)CN(C)C(c1ccoc1C1CC1)=O)C(C)C 17670,c1(SCC(N2C(CN(C(c3n(C(C)C)ncn3)=O)C)CCC2)=O)cccc[n+]1[O-] 17671,c1(-c2sc(C(=O)OC)c(C)c2)ccnc(OC)c1SC 17672,C1(NC(C(=Cc2cn[nH]c2)C)=O)CCN(C(c2cc(F)c[nH]2)=O)C(C)C1 17673,Cc1cc(C)n(C(C)C(N2CCCC2CNC(=O)C=CS(C)=O)=O)n1 17674,Cc1cc(=O)oc(C)c1C(=O)NC1CCN(C(=O)C(C)Cc2ccc(O)cc2)C1 17675,N1(C(c2cnn(CCC)c2C)=O)CCCCC(CNC(C2(F)CCOCC2)=O)C1 17676,c1(CC)ccccc1C(=O)NC1CCC1NC(c1cn(CCO)nc1C)=O 17677,CN=C(NCC(N1CCOCC1)c1ccco1)N1CCN(c2nncn2C)CC1 17678,n1(CC)cc2ccc(C(N3CC(NC(c4scnc4CC)=O)C(O)C3)=O)cc2n1 17679,C=Cc1cc(C(=O)NCC2(O)CCN(C(=O)CC3CCCN(C)C3)C2)cc(F)c1 17680,C12(C(N(C3CCN(C(=O)CN4CCCC4C)CC3)CC)=O)CCC(F)(CC1)C2 17681,CCC(CC(=O)N1CCC(CNC(=O)CNS(=O)(=O)CC)(COC)C1)SC 17682,C(CCN(C)C(C1CCS(=O)(=O)N1)=O)(C(C)(C)C)NC(Cc1c(C)occ1)=O 17683,N1(C(Cc2c(C)cc(Cl)cc2)=O)CC2CN(C(=O)CC34CCCC3C4)CC2C1 17684,N1(C(C2(CC)COC2)=O)Cc2ccccc2CC1C(N1C(C)CCC1C)=O 17685,c1(SCC(=O)NCCOCCCNC(c2n[nH]cc2F)=O)cccc(F)c1 17686,CC12CC(NC(=O)CCC3CC3)(C1)C1(CN(C(c3cncc(N)n3)=O)C1)O2 17687,c1(-c2cc(C(=O)NCc3cc(Br)ccc3O)c(F)nc2)ccc(F)c2[nH]ncc12 17688,O=C1CC(N=c2[nH]c3c(c(=NCCC4CCOCC4)[nH]2)CCCC3)CN1 17689,C(CC(=O)NCC#CCNC(C1(COC)CCC1)=O)SC 17690,c1(OC)cncc(C(N2CC(NC(=O)COC3(C)CCCC3)CC2C)=O)n1 17691,N(C)(C1CCc2cc(Cl)ccc21)C(CC1N(C)CCSC1)=O 17692,N1(C(C(C)C)=O)CCC(C2CC2)(CNC(c2coc(O)n2)=O)C1 17693,c1(OC(C)C)cccnc1C(N1CC2CC2(CNC(C2CC2C)=O)C1)=O 17694,c1(C(=O)NCC(C2(O)CCN(C(=O)CNC(N)=O)C2)C)cc2c(cn1)OCCO2 17695,Cc1ccc(O)c(C(=O)NCc2c(C)noc2C)c1.c12cc(n[nH]1)C(=O)NOC2 17696,C12(C(=O)NCC(CC)NC(=O)COC3CCCCC3)CCC(C1)C(C)(C)O2 17697,N1(CCC)CCCC(C(=O)NC2CC(O)(CNC(=O)C=COCC)C2)C1 17698,c1(C(=O)NCC2(F)CCC(NC(Cc3nc(C)sc3)=O)C2)c(Cl)ccc(O)c1N 17699,C=CC1(C(=O)NCCOCCN(C)C)CCN(C(=O)CC2CCCN2C)C1 17700,c1(C(=O)NC2(COC)CN(C(=O)C(C)(C)F)C2)cc(C)c(OC)c(C)c1 17701,C1(C(=O)NC2(CC(N3CCC(C(=O)NC)C3C)=O)CC2)CCC(=O)N(C)C1 17702,c1(C(=O)NCCCC(C)NC(=O)C(F)C2CC2)ccc(C(F)F)c(F)c1 17703,C1(NC(CC(CC)OC)=O)CCN(C(c2cc3nccnc3[nH]2)=O)CC(C)(C)C1 17704,N1(C(c2c(C(C)C)c[nH]c2)=O)CCC(F)(F)C(NC(=O)C2CC2)C1 17705,C1(OC)CCC2(C(N3CC(CCNC(C4CC(N(C)C)C4)=O)C3)=O)CC12 17706,C(=O)(C(C)(C)CCS(C)(=O)=O)NC(C)CNC(=O)C#CC1CCCCO1 17707,c1(C(=O)NCC(C(C)C)NC(C2CC3CCC2O3)=O)ccc2ncnn2c1 17708,Cc1coc(C)c1C=CC(=O)N(C(C)CCNC(=O)CC(C)(C)CN(C)C)C 17709,C1(CC(=O)NC2CCC2NC(C2CC=CC2)=O)CCCCC1(F)F 17710,C1(NC(CC2(C)CC2)=O)CC2COCC(C1)C2NC(c1cnn(CCO)c1)=O 17711,C(=O)(C1=CC2CCC=CCCC12)N1CCC(NC(CS(=O)(=O)NC)=O)C(C)C1 17712,C(c1ccccc1F)=CCC(=O)NCC(CC)(C)NC(c1cnc(O)n1C)=O 17713,CC(C(=O)N1CC(O)CC1CC(N1CC(C(=O)N(C)C)C1)=O)S(C)(=O)=O 17714,C1(NC(CC2(OC)CC2)=O)CC2CCC(C1)N2C(C12CCC(F)(CC1)C2)=O 17715,c1(C(N2CCN(C(Cn3ncc(C)c3)=O)C(CO)C2)=O)c(C)[nH]c2ccccc12 17716,C(c1ccc(C(F)(F)F)cc1)=CC(=O)NC1(C)CCN(C(c2ccsn2)=O)C1 17717,C12(NC(c3ncn(CC)c3)=O)CC1CN(C(=O)Cc1csc(C)c1)C2 17718,c1(C(=O)NC2CC(OCC(=O)N(CCCOCC)C)C2)ccc(C)cc1C(=O)C 17719,C12(NC(Cc3cn(CC)nc3)=O)CCC1CN(C(=O)C=CC1CCOCC1)C2 17720,CC1=C(C(=O)NCCC2CCN(C(=O)CCCc3ccncc3)C2)CCO1 17721,C(c1ccc(O)cc1)=CC(=O)Nc1cc(-c2cccnc2)ccc1OC(F)F 17722,CC1(C)CN(C(=O)CC2OCCCO2)CCC1C(=O)NCCC(O)C(F)(F)F 17723,C1(CC)(NC(=O)Cc2cnoc2)CCN(C(=O)CCCC2CCOCC2)CC1 17724,C1(O)(CNC(C2CC23CCCC3)=O)CCN(C(c2cscc2C(F)(F)F)=O)C1 17725,Cc1noc(C)c1C(C)C(N1CC(C(N)=O)(N(C)C)C1)=O 17726,C(=O)(CCCC(C)(C)C#N)N1CC(NC(C2(CC)CCCC2)=O)C(C)C1 17727,c1(COC)nc(C)c(C(N2CCCC(CNC(C3CN(C(C)C)C3)=O)C2)=O)s1 17728,c1(C(=O)NCC2CN(C(CCOCCOC)=O)C2)ccc(N)c(C)c1Cl 17729,c1(C(=O)NC2C(NC(COC)=O)COCC2)ccc2nc(C)oc2c1 17730,Cc1cn(C)cc1C(=O)N(CCC(=O)N(C1C=CC(CSC2CC2)C1)C)C(C)C 17731,C1(C(=O)NCCOC2CCC2)CN(C(C2CC23CC3)=O)CC1F 17732,CC(C)(C)CC(=O)NCC(=O)NC1CC(CNC(=O)CSc2ccc(F)cc2)C1 17733,N1(C(COCC=C)=O)CC2(CCC2CNC(=O)C(=O)NOC)C1 17734,c1(C(N(C(c2ccccn2)C)C)=O)c[nH]n(C)c1=O 17735,CC(C(C)(C)NC1COCC1C(=O)OC(C)(C)C)NC(=O)C(N1CCC(C)C1)=O 17736,Cc1nc(C(N2CCS(=O)(=O)C(CCNC(c3cnco3)=O)C2)=O)c(=O)[nH]c1C 17737,Cc1nc(C2CN(C(=O)C(C3CCCO3)NC(=O)CCNC(N)=O)C2)n[nH]1 17738,N1(C(c2ccc(C)cn2)=O)CCC2(NC(c3cn(C)ccc3=O)=O)CC2C1 17739,c1(CCC(=O)OCC)cc(=NC(C)CC(C)NC(=O)CCSC)[nH]c(C)n1 17740,C1(C)(C(N2CC(O)(CN(C(=O)Cc3n[nH]c(=N)s3)C)C2)=O)Cc2ccccc2C1 17741,N(C1COc2ccccc21)C(C1N(Cc2cc(OCC)cc(Br)c2)CCC1)=O 17742,N1(C(CNC(=O)OC)=O)CC2C(CNC(=O)C(c3ccc(F)cc3)N(C)C)C2C1 17743,C1(CC(=O)NCc2ccccc2F)C2CN(C(=O)CC3CCOC3)CC12 17744,C1(CC(=O)NCc2cc(C)ns2)CN(C(=O)CCc2cncs2)CCO1 17745,C(=O)(C(C)(C)C(=O)N(C)CC1CCCN1C(=O)CCc1csc(C)n1)NC 17746,C(=O)(C(F)(CNC(=O)C1=CCN(C)C1)C(C)C)N(C)Cc1cccc(C)n1 17747,N1(C(C2CC(=O)NC2)=O)CC(NC(c2cncnc2)=O)C(F)(F)C1 17748,CCCC(C)(C)C(=O)NCC(O)CCNC(=O)CNc1cccnc1 17749,c1(C(=O)NCC(CNC(=O)COCC2CCC2)CO)cc2c(s1)COCC2 17750,C(=O)(C1=C(Cl)CCCC1)NC12C(CN(C(C(C(C)C)n3cnnn3)=O)C1)C2 17751,CC(Cc1cn[nH]c1)CN=c1[nH]c2c(c(=NCC3CC3C3CCOCC3)[nH]1)SCC2 17752,C12(C(N(C3CCN(C(=O)CC4CCC4)CC3)C)=O)CCCC1CC(=O)CC2 17753,C1(CNC(C2(C(=O)NC)CCC2)=O)C2CCC(C2)N1C(c1ccc(C(N)=O)[nH]1)=O 17754,N1(C(C2C(C)C2(F)F)=O)CCN(C(c2cscc2C(F)F)=O)CC(C)(C)C1 17755,CC1CC(N(C(=O)C(=O)N(C)Cc2ccc(Cl)cc2F)C)CC(C)O1 17756,Cc1ccc(C(=O)NCCCCCN(C)C(C2(C)CC2C)=O)c2ncccc12 17757,N1(C(C2CC(C(=O)OC)C2)=O)CCC2CC12C(=O)N(CC(O)CO)C 17758,N1(C(C(=O)NCCCCCCCC)=O)CCc2sc(NC(=O)CCF)nc2C1 17759,CC1CN(C(C2CCCC(CF)C2)=O)C(C)CN1C(=O)CC1CSCCO1 17760,C1(C(=O)NCCCCCC=C)CCN(C(=O)C(C)(C)C(F)F)CC1C 17761,C(CCCC(C)(F)F)NC(CNC(C(c1ccnn1C)C)=O)=O 17762,CCCCC(C)C(=O)N1CC(CNC(=O)CCOCC)C(O)C1 17763,Cc1c[nH]c(C#N)nc1=NCCNC(C1COc2ccc(F)cc2C1)=O 17764,C1(CCNC(c2cccc(=S)n2O)=O)CCN(C(=O)C(O)C2CC2)CC1(F)F 17765,c1(C(=O)NC(c2cn(C(C)C)nn2)CCC)ccc(Cl)cc1-n1cncn1 17766,N#CC1CN(C(C2CCCN2C(=O)CC2CC(OC3CC3)C2)=O)CC12CCC2 17767,c1(C(N(CCCCCC)C(=O)CN(C)Cc2ccco2)=O)ccc(OC)cc1C 17768,CC(C)C(O)CC(=O)N(C1CCN(C(C23CSCC2C3)=O)CC1)C 17769,C1(CNC(c2nc[nH]c3ncnc2-3)=O)CN(C(=O)C(F)(F)C2CC2)CC12CCC2 17770,c1(C(c2n(CC)nnn2)NC(C2CCC2)C2CC2)ccc(OC)cc1[N+](=O)[O-] 17771,C1(NC(C=C(C)C(C)C)=O)CCCCC1CNC(c1ccno1)=O 17772,C1(C(=O)NC(CNC(c2ccc(C(F)(F)F)s2)=O)C2CC2)CCCCS1 17773,n1(CC)nnc2c1CCC(C(=O)NCC1CCN(C(C3COC(=O)N3)=O)CC1)C2 17774,c1(C(=O)NC2(CCNC(C3C(C(=O)OC)C3)=O)CC2)cccc2c1NC(=O)CO2 17775,C(=O)(C(CC=C)CC(C)C)NCC1C2CN(C(COc3ccc(C#C)cc3)=O)CC21 17776,c1(C(N2C(C(=O)NCC(C)CO)C=CC2)=O)cc(F)ccc1O 17777,C1(NC(c2ccc3occc3c2)=O)CN(C(C2CC2CF)=O)CC2(CCC2)C1 17778,n1(CC)cc(-c2ccc(CN(CCO)Cc3ccc(F)cc3)cn2)ccc1=O 17779,c1(C(N2CCC(NC(C3(SC)CCC3)=O)C(O)C2)=O)ccc(P(C)(C)=O)cn1 17780,c1(C(=O)NCCOCCC(=O)NCC2(SCC)CC2)ccc(C)cc1C 17781,C(=O)(CCS(=O)(=O)N(C1CCC(NC(=O)CCc2ncc(C)[nH]2)C1)C)OC 17782,O(NC(=O)C(C)(C)C1CCCN1C(=O)CN1CCCCC1)CC(=O)NC(N)=O 17783,C1(NC(C=Cc2nc(C)sc2)=O)CC(CNC(=O)CC2(O)CCC2)C12CCC2 17784,c1(OC)cnc(C(N2CCCC2CCNC(=O)C=C(C)C(C)C)=O)nc1 17785,N1(C(c2cn(CCC)nn2)C(=O)NC2CCCC2)C2CCC1CN(C)CC2 17786,C1(CC(=O)Nc2ccc(Br)nc2)COCCN1Cc1ccc(-c2ccccc2)s1 17787,CCCCC(C)(F)C(=O)N1CC(NC(C23CC(C)(C2)OC3(C)C)=O)C(O)C1 17788,C(=O)(C(CNC(=O)C1=CC2(CCOC2)C1)CC(C)C)Nc1c(COC)cccc1 17789,c1(C2(N(C(=O)Cn3cc(C(F)(F)F)cn3)C(C)C)CC2)ccnc2ccccc12 17790,C12(C(=O)OC)CCCCC1CN(C(c1c(OC)c([N+](=O)[O-])ccc1)=O)C2 17791,N1(C(C2C(OCC)C2)=O)CC2(C1)CN(C(=O)C(N1C(=O)CCC1=O)C)C2 17792,N1(C(CSCC(C)C)=O)Cc2ccccc2CC1CNC(=O)C(C)SC(C)C 17793,NC(=O)CCCC(=O)N1CCC(C2OCCC2Cc2ccccc2)CC1 17794,CC1CCN(C(=O)Cc2cncc(C(F)(F)F)c2)CC1c1ccc(F)cc1 17795,CCC(C)CCCCC(=O)NC(CC(=O)N(C)Cc1ncco1)C(C)OC 17796,CN1CCN(c2ccc(C(N3CC(NS(=O)(=O)CC4CC4)C(O)C3)=O)cc2)CC1 17797,c1(C(N2CC(O)CC(NC(CCc3nc(=N)[nH][nH]3)=O)C2)=O)[nH]nc([N+](=O)[O-])c1Cl 17798,c1(C(N2C(CNC(=O)CC3NC(=O)NC3=O)CCC2)=O)ccc(CO)cc1F 17799,N1(C(c2c(C)c[nH]n2)=O)CCCC(NC(c2ccsc2Cl)=O)C1C 17800,c1(C(N2C(C3(NC(C(CCSC)O)=O)CC3)CCCC2)=O)cc([N+](=O)[O-])c[nH]1 17801,CN1CCC(C(=O)NC2CCC3(CC3)C2)(NC(C2C=CCCC2)=O)C1 17802,C1(C(=O)NCCOCCCC#C)CCN(C(C2CC(C)CCO2)=O)C1(C)C 17803,C1(CNc2c(C)c(NCCC(N)=O)ncn2)CCC2(C1)CC2(F)F 17804,C1(C2CC2)(CNC(c2c(CCC)n[nH]c2)=O)CCN(C(=O)CC(C)(F)F)C1 17805,C(=O)(CCCC(c1ccccc1)NC(=O)Cc1cocn1)OC 17806,C(=O)(CCCC(F)(F)F)NC(CN(C)C)C(N1C2CCC1CC2)=O 17807,C1(F)(CNC(c2cccc(CCC)c2)=O)CCN(C(=O)C(F)=CC2CC2)CC1 17808,c1(Cn2cc(-c3c(C)ocn3)nn2)cccc(C(=O)NCC2CSCCS2)c1 17809,c1(NC(=O)NC2CCCN(C(C3CC(O)C3)=O)C2)ccc2nn[nH]c2c1 17810,C(=O)(CCCNC(C)=O)N(C1CCN(C(=O)CC(=O)N2CCOCC2)C1)CCC 17811,C1(F)(CNC(=O)CSC(F)(F)F)CC2CCC(C1)N2C(=O)CC1CS(=O)(=O)C1 17812,Cn1cnc(NCC2C(Cn3cc(CN4CCNC4=O)nn3)C2(F)F)cc1=O 17813,c1(C(=O)NC2C(CNC(C(COC)(F)F)=O)CCCC2)cnc2c(c1)CCC2 17814,c1(CC(=O)NCCC2CCC(NC(=O)C3=CCCC3)C2)cccnc1C(F)(F)F 17815,C1(C)(CNC(C2C3CN(C(c4nc(C)sc4C)=O)C2C3)=O)NC(=O)NC1=O 17816,S(=O)(=O)(c1cnc(C(C)C)[nH]1)N1CCC2(C(CC)C2)C1 17817,NS(=O)(=O)c1cc(C(N2CCC(NC(=O)C(F)(F)c3cscn3)C2)=O)ccc1Cl 17818,c1(C(N2CCC(CCC(C)O)CC2)C(=O)NC2CC2)ccc2c(c1)CCCO2 17819,c1(C(N2CCC(N3CCN(C(CCSC)=O)CC3)C2)=O)c(C)cc(O)nc1C 17820,N1(C(CCC(C)N(C)C)=O)CCC=C(C(=O)N2CCC(C)(C#N)CC2)C1 17821,Cc1ccc(CC(=O)NCC2CC(CNC(c3ccc(C(F)(F)F)s3)=O)CO2)o1 17822,c1(OC(CC)CC)ccc(C(=O)NCC2CC2CNC(c2cn(C)cn2)=O)cc1 17823,C1(C(=O)O)(COC)CCCS1(=O)=O.c12cn(C)nc1C(=O)NCCn1cc-2nn1 17824,c1(C(N2CC(COC)N(C(C3CCC(C)(C)O3)=O)CC2)=O)ccc2cc[nH]c2n1 17825,C1(NC(CC2(C(=O)OC)CC2)=O)CCCCN(C(C2CC(F)C2)=O)C1 17826,N1(C(CCCN(C(C)=O)C)=O)CCCC(C(=O)Nc2cccc(CF)c2)C1 17827,c1(NC(C2(C)CN(c3ncnc(C)c3Br)C2)=O)oc2ccccc2c1C 17828,C1(C(N(C)CC2CCC2)=O)CCCC1CNC(C1CS(=O)(=O)C1)=O 17829,C1(C)(C(=O)NC2(C)CN(C(=O)CC(C)(O)c3ccccc3)C2)CCCCNC1=O 17830,CC(C#N)C(=O)N(CC(O)CN(C(=O)CN(CCc1ccccc1)C(N)=O)C)C 17831,C1(CNC(CC(C)SC)=O)(CO)CCN(C(c2coc(C(N)=O)c2)=O)C1 17832,C#CCCCC(C)C(=O)NCc1ccc(C(N2CCCC(C)(C)C2C)=O)cn1 17833,N1(C(C(CC)(C)C)=O)CCN(C(C2CCCC23CCC3)=O)C(C)C1 17834,c1(C(=O)NC2(C)CC(NC(C3N(C(C)=O)CC(O)C3)=O)C2)cc(O)cc(C#N)c1 17835,Cn1cnc(C=CC(=O)NCC(=O)NC2COCCOC2)c1 17836,n1(CC)cc2ccc(C(N3CC4CCOC4(CNC(=O)CSC)C3)=O)cc2n1 17837,c1(C(=O)NC2CCCC(NC(C(C)(C)C3CCOCC3)=O)C2)c[nH]cc(F)c1=O 17838,c1(CN(C(=O)C(C2(O)CCCNC2)(F)F)C)nc2ccccc2n1C 17839,Clc1ccc(-c2cc(-c3nc(C4CC45CC5)nn3C3CCOC3)n[nH]2)cc1Cl 17840,c1(CNC(C2(C)C=CCC2)=O)cccc(NC(=O)CC2CCSC2)c1 17841,C1(C)(C(=O)NC(C)Cn2ccnc2)CCN1C(=O)COC1CCCCC1 17842,C1(C(=O)NC2(CO)CCN(C(C34CC(C)C3C4)=O)CC2)CN(CP(C)(C)=O)C1 17843,C12CN(CC1C)C(=O)C(C)n1cc2nn1.c1(NCCN(C)C)csc(C)c1C.CO 17844,c1(-n2cc(C3CN(C(C4C(CC)CCC4)=O)C3)nn2)cc(F)ccc1C 17845,N1(C(c2ccc(OC)cc2)=O)CCN(C(c2cc(OC)no2)=O)C(CF)C1 17846,c1(OC)cc(C(N2CCC(NC(=O)C=CC(C)(C)C)C(CO)C2)=O)ccc1C 17847,c1(C(N2C(C)CN(C(=O)C(N3CCOCC3)C)CC2)=O)cn2cnnc2cn1 17848,C1(CCNC(c2[nH]cc(C)c2C)=O)CCN(C(=O)C(C)n2ccnc2)CC1(F)F 17849,N1(C(C=CCN(C(C(=Cc2ccco2)C)=O)C)=O)CCC(F)(C(N)=O)CC1 17850,C(c1cccs1)=CC(=O)N(CC(CC)NC(=O)CC1CCOC1)C 17851,c1(C(=O)NCC2N(C(C(C=C)OC)=O)CC(F)C2)cc(C)c(C#N)c(C)c1 17852,C=CCC(C(=O)NC(C=C)CO)NC(=O)C=CC1CCCN1C 17853,C1(CNC(CSCC=C)=O)CN(C(C2COCOC2)=O)CCC1C 17854,CN1CC(NC(N2CCCC2c2ccc(Cl)nc2)=O)C2(CC2)C1 17855,C=C(C)C(C)(C)C(=O)NCCN(C)C(C1CCC(C#N)C1)=O 17856,CC1CC(C(=O)Nc2nccc(CSc3ccccc3)n2)CCN1C 17857,N#CC1(c2ccccc2)CC(c2nc(COc3ccccc3)no2)C1 17858,N1(C(COCCC=C)=O)CCC(CC)C1CNC(=O)CCn1ccnc1C 17859,C1(C(=O)NC2(CNC(c3ccc([N+](=O)[O-])s3)=O)CCOC2)Cc2nccnc2C1 17860,c1(NC(=O)C(C)(CO)CO)ccc(C(F)(F)F)cc1O.C12(CC)CN(C1)C2=O 17861,C1(CCC)CN(C(=O)C=CBr)CCN1C(C1CCC1(C)C)=O 17862,c1(CN(C(=O)CSCC(=O)Nc2ccccn2)C)ccc(Cl)cc1 17863,C(=O)(C1CCc2c[nH]nc21)NC1CCC(CC(=O)N(c2cccc(O)c2)C)CC1 17864,C1(C(=O)NCC2CCN2C(=O)C(F)(F)CC2CC2)CCC([N+](=O)[O-])CC1 17865,CCC(CCOC)NC(C1CC(NC(=O)C(F)OC(F)(F)F)C1)=O 17866,Cc1nc(O)nc(O)c1N(C)C(c1cccc(CN2CCCC2CN(C)C)c1)=O 17867,c1(CC=CC(=O)N(C(CNC(C=CC(CC)=CC)=O)C)C)ccccn1 17868,C1(C(=O)NCC(C)(C)NC(C(c2cccc(OC)c2)C)=O)OCCOC12CCC2 17869,N1(C(c2n(C(C)C)ccn2)=O)C2CCCC1CN(C(C1CCCS1)=O)C2 17870,CC1C(NC(C2(CN(C)C)CC2)=O)CCN1C(=O)CC(F)(F)F 17871,N1(C(CC(CC)OC)=O)CCC(C2(O)CN(C(C3(CO)CCC3)=O)C2)CC1 17872,N1(C(c2ccc(C)nc2C)=O)CCC2C(CCN2Cc2cc(Br)cc(Cl)c2O)C1 17873,CCC(C)CC(=O)C(=O)N1CCOC(C(=O)NCC2(C)C=CCCC2)C1 17874,N1(C(c2c(F)cccc2F)=O)CCCC2(C1)CN(Cc1cncnc1)CCO2 17875,Cc1csc(C(=O)NCC2(CNC(=O)C(F)F)CC2)c1Cl 17876,c1(C(=O)NC(CC=C)CNC(=O)Cc2csc(=N)[nH]2)nn(C)c(Cl)c1Cl 17877,C1(C(N(CCN(CC=C)C)CC)=O)C=CCN(C(=O)C(C)(O)C2CCC2)C1 17878,C1(NC(c2cn(C)nc2-c2ccoc2)=O)CCN(C(=O)C(Cl)=CCl)CC1F 17879,O=C1NCCCCC1C(=O)NC1CC(C(F)C(=O)NCCCc2nncs2)C1 17880,C1(O)(CC(=O)NCC(CC=C)NC(=O)CCc2cccnc2F)CCCCCC1 17881,N1(C(c2c(C(C)C)nns2)=O)CCC(CNC(C2(C#N)CC3CC3C2)=O)C(C)C1 17882,C1(OC)(OC)CCC1C(N1CCCC1CCC(=O)NCC(C)(C)F)=O 17883,c1(C(N2CCCC(c3ncc[nH]3)C2)=O)cccc(-n2cnnn2)c1 17884,c1(C(=O)NC(C)CN(C(=O)C(O)Cc2ccccn2)C)cnc2[nH]ncc2c1 17885,c1(C(=O)NC2CN(C(C(CSC)(C)C)=O)CC23CC3)ccn2ccnc2n1 17886,c1(NC(=O)C=Cc2ccc(C(F)F)o2)ccc2[nH]c(-c3ccco3)nc2c1 17887,C#Cc1ccc(F)cc1C(=O)NCC(C)(C1CCC1)NC(c1cn(CC)nn1)=O 17888,N1(C(CC)=O)CCCC(C(=O)NC(CNC(c2ocnc2C(F)F)=O)C2CC2)C1 17889,N(C1CC2(CC2)Oc2c(F)cccc21)C(C1(F)CC=CCC1)=O 17890,C12(CNC(CCC=C)=O)CC1CN(C(c1cc(C(=O)OC)sn1)=O)C2 17891,c1(SCC)cccc(CC(=O)NCC(CC)NC(c2ccc(C(F)F)nc2)=O)c1 17892,Cc1cc(C)c(C(N2CCC(NC(c3cn(C(C)(C)C)nc3Br)=O)C2)=O)cn1 17893,CCCCCC(=O)N(CCCNC(c1ccc(-c2nc(C)no2)cc1)=O)C1CC1 17894,N1(C(c2cc(C(=O)OCC)nn2C)=O)CCCC(CNC(C2CCSC2)=O)CC1 17895,C1(NC(Cc2ccc(C(C)=O)s2)=O)CN(C(c2ccccc2)=O)CC1C 17896,CC#CCCCC(=O)NCC1CC(NC(=O)Cc2noc(C)c2C#N)CC1O 17897,N1(C(C2C(C(C)C)C2)=O)CCC(C)(CCNC(c2cc(Cl)n(C)n2)=O)C1 17898,C1(NC(C2(C(C)=O)CC2)=O)CCC(C)(C)CC1CNC(=O)C(C)(C)c1ccns1 17899,C1(CC)CN(C(C2CC(SC)C2)=O)CCN1C(=O)CC1CC(C(=O)OC)C1 17900,N1(C(CC(CC#C)NC(c2cccc(C)c2C)=O)=O)CC2(C1)OC(=O)NC2C 17901,C1(CC)CCCN(C(=O)C(n2ccnc2C)C)C1C(=O)NC1COCC(C)(C)C1 17902,Cc1cc(C(N2CCC3(C2)CN(C(=O)C(C)C(F)(F)F)C3)=O)c(Br)c(C)c1 17903,c1(NC(C2N(C(CCc3ccc(C)cn3)=O)CC2)=O)ncc([N+](=O)[O-])cc1I 17904,c1(C(=O)NC(C(C)NC(C2CCOCC2(C)C)=O)CO)cc2cc(Cl)cnc2[nH]1 17905,c1(C(=O)NCC(CC)NC(C2CSC2)=O)cc2cc(C)c(Cl)cc2[nH]1 17906,CC1CN(C)C(C)CN1C(C1CC2CCC1N2Cc1ccc(C(=O)O)cc1)=O 17907,c1(C(N2CCC(C)(CNC(CC3C=NN(C)C3=O)=O)C2)=O)cc2ccncc2s1 17908,Cc1ccc(NC(=O)CC2CN(Cc3ccc(-c4ccc(C)s4)cc3)C2)c(O)c1 17909,c1(C(=O)NC2CCC(C)(CNC(C3C(C)=C3)=O)C2)cc(C)nc2onc(C)c12 17910,c1(C(=O)NC2C(C(N3CC(SC)C3)=O)COCC2)ncnc(O)c1F 17911,C1(C(=O)NCC2CC(NC(C(Cn3ccc(C)n3)C)=O)C2)CCC(=O)NC1 17912,C1(CC(=O)NCC2C(NC(COCC(C)C)=O)C2)CC(OC(C)(C)C)C1 17913,c1(OCC)ccc(CC(=O)NCC2(CNC(=O)CN(C)C3CC3)CC2(F)F)cc1 17914,c1(C(=O)NC(C(C)NC(C(CC#C)O)=O)(C)C)[nH]cc2c1CCCC2 17915,c1(C(N2C(CN(CCCC3CCOC3)C)CCCC2)=O)cc2sccc2[nH]1 17916,N1(C(C2C(C(C)(C)C)CC2)=O)CCC(O)(Cn2cc(C3(CO)CC3)nn2)C1 17917,C1(C)(N(C)CC)CCN(C(C2(N(C)C(c3cncnc3)=O)CC2)=O)C1 17918,CCCC(C(=O)OCC)N1CC2C(C1)N2C(=O)CCCO 17919,c1(CC(=O)NC2C(SC)CN(C(c3cnc(O)o3)=O)C2)ccc2c(c1)NC(=O)C2 17920,N1(C(CCSC)=O)CCN(C(C2(CO)CCC2)=O)CC1c1ccccc1Cl 17921,c1(OC)nc(Cl)ccc1C(=O)NC(C)CC1CN(C(=O)C(c2ccc(Cl)s2)C)C1 17922,c1(N2CCC(CC)CC2)[nH]c(=NC(CCO)CC(C)C)nc2c1ncn2C(C)C 17923,C1(O)(C(C(=O)NCC=C)NC(=O)C=CCC2(N(C)C)CCC2)CCCCC1 17924,C#CCC(CC(F)F)C(=O)N1CCC1C(=O)NC(=O)N(CC(=O)N(C)C)C 17925,c1(N(C(CNC(C(C(C)C)OC)=O)C)C)cc2nnc(-c3ccccc3)n2cn1 17926,C(=O)(C1Cc2c(Cl)cccc21)NCCC1(C)CCN(C(CCCOCC=C)=O)C1 17927,c1(NC(C=CC2N(C(CN3CCC(OC)C3)=O)CCC2)=O)ccc(Cl)nc1C 17928,N1(C(C(C=C)(C)C)=O)CC(NC(c2cc(C(C)C)on2)=O)CC2(CCC2)C1 17929,N1(C(c2n(CC)ncc2)=O)CCOC(C)(CNC(c2nn(C)nc2Br)=O)C1 17930,C1(CNC(=O)NC(C)COC(F)(F)F)Cc2ccc(F)cc2C1 17931,C12(C(N3CCC4(NC(=O)C=Cc5ccco5)C(C3)C4)=O)CCC(F)(CC1)CC2 17932,Cc1ccc(-n2cc(C(=O)NC(Cc3ccccn3)C(=O)O)nn2)cc1 17933,N1(C(C2N(N=O)CCC2)=O)CC(F)(F)CC1CCNC(c1ccccc1CO)=O 17934,C1(C(=O)NCC=CCC(N2CCC(C)C2)=O)C2C3CCC(C3)C12 17935,Cc1ccc(Cl)c(C(=O)NCC2CCCCN2C(=O)Cc2cc(C)ccc2C)c1 17936,c1(C(C)C)ccc(C(=O)NCC2C3CCC(C3)N2C(C2(C)CCOC2)=O)c(F)c1 17937,c1(C(N2CCC(C(=O)NCCc3c[nH]nc3C)(OC)C2)=O)cc2ccccc2o1 17938,c1(C(=O)NCC(CCCC)NC(=O)CCC(CC)OC)c[nH]c(=NCC)s1 17939,N1(C(C(CC)SC)=O)C(C(N2CCC(C(=O)OC)C2(C)C)=O)CCC12CC2 17940,Cc1ccncc1-c1cn(CC(N2CCCC(COc3ccccc3)C2)=O)nn1 17941,Cn1c(C(N2CCCC3C(=O)NCC23)=O)c(Cl)c2ccccc12 17942,N1(C(CC(=C)C)=O)CC2CC(NC(c3cc(OC)cs3)=O)C(C2)C1 17943,N1(C(COCCN(C)C)=O)CC(C)(NC(=O)Cc2csc(S)n2)C1 17944,c1(C(=O)NCCCCCNC(c2cncc(N)n2)=O)ccc(S(N)(=O)=O)cc1Cl 17945,c1(CC)cc(C(=O)NCCN(C(C2SCCC2C)=O)Cc2ccccc2)nn1C 17946,C1(C(=O)NC(c2cnc(C)s2)C)CCC(C)(C)N(C(=O)CC2=CCCCC2)C1 17947,c1(OC)ccc(OC)c(CCC(N2CC(NC(C3CCO3)=O)C(C)(C)C2)=O)c1 17948,N1(C(C=Cc2nc(C)sc2)=O)CCCCC1C1CCCN1C(=O)C(O)C1CCC1 17949,n1(C(C)C)cc(C(=O)NCCC(C)N(C)C(c2cc(F)n[nH]2)=O)c(Br)n1 17950,C(=O)(C(C)(C)C(=O)c1ccccc1)N(CCC=C)C(=O)CN(CCO)CCOC 17951,c1(C(=O)NCC(C)NC(c2n(C(C)C)ccc2)=O)cc(Cl)ccc1F 17952,C1(O)(CNC(COCC=C)=O)CCCN(C(=O)CO)C1.C12CCC1NC(=O)C2 17953,c1(C(N(CC(C)NC(c2cn(C3CCC3O)nn2)=O)C)=O)cc2ccsc2s1 17954,C1(C#N)(C(=O)OC)CC2CCC1CC2NC1CCCC1c1ccccc1 17955,C1(NC(CN(C(COC)=O)C)=O)CC2CC1CN(C(=O)Cn1ccnc1C)C2 17956,CC(C(=O)NCC1CCN(C(=O)Cc2cncs2)CC1CO)C(F)(F)C(F)F 17957,c1(C(N(C2CCCN(C(=O)C(O)C3CCCC3)C2)CC)=O)cc2cnccc2[nH]1 17958,C1(NC(C2N(CC#C)CCC2)=O)CC2(CCCN(C(=O)C(F)C(C)(C)O)C2)C1 17959,C=C1CC(C(F)(F)F)(C(=O)Nc2cc(COCCCF)on2)C1 17960,c1(C(C(=O)NCC(CO)NC(COCCC=C)=O)(F)F)ccc(Cl)cc1 17961,CNS(=O)(=O)NCC(=O)NCCOCCNC(=O)Cc1conc1C 17962,C1(CCC)CCCN(c2cccc(C(N3CCCC3)=O)n2)C1 17963,N1(C(CCCNC(=O)OC)=O)CC(O)CC1(C)C(N1CCC1CF)=O 17964,Cn1cccc(-c2cccc(C3CC3C(=O)Nc3ncc(Br)nc3Cl)c2)c1=O 17965,C1(O)(C(C)NC(C2C(CC)CCC2)=O)CCN(C(C2CN(C)C(=O)N2)=O)CC1 17966,n1(CC(C)N(C)C)cc(Br)c(O)nc1=O.N12C=CC(=NCc3cn1nn3)N2 17967,C(c1ccc(F)cc1)=C(C)C(N1CCC(C)(NC(=O)CN2CCCCS2(=O)=O)C1)=O 17968,c1(-c2cn(CC(CN)OC)nn2)ccc(C(F)(F)F)cc1Cl 17969,C(=O)(C(C)CC(F)F)NC(CN(C(c1ccc(C(N)=O)cn1)=O)CC)C 17970,N(C(=NCCCN1CC(C)OC(C)C1)N1CCN(C2CC2)C(=O)C1)CC(=C)C 17971,c1(C(N)=O)ccc(C(=O)NCc2cn(CCNC(N)=O)nn2)cc1 17972,C=CC(C)(C)CC(=O)N1CCC(CO)(NC(=O)C(CC2CCCCC2)CCC)C1 17973,Cc1ccn(C)c1C(N1CC(O)(C(C)NC(=O)CCc2ccnc(Cl)c2)C1)=O 17974,C(=O)(C1=CCC2CCC1N2C(=O)C(Cl)Cl)NC(C)Cc1ccco1 17975,c1(OC)cc(Br)ccc1C(c1nnnn1Cc1cccc(OC)c1)NCC(N)=O 17976,c1(OC)cc(-c2nc(-c3nc(C(C4CCC(C)CC4)C)no3)cs2)c(F)cc1O 17977,C1(NC(CCCC#C)=O)CCCC12CN(C(c1cccnc1OCCOC)=O)C2 17978,C1(NC(CCOCC#C)=O)CC2(C1)CC2NC(c1cnn(-c2ccccn2)c1)=O 17979,C1(CNC2CC(CNC3(CC(=O)OC)CCC3)C2)CCCC1C 17980,c1(C(=O)NCC2C(NC(CC(C=C)C)=O)CCCC2)ccc(C(F)(F)F)c(N)c1 17981,C1(NC(CCC2(C)CC2(F)F)=O)CN(C(=O)Cc2cccc(O)c2)CC1F 17982,c1(-c2scc(C)n2)ccc(C(=O)N(C2CN(C(C3(C)CCCN3C)=O)C2)C)cc1 17983,c1(CCC(=O)NC2(CNC(CCC(CC)C)=O)CCOC2)cnc2ccccn12 17984,N1(CC(=O)N(c2nc3ccccc3o2)CC)CCC(C2CC(F)(F)C2)C1 17985,c1(C(=O)NCC(c2ccc(C)cc2)NC(C2(C3CC3)CC2)=O)cnc2n1CCS2 17986,CC1CN(C(c2cn(CCNC(=O)C(C)(Cl)Cl)cn2)=O)CC1(C)CO 17987,C(=O)(CCCC(F)(F)CO)NC1C(SC)CN(C(c2c[nH]nc2[N+](=O)[O-])=O)C1 17988,N1(C(=O)Cc2ccc(Br)cn2)CCC(F)C(NCc2cc(O)cc(F)c2)C1 17989,N1(C(C2C(C)CCO2)=O)CCC(F)(C(N2CC(C3CCCO3)C2)=O)C1 17990,N1(C(C(C)c2ccco2)=O)CCC(O)C(N(C)C(c2cc3n(n2)CCO3)=O)C1 17991,CC1CC(C(=O)OCCNC(C)C=Cc2ccc(=O)n(CCO)c2)CC(=O)N1 17992,N1(C(C2(CC=C)CCC2)=O)CC(NC(c2cn(-c3ccccc3)nn2)=O)C(C)C1 17993,C1(CCNC(CC(C)F)=O)CCCCN1C(c1ccc(-c2cccnc2)cc1)=O 17994,c1(OC)ccccc1C(=O)NC1CC2(C1)CC2C(=O)NCc1c(C)n[nH]c1C 17995,CC1(C)C(CC(=O)NCc2nc(C3CC3)cs2)CCN1C(=O)CC1(C#N)CC1 17996,C1(C(=O)NC2C(NC(c3ccc(C)o3)=O)CCC2)CCCN(C(=O)C(C)(C)C)C1 17997,C1(C(N2CC(C#N)C2)=O)CC(OC)CCN1C(C1CC2CCC(C1)C2)=O 17998,c1(CN(C(C2(F)CCN(C(=O)OC(C)(C)C)C2)=O)CC)ccc(Cl)c([N+](=O)[O-])c1 17999,N1(C(C2(F)CN(C(CS(CC)=O)=O)C2)=O)CC(C)OC(C)(C)C1C 18000,c1(-c2cncc(OC)c2)ccc(CN2CCCC2(C)CO)c(C)c1 18001,C(=O)(C1(C)CCn2c(C)nnc21)N1CC(NC(c2ncc(C)cn2)=O)C(O)CC1 18002,c1(C(=O)NC2CCCC3CN(C(CCOC)=O)CC32)cccc(S(N)(=O)=O)c1C 18003,N1(C(c2ccc(C#C)c(Cl)c2)=O)CC(NC(C)=O)C2(CCOCC2)C1 18004,c1(NC(C2(C)CCN(C(C(C)(C)CCl)=O)CC2)=O)c(F)cccc1C#N 18005,Cc1cccc(C(O)C(=O)NC(C)CN(C(=O)CC2CC3C=CC2CC3)C)c1F 18006,C1(NC(c2ccc(N(C)C)cn2)=O)CC2CCC1C(NC(=O)C1=CCCOC1)C2 18007,C1(CC(N2C(CCNC(=O)C(F)C3CCC3)COCC2)=O)CC(=O)NC(=O)C1 18008,c1(C(N2C(CNC(c3ccn(C)c3)=O)CCCCC2)=O)c[nH]c2cc(O)ccc12 18009,N1(C(C(Cc2ccccc2)OC)=O)CCC2(C1)CN(C(=O)C(O)C(C)C)C2 18010,N1(C(c2cc(SC)c(C)o2)=O)CC(C)N(C(c2cn(C)c(C)cc2=O)=O)CC1C 18011,CCC1=NOC(C(=O)NCCCN(C(c2cnc(CC(C)(C)C)s2)=O)C(C)C)C1 18012,c1(CNC(C(CC)NC(C2CC(C)(C)CCO2)=O)=O)cccc(C#N)n1 18013,C(=O)(CC1c2ccccc2CCN1C(=O)C(=O)NC(C)C)N1CC(CC)OCC1 18014,N1(C(C2CCC(CCC)CC2)=O)C(CNC(c2cc(Cl)cs2)=O)CC2COCC12 18015,N1(C(c2ccc(C)cc2)=O)CC2(CC(NC(c3cnc(N)c(Br)c3)=O)C2)C1 18016,C1(Cn2cc(-c3c(CC)cccc3)nn2)CCN(C(=O)C(F)(F)Cl)CC1(F)F 18017,N1(C(C)=O)CCC(NC2(C(=O)N(C3CCN(C)C3=O)C)CC2)CC1 18018,N1(C(C(COC)C)=O)CCOC2(CCN(C(C3CC(=O)C3)=O)C2)C1 18019,c1(C(=O)NCCN(C)C(c2cc(C3CC3)ncn2)=O)cccc(C2(F)COC2)c1 18020,CCCC(CCC)CC(=O)NCC1CN(C(c2cnn(CC)c2)=O)CCC1C 18021,n1(CC(=O)NCCC(CNC(c2ccc(C)o2)=O)O)cc(Br)c(C)n1 18022,N1(C(C=NOC)=O)CC(CNC(=O)Cc2cccc(F)c2F)CC2(CCC2)C1 18023,CC1CCCn2cc(C(=O)NCC3CC3NC(C3CN(S(N)(=O)=O)C3)=O)nc21 18024,CCC(O)(C(=O)NCCCCC(C)NC(c1nc(C)cs1)=O)c1ccccc1 18025,N#CC1CCCCC1NC(C1(CCNC(C23CCC(C2)OC3C)=O)CC1)=O 18026,CN1CC(NC(C2CC23CC(NC(=O)CC2CCC(C)(C)O2)C3)=O)C(C)(C)C1 18027,Cc1cc(Cl)cc(Cc2nc(-c3ccc(C)c(C(C)C)c3)no2)c1O 18028,N1(C(C(C)OC(C)(C)C)=O)CCCN(C(=O)COC2CCCCC2)CC1 18029,c1(C(=O)NCC(CC(C)C)NC(c2c(C)ccnc2)=O)c(C)nc(O)nc1S 18030,n1(CC)nc(C(=O)NCC2CC2CNC(=O)CCCN(C)C(C)C)c(Br)n1 18031,c1(CC(N2C(CNC(C3(C#N)CCCO3)=O)CC2)=O)cc(F)ccc1Cl 18032,CC(C)CC(O)CNC(C1CCC(C2CC2)N1C(=O)CCn1cnc(=N)[nH]1)=O 18033,N1(CC)CCN(C(=O)CCC(=O)C(C)(C)C)C(=O)C12CCCC2 18034,N1(C(CC(C=C)CC)=O)CC2(C(=O)N(C)Cc3cncnc3)CC1CCO2 18035,c1(CC(=O)NCCC2(O)CN(C(c3c(C)coc3C)=O)C2)cccc(Cl)c1Cl 18036,C1(C(N(CCNC(C(c2ccc(OC)cc2)CC)=O)C(C)C)=O)CSCC(=O)N1 18037,C1(NC(c2conc2C2CCC2)=O)CCCN(C(C2CC=CCC2)=O)C1 18038,c1(C(N2CCC(C(C)NC(c3ncccc3F)=O)C2)=O)cc2nc[nH]c2cc1F 18039,C(c1ccc(C)c(C)c1)=CC(=O)NC(CCOC)CNC(=O)C(C)C1CC1 18040,c1(C(N(CC(C)N(C(C(CCC)CC)=O)C)C)=O)ccc2c(c1)CN(C)CC2 18041,C=CCC(C(=O)NCC1(CN(C)C(C2CCC3CC3CC2)=O)CC1)C(C)C 18042,C(=O)(C(C)(F)C(F)(F)F)NCC(C(C)C)(C)NC(C1CCN(C(N)=O)CC1)=O 18043,Cc1cc(Cl)cc(CNCC2OCCN(C)C2c2ccccc2)c1O 18044,C(C(CC(=O)NC1CCN(C(C2CCCS2)=O)CC1)C(F)F)N(C)C 18045,C1(NC(CCOc2c(CC)cccc2)=O)CCCCN(C(c2cnns2)=O)C1 18046,C=C(Cl)CC(C(=O)N1CCC1C)NC(c1nnn(C)c1C)=O 18047,C(=O)(C(C)(C)C(=O)NC1CCCN(C(c2cc(Cl)sc2Cl)=O)CC1)NC 18048,C1(NC(c2c(CC)oc(C)c2)=O)CN(C(=O)CC(C)N2CCCC2=O)CC12CC2 18049,C(=O)(C1=CCSC1)NCCC(CNC(CC(C)C)=O)O 18050,N1(C(CN(c2ccncc2)C)=O)CCC2CC1CN2C(c1csc(Cl)c1)=O 18051,CC1CC(C)N(C(=O)C2=CCCSC2)CCN1C(c1ccc(Cl)c(C#N)c1)=O 18052,N1(C(C2=CCCC2C)=O)CCC2CC(n3cc(C4CC4)nn3)CCC2C1.C1(Br)CC1 18053,C1(CCC(=O)NCCN(C(C)C)C2CC2)CCN(C(N2C(=O)CNC2=O)=O)CC1 18054,C1(NC(CCC#CC)=O)CCSC12CN(C(=O)CCOc1cccc(C)c1)C2 18055,C=CC1(C(N2CC(C(=O)NC)C2)=O)CCN(C(C2CC2C2CCC2)=O)CC1 18056,CC1(C)CC(NC(=O)CCN(C(=O)CCc2ccsc2)C2CC2)C1 18057,C1(C(=O)NCc2cn(CC(=O)Nc3cn(C)nc3)nn2)C2CCC(F)C12 18058,N1(CC(=O)NC2CN(C(C(C(C)C)F)=O)CC2C)CCc2ccccc21 18059,C12(NC(c3n(C)ccc3)=O)CN(C(C3CCOCC3)=O)CC1CS(=O)(=O)C2 18060,N1(C(c2ccc(NCC)cc2)=O)CCCC(F)(CNC(=O)CC2CC3(CC3)C2)C1 18061,Cc1ccc(NC(C2(CCNC(C34CC(C)(CCO3)C4)=O)CCC2)=O)cc1CO 18062,CCCCCCCC(=O)NCC(C)(O)CNC(C1CNC(=O)CC1(C)C)=O 18063,c1(C(N2CCCC(C(C)NC(C(C)N=[N+]=[N-])=O)C2)=O)ccc(O)c(F)c1 18064,c1(C(N2CCCC(C)C2CNC(C2(N(C)C)CCC2)=O)=O)cccc2ccnn12 18065,Cc1oc2ccccc2c1C(N1CC(NC(C2CCCCS2)=O)CC1(C)C)=O 18066,C1(NC(C(C)C)=O)CN(C(=O)C(F)=CCCF)CCC1c1ccc(F)cc1 18067,c1(CCC(=O)N(CC(C)O)CCNC(C(C)NC(C)=O)=O)ccc(Br)nc1 18068,C1(C(=O)Nc2cccc(C(F)F)n2)CC(O)CCN1C(c1cccc(Cl)c1Cl)=O 18069,Cc1ccc(C(=O)NCC2CN(C(C3CN(C)CC(C)O3)=O)CC2C)nc1F 18070,CC1CN(C(=O)C=CI)CC2(CCN(C(c3cc(O)nc(O)c3)=O)C2)O1 18071,C(=O)(CC(C)C(F)F)NCC1(CNC(c2c(C)cncc2)=O)CC12CCC2 18072,Cc1ccc(CCc2nc(-c3ccc(Br)cn3)nn2CCN(C)C)c(C)c1 18073,C1(NC(CC(=C)I)=O)CC(C)CN(C(c2ccc(C)nc2)=O)C1 18074,c1(-c2cn(C3CCN(C(C4CCCO4)=O)C3)nn2)ccc(Cl)c(Cl)c1 18075,CC(C)(C)CCC(F)C(=O)N1CCC(CCC(=O)NCCOCCCF)C1 18076,C1(N(C)C(=O)NCCc2nc(-c3ccccc3)no2)CCCCC1C(F)(F)F 18077,C1(C(N(C(C)C(=O)OC)CC=C)=O)CN(C(=O)C(C)c2cc[nH]n2)CC12CC2 18078,CCC(C)(CO)C(=O)NCC(F)CNC(=O)CN1CCOC1=O 18079,C1(C)(CC(=O)N(CC(=O)N(CCOC)CC2CC2)CCC)CC1(F)F 18080,C1(CNC(NCC(CC)CC(F)(F)F)=NCCF)CCC2(CCCC2)CC1 18081,C1(O)(C(=O)NCc2nc(CNC(CCC(C)OC)=O)sc2)CCCC(C)(C)CC1 18082,Cc1cc(C)c(C(N2CCC(=CCNCc3cnc(C4CC4)s3)CC2)=O)c(C)c1 18083,C1(CNC(C2(CC#C)CC=CCC2)=O)N(C(=O)Cc2cnsc2)CCC1(C)C 18084,C1(NC(C2(Cl)C(C)(C)C2)=O)CCCN(C(c2nc(=N)cc[nH]2)=O)C1 18085,c1(C(N(C)CC2N(C(COCCC#C)=O)CC(F)C2)=O)cc2c(C)cccn2c1 18086,c1(C(C)=O)csc(C(=O)NCC2(O)CN(C(C3CC3(C)C)=O)C2)c1 18087,N1(C(CC(C)OC)=O)CC(CNC(=O)CN(C(=O)C(C)C)C)C2CCCC12 18088,N1(C(C(=O)NC(C)C)=O)CC(NC(=O)C(c2ccccc2Cl)O)CC12CCC2 18089,C1(NC(C(C)=C2CCC2)=O)CC(F)(F)CC1NC(c1ccc(-c2ccco2)o1)=O 18090,c1(OC)cc(N(C)CCN(C)C(C2CCOC(C(C)C)C2)=O)nc(C(F)(F)F)n1 18091,c1(C(=O)NC2C(CNC(=O)CCC3CCCCO3)CCC2)cc(Cl)cnn1 18092,C1(NC(n2c(C)cnc2)=O)CN(C(C2CCCN2S(C)(=O)=O)=O)CC1C 18093,S(=O)(=O)(c1ccc(F)cc1)NCCC(=O)N(c1ccccc1)CC(C)C 18094,c1(NC(C2(SC)CN(C(c3cc(O)nc(O)n3)=O)C2)=O)cc(C)cnc1C 18095,c1(C(=O)NCC(CN(C(CC(C=C)C)=O)CC)(C)C)cc2cccnc2o1 18096,C1(NC(COCC(N2CCCC2)C)=O)CC2CC1N(C(c1cnnc(O)c1)=O)C2 18097,c1(NC(c2ccc(C(=O)NC34CC(C(=O)O)(C3)C4)cc2Cl)=O)cccc(Br)c1Cl 18098,C(=O)(C(C)(C)C(C)NC(C1CCNC1=O)=O)NC1(C#C)CCOC1 18099,C(=O)(CC(C(F)F)NC(=O)CC1CCSC1)NCCCCC 18100,C(=O)(C1=CCCCO1)N1CC(NC(c2c(C)oc(C(F)(F)F)n2)=O)C2C1C2 18101,CC1(C)CC(C(O)CNC(=O)CNC(c2cccs2)=O)C1 18102,C1(C(=O)NCCCC(C)NC(C2(C(=O)NC)CC2)=O)CN(C(C)C)CCO1 18103,Cc1nc2c(Cl)cccc2cc1C(=O)NC(CNC(C1CNC(=O)N1)=O)C1CC1 18104,c1(NC(C(N2CCC(C(=O)OC)(C(=O)OC)C2)=O)=O)c(C)cc(Cl)nc1I 18105,C1(CC(=O)OCC)CCCCC1(O)CNc1cccc(-c2ccccc2C)c1 18106,C1(NC(C2CCCC2)=O)CCOC12CCN(C(C1COC3COCC13)=O)CC2 18107,c1(C(=O)NCC(CNC(C(C=C)O)=O)CO)ccc2c(c1)OCCC2 18108,C1(CNC(C2N(CC)CCC2)=O)CCCN(C(=O)CCC(C)(C)N(C)C)CC1 18109,N1(C(C2CC(=O)NC2)=O)CCOCC(F)(CNC(C2CC2c2ccsc2)=O)C1 18110,c1(C(=O)NC(C(C)NC(CCN(C(CCC)C)C)=O)C)cc(C)nc(O)n1 18111,c1(OC)ccc(CC(=O)NCC2CC2NC(=O)CSc2nncn2C2CC2)cn1 18112,N1(C(C(=O)Nc2c(C)noc2C2CC2)=O)CCC2(CCOC2=O)C1 18113,CCCCCCCCC(=O)NC(c1cccnc1)C(=O)NCc1cnc[nH]1 18114,N1(C(c2ncc(C(F)(F)F)[nH]2)C(=O)NCCCC)CC(OC)CC(O)C1 18115,C(=O)(C1CCC(=O)c2cccn21)N1CCN(C(C2C(C)C2C)=O)C(CO)C1 18116,N1(C(=O)OC(C)(C)C)CCCCCC(NC(=O)NCC2CC23CC3)C1 18117,N(C(=NCCCP(C)(C)=O)NCCSC)CC(c1cc(OC)cc(OC)c1)(C)C 18118,C1(CNC(C2CCC(OC)CC2)=O)C2CCCC1N(C(=O)CC(C)SC)C2 18119,CN1CCC(C2(C(=O)OCC(C)(C)CC(F)(F)F)CC2)CC1 18120,CC1CCC(CNC(=O)Cc2ccno2)CN1C(c1cccc(C(F)F)c1F)=O 18121,N1(C(C(Cc2cc[nH]n2)NC(C2CN(C)C(=O)C2)=O)=O)CCN(C)C2(CCC2)C1 18122,c1(C(=O)NC2(CO)CN(C(C3OCC(C)C3)=O)C2)ccc(C#N)c(O)c1 18123,CCC(C(C)CN(C)C)NC(=O)C(Cc1cc[nH]n1)NC(=O)CCc1ccco1 18124,c1(C(=O)N(c2ncncc2I)CC2(F)CNC2)ccc(Cl)c(F)c1 18125,C(=O)(C(O)P(C)(C)=O)N1CCCC(NC(CS(N2CCC(C)CC2)(=O)=O)=O)C1 18126,c1(OC)c(C(=O)NC(C)CCCCNC(c2c(C)ncn2C)=O)cc(F)cc1F 18127,CC1(C)CC(C(=O)O)CN1Cc1cc(C#N)ccn1 18128,C1(C(C)NC(C(CC)N(C)C)=O)CCCN(CC(=O)Nc2cnccn2)C1 18129,N1(C(C2CC(C(C)C)C2)=O)CCCC(C)(CNC(C2(C)CCCCO2)=O)C1 18130,c1(SCCNC(N2C(c3scc(C(=O)OCC)n3)CCC2)=O)cccc(Cl)c1C 18131,c1(C(N2CC(NC(c3c(NC)nccc3)=O)C2)=O)ccc(-n2ccnc2)cc1C 18132,N1(C(Cc2nc(C)sc2)=O)CC2(CNC(C3CCSC3)=O)CC1CO2 18133,O=C(C1=Cc2cc(Cl)ccc2OC1)NC1C2CC1N(C(=O)COC(F)(F)F)C2 18134,CC(C)C(C(=O)NC(C1(C)CN(C(=O)C(=O)NCC2CC2)C(C)(C)C1)C)C(C)C 18135,C1(NC(=O)OC(C2CCCCO2)CC)CCC(OC)CC1OC(C)(C)C 18136,C(=O)(C(C)CC(F)F)N1C(C=CC(=O)N(CC)Cc2cn(C)nn2)CCC1 18137,C1(C(=O)NCCc2cc(C(=O)NCC3CCSC3)no2)C2CCC(=O)C12 18138,N1(C(CC(C)OC)=O)CCC2(CCCN(C(c3scc(Cl)c3Cl)=O)C2)C1 18139,C(C(C)(O)C(C)CC)NC(C(C)NC(C1(CC#C)CCCO1)=O)=O 18140,Cc1ncsc1C(=O)NCC(O)CN(C(C1CCC1c1ccccc1)=O)C(C)C 18141,C1(C(C)=O)CCN(C(=O)C(=O)N(C(c2ccccc2)CC2CCOCC2)CC)C1 18142,c1(C(N2CC(CCCCNC(CCC=C)=O)C2)=O)nnn(COCC)c1N 18143,c1(C(=O)NC(CC(C)NC(CNC(=O)NC)=O)C)cc(C(C)C)ccc1F 18144,CN1C2CC(O)C1CC(c1nnnn1C1CC1)(NCC1CCOC1=O)C2 18145,N1(C(COCC(=C)C)=O)CC=CCC1C(=O)NC1CC(C)OC1=O 18146,C(=O)(CC(O)C(C)CC)NC1(CC=C)CCN(C(=O)CC2OCCO2)CC1 18147,C(=O)(CC(CNC(=O)C(C(C)C)NC(=O)N(C)C)c1ccc(Cl)cc1)OC 18148,n1(CC)nncc1C(=O)NC(C)C=CC(N1CCC(N(C)C)C1)=O 18149,c1(C(=O)NCCC2CCN(C(C3C(C=C)C3)=O)C2)c(-n2cccc2)sc(C)c1C 18150,C1(S(C)(=O)=O)(CNC(c2c(SC)cc(Br)cc2)c2nnnn2C(C)C)CCCC1 18151,OCCC#CCN=c1ccnc(NCCn2cc(Br)ccc2=O)[nH]1 18152,N(C(=NCCC)NCC1CC1C1CCCO1)CC.c12cccc(c1)C1CC1N2 18153,c1(-c2ccc(-c3n(CCOC=C)ccn3)s2)ccc(CCO)nc1 18154,c1(CC)nc(C(=O)N(CC(N2C(CO)CC2C)=O)CC2CC2)co1 18155,N1(C(c2c(COC)cco2)=O)CC2CC1CN2C(c1cc(C(C)C)on1)=O 18156,CC1CN(C(C2CCCC2CNC(C2CC(O)CN2C)=O)=O)CCS1 18157,Cc1nc(Cl)ccc1CC(N1CC(OC2CCN(C(=O)C(C)C3CC3)CC2)C1)=O 18158,c1(C(=O)NCCN(C(C2CN(C)C(=O)N2)=O)CC)cc2[nH]ccc2s1 18159,C1(CNC(c2c(C)coc2C)=O)CC(C)(C)CCC1NC(=O)CC1CC(F)(F)C1 18160,c1(C(=O)NC2(CO)CCCN(Cc3ccccc3)C2)cccc([N+](=O)[O-])c1O 18161,C1(NC(C(CC)(C)C)=O)CC2CN(C(=O)C=Cc3ccn(C)c3)CC2C1 18162,C1(NC(c2ccc(CC)[nH]2)=O)CCCC(CNC(c2cn(C3CC3)nn2)=O)C1 18163,N1(C(CSCCOC)=O)CC=C(C(=O)NC2(CO)CCOC2)C1 18164,C(C(C)(C)CN(C)C(c1ccc(CSC)o1)=O)NC(CSCC=C)=O 18165,C1(C(=O)NC2CC(N(C(c3ncn(CC)c3)=O)C)C2)CC(C(C)C)=NO1 18166,c1(C(=O)NCc2ccnc(-n3cccn3)c2)cc(F)c2c(c1)OCCO2 18167,O=S(=O)(c1[nH]c(=NCC(O)c2cccnc2)ccc1Br)NC1CC2(CCC2)C1 18168,N1(C(C(C)C)=O)CC2CCOCC2(NC(=O)CCOCC(F)(F)F)C1 18169,C(=O)(CCCC(C)(C)C)N(C1CCN(CCC2CCCCO2)CC1)CCC 18170,C1(NC(c2ccc(OCCCOC)cc2)C)CCCC(C)(C)C1 18171,c1(C(=O)NC(CCC)CNC(c2cnc(COC)s2)=O)cncc(Cl)c1 18172,C1(NC(C2C=C(C)CS2)=O)CCC(C)(CNC(=O)Cc2csnn2)CC1 18173,N1(C(c2nccc(C(F)F)n2)=O)CCCCC2(CCN(C(C3CC3(Cl)Cl)=O)C2)C1 18174,c1(C(N2CCC(NC(COCCC(C)C)=O)(CF)C2)=O)nnn2c1CCCC2 18175,CCC(C)(CCC(C)C)C(=O)N1CC(NC(=O)CCc2cnn(C)n2)C2(CC2)C1 18176,c1(CC(=O)NC(C(C(C)C)NC(=O)OC(C)(C)C)C)cnc(O)nc1O 18177,C1(C(N(CC(CO)CC(C)C)CC)=O)CCC2(CCN(C(=O)OC(C)(C)C)C2)C1 18178,N1(C(C(C(=O)OC)OC)=O)CCCC2CCCC12 18179,CC1(C)CC(C(=O)NC2CC2NC(c2cnc(-c3cccs3)s2)=O)=NO1 18180,c1(CC(=O)NC2CC3(C(NC(CCCC#C)=O)C3)C2)c(C)nc(CC)nc1C 18181,c1(OC)ccc(CC(N2CCC(NC(C3(O)CCSCC3)=O)C(O)C2)=O)cc1Cl 18182,N1(C(c2cc(CNC(COCCCCC)=O)[nH]n2)=O)CCCC(C)C1CO 18183,O=C(NOCC1CCCOC1)C(=O)NC1CCCCC1 18184,CCCC(CC)CCC(=O)NCCC1(O)CCN(C(c2cc(F)cc(Cl)c2)=O)C1 18185,CN1CC2CC1CN2C(=O)C(=O)NC(CN1CCCC1c1cncc(Br)c1)(C)C 18186,C1(NC(=O)C(=Cc2c[nH]cn2)F)CCCN(C(C2CC3(C2)CC3F)=O)C1 18187,c1(C(N2C(CCC(=O)Nc3ccnc(F)c3F)CCC2)=O)ccnc([N+](=O)[O-])c1 18188,Cc1cc(C(=O)OCc2cnoc2C2CC2)nnc1C 18189,C1(c2nc(C(F)(F)F)no2)(CC=C)CCN(C(n2cnnn2)=O)CC1 18190,N1(C(CCc2nnc(C)n2C)=O)CCC(CNC(=O)C(C)C2CCC2)C12CCC2 18191,N1(C(c2c(OC)nccc2)=O)CCN(C(=O)C(C)c2cc[nH]n2)CC12CC2 18192,C1(C(N2C(CC)CN(C(=O)C(O)CC(C)C)CC2)=O)COc2cc(F)ccc2C1 18193,N1(C(c2n(C)c(O)nc2)=O)CC(NC(C2CC2c2ccc(Cl)s2)=O)CCC(O)C1 18194,CCC(CCCC(=O)NOCc1ccccc1)NC(C1CC2(CC2)C1)=O 18195,Cc1csc2ncc(C(=O)NCC3CCCN(C(C4CNC(=O)C4)=O)C3)c(=O)n12 18196,C1(N(C(C)=O)C)CCCCC12CCCN(C(=O)C1CC1)C2 18197,c1(CCC(N2CC3(CN(Cc4cncc(C)n4)C3)C2)=O)c[nH]c2ccc(F)cc12 18198,C(CC(=O)NC1(C)CCCC1(C)C)(C(C)OC)NC(CC=CCCCCC)=O 18199,c1(CC)oc(C)cc1C(=O)OCc1ccnn1C(F)(F)F 18200,N1(C(CN(S(CC)(=O)=O)C)=O)CCC2(CC1)CC2CNC(=O)CC(C)CN(C)C 18201,CC1C(=O)N(C)CCN1Cc1nc(-c2sccc2CO)cs1 18202,N1(C(CN2C(C)CCCC2)=O)CCC(NC(=O)CC2CCC(=O)NC2)C(C)(C)C1 18203,N#Cc1cc(N2CCCC2CNC(c2cccc3c2ncn3C)=O)ccc1[N+](=O)[O-] 18204,C=C(C)CCC(=O)NC1CCCC1NC(=O)CCC(=O)c1ccccn1 18205,c1(C(N2CC(C)N(C(=O)CC3CCC4CC4C3)CC2)=O)cc2ncccc2[nH]1 18206,C1(C(=O)NCC(C)(C)NC(Cc2c(C)noc2)=O)CCS(=O)(=O)C1 18207,C1(NC(C(=O)OCC)=O)CCC(CCC(=O)NCCSCC(N2CCCC2)=O)C1 18208,C1(CCOC)CN(C(C2CCCN2C)=O)CCN1C(=O)CP(C)(C)=O 18209,N1(CCCCC(C)C)CC2(CCC(CNC(C3CCCCO3)=O)O2)C1 18210,C1(CNC(c2[nH]cc(CC)c2)=O)(OC)CCN(C(C2CC(=O)N(C)C2)=O)CC1 18211,c1(C(=O)NCC2(F)CC(NC(C(C(CC)C)O)=O)C2)cc(F)cc([N+](=O)[O-])c1 18212,N1(C(c2c(C)cc(O)cc2)=O)CCN(C(=O)CCCN=[N+]=[N-])CCC1C 18213,C(=O)(NNC(=O)C(C)(C)CCCCNC(c1cccnc1)=O)c1c(C)ccs1 18214,n1(CCNC(C(C)C2CCCC2)=O)cc(C(=O)NC2(C)CSC2)cn1 18215,CC1(C)C(C)(C)C1(F)CC(N1CCN(C(c2cnc(Cl)c(Cl)c2)=O)CC1)=O 18216,C1(NC(CC(C)(C)C2CCCCC2)=O)CCN(C(=O)CCCC#N)CC1O 18217,N1(c2ncnc(C)c2Br)CCC(F)(F)C(C(=O)NC2CCCC(O)C2)C1 18218,c1(NC(C)=O)ccccc1C(F)(F)C(=O)NC1CC(C)N(C(=O)CC(C)C)C1 18219,C1(C(N(CC(C)(C)NC(=O)CC(F)(F)Cl)C)=O)CCCC1S(C)(=O)=O 18220,c1(C(=O)NCCOCCOCC(=O)NCCCNS(CC)(=O)=O)ccc(O)nc1 18221,c1(NC(C2N(C(c3c(C)cnnc3)=O)CC=C2)=O)ncc(Br)c(C)c1[N+](=O)[O-] 18222,N1(CC(=O)NCCc2c(Cl)cccc2Cl)CCC2(CC(=O)NC2=O)C1 18223,c1(CC(=O)NC2C=CCN(C(C(C)Oc3ccccn3)=O)C2)c(Cl)cccc1Cl 18224,N1(C(c2c(OC)c(Cl)ccc2)=O)CCN(C(C2CC=CC2)=O)C2CCCCC2C1 18225,C1(C(=O)NCC2C(CNC(Cc3c(C)cnn3C)=O)C2)CC2CC(=O)C1C2 18226,C1(C(N(CC)CC2CCCN2C(=O)CC#N)=O)Cc2cccc(F)c2O1 18227,N1(C(c2cc(-c3ccc(C)o3)[nH]n2)=O)CCC(C(N)=S)CC1 18228,C1(CC)CCN(C(=O)CC2CN(C(c3cc(C)[nH]n3)=O)C2)C1CNC(C)=O 18229,c1(CC(=O)NC(CC)CNC(C2(C)C=CCC2)=O)ccc(OC)cc1Br 18230,C1(=O)CC(C)C(=O)N(C2CC2)CC(=O)N(C)CC(=O)O1.C(C)(C)(C)NCC 18231,Cc1cc(Br)cnc1C(c1nnnn1C1COC1)NCCC1CCC(C)(C)C1 18232,CCC(CN(C)C(c1cnsn1)=O)NC(C1CCCO1)=O 18233,S(=O)(=O)(CC(=O)NC1COCC1CNC(c1c[nH]nc1OC)=O)N(CC)CC 18234,Cc1ncc(C=CC(=O)NCC2CCN(C(C3(O)CCOC3)=O)C2)c(O)n1 18235,c1(C(N2C(C3(NC(Cc4nc(C)[nH]n4)=O)CC3)CCC2)=O)nc(O)c(C)s1 18236,N1(C(C2N(C)CSC2)=O)CCCC(c2cn(-c3ccn(CC(F)(F)F)n3)nn2)C1 18237,N1(C(C(N2C(=O)CCC2=O)C)=O)CCC2(CC1)CC(NC(=O)CC(C)(C)C1CC1)C2 18238,c1(C(=O)NC2C3(CC(NC(C(CCC)OC)=O)C3)C2)ncc(C)nc1OC 18239,Cc1cccc2c(C(N3CC(C)CCC3CNC(=O)CC(F)(F)F)=O)nccc12 18240,C=CC1(C(=O)NC2(CC3CC3)CC2)CCN(C(C2CC=CC2)=O)CC1 18241,C=CCC(CO)NC(=O)COCCNC(C1CC12CC2)=O 18242,C1(NC(C(C)Oc2cccnc2)=O)CC(C)N(C(=O)CCC2CC2(F)F)C1 18243,c1(NC)cnccc1C(N1CCC(NC(C2(C)COCCO2)=O)C1C)=O 18244,c1(C(N)=O)cccc(OCC(N2CC=CC(NC(c3ccc[n+]([O-])c3)=O)C2)=O)c1 18245,c1(OCC)cc(C(N2CCC(CNC(=O)C3=CCC(C)CC3)C2)=O)cc(Cl)c1O 18246,C1(NC(c2cc(C)c(O)nc2)=O)CC2CCC(C1)N2C(C1(C)CC1(C)C)=O 18247,CCCCCC(CC)C(=O)N1CCC(CNC(=O)CCC2CC2)(COC)CC1 18248,N1(C(CCc2cncc(C)c2)=O)CC2CN(C(c3ccc(C)nn3)=O)CCC12 18249,C(=O)(CC(C(C)OC)NC(c1ccc(O)cc1F)=O)NCCCCCC=C 18250,c1(CN2CC3C(C(=O)NCc4ccc(F)cn4)C3C2)cccc(O)c1F 18251,C1(C(=O)NCCC(CNC(c2cn(C)nc2O)=O)O)CCC(=O)CC1(C)C 18252,N1(C(C2C(C)OCC2)=O)CCC(NC(=O)CSc2cnn(C)c2)C12CCC2 18253,c1(C(N(C2CC(NC(C3(C)CS(=O)(=O)C3)=O)C2)C)=O)cc2c(cc1O)CCCC2 18254,c1(OCC)ncc(C(=O)NC2CC(CNC(c3ncn(C)n3)=O)C(O)C2)cn1 18255,Cc1cc(C(N2CC3C(CN(C(=O)Cc4ccco4)C)C3C2)=O)cc(C)c1N 18256,C(=O)(C(C)P(C)(C)=O)N(CCOC)CCNC(=O)Cc1c[nH]ccc1=O 18257,CC1CCN(C(c2scnc2C2CC2)=O)CC1CNC(=O)C=Cc1ccsc1 18258,C1CCCCCN=C2C=CC(=CN2)S(=O)(=O)N1CC(C)C.C(C(C)(C)C)SC 18259,C(=O)(CCC(F)(F)C(F)F)NC1C(NC(C2OCCN(CC)C2)=O)CC1 18260,Cc1ncc(CC(=O)NCCCCCNC(C2(C)CC2F)=O)[nH]1 18261,C1(CC(=O)N(C)CC2CCCN(C(c3c(C)nc(O)[nH]3)=O)C2)CCCCC12CC2 18262,N1(C(c2c(CC)ncs2)=O)CCOC2CCN(C(=O)C(C)c3ccsc3)CC12 18263,c1(C(=O)NCCN(C(CC(C)OC)=O)CCCN(C)C)csc(C)c1C 18264,c1(OCCOC)cc(F)ccc1NC(=O)CCN1CCSC1=O 18265,c1(C(CC)=O)cc(C(N2CCC(CCNC(C3CC4CC3C4)=O)C2)=O)ccc1F 18266,c1(OCC(C)O)ccccc1NC(=O)NCC1CCCC(C(F)(F)F)C1 18267,n12cc(nn1)C2.c1(C(N2CC(N(C(C)C)C)C2)=O)cc(C(N2CCCC2)=O)c[nH]1 18268,C1(O)(CNC(c2ccc(C(F)F)nc2O)=O)CCCN(C(C2(F)CCOC2)=O)C1 18269,C1(n2ncc(NC(N(C(CC)(C)CC)Cc3cccs3)=O)c2)CCN(C)CC1 18270,C1(NC(=O)CCOC2CC2)COC2(CCN(C(=O)CCN3CCOCC3=O)C2)C1 18271,Cc1ccc(C(=O)NC2CC3CN(C(C4(F)CCCC4)=O)CC23)c(C(C)C)n1 18272,C(=O)(CCCCCC#N)N1C(C)(C)CC(NC(C2CC23CCC3)=O)C1 18273,c1(C(=O)NCCCCC2CN(c3c(C)cnc(C)n3)C2)cc(C)c(C)cc1Cl 18274,c1(C(=O)NC2C(C=C)CN(C(=O)CCSCC)C2)ccc2nc(S)oc2c1 18275,N1(C(c2ccccc2Oc2cccnc2)=O)CCN(C(C2CC2F)=O)C(CF)C1 18276,c1(C(=O)NC(C(C)NC(C2(CC)COC2)=O)C)cccc(P(C)(C)=O)c1 18277,C1(C(=O)NC(CC=C)CO)CN(Cc2ccccc2C(=O)O)CCS1 18278,c1(C(=O)NCCOCCCNC(C2(C)CC2(F)F)=O)cc2ccncc2s1 18279,N1(C(CCOc2cn(C)nc2)=O)CCN(C(c2cnn(C)c2)=O)CC12CCC2 18280,N1(C(C2(CC)CC2(F)F)=O)CCC(C2(NC(C3CCCCCC3)=O)CC2)C1 18281,c1(C(N2CC3C(NC(=O)C4=CCCC4)C3C2)=O)ccc2c(c1)C(=O)NCCO2 18282,N1(C(C(C)O)=O)CC2(CC2C(=O)Nc2ccc(N3CCCCC3)nc2)C1 18283,C1(C(N2C(C(=O)OCC)CCC2)=O)CN(Cc2csc(Cl)n2)CCO1 18284,N1(C2CN(CC(=O)NCCC)C2)CC(Cc2nnnn2CC)CC1=O 18285,c1(C(=O)NC2C(CC)N(C(=O)C(CC)(CC)OC)CC2)cncc(F)c1C 18286,C1(CN(C(c2c(OC)csc2)=O)C)COCCN1C(=O)CCCc1n[nH]c(=N)s1 18287,N1(C(C(C)(CO)NC(C2CC(C(=O)OC)C2)=O)=O)CCCC(C)(C#N)C1 18288,S(=O)(=O)(c1cccc(Br)c1)N1CC2(CCN(C(C(CC)c3ccccc3)=O)C2)C1 18289,c1(OC)cc(CN2CC3CCC2CN3C(c2c(O)cccc2F)=O)cc(F)c1O 18290,CCC(O)C(C)(C)C(=O)NOCC(N1CC2CCC2(C(=O)OC)C1)=O 18291,C1(CC)CNC(=O)CN1C(C1CC=CCN1C(=O)C(C)NC(C)(C)CC)=O 18292,N1(C(C2C(C)OC(=O)N2)=O)CC2CN(C(C3CCC3)=O)CC2(C(F)(F)F)C1 18293,c1(C(N(C2CCN(C(C3CCC3(F)F)=O)C2)CCC)=O)ccnn1CC 18294,CCC(C)(C)C(O)C(=O)NCCCN(C)C(C1CC1c1ccoc1C)=O 18295,c1(C(C)C)nocc1C(=O)NC1CC1CNC(=O)C(C)CC1CC1 18296,C(=O)(C(CCCCSC)N(C)CCOCc1ccccc1C)NC 18297,C1(O)(C(=O)NCCC2(C(=O)OC)CCCC2)CCNCC1 18298,C1(C(=O)NC)CCC(C)N1C(=O)OC(C)(C)C.n12cnc(c1)NCC2 18299,Cc1nn(C)c(Cl)c1C=CC(N1CC(CNC(=O)Cn2ccc(O)nc2=O)C1)=O 18300,N1(C(C2(NC(c3n[nH]c(O)n3)=O)CSC2)=O)CC2(C1)NC(=O)NC2=O 18301,c1(OC)cccc(CCCN(C)CC2CCCN(C(c3cncn3C)=O)C2)c1 18302,C1(C(=O)NCCN(C(=O)CCCc2cccnc2)CC)CCCC(N(C)C)C1 18303,CC(CCNC(=O)COC1CCOC1)CCNC(c1nc[nH]c1C(C)(C)C)=O 18304,c1(SCC(=O)NCCN(CCC)C(c2nocc2C(C)(C)C)=O)ccccc1F 18305,c1(C(=O)NCCC(C)NC(C2(COC)CCOCC2)=O)ccc2nc(C)sc2c1 18306,C1(CC(=O)NCCCCNC(C2CC(CC(=O)OC)C2)=O)CCCC(=O)N1 18307,C1(NC(c2n(CC)ncn2)=O)CCC2CN(C(c3nccnc3N)=O)CC2C1 18308,c1(CC(=O)N(CCN(C(C(C=C)(C)O)=O)C)C)ccc2ncsc2c1 18309,CC(C)CC(CC(C)C)C(=O)NC1CC1NC(C1(Cl)CC1)=O 18310,N#Cc1cc(F)ccc1-c1cccc(-c2nc(C(N3CCCC(O)C3)=O)cs2)c1 18311,CC1C(C)N(C(=O)C=Cc2ccccc2F)CCN1C(c1nnc(O)nc1O)=O 18312,Cc1c(C(N2CC(=O)CC2C(=O)NC(CC2CC2)C2CC2)=O)nnn1C 18313,N1(C(C2N(C)C(=O)NC2)=O)CCC(C2CC2)C1CNC(=O)CC1(CO)CC1 18314,C(=O)(CC(O)CC(C)(C)C)NCC1N(C(c2nc(OCC)sn2)=O)CC=C1 18315,N1(C(=O)NCC2(OC)CC2)CCC(O)C(C(=O)NCCC(C)OC)C1 18316,c1(C(=O)NC2CC(C)(NC(=O)CC3CC34CC4)C2)csc2c1CCCC2 18317,Cc1nc(NCC(C)C(C)(F)F)cc(=NCc2c[nH]nc2C2CC2)[nH]1 18318,c1(OC)nc(C)ccc1C(=O)NC1CN(C(c2cnc(O)cc2O)=O)CC12CC2 18319,C(CCC(C)(C)C(=O)NCC(C)(C(=O)OC)OC)NC(c1ncc(CC)cn1)=O 18320,c1(C(N(C2CCCN(C(=O)Cc3cnns3)C2)C)=O)cnc2c(c1)NCC2 18321,C(C1CN(C(C2CC2c2ccco2)=O)CC1C(=O)NC1CC(C)C1)=CC 18322,N1(C(CC)CC)CC(C(=O)NCCCN(C(c2cccs2)=O)CC)CC1=O 18323,N1(C(c2c(C)nco2)=O)CC(C)(C)OCC1CNC(C1(C)CC2CCC1O2)=O 18324,C1(C)(CC(NOCCOC)=O)CCCN1C(c1nnn(CC)c1C)=O 18325,CC1CN(C(=O)C(C)(C)C)CC1CCNC(C1(C#N)CCC1)=O 18326,CC(CO)C(C)N=c1[nH]c2cc(Cl)c(S(=O)(=O)NCCC3(C)CCCC3)cc2s1 18327,C1(C(C2CCCC2)NC(CSS(C)(=O)=O)=O)CCCN1C(=O)CC1CC=CC1 18328,C(=O)(CC(COC)COC)N1C(C(=O)NC(CCC)C(N)=O)CSC1 18329,c1(C(N(C(C)CNC(c2sccc2C)=O)CC)=O)cc(F)ccc1OC 18330,C(=O)(C#CC1CCCC1)N(CCCNC(c1c(C)cnn1C(C)C)=O)CCO 18331,CC1(C(=O)NC(CNC(c2cc(O)ncn2)=O)C2CC2)CCC(F)(F)CC1 18332,N1(C(C2(NC(CCc3ccc(C)o3)=O)CCC2)=O)CCCCCCC1C 18333,N1(C(=O)NC(CN(C)C)C(=O)N2CCCC2)CCOC(C(F)(F)F)C1 18334,C(=O)(CS(=O)(=O)CC(C)C)NCC1(O)CN(C(c2cnc(C)[nH]2)=O)C1 18335,CC(C)(CC(=O)NC1CCCN(C(c2nccc3c[nH]nc23)=O)C1)CC(F)(F)F 18336,CCC(C(=O)N1CC2CC2(CNC(C2CN(C3CCC3)C2)=O)C1)C(F)(F)F 18337,CC(CCNC(=O)CC1CCCO1)NC(=O)C=C1CC1 18338,CCC(CC)(CO)C(=O)N1CCC(O)C(NC(=O)C=CC2CCC2)C1 18339,CC(C)CC(O)C(C)C(=O)N1CC(C(=O)NCC2CCC(C)(C)O2)C(C(C)C)C1 18340,N1(CCNC(CC(C=C)C)=O)CCN(C(=O)CC2CCC(C)(C)C2)CC12CCC2 18341,Cc1ccc2oc(CNC(C3CCCCN3C(c3ccccc3)=O)=O)nc2c1 18342,CC(C)(C)CC(C)(C)C(=O)NC1CCN(C(=O)CC2CCCC3(CCC3)O2)C1 18343,CN1CCOC(C(=O)NCCCCCCNC(=O)COC(F)F)C1 18344,c1(C(C(=O)NCCC2(O)CN(C(C(C)SCC)=O)C2)C)ccc(F)c(F)c1 18345,c1(N2CCN(C(C(=O)NCC=C)COc3ccccc3)CC2)ccccc1C#N 18346,c1(CNC(C2(F)CCN(C(C=Cc3cn(C)nc3)=O)C2)=O)nnc2n1CCC2 18347,C=CCC(C)(C)CC(=O)N1CCC(C)C(CNC(=O)C(CC)C(=O)OCC)C1 18348,c1(C(N(CCNC(=O)C(C2(O)CCCCC2)(F)F)CC)=O)cnc2nccn2c1 18349,N1(C(CC2CC(OC)C2)=O)CCN(CCN(C)C(C2CCCS2(=O)=O)=O)CC1 18350,C(CCN=c1cc[nH]cc1S(=O)(=O)NC1CCCc2c1cnn2C)SC 18351,c1(C(=O)NCC(c2ccccc2)NC(C(C)CO)=O)cc(=O)c2cc(Cl)ccc2o1 18352,c1(C(=O)NCC2N(C(CNS(C)(=O)=O)=O)CC(F)C2)c(OC(F)F)cccc1F 18353,c1(C(C)=O)cc(C(=O)NCC23CN(C(C45CCC4C5)=O)CC2CCO3)ccc1O 18354,c1(C(=O)NCC(C)NC(c2snc(O)c2Cl)=O)ccc(C2COC2)cc1 18355,C1(NC(N(CC2=CCSC2)C)=O)CCCC1(C)CN(C)C 18356,n1(CC)ccc(C(=O)NC(CNC(=O)C(C)n2cnnn2)CO)n1 18357,C1(C(=O)OCC)CN(C(=O)C(C2CCCCC2)NC(=O)OC)C2(CCOCC2)C1 18358,c1(OC)cccc2cc(C(C)NC(=O)NCc3ccc(C#N)c(OC)c3)oc12 18359,c1(C(=O)NC(C(C)NC(=O)CCC2CC2)(C)C)cc2ccccc2n1C 18360,CCCCCC(C)CC(=O)NC(C(=O)NCC1(CN=[N+]=[N-])CC1)C(C)(C)C 18361,C(=O)(CC(C)CC(C)(C)C)NCC1(F)CCCN(C(CCN(CC)CC)=O)C1 18362,Cc1cc(C(=O)N(CCCCNC(=O)C(C)(C)N(C)C)C)ccc1OC(F)(F)F 18363,c1(C(C)(C)C)cccc(CNC(C2CC2C(=O)Nc2cnc[nH]2)=O)c1 18364,CCC(C)(C)C(O)C(=O)N1CC(F)CC1CN(C(=O)CC1CC1)C 18365,CC1CN(C(C2CC(O)CN2C(c2ccc(CO)s2)=O)=O)CCC1N(C)C 18366,CC1CCCN(C(=NCC(O)C2CC(F)(F)C2)NCc2cccs2)C1 18367,N1(C(COc2c(OCC)cccc2)=O)CCC(C)(C(=O)N(C)CC#N)C1 18368,c1(OC)ccc2[nH]cc(C(N3CCC4CCC(C3)N4C(=O)CO)=O)c2c1 18369,c1(C(=O)NCC23C(CN(C(Cn4c(C)csc4=O)=O)C2)C3)cccn2cncc12 18370,C(=O)(CCCCCN(C)C)N(C(C)C)CCN(C(=O)Cn1ncccc1=O)C 18371,Cc1cncc(CC(=O)NC23COC(CNC(c4cc(CO)c(C)o4)=O)(C2)C3)c1 18372,Cn1ncc2c(N3CC4CCN(Cc5c[nH]c6ncccc56)CC4C3)ncnc12 18373,C1(NC(C2(C)CNC(=O)C2)=O)CCCCN(C(=O)Cc2ccnn2C2CCC2)C1 18374,c1(C(=O)NCCN(C(c2cn(CC)cn2)=O)CC)ccccc1NC(N)=O 18375,C1(N(CCC)C(C2CCCC2O)=O)CCN(C(C2CC2c2ccncc2)=O)CC1 18376,N1(C(c2cn(CCCC)nn2)=O)CC2CC1C2NC(c1snnc1CC)=O 18377,Cc1cc(CCCNC(=O)C(C)Sc2ccccn2)oc1C(=O)O 18378,c1(C(N(CCN(C(CC(CC)OC)=O)C)C)=O)[nH]cc2c1CCS2(=O)=O 18379,Cc1cccc(C(=O)NCCC2(O)CN(C(=O)CCOc3cccnc3)C2)c1 18380,C1(NC(C2CCC(C)(C)O2)=O)CN(C(=O)C=Cc2cc[nH]n2)Cc2nccn2C1 18381,C=CCCC(C(=O)OC)NC(=O)CCCCN(C(=O)C=C=C(C)C)C 18382,c1(C2C(C)C2)ccc(CCC(=O)NCCCCN(C)C(c2coc(Cl)c2)=O)o1 18383,C(CC(=O)N(CC(C)CC)C)(C(F)(F)F)NC(C(CC#C)C1CC1)=O 18384,c1(C(C(=O)NCCOC2CN(C(COCCOCC)=O)C2)(C)C)cccc(C#N)c1 18385,c1(C2(NC(C3CCOC3)CC)CCC2)c(F)cccc1F 18386,c1(C(N2CC(C)C(NC(=O)CCOC3CCC3)C2)=O)cc(F)ccc1Br 18387,CC1CC(c2nnnn2C)(Nc2ccc(Cl)c(Cl)c2)CC(C)O1 18388,C(c1ccncc1C)=CC(=O)NCCc1c(CNC(CC=C(C)C)=O)nco1 18389,CC1(C)C2COC1(C(=O)NCC(C)(C1CC1)NC(c1cc(Cl)c(Cl)s1)=O)C2 18390,C1(C(=O)NC2CC(C(N(c3cn(CC)nc3)C)=O)C2)C2CCCC(=O)C12 18391,C12(CNC(c3cnc(C4CCCCC4)s3)=O)CC(CO1)N(C(=O)C1CC1)C2 18392,C1(CNC(C2N(C(CC3N(C)CC=CC3)=O)CCC=C2)=O)CC(C(N)=O)=NO1 18393,c1(C(N2C(CNC(C3C(C4C(C)C4)C3)=O)CC2)=O)cnn2cc(C#N)cnc12 18394,CC(C)(CNC(=O)Cn1cc(Cl)cn1)C(=O)N1CC2C=CC2C1 18395,c1(CC(=O)NC2CC(F)CN(C(c3c[nH]ccc3=O)=O)C2)cccc2sccc12 18396,CC(C)C(C(=O)NC12CC1CN(C(C1(N(C)C)CCCC1)=O)C2)C1CCC1 18397,c1(OC)nc2ccccc2c(Cl)c1Br.C1(OC)CCCNC(=O)N1C1CC1 18398,c1(-c2nc(C3N(C)CCNC3)on2)ccnc2[nH]ccc12 18399,c1(C(=O)NCCCCCNC(CCCC(=O)NC(C)C)=O)ccnc2c1CCO2 18400,C(=O)(C(C)(C)C(F)F)NCC(O)(C(F)(F)F)c1ccc(F)cc1.n12cc(nn1)C2C 18401,C1(NC(CC2CC(C)C2)=O)CCCC1NC(=O)C(c1ccc(Cl)s1)=O 18402,NC1CC(C)(C)Oc2ccc(F)cc21.Cc1cc(=NCC=CC(=O)N(C)C)[nH]cn1 18403,C1(C#N)(C(=O)NCC(CNC(=O)C(C(C)C)N(C2CC2)CC)OC)CC1(C)C 18404,N1(C(c2c(C)nco2)=O)CCOC2(C1)CN(C(c1cc3c(C)n[nH]c3cn1)=O)C2 18405,C1(C(=O)NCCCN2CCC(NC(C3CS(=O)(=O)C3)=O)CC2)CCc2nncn2C1 18406,CP(C)(=O)c1cccc(C(=O)NCC2CCC2NC(C2CC3CCC3C2)=O)c1 18407,c1(OC)cc(C(=O)Nc2cccnc2O)ccc1I 18408,Cc1nc2nccc(C(N3CC(N(C(=O)CCC4CC(F)(F)C4)C)C3)=O)n2n1 18409,C1(C(N2C(CCNC(C(COC)O)=O)CCC2)=O)CN2CCN1CC2C 18410,N1(C(C=C(CCC)C)=O)CC(C2CC2)(C(=O)NCCCCC2CC2C)C1 18411,c1(C(=O)NC(CCN(C(C=C(C)Cl)=O)C)C(C)(C)C)sc2cncn2c1C 18412,C=CC1(CC(N2CCC2N2CCCCC2)=O)CN(C(=O)C(O)CCSC)C1 18413,S(=O)(=O)(c1c2ccccc2nn1C)NCC.CN=c1[nH]cc(C(N2CCCC2)=O)s1 18414,C12(C(N3CC(C)(NC(CC(CC)C4CC4)=O)C3)=O)CCCC(C1)OC2 18415,n1(CC(=O)N(C2CN(C(C3C(C(C)C)C3)=O)C2)C)cc(S(N)(=O)=O)cn1 18416,c1(C(N2CCN(C(C(C)OC)=O)CC2CCO)=O)cc(C)cc2c1OCC2 18417,N1(C(CC2(C)CN(C(c3ccc4n[nH]cc4c3)=O)C2)=O)CCCCC(C)(F)C1 18418,N1(C(CCCC2C(C)C2)=O)CC(CNC(=O)C2=CSCCO2)OC2(CCC2)C1 18419,c1(CC)ccc(CCNC(=O)C(=O)NC2CC(C(=O)N(c3ncc[nH]3)C)C2)cc1 18420,C1(C(N2CC(CC)C2)=O)(CNC(=O)COc2ccsn2)CC12CCC2 18421,N#Cc1cnc(C(=O)NCC2C=CC(NC(=O)CC3(O)CCCCC3)C2)c(Cl)c1 18422,CC(O)C(C)C(=O)N1CCN(C(=O)C(CN(C)C)N(c2ccccc2)C)CC1 18423,C1(NC(=O)CCn2cncn2)CCC(CNC(c2cc(-c3cccs3)[nH]n2)=O)C1 18424,N1(C(CC(C)C(F)(F)F)=O)C(C)CC2CN(C(=O)Cc3c(Cl)cnn3C)CC12 18425,n1(CC)cnc2c(NC(C)COC(C)C)[nH]c(=NCCN3CC4CC4C3)nc12 18426,c1(C(N2CC(C)C(NC(=O)C=CC3(C)CCOCC3)C2)=O)cc2cnn(C)c2s1 18427,C(C(C)(C)C(=O)N1CCN(CC(C)(C)NC(C2CC(=C3CC3)C2)=O)CC1)SCC 18428,c1(C(N2C(CNC(C3CC4C=CC3O4)=O)COCC2)=O)cc(Cl)ccc1Cl 18429,c1(C(N2CC(NC(CN(c3ccccc3)C)=O)C3C2C3)=O)cc2occc2s1 18430,C12(C(N3CC(CNC(C(F)=CC)=O)N(C)CC3)=O)CCCN(CCC1)C2 18431,c1(C(=O)NC2CCC(NC(C(CC)(C)C#N)=O)C2)cnn2cccc(Br)c12 18432,C1(COc2cccc(C(=O)OC)c2)C(C)CCN1C(=O)COCC(F)(F)C(F)F 18433,c1(CC)nc(=N)[nH]cc1C(N1CC2CC1CN2C(C1CC2C=CC1C2)=O)=O 18434,c1(N2CC(CNC(C(CCC)NC(N)=O)=O)OCC2)ncc2c(ncn2C)n1 18435,C(C1=NOC2CC12)(c1nnnn1C1CC(F)(F)C1)NCC(C(C)C)(C)C 18436,C(=O)(CCCCCCSC)N1C(CNC(C(C=C)(C)CC)=O)CC2CC21 18437,c1(C(=O)NCC2COCC2NC(C2CCO2)=O)nc2n(c1Cl)CCCC2 18438,C(c1nc2ccccc2s1)=CC(N1C2(CNC(CC(CCC)O)=O)CC(C1)C2)=O 18439,CCC(CCCC(=O)N1CCCOCC1C)NC(C1CC(C)CCO1)=O 18440,c1(CC(=O)NC2CC(F)(CNC(=O)Cc3ccccc3O)C2)cc(F)ccc1Cl 18441,N(C1CCc2cc(Br)ccc21)C(c1c(OC)c(O)ccc1)c1nnnn1C 18442,c1(C(C(=O)NCC2N(C(C)=O)CC2)O)cnccc1C.N12CC(C1)C2=O.N 18443,c1(COC)nc(C)cc(=NCC2CN(C(c3cnc(C)nc3C3CC3)=O)C2)[nH]1 18444,N1(C(C(C)OCC2CC2)=O)CCCC(C)(CNC(c2ncccc2F)=O)C1 18445,Cc1coc(C=CC(=O)NCC(CC(C)C)NC(c2coc(Br)c2)=O)n1 18446,C(c1ccccc1Cl)=C(C)C(=O)NC1CCN(C(=O)CC2(C)OCCO2)CC1C 18447,Cc1nccn1CCC(=O)NCC1CC(NC(c2ncoc2C(C)(C)C)=O)C1 18448,c1(C(N2C(CC(=O)N(C(CC(CC)C)C)C)COCC2)=O)cc(C)cc(O)c1 18449,CON1CC(C(=O)NCC2(C(N3CCC(OCC(N)=O)C3)=O)CC2)CC1=O 18450,C1(NC(c2n(C(C)C)ccn2)=O)CCCC(CNC(c2cc(O)n(C)n2)=O)C1 18451,C(=O)(C(COC1(CC)CC1)C(F)(F)F)N1CCC(NC(C(C)OCC)=O)C1 18452,Cc1cc(=NCCN2CCCn3nccc32)[nH]c(NC2CCC(F)(F)C2)n1 18453,CCC(C)CC(C)C(=O)NCCCCNC(=O)CNC(=O)Nc1ccc(C)cc1 18454,C(=O)(CCCC(O)c1ccccc1)N(CC(C)NC(C1CCC(N=[N+]=[N-])C1)=O)C 18455,N1(C(C2C(C)(CC)C2)=O)CCCCC12CC(NC(=O)Cn1ccnc1C)C2 18456,N1(C(c2c(=O)ccn(C)c2)=O)CCN(C(c2ocnc2C(F)F)=O)CC12CC2 18457,C1(NC(c2c(C)nn(C)c2)=O)CCCCC12CCN(C(=O)COC1CCOC1)C2 18458,C=C(C)CC(C(=O)N(CC(=O)NC(c1cccnc1C)C)C1CC1)OC 18459,C1(C(=O)NC2C(C#C)CCC2)CNC(=O)CN1C(=O)COC1CCC1 18460,Cc1ccc(NC(=O)CCNc2nc(C)c(C)[nH]2)cc1S(=O)(=O)NC1CC1 18461,N(C1CCCc2c(F)cccc21)C(C(=O)NCCCC=C)=O 18462,C#CC1CN(C(C2CN(C(c3ns[nH]c3=O)=O)CC2(C)C)=O)CCN1C 18463,C1(CC)CC(C(=O)NC2(CNC(c3ccc(Cl)nc3C)=O)CC2)CCC1=O 18464,c1(C(=O)NCC(CC=C)NC(=O)C(c2cnn(C)c2)O)nc(Cl)sc1C(C)C 18465,C1(NC(C=C2CCC(C)CC2)=O)CCN(C(c2cc(Cl)n(C)n2)=O)C12CC2 18466,c1(C(=O)NC(C)CNC(C2CCCC2)=O)ccoc1I 18467,N1(C(C(C(C)(C)C)=O)=O)CC(CNC(C2CC(F)(CO)C2)=O)CC12CCC2 18468,N1(C(c2cc(OC)ncc2)=O)C2CCC1CN(C(C1CC1c1ccnn1C)=O)C2 18469,c1(OC)nccc(C(=O)NCC2(O)CC(CNC(=O)CCOC(C)=O)C2)n1 18470,CC(C)C(C(=O)NCC1CN(C(=O)CCCn2cccc2)CCO1)C1CCC1 18471,N1(C(C(C)=C2CC2)=O)CCC2(C1)CN(C(c1ccc(F)c(O)c1F)=O)C2 18472,C1(CNC(C2C(C)=C2)=O)CCC2CN(C(c3ccc4ncnn4c3)=O)CCC2C1 18473,n1(CC)nc(CN2CC3CC2(C)C3)c2c1CCOC2 18474,C1(NC(C2(CCOC)CC2)=O)CN(C(c2cncn(C)c2=O)=O)C2CCCCC12 18475,C#CC(C)(C)C(=O)NC1CCC(C(=O)NCC2CC2C)CC1 18476,Cc1nn(C)cc1C(C)NC(c1conc1C(C)NC(=O)CC1C=CCC1)=O 18477,c1(C(N2CC(N(C(c3c(C)cn(C)c3)=O)C)C(F)C2)=O)ccc2nonc2c1 18478,c1(C(N(CC(C)O)CCNC(COCCCC#C)=O)=O)ccc2c(n1)NC(=O)CO2 18479,C1(C)(C(=O)NCCOCCCNC(C(C2CCCO2)OC)=O)CC2(CCC2)C1 18480,C(=O)(C1=CC2CCC1C2)NCc1ccc(C(C)NC(C2(CF)CCC2)=O)cc1 18481,C1(CNC(C(C)(C)SC(F)(F)F)=O)CN(C(c2cnns2)=O)CCO1 18482,C(CCC(C(=O)NCC1(O)CCSC1)NC(=O)CC(C)C)OC 18483,N1(c2nnc(CC)s2)CCC(NC(=O)CNC(c2cscn2)=O)C(C)C1 18484,N1(C(c2c(CC)onc2)=O)CC(NC(C2COC(C)C2)=O)C2CCCC12 18485,N(C1c2ccccc2CC1NC(=O)C1CCCc2ccnn21)C(CCC(C)C)=O 18486,c1(-c2nc(C3(c4ccc(C(=O)OC)cc4)CCOCC3)on2)cnc(F)cc1C 18487,C(CCN=C(NCc1cncc(O)c1)NC1CCOC(C)C1)OC(C)C 18488,C1(CN(C)C(c2nnn(C)c2C(F)F)=O)CN(C(C2C(C)(C)C2(F)F)=O)CCO1 18489,C#Cc1ccc(C(N2CCCC2CN(C(=O)C(F)CC)CC)=O)c(OC)c1 18490,C(=O)(CCC(F)(F)CN=[N+]=[N-])NCCC1N(c2nnc(CCC)s2)CCC1 18491,N1(C(COC(C)(C)C)=O)CCCC2CCN(C(=O)C(F)(F)CN3CCCC3)CC12 18492,Cc1cnc(C)c(C(=O)NCC2CC2CNC(c2n[nH]cc2C(C)C)=O)c1 18493,c1(C(=O)NC2CC(C)N(C(=O)CCC(C)(C)O)C2)ccc(C#N)c(Cl)c1 18494,C1(C(=O)NCC(CC(C)C)NC(c2[nH]cc(CC)c2)=O)CC2(C1)CC(C#N)C2 18495,c1(C(=O)N(c2ccc(Cl)cn2)C2CC2)ccc(C2CCNCC2)cc1 18496,c1(OC)cccc(C(N2CCC(N(C)C(C3C(C)(C)C3(F)F)=O)C2)=O)c1[N+](=O)[O-] 18497,C(=O)(N(OC)C(C)C)c1c(CNC(C2C(C=C)OCC2)=O)cnn1C 18498,N1(C(c2cc(COC)sc2)=O)CC(CNC(c2cscc2COC)=O)C(C)C1 18499,C(C1CCCCCC1)=CC(=O)NC1(CCNC(C2(C)CCCOC2)=O)CCCC1 18500,C1(C(C)(C)C)CCN(C(=O)C(=O)NCC(C2CCCC2)=O)C(C(N)=O)C1 18501,c1(NC(COC)CC2CC2)[nH]c(=NCCC2CC=CCC2)nc2c1ncn2C 18502,N1(C(C(C)NC(c2ccoc2)=O)=O)CCN(C(=O)CN2CCSCC2)C2CCC12 18503,C(=O)(C(C)C1=CCCC1)NC(CCCNC(C=CC=CC)=O)c1ccccc1 18504,C1(CNC(CCCOC)=O)CCC(F)(CNC(=O)CC2CCCC(C#N)C2)CC1 18505,c1(C(C)=O)cc(C(=O)NCCCC(C)NC(C23CCC(OC)C2C3)=O)n(C)c1 18506,N1(C(C(CCCC)C)=O)Cc2n[nH]cc2C1C(=O)NCCc1nnc(C)s1 18507,CN1CCC(C)(C(=O)NCC(O)CCNC(=O)C(CN(C)C)N(C)C)CC1 18508,c1(CN2CC(NC(=O)CCN3CCC3)CC(F)(F)C2)ccc2c(c1)OCCO2 18509,N1(C(CC=C=C)=O)CCOC2CN(C(c3[nH]c(=N)ccc3C)=O)CC12 18510,N1(C(C2(CC#C)CC2)=O)CCc2nc(O)cc(C(=O)NC3CCN(C)C3C)c2C1 18511,C12(C(=O)NC(C)CCNC(C3C4(CC4)C34CC4)=O)CCCC1OCC2 18512,c1(CC2OCCN(C(C34CCC(OC)C3CC4)=O)C2)ccc(F)cc1C#N 18513,c1(OCC)cccc(C=CC(=O)NC2CCCN(C(C3(C)CNC(=O)C3)=O)C2)c1 18514,CC1(C)CCN(C(=O)C=Cc2cccnc2)CC1CNC(=O)Cc1cc(Cl)cs1 18515,CC1CCCN(C(=O)COCC(F)F)C1CN=c1[nH]nc(C2CCCC2)s1 18516,S(=O)(=O)(c1c[nH]ccc1=NCC1CCCOCC1)NCc1c(Cl)cn(C)n1 18517,N1(C(CNC(CC)=O)=O)Cc2nccn2CC(NC(=O)CC2CCCCO2)C1 18518,c1(OCCC(=O)NC2CC(NC(=O)CC3CCCCCC3)C2)ccc(F)cc1Cl 18519,C1(C(N2CCC(c3cc[nH]n3)C2)=O)COC2(C1)CN(C(c1cccnc1O)=O)C2 18520,C#Cc1ccnc(C(=O)N(CCCOCCNC(=O)C(C(C)CC)OC(C)=O)C)c1 18521,C(CC(=O)N1CC(C)(CCO)C1)(C(C)OC)NC(C(C)OCCOC)=O 18522,C1(NC(c2cc[nH]n2)=O)CN(C(c2cscn2)=O)C2(CCC2)C1 18523,C1(C(=O)NCC2OCCN(C(C3(n4cccn4)CC3)=O)C2)CCCCNC1=O 18524,c1(C(=O)OC)cc(CN2CCOC(c3nc(C(F)(F)F)n[nH]3)C2)cc(N)c1 18525,C(=O)(N=c1[nH]nc(Cl)c(C)c1C)c1c(C)nc(-c2ccccc2)s1 18526,N1(C(C2C(NC(C3(OC)CCSC3)=O)CC=CC2)=O)CCOC(C)C1C 18527,C1(C(=O)NC(C)C=CC(=O)NCCN2CCC2)OCCCC1(C)C 18528,S(=O)(=O)(c1ccc(S(=O)(=O)N2CCCC2)cc1)N1CCC(C#CC)C1 18529,C=Cc1ccc(CNC2CCC23CNC3)cc1 18530,c1(C(=O)NC2CN(C(Cc3ccc(C)o3)=O)CC2(C)C)cc(Cl)cc2c1CCC2 18531,Cc1cc2c(cc(C(N3CC4CCN(C(=O)CO)C4C3)=O)n2CC2CC2)s1 18532,C1(NC(c2c(C#C)cn(C)n2)=O)CCN(C(=O)C(C)OCCOCC)CC1(C)C 18533,C12(NC(CC3CN(C(C(CC#C)O)=O)CC34CC4)=O)CCC(C1)C(O)C2O 18534,c1(C(N2CCC(NC(c3ccn4c3CCCC4)=O)C2)=O)cc2c(cc1Cl)NCC2 18535,CCC(F)(F)CC(=O)N1CC(O)(C(C)NC(C2CCC(C)O2)=O)C1 18536,C1(O)(CNC(Cc2c(C)cccc2)=O)CCCN(C(c2c(C)noc2C)=O)CC1 18537,c1(SC)cc(C(N2CCC2CNC(=O)C2CC2)=O)nn1C 18538,C(=O)(CCC(C)(C)C#N)N1CCCC(CC=C)(NC(=O)CC(O)CC2CC2)C1 18539,C1(NC(CC=C=C)=O)(CNC(=O)C(C2(OC)CCOCC2)(F)F)CCOCC1 18540,C1(C(N2CCOCC2)=O)CN(Cc2ccnc(Br)c2)CC(F)(F)C1 18541,c1(CC(=O)N(C(C)CCNC(c2c[nH]c(Br)c2)=O)C)cccc2ncccc12 18542,Cc1cccc(C(=O)NC2CCN(CCNC(c3cc(C)n(C)c3)=O)CC2)c1N 18543,Cc1ncn(C)c1C(N1CC(n2cc(CNC(c3csc(=N)[nH]3)=O)nn2)C1)=O 18544,c1(C(=O)NC2CCC(C(=O)NCCC=C=C)CC2)cc2occc2[nH]1 18545,C1(NC(=O)CC=C(Cl)Cl)CCCCCN(C(c2ccc3cnnn3c2)=O)C1 18546,N1(C(C=C(C)C(C)(C)C)=O)CCCCCCC1C(N1CC2CCOC2C1)=O 18547,CC(C(=O)NC1CCN(C(=O)C(c2cc(F)ccc2F)=O)C1)C1=CCCC1 18548,Cc1oc(S(C)(=O)=O)cc1C(=O)NCC1CC(O)CN1C(C1CC12CCCC2)=O 18549,N1(Cc2ccc(OC)c(I)c2)CCC(Nc2ncc(F)cn2)C(C)(C)C1 18550,N1(c2nnc(C(C)C)o2)CCC2(CC1)CN(C(=O)C(F)C1CCOC1)CC(C)O2 18551,c1(N2CCN(C(C)C)CC2)ncc([N+](=O)[O-])cc1F.c1(C2C(C)N2)ccc(F)cc1 18552,N1(C(C2=CC(C)(CC)C2)=O)CC2CCCC2(NC(=O)CCc2ccn(C)n2)C1 18553,N1(C(C2CC(C)SCC2)=O)CCC2(C1)CN(C(=O)Cn1cccc1)CCO2 18554,n1(CC)cc(C(N2CC(C(O)C(=O)NC3CC(C(C)C)C3)C2)=O)nn1 18555,C1(NC(c2ccc(C)nn2)=O)CN(C(C2(CC#N)COC2)=O)CCC12CCC2 18556,N1(C(C(C(C)C)n2cnnn2)=O)CC2(CCC2CNC(=O)C(=O)N2CCCC2)C1 18557,N1(C(C2=CCCN(CC)C2)=O)CCSC2(CCOCC2)C1 18558,c1(C(=O)NCCCCNC(C(C)OCOC)=O)cnn(CCCN2CCCC2)c1 18559,C1(NC(c2ccc(C)o2)=O)CCCCC12CCN(C(c1cncc(F)n1)=O)C2 18560,C1(C(N2CC(CC(C)NC(CCNS(CC)(=O)=O)=O)C2)=O)CCCN1C 18561,N#Cc1ccc(C(N2CC3CC3(NC(=O)CCC3CCCCCC3)C2)=O)[nH]1 18562,c1(CC(=O)NC2C(COCC(=O)NC3CC(F)(F)C3)CC2)ccc(C(F)F)cc1 18563,c1(C(N(CCN(C(C(CC)C)=O)C)C)=O)cccnc1-n1ccnn1 18564,c1(NC(C2(F)CCN(C(C(CC)O)=O)C2)=O)ccc2c(c1)OCCO2 18565,CONC(=O)C(C)(C)CCNC(c1ccc(C(C)C)o1)=O 18566,c1(C(=O)NCCC(C)CCNC(=O)CS(C)(=O)=O)cc(C(F)F)cc(F)c1 18567,C1(NC(CCC(C)OC)=O)C(C)CCN(C(=O)COCCN(C)C)C1C 18568,C1(NC(C2CCN(C)C2)=O)CCCC(C(N)=O)C1.N12CCN(CC1)CC2=O 18569,C(=O)(C1=CCS(=O)(=O)C1)N1CCC(O)(C(C)CNC(c2cc(O)nc(Cl)c2)=O)C1 18570,CS(=O)C=CC(=O)N1CCC(CCCNC(=O)C(C)(F)c2ccon2)CC1 18571,c1(C(=O)NCC2CC(NC(=O)Cn3ccnn3)C(O)C2)coc2ccc(F)cc12 18572,Cn1c(C(=O)NCC(O)CNC(c2ccc(Cl)o2)=O)cc2c1CCOC2 18573,N1(C(C(C)OCOC)=O)CCC2(CCC(NC(c3ccc4n[nH]cc4c3)=O)C2)C1 18574,C1(CNC(C(N2CCC(C#C)(O)CC2)C(C)C)=O)CC2(CO1)CC(F)(F)C2 18575,c1(CNC(=O)NC2CCN(CCC(=O)OC)CC2)cc(C)c(C(F)F)cn1 18576,c1(CC(=O)NCC2(CNC(c3c(C)onc3)=O)CCC2)cn(C)nc1Cl 18577,c1(CNC(CNC(=O)NC)=O)ncc(C(=O)NCC2C=NNC2=O)o1.C1CCN1 18578,CC1CC(C(=O)NC2CCCC2CN(C)C)N1C(C1CSC1)=O 18579,c1(C(=O)NCC(C(N2CC(C)(CC)C2)=O)C)n[nH]c2c1COC2 18580,C1(NC(NNC(=O)C2CC(OC)C2Sc2ccccc2)=O)CCn2ccnc2C1 18581,N1(C(CN2CCN(C)CC2)=O)CCN(Cc2ccc3nonc3c2)CC12CC2 18582,c1(C(=O)NCCN(C(C2CC(CCC)C2)=O)C)occ(C)c1C 18583,N1(C(C2(C(=O)NC)CC2)=O)CC(O)(C(=O)NCC2(OC)CC(C)C2)C1 18584,N1(C(C(CNC(C(CC2CC2)OC)=O)C)=O)CCc2ccc(C#N)cc21 18585,c1(C(=O)NCC2CCN(C(c3cn(CC)nc3)=O)CC2O)cccc2c1CCN2 18586,c1(C(N2CCC(C)(C(=O)NC(C(C)SC)C)C2)=O)cnc2cc[nH]c2c1 18587,c1(CC(=O)NC2C(NC(C3(C#N)CCCC3)=O)COCC2)ccc2c(c1)CCO2 18588,N1(C(c2c(C)cc(C)s2)=O)CCC(CNC(c2c[nH]nc2C2CC2)=O)C(C)C1 18589,C(c1ccc(Cl)c([N+](=O)[O-])c1)=CC(=O)NCC1N(C(c2nc(C)oc2)=O)CC1 18590,c1(C(C)C)cc(C(=O)N(C2CCN(C(c3coc(Cl)n3)=O)CC2)CCO)n(C)n1 18591,C1(CNC(c2cc(C)ns2)=O)CN(C(=O)CC(O)C2CCCC2)CC1C(F)(F)F 18592,C(=O)(C1=CCOCC1)N1C(C2(NC(COC3CN(C(C)=O)C3)=O)CC2)CCC1 18593,N1(C(=O)NCc2cncn2-c2cccc(Br)c2)CCCN(CCO)CC1 18594,c1(SC)nn(C)cc1C(N1CCCC1(C)CNC(=O)Cn1cc(CSC)nn1)=O 18595,N1(Cc2c(N3CCCC3)ccc(C)c2)CCN(CCCOC(C)C)C(C)(C)C1 18596,N1(C(C(c2cc(C(C)=O)[nH]c2)N(C)C)=O)CCN(C(C2CCC(=O)NC2)=O)CC1 18597,c1(NC(Nc2cccc(C)c2)=S)ccnc(P(C)(C)=O)c1 18598,C1(NC(c2cc(OC)no2)=O)CC2CCC1CC2NC(C1CCCC1(C)C)=O 18599,C=C(C)C(C)(O)C(=O)N1CC(O)(CCNC(c2ccc(C)nc2)=O)C1 18600,Cc1ccc(Br)c(N)c1C(=O)NC1CCN(C(=O)C(Cl)=CCl)C1 18601,CCC(C)C(C(=O)NCC1CC2(CC2)CO1)NC(=O)Cn1cnnc1O 18602,N1(C(CN(CCOC)C)=O)C2CCC1CC(NC(C1(C)CCC(O)CC1)=O)C2 18603,Cc1cc(CC(N2CCC(N(CCO)Cc3cnc(S)[nH]3)C2)=O)n(C)n1 18604,CC1(C(=O)NCC2CCCC(NC(c3cnc(C4CC4)o3)=O)C2)CC2(CCC2)C1 18605,c1(C(=O)NCC(CC=C)NC(C2COCCN2CC)=O)ccc2nccnc2n1 18606,C1(C(=O)NC(C)CCCNC(c2cc(C(C)(C)C)ccn2)=O)COC2(CCC2)C1 18607,CC1CCC(NC(C2CCC(C)(C)CC2)=O)CN1C(C1CN2CCC1CC2)=O 18608,c1(CC)ccc(C)cc1C(N1CCCC1C(C)NC(c1[nH]nnc1C)=O)=O 18609,C1(C(=O)NCC2(C(N(CCN(C)CCO)C)=O)CC(C)(C)C2)CC(=O)NC(=O)C1 18610,C1(NC(=O)C(O)C(F)F)CN(C(=O)Cc2ccc3nonc3c2)C2(CCC2)C1 18611,C1(N(C(c2cccn2C(C)C)=O)CC)CCCN(C(c2ccc(CF)cc2)=O)C1 18612,c1(C(=O)NC2C(NC(c3ccc(C4OCCO4)cc3)=O)COC2)ncc(F)cn1 18613,Cc1cc(C(=O)NCCNC(c2cnc(C3CC3)s2)=O)c(C)n1CC(F)(F)F 18614,c1(C(N2CC(C(=O)NCc3nn[nH]c3C(F)(F)F)C2)C)ccccc1F 18615,C1(C(CNc2ccc(C)c(C3CC3)c2)OC)CCC(F)(F)CC1 18616,c1(NC(CSCCNC(=O)NC)=O)cc(F)ccc1F.c1(C(C)C)ccnn1C 18617,C1(F)(C(=O)NCCC2(CNC(C3CC=CCC3)=O)CC2)CC1(Cl)Cl 18618,C(=O)(C1CCCc2ncnn21)N1CCC(CC(=O)Nc2cnc(C)c(F)c2)C1 18619,C(=O)(CC(C)O)NCC(C)=CC(=O)NCc1nn[nH]n1 18620,c1(C(=O)NC(CC)CNC(c2ccc(C(C)C)cc2C)=O)c(C)nc(C)nc1C 18621,Cc1nccc(C(=O)NCC2(CNC(c3csc(F)c3)=O)CCCCC2)c1N 18622,c1(C(=O)NC2C(NC(C(C)C#N)=O)C2)c(F)ccc(F)c1Cl 18623,c1(CC(N2C(CCNC(=O)CC3CCC4CC34)CCC2)=O)cccnc1F 18624,N1(C(CC(C=C)(C)C)=O)CC2CN(c3ncc(C(=O)OC)cc3Cl)CC2C1 18625,c1(C(=O)NCC2(CC(=O)N(C)Cc3ccon3)CC2)cc(Cl)n(C)n1 18626,N1(C(c2c(OC)csc2)=O)CCOCC1C(=O)Nc1cncc(C(F)(F)F)c1 18627,C1(CC(N2C(CNC(C(C)n3cccc3)=O)CCC2)=O)SC(=N)NC1=O 18628,C(CCC(C(=O)NC(C)(C)C)N(CC(C)OC)CC=C(C)C)OC 18629,C1(C(=O)NCCC2(C)CC2(F)F)(OC)CCN(C(c2nc(C)sc2C)=O)C1 18630,c1(C(=O)NC(CC(=O)NC2CC(OCC)C2)C2CC2)cc(OC)n(C)n1 18631,C(CC(F)(F)F)SCC(=O)NC(C1CN(C(c2cn(C(C)(C)C)nn2)=O)C1)C 18632,c1(C(N(C(CNC(C2CC2OCc2ccccc2)=O)C2CC2)C)=O)cnn(C)c1F 18633,C1(C(N(C2CCCN(C(=O)CC3=NNC(=O)C3)C2)C)=O)CCCC12CCOCC2 18634,C12CCCCC1NC(=O)c1cnn(c1N)Cc1cn2nn1.C1(C(C)O)CCC1 18635,C1(CNC(c2cc(C)[nH]n2)=O)CC2CC2N1C(=O)CC(F)(F)Cl 18636,C(CC(=O)NOCCN1CCCC1=O)(C(F)(F)F)NC(C(CCC)=CCC)=O 18637,N1(C(CCCOCCOC)=O)CC2CC1C2C(=O)NC1C=CC(CO)C1 18638,c1(C(N2C(C(C)NC(C(CC)=CCCC)=O)CCC2)=O)nc(O)sc1C 18639,C(=O)(C(C(C)C)NC(=O)COCCSC)NC(CC)CO 18640,C1(CN(C(C(CC)SC)=O)CC)CCN(C(c2c[nH]cc2Br)=O)CC1 18641,NS(=O)(=O)c1sccc1C(=O)NCCN(C(C1COCCO1)=O)C1CC1 18642,c1(C(=O)NCCCC(CCC)NC(=O)CNS(N)(=O)=O)cc(F)cc2nc[nH]c12 18643,C1(C(=O)NCC(COCC)O)CSCCN1C(c1ocnc1C1CC1)=O 18644,c1(C(N2C(CNC(c3[nH]cc(C(N)=O)c3)=O)CCC2)=O)ccc2c(n1)NCCO2 18645,c1(C(c2n(CC)nnn2)NC(C(C)C)c2cncs2)ccc(C(F)F)cc1 18646,c1(C(=O)OC)cc(=NCC2CCCN2C(=O)CSc2cccc(F)c2)[nH]cn1 18647,c1(C(N(CC(=O)NCCC(C=C)C)C2CC2)C)ccccc1C 18648,N1(C(C=CC(=O)OCC)=O)CCOC2CCN(C(=O)C(C)Cn3ccnc3)CC12 18649,C1(CN(C(C(C=CCCC)O)=O)C)CN(C(=O)C=CCCCCC)CCO1 18650,c1(C(=O)NC2CCN(C(c3cn(CCC)nc3)=O)C(C)C2)ccc(C)c(C)c1N 18651,CC1CCC(CNC(c2cc(CNC(c3coc(C4CC4)n3)=O)cs2)=O)N1C 18652,C1(CNC(C(C)(C)OCC)=O)CCC(CN(C(=O)CCc2cn[nH]c2)C)CC1 18653,c1(NC(C(CC)N(C(C(CC)OCC)=O)C)=O)cc(C)cnc1O 18654,N1(C(C=C(C)CNC(=O)CCn2ccc(C)n2)=O)CCCCC1C1CCC1 18655,N1(C(c2cc(OC)nn2C)=O)CC(C)N(C(c2cc(C)n(C)c2)=O)CC1C 18656,Cn1c(C(c2nnnn2C2COC2)NCCCc2ccccc2)ccc1Cl 18657,N1(C(c2c(N3CCCCC3)cccc2Cl)=O)CC2CCC(C1)C2.N1CCCC1 18658,c1(NC23CC(C(=O)NCc4cncnc4)(C2)C3)cc(N2CCCC2)ncn1 18659,C1(NC(CCCCC#C)=O)CC(C2CCN(C(c3c(N)sc(C)c3C)=O)C2)C1 18660,c1(NC(C2(F)CN(C(c3cc(Br)ccc3Cl)=O)C2)=O)cnc2ccc(F)cn12 18661,c1(C(=O)NCC(C2CCCCC2)(C)NC(C(C)NC(=O)OC)=O)ccc(Br)o1 18662,N1(C(CSCCNC(c2cccn(C)c2=O)=O)=O)CC2(CC=CC2)C1 18663,N1(CC(=O)NCCOCC(=O)NC2CC2(F)Cl)CCCCS1(=O)=O 18664,N1(C(c2scnc2C2CC2)=O)CC2CCC(C1)N2C(C1CCCC1O)=O 18665,C(=O)(C(F)(CNC(=O)CCc1nncs1)C(C)C)NCCC(=C)C 18666,C1(CN(C(c2cc(Cl)cn2C)=O)CC)CCN(C(c2nncs2)=O)CC1 18667,C1(NC(C2CC(C#C)(O)C2)=O)CCN(c2nc(C)ns2)CC1F 18668,C(=O)(CCCC(=O)N1CCCN(C(=O)CNC(=O)CCCCO)CC1)OC 18669,c1(C(=O)NCC2CC2)cc2c(s1)CCN(C(=O)CN1CCCCC1=O)C2 18670,CC(O)C(C)(C)C(=O)NCC#CCNC(C1CC(O)CN1C(=O)OC(C)(C)C)=O 18671,C1(Oc2ncc(OC)nc2)CCN(C(=O)C(CN(C)C)NCCO)CCC1(F)F 18672,N1(C(c2ccc(C(C)=O)cn2)=O)CC(CNC(=O)C(C2CCCCC2)F)CC(C)C1 18673,C1(C(=O)NCC2CN(C(=O)CO)CCC2(F)F)Cc2cncn2C(=O)N1 18674,c1(OC)cccc(NC(C2(C)CCN2C(c2cccnc2O)=O)=O)c1 18675,C1(NC(CCC#C)=O)COC2(CNC(c3cc(Cl)sc3Cl)=O)CC1C2 18676,C1(NC(C2CN(S(CC)(=O)=O)C2)=O)CC(F)CN(C(c2csc(C(F)F)n2)=O)C1 18677,C1(NC(C2CC23CC3)=O)C2COCC1CN(C(=O)CCc1ncc(F)cn1)C2 18678,Cc1ccc(Cl)c(C(=O)NCCN(CC(C)O)C(=O)CN2CCC2C)c1 18679,C1(CN(C(=O)CC2(C)CC2(F)Cl)C)CCN(C(C2(O)CCCCC2)=O)CC1 18680,c1(OC)ccc(N)c(C(N2CCC(NC(C3CC3(C)C)=O)C2(C)C)=O)c1 18681,c1(C(=O)OC)cc(Br)cc2c1CCN2C(=O)Cc1ccc(F)cc1Cl 18682,c1(C(=O)NC(C)(C)CNC(c2cnn[nH]2)=O)ccc(F)c(Cl)c1N 18683,CN1CC(NC(=O)CNC(=O)CNC(c2n[nH]c3c2CCC3)=O)C2(CC2)C1=O 18684,CC1(C)OCCCC1C(=O)NCC1CN(Cc2ccccc2)CCCO1 18685,N1(C(CSC)=O)CC(NC(=O)Cn2nc(C)c3cccnc23)C2CCCCC12 18686,c1(C(C(=O)N(C2CN(C(=O)CC3CCCC(O)C3)C2)C)(C)C)cccc(C#N)c1 18687,C1(NC(C(C(C)(C)O)F)=O)CC(C2CCN(C(=O)CCc3nc(=N)[nH][nH]3)CC2)C1 18688,C12(C(N3CC(C)(NC(C(C)CSC(F)(F)F)=O)C3)=O)CC3CC(C1)CC(O)(C3)C2 18689,c1(NC2CCC2)ccc(C(=O)NC2C(NC(C(C3CC3)OCC)=O)CC2)nc1 18690,CN1CC(C)(C(N2CC(N(C)C(c3cc(C4CC4)ns3)=O)C3(CC3)C2)=O)CC1=O 18691,C(=O)(C(CC(C)(C)C)NC(=O)OC(C)(C)C)Nc1ccc(C(C)O)cc1 18692,C(C(C)C(=O)NC(C)CNC(c1cnc(-c2ccoc2)s1)=O)OC 18693,c1(CC)cccc(C)c1C(N1CCCC(O)(CNC(=O)CC2CC2C2CC2)C1)=O 18694,CC(CC(=O)NCC1(C(=O)N(CC(C2CCCC2)O)C)CC=CC1)C1CCCO1 18695,C1(NC(c2cn(CC3CC3)nn2)=O)CCCN(C(c2ccc(Cl)nc2)=O)CC1 18696,Cc1cc(C#N)nc(N2CCC(NC(c3ccc(-c4ccco4)[nH]3)=O)C(C)C2)n1 18697,c1(C(=O)NC2CC(NC(=O)Cc3cccc(O)c3)C2)ccc2c(c1)CC(=O)N2 18698,c1(CC)cc(C(N2CCCC2CNC(C2(F)C(C)(C)C2(C)C)=O)=O)cn(C)c1=O 18699,c1(C(N2C(CC(=O)Nc3ccc(C)c(F)c3)COCC2)=O)c(O)cc(O)cc1O 18700,Cc1cc(-c2ccnc(NC(c3ccccc3N(C)C(C)C)=O)c2)ccc1F 18701,N1(C(C(c2c(C)cccc2)C)=O)C2CCCC1CN(C(C1CCN(C)C1=O)=O)C2 18702,n1(CC)cc(Cl)cc1C(N1CC(CCNC(c2ccc(C#N)[nH]2)=O)C1)=O 18703,N1(C(C2(CC)CCC2)=O)CC2(CCN(Cc3nnc(C(C)C)s3)C2)C1 18704,C1(C(=O)NCCCc2c(C)n[nH]c2)CCN(C(c2[nH]nnc2C(F)F)=O)CC1O 18705,C1(C)(C(=O)NCC2(NC(C3CCCN(C)C3)=O)CC2)Cc2ccccc2C(=O)O1 18706,c1(C(=O)NCC(CC)N(C(=O)C=Cc2ccc(C)s2)C)ccc(=N)[nH]c1 18707,C1(=CC(CC)C)CCN(CCC#N)CC1.C12CCC(CC1)C(=O)N2C1CC1 18708,C(=O)(NNc1ccc(F)c(Br)c1)C(=O)OC(C)(C)C.CC1CCCCC1CN 18709,N1(CC(=O)N(CCCNC(C)=O)CC)CCC(NC(C)=O)CC1 18710,C1(NC(C(C)=C(CC)C)=O)CC2(CCN(C(=O)COC3CCOC3)C2)C1 18711,CCC(C)(CCNC(=O)CCCn1ccnc1)NC(=O)C(C)n1ccnc1 18712,c1(C(=O)NCCNC(C(c2ccc(Cl)cc2)(C)N(C)C)=O)ncccc1Cl 18713,c1(OCC)ccc(F)c(F)c1-c1cncc(C(N2CCC(OC)C2)=O)n1 18714,C1(CNC(C(C2CCOCC2)C)=O)CC2CCC(C1)N2C(C1CCS(=O)(=O)N1)=O 18715,C1(OC)CN(C)C(C)(C(N2CCCCC(CNC(C3(O)CCCCC3)=O)C2)=O)C1 18716,C1(CNC(c2c(C)n(C3CC3)cc2)=O)CN(C(=O)CC(C)CN(C)C)CCCO1 18717,N1(C(C(COC)OC)=O)CC(NC(c2ccc(OC)c(Br)c2)=O)CC1(C)C 18718,Cc1cnccc1CNC(=O)C(CCF)NC(c1cnccc1C)=O 18719,C#CCC(C)(C)C(=O)N1CCC(C)C(NC(c2cncc(C(C)C)c2)=O)C1 18720,c1(C(=O)NC2C(C)CN(C(c3ccnc(O)c3)=O)C2)cccc2c1OCCCO2 18721,c1(OC)ccnc(C(=O)NC2CCCCC2NC(=O)C(O)CN2CCCC2)c1N 18722,C12(C(N3CCC(CN(C)C(C4CC4(Cl)Cl)=O)CC3)=O)CC(C)(C1)OC21CCC1 18723,OC1COc2c(NCc3cc(Cl)sc3Cl)cnn2C1 18724,C#CCCCCCC(=O)N1CCC(N(C(c2cc(CO)[nH]n2)=O)CC)CC1 18725,c1(COC(CCC2(O)CCN(C(=O)OC(C)(C)C)CC2)=O)cc(Cl)cc2c1OCC2 18726,C#Cc1cccc(CC(=O)NC2CCOC2C(N2CCNC(=O)C2CCC)=O)c1 18727,C1(CNC(C2N(C)CC(O)C2)=O)CC2(CCC2)CN1C(=O)CC1C=CCC1 18728,Cc1ccnc(CNC(=O)C(C2CC2)N(C(=O)C(C)C(C)C)C)n1 18729,C=C(Br)CCC(=O)NC(c1ccccc1)CNC(=O)CC1CCCCCO1 18730,c1(C(N(CC(=O)NC2(CC(=O)OC)CC2)CC2CC2)=O)nnnn1C 18731,C=CCCCC(C)(C)C(=O)N1CCC(NC(c2ccc(C)c(Br)c2C)=O)CC1 18732,C=CCC(CC(=O)NCC(=O)N(C)C1CC1)NC(C1CCOC(CC)C1)=O 18733,N1(CC2(NC(CCOC)=O)CC2)CCN(C(C2OCCOC2C)=O)CC1 18734,c1(N(CC(CN(C)C)(C)C)C)nc(N2CCC(C)(C)C2)nc2c1cnn2C 18735,C(=O)(C(C)(C)CC(=O)OC)NCC(CC=C)C(=O)Nc1ccc(Cl)cc1 18736,n1(C(C#C)C2CCC2)cnc2c(N3CC(N(C)C(C)=O)C3)ncnc12 18737,c1(C(N2C(CNC(C(C)NS(C)(=O)=O)=O)CC2)=O)ccc(C2CC2)cc1F 18738,CC#CC1CCN(C(C2CCN(C(=O)CC3CCC=CCC3)C2)=O)C1 18739,C#Cc1ccc(C(=O)NCC2(NC(c3ccsc3COC)=O)CCC2)cc1Cl 18740,c1(C(=O)NCCOCCCNC(C(C)SC(C)C)=O)ccc2cn(C)nc2c1 18741,C(=O)(C1CCCn2cnnc21)NC1C(CNC(c2cccc(C(C)C)c2)=O)C1 18742,CC(C)CC(C)CC(C)C(=O)C(C1(c2cn[nH]c2)CCC1)=O.N1(CCN)C(=O)CNC1=O 18743,C(=O)(N(CCC(=O)OC)OC)C12C(CN(C(C(CC(=C)C)OC)=O)C1)CCC2 18744,c1(C(N(CCCN(C)C(C2(O)CCOC2)=O)C)=O)cccc(O)c1F 18745,Cc1ccc2oc(C(=O)NCC3(F)CC(NC(c4cc[n+]([O-])cc4)=O)C3)cc2n1 18746,c1(C(=O)NC(CNC(C2(C(C)C)CCCO2)=O)C)cnc([N+](=O)[O-])n1C 18747,C(C(CNC(C1CC1c1cnsc1)=O)C(F)(F)F)NC(=O)COCC(F)(F)C(F)F 18748,C(=O)(C#CC1(C)CCCO1)NC(C)CNC(c1cnn(C)c1C(F)(F)F)=O 18749,CC1=NOC(C)(C(=O)NCC2(C(N)=O)CN(C(=O)CSC(F)(F)F)C2)C1 18750,C1(O)(CCNC(c2c(CC(C)C)onc2)=O)CCN(C(=O)COCCN(C)C)C1 18751,N1(C(c2cn(CC(=O)NCCN(C3CC3)CC)nn2)C)CCN(C)CC1 18752,CC(C(=O)NC1CCCC1N(C)C)C(C)NC(=O)CN1CSCC1=O 18753,N1(C(C2(CC=C)COC2)=O)CCCC(CC)(NC(=O)Cn2ccc([N+](=O)[O-])n2)C1 18754,C1(CC(=O)NC2CCN(C(c3cnc(S)[nH]3)=O)CC2O)CC2CCC1CC2 18755,N1(C(c2c(COC)ccs2)=O)CCCCC2(CCN(C(c3cnc[nH]3)=O)C2)C1 18756,N1(C(c2ncc(OC)cn2)=O)CCC(NC(c2cc(C)c[nH]2)=O)C(C)(C)C1 18757,c1(C(C(=O)NCC2(NC(C3C(C)(Br)C3)=O)CC2)=O)cc(F)ccc1F 18758,C1(C(C)C)CNC(=O)CN1C(C1CC12CC(NC(c1nccn1C)=O)C2)=O 18759,C1(OC)CC2(C1)CN(C(=O)C(CNC(c1ncccn1)=O)C(C)C)C2 18760,C1(C(N(Cc2cn(CC(N3CCOCC3)=O)nn2)O)=O)Cc2nccnc2C1 18761,C1(SC)CC(CC(=O)NCCN(C(=O)C(C)C2CCCC2)CC(C)O)C1 18762,N1(C(Cc2ncn(C)c2)=O)CC(C(=O)NC(c2nc[nH]n2)C2CC2)C2(CC2)C1 18763,O=C(C(C(F)(F)F)C(F)(F)F)NCC12CC(NC(=O)C(F)=C3CCCC3)(CO1)C2 18764,C(=O)(C1=CCC(C)CC1)NCC1OCCN(C(CCc2ccc(OC)cc2)=O)C1 18765,Nc1cccc(C(n2ccnc2)NC2CCOC(CSc3csc(Br)c3)C2)c1 18766,C1(NC(CCC)=O)CCC12CN(C(=O)CCC(c1ccccc1)N(C)C)C2 18767,Cc1ncc(NC(C2CN(C(c3cncc(Cl)c3)=O)CCN2)=O)c(C)c1Br 18768,N1(C(c2c(OC)csc2)=O)CCOCC(NC(c2cc(F)cnc2Cl)=O)C1 18769,Nc1c(CN2CC3CC3C2C(F)(F)F)ccnc1Br 18770,CC1=CCC(C(=O)NCC2CC2NC(c2ccc(NC3CC3)nc2)=O)CC1 18771,c1(CNC(=O)CNC(=O)CNC(C2C3CCCC23)=O)ccnnc1 18772,C(C(C)(C)C(=O)N1CCC(O)(CC)C1)NC(c1ncn(CC)c1)=O 18773,C1(CNC(c2cnc(CC)s2)=O)Cc2ccccc2CN1C(C1CS(=O)(=O)C1)=O 18774,Cc1cc(C#N)ccc1C(N1CCC2(CC2NC(C2CC3(CC(=O)C3)C2)=O)C1)=O 18775,CCCCCCCCC(C)CC(=O)NCc1ccc(OC)cc1 18776,C#CC1CCCC(CNC(=O)C(C(C)C)NC(C2C(C)C2C)=O)C1 18777,C1(CC)(CO)CCN(C(C2CSCN2C(=O)C(C(=O)OCC)OC)=O)C1 18778,C(=O)(C(C)CCCC(C)=O)N1C2CC(C(N=c3ccn(CCOC)[nH]3)=O)(OC2)C1 18779,N1(C(CC2(C)CN(C(c3cc(C(F)(F)F)nn3C)=O)C2)=O)CCC(O)CC1.CO 18780,N#Cc1cc(NC(=O)NCC23CC(CCO2)C3)co1 18781,c1(OC)ncccc1C(c1nnnn1C)NC(C1CCC1)C 18782,c1(NC(=O)CC2(C3(C#N)CC3)CC2)cccc(F)c1Cl.C12CCN(C1)CCN2C 18783,N1(C(C(c2cccnc2)C)=O)CCC2CC(CNC(=O)CCF)CCC2C1 18784,C1(CC(C)C)CC(C(=O)NCCCNC(c2cc(=O)cc[nH]2)=O)CC(=O)N1 18785,C1(CC(=O)NC(C(C)CO)C)CCN(C(=O)CCN2CCCC2=O)CC1 18786,N1(C(c2cc(CC)nn2C)=O)C2CCCC1CC(NC(C1CC1(C)Br)=O)C2 18787,c1(CN2C(C(=O)OC)(CO)CCC2)cc2nccc(Cl)c2s1 18788,N1(C(=O)NC(Cc2cccc(C)c2)C2CC2)CCCC(O)(c2cnn[nH]2)C1 18789,C12(C(=O)NC(CC)CNC(=O)COCC3CCOC3)CSC(C1)C2 18790,c1(CC)nccnc1C(=O)NCC1CCN1C(=O)C(=CC1CCCC1)C 18791,C(=O)(C(CNC(=O)Cc1nocc1C)CC(C)C)NCC(CSC)OC 18792,CC1(C)CCCCC1CC(=O)NCC(C)(C)CNC(=O)CC12CC(C1)C2 18793,N1(C(CCCOC(C)=O)=O)CC2(COC(CNC(=O)C(F)CC3CCC3)C2)C1 18794,S(=O)(=O)(c1ccc(N2CC(CO)C3(CC3)C2)c(C#N)c1)NCCCN(C)C 18795,c1(NCC(C)(C)NC(Cc2ccc(OC)cc2)=O)ccc(C#N)cc1[N+](=O)[O-] 18796,C1(NC(CCNS(CC)(=O)=O)=O)CC2CC1N(C(C1(O)CCOC1)=O)C2 18797,C12(NC(CCc3ccnc(C)n3)=O)CCCC1N(C(=O)CSCC(N)=O)CCC2 18798,Cc1cc(Cl)cc(C(=O)NCC2(NC(C3CCC(=O)N3)=O)CCCC2)c1C 18799,C=CC(CCC)CC(=O)N1CC(C(=O)NCC2CCOC(C)(C)C2)C(F)(F)C1 18800,c1(OC)cc(C)ccc1C(N1CCCC(CNC(c2cc(Cl)c[nH]2)=O)CC1)=O 18801,C1(CNC(c2cccc(CC)c2)=O)COCCN(C(=O)CCOCC2CCC2)C1 18802,c1(C(=O)NCC(O)CNC(C2CC2C2CCC2)=O)ccc2ccc(Br)cc2c1 18803,c1(C(=O)NCC(CCCC)NC(=O)C(C)CF)ccc2n[nH]c(C)c2c1 18804,N1(C(c2ccc(Br)cc2)=O)CCC2CCCC2C1 18805,c1(-c2cn(C3CCC(n4cc(CCS(C)(=O)=O)nn4)CC3)nn2)cc(C#N)ccn1 18806,C1(NC(c2cc(SC)oc2C)=O)CCN(C)C12CCCN(C(=O)C=CCO)C2 18807,c1(C(=O)OC)ccc(C(=O)N(C)CC2CN(C(=O)C(C)c3ccco3)C2)c(Cl)c1 18808,C1(C(=O)NCC2C(C)CC2)N(C(c2coc(N(C)C)n2)=O)CC12CCCC2 18809,CCC(CC(=O)N(C1CN(C(C2CC=CCO2)=O)CCC1O)C)C(C)C 18810,C(C)(N=c1[nH]c2c(c(=NCCCc3cccnc3)[nH]1)CSC2)c1nc(CC)[nH]n1 18811,Cc1nnn(NC(=O)C(CNC(c2ccc(N)cn2)=O)CC2CC2)c1C 18812,c1(CNC(C(c2ccnn2C)C)=O)cc(C(=O)NCC2(F)CCOCC2)ccn1 18813,C1(F)(C(N(C(c2ccccc2)CNC(=O)CC(C)(C)O)C)=O)CCC(F)(F)CC1 18814,C1(CNC(CCSC)=O)CC2(CCN(C(c3cc(C(F)F)ccn3)=O)CC2)CO1 18815,C(=O)(CCCS(C)(=O)=O)N1CCN(C(C(C)NC(=O)NC)=O)C(C)C1 18816,c1(C(=O)NC(C2CCN(C(=O)CCc3ncc[nH]3)CC2)C)cc(Cl)cnc1O 18817,CCC(CCCC(=O)N(CC1CCC1)CC1CC1)NC(c1cc(C)cc(C)c1)=O 18818,c1(C(=O)OC)cnc(NC(C2CC23CN(Cc2ccc(F)c(Cl)c2)C3)=O)c(Cl)c1 18819,N1(C(N)=O)CCC(NC(=O)C(C2(O)CCC2)NC(C23CSCC2C3)=O)C1 18820,Cc1c(C(=O)NCC(C)CNC(=O)C(C(C)C)NS(C)(=O)=O)cccc1Br 18821,CCC(C)(C)C(=O)N1CCOC(CCNC(=O)CCn2cncn2)C1 18822,N1(C(c2ccc(NC)cc2)=O)CCN(C(=O)COCCO)C(CO)C1 18823,N1(C(c2ccoc2Cl)=O)CCC(N(c2ncnc(C(C)(C)C)n2)CCO)CC1 18824,c1(N(C)Cc2ccccc2F)nc(=NCC2(C)CCCC2O)[nH]c2c1CCC2 18825,n1(CC)cc(C(=O)NC2C3CCN(C(c4sc(C)nc4C)=O)C23)c2ccccc12 18826,c1(CC(=O)NC2CC(C)N(C(c3cccn(O)c3=O)=O)C2)c(F)cccc1F 18827,N1(C(CN(CC#C)C(C2CCCC(OC)C2)=O)=O)CC2CCCC(O)C2C1 18828,O=C(C1=CCOC1)NCCCC(c1ccccc1)NC(C1CCCCCC1)=O 18829,CC1CCC(C)(C(=O)NCCNC(c2ccnc(Oc3ccccc3F)c2)=O)C1 18830,N1(C(C#C)C)CCN(C(=O)C(CCF)NC(c2cnncc2C)=O)CC1 18831,C(=O)(Nn1cccc1)C1C(C(=O)OC)C1 18832,c1(C(=O)NCCNC(=O)CNC(=O)NC2CC2)cc(CCP(C)(C)=O)[nH]n1 18833,Cc1cccc(C(=O)NCCCCCCNC(=O)CC2(C)CCCO2)c1N 18834,N1(C(c2c(CNC(c3n(C=C)nnc3)=O)cco2)=O)CCC2C(CCN2C)C1 18835,N#Cc1cc(C(=O)NCCN2CCN(C(=O)C(O)C3CCC3)CC2)c[nH]1 18836,C1(C(=O)NC(C2CCN(C(C3COC(=O)O3)=O)CC2)C)CCSC(C)C1 18837,C1(F)(CNC(c2ccnc(O)c2)=O)COCCN(C(=O)C(O)c2cnc[nH]2)C1 18838,Cc1cc(C)c(C(=O)NC(Cc2ccoc2)C(=O)NCc2ccc(C#N)s2)s1 18839,C1(C(C)C)N(C(C2CC2C)=O)CC12CCN(C(c1nc(C3CC3)cs1)=O)CC2 18840,N1(C(CC(CCC)(C)C)=O)Cc2cccc(CNC(=O)C(COC)CC)c2C1 18841,N1(C(Cc2scc(C)c2)=O)CCC(CF)(NC(=O)C(C(C)C)n2cnnn2)C1 18842,C1(C(=O)NCC2CC(F)CN2C(C2(F)CCCCC2)=O)CCCC1C1CC1 18843,c1(C(=O)OC)ccc(C=CC(=O)NC2CCN(C(=O)C=CCOC)C2C(C)C)o1 18844,C(=O)(C1=CCOCC1)N(C1CCCN(C(c2c(COC)cccn2)=O)C1)CCF 18845,C(=O)(CC(C(F)F)C(C)(C)C)N1CC(CNC(C(CCN2CCC2)NC=O)=O)C1 18846,Cc1cc(Cl)cc(C(N2CCCC2CCNC(c2ncnn2C)=O)=O)c1O 18847,Cc1cc(NC2CCSC2C)ncc1S(=O)(=O)N1CCC(c2ccncc2)CC1 18848,C1(C(=O)NCc2n(CC)ncn2)CC=CC(NC(=O)C(C(C)C)NC=O)C1 18849,C1(C(N2C(COC)(CNC(=O)C3=CCOCC3)CCC2)=O)CCCCC12CCC2 18850,c1(CCC(=O)NC2CN(C(=O)CCc3ccoc3)C2)cccc(F)c1 18851,c1(C(N(C2CCC(NC(CSCC)=O)C2)C)=O)cnc2cc(C)ccc2c1 18852,c1(C(=O)OC)ccc(CC(C)C)nc1N1CC2CC(NC(=O)CC3CC3C)C2C1 18853,c1(C(=O)NCC2CN(C(C3C(C)CC3)=O)C2)cc(Cl)ccn1 18854,N1(C(c2c(OCC)nccc2)=O)CC2CC(C1)N(C(=O)CCc1ncc(C)[nH]1)C2 18855,c1(OC)ccc(-c2ccnc(C(N3CCC(F)(c4cn(C(C)C)nn4)C3)=O)n2)cc1 18856,c1(C(=O)NC(CC)CNC(c2csc(C)n2)=O)sc2ccccc2c1Cl 18857,c1(C(=O)NC(CN(C(c2cccc(SC(F)(F)F)c2)=O)CC)C)cc(C)n(C)c1 18858,CC1=NS(=O)(=O)NC=C1C(=O)N1CC(NC(=O)C2=C(C)OCC2)CCC1C 18859,c1(C(=O)NC(C(C)C)CNC(C2CC23CCC3)=O)nn(C)c(C(F)(F)F)c1Cl 18860,C1(NC(C(C2CCN(C(c3c(CC)c[nH]n3)=O)C2)(C)C)=O)C2CCCCC12 18861,c1(NCCCC2C(O)CCC2)nccc(=NCCOC2CCOCC2)[nH]1 18862,C(=O)(CCCCCCCC1CC1)N1C(CNC(c2cn(C)c(=O)cc2)=O)CCC1 18863,c1(C(=O)OC(c2cccc(C#N)c2)C)ccnc(Cl)c1N 18864,c1(NC(C2CCN(C(Cn3ncc(CC)c3)=O)CC2)=O)ccc2ccncc2c1 18865,N1(c2ncc(C(=O)OCC)s2)CCCC2(CC(NC(=O)C(C)c3ccco3)C2)C1 18866,C1(NC(c2ccc(C(C)(C)C)cn2)=O)CC2CC(NC(=O)C3=CCCS3)CC12 18867,C1(NC(CNC(CN(C)C)=O)=O)CCOC12CCN(C(=O)CC(F)(F)F)CC2 18868,C=CCCCC(=O)NC1CCC(NC(C2(COC)COC2)=O)CC1 18869,c1(CN2CC(NC(C(CCC)C)=O)C(C)C2)nn2c(=O)cc(C)nc2s1 18870,C(=O)(C(C)CC(F)F)NC(C(=O)NCC1(OCC)CCC1)Cc1ccoc1 18871,N1(C(C2C(OC)CCC2)=O)CCc2[nH]nc(CNC(=O)CC3(OC)CC3)c2C1 18872,C1(NC(=O)C=CC=C(Cl)Cl)CN(C(c2cnc3n2CCC3)=O)CC12CCC2 18873,Cc1csc2ncnc(N3CCC(C)(C)C(CNC(=O)C(C)S(N)(=O)=O)C3)c12 18874,C(=O)(CC(c1ccccc1)OC1CC(N)C1)NCC1(OC)COC1.C(=O)NCC 18875,C1(C(=O)NCCNC(c2cc(F)cc(N)c2F)=O)(CC)CCC(F)(F)CC1 18876,N1(C(Cc2c(C)nccc2)=O)C2CCC(C2)C1C(=O)NOC(C)C 18877,CCCC(C)CC(=O)NC(C)CN(C(c1ccncc1C1CC1)=O)CC 18878,c1(C(=O)NC2CC(CNC(c3c(OC)ccnc3)=O)C2)ccc2ncccc2n1 18879,CCN=c1[nH]cc(C(=O)NCC(F)CNC(=O)C(c2cccc(C)c2)C)s1 18880,c1(C(N2CC3(C2)SCCC3NC(=O)C(F)(F)C2CC2)=O)cccc2sccc12 18881,Nc1nc2ncccc2cc1C(=O)NC1(CO)CCN(C(=O)CC2CCCC2)C1 18882,N1(CCc2ncn(C)c2)CCc2onc(C3CC3)c2C1 18883,Cc1nc2cccc(NC(=O)NCC(C)(C)CC#N)c2[nH]1 18884,c1(C(N2CCCOCC2C)C(=O)NCC(=C)C)cccc(C(F)(F)F)c1F 18885,N1(C(C(C2(O)CCCC2)OCC)=O)CCSC12CC(OC)C2 18886,S(=O)(=O)(c1ccc(NCCCc2cccnc2)c(Br)c1)NC(C)CS(C)=O 18887,CC1CC(NC(=O)NNC(=O)c2cn(C)nn2)CCN1C 18888,S(=O)(=O)(CCC(F)(F)F)N1CC(C)(CC(N2CCC(OCCF)C2)=O)C1 18889,N1(C(CC2C(CC)CC2)=O)CCN(Cc2ccc(NC(=O)C=C3CC3)cc2)CC1 18890,c1(C(=O)NC2C(NC(CSc3nc(C)[nH]n3)=O)C2)cc(N)cnc1C 18891,C(CC(C(=O)N1CCC(NC(=O)CC2CCCC23CC3)C1)OC)OC 18892,C1(NCc2cnc(CC)[nH]2)CCN(c2ccccc2)C1=O 18893,C(CC(=O)N(CCCNC(=O)C(O)Cn1cncn1)C1CC1)(C(F)(F)F)OCC 18894,Cc1nsc(NC2CC2)c1C(=O)NC(CNC(C1CCCCC1CO)=O)C1CC1 18895,C(=O)(C1=NNC(=O)CC1)NCC1(NC(c2nccc(C)c2)=O)CCOC1 18896,N1(C(c2cncc(N)c2)=O)CCC2C(C1)CN2C(c1cccc2sccc12)=O 18897,C1(O)(C(=O)NCC2CC(NC(COC(CC)C)=O)C2)CCCC1 18898,C(=O)(C1=CC2(CN(C(=O)CC3CCCC(O)C3)C2)OC1)NC(c1ccnn1C)C 18899,c1(OC)ccccc1CC1(O)CC(COC(C2CC2(F)F)=O)C1 18900,CC1(C)COc2ccc(C(=O)NCCC3(O)CN(C(=O)C4=CCCC4)C3)cc21 18901,N(C1CCCc2ccc(F)cc21)C(=O)NNC(=O)C(=O)NC1CCCCC1 18902,C(=O)(C(C)CC(F)(F)F)NCc1c(C(=O)NCC2(CC)CCCO2)cco1 18903,C1(NC(C2CCC(C)C2)=O)CC2CC(C1)N(C(=O)CCCCCN(C)C)C2 18904,c1(OC)ccc(C(c2ccc(C)s2)NC(Cc2ccccc2)C2CC2)cc1Br 18905,c1(C(=O)NC23CC(C(=O)NC4CC(C)OC4=O)(C2)C3)cn(C)c(=O)cn1 18906,c1(C(N(C(CN(C(C(C)NC(C)(C)C)=O)C)C)C)=O)ncc(F)c2ccccc12 18907,C1(CNC(=O)CC2CCCO2)CCCN1c1ccncn1 18908,O=C(CC(C(F)(F)F)NC(C1(n2cccn2)CC1)=O)NCCC1CC1 18909,C(=O)(C#CC1(C)CC1)NCC=CCNC(CS(=O)(=O)NC)=O 18910,N1(CC)CCOC(C(=O)NC(CCN(C)C(C2(C3CC3)CCC2)=O)C(C)C)C1 18911,c1(C(=O)NCC(C)CC(=O)NCC2CC3C=CC2CC3)ccc2n[nH]cc2c1 18912,N1(C(CNCCC=C)=O)CCc2ccccc2C1CCNC(=O)COCC1CC1 18913,c1(C(=O)NCc2c(CCNC(C(C)OCCC#C)=O)ocn2)cc(C)c(C)o1 18914,Cc1ccc(F)c(O)c1C(N1CC2CC(NC(C3CCCCC3)=O)CC1C2)=O 18915,C1(NC(c2cnc(C(C)O)s2)=O)CC(C)N(C(=O)Cc2cnn(C)c2C)C1 18916,C1(C(=O)NC(c2cc(F)cc(Cl)c2)CNC(C)=O)CCC(=O)NC1=O 18917,C1(F)(Cc2cn(CCC3(C)CC3)nn2)CCN(C(=O)CC2NC(=O)NC2=O)CC1 18918,C1(NC(CC(C)(C)O)=O)CC12CCN(S(=O)(=O)c1ccccn1)CC2 18919,C12(CC(N3CC(CN(C(=O)CCCF)C)OCC3)=O)CCCN1CCC2 18920,N1(C(CC(C)SC)=O)CCCC(C2CN(C(c3c(C(F)(F)F)ncn3O)=O)C2)C1 18921,C1(NC(c2ncc(NC)nc2)=O)CCN(C(=O)CC2CC3(CC3)C2)CC1C 18922,C1(C(=O)NC(C(C)(C)C)CNC(=O)C(N)=O)CCn2c(O)nnc2C1 18923,c1(C(N2CCCC(CC3CC3)C2)C(=O)NCCC)ccc(OC)c(Br)c1F 18924,C1(NC(C2C3CC4C(C3=O)C24)=O)CCCN(C(c2[nH]cc3c2CCC3)=O)CC1 18925,CC1(C)CC(N=c2ccnc(C(F)(F)F)[nH]2)CN(C(c2cccnc2O)=O)C1 18926,N1(C(C(CNC(CC2(OCC)CCC2)=O)(C)C)=O)CCC2(CNC(=O)N2)C1 18927,C(C(C)(C(=O)NC(C1CCCC1O)C)NC(C1CCC(=O)O1)=O)SC 18928,C1(NC(CCOC)=O)CN(C(c2sc(Br)nc2C)=O)CCC1CO 18929,Cc1nc(CN2CC(C(=O)N=c3cc(C4CC4)o[nH]3)OC(C)(C)C2)nc(O)c1F 18930,c1(OCC(CNC(=NC)NC2CCOCC2)O)ccc(C(F)(F)F)cc1 18931,C1(OC)CC2CC(C(=O)NC34CC(NC(=O)COC(C)=O)(C3)C4)CC12 18932,c1(C(N2C(C)CCC(NC(C(C)=C(CC)C)=O)C2)=O)cc[nH]c2nccc1-2 18933,C1(NC(C(=O)NCC(CC)O)=O)CCCN(c2ccccc2C)C1 18934,C1(NC(C(CSC)O)=O)CC2CCC1N2C(c1ccc(Cl)cc1N)=O 18935,Cc1cccc(OCC(C)NC(=O)C(C)N(C(C2CCCCC2)CN(C)C)C)c1 18936,N1(C(C(C)N(C(=O)C(C)N(CCOC)CC)CC)=O)CCn2ccnc21 18937,C#Cc1cccc(CCC(=O)NCCCN(C(=O)CNS(N)(=O)=O)C(C)C)c1 18938,C1(NC(C(C)CF)=O)CC2CN(C(c3cc(Cl)no3)=O)CC2C1 18939,c1(C(N2CC(CC(C)NC(c3n(CC)cc(Cl)c3)=O)C2)=O)cc(C#N)cn1C 18940,c1(CC(C(=O)NC2CN(C(c3cc(COC)sc3)=O)C2)O)cc(Cl)cc(Cl)c1 18941,N1(C(c2c(CC)nc(C)o2)=O)CCC2(CC1)CCN(c1nnc(C)o1)CC2 18942,Cc1cnc(C(N2CCC(NC(C3CC3C(N)=O)=O)C(O)C2)=O)cc1Cl 18943,n1(CC)nncc1C(=O)N(CCCNC(=O)CSCc1ccncc1)C(C)C 18944,c1(OC)cc(F)c(C(N2CC(C)(NC(c3cc(C)cs3)=O)C2)=O)c(F)c1 18945,C1(C(=O)NCC(C)CN(C)C(c2ccccc2F)=O)CCCC(C)CC1 18946,Cc1ccc(S(=O)(=O)N(C2CC3CNC2C3)C2(C#N)CCC2)cc1F 18947,CCC(CC(C)C)C(=O)N1CC2CCC1C(CNC(=O)C(C)NS(=O)(=O)CC)C2 18948,N1(C(C=C(CCC)CCC)=O)CCCN(C(=O)C(C)OC(C)(C)C)C(C)C1 18949,N1(C(c2n[nH]c(C)c2Cl)=O)CC=C(C(C)(C)C(=O)N(C2CCN(C)C2)C)C1 18950,c1(C(N(C(C)CNC(=O)CSCCC(C)C)CC)=O)ccc(O)nc1C 18951,C1(C(N(CC(C)C)CC(=O)NCC2CC2Cl)=O)CCCC(C)(C)C1 18952,c1(OCCC)cccnc1C(=O)NCC1CCCCN1C(C12CCC(CO1)C2)=O 18953,N1(C(C(n2cc(Cl)cn2)C)=O)CCC2(C)CN(C(C3CCC4CC34)=O)CC12 18954,CC1(C(=O)NCc2occc2C(=O)NCc2ncccc2Cl)CC2CC2C1 18955,C12(C(=O)NC3C(NC(C(C)(C)COCC(F)F)=O)COC3)CC1COC2(C)C 18956,c1(CC(=O)NCCCCN(C)C(C2(C)CCCOC2)=O)ccc(Cl)cn1 18957,C1(C(N2CCCC(CC)C2)=O)CC12CCN(Cc1ncc(Cl)nc1Cl)C2 18958,c1(OC(C)=O)ccc([N+](=O)[O-])cc1C(N1CCN(C(=O)CS(C)(=O)=O)C2CC12)=O 18959,C(=O)(C1=CC(C)(C)C1)N1CCC(C(=O)Nc2c(CC)nn(C)c2)C1 18960,Cc1ccc(=O)n(CC(N2CCN(C(c3ccc(C)c(C)n3)=O)C(CO)C2)=O)c1 18961,N1(C(C(C(CC)O)C)=O)CCC2(CCN(C(c3ccnnc3C)=O)C2)C1 18962,N1(C(C(CCOC)C)=O)CCN(C(c2cccc3nc(C)nn23)=O)CC2(CC2)C1 18963,CCCS(=O)(=O)C(C)C(=O)N1CC(N(C)C(c2c[nH]c(=N)nc2C)=O)C(C)(C)C1 18964,C1(C(=O)NC(COCC)C(C)C)CC2(CC2)CN1C(=O)C(c1ccnn1C)C 18965,C1(C(N(CC(C)(C)NC(CCN(C(C)=O)C)=O)C)=O)CCCN1C(=O)C(C)(C)C 18966,N1(C(C(COC)(C)O)=O)C2CCC1CC(N(C(=O)CCc1ccoc1)C)C2 18967,C#Cc1ccc(Cl)c(C(=O)NC2CC(CNC(=O)CSS(C)(=O)=O)C23CCC3)c1 18968,C(=O)(CC(C)COCC)N(C(C)C(=O)N(C)Cc1ccnn1C)CCC 18969,Cc1nc(N2CC3(CCC(NC(=O)Cn4cc(Cl)cn4)CC3)C2)c2ccsc2n1 18970,c1(CC)ccc(C(=O)NC2CN(C(=O)C(N3CCNC3=O)C)CC23CC3)cc1F 18971,S(=O)(=O)(c1cccnc1N1CCCN(C)CCC1)N1CCN(C(C)CO)CC1 18972,c1(C(N(CC(C)(C)NC(CC(C)F)=O)C)=O)cnn(CCO)c1C(F)(F)F 18973,C(=O)(C(O)CC(F)F)N1CCC(N2CCC(NC(c3cscn3)=O)CC2)CC1 18974,c1(CNC(CCC(=C)C)=O)nc2c(s1)CCN(C(=O)C(C)(C)N1CCCCC1)C2 18975,C12(C(=O)NCC(C)(CO)NC(c3c(OC)scc3)=O)CCCC1C2(F)F 18976,c1(OC)ccc(C=CC(=O)NC(C2CCCN2C(C2C=C2C)=O)(C)C)c(C)c1 18977,C(=O)(C(C)(C)CC(F)F)NC(CCN(C(c1[nH]cc(C(C)=O)c1)=O)C)C 18978,N1(C(C(COC)NC(CCCOCC)=O)=O)CCC(C)C(CO)C1 18979,N1(C(CCC(=O)c2cccs2)=O)CCCC2(CCCN2C(C2CC2F)=O)C1 18980,c1(C(=O)NCC(C2CC2)NC(CC2C(C)(C)CCCO2)=O)scc2c1OCCO2 18981,C(C)(C)(CCCCC(=O)NCC1CCC1NC(c1sc(OC)nc1Cl)=O)OC 18982,C1(S(N)(=O)=O)(C(N2CC(NC(=O)C(C(C)C)OC)CC(OC)C2)=O)CCCC1 18983,CCC(CC(=O)NCCC(C)(C)NC(=O)CS(=O)(=O)N1CCOCC1)SC 18984,c1(CSCC(=O)NC2(CCNC(C(C)NS(C)(=O)=O)=O)CC2)ccccn1 18985,C1(COC(CCCCN=[N+]=[N-])=O)CCC2(CCOCC2)CO1 18986,C1(C(N2CC(C3CN(C(C(C=C)O)=O)C3)C2)=O)CCc2n[nH]c(C)c2C1 18987,N1(C(COCc2onc(CC)n2)=O)CCC(CNC(=O)C=C(C)Cl)C(CO)C1 18988,C(CC(=O)NC(c1cnn[nH]1)(C)C)(CC(C)C)NC(c1c(CC)n(C)nn1)=O 18989,Cc1cnc(NCC(F)C2CCC2)c(S(=O)(=O)NCC2CCC(C)(C)O2)c1 18990,C1(=O)C(C(C)C)CN1.S(=O)(=O)(CCNS(C)(=O)=O)COC(C)C 18991,N1(C(c2cncc(C)n2)=O)CC(CNC(=O)Cc2ccc(F)cc2)CC(C)C1 18992,C#CCCCCCCC(=O)N(C1(S(C)(=O)=O)CC1)CCN(C(=O)C1CC1)CC 18993,c1(C(=O)NC(CC(C)NC(c2cnc(CC)[nH]2)=O)C)cnc(N)c(N)c1 18994,C(=O)(C1Cc2ccc(Cl)cc21)N1CC2CCN(C(CNC(C)=O)=O)C2CC1 18995,c1(C(CNC(C2(C)CCCS2)=O)NC(=O)CN2CC=CC2)ccc(F)cc1F 18996,C#CCCN=C(NCc1ccc(C(C)(C)C)cc1)N1CCC(CS(C)(=O)=O)C1 18997,C1(NC(C2(C(=O)OC)CC2)=O)CCN(C(=O)C=C2CCOCC2)CC1C 18998,N1(C(C(C)OCCCC)=O)CC(C)(C)CCC1CNC(C1(c2cccs2)CC1)=O 18999,C1(COC)CN(C(=O)C(O)CCSC)CCN1C(=O)CSCCC#N 19000,CC1CN(C(C2(F)CCCCC2)=O)CCN1C(c1ccnc(-n2ccnc2)c1)=O 19001,Cc1ccncc1-c1cn(CCC2CN(C(=O)CC3CCC(C)CO3)C2)nn1 19002,C1(C(=O)NC(C(C)NC(=O)CSCC(N)=O)C)(CF)CCOCC1 19003,c1(OC)cc(C#N)ccc1NC(C1(C)CCN1C(c1cnc2[nH]ncc2c1)=O)=O 19004,CC(N=c1[nH]c(=NCc2cn3ccccc3n2)[nH]c2c1COC2)c1ccc(Br)s1 19005,c1(C(=O)NCCC#C)cnc2ccc(-c3ccc([N+](=O)[O-])c(F)c3)cn12 19006,C1(NC(=O)OC(C)(C)C)CC(CNc2c(Br)noc2C(=O)O)C12CCC2 19007,C1(c2noc(C(C)CCc3ccco3)n2)(NCC)CCCCCC1 19008,Cc1ccc(C)c(C(=O)NOC(CC(C)C)C(=O)N2CC(Cc3ccco3)C2)c1 19009,c1(C(N(C)Cc2c(C)ccc(C)c2)=O)cccc([N+](=O)[O-])c1N1CCOCC1 19010,C1(=CC(=O)NC(CC(C)NC(=O)COC2(C)CCC2)C)CCC(C)(C)CC1 19011,c1(NC(C2N(C(COCCOCC#C)=O)CC=C2)=O)ccc(C)cc1CC 19012,C1(C(=O)NCC2(C)CCN(C)C2)(CC)CCCN1C(c1ccc(F)cc1)=O 19013,CC(C)CC(C(N)=O)N(C(=O)C(C1CC1)N(C)C(C1CC12CCCC2)=O)C 19014,C1(C(=O)NCC(O)C(C)(C)O)(NC(C(c2cncnc2)C)=O)CCN(C)C1 19015,Cc1cc(C(=O)NCC(C)(C(C)C)NC(c2ncn(C)n2)=O)n(C(C)C)n1 19016,C1(C(N(CCC(=O)N(CC(CC)C)C)C)=O)CCC2CC12 19017,C1(CC)CN(C(=O)CC2(N(C)C(c3ccc(Cl)cc3)=O)CC2)CC(C)O1 19018,C(=O)(C(F)(F)C(F)F)N(CCN(C)C(C1CC1c1ccc(F)cc1F)=O)C 19019,c1(C2(C(N(CCCNC(C(CC)C)=O)CC)=O)CCOCC2)ccc(Cl)cc1Cl 19020,C(CCCCCCC(=O)NC(CO)C(C)NC(c1nc(C)oc1C)=O)SC 19021,CCC(CC(=O)N1CC(C(N)=O)C1)NC(=O)Cc1ccc(C)cc1 19022,CCC(C)(C#N)C(=O)N(CCCCN(C)C(C1C(C)C1(F)F)=O)C 19023,N1(C(C(C(C)C)C(C)NC(c2cncc(O)c2)=O)=O)Cc2cccc(F)c2C1 19024,C1(CC(=O)NCc2cccc(CNC(C3CC=CCC3)=O)c2)(OC)CCOCC1 19025,CCC(O)CC(=O)NCC(C)NC(C1(NC(C)=O)CCC1)=O 19026,c1(C(=O)NCC(CNC(C(C)NC(COC)=O)=O)F)ccc(=O)n(CCF)n1 19027,N1(C(CCSCCC)=O)CC2(C1)CN(C(c1cc[nH]c1C1CCCC1)=O)CCO2 19028,n1(CCNC(c2cc(CO)on2)=O)cc(C(=O)NC2CCOC2)nn1 19029,c1(C(=O)NCCC2(OC)CN(C(=O)C(C)NC(N)=O)C2)cccc2nsnc12 19030,C(C(O)C(=O)NCCCC1CCCN1C(c1cc(-c2ccoc2)[nH]n1)=O)SC 19031,C1(CC(=O)NCC(N2CCOCC2)C)(OC)CN(C(=O)C=C2CCOCC2)C1 19032,c1(CC(=O)NC23CC2CN(C(C2CCOCC2)=O)C3)c(F)cccc1Cl 19033,c1(CC)ccc(NC(C2(F)CCN(C(c3nn(C)cc3Cl)=O)C2)=O)cn1 19034,c1(C(=O)NC(=O)NC)ccc(-c2nnnn2C2CC2)cc1.C(CCC)=CCO 19035,N1(C(CC2N(C(C3C(C)(C)OCC3)=O)CC(O)C2)=O)CCC2(CCC(O)C2)C1 19036,c1(C(=O)NC(CN(C(c2ccc(CCC)s2)=O)C)C)cnc(OCC)cn1 19037,C1(C(N2CC(CNC(C(CC)(C)O)=O)(COC)C2)=O)CC(C)CC(=O)N1 19038,c1(C(=O)NCCC2CSCCN2C(=O)CC2CSCCS2)cccn2ncnc12 19039,Cn1cc(I)c(CN2CCC(CC(N3CCCC(C4(C)COC(=O)N4)C3)=O)C2)n1 19040,c1(C(=O)NC(C)CCNC(c2cc(O)n(C)n2)=O)cnn2cc[nH]c12 19041,CC1CN(C)CCC1NC(C1CC2(CCC2)CO1)=O.C12(CC1)N(C)C2=O 19042,c1(C(=O)NCCC2CCCN(C(=O)CC(F)(F)F)C2)ccn2ccsc12 19043,N1(C(c2c(C)nccc2)C(=O)NC(C)(C)C)CC(C)(C)c2ccc(Cl)cc21 19044,C1(NC(C(C)=CC)=O)CCCN(C(c2ccnc(N3CCC(C)C3)c2)=O)CC1F 19045,C1(C(N2CC(CNC(CCCCOC)=O)(COC)C2)=O)CC2CCCN(C1)C2 19046,c1(C(=O)NCC2CN(C(C3(OC)CCCC3)=O)CC2O)cc2oc(C)c(C)c2[nH]1 19047,N1(C(C2(C#N)CCC2)=O)CC(NC(=O)CCCn2ccnn2)C2(CCOCC2)C1 19048,CC(O)CCCC(=O)N1CCCC1C(C)(C)NC(c1cnccc1Cl)=O 19049,c1(CN(C(=O)C(c2ccccc2)C)CC=C)ccc(F)cc1F 19050,C1(n2cc(C(C(C)C)O)nn2)CCN(C(=O)COc2ccccc2Br)CC1 19051,CCCCC(=O)C(=O)N1CCN(CC(=O)NC2CC3CCCC3C2)CC1 19052,C(=O)(C(C)CC(C)C)NC(C(=O)N(CCC#C)C)COCC 19053,N1(C(CCC(=O)NC)=O)CCOC2(C1)CN(C(c1cc(C)cnn1)=O)C2 19054,N1(C(c2c(C(=O)OC)cco2)=O)CCN(C(C2(C)CCCS2)=O)CC1C(C)C 19055,N1(C(c2cccc(CCN(C)C)c2)=O)CC2CCN(C(C3CCC4CC34)=O)C2C1 19056,N1(C(C2C(NC(c3ccc(C)s3)=O)CCO2)=O)CCN(C)C(CN(C)C)C1 19057,C1(NC(C=Cc2nc(C)sc2)=O)CCC(O)CN(C(=O)C(C)(O)C2CCC2)C1 19058,c1(CC)cc(C(=O)NCC(C)CNC(=O)C(C(C)(C)C)n2ccnn2)ccc1Cl 19059,Cn1c(C(N2CCOC(C(=O)NC3CCC(CCO)CC3)C2)=O)ccc1C#N 19060,C1(CC(=O)OC)CN(C(=O)Nc2ccc(-c3nc(C)c(C)[nH]3)cc2)C(C)(C)C1 19061,C1(CNC(c2cccnc2C2CC2)=O)CCC(C(=O)NC2CCCC(O)C2)CC1 19062,N1(C(c2ccc(C)[nH]2)=O)CC2C3CCC(C2C1)N(c1nnc(C2CC2)s1)C3 19063,c1(C(C)C)ncsc1C(N1CC(CNC(=O)CNC(N)=O)C1)=O 19064,CCC(CC(=O)NC(C)(Cc1ccccc1)C(F)F)c1ccccc1 19065,N1(C(CCC2CCCN(C(CC(=O)OC(C)(C)C)=O)C2)=O)CC=C(C(=O)O)C1 19066,C(CCCCC(=O)NCC1CC=CCO1)N(C(C(C1CC1)OCC)=O)C 19067,N1(C(CNC(=O)CC(F)(F)F)=O)CCCCCCC1C(N1CCC(CF)C1)=O 19068,N1(C(CCSCC(C)C)=O)CCC(C)(NCC2CCC2CF)C1 19069,OCCC(N=c1nc(N2CCCC3(CC(O)C3)C2)c2[nH]ccc2[nH]1)C1CC1 19070,C(c1ccccc1Cl)=CC(=O)NCCCC(C)(C)NC(C1C(C)C1C)=O 19071,N1(C(C2CCN(C)C2)=O)CC2CCC2(CC(N2CCC3CCCC23)=O)C1 19072,c1(C(N2CCC(N(C)C(C3CC(C)(C)CN3C)=O)CC2)=O)nccc2[nH]ccc12 19073,N1(C(c2c(C)cncc2)=O)CCN(C(=O)COc2cccc(O)c2)CC1C 19074,c1(OC2CN(C(=O)C(F)=CCCF)C2)ccccc1NC(=O)C=Cc1ccsc1 19075,c1(NC(CC2N(C(C3CNC(=O)O3)=O)CCC2)=O)nc(Br)ccc1Cl 19076,Cc1nc(C(N2CCC(C)(NC(C3CC4C=CC3C4)=O)C2)=O)c2ccccn12 19077,N1(C(C2C(CC(C)C)C2)=O)CCCC12CCN(C(=O)Cn1nc(O)ccc1=O)CC2 19078,N1(C(C(n2cnc(C#N)n2)C)=O)CC(C)N(C(C2CC(Cl)(Cl)C2)=O)CC1C 19079,c1(C(N2CCC(NC(C3(C)C(CC)CCC3)=O)C(F)C2)=O)cc2ccccc2[nH]1 19080,C1(CNC(C(C)=C(C)C)=O)CCN(C(C2CNC(=O)N2)=O)C12CCC2 19081,c1(OC)ccc(C(F)F)cc1C(=O)NC1CC(O)CN(C(=O)CSC(F)(F)F)C1 19082,c1(NC(N(CC#C)C(C)C)=O)ccc(OC(C)C)cn1 19083,CCC(C)C(C(=O)NC)NC(=O)C(C)C1C(C(N2CCC2c2ccn(C)n2)=O)C1 19084,CC1CN(C(=O)CC2COCCN2Cc2cc[nH]c2)CCC1=O 19085,CC(C)C(CNC(=O)CCC(C)(C)F)C(=O)Nc1cn(C)nc1O 19086,C#CCCCCCCC(=O)NC(C1CCN(C(=O)CSC(C)(C)C)CC1)CO 19087,N1(S(CC(C)C)(=O)=O)CC2(CCN(C(c3ccn(C(F)F)n3)=O)C2)C1 19088,c1(C(=O)NCC2N(C(C(C)n3cccn3)=O)CC(O)C2)cncc2ccccc12 19089,C1(C(N2CCN(C(C(C(=O)OCC)(C)C)=O)CC2CF)=O)CCn2ncnc2C1 19090,N1(C(C(C)(F)F)=O)CCOC2(CCN(C(=O)C=Cc3c(F)ccc(Cl)c3F)C2)C1 19091,N1(C(c2cnccn2)C(=O)NCCCC)CCC(C(N)=O)C(C(C)C)C1 19092,c1(N2CC3C(N(C)C)C3C2)nc(=NCC2(C3CCC3)CC2)[nH]c2c1SCC2 19093,N1(C(CSCC#C)=O)CCC(C)(C(=O)NC(C)(C)CCOC)C1 19094,C(C(=O)NCC1CCCC1NC(c1nccn1C(C)C)=O)(C(C)C)n1ncc(C)c1 19095,c1(C(=O)NC(CC)CN(C(=O)C(O)C2CC2)C)cn(C(C)(C)C)cn1 19096,CN1CCn2ncc(C(=O)NC3CC4CCC(C3)N4C(c3nccn3C)=O)c2C1 19097,N1(C(C(C)SC(C)C)=O)CC2(C(=O)OCC3CC4(CCC4)C3)CCC1CC2 19098,c1(CNC(c2c(C)nco2)=O)cccnc1CNC(c1cc(Cl)cn1C)=O 19099,N1(C(C)=O)CCC(CNc2coc(CNC(C3CCCC3(F)F)=O)n2)CC1.CC.N.C 19100,c1(CNC(c2cc(C(C)(C)C)on2)=O)c(F)cc(Br)cc1F 19101,c1(C(C)=O)cc(=NCC(C2CC2)NC(=O)Cc2ccc(Cl)nc2)[nH]cc1[N+](=O)[O-] 19102,c1(CN(C)CC2(C(N=c3c(C(C)=O)c[nH][nH]3)=O)CC2)cc(Br)cnc1Cl 19103,C1(C(=O)NCC(CO)NC(=O)COCC(F)(F)F)CCNC1=O 19104,CCC(C)(C)C(O)C(=O)NCC#CCNC(C1CCC2(CC1)CC2)=O 19105,N1(C(CC(CC)SC)=O)CC2CN(C(C3(OC(C)C)CC3)=O)CC(C1)O2 19106,c1(NC(c2csc(C(=O)Nc3ccccc3I)n2)=O)ccc2c(c1)COC2 19107,N1(C(C(C)n2cccc2)=O)CC2CC1(C(=O)NC1CCOC1(C)C)C2 19108,C(=O)(C(C)CS(C)(=O)=O)NC1C(NC(c2ccc(-c3nc(C)[nH]n3)cc2)=O)C1 19109,C1(C(=O)NCC2CN(C(C(=O)N(C)C)=O)CC23CCC3)CCc2cnn(C)c2C1 19110,c1(C(=O)NC2CCN(C(=O)CSC(F)(F)F)C2)cc(F)c(F)c(F)c1 19111,C(=O)(C1=CCCN(Cc2ccc(Cl)c(I)c2)C1)Nc1cc(C(=O)OC)cc(F)c1 19112,c1(N(CCC)Cc2cc[nH]c3nccc2-3)cccc2ccccc12 19113,C1(C(C)(C)NC(COCCC=C)=O)CCN(C(=O)C(C2CCCCCC2)C)CC1 19114,c1(C(N(CCCCNC(CCC=C=C)=O)C)=O)cc2c(C)c(F)ccc2[nH]1 19115,N1(C(C(C(C)C)NC=O)=O)C2CCC1CN(C(=O)CN1CC=CC1)CC2 19116,c1(C(=O)NC23C(NC(CC(C)O)=O)CC(CC2)C3)ccc2nnc(S)n2c1 19117,N1(C(c2cc(C)c(C)o2)=O)CC2(CCC2)CC1CNC(=O)CC(C)(O)C1CC1 19118,C#Cc1ccc(CNC(C2CCCCN(C(C3(N(C)C)CCC3)=O)C2)=O)cc1 19119,c1(C(=O)NCCCN(C(c2c[nH]nc2NC(C)C)=O)CC)ccccc1NC 19120,N1(CCNC(C(CNC(C2(F)CC2)=O)N(C)C)=O)CCNC(=O)C1 19121,c1(C2(C(N(CCCNC(CCC=C)=O)CC)=O)CCC2)ncccc1F 19122,Cn1c(C(=O)NCCC2COCCN2C(C2CC2(C)C)=O)cc2ccsc12 19123,C1(C(N(C(c2nn[nH]n2)C)C)=O)N(C(C2CCN2C(C)(C)C)=O)CC12CCCC2 19124,C(=O)(CC(C)P(C)(C)=O)NCC(CNC(c1c(C(C)C)c[nH]n1)=O)C(F)(F)F 19125,C(c1cc(Br)cs1)=CC(=O)NC1CCCN(C(C2CCNC2=O)=O)C1 19126,N(C1COc2ccc(Cl)cc21)C(C1C2CN(C(c3ncccn3)=O)CC21)=O 19127,Cc1ccc(F)c(CNC(C2(C)CCCN(C(=O)C(C)OCCN(C)C)C2)=O)c1 19128,C(C)(CCCCNC(=O)C(c1cccc(Br)c1)O)NC(c1cc(C)[nH]n1)=O 19129,C(CC(CC)C(=O)NC(Cc1ccoc1)C(N1CCOCC(O)C1)=O)=CC 19130,C(=O)(CCS(=O)(=O)CC(C)C)NCC1CC(CNC(CN(C)CC)=O)OC1 19131,c1(CC)nc(C)c(C(=O)NCC2(CCNC(=O)C(C(C)C)NC=O)CC2)o1 19132,c1(C(=O)OC)cc(C)[nH]c(=NCC(C)(C2CC2)NC(=O)CC(=O)NC2CC2)n1 19133,C1(C)(NC(CC=C=C)=O)CCN(C(=O)CC(C)C)CC1 19134,c1(C(N2CCC(N(C(c3cc(C)c(O)cc3)=O)C)C2)=O)ccc2nc(O)[nH]c2n1 19135,c1(OCCC(=O)NCC2CC(NC(C3N(C(C)C)CCC3)=O)C2)cccc(F)c1 19136,CCCC(C)(O)CC(=O)N(c1ccc(C)c(-n2cnnn2)c1)C(CC)=O.C 19137,N1(C(c2ccc(C)o2)=O)CCN(C(=O)CCN2CCOCC2)C(SC(F)F)C1 19138,N1(C(C=CC2CCN(C(CCCOC(C)C)=O)CC2)=O)CCCC(N=[N+]=[N-])C1 19139,c1(C(N2C(CC(=O)NC)CN(C(=O)C(F)OC)CC2)=O)cc(C)c(C)cc1C 19140,CC1CCCN(CCNC(=O)CC2CCN(C(C3(C)CNC(=O)N3)=O)C2)C1 19141,N1(C(c2ccc(C(C)(C)C)[nH]2)=O)CC2CCCC2(Nc2ccnc3ncnn23)C1 19142,c1(NCc2c(C)nc(C)s2)nc2ccccc2nc1N1CCC(O)CC(C)(C)C1 19143,c1(C(N2CCC(CNC(C(C=CC)O)=O)C(C)C2)=O)cc(C)cc(OC)c1O 19144,N1(C(C(CC=C)C)=O)CC(CNC(c2cc(CCC)oc2C)=O)C2(CC2)C1 19145,O=C1CCC(=O)N1C1CCNC1.c1ccc(-c2ccco2)nc1 19146,C12(CC(=O)NCCC3CN(C(C45CCN(CC4)CC5)=O)C3)CCCCC1C2(F)F 19147,c1(N2CCC(SC)CC2)ccnc2c1CCCC2O 19148,N1(C(c2cn(Cc3cnns3)nn2)C)CCN(C(=O)CC2CC(F)C2)CC1 19149,CCC(c1cccc(Cl)c1)=CC(=O)NCC(CC)NC(c1ncoc1CC)=O 19150,C12(CNC(c3cc(C)c(C)o3)=O)CCCCC1CN(C(c1ccc[n+]([O-])c1)=O)C2 19151,C#CCCCCCCC(=O)NCC1(O)CCN(C(=O)C(C2CCCCC2)C)CC1 19152,C(CCCCC(=O)N(C(CNC(c1ccncc1C)=O)C1CC1)C)OC 19153,N1(C(C(C=C)(C)C)=O)CC2CCN(C(=O)CCOc3cc(C)cc(C)c3)C2C1 19154,C1(CCC(=O)NCCOCCC)CCCCN(C(C2CC3(CC(=O)C3)C2)=O)C1 19155,c1(NC(C2C=CCN2C(c2ccc(F)c(Cl)c2)=O)=O)cccc(F)c1Cl 19156,N1(C(Cc2cnc(C)s2)=O)CC2(CCC2NC(C2CCCC(=O)N2)=O)C1 19157,Cc1nc(CC(=O)NCC(O)CN(C(=O)C(C)(C)CN(C)C)C)c(C)s1 19158,c1(C(=O)OC)ccc(NC(=O)NC2CCC(F)CC2)c(OC(C)C)c1Cl 19159,c1(C(=O)NC2C(NC(Cc3ncc(C)o3)=O)C2)cncc(N)c1C 19160,n1(CC)nc(C(=O)NCC2COC(CNC(c3sncc3C)=O)C2)cc1O 19161,c1(CNC(=O)CC(C2CC2)NC(c2ccc(Cl)cc2)=O)cccc2[nH]ncc12 19162,N1(C(C(C)(CO)OC)=O)CC2CN(C(C3CCC(C)(C)OC3)=O)CC(C1)O2 19163,CC1(C)CCC(C)(NC(=O)CONC(C2CCCC(C#N)C2)=O)CC1 19164,C1(CNC(C2N(CC)CCC2)=O)(NC(=O)CCC(F)F)CCC(C)(C)CC1 19165,N1(C(COCC=C)=O)CC2CCC1CN2C(c1cc(CC(=O)OC)on1)=O 19166,C1(C2(O)CCOCC2)(C(N2CC(F)(CNC(c3c(CC)onc3)=O)C2)=O)CC1 19167,C1(C(=O)NCC(C)CNC(=O)CCCN2CCCC2)CC(C)OC(C)C1 19168,CCC(C)CCC(=O)N1CC(O)CC1C(=O)NCC1CCOC1C1CC1 19169,c1(C(N(CCC)CCNC(=O)C(C)(C2(C)CC2)OC)=O)cnn(C)c1C#N 19170,C1(NC(CC)=O)CCCC1C(=O)OC1(CO)CC(C)C1 19171,c1(OC)cc(C#N)ccc1C(=O)N(C)Cc1ccc(C)cn1 19172,C1(NC(C2(NC(C)=O)CCCC2)=O)CCCN(C(C2CC(=O)NC(=O)C2)=O)C1C 19173,Cc1n[nH]c(C)c1C(=O)NC(Cc1ccc(F)cc1)CC(=O)NCC1CCC1 19174,c1(C(N2CCC(NS(CCC)(=O)=O)C2)=O)cc(Cl)cnc1O 19175,c1(OC)ccc(C(=O)NCC2(NC(=O)C(C)=CC(C)(C)C)CCOC2)nc1Cl 19176,c1(CC)[nH]c(C(=O)NC2(C)CC(NC(=O)C(C)(O)CC)C2)nc1Cl 19177,Cc1ccc(F)c(C(N2CC3CC2C3NC(=O)C2=CCOC2)=O)c1 19178,C1(C)(CNC(CCOC)=O)CCCN(C(C2(C(F)F)CC2)=O)C1 19179,N1(C(C2CSCCN2C(=O)CN(CCO)CCO)=O)CCc2ccccc2C1 19180,c1(C(=O)NCCCOCCN(C(C(F)=C(C)C)=O)C)ccc(C(F)(F)F)s1 19181,N1(C(=O)NC(CC)CNS(C)(=O)=O)CC2OC(=O)N(CCCF)C2C1 19182,Cc1c(NC(C2CC(C)CN2C(C2C=CC(=O)N=N2)=O)=O)cc(Cl)cc1Br 19183,c1(SC)nc(=NCC(C)N(C)C(c2ccc3cc[nH]c3n2)=O)s[nH]1 19184,C1(CNC(C(C)OCCOC)=O)CCC(NC(C2(COC)COC2)=O)CC1 19185,c1(C(=O)NCCCN(C(C2(C)CC(=C)C2)=O)C2CC2)ccnc(C2CC2)c1 19186,N1(C(c2ccc(C)n2C)=O)CCN(C(c2n[nH]cc2F)=O)C(CS(C)(=O)=O)C1 19187,C(C#Cc1cn(CCF)nn1)NC(C1CCOC1)=O 19188,O=C(N=c1[nH]ccc2cc(Br)ccc12)C1CC2CC2N1C(c1ncccc1Cl)=O 19189,C1(NC(C=C2CCC(C)C2)=O)CCCCCCC1(C)C 19190,C(=O)(CCCC(F)F)NC(C1CCCCN1C(=O)C1=NOCC1)C 19191,c1(C(=O)NCCC(C)NC(=O)C=C(C2CC2)C2CC2)ccnc(N(C)C)c1 19192,N1(C(c2c(CC)scc2)=O)CC2CC(C1)CN(C(=O)C(C)(C)CC)C2 19193,N12CCC3(CCC(C3)NC(=O)C=C(C)C1)CC2.C1(CC)(COC)CCCCO1 19194,C1(C(N2CCOC(c3ccc(C)s3)C2)C(=O)NCCC)CC2(CCCO2)C1 19195,NS(=O)(=O)N1CC(C(=O)NC2CCCN(C(C3CCN(C4CC4)S3(=O)=O)=O)C2)C1 19196,c1(CC)noc(C(=O)N(C2CN(C(c3cn(CC)nc3C)=O)C2)C)c1C 19197,C(=O)(C(C#N)C1CC1)N1CC(CCN(C(C)(C)C)C(=O)OCc2ccccc2)C1 19198,C1(CNC(C(C)OCC)=O)CN(C(=O)Cc2sc(C)cc2C)CC1O 19199,c1(OCCC(=O)NCC2(OC)CN(C(C3C(COC)C3)=O)C2)ccc(Cl)c(F)c1 19200,C1(CN(c2ccc(Br)cc2)C)CCC(=O)N(C(=O)CSC2CCOC2)C1 19201,N1(C(C2CC3(CC(NC(CC(C(C)C)C)=O)C3)C2)=O)CC2(CCCN2C)C1 19202,CC1CC(C)(C)N1C(=O)C=CCC(C)(C)NC(=O)CSC(C)(C)C 19203,c1(C(=O)NCC(C)N(C(Cc2cc(COC)on2)=O)C)ccn2c1CCCC2 19204,C(CCCCCNC(c1c[nH]nc1C1CCC1)c1nnnn1CCCSC)OC 19205,CC(c1ccccc1)=CC(=O)NCC1CC(NC(c2cc(Cl)nn2C)=O)C1(C)C 19206,C1(C(=O)OC)CN(Cc2cccc(CO)n2)C2CCOCC12 19207,C(=O)(C(C(C)C)NC(=O)C(C)NC(C)=O)N1CC(C)(NC(C2(C)CC(=C)C2)=O)C1 19208,N1(C(c2c(CC)oc(C)c2)=O)CCN(C(=O)CC(F)(F)Cl)C2CCCCC2C1 19209,c1(SC)ccc(C(=O)NC2CCN(C(=O)CS(C)(=O)=O)C2C)cc1[N+](=O)[O-] 19210,CCC(C)(CC)C(=O)NC1CCN(C(c2sc(C)nc2C)=O)C(C)C1 19211,N1(C(=O)NC(C)Cc2ccccc2)CCC2(CCC2(C)C)C1 19212,c1(C(N2CC3CC(CNC(C4(CC)CC4)=O)C3C2)=O)cc(OC)c(O)c(Cl)c1 19213,N1(C(C=CC)=O)CCC(C(=O)NC2CC(CO)C23CCC3)=C(F)C1 19214,c1(C(=O)NC(C)CNC(=O)CC2CCCCC2)cn(C(C)(C)C)nc1C(C)(C)C 19215,N1(C(C2(CCOC)CCC2)=O)CCN(C(=O)CC2CCCC2)C(C(F)F)C1 19216,CC1CCC(C(=O)NOCCCC(C)(C)C)N1C(=O)C(=O)NC1CCC1 19217,C1(NC(c2ccncc2O)=O)CCN(C(c2cnc(-c3cnccn3)s2)=O)CC1 19218,Cc1c(C(=O)NC2CCC(CNC(c3ncc[nH]3)=O)C2)cnn1CC(C)(C)O 19219,Cc1nc2c(C)cc(C(=O)N(C(CO)CC(C)C)C)cn2n1 19220,c1(C(N2CC(CN(C(=O)C(c3cncnc3)=O)C)C2)=O)cccc(S(C)=O)c1 19221,C1(C(=O)NC(CCCNC(Cc2ccc(C(=O)NC)cc2)=O)C)CC(F)(F)C1(C)C 19222,N1(C(c2c(CCC)[nH]cc2)=O)CCC2(CCC2)C(NC(=O)CCS(N)(=O)=O)C1 19223,CCC(CC1CCCC1)C(=O)N1CC(COC)(NC(=O)Cc2nonc2C)C1 19224,c1(CC(N2CC(CCNC(C(C(C)OC)O)=O)C2)=O)cn2ccccc2n1 19225,CC1CCC(CNC(C2C=CC=CC=C2)=O)N(C(=O)Cc2cn(C)cn2)C1 19226,C(=O)(CCCCCC#N)NC1CCCN(C(c2c(C)noc2C(F)F)=O)C1 19227,C(=O)(C1COc2ccccc21)N1CC(CN(C(C(C)OCC2CCCO2)=O)C)C1 19228,C1(CC(=O)NCCC(C)N(CCC)C)CCN(C(c2cscc2C)=O)C1 19229,c1(C(=O)NCC(=O)NC(C#C)CC2CCC2)c(F)cc(Cl)cc1Cl 19230,C1(C(F)F)(CNC(C(C)O)=O)CCN(C(=O)CCN(S(C)(=O)=O)C)C1 19231,N1(C(C)C)CCN(C(=O)C(CCF)NC(C2CCC(C(N)=O)C2)=O)CC1 19232,C(=O)(CC(C)(C)C)NC(C1CCN(C(c2cnc(C(C)C)[nH]2)=O)CC1)C 19233,[N-]=[N+]=NC(CCC(N)=O)C(=O)NCCCc1cc(CO)on1 19234,C1(NC(C2(NC(C3C=CCC3)=O)C(C)C2)=O)CC2(CCC2)C1 19235,CCC(CC)(CO)NC(c1cncc(CNC(C2CCN(CC)C2)=O)c1)=O 19236,CCCC(O)(CCC)CC(=O)N1CCC(NC(c2ccc3nccn3c2)=O)C1 19237,N1(C(CCOCCN(C)C)=O)CC(CN(C(=O)CCOCC2CC2)C)C2(CC2)C1 19238,C(=O)(C(CCC)c1ccc(Cl)cc1)N(CC(C)NC(C=C(CCC)C)=O)CC 19239,C#CC1(C(=O)NCC(C)(F)C(C)(C)F)CCN(C(=O)CN(C2CCCC2)C)C1 19240,C1(N(c2ncc(Br)cn2)C(C2CCCO2)=O)CC2CCC(C1)N2 19241,C(=O)(C(F)C1=CCCCC1)N1CCC(O)(C(C)NC(C2C(CC)C2)=O)CC1 19242,c1(NC(C(C)C)C2CC2)nc2ccccc2nc1NCC1CCC(C)(C)O1 19243,C1(=O)NNc2ccc(cc2)S(=O)(=O)CN1.c1(OCCC)ccccc1C(F)(F)F 19244,C(c1ccoc1)=CC(=O)N(CC(Cc1ccccc1)NC(C1C(C=C)C1)=O)C 19245,C1(N(C(C(c2ccccc2)NC(C2CCC(=C)CC2)=O)=O)C)CCCC(C)(C)C1 19246,c1(C(=O)NCc2cc(C)c(C)nn2)coc2c1CN(C(=O)CC1CCOC1=O)C2 19247,C(=O)(CC(CNC(C1C=CCS1)=O)OC)NC1CCN(CC)C1 19248,C(CC1CCC1)(C(=O)NCC(O)C(C)C)NC(C(C)SCCCC)=O 19249,C1CCCCCC(=O)N1.C1(C)(c2cn(CCCCSC(C)=O)nn2)CCOCC1 19250,C(C(C(C)C)NC(c1ocnc1C(C)C)=O)NC(C(=O)NCCOC)=O 19251,C(=O)(C(CC)NC(=O)CC1(N(C)C)CC1)NC(CC)CSC 19252,C=C(Br)CC(C)(C)C(=O)NC1CCCCN(C(c2cc(COC)on2)=O)C1 19253,c1(C(=O)NCCN(C(=O)Cc2cc[nH]n2)CC)cc(C(C)=O)cs1 19254,C(CCC1CCC1)(C(=O)NCCc1ccon1)NC(c1cc(CO)on1)=O 19255,c1(C(=O)NCC(C)(CO)NC(c2nc(Br)c[nH]2)=O)c(F)cc(F)cc1F 19256,C1(C2CC2)(NC(C2CC(F)(F)C2)=O)CCN(C(C2CCCN2C2CC2)=O)C1 19257,c1(C(C)C)nc(NCCCC2CC2)cc(=NC2CCC3CC2C3(C)C)[nH]1 19258,CN1CC(NC(=O)CC2CN(C(C3CC4(CC4)C3)=O)CCO2)C2(CC2)C1 19259,CC1=C(C(=O)N2CC3=C(C2)CN(C(c2c(C)ncn2O)=O)C3)C(=O)OC1(C)C 19260,N1(C(CCCC(C)=O)=O)CC(C)CN(C(=O)CCc2c[nH]c(=N)[nH]2)C(C)C1 19261,c1(C(=O)NC2CC(CNC(C3(F)CCC3)=O)C23CCC3)cccc(C(F)F)c1F 19262,C1(CNC(C2(C(C)(F)F)CC2)=O)(NC(C2CCCCS2(=O)=O)=O)CCCCCC1 19263,C#CC1(C(=O)N(C(C)CCCC)C)CCN(C(C2CCC(COC)C2)=O)CC1 19264,C1(NC(C(C)(C)CF)=O)CCN(C(=O)Cn2ccccc2=O)CCC1CO 19265,CC1CCCN(C(=O)Cc2cccc(Cl)c2)C1CNC(=O)CC1CCCN(C)C1 19266,CCC(CNC(c1nnnn1CCSC)C1(CSC)CC1)CCO 19267,c1(CN(CC)Cc2cn(C)cn2)csc(-c2cnn(-c3ccccc3)c2)n1 19268,N1(C(C(COCC)C)=O)CCC2CN(C(=O)C=CC3CCCN3C)C2C1 19269,c1(C(N2CC(CC=C)(NC(C3CCC(COC)O3)=O)C2)=O)nccc(C)c1N 19270,CCCC(C)CCNC(=O)CCOCCNC(=O)CC1CCOC1(C)C 19271,Cn1c(N2CCC(C3(NC(=O)CC(C)(F)F)CC3)C2)c(C#N)c(=O)n(C)c1=O 19272,c1(C(N2CCCC2Cn2cc(COC(C3C(CC)C3)=O)nn2)=O)ccc(CO)cc1 19273,C(=O)(C(C(C)(C)C)n1cc(CCS(N)(=O)=O)nn1)NN1CC(S(C)=O)C1 19274,CCC(C)(CNC(=O)C(C1(O)CCCCC1)=CCC(C)(C)NC(=O)COC)CC 19275,c1(NC(Cc2nccc(CC)c2)=O)ccc2c(c1)CCC2N(C)C 19276,C12(C(NOCCOC)=O)CC(CO1)N(C(C1CC1c1cccc(F)c1)=O)C2 19277,C1(C(N(CC(C(=O)NC2(CC#C)CCC2)(C)C)C)=O)CC12CCCCC2 19278,Cc1ccc(C(=O)NC2CC(N(C(=O)CC(C)C3CC3)C)C2)c(O)c1C 19279,C(=O)(C1=NOC(CNC(C2CNC(=O)C2)=O)C1)NCCOCCCC 19280,c1(OC)c(C(=O)NC2CC3(NC(=O)C#CC4(C)CC4)COC2C3)cccc1F 19281,c1(NC(c2n(CC)ccn2)C)[nH]c(=NCCCn2cccn2)nc2ncn(C)c12 19282,Cc1nc(C2CC2)ccc1C(=O)NCC1CN(C(=O)C(F)C(F)(F)F)CCC1C 19283,C(CCN(C)C)(CN=c1[nH]c(=NCc2csnn2)[nH]c2cc[nH]c12)OCC 19284,N1(C(COC(C)C)=O)CC2CN(C(=O)Cn3nc(Cl)ccc3=O)CC2C1 19285,c1(C(=O)NCCOCCNC(C(C)NS(CC)(=O)=O)=O)ccc(CO)cc1F 19286,C1(Cc2cn(C3C=CCC(C(N4CCCOCC4)=O)C3)nn2)CCCS(=O)(=O)C1 19287,C1(C(=O)NC2(CO)CN(C(CC3(C)CC3F)=O)C2)CC2(C1)CC1(CCC1)C2 19288,C(=O)(CCC(=O)NN(C)C)N1C(CNC(c2ncn(C(C)C)c2)=O)CC(O)C1 19289,N1(C(C2N(CC#C)CCC2)=O)CCOCC(NC(=O)C(C)N(C)C)C1 19290,C1(C)(C(=O)NC2CCN(CC)C2)C=CCN1C(c1cc(Cl)cs1)=O 19291,c1(C(=O)NC(C2CCOC2)CNC(c2c(C(C)=O)ccs2)=O)cc(F)ccc1N 19292,c1(N2CC(C(NNC(c3ncc(C)c(O)c3)=O)=O)C2)cccc(Cl)c1[N+](=O)[O-] 19293,C1(c2cn(C)nc2)CN(C(C2C3CCCCC23)=O)CCN1C(C1(CCF)CC1)=O 19294,N1(C(c2c(C)cc(C)nc2)=O)C2COCC1CC(NC(C1(F)CC=CCC1)=O)C2 19295,c1(C(=O)NCC2N(C(C(C(C)C)C)=O)CCC2)ccn(C(=O)OC(C)(C)C)n1 19296,C1(NC(c2cnc(F)c(Cl)c2)=O)CCC2CCN(C(C3CC3(F)F)=O)C1C2 19297,Cc1ccc(Cl)c(C(=O)NC2CC(CNC(=O)Cc3nccn3C)C2)c1N 19298,C1(C(=O)NCC23CC(CN2C(c2sccc2Cl)=O)C3)(OC)CCS(=O)(=O)C1 19299,CC1CCc2sc(C(N3CC4CCCC3C4CNC(=O)C(C)C)=O)cc2C1 19300,C12(C(=O)NCCC(C)N(C(=O)C(C)OC3CCCC3)C)C=CC(CC1)C2 19301,N1(C(C=CC(C)(C)NC(Cc2scc(C)c2)=O)=O)CCC(C)C2(CCC2)C1 19302,C1(C(C)NC(C(C)OCCCC)=O)CCCN(C(c2cccs2)=O)C1 19303,c1(C(N(C2CCCCC2)CCNC(C(C2CCOC2)OC)=O)=O)c(C)ccn1C 19304,C1(NC(C2CCC=CCCC2)=O)CCC2CN(Cc3ccncc3Cl)CC2C1 19305,C(CN=c1nc(C2CC2)[nH]s1)C1CC(NC(CC2N(C)CCC2)=O)C1 19306,c1(C(N2CCC(CN(C(=O)C=CS(C)=O)C)C2)=O)ccc(F)c2ccoc12 19307,N(C(=NCC#Cc1cccc(C(F)(F)F)c1)N1CCC(C(C)(C)C)C1)CCOC 19308,C1(CCC)CCC(NCC2CCC2C(F)F)CC1 19309,c1(OC)ccc2cc(C(=O)NCC3CN(C(=O)C(C)S(C)(=O)=O)CCO3)[nH]c2n1 19310,C1(NC(c2ccc3[nH]ccc3n2)=O)CC2CCC1N(C(c1cscn1)=O)C2 19311,c1(NC2CC(C)C2)cc(N2CCOC(CNC(C)=O)C2)ncn1 19312,CC(C)C(C(C)NC(c1csc(Cl)c1)=O)NC(c1sccc1CC#N)=O 19313,C=CC1COCC1NC(=O)CN(C(=O)C(C)(C)CC)C1CCC1 19314,c1(C(=O)NCCNC(C(C2CC2)OC)C)n[nH]cc1C1CCC1 19315,N1(C(c2sc(C)c(O)n2)=O)CCCC2(CCC2NC(=O)CCCc2cccs2)C1 19316,CCCCCCCCC(=O)NCc1ccoc1C(=O)NCc1snnc1C 19317,c1(CCC(=O)OCC(=O)Nc2scc(C)n2)cccnc1Cl 19318,N1(CC(=O)NC2CCC(N(C(c3cncc(CC)c3)=O)C)C2)CCC(=O)NC1=O 19319,c1(CC(=O)NCCCOCCCNC(C(CC(=C)C)C)=O)cccc([N+](=O)[O-])c1 19320,C1(N(C(c2c(C)scc2)=O)C)CCCC(N(C(=O)COC2(C)CCC2)C)C1 19321,c1(C(=O)NCCCCC2CN(C(C3CC4(C3)CC4F)=O)C2)ccc(CO)cc1F 19322,c1(CCC)cc(C(=O)NC(C)(C(=O)NCCCCN(C)C)C2CCC2)no1 19323,N1(C(C(CC)F)=O)CCC(C)C(NC(c2ccn(C3CCC3)n2)=O)C1 19324,C1(NC(c2cc(C)c(C)o2)=O)CCC2CC1CN2c1nnc(-c2ccon2)s1 19325,C1(O)(CNC(C(C)OCCN(C)C)=O)CCCN(C(c2ncccc2N)=O)CC1 19326,C(=O)(C(F)C(F)(F)F)NC(c1c(CC)cccc1)CNC(=O)CC(=O)NC 19327,C(=O)(NNc1cc(F)c(F)c(F)c1)c1n(CCN)ncn1 19328,CC1CCN(C(C2(CO)CCN(C(=O)C3=CCCSC3)C2)=O)CC1(C)C 19329,C12(C(N3CC(C(C)C)C3)=O)CC(C)(CN1C(C1NC(=O)OC1C)=O)C2 19330,N1(C(C(COC)NC(C)=O)=O)CCN(C(C2CCC3(CC2)CC3)=O)CC1CC#N 19331,S(=O)(=O)(c1cccc(=NCCOC2CCCC2)[nH]1)OC(C(CC)C)C 19332,CCC(CC)C(=O)N1CC(NC(C2(Cc3cccc(F)c3)CC2)=O)C(C)C1 19333,C(=O)(CCCC#N)NCC(CC)N(C(=O)C(N1CCCC1)C1CC1)C 19334,C(=O)(C(C)C(C)(F)F)NC1(C)CC(NC(c2c(C(C)C)n[nH]c2)=O)C1 19335,Cc1cc(C)c(C(=O)NCCOCCNC(=O)C(C)Cc2cnn(C)c2)c(Cl)n1 19336,CN1CCN(C(=O)CCc2cccnc2)CC1C(=O)NC1(CO)CCOC1 19337,N1(C(CN(CCOC)C)=O)CC2CCC1C(NC(=O)C(C(C)(C)C)C1CCC1)C2 19338,Cc1ccccc1C1(C(=O)NCCC2CCCN2C(c2ccc(F)s2)=O)CCC1 19339,c1(C(=O)NC2(CN(C(C3(C(C)C)CNC(=O)C3)=O)C)CC2)ncc2ccccn12 19340,Cc1noc(C(C)OC2CC(OC(C)(C)C)C2)n1 19341,C1(c2c(C(=O)OC)c(C)no2)CCN(c2cc(NC3CC(C)(F)C3)ncn2)CC1 19342,CS(=O)(=O)CCC(=O)N1CCC(C2OCCC2NC(=O)CO)CC1 19343,C1(NC(c2c(OCCC)cccc2)=O)CN(C(C2CSCCS2)=O)CCC1F 19344,C(=O)(C(C)CNC(=O)C(Cn1ccnn1)NC(=O)CCn1cccc1)OC 19345,C(=O)(C1=C(C)OCCS1)NC1CC2CN(C(c3nn(C(CC)C)c(C)c3)=O)C1C2 19346,C(=O)(C(F)CCC(C)C)NC12C(NC(C3N(C(CC)=O)CSC3)=O)CC(CC1)C2 19347,C12(C(N3CCC(C)(NC(=O)CCN4CCOCC4)C3)=O)CC1CCC2(F)F 19348,C1(C(=O)NCCC2(NC(c3c(OC)scc3)=O)CC2)CCCC(C(N)=O)C1 19349,N1(C(C#CC(=O)N(C)C)=O)CC=C(CCNC(C2(F)CCS(=O)(=O)C2)=O)CC1 19350,C(=O)(C1=CCCCC1)N(CC(CC)NC(c1cccc(-c2cccs2)n1)=O)C 19351,CCCC(CCCNC(=O)C(C(C)O)NC(=O)OCC)OC(C)(C)C 19352,CS(=O)c1cccc(C(N2CCN(C(=O)CCc3cnc[nH]3)C3CCC23)=O)c1 19353,C(CC(C)(C)C)(C(=O)NCCOCCCNC(=O)CCCN(C)C)OC 19354,c1(C(=O)NCC(C)CNC(=O)CCc2cncs2)ccc2c(n1)NCC2 19355,C1(N(C(c2ccc(C3COC3)cc2)=O)CC)CCCN(C(c2cn[nH]c2)=O)CC1 19356,c1(CCC)ncc(S(=O)(=O)NC2CCCCC2OC)n1-c1ccccc1 19357,c1(C(N(CCCNC(C(C2CCCC2)OCC)=O)C)=O)c(C)nn2ncccc12 19358,C1(NC(c2c(CCC)nns2)=O)CN(C(=O)C(C)S(N)(=O)=O)CC12CCC2 19359,N1(C(c2c(C)[nH]c(C(C)(C)C)c2)=O)CCC2(CC(NC(=O)COCCF)CO2)C1 19360,C1(CNC(C2(CC#C)CCCC2)=O)CCC2(CN(C(C3CCCO3)=O)C2)O1 19361,c1(CC)nc(C)cc(=NC(=O)c2ccn3ncc(I)c3n2)[nH]1 19362,Cc1cc(C)c(CC(=O)NC2CC(N(C)C(c3ccc(C#N)[nH]3)=O)C2)s1 19363,c1(C(=O)NCC2=CCN(C(C3CC34CCCC4)=O)CC2)ccc2nn[nH]c2c1 19364,C#CCCCCCCC(=O)NC1(C)CCN(C(c2cc3c(nn2)CCCC3)=O)C1 19365,c1(OC)cccc(C)c1C1(C(=O)OCCSc2cc(OC)ccc2F)CC1 19366,C#Cc1cn(C)nc1C(=O)NC(C)CC(=O)N(CC(N)=O)CC(C)C 19367,c1(CC(=O)NCC(CNC(c2cc(C)c(C)o2)=O)F)ccc(F)c(Cl)c1F 19368,N1(C(C(C)NC(=O)NC)=O)CC2CC(NC(c3ccnc(C)c3Cl)=O)C1C2 19369,Cc1nc2ccc(C(=O)NCC3CCCC3NC(=O)CC3CC3(Cl)Cl)cc2n1C 19370,N1(C(c2cnc(CCC)s2)=O)CCCC(CN(C(C)C(=O)NC)CCC)C1 19371,N1(C(C(CC)OCC)=O)CCC2CCN(C(=O)CCc3cscn3)CC2C1 19372,C1(N(CC(=O)NCC)C)CC12CCN(c1nc(C(C)C)ns1)CC2 19373,CC(C)(C)CC(O)CC(=O)NC1CCN(C(c2c(N)cccc2F)=O)CC1 19374,C(=O)(CCCCCCN=[N+]=[N-])NCC1CCCN(C(C(OC)OC)=O)C1 19375,C1(C(N2CC=CC(O)C2)=O)(NC(c2cc(COC)no2)=O)CCC(C)(C)C1 19376,N12CC(O)CC1C2=O.C1(NC(=O)OC(C)(C)C)CC(NC(C2(Cl)CC2)=O)C1 19377,C1(NC(=O)NC(C)C)CCCC(Nc2nnc(C(C)C)s2)C1 19378,N(C(C)=[SH]n1nc(-c2ccc(F)cc2)o1)(c1c(C)cccc1)C1CCCC1 19379,c1(OC)ccc(C)c(C(N2CC(NC(=O)C(C)CSC)C(C)(C)C2)=O)c1 19380,C1(NC(C(C)C2CC2)=O)CN(C(=O)CCc2cccc(Cl)c2)CCC12CCC2 19381,Cc1cc(N)cnc1-c1nc(CC2N(C3CC3)CC2(C)C)nn1-c1ccccc1 19382,C(=O)(C1=NOC(C)C1C)N1CCC(NC(c2cc(C(C)C)on2)=O)(CO)C1 19383,Cc1cnc(C(N2CCC(NC(c3cc(F)c[nH]3)=O)C(CO)C2)=O)c(C)c1 19384,CC(CC(C)(C)C)C(=O)NCc1cc(C(=O)NCCCC2CC2C)n[nH]1 19385,CC1CCN(C(c2cn(CCO)nn2)=O)CC1C(=O)N(CC(F)F)C1CC1 19386,C(=O)(C(C)(C)C(C)C)N(CC(CNC(Cc1ncc(C)s1)=O)O)C 19387,C(CCCCCNC(C1CCCN1C)=O)NC(C=CCCC=C(C)C)=O 19388,C(=O)(CCCCC(=O)N1CCC(C)N(C(C2CCCN(C(N)=O)C2)=O)CC1)NC 19389,CC1CC(=O)NC(C(=O)NCC2(CNC(c3nocc3C3CC3)=O)CC2)C1 19390,N1(C(C(C)NC=O)=O)CCC2CN(C(c3cnc(O)nc3O)=O)CCC12 19391,N1(C(C(C(C)C)OC)=O)CC(CNC(c2cccc3nn[nH]c23)=O)CC12CCC2 19392,C12(C(=O)NCC(C(C)C)NC(=O)C(C)(C)c3cncs3)CC3CC(CC1C3)C2 19393,c1(C(N(CCN(C(CSCC)=O)C(C)C)C)=O)nc(C)ncc1Cl 19394,N1(C(c2c(C)noc2N)=O)CCCC(NC(=O)CC(O)C2CCCC2)CC1 19395,C12(C(=O)NC3CCN(CC)C3=O)CC(CCO1)N(C(=O)Cc1cc(C)cs1)C2 19396,C(=O)(CC(=O)NC(C)CNC(=O)C(C)C1CCC1)NCC#C 19397,N1(C(C2CC(CN(C)C)C2)=O)CC2CCCC(NC(=O)C(C)(C)F)C2C1 19398,CC(C)CC(C)CC(=O)N(C1CCCN(C(=O)CC2=NNC(=O)C2)C1)CC1CC1 19399,CC1CCCC(C(N2CCN(c3ccc(C(=O)O)cc3)CC2)=O)C1C 19400,CC1CN(C(c2ncc[nH]c2=O)=O)CC(CCNC(c2cn(C)nn2)=O)O1 19401,C(=O)(CC(F)(F)C(F)F)N(CCCNC(=O)CNC(C1CCCCC1)=O)C 19402,C12(C(N(CCC3CCN(C(c4nc(C)sc4C)=O)CC3)C)=O)CC3CC1C2C3O 19403,N1(C(c2nnc(C)o2)C)CCCC(CNC(c2cn(C3CCOCC3)nn2)=O)C1 19404,C(=O)(CCC(=O)NN(C)C)N1CC(C2CC2)(C(=O)NC(C2CCCCO2)CC)C1 19405,Cc1cc(NC2CCOc3ccccc3C2)ncc1S(=O)(=O)N(C)Cc1ccns1 19406,C1(N(C)C)(CNC(C2(NC(C3C(C(C)C)(CC)C3)=O)CCC2)=O)CCCC1 19407,c1(C(N2CCCC(CNC(CSC(C)(C)C)=O)C2)=O)cccc2nonc12 19408,N1(C(c2cnco2)=O)CCS(=O)(=O)CC1c1ccc(COc2ccccc2)cc1 19409,N1(C(C2CC=CC(NC(C(CC)(C)O)=O)C2)=O)CC=C(CO)CC1 19410,C(=O)(C(Cn1cccn1)NC(=O)C(C=C)OC)N(C(C#C)C)C 19411,C(=O)(C#CC1CCCO1)N1CCC(NC(c2c[nH]c3nccc-3c2)=O)C(O)C1 19412,c1(C(=O)NCC2CCCC(NC(C(C)c3cccs3)=O)C2)ccc2nccn2n1 19413,C=CCC(C(=O)NCC1CC2CCC(C1)N2C(=O)C=NOC)C(C)(C)C 19414,C12(C(N3C4CN(C(CC5(C)CCC5)=O)C(C4)C3)=O)CCCCN1CCC2 19415,C(C)(CNC(c1ccc(-c2nncn2CC)cc1)=O)(C(C)C)NC(CC)=O 19416,C#CCCC(O)C(=O)NCCNC(C1CCC(Cc2cccc(Cl)c2)C1)=O 19417,CC(C)(C(=O)NC(CNC(=O)C(C)(C)n1cnnn1)CC(F)(F)F)C(F)(F)F 19418,CC1(C(=O)NCCc2n[nH]cc2C(=O)NCCC2CC(O)C2)CCCC1O 19419,N1(C(c2c(F)ccc(C)c2)=O)CCC2(CCCN2C(C2CSCCS2)=O)C1 19420,N1(C(c2cc(C)cc(F)c2N)=O)CCC2(CCCC2NC(c2ccon2)=O)CC1 19421,CC(C)C(CC(=O)NCCCc1ccsc1)NC(c1c[nH]nc1C(F)F)=O 19422,C(C(C)(C)C(=O)NC1C2CN(C(C3CCCN3C(C)=O)=O)CC12)NC(C)=O 19423,c1(-c2cn(C3CC(C(=O)OC)C3)nn2)cc(F)c(F)c(F)c1 19424,C(C(=O)NCc1ccoc1C(=O)NC(CO)C1CCC1)(C(C)(C)C)OC 19425,CCCC(C)C(=O)NC(C)(CNC(=O)Cc1nccc(OCC)n1)C1CC1 19426,C1(C(C)C)COCCN(C(=O)C=CC(C)NC(=O)CC(F)(F)F)C1 19427,N1(C(C2CCCN(C(C)=O)C2)=O)CCCC2CN(CCC3CCCCCC3)CC12 19428,C(=O)(C(F)CC(C)(C)NC(=O)CC(C)(C)CC)N1CCCC(C=C)C1 19429,C1(N(CCC)C(c2[nH]cnc2C)=O)CCN(c2nnc(C3CC3)o2)CC1 19430,c1(N2C(C)CN(C(c3cc(=O)cc(Cl)[nH]3)=O)CC2)ncc(C#N)cc1Br 19431,c1(C(=O)NCC(C)NC(c2c(F)ccc(F)c2O)=O)c(F)ccc2nc[nH]c12 19432,C1(NCCCn2c(C)ncc2)CN(C(=O)CC2(c3ccccc3)CC2)CC12CC2 19433,c1(C(=O)NC(C)C(C)NC(c2sccc2-n2ccnn2)=O)cccc([N+](=O)[O-])c1 19434,C(CC(C)(C)NC(=O)CCOCC1CCC1)=CC(=O)N(CCCC#C)C 19435,C1(C)(CNC(C(C2CCN(C(c3coc(C4CC4)n3)=O)C2)C)=O)CCCOC1 19436,Cc1cc(CC(N2CCC(F)C(NC(c3ccoc3Cl)=O)C2)=O)ccc1CO 19437,N1(C(c2c(C)ccs2)=O)CC2CCC(NC(c3ccc4n[nH]cc4c3)=O)(C2)C1 19438,C(=O)(CCCCCS(N)(=O)=O)NC(CC(C)NC(c1c(CSC)cccc1)=O)C 19439,CC(C(=O)NCc1cn(C2CN(C(c3ncccc3Cl)=O)C2)nn1)C(C)(F)F 19440,C12CCN(C1)C2=O.C1(C2CCCO2)(CN(CC(=O)NC)C)CCCC1 19441,C(=O)(C(C#N)C(C)(C)C)N1C(CC)CN(C(c2c(C)ncnc2O)=O)CC1 19442,C1(CNC(C=CCCC)=O)CCN(C(=O)C(C)CSC)CC1C1CC1 19443,CN1CC2CCN(C(=O)CC3CC3CNC(C3CS(=O)C3)=O)CC2C1 19444,c1(C(=O)NC2CC(C)N(C(c3ocnc3C(F)F)=O)C2)ccc2c(c1)CCC2 19445,C(=O)(CS(=O)C(F)(F)F)NCC1C(N(C)C)CN(C(CC=CC=C)=O)C1 19446,CCCCCC(COC)C(C)NC(=S)NCCC(F)(F)F 19447,N1(C(C2N(C(C)(C)C)CC2)=O)CCCC2CN(C(=O)C3CC3)CC12 19448,N1(C(c2c(CC#N)cccc2)=O)CCCCC(NC(C23CC(CF)(CO2)C3)=O)C1 19449,C=CCC(CC(F)F)C(=O)NCC12CC1CN(C(c1cccc3ncnn13)=O)C2 19450,C1(CNC(C2CC(C)OCC2)=O)COCCN(C(c2ccnc(C(N)=O)c2)=O)C1 19451,c1(CNC(C(=O)NC(CC)CC2CCCO2)=O)cccc(F)c1Br 19452,c1(C(=O)NC(C(C(C)C)O)c2ccccc2)n[nH]c2c1CCCCC2 19453,N1(C(C=Cc2c(OCC)cccc2)=O)CC(C2CN(C(=O)C3=NOC(C)C3)C2)C1 19454,CCC(CC(=O)NC1CCCC(NC(C2CC(O)CN2C(C)=O)=O)C1)C1CC1 19455,CN1CCC(NC(=O)CCF)C12CCCN(C(c1cccn3nncc13)=O)C2 19456,C12(NC(C3CCCN(C(C(C)(C)C)=O)C3)=O)CCCC1NCC2 19457,C12(CNC(c3c(C(C)C)cccc3)=O)CCCC1CN(C(=O)C(C)N(C)C)C2 19458,c1(N(C)C)ncc(C(=O)NCC2CC(O)CN2C(c2ccc(O)nc2)=O)cc1Cl 19459,c1(CN(C(=O)NC2CCC(c3ccc(F)cc3)C2)CC)csc(C#N)c1 19460,N1(C(c2ccccc2)CC)CCN(Cc2ccc(Br)cn2)C(CC)C1 19461,C(=O)(C1=COCCO1)NCC(C)(C1CCC1)NC(c1cc(CN(C)C)on1)=O 19462,C(=O)(C1=C(Cl)CCOC1)NCC1N(C(CCCCCN(C)C)=O)CC(O)C1 19463,Cc1nc(C)n(O)c1C(=O)NC1CCCN(C(=O)C(C)(C)C(N)=O)C1 19464,N1(C(CC(C)n2ccnc2)=O)CCCC(CNC(C2(C3CCCO3)CC2)=O)C1 19465,C1(C(N2CCC(C(C)NC(=O)C(C)(C)F)CC2)=O)CC2(CCO1)CC2 19466,c1(Oc2ccc(C(=O)OC)cn2)cc(NCCO)cnc1-c1ccc(SC)cc1 19467,N1(C(C=CCN(C)C(c2ccc([N+](=O)[O-])o2)=O)=O)CCC2CCCCC2C1 19468,C1(C(N2CC(COC)(NC(=O)Cc3sc(O)nc3O)C2)=O)C2CCC1(C)C2(C)C 19469,Cc1ccc(C)c(NC(=O)CCC(C)NC(=O)CCc2nncn2C)c1 19470,Cc1cc(C(N)=O)cc(C(=O)N(C)CCN(C(C2CCCC2(F)F)=O)C(C)C)c1 19471,N1(C(c2c(OC)n[nH]c2)=O)CCC2(CC1)CN(C(=O)COC1CC=CC1)C2 19472,C=CCC(C)(C)C(=O)NC1CCC1NC(c1cccc(C(C)=O)c1)=O 19473,O=S(=O)(c1ccc(N2CCC3(C2)CC(F)(F)C3)c(Br)c1)NCC1CSCCS1 19474,C=CCC(C)(CC)C(=O)N1CCC(C)(CC(=O)NCCc2cc[nH]n2)C1 19475,N1(C(c2nsnc2O)=O)CCC(F)(C(=O)NCCN2CCCC2=O)C1 19476,CC(O)(CNC(=O)C(C1CCC1)NC(c1cc(O)ccc1F)=O)C(F)(F)F 19477,N1(C(C(C)OCC#C)=O)CCC2CCC(NC(c3ccc(Br)cc3)=O)C12 19478,C1(C(=O)NCc2cc(C(=O)NCCC3(C)CCCO3)no2)CCC(O)CN1C 19479,c1(OC)ncc(Cl)c(N2CCCC(NC(C3(ON4CCCCC4)CCC3)=O)C2)n1 19480,N1(C(CCN(C)C(c2[nH]ccc2C2CC2)=O)=O)CC=CC(O)C1 19481,N1(C(c2c(C)nsc2)=O)CCC(C(C)NC(=O)CC2CCCO2)CC1 19482,Cn1nc(CO)c2c1CN(C(c1cc(-c3ccccc3)ns1)=O)CC2 19483,c1(CC(=O)NCC2(OC)CN(C(C(CC=C)(C)C)=O)C2)ccc(S(C)=O)cc1 19484,C1(C(=O)NCCc2c(C(N(CCC(=O)NC)C)=O)c[nH]n2)OCCOC1C 19485,O=C(CC1CCOC1)NOCC(=O)NCCOCCSc1nc[nH]n1 19486,C(C(C)(C)C(=O)NCC1CCC(CC)CC1)NC(CCSCCC)=O 19487,O=S(=O)(c1ccc(Cl)c2ccccc12)NC1CCc2nn(C3CCSC3)cc2C1 19488,C1(CC=C)(NC(=O)CC(C)F)CCCN(C(c2cc(C(F)F)ccc2Cl)=O)C1 19489,CC(C(=O)NCC1(O)CCCN(C(c2ccn3c2CSCC3)=O)C1)C1=CCCC1 19490,CC(C(=O)N1CCCC1C(C)NC(C1(C)CCC(=O)N1)=O)S(N)(=O)=O 19491,Cc1cccc(F)c1C(=O)NC1CC(N(C)C(C2CC3COCC3C2)=O)C1 19492,N1(C(CSCC#C)=O)CCC(NC(=O)C(C(C)C)n2cnnn2)C1C1CC1 19493,C(=O)(CC(C)CNC(C1CCNC(=O)C1)=O)N(C(COC)COC)C 19494,c1(C(=O)NCCN(C(C2(C)CC2C(F)(F)F)=O)CC)ccc(C)cc1C 19495,C1(C(=O)NCC(=C)Br)CC2CC1CN(C(=O)CCC1OCCO1)C2 19496,N1(C(C=C(C)C(C)(C)C)=O)CC(N=[N+]=[N-])CC1C(=O)NCc1cscn1 19497,N1(C(=O)CCc2cccs2)CCCN(C(C2CC3CC2CC3O)=O)CC1 19498,N1(C(C2(F)CCC(C)CC2)=O)CCOC2(C1)CN(C(=O)CCC1CC1(C)C)C2 19499,c1(OCC)ccc(C(=O)NCC2CN(C(c3ccnc(C)c3)=O)CC2C)cc1O 19500,C1(N(C(c2n(CC)ncn2)=O)C)CCCCN(C(=O)C=Cc2ccc(C)cn2)C1 19501,N1(C(C(Cc2cn(-c3c(C(=O)O)ccnc3)nn2)O)=O)CCNC(=O)C1C 19502,N1(C(CC=CC=C)=O)CCC(CNC(=O)CC(C(F)(F)F)OC)C(F)(F)C1 19503,CC1(NC(=O)CNC(N)=O)CCN(C(C2CCCC(F)(F)C2)=O)CC1 19504,C1(C(=O)NC(C(=O)NCCC(=O)NCC)Cc2cn[nH]c2)CCCCCCC1 19505,n1(CCC(=O)NC(CC(CC)=O)C(=O)O)ccc2ccc(F)cc12 19506,N1(C(C2(NC(CN=[N+]=[N-])=O)CCC2)=O)CC=CC(O)C1 19507,c1(CC)onc(OC(c2cc(-c3cn(C4CN(CC)CCO4)nn3)c[nH]2)=O)c1C 19508,C(C(O)C(=O)N(CC(C)NC(=O)C(CN(C)C)N(C)C)C)=CCCC 19509,c1(NC(C2CCC(N(C(=O)COCC3CCCO3)C)CC2)=O)nnc(O)cc1O 19510,c1(CCC)nc(C)c(C(=O)NCC2CC(NC(=O)C=Cc3cccs3)C2)s1 19511,CCC(CC)(CCNC(=O)CN1CCC(=O)CC1)NC(C1C(C)(C)C1(C)C)=O 19512,C(CCC(C)(C)C)(c1n(CC=C)nnn1)NCc1ccc(-n2cncn2)cc1 19513,c1(OC)cc(C(=O)NCCC2CCN(C(c3ccc(Cl)cn3)=O)CC2)nc(C)c1 19514,C1(N(C(c2nc(C)sc2)=O)CC2CC2)CCN(C(=O)CC2(O)CCOC2)CC1 19515,Cc1nc(N2CCN(C(C34CCOC3CCOC4)=O)CC2C)c(Cl)cc1C#N 19516,C1(CNC(COCCCC)=O)CC2(CCN(C(c3cc(C4CC4)ns3)=O)CC2)C1 19517,N1(CC(=O)N(CCCC)CC)CC2CCC(NC(=O)CNC3CCOC3)CC2C1 19518,c1(CC)nc(C(=O)NC(CNC(C2CCOC2)=O)C(C)C)c(N)s1 19519,c1(C(=O)NC2CC(NC(C3(c4ccn(C)c4)CC3)=O)C2)csc(S(N)(=O)=O)c1 19520,c1(C(C)=O)ncc(C(=O)NC2CCC(NC(=O)C(C)n3cnnn3)C2)s1 19521,C1(C(=O)NCC(C)CNC(=O)CC2COC(=O)N2)CCC12CCC2 19522,N1(C(C(C)C2CCCO2)=O)CCC2CCN(C(c3ccc(O)nn3)=O)CC2C1 19523,c1(C(C)C)nnc(C=CC(=O)NC2CCCCC2NC(=O)CCn2cccn2)o1 19524,Cc1cccc(C)c1NC(=O)C(N1CCCC(CC(=O)N(C)C)C1)CC1(C#N)CC1 19525,C(c1cc(Cl)ccc1Cl)=CC(N1CC(CNC(C2(COC)CCC2)=O)C2C1C2)=O 19526,c1(OC)ccc(C(N2CC(NC(=O)CC(C)OC)C(F)C2)=O)c(F)c1 19527,C(C)(CC(=O)N1C2CCC1CC(NC(C1CCC1)=O)C2)(C(F)(F)F)N(C)C 19528,C(=O)(C(F)CC(C)(C)NC(c1ccc(O)cn1)=O)N1CCN(C)CC1 19529,C(C(C(=O)NCC(CC)NC(=O)C(c1cncn1C)O)c1ccccc1)OCC 19530,S(=O)(=O)(c1cnn(C)c1)N1CC(CC(N2CCC(N(C)C3CC3)CC2)=O)C1 19531,S(=O)(=O)(c1cc(C)c(C)s1)NC(C1CCCN(CCOC)C1)C 19532,c1(OC)ncc(C)cc1-c1ccc(C2(NC(c3c(Cl)cnn3C)=O)CCC2)cc1 19533,N1(C(CCC#CC)=O)CCc2nc(CNC(c3cc4n(c3)CCCC4)=O)sc2C1 19534,C1(CNC(c2cc(C(F)F)cs2)=O)CCCN(C(c2conc2C2CCC2)=O)C1 19535,C1(C(C)OC(=O)CC(c2cccnc2)NC(=O)OC(C)(C)C)CC2(C1)CC(O)C2 19536,c1(C(=O)NC(CNC(C2C(C)C2C)=O)C2CC2)ccnc(NS(C)(=O)=O)c1 19537,N1(C(Cc2n(C)cnc2)=O)CCN(CCNC(N)=O)CC1 19538,c1(C(=O)NCCN(C(C=CSC)=O)C)cccc2c1OCCN2 19539,C1(C2CCCN(C(=O)C3=CCCC3)C2)(NC(c2cc3cnccc3o2)=O)CC1 19540,c1(CC)nn(C)c(Cl)c1C(N1CCC(C)(CNC(C2CC23CCC3)=O)C1)=O 19541,c1(C(N2CCC(O)(CCNC(c3coc(Cl)c3)=O)CC2)=O)ccn2nccc2n1 19542,C(C(=O)NCc1ccnc(O)c1)(C(C)C)NC(CN(C(C(C)C)=O)C)=O 19543,C12(NC(COC(C)C)=O)CCC(NC(c3cc(Cl)ncn3)=O)(CC1)C2 19544,CCC(CC(=O)N1CC(O)(CN(C)C(c2cc(C(N)=O)ccn2)=O)C1)C1CCC1 19545,c1(C(=O)NCC2CCCCN(C(C(C=C)O)=O)CC2)c(C)nn2c(C)cccc12 19546,N1(C(C(=O)NC)CC(C)c2ccccc2)Cc2ccccc2C1COC 19547,C(C)(C)(CCCC(=O)N1C2CCCC1COC2)NC(C(CC)COC)=O 19548,S(=O)(=O)(c1ccc2ccccc2c1)N1CC2N(C(=O)C(F)Cl)C(COC2)C1 19549,N1(CC)CCCCC1CNC(C1CC(=O)N(C2CCCC(C)C2)C1)=O 19550,C12(CC(=O)NCCCCCN(C(C3CC(SC)C3)=O)C)COCC(C1)C2 19551,C1(CNC(CC(CNC(=O)C(N2CCOC2=O)C)OC)=O)CCCCC1(C)C 19552,c1(C(N(C(CNC(C2(C)C(C(=O)OC)C2)=O)C)C)=O)cc(-c2ccncc2)on1 19553,C(=O)(C(C)CC(C)(F)F)NC1C(NC(C=CSC)=O)COC1 19554,C1(C(=O)NCCC(N)=O)C=CCN1C(=O)CC1COC(=O)C1 19555,Cc1cc(C(=O)NC2CCC2NC(=O)C=CBr)cc(Cl)c1Br 19556,c1(NC(COC)=O)ccc(C)c(C(=O)NC2CC(NC(=O)CC3COCC3O)C2)c1 19557,C12(C(=O)NCCCC3(NC(C4C(C)OCC4)=O)CC3)CC3CC1C2C3 19558,C1(C(=O)Nc2n[nH]c(-c3ccc(Cl)c(Cl)c3)n2)CCn2c(O)nnc2C1 19559,C1(C(N2CC3C(C(=O)OC)(C3)C2)=O)CCCCN(C(=O)Cn2cccn2)C1 19560,C(=O)(C(CC(C)C)C(N)=O)N1CCCC(O)(c2cn(Cc3c(C)sc(Br)n3)nn2)C1 19561,C(=O)(C(F)(F)C(F)(F)C(F)(F)F)NCC(CO)NC(C1(C)CC(O)C1)=O 19562,N1(CC)CCOCC1C(=O)N(CC(C)(C)CNC(C1CCCC1OC)=O)C 19563,N1(C(c2n[nH]c(CC)c2Br)=O)CC(C)(C)CC1CNC(C1CCC1C)=O 19564,c1(C(C)C(=O)NCCCNC(=O)CC2NC(=O)NC2=O)ccc([N+](=O)[O-])cc1F 19565,N1(C(C2C=CCCC2)=O)CC2CC1(C(=O)Nc1ccccc1)C2 19566,C1(C(C(=O)NC)N(C2CC(n3cncn3)C2)C)CC2CCC1C2 19567,C(=O)(C1SCCc2ccccc21)N1CC(CNC(C(=O)NCC)=O)C(C)C1 19568,c1(CC(C)C(=O)NCCC2(O)CCN(C(=O)CC3(C#N)CC3)C2)cccc(F)c1 19569,Cc1ccoc1CNC(c1cnns1)=O 19570,C1(C)(CNC(C(C)C2CCCC2)=O)CCN(C(=O)CC2SC(=N)NC2=O)CC1 19571,N1(C(CC(CC)C)=O)CCCCC2(CCN(C(c3ccccc3SCC)=O)C2)C1 19572,c1(C(=O)NCC2CN(C(C3C(C=C)C3)=O)C(C)(C)C2)cc(Cl)cc(Cl)c1O 19573,Cc1ccc(SCCC(=O)NCC2CN(C(=O)OC(C)(C)C)CC2O)cc1C 19574,C1(NC(C2=NNC(=O)C2)=O)CCCC2CN(C(C3CC=CC(O)C3)=O)CC12 19575,CC(C)CC(O)C(=O)NC(Cc1ccco1)C(=O)N(C)CC1(O)CCC1 19576,O=C(CCCCCCCO)N(C1CCN(C(c2cncc(Br)c2)=O)C1)CCO 19577,C12(C(=O)NCCCCC)CCCC1CCN2C(c1ccc(CC)cn1)=O 19578,Cc1ccc(C(N2CC3(CCC3NC(=O)C(C)OCC3CC3)C2)=O)c(Br)c1 19579,C(=O)(CCC(CC)OC)NC1CCN(C(CCCC)=O)C1CC 19580,CCC(CC(F)F)C(=O)N1CCCC1CN(C)C(c1c(F)ccc(C)c1N)=O 19581,C1(CC)CN(c2ccccc2)CCN1C(c1cc(-c2ccccn2)[nH]n1)=O 19582,Cc1cc(C(c2nnnn2CCC2(C)CC2)NCC2CC23CC3)c2c(c1)CCC2 19583,C(CC(C(C)(C)C)NC(=O)C(O)c1ccsc1)N(C)C(c1cc2n(n1)CCO2)=O 19584,C1(C(=O)NCC(C)(C)NC(CCC=CC)=O)CCN(C(=O)C(C)(C)C)CC1 19585,C(=O)(C(F)(F)C(O)C(C)C)N1CCCCC(NC(c2c(C)nc(CCC)o2)=O)C1 19586,C1(C(=O)NCC(CNC(=O)COC2CCC2)OC)CCOC1c1cccnc1 19587,N1(C(=O)NC(c2nc(=O)[nH][nH]2)C)CCCC2(C=CCO2)CC1 19588,N1(C(C2C(C#C)C2)=O)CCN(C(=O)COc2ccc(Cl)c(Cl)c2)CC(O)C1 19589,c1(C(=O)OC)ccc(F)c(C(=O)NCC2CC(NC(=O)C(F)(F)C(C)O)C2)c1C 19590,C1(C(N2CC(C)OCCC2)=O)CCCCCCN1C(=O)CCCCC#N 19591,C1(NC(CN(c2ccncc2)C)=O)CCC2CN(C(C3CC(=C4CC4)C3)=O)CC12 19592,CC(C)C(Cc1ccccc1)C(=O)NCCC(C)N(C)C(c1cc(C#N)c[nH]1)=O 19593,c1(NC(C2N(Cc3ccc(C)[nH]3)CCNC2)=O)cc(C#N)ccc1O 19594,C1(NC(c2c(CCC)n[nH]c2)=O)CN(C(C2C(C)(C)C2(C)C)=O)CCC1O 19595,CC1(CNC(N2CCC(C(=O)OC(C)(C)C)CC2)=O)OCCc2sccc21 19596,N1(CC)CC(C(N2CC3CC2C3NC(c2nccnc2N)=O)=O)CCC1=O 19597,c1(C(N2CCCCC2c2cccc(O)c2)=O)ccc(C2CC2)cc1I 19598,c1(C(=O)OCC)ccc(N(C2CCCN(C(c3cc(C(F)F)[nH]n3)=O)C2)C)nc1 19599,C1(CC(=O)N(CC(C)N(C(c2c(SC)ccs2)=O)C)C)CN2CCN1CC2 19600,C(=O)(CN1C(=O)CSc2ccccc21)N1CC(NC(C2C(C)CCC2)=O)(CO)C1 19601,c1(SCC2CC(N(C(C=C)C3CC3)C)C2)cccc(OCC(=O)OC)c1 19602,N1(C(C2(CC)CCC2)=O)CCC(C(F)C(=O)N(C)CC2(C)CC2)C1 19603,O=C1CCC(C(N2CCN(C(c3cn(C4CC4)cn3)=O)C(CO)C2)=O)CCO1 19604,c1(CC)cc(C2CC2)nc(NCc2cn(Cc3nnc(C)o3)nn2)n1 19605,C1(NC(CC)=O)(NCC(c2ccc(C(C)C)cc2)=O)CCOCC1 19606,c1(OCC)ccc(C(=O)NC2CCCN(C(=O)COC(C)C)C2)nn1 19607,C#CC12CCC(C(N3CCC4(CC3)CC4CNC(=O)C=CBr)=O)(CC1)CC2 19608,C1(N(C(=O)Cc2cc(C)[nH]n2)CC)CCCN(C(=O)C(CO)NC(=O)OC)C1 19609,c1(NC(C(C)NC(C(C)OC)=O)=O)cnc(F)nc1 19610,C1(CNC(C(C)C(F)F)=O)C(O)C(O)CN1C(=O)CC1CCCC1 19611,C1(N(C)C(c2cc(-c3cccnc3)no2)=O)CCC(NC(C2CC2(Cl)Cl)=O)CC1 19612,N#Cc1ccc(C=CC(=O)NCCNC(=O)Cc2csc3ccccc23)cc1 19613,c1(OC)ccc(NC(C2(C)CN(C(c3cc(F)ncc3Br)=O)C2)=O)c(F)c1 19614,CC1(F)CCN(C(=O)CC2CCN2C(c2ccccc2F)=O)C1 19615,c1(C(=O)NCC(N(C(=O)C=CC2CCCC2)C)C2CC2)cc2cccn2c(O)n1 19616,N1(C(c2cc(C)oc2)=O)CCC(CNC(=O)CCOCC(C)C)CC1C 19617,N1(C(c2scc(C)c2C)=O)CCC2(CC2NC(C2CC(C(C)C)=NO2)=O)C1 19618,C1(NC(CCCCCSC)=O)CCN(C(=O)CC2C=CS(=O)(=O)C2)CCC1(F)F 19619,C1(CCNC(C23CC(C)(C2)C3)=O)CCCCN1C(=O)CC1(C)CCCO1 19620,CN1C(=O)CC(C(=O)Sc2ccccc2)C1SCC#N 19621,Cc1c(Br)cc(C(N2CC3CC3(C(=O)NCc3ccc[nH]3)C2)=O)cc1Br 19622,C(=O)(C(O)CC(N)=O)N1CC(NC(C23CC(OC)C2C3)=O)C(O)C1 19623,c1(NC2(CC(=O)NC(CC(C)C)CO)CCC2)ncnc2c(Br)csc12 19624,N#CC1(C(=O)NC2CC(NC(=O)CCF)C2)CCCC(=O)C1 19625,C1(NC(=O)CC2CCCC2)CC12CCC(NC(c1ccc(Cl)cn1)=O)CC2 19626,N#Cc1ccccc1CNC(=O)C(CN=[N+]=[N-])NC(=O)CC1(O)CCOC1 19627,N1(C(c2cnc(CC(C)C)s2)=O)CCN(C)C(CNC(=O)C(C)CN(C)C)C1 19628,CC1CN(C(C2(C)CCCN2C)=O)CCC1C(N1CCCC(C(N)=O)C1)=O 19629,CCCCC(CC)CC(=O)N(C)CC1(NC(C2Oc3ccccc3C2C)=O)CC1 19630,C1(C(N2C(C)CCC(=O)C2)=O)CCCCCCN1C(c1cc(C(N)=O)[nH]n1)=O 19631,c1(NC(C2CCCN(C(c3cc(CC)ncn3)=O)C2)=O)cccc(F)c1O 19632,C1(CC(=O)N(C2CCCN(C(C3C(Cl)(Cl)C34CC4)=O)C2)CC)COCCOC1 19633,C(=O)(C(CC(N)=O)NC(=O)C(C)C(C)COC)NCC(CC)(C)OC 19634,c1(C(N(C2CCN(C(=O)C=Cc3cccs3)C2)C)=O)cc(C(F)(F)F)ccn1 19635,N1(C(CC(=O)NCC2CC2)=O)CC2CCC1CN2C(=O)Cc1cc[nH]n1 19636,C1(C)(CNC(c2n(C)ncc2)=O)CCCN1C(=O)CCc1ccc(CO)cc1 19637,Cc1ccnc(C(=O)N(C2(C)CCN(c3nnnn3C)C2)Cc2ccccc2)n1 19638,c1(OC)sc(C(=O)NCC2(F)CN(C(=O)C(C)(Cl)Cl)C2)cc1Br 19639,C1(C(N(CC(CNC(C(C)=C(C)C)=O)(C)C)C)=O)CCCCC(F)(F)C1 19640,CC1C(NC(=O)Cc2n[nH]cc2Br)CCCN1C(c1ccc(F)c(F)c1)=O 19641,c1(OC)cccc(F)c1C(=O)NC1CCN(C(C2CCC(F)CC2)=O)C1 19642,N1(C(C(c2cn(C)nc2)=O)=O)CCCC2(NC(=O)COC3CCCC3)CCCC12 19643,Cc1c(C(=O)NC23CC(NCc4cc(O)ccc4F)(C2)C3)cncc1Br 19644,C(CC(c1nnnn1C1CC1)C1CCCO1)(C(C)C)(OCCOC)NCCSC 19645,c1(N2C(CNC(C3(C(=O)NC)CC3)=O)CC3COCC32)ncc2scc(Br)c2n1 19646,CC1CC(C(N2CCC(CF)C2)=O)CCN1C(=O)CCc1cnccn1 19647,c1(CCC)ncc(C(=O)NCC2CCN(C(=O)C(C)c3ccsc3)C2)s1 19648,N1(c2nc(C)c(Br)cn2)CC(C)(C)CCC1CNC(=O)C(C)Cc1cnc[nH]1 19649,C1(C(=O)NCCN(CCCF)C)CC(O)CCN1C(c1ccn(C(F)F)n1)=O 19650,C#CCC(CC(=O)N1CCC=CC1COC)NC(C1CC(F)(F)C1(C)C)=O 19651,C1(C(C2CCC2)NC(=O)CC2CCCCO2)CCCCC1 19652,c1(C(=O)NC2C3(CC(NC(C(CC=C)(F)F)=O)C3)C2)ccc2cnc(C)n2c1 19653,N1(C(C2(OC)CCSC2)=O)CCOC(CNC(=O)COc2cnn(C)c2)C1 19654,c1(NCc2c(C)cc(C)cc2C)nc(C)cc(=NCc2ncccc2C(F)F)[nH]1 19655,c1(C(N2CCC(OCc3ccccn3)CC2)=O)cnccc1Cl 19656,c1(CC(N2CC=C(CNC(C3CC3CN(C)C)=O)CC2)=O)ccc2[nH]ccc2c1 19657,CC(C)(C)C(O)C(=O)NCC1CC(NC(c2cccc(-c3cnco3)c2)=O)C1 19658,C(CC(C(=O)O)NC(=O)CCc1cncnc1)c1cn(C(COC)COC)nn1 19659,CCCCS(=O)(=O)CC(=O)N1CC2C(Cc3ccccc3)C2C1 19660,C1(NC(c2c(C)c[nH]n2)=O)CC2C1CCN2C(=O)C=C1CCCCC1(C)C 19661,N1(C(C=C(C)C2CC2)=O)CCSCC1C(=O)NC(C)C(N)=O 19662,c1(C2(C(=O)NC(CNC(C=CC(=O)OCC)=O)C)CC2)ncccc1F 19663,C1(CNC(=O)OC(C)(C)C)(COC(C2C=CCCC2)=O)CC2(CC(F)C2)C1 19664,Cc1cc(C(N2CC(O)(CNC(=O)CC3(O)CCCN(C)C3)C2)=O)cc(C)c1F 19665,c1(-c2c(CC(=O)N(CCOC)Cc3ccccc3)scc2)ccc(C)c(C)c1F 19666,CCC(CC)CCC(=O)NC1CN(C(c2cnn3cccc3c2)=O)CC1O 19667,c1(OC)ccc(CNC(=O)C(c2ccc(I)s2)N(CCF)C2CC2)cc1 19668,C1(CC)CCC(C(=O)N(CC(O)CNC(c2csc(COC)n2)=O)C)O1 19669,C1(C(=O)NCC(C)(C)F)C2CC(O)C(C2)N1C(c1cccc2[nH]ncc12)=O 19670,C1(C)(CNC(=O)NC(CS(CC)(=O)=O)C)CCCCC1(F)F 19671,CC1(CCNC(C2(C)C=CCC2)=O)CCN(C(c2csc(Br)n2)=O)C1 19672,C(=O)(C1=CCOCC1)NC1CCC(NC(C2C(C#C)C2(C)C)=O)CC1 19673,CN1CC(C(N2CC(N3CCN(C(=O)C=Cc4ccc[nH]4)CC3)C2)=O)NC1=O 19674,N1(C(C2(COC)CCCCC2)=O)CCN(C(=O)C(F)C(F)(F)F)C(C)C1 19675,C=CC(C)(C)CC(=O)NCC1(C)CCCN1C(=O)C=Cc1scnc1C 19676,CN(CCCC(=O)N1CCN(C)CC1CNC(=O)CC1CC(O)C1(C)C)N=O 19677,c1(C(=O)NC2(C)CCN(C(C3(CCO)CC3)=O)C2)ccc(Br)cc1[N+](=O)[O-] 19678,c1(CNC(C2(CNC(CCc3onc(C)n3)=O)CC2)=O)cc(O)ccc1F 19679,c1(C(N(CCCCCNC(C(C)OC2CCOC2)=O)C)=O)ccc(N(C)C)cn1 19680,N1(C(CCCC#CC)=O)CC(CNC(=O)C(O)CC(C)C)CC(C)(C)C1 19681,N1(C(CSC2C(=O)OCC2)=O)CCC2(C1)CN(C(c1c(Cl)nsc1Cl)=O)C2 19682,N1(C(CC2C(C(=O)OC)C2(C)C)=O)CCC(NC(c2nn(C)cc2C)=O)C(C)C1 19683,c1(C(N(CCOCCNC(C2C(OC)CC2)=O)C)=O)csc2nccn12 19684,c1(C(=O)NCC(C)NC(c2n(CC)nc(C)c2)=O)ccc(F)c(C)c1C#N 19685,N1(C(c2occ(C)c2)=O)CC(C)(C)CC1C(=O)NCc1ccc(Cl)o1 19686,CC1=NOC(C)(C(=O)NCC(CO)NC(C2CCN(C)C2=O)=O)C1 19687,c1(C(N2C(CNC(c3ccc(C#C)cn3)=O)CCC2)=O)noc2c1CCCCC2 19688,C=CCC(C(=O)N(CC(C)O)CCNC(C12CCC(OC)(CC1)C2)=O)C(C)(C)C 19689,CCC(CC(F)F)C(=O)N1CCC1CNC(=O)CCNS(=O)(=O)CC 19690,N1(C(C(C(C)C)OC)=O)CC2C(NC(=O)CC(C)(C)C(C)(F)F)CS(=O)(=O)C2C1 19691,C1(NC(C2(OC)CCN(C(C(COC)COC)=O)C2)=O)CN2CCC1(F)CC2 19692,Cn1nc(C(N2CCC(N(CCO)C(C3CCNC3=O)=O)C2)=O)cc1F 19693,C(=O)(C(F)C1=CCCCC1)NCc1ccc(CNC(C2C(=C)CC2)=O)c(F)c1 19694,C(=O)(CCC(F)(F)F)NC1CCCC(CC(=O)Nc2c(CC)nn(C)c2)C1 19695,c1(C(N(C)CC2(CNC(C3CC3Cl)=O)CC2)=O)ccc(CN2CCCCC2)o1 19696,c1(C(=O)NC(C)(CNC(C2COCOC2)=O)C2CC2)c[nH]c2nccc-2c1 19697,N1(C(CC(C)(C)C)=O)CC2(CCCN(C(c3cccc4nscc34)=O)C2)C1 19698,C(=O)(C1=CNC2=NCCCN12)NCC1N(C(CC2C(OCC)COCC2)=O)CCC1 19699,c1(C(N2C(C(C)NC(c3n(CC)c(O)nc3)=O)CCC2)=O)cc2ccccn2n1 19700,c1(C(N2CC(C(C)NC(=O)C(C)C(F)F)C2)=O)ccc(N)c(F)c1F 19701,c1(C(N(C2CCCCN(C(C=CC(=O)N(C)C)=O)C2)C)=O)ccnc2c1CCC2 19702,c1(C(=O)NCCCCC(=O)N(C2C(C)CN(C)CC2)C)nccc2[nH]ccc12 19703,C1(NC(CC(=O)OCC)=O)CN(C(c2ccnn2CC)=O)CC12CCC2 19704,N1(C(c2c(C)scn2)=O)CCCC(N(C(=O)Cc2cc(Cl)cs2)C)CC1 19705,n1(CC)ccc(C(=O)N(CC(C)(C)NC(c2cc(C)c(Cl)s2)=O)C)cc1=O 19706,N1(C(c2scc(C)c2C)=O)CCN(C(C2CCN2C2CCCC2)=O)C(CF)C1 19707,N1(C(C(C)NC(N)=O)=O)Cc2nccnc2CC1C(=O)NC(C1CCOCC1)C 19708,C1(NC(COCCCOC)=O)CN(Cc2cc(C3CCCCC3)on2)CCC1C 19709,CC(N=c1ccc(C#N)n[nH]1)C1CCN(C(C2CCc3nn[nH]c3C2)=O)C1 19710,C1(NC(CN(S(CC)(=O)=O)C)=O)CCCCC1NC(=O)C=Cc1ncco1 19711,Cc1cccc(SCC(=O)N(C2CCCC(NC(=O)CC(C)(C)C)C2)C)c1 19712,c1(C(=O)NC(CN(C(C(C(C)C)OCC)=O)C)CC)nc(C)c(C)nc1C 19713,CCC(CC(C)C)C(C(=O)Nc1c(C)cc(C)cc1C)N1CC2CCC(C1)O2 19714,c1(C(=O)NCCCCNC(C2CC3CCC2C3)CC)cc2ccccc2o1 19715,N1(C(c2ccc(C)nc2C)=O)CC(NC(=O)CN2CC(=O)NC2=O)C(C2CC2)C1 19716,C1(C)(C(=O)NCCOCCN(C)C(c2cc(Br)cn2C)=O)CCCNC1=O 19717,N1(C(Cc2cn(CC)nn2)=O)CC(NC(=O)CNC=O)CC(F)(F)C1 19718,C(CCCCC(=O)NC(C)CCN(C(=O)Cc1cc(C2CC2)no1)C)OCC 19719,N1(C(C2C(OCC)C2)=O)CCC(NC(=O)C(N2CCCCCC2)C)C(C)C1 19720,C#Cc1cc(NC(=O)C(C)N(C(C2(C)CC2(C)C)=O)C2CC2)cc(F)c1 19721,c1(C(CNC(C(=O)NC2C(OC)CCC2)=O)OC)ccncc1F 19722,N1(C(C(C)N(C(CSC(C)C)=O)C)=O)CCCC(C)(O)C1 19723,C12(CNC(CCN(CCC)C)=O)CN(C(=O)CC=C(C)C)CC1CCO2 19724,c1(C(=O)NC(CCNC(c2nc(C)nn2C)=O)(C)C)nccc(N)c1Cl 19725,CC1CC(C(=O)NCC23CC(CNC(C4CC5CC5C4)=O)(CO2)C3)CC(C)C1 19726,c1(OC)cc(Br)c(C(=O)NCCNC(c2nccc(C)c2N)=O)cc1OC 19727,N1(C(C2CC(=C)C2)=O)CCC(C(=O)OC)C(O)C1.c12nccc(n1)N2 19728,c1(C(=O)NCC(CN(C(c2nc(C(C)=O)sc2)=O)C)C)nnc(C)cc1O 19729,Cc1noc(C)c1S(=O)(=O)N1CC2CN(S(=O)(=O)CCBr)C2C1 19730,c1(OC)cc(C(=O)NCC2CN(C(C3(OC)CCC3)=O)C2)cc2cn(C)nc12 19731,c1(NC(C(=O)Nc2cc(C)sc2C)=O)c(C)ccc(F)c1[N+](=O)[O-] 19732,C(=O)(N=c1ccn(CCC2CC2)[nH]1)C12CC(CNC(Cn3nnc(C)n3)=O)(C1)C2 19733,c1(C(=O)NCC2(O)CCCN(C(C3ON=C(CC)C3)=O)C2)cccn2nccc12 19734,N1(CC(=O)NCCC)CCS(=O)(=O)C(CCNNC(=O)CC2NC(=O)NC2=O)C1 19735,CCS(=O)(=O)CCC(C(=O)N1CC2CCC1C(CSC)C2)NC(=O)OC(C)(C)C 19736,N1(C(C(CC)CC2CCCCC2)=O)CC(C)CN(C(=O)Cn2cccn2)CC1C 19737,N1(C(C(C=C)C)=O)CC(O)(C2(CNC(=O)COCc3cccc(C)c3)CC2)C1 19738,c1(CCC)nc(=NC(C)CN(C(=O)Cn2cc3ncccc3n2)C)s[nH]1 19739,N1(C(c2c(CC)cno2)=O)CCC2C(C(=O)NCCCCC3CC3)C2C1 19740,c1(C(=O)NCC2(O)CCN(C(C3(C)CC3(F)F)=O)CC2)coc2ccc(O)cc12 19741,C1(N(C)C)CN(C(C2CC2(Cl)Cl)=O)CC1CNC(c1csc(O)n1)=O 19742,c1(C(N2C3CC(NC(CCC(C)(C)F)=O)CC2CC3)=O)cnnc2ccccc12 19743,c1(NC(C)=O)ccccc1SCC(N1CC(C)(NC(=O)CC2CCC(O)C2)C1)=O 19744,N=c1[nH]c(=NCC2CCC3CC23)[nH]c(=NCCCCCC(=O)NC2CC2)[nH]1 19745,c1(C(N2C(CCC)(C(=O)OCC)CCC2)=O)ncn2c1CCNCC2 19746,CCC(CN(C)C)CC(=O)NCC1(O)CN(C(=O)CCC(C)N(C)C)C1 19747,c1(NCC(N2C(CC)CC(C(F)(F)F)CC2)=O)ccc(CO)c([N+](=O)[O-])c1 19748,N1(C(C(c2ccc(Cl)cc2)CC)=O)CC2CN(C(=O)OC(C)(C)C)CC2(C)C1 19749,C12(C(N3C(CN(C(CCCC(C)C)=O)C)CCC3)=O)CC=CCN1CCC2 19750,C1(NC(c2c(CC)csc2)=O)COCCN(C(c2cn(C(C)C)cc2C)=O)C1 19751,Cc1cc(CO)oc1C(=O)NCC1(F)CC(CNC(=O)CC2CC3CC3C2)C1 19752,C(C1CN(C(=O)Cc2cnn(C)c2C)CC1C(=O)NCCCN1CC=CC1)=CC 19753,C1(NC(C2CCN(C)C2)=O)CC2(C1)CC(NC(c1cc(C(F)F)no1)=O)C2 19754,C1(C(N2CCN(C(c3c(CC)ncs3)=O)CC2COC)=O)CCc2nn[nH]c2C1 19755,C(C)(C(=O)NOOC)(N(C(C1CCC(Cc2cccc(C)n2)C1)=O)C)C1CC1 19756,c1(CC)nccnc1C(=O)NCC(C)N(C)C(C1CCC1(F)F)=O 19757,C1(CNC(c2c(F)ccc(OC)c2)c2nnnn2C)CCOC2(CCC2)C1 19758,Cc1cc(F)cc(C(=O)NCC2CN(C(C3CC4(CC4)CO3)=O)CC2(C)C)c1N 19759,n12c(C)cc(c1C)C=CC(=O)NC1CC1NC(=O)C2.C(=O)(C(C)CC)N.CCC 19760,N1(C(c2c(C)nn[nH]2)=O)CCCCCCC1C(N1CCC(C)(CO)C1)=O 19761,Cc1cn(C)nc1CNC(=O)CONC(C1(C)CNC(=O)N1)=O 19762,C(=O)(C1=CCN(C(=O)CC(C)C2CC2)C1)N(C(CC(CC)C)C)C 19763,N1(C(=O)Nc2cc(F)ccn2)CCn2cc(-c3cccnc3OCCO)nc2C1 19764,C1(C(=O)NC23CN(C(c4cc(C)n(C)n4)=O)C(CC2)C3)CNC(=O)CC12CCC2 19765,C#CCC(CC#C)C(=O)N1CC2CCN(C(=O)CCC(C)SC)C2C1 19766,C(=O)(C1CCCc2nncn21)NCCNC(c1c(C(F)F)ccc(C)c1)=O 19767,N1(C(CSCc2ccc(C(C)C)cc2)=O)CC2CC1CCC2NC(C1(C)CC1)=O 19768,c1(C(=O)NC2CC(C)(NC(C(CC)COC)=O)C2)cc(O)cc(F)c1 19769,N1(CC(c2c(C)ccnc2)=O)CCC(C#N)(C2CC2)CC1 19770,C1(CNC(C=CC=CC)=O)CN(C(c2n[nH]cc2C2CCC2)=O)CCC12CCC2 19771,C1(C(N(C2C(C)CC2)C)=O)CCC2CCC1N2C(c1cnn(C)c1Cl)=O 19772,N#CC1(C(=O)NCC2CC(NC(C3(S(N)(=O)=O)CCC3)=O)C2)CC2CC2C1 19773,C=CC(C)(O)CC(=O)NC(CC(F)F)C(=O)NCC(C)C(=O)OCC 19774,CCC(CC1CCCCC1)C(=O)NC1CCCCC1CNC(c1[nH]ccc1C)=O 19775,N1(C(CC2CC(CC)C2)=O)CCCC(C)(CNC(=O)CS(=O)(=O)NC2CC2)C1 19776,CC(C)C(C)(C)C(=O)NCc1nc(C(=O)NC2CNC(=O)C2)co1 19777,C1(C(=O)OC)Cc2ccccc2C1NC(=O)CC1C(=O)ON=C1C 19778,C1(F)(C(N(C)CC2C(C)C2)=O)CCN(C(C2CC(C)(C)CCO2)=O)CC1 19779,C12(NC(C3(CF)CCNC3)=O)CC(c3ccccc3)(C1)C2 19780,Cc1cccc(C(=O)N(CC(C)N(C(=O)CCSc2ccccc2)C)C)c1C 19781,Cn1c(C(=O)NC(c2ccco2)c2cccs2)ccc1C=O 19782,c1(C(=O)NC2CCC(NC(c3coc(O)n3)=O)CC2)ccc2c(c1)CCCC2=O 19783,C1(CNC(CCOCC#C)=O)CN(C(c2c(N)cnn2C)=O)CCC1C 19784,C1(C(N2CC(NC(C(C)=CC)=O)C(CC(C)(C)C)C2)=O)OC(C)(C)OC1(C)C 19785,C(CCCCC(=O)N(C1CCN(C(c2cc(C)co2)=O)C1)C)OCC 19786,c1(C(N(CC(=O)Nc2ccc(SC)nc2)CC#C)=O)[nH]ccc(=O)c1C 19787,CC1(C)C=C(C(=O)NCC2(NC(=O)C=CCN3CCCC3)CCCCCC2)C1 19788,C(=O)(CC(C)(C)C(F)F)NCCCC(C)NC(=O)CC1CCS(=O)(=O)C1 19789,c1(CNC(=O)Nc2cccc(CN(C)C(=O)OC(C)(C)C)c2)cccc(Br)c1F 19790,c1(OCC)ncc(C(N2CCC2C(=O)NC)=O)cc1-c1cccc(C(C)(C)O)c1 19791,C1(NC(C(C)=CC2CC2)=O)CCC(C)N(C(=O)CCCn2ccccc2=O)C1 19792,C(=O)(CC(C)(C)NC(=O)C=CC1CCOC1)NC1C(CN(C)C)C1 19793,C1(C)(CNC(c2ccc(C(C)C)o2)=O)CN(C(=O)COC2(C)CCC2)CCO1 19794,n1(CC(=O)N(CCC(=O)NC2CCN(C(C)C)C2)C(C)C)ncn(C)c1=O 19795,N1(C(C2(CCC)CCC2)=O)CC2(CCC(CNC(=O)C(C)CC(C)(F)F)O2)C1 19796,Cc1cc(-n2cc(C(C(C)C)NC(=O)C(CO)NC(N)=O)nn2)cc(C)c1 19797,c1(OC(C)C)nccc(C(=O)NCC(CO)NC(C2(CO)CCC2)=O)c1F 19798,C1(CNC(c2nnc(CC)s2)=O)CC2COCC2N1C(c1sncc1C)=O 19799,N1(C(c2ccc(CC)s2)=O)CCC(NC(c2c(C(F)F)nn(C)c2C)=O)C(C)C1 19800,C1(CCC(=O)Nc2cccc(CC)c2)CCCCN(C(c2cccnc2C)=O)C1 19801,C(CNC(=O)COCCN(C)C)(CC(F)(F)F)NC(c1c(C)cno1)=O 19802,C1(C(N2CCC(CCO)C2)=O)CCCN(C2CC2)C1 19803,Cc1ccc(CC(=O)NC2CCCC(CNC(C34COC(CF)(C3)C4)=O)C2)cc1 19804,C1(NC(c2ccncc2Cl)=O)CC2CN(C(C3CCCSC3)=O)CC12 19805,C1(N(C)C(c2coc3c2COC3)=O)CCCC2CN(C(=O)CC3CC34CC4)CC12 19806,c1(C(N2CCC(O)(CNC(C3(C(=O)OCC)CC3)=O)C2)=O)cc(=O)cc(Cl)[nH]1 19807,N1(C(c2cc(Br)ncc2Br)=O)CCC2CN(c3ncc(F)cn3)CC2C1 19808,c1(C(=O)NC(C(=O)NCCNC(=O)NC)CCOC)cccc2ccoc12 19809,C1(C(N2CC(CNC(=O)CC3CC3(Cl)Cl)OCC2)=O)CCOC2(CCC2)C1 19810,C1(N(C(=O)C(C)n2cccn2)CC(=O)NC(C)C)CCCC12CCNCC2 19811,c1(C(=O)NC(COC)CC(C)(C)C)ccc2n1CCNC2 19812,N1(C(c2nc(CNC(C3N(C)CCOC3)=O)oc2)=O)CCC(O)C(O)C1 19813,C1(C(=O)NC23CCC(NC(Cc4cnc(C)[nH]4)=O)(CC2)C3)CCC(=O)CC1(C)C 19814,Cc1cccc(F)c1CC(=O)Nc1nc(CNC(=O)Cc2cncn2C)cs1 19815,c1(C(=O)NCC(CC)NC(C2CNC(=O)N2C)=O)ccc2ccc(O)nc2n1 19816,CC1CCCN(C(c2cccnn2)=O)C1CCNC(c1cc(F)ccc1Br)=O 19817,N1(C(C(C)OCCCC)=O)CCCC(C)(CNC(C2(C)CCCO2)=O)C1 19818,N#Cc1ccc(CN2CCC(C(=O)Nc3nn(CC(F)(F)F)cc3Br)C(O)C2)nc1 19819,c1(CC)nc(O)c(C(=O)NC2CCCCC2CNC(C2(C)CC=CC2)=O)cc1C 19820,N1(C(CC=CC=C)=O)CCN(C(=O)COCCCF)CC1C1CCC1 19821,C1(C(=O)NC2(C(C)O)CC2)CCCC(NC(C2COCC2(C)C)=O)C1 19822,N1(C(c2cc(I)c(F)cc2F)=O)CCC2C(CCN2Cc2cccc(Br)c2Cl)C1 19823,N1(C(Cn2c(CC)nnn2)=O)CCC2CCC(C1)N2Cc1cc(C(C)(C)C)on1 19824,C(C(C)C(F)C(=O)NCc1csc(C)c1C)NC(c1ncn(CC)c1)=O 19825,CC1C(C(=O)NC23CC(NC(C4OC(C)(C)OC4(C)C)=O)(C2)C3)C(O)C(=O)N1C 19826,c1(NC(C2CCCCN2C(c2ccnnc2O)=O)=O)cc(Cl)ccc1CO 19827,CCC1=C(C(=O)NC2CCN(C(c3cnn4c3OCCC4)=O)CC2C)SCCO1 19828,c1(NC(C2CN(C(C(COC(C)C)NC(C)=O)=O)C2)C)nccc(C)n1 19829,C1(C(=O)NCC(C)(C)NC(c2cc(C(F)(F)F)no2)=O)C2CC2C2CC12 19830,C1(CC(=O)NC2C(OC)CCCC2)C2CCCC2N1C(c1nscc1C)=O 19831,N1(C(CCN(C(c2c[nH]c(=S)cn2)=O)CCO)=O)CCC2(C=CCO2)C1 19832,N1(C(c2ncc(C)cc2F)=O)CCC2C(CCCN2C(=O)CC(C)(F)F)C1 19833,C1(C(=O)NCC23OC(C)C(NC(c4cccs4)=O)(C2)C3)CCCC1S(C)(=O)=O 19834,CCS(=O)CC(=O)NCC(c1ccc(F)cc1)NC(C1(OC)CC1)=O 19835,Cn1nc(C2CCC2)cc1C(=O)NCCCCCCNC(C12CCC1C2)=O 19836,C(=O)(CC(C)NC(N)=O)NCC(C)CN(C)C(c1sccc1Br)=O 19837,N1(C(C(C(CC)C)O)=O)CCCC2(C1)CN(C(=O)CN1CCP(C)(=O)CC1)C2 19838,CC1(C)CCOC(CNC(C2C(O)CCN2C(C2CN3CCN2CC3)=O)=O)C1 19839,c1(C(=O)NCC(CC=C)NC(c2cscc2C)=O)cc(N(C)C)ccn1 19840,c1(CCc2ccsc2)nc(C2Cc3ccccc32)nn1-c1nc2ccccc2s1 19841,c1(CCNC(c2cc(C)c(Br)s2)c2n(C(CC)C)nnn2)c(Cl)cccc1Cl 19842,N#CC1(C(N2CC(CNC(=O)CCCCCNC(N)=O)C2)=O)CC2CCC1CC2 19843,C(=O)(C(CC(N)=O)NC(=O)COC1CCCOC1)NCC(C=C)O 19844,C=CCCCC(=O)NCCC1(C(=O)NC2(C3CCC3)CC2)CCC1 19845,CC(C(C)(C)CO)NC(=O)C(C)(C1CC1)N(C(=O)COc1ccsn1)C 19846,c1(C(=O)NCC2(C(F)F)CCN(C(C(CC)OCC)=O)C2)c(Cl)ccc(C)c1O 19847,N1(C(C2CCC(C)CC2)=O)CCC(NC(c2cnn(C3CC3)c2)=O)CC(C)(C)C1 19848,c1(NC(CC(C)C)C)cc(S(=O)(=O)NC(c2ccc(Cl)cc2)CF)ccc1C#N 19849,N1(C(CCCC)=O)CCN(C2CCC(NC(C3(C)CCC(=O)N3)=O)CC2)CC1 19850,C1(NC(c2cn(C)nc2C2CC2)=O)CCCCN(C(=O)CO)CC1 19851,N1(C(C(CC)OCC)=O)CCc2nc(CNC(c3cn(C)nc3C)=O)sc2C1 19852,C(N=c1ccnc(NC2CCCn3ncnc32)[nH]1)C1(N(C)C2CC2)CCCSC1 19853,C(=O)(C(CC)NC(C)=O)N(CCNC(C1CCCN1C(=O)C(F)(F)F)=O)CC 19854,C(CCCCCC(=O)NCCC1CCC(=O)N1)NC(C(=Cc1cn[nH]c1)C)=O 19855,C12(CNC(c3c(C)coc3C3CC3)=O)CCCC1CCN2C(c1ccncc1)=O 19856,N1(C(CC(=O)OC)=O)CC2(CO)CC1(C(=O)NC1CC(O)CC1O)C2 19857,C(=O)(C(C(C)CC)N(C(=O)CCN1CCCCC1)C)N(CC#C)CCO 19858,C1(NC(=O)CCC(F)F)CN(C(c2nccc3[nH]ccc23)=O)CC1C1CC1 19859,c1(CNC(C2N(C(C)C)CCC2)=O)ccc(CNC(C2CC2(C)C)=O)cc1F 19860,N1(C(C2N(C)C(=O)CC2)=O)CCC(O)(C2CCN(C(=O)C3=CCC3)CC2)CC1 19861,N1(C(CSCCCC)=O)CCC2(CC1)CCN(C(C1CCC3CC3C1)=O)C2 19862,N1(C(C2CCC(N(C)C)CC2)=O)CC(NC(=O)CS(=O)(=O)CCO)C(C2CC2)C1 19863,c12ccccc1N(C)C(C)C(=O)N2.C1CC(=O)N1.CCCNC(=O)OCC 19864,c1(C(=O)NCCNC(c2nocc2Cl)=O)c[nH]c2ccc(Cl)cc2c1=O 19865,c1(C(=O)OC)ccc(N2CC(CCNC(=O)C(c3ccnn3C)C)(OC)C2)nc1 19866,c1(NC(C2CCCC2NC(c2cn(-c3ccccc3)nn2)=O)=O)c[nH]nc1Br 19867,c1(OC)ccncc1C(=O)NC(C)CCNC(C1(Oc2cccc(C)c2)CC1)=O 19868,Cc1ccncc1CC(=O)NCC(C)(C)NC(c1cnc(N2CCOCC2)s1)=O 19869,c1(C(=O)NC2C=CC(C(=O)NC(c3ncc[nH]3)CC)C2)ccnc(C)c1C 19870,Cc1cccc(-c2cncc(C(=O)NCC(O)CCNC(C3CCCS3)=O)c2)c1 19871,CCCC(O)CC(=O)NC1CCC1CNC(=O)CCNC(=O)C(C)(C)C 19872,CC(C)(C)C(CNC(c1ocnc1C(F)(F)F)=O)NC(c1c[nH]c(C(N)=O)c1)=O 19873,C1(NC(C(=O)NCC)=O)C2CCCN(Cc3cc(C)ns3)C2C1(C)C 19874,c1(C(N2CC(O)(CCNC(C3C(C)(C(F)F)C3)=O)C2)=O)cccc([N+](=O)[O-])c1N 19875,Cc1cc(CC(=O)NC(C)CCN(C(c2[nH]nnc2C)=O)C(C)C)cs1 19876,C1(CC)CN(C(c2cncn2C)=O)CCC1CNC(c1ccnn1C)=O 19877,C1(C(=O)NC(c2ccccc2F)CC)CC(F)CN(C(c2cc(O)ncn2)=O)C1 19878,N1(C(C(CC(C)C)(F)F)=O)CCCC2(C1)CN(C(c1ccnn(C)c1=O)=O)C2 19879,C(=O)(CS(=O)(=O)NC(C)(C)C)NCC(C)CNC(C1CC1c1nccs1)=O 19880,c1(C(N2C(C)CN(C(C3(C)CC=CCC3)=O)CC2)=O)cccn2ccnc12 19881,N1(CC)CC(C(=O)NC2CN(C(C3(F)CCCC3)=O)CC2C)CC1=O 19882,c1(C(=O)NCC2CC(NC(=O)C(F)(F)c3nccs3)C2)cc2c(Cl)cncc2s1 19883,c1(C(N(CCCNC(C(CCC)NC(C)=O)=O)CC)=O)c(Cl)ccc(Cl)c1O 19884,C12(CNC(C(C)(C)SC)=O)CCC(CN(C(C34CCC(C)(C3)OC4)=O)C1)C2 19885,CC1CC(O)CN(C(=O)NCc2ccccc2)C1.C12CN(CCO1)C2 19886,C1(CNC(CN(CCC#C)C)=O)C(C2CC2)CCN1C(=O)C#CC1(C)CC1 19887,Cc1cccc(Cl)c1C(N1CC(CC(N2CCC(CF)CC2)=O)C1)=O 19888,c1(C(=O)NC2CCC(C)N(C(C3C4CC5C(C4)C35)=O)C2)ccc2nn[nH]c2c1O 19889,CC(C)CC(CNC(=O)CCc1nccc(C(=O)O)n1)N(C)C 19890,N1(C(C(=O)NCC=C)c2cccs2)CCc2ncncc2C1 19891,C1(C(=O)NCCCCC2CCCN(C(c3cnc(C)[nH]3)=O)C2)COC2(CCC2)C1 19892,c1(NC(C)=O)ccc(NC(=O)CC2CCCN(C(=O)CCCCC#N)C2)cc1C 19893,c12ccc(CO)c(c1)NC2=O.c1(COC)oc(C2CC2)nc1C 19894,C(=O)(C(CC(C)C)NC(C1(NC(c2ccccc2C)=O)CCOC1)=O)OC 19895,c1(C(C)=O)ccc(C(=O)NCC2CC(C)N(C(=O)OC(C)(C)C)C2)cc1Cl 19896,Cc1ncc([N+](=O)[O-])n1CC(=O)NC1CC(C)(CNC(C2CC(C)CCO2)=O)C1 19897,C12(CNC(C(CC(C)C)N(C)C)=O)CN(C(c3cc(Cl)no3)=O)CC1CCO2 19898,Cc1sc(O)nc1C(=O)N(C)CC1CCN(C(=O)COCC(F)F)C1 19899,c1(CC2CN(C(c3ccccc3F)C)C2)c(F)cc(C(F)(F)F)cc1F 19900,C1(C(=O)NCC(=O)N(CC)CC)CCC(C(C)C)N1C(c1cc(CO)c(C)o1)=O 19901,C1(CC)CCN(C(=O)CCN(CC)CC2CC2)C1.C1(C)(C)CNC(=O)CO1 19902,c1(CC(N2CC(O)(C(C)NC(C=C(C)C3CC3)=O)C2)=O)cc(F)ccc1F 19903,C1(CNC(c2ccc(F)cc2)=O)CCC2(CN(C(C3(CO)CCC3)=O)C2)O1 19904,C1(SC)CN(C(=O)CC(F)(F)F)CC1C(=O)NC1CC(N(C)C)C1 19905,O=C(C1=CS(=O)CCC1)N1CCN(C(c2ccccc2Cl)=O)C(CC2CC2)C1 19906,c1(C(=O)NC(CC2CN(C(C3(CC#C)CC3)=O)C2)C)ccn(CC)c(=O)c1 19907,c1(C(=O)NCC2CN(C(c3n(C(C)C)ccc3)=O)C2)cc2n(c1)CCC2 19908,c1(C(=O)NC2(C)CCN(C(=O)CC3CCCC(=O)C3)C2)onc2c1CCCC2 19909,N1(C(Cc2n(C)c(S)nn2)=O)CCCC(F)(CNC(=O)CC2CNC(=O)O2)C1 19910,Cc1ccn(CCNC(=O)CN(C(=O)C(O)NC(c2cccnc2)=O)C)c(=O)c1 19911,c1(C(N2C3C(NC(c4ccc(C)nn4)=O)C(C3)C2)=O)n[nH]cc1[N+](=O)[O-] 19912,C1(CC)CC(O)CN1C(=O)C(CC1CCC1)NC(=O)C=CC(=O)OC(C)(C)C 19913,N1(C(C(C)=CC)=O)CCCC2(CCCCC2NC(=O)CC(C)CCC=C(C)C)C1 19914,N1(C(C(CC)SC)=O)CC(NC(c2nccc3[nH]ccc23)=O)C2(CCOCC2)C1 19915,CCC(CC(F)F)C(=O)NC1CN(C(c2ccc(Cl)c(F)c2F)=O)C(C)(C)C1 19916,S(=O)(=O)(CCCCCl)NC1CCC(C(=O)NC2CCN(Cc3ccccc3)CC2)C1 19917,C=CCCCCC(=O)NC(CO)C(C)NC(c1ccnc(OCCOC)c1)=O 19918,N1(C(C2CCC2)=O)CC2C3CCC(C2C1)N(C(c1c(F)cc(F)cc1Cl)=O)C3 19919,CON1CCC(C(=O)NCCCCCNC(=O)C(c2cncnc2)C)CC1 19920,N1(C(C=C(C)C(F)F)=O)CCC(NC(C23CCC(C2)C3)=O)C(C(C)C)C1 19921,c1(C(N2CC(NC(=O)C=C(Cl)Cl)C(CO)CC2)=O)ccn2nccc2n1 19922,c1(Oc2ccc(OC)cc2C=Cc2cccnc2)cccc2sc(C(F)F)nc12 19923,c1(C(=O)NCC2(NC(C(CCCC)O)=O)CCOC2)ccc2c(c1)NC(=O)C2=O 19924,c1(C(=O)NCC2CC(OC)CN2C(=O)C(C)NC(C)(C)C)ccc2ccsc2c1 19925,CC1CCN(C(C2CCCC3CCCN23)=O)C(C2CCC(C)O2)C1 19926,c1(C(=O)OC)ccoc1C(=O)N(CCCCNC(c1ccc(C(F)(F)F)[nH]1)=O)C 19927,S(=O)(=O)(C=Cc1ccccc1)NC1C(F)(F)CCN(C(=O)CN2CCOCC2)C1 19928,N1(C(C(CSC)C)=O)CC(O)CC1CNC(c1nc(C2CC2)cs1)=O 19929,C12(C(=O)NCC3C(NC(CSCCOC)=O)CCCC3)CCN(CC1)S(=O)(=O)C2 19930,CCC(C)(CNC(=O)C=Cc1ccncc1)C(=O)N(C)CC1(C)CCCC1 19931,N1(C(CC(CCC)O)=O)CC2(CCC2)CC1CNC(C1(NC(C)=O)CCCC1)=O 19932,c1(C(=O)NCC(CNC(CC2(OC)CCCCC2)=O)F)c(C)cc(F)cc1C 19933,N1(C(c2cccc(COC)n2)=O)CCC2CCN(C(c3ccoc3Cl)=O)CC12 19934,C1(NC(C2C(C(C)C)OCC2)=O)CC=C(C(=O)NCc2ccoc2)C1 19935,CC(C(=O)NCC1CC2(C1)CN(C(=O)Cc1cccc(C#N)c1)C2)C(C)(F)F 19936,C1(C(=O)N(C2CC3CC3C2)C)(OC)CCN(C(=O)Cn2c(O)nnc2O)C1 19937,O=C(CCC(F)F)NCCCCNC(C1(CC2CCCC2)CCCC1)=O 19938,C(=O)(CCC(N)=O)N1CC(O)(C(C(=O)N(CC(C2CC2)OC)C)F)C1 19939,C1(C(=O)NC2C=CC(CNC(C3(C(F)F)CCCC3)=O)C2)(OC)CCSC1 19940,c1(OC)ccc(CC(=O)N(C)Cc2cc(Cl)ccc2C)c(Br)c1 19941,c1(OC2CCCC(C(=O)NCCNC(CC(=C=C)C)=O)C2)ccccc1C#N 19942,C(C1CCCC1)=C(C)C(=O)NC1C=CC(CC(=O)NCC2CC2Cl)C1 19943,C(=O)(C1=CCCCCC1)NC(C(N1CC[Si](C)(C)C1)=O)CC1CCOCC1 19944,c1(NC(COC(C(CCOC)C)=O)=O)ccc2c(c1)CCC2 19945,Cc1cc(C)n(C(C)CC(=O)NC(C2CCCN2C(=O)CCC(=O)C2CC2)C)n1 19946,C(=O)(C(C)CC(=O)c1ccccc1F)NCCNC(C(N1CCNC1=O)C)=O 19947,C1(CC(C)C)CCN(C(=O)CC2CCCC(NC(c3cc(C#N)cs3)=O)C2)CC1 19948,c1(OC)cc(C(=O)NCCCN(C(=O)C(C)C(F)F)Cc2ccccc2)ncn1 19949,c1(C(N2CC(CNC(C3CC(OC(F)F)C3)=O)C3(CC3)C2)=O)cccc(F)c1Cl 19950,c1(C(N2CC(O)CC(NC(c3cc(C#N)sc3)=O)C2)=O)cc2nc[nH]c2cn1 19951,Cc1sc(=O)n(CCC(N2CCCCC2CCNC(=O)CC(C)N(C)C)=O)c1C 19952,C1(NC(c2ccc(O)cn2)=O)C2CCC1CN(C(=O)C=Cc1ccco1)C2 19953,C(C)(C)(C(=O)OC(C)(C)C)NC(CC)=O.C1(Cc2ccco2)C(=O)O1 19954,N1(C(CC=CCNC(C2(CCN=[N+]=[N-])CC2)=O)=O)CC2CCCCC2C1 19955,N1(C(C(CC)CC2CCCC2)=O)CCN(c2nc(C)cc(C)n2)C(C)C1 19956,O=C(C1=CC2(CCN(C(=O)C(F)n3ccnc3)C2)C1)NCC1(CC2CC2)CC1 19957,N1(C(=O)CC(F)F)CCN(C(c2ccc(C(F)(F)F)cn2)=O)C(CF)C1 19958,C(=O)(C(C)(C)C1=CCN(C(=O)CC=CCCCCC)C1)NCCCC 19959,N1(C(C(C2CC2)OC)=O)CCCC(N(C)C(c2cccc(F)c2SC)=O)CC1 19960,c1(C(=O)NCC(CC(C)C)NC(C(COC)(C)C)=O)cnn2cc(C)cnc12 19961,N1(C(c2scc(C(C)=O)c2)=O)CCCC(C)(NC(=O)CCN2CCCC2=O)C1 19962,CC(CC(F)(F)F)C(=O)NCC(C)(C)CCNC(c1cccc(NCC#N)c1)=O 19963,c1(C(N(CCCCCNC(=O)CNC=O)C)=O)ccc2ocnc2n1 19964,C1(Nc2c(C(=O)OCCOCC3CCCC3)cccc2)CCc2c[nH]nc2C1 19965,N1(C(CCOCc2c(C)ncs2)=O)CC2CC(NC(=O)COCC(F)F)C1C2 19966,N1(C(C(F)=C(C)C)=O)CCN(C(C2CC2(Cl)Cl)=O)C(C(C)C)C1 19967,N1(C(CC(n2c(CC)ncc2)C)=O)CCCC2CN(C(=O)CC(C)OC)CC12 19968,Cc1nc(NCc2csc(Cl)c2)cc(=NC(C)C2CCN(C)C2)[nH]1 19969,C1(N(C)C(c2cncnc2)=O)CCCC2CN(C(=O)CC3(O)CCCC3)CC12 19970,c1(C(N2CC(COC)N(C(=O)CCNC(C)=O)CC2)=O)cc2oc(C)cc2[nH]1 19971,C(c1c(C)nn(C)c1Cl)=CC(N1CC(OC)(CNC(c2cnc(=N)[nH]c2)=O)C1)=O 19972,c1(C(=O)NC(C)CC(C)NC(=O)C=CC(=O)NC2CC2)cccn2c(O)nnc12 19973,N1(C(c2c(COC)cno2)=O)CC(c2cccc(CO)c2)C(c2ccccc2)C1 19974,Cn1cc[nH]c(=NCC2CN(c3ncccn3)CCO2)c1=O 19975,C12(C(=O)NC3CCN(C(=O)Cc4ccsc4)CC3)CCCCC1C2Br 19976,O=C1CCOCCN1Cc1cn(CC2CCN2C(=O)CCc2cc(Br)ccc2F)nn1 19977,C(CC(C)C(=O)NCC(CNC(=O)Cc1ccncc1Cl)CO)=CC 19978,C1(CCOC)(NC(c2ccc(Br)o2)=O)CCN(C(=O)Cc2ccco2)C1 19979,c1(C(N2CC3(CCN(C(C4(NC(C)C)CC4)=O)C3)C2)=O)cccc2ccn(C)c12 19980,n1(CC)cncc1CC(N1CC(c2ccccc2)(CO)C1)=O 19981,CC1(C)CC(NC(=O)Cc2ccc(Br)cn2)CN(C(C2COCCO2)=O)C1 19982,Cc1c(Cl)nc[nH]c1=NCC(O)CNC(C1CCCCC12CCC2)=O 19983,N1(C(CSCC)=O)CC(NC(C2CCCN(S(C)(=O)=O)C2)=O)C(n2ccnn2)C1 19984,C(=O)(CC1=CCN(C)CC1)NCC1(C(N2CC(C)C(F)C2)=O)CC(=C)C1 19985,c1(C(=O)NCCC2(COC)CC2)cc(C)n(C)c1.C12(CC1)C(=O)NC2 19986,c1(C(N(C(CN(C(C(COC)OC)=O)C)C)C)=O)ccc2ncccc2c1F 19987,O=C(CCC(F)(F)F)NCC1CC1NC(c1cnn[nH]1)=O 19988,c1(CNC(CC(C)CF)=O)nc(CNC(=O)C(C)c2ccco2)cc(O)n1 19989,C1(N(C(c2cccc(CC)n2)=O)C)CCC2CN(C(=O)CCc3cnc[nH]3)CC12 19990,C1(C(=O)NCC(C)(CNC(c2cc(C3CC3C)on2)=O)OC)CC2(CCC2)C1 19991,N1(C(=O)C=CC=C(Cl)Cl)CCC(F)(CNC(C2CC(C(F)(F)F)C2)=O)CC1 19992,c1(C(N2CCC3(NC(c4ccsc4)=O)C(CC2)C3)=O)cc2c(O)ncnc2cn1 19993,C(=O)(C(F)CCC(C)(C)C)N1CCC(CC#C)(C(=O)NCC2CC2(Cl)Cl)C1 19994,C1(C(N2CC(O)(CCNC(c3n(C)c(Cl)nc3)=O)C2)=O)CC1C1CCCC1 19995,C#CCC(CC(F)F)C(=O)NC1(C)CCCN(C(C2CCC=CCCC2)=O)C1 19996,CCCC(CCC)C(=O)NC1CCN(C(c2c[nH]nc2Br)=O)CC1CC 19997,C(=O)(CN1C(=O)COc2ccc(Cl)cc21)N1C(C)(C(N2CCC(CN)CC2)=O)CC1 19998,C(c1cccc(F)c1)=CC(=O)N(CCCN1CCCC(O)C1)CCC#N 19999,C1(CNC(C(=Cc2cn[nH]c2)C)=O)CN(C(=O)C(F)C(C)(F)F)CC1(C)C 20000,N1(C(C(C(C)C)C)=O)CCC2(CC2NC(c2ncccc2F)=O)C1 20001,C1(CC(=O)N(CC(C)N(C(C)=O)C)C)C(=O)NN=C1C.C1(C2C(=O)N2)CCCCC1 20002,C1(C(N(CCN(C)CCO)C)=O)CC2CCC1N2C(=O)CCCOC(C)(C)C 20003,C1(NC(C(C)n2cncn2)=O)CC2(CCCN(C(C3CC4CCC3C4)=O)C2)C1 20004,N1(C(C(C)(C)CCF)=O)CCC2CN(C(C3CC(=O)OC3(C)C)=O)C2C1 20005,C1(NC(c2occ(C)c2)=O)CCC2CN(C(C3CC4(CCCC4)CO3)=O)CC2C1 20006,C(C(N=[N+]=[N-])C(=O)NCC(O)CNC(c1csc(C(C)C)n1)=O)OCC 20007,CC1(C)C(C)(C)C1(F)C(=O)NCC(C1CC1)NC(c1cnn(C(C)(C)C)c1)=O 20008,C(=O)(CC(C)(C)CN(C)C)NCc1nc(CNC(C(CC)C)=O)sc1 20009,c1(NC(N(CCCN=[N+]=[N-])C)=O)ccccc1C1CCC(=O)N1 20010,c1(C(=O)NCC2N(C(c3cc(OC)no3)=O)CC(O)C2)cccc2c1CNC2=O 20011,CC1(CNC(=O)CC2CCCO2)CN(C(c2ccsc2C(F)(F)F)=O)CCO1 20012,CN=c1[nH]c(=NCC(C)F)[nH]c(=NCCc2ccc3n[nH]cc3c2)[nH]1 20013,CC1(NC(=O)CC2(O)CCC2)CCC(NC(C2CS(=O)C2)=O)CC1 20014,c1(CC)ccc(C#N)cc1COC.C12CCCCN1CCNC(=O)C2 20015,C1(NC(CS(N)(=O)=O)=O)CC(C2CCN(C(c3n[nH]c4c3CCOC4)=O)CC2)C1 20016,C1(n2cc(C(C(OC)OCOC)C)nn2)CN(C(c2conc2C)=O)CC1C 20017,c1(C(N2CC(CC(C)NC(=O)CCS(C)(=O)=O)C2)=O)ccc2c(c1)OCO2 20018,N1(C(c2cc(CCC)[nH]n2)=O)CCC(O)C(NC(c2ncoc2CC)=O)C1 20019,c1(NC(C)=O)ccc(C(=O)NCCCN(C)C(c2ccc(CO)cn2)=O)cc1F 20020,C1(C(N2CCC(CO)C(O)CC2)=O)CC12CCN(C(C1(CO)CC1)=O)CC2 20021,N1(C(N(C)C)=O)CCC(C(=O)NCC(C2CCCC2)NC(=O)CC2(C)CC2)C1 20022,O=C(C1=COCCO1)N1CC2CC2(CNC(C2(n3cncn3)CC2)=O)C1 20023,CC(=O)C(C)CC(C)C(=O)NC(C(=O)NCCSCCCO)C1(O)CCC1 20024,c1(C(N(CCNC(c2c[nH]nc2Cl)=O)CC)=O)cc(OC)cc(C)c1 20025,C1(CC(NOCCOC)=O)CC2(C1)CN(C(=O)CNC(=O)CC(F)(F)F)C2 20026,c1(-n2cc(C3C(=C)CC3)nn2)ccncc1Br 20027,c1(C(N(C2CCN(C(C(C(C)C)OC)=O)C2)C)=O)cc2nccn2c(O)n1 20028,C1(CN(C(=O)CC2CC(SC)C2)CC)CCN(C(=O)C(c2ccccc2)C)CC1 20029,N1(C(=O)CN2CCOCC2)CC2(CC(S(=O)(=O)N3CC(N4CC(O)C4)C3)C2)C1 20030,c1(C(=O)NCC(C)N(C(=O)CN(C)C(=O)OC)CC)cc2nc(C)sc2[nH]1 20031,N1(N(C(CC(C)C)=O)C)CCN(C2CN(c3nncs3)C2)CC1 20032,C(CCN=c1[nH]c(=NC2CCc3cccnc32)c2sccc2[nH]1)=CCCC 20033,C(O)(C(=O)O)(C(F)(F)F)c1cn(C(C(=O)NCc2c(C)oc(CO)c2)C)nn1 20034,N1(C(COC)=O)CC2CCC2(CNC(=O)C(C2CCCCCC2)O)C1 20035,C1(C)(CNC(COc2ccc(C)cc2)=O)CN(C(=O)CCCCCF)C(C)(C)C1 20036,c1(C(N2CC(CNC(C(C)n3ccnc3)=O)N(C)CC2)=O)cnc2occc2c1 20037,C1(NC(c2cc(SC)oc2C)=O)CN(C(C2(C)CCCCO2)=O)CCC1O 20038,N1(CC)CCCN(C(C2OCCC2NC(=O)C(C2CCCCC2)O)=O)CC1 20039,C(CCC(C)(C)NC(c1sc(C(C)C)nc1C)=O)NC(C(COC)OC)=O 20040,C1(C(N2CC(OCC(=O)NC)C2)=O)CCC(O)CN1C(C12CC(C#N)(C1)C2)=O 20041,n1(CC(=O)NC(c2cn(-c3ccsc3C(=O)O)nn2)C)cnnc1O 20042,C(=O)(CC(C(=C)C)OCC)NCC(C(N1CCC(C#C)C1)=O)C 20043,CC1CN(C(c2ccon2)=O)CC(CCNC(c2ccoc2C(F)(F)F)=O)O1 20044,CC1=C(C)CC(C(=O)NCCC(C)(C)CNC(C2CC3CC3C2)=O)CC1 20045,C1(NC(C(C)C#N)=O)CN(C(c2ccc(CN3CCOCC3)s2)=O)CC12CC2 20046,c1(N2C(=O)N3CC4(CCSC)C(C(C)C3(C)C2=O)C4)coc2c(OC)cccc12 20047,CC(C)CC(C)(CNC(=O)COC1CCN(C)CC1)NC(c1cnccc1Cl)=O 20048,CCCCC(CNC(=O)COc1ccon1)NC(=O)C(C(C)C)c1ccncc1 20049,CC(C)CC(C)(CNC(c1ccc(C(N)=O)s1)=O)NC(c1ncc(F)cc1F)=O 20050,c1(CC)nnc2cc(NCC3(CNC(C4CC(N(C)C)CCO4)=O)CC3)ncn12 20051,C(CCCC(=O)NCC(C)(CO)NC(=O)COc1csc(C(F)(F)F)n1)N(C)C 20052,C1(NC(CC(C)(C)C2CC2)=O)CN(C(c2cccc(N)c2O)=O)CCC1CO 20053,N1(C(C2N(C(C)=O)CCCC2)=O)CCC(C)C(NC(c2cnc(C(N)=O)s2)=O)C1 20054,c1(C(N2CCC(NC(CNC(=O)OC)=O)C(O)C2)=O)cc2c(C)[nH]nc2s1 20055,N1(C(c2c(C)cc[nH]2)=O)CCN(C(=O)C(C)Cc2cccc(F)c2)CC(C)(F)C1 20056,c1(N2CCC(OCC(C)C)CC2)ccnc2cc(O)ccc12 20057,c1(C(N2CC(NC(CC(C=C)C)=O)C(C)C2)=O)cc(Cl)ncc1O 20058,C1(C(N(C)CC2CCN(C(=O)OC(C)(C)C)CC2)=O)CC2CC(C1)CS(=O)(=O)C2 20059,O=C(CC1=CCN(C(=O)CC2CCCCO2)CC1)N1CCCN(C2CC2)CC1 20060,c1(N(CC)CC)ccc(C(=O)NCCNC(=O)C(C)NC(C2CCC2)=O)cn1 20061,N1(C(C2CCC(C(C)(C)C)O2)=O)CCN(C(=O)Cc2cccc(F)c2)CC1CF 20062,CC(=O)C(C)CC(C)C(=O)N1CCN(C(=O)C#CC2CCC2)C(C(C)(C)C)C1 20063,N1(C(C(C=C)(C)C)=O)CCC(C2CC2)(NC(=O)C(C)SC(C)C)C1 20064,C1(C)(C(N2CCCC(=C)C2)=O)CCN(C(c2cc(C)ccc2F)=O)CC1 20065,Cn1cc2c(n1)CC(OCCNC(N1CCCC(C)(C(F)(F)F)C1)=O)CC2 20066,N1(C(C=CC)=O)CCC(C(=O)NCC2CSCCO2)C1C(C)C 20067,C(=O)(CCC(=O)N(C)C)N1CC(CCCCNC(C(C)OCC(C)C)=O)C1 20068,Cn1cc(C(=O)NCCC2(NC(=O)C(O)C3CCC3)CC2)c(-c2cnccn2)n1 20069,C(=O)(CC(C(F)F)NC(=O)CC1CC(F)(F)C1)NCC1N(C)CCOC1 20070,C1(NC(c2ccn(CCN(C)C)n2)=O)CCC(NC(=O)CC2CCC3CC23)CC1 20071,C1(NC(c2nc(C)oc2)=O)CCCCC12CCN(C(C1CSC1)=O)C2 20072,C(=O)(C(CC1CCCC1)C(C)C)NCC1(NC(C=C(C)C2CC2)=O)CCOCC1 20073,c1(C(N2CCC(OC)CC2)C(=O)NC(C)C)ccc(OC(F)F)cc1Cl.OC(F)F 20074,C1(n2c(-c3ccc(CN4CCCC4)o3)nc(C(C)C3CC3)n2)CCOC(C)(C)C1 20075,CC1CCCC(C(=O)NCCCOCCC(=O)NCc2ccn(CCF)n2)C1 20076,C(=O)(C1=CCCCCC1)NC(C)CCCCNC(=O)CNC(C1CCCCC1)=O 20077,c1(CSCC(=O)N(C)CC2CN(C(=O)C(C3CCCCC3)O)C2)ccccc1 20078,c1(C(=O)NC2C(CNC(c3cnn(C)c3Br)=O)C2)cc(F)cc(Cl)c1N 20079,C=C(C)CC(C(=O)NCC1CSCCO1)NC(=O)C=C1CCOCC1 20080,N1(C(c2ccc(CSC)o2)=O)CCC2CN(C(C3CC3c3ccsc3)=O)C2C1 20081,CCCCC(O)C(=O)NCC1(F)CC(CNC(=O)CC2(c3ccon3)CC2)C1 20082,C1(C(=O)NCC2CC(OC)C2)(NC(c2cnncc2C)=O)CCN(C)C1 20083,Cc1ccc(C(=O)NCC(CNC(c2cn(C)nc2C)=O)C(F)(F)F)cc1Br 20084,N1(C(CC)=O)CC(N(C)OC)C1.c12n[nH]cc1C(=O)NC2 20085,C(=O)(CCC(F)(F)C(F)F)NC(C1CCOC1)CNC(c1c(C)cnnc1O)=O 20086,N1(C(C(COC)(C)OC)=O)CCC2(CC1)CN(C(c1cocc1C)=O)C2 20087,c1(C(N2CCSCC2)C)cn(CC2C=CCN2C(c2cc(C(=O)O)on2)=O)nn1 20088,N1(C(CC(C(C)C)O)=O)CCC(C2(O)CCN(C(=O)CN3CCCC3=O)C2)CC1 20089,c1(OC)c(C(=O)NC(CNC(=O)Cc2ccc(C)nc2)CO)ccnc1Cl 20090,c1(C(=O)NCC2CC(CNC(CSS(C)(=O)=O)=O)OC2)cc2ccnc(Cl)c2s1 20091,c1(C(N2CCC(N(C(C(CC)NC(N)=O)=O)CCO)C2)=O)cnc(C)c(C(C)=O)c1 20092,c1(CC(=O)N(c2cccc(OC)c2)C(C)C)cccc2ccncc12 20093,C(c1c(C)noc1C)=CC(N1C(C2CCCN(C(CS(CC)=O)=O)C2)CCC1)=O 20094,C1(CNC(C2COC3(CCC3)C2)=O)CN(C(=O)C2=CCCSC2)CC12CCC2 20095,c1(C(N(C2CCCCN(C(=O)C(C)(F)C(C)(C)F)C2)C)=O)ccn2nncc2c1 20096,Cc1nnc2ccc(C(=O)N(C)CC3(CNC(C4(O)CC4)=O)CC3)cc2c1C 20097,CC1CC(CNC(=O)Cc2cscn2)CN1C(=O)CCN1CCCCC1 20098,CCCC(C(=O)N1CCCN(C(c2oc(SC)cc2C)=O)C(C)C1)S(N)(=O)=O 20099,C1(N(C(=O)C(O)CC2CC2)CC)CCCN(C(c2oc(C)cc2C)=O)C1 20100,C#Cc1cnc(N2CCN(C)CC2CNC(=O)Cc2ccn(C(C)C)n2)nc1 20101,CCC(C)(C)CC(=O)N(C(CC(F)F)C(=O)N1CCS(=O)(=O)CC1)C 20102,C(CC(=O)NCCN(C(=O)CC1(C)CCC1)C(C)C)OCCC 20103,CCC(COC)C(=O)NCC(C)(C)C(=O)N(CC(C)C(=O)OCC)C 20104,N1(C(C=CC)=O)CC(C)(C)CC1C(=O)NCC1COCCO1 20105,C1(NCc2c(C)nsc2C)CC(NC(c2ccc(-c3cc[nH]n3)s2)=O)C12CCC2 20106,C(CCCOC)(C(=O)N(C)Cc1cnccc1C)NC(C(CCC)O)=O 20107,C(=O)(C1CCCc2nc[nH]c21)N(CC(C)NC(C1(C)CC2(CCC2)C1)=O)C 20108,CC1CCC(C(=O)NC2CC3(CCC3)C2O)N(C(=O)Cn2cc(CO)nn2)C1 20109,N1(CC(=O)N(C2CCCC(NC(c3ccnc(S)c3)=O)C2)C)CCNC(=O)C1 20110,c1(C(=O)NC2C(C(=O)NCCN(CC)CC)CC2)cccc(C)c1O 20111,c1(OC)cncc(C(=O)NCC(C)(CO)NC(=O)Cc2nc(C3CC3)cs2)n1 20112,c1(C(=O)NCC2C(OCC)CC2)c(CNC(=O)CC(C)(C)O)cnn1C 20113,C1(F)(C(C)NC(C(CC)=CC)=O)CCC(NC(=O)CCCc2cccnc2)C1 20114,Cc1ccc(OCC(=O)NC2CCCC2NC(c2cc[n+]([O-])cc2)=O)cc1 20115,c1(CC(=O)N(CC(C)O)CCNC(C2(CC=C)CCC2)=O)c(C)cccc1C 20116,c1(C(N2C(CCN(C)C)COCC2)C(=O)NC2CCCC2)cc2ccncc2o1 20117,C1(CC=C)(NC(=O)C(O)C2CC2)CCN(C(C2CC2F)=O)C1 20118,c1(C(=O)NC(CCOC)CNC(=O)C(C)(C)C)ccc(OC)c(OC)c1OC 20119,CC(=O)CCCC(C)C(=O)N1CCCC1C(C)NC(=O)C(C)NC(C)=O 20120,C1(C(=O)NCC23OCC(NC(c4ccnc(C)n4)=O)(C2)C3)COCC(C)(C)O1 20121,c1(CC)ccc(-c2nc(C(=O)NCCN(C(=O)C(C3CC3)SCC)C)cs2)cc1 20122,N1(C(C(c2cc(Cl)sc2Cl)C)=O)CCN(C(=O)C(Cl)=CCl)CC1C 20123,Cc1ccc(C(N2CCC(CO)(NC(=O)CCn3ccnn3)CC2)=O)cc1F 20124,CC(CNC(c1[nH]nnc1C1CC1)=O)C(F)C(=O)N1CCC(F)(F)CC1 20125,C1(NC(c2n(C)cc(Cl)c2)=O)CS(=O)(=O)CC1NC(C1CCS(=O)(=O)CC1)=O 20126,c1(CC(=O)NCC(C2CCOC2)NC(C2(CC=C)CC2)=O)csc(COC)n1 20127,C#Cc1cn(C)nc1C(=O)N(C1(C(=O)NC(C)C(C)CO)CC1)C 20128,N1(C(c2n(C(C)C)ccc2)=O)CCCC(NC(=O)C(C)(C)c2cncnc2)CC1 20129,N#Cc1cnc(NC(C2CCCN2C(c2cc(F)cc(I)c2)=O)=O)c(Cl)c1 20130,c1(CC#N)ccccc1C(=O)NCC1CCN(C(=O)CC2CC3C=CC2C3)CC1 20131,c1(CC(C)C(=O)NCC(Cc2ccc(Cl)cc2)CO)ccc(O)cc1 20132,CC1(NC(C2CCC=CC2NC(c2cncc(C#N)c2)=O)=O)CCCC1(F)F 20133,c1(C(=O)NC2(C(N(CC)Cc3scnc3C)=O)CC(C(N)=O)C2)cc(CO)[nH]n1 20134,N1(C(C(C)NC(=O)C(C)(C)C)=O)CC2CCC(CNC(=O)CCC3(C)N=N3)(C2)C1 20135,N1(C(c2c(CCC)cccc2)=O)CCC(NC(=O)CCC(C)N(C)C)C(CO)C1 20136,C(=O)(N=c1ccc(C(C)(C)C)n[nH]1)c1c(OC)cc(C)cc1.C1(C)C(=O)O1 20137,C1(CCC)CCC(CNC(c2cnn(C3CCNCC3)c2)=O)CC1 20138,C1(F)(CNC(c2c(COC)onc2)=O)CCCN(C(c2csc(CO)n2)=O)C1 20139,C(=O)(C1=CCN(C(c2coc(CO)c2)=O)CC1)N1C(C(C)O)COCC1 20140,N1(C(CC)=O)CCC2CN(C(C3CC(=O)C34CCC4)=O)C2C1.C1CCC1(OC)OC 20141,C(=O)(C(C)(C)C(C)C)NC1(COC)CCN(C(C=Cc2n(CC)ccn2)=O)C1 20142,C(C(N=c1[nH]c(=NC2CCN(C)C2C)[nH]c2ccsc12)C(C)C)OC 20143,N1(C(c2c(CC)scc2)=O)CCCC12CCN(C(c1n[nH]c(C)c1[N+](=O)[O-])=O)C2 20144,C(=O)(C(C)(C)C1=CCN(C(c2sccc2F)=O)C1)NC1C(O)CCC(C)C1 20145,N1(C(c2cnc(Cl)n2C)C(=O)Nc2c(C)cc(F)cc2)CCCC2(CCC2)C1C 20146,c1(C(=O)NC(CC(C)NC(Cc2c(CC)con2)=O)C)cc2cc(Cl)ncc2[nH]1 20147,c1(C(=O)NC(CCNC(C(COC)OC)=O)(C)C)cnc2cnccc2c1 20148,C(C(COC)C(=O)NCCCCCN(C(=O)Cn1nccn1)C(C)C)OC 20149,CC1CC(CNC(=O)CCCN(C)C)CN1C(=O)CC12CCCC1C2 20150,c1(CC)nc(NC(=O)CCOCCCNC(=O)C(C)NC=O)n[nH]1 20151,Cc1cc(F)c(C(c2nnnn2C)NCc2cn3ccccc3n2)c(F)c1 20152,CC#CCC(C(=O)N1CCC(CC(C)C)C1)NC(=O)CN1CC(C)(C)C1 20153,C1(CC(N2C(CNC(=O)CC3CCC(F)(F)C3)CC2)=O)CCCC(F)(F)C1 20154,CC(C)CC(CNC(C1C2CCC(C2)C1C)=O)C(=O)NCC#CC1CC1 20155,C(c1ccc(OC)c(OC)c1OC)=CC(N1CC(NC(C(=O)NC)=O)C(O)C1)=O 20156,CN1CCC(N(C(=O)C(=O)NCC2C(C)(C)C2(C)C)C)CC1 20157,C1(C(=O)NCCC(C)NC(c2cn(C)c3ccsc23)=O)Cc2ccccc2O1 20158,c1(CC)ccc(N)c(C(=O)NCC(O)CNC(C2(Cl)CC23CCC3)=O)c1 20159,c1(NC(CCC(CC)NC(=O)CC2C(=O)NN=C2C)=O)ccc2cc[nH]c2c1 20160,C(=O)(C1CCc2ccccc21)N(C1CN(C(CN(CCOC)C)=O)CC12CC2)C 20161,Cc1cc(-c2ncc(Cl)cc2C(=O)NCC2CCC(F)C2)cc2c1NC(=O)CC2 20162,c1(NC(C)=O)cc(F)c(S(=O)(=O)NC(c2ccc(C#N)cc2)(C)C)c(F)c1Cl 20163,CC(N=c1ccnc(Cl)[nH]1)C1CCN(C(=O)Cc2ccc(C(F)F)cc2)C1 20164,C(C(COC)CC(=O)N1CC(F)(CNC(=O)CC2CC2(C)C)C1)OC 20165,c1(CC(C(=O)NC(CNC(COCCCCC)=O)CC)O)ccc(Cl)cc1 20166,CC1C(NC(=O)CN(C)C)CC2CCC1N2c1ccnc(-c2cccc(Cl)c2)n1 20167,C1(CC(=O)NC2C(C)N(C(c3sc(F)cc3Cl)=O)CC2)Cc2cc(F)ccc2O1 20168,N1(C(C2(NC(CCN(C)CC)=O)CC(CO)C2)=O)CC2(C)CC1(CO)C2 20169,N1(C(C2N(C(C(CC#C)C3CC3)=O)CCC(CC)C2)=O)CCCCN(C)CC1 20170,CCCC(CCC)CC(=O)N1CC(NC(=O)C(O)Cc2cccc(Cl)c2)C(C)C1 20171,N1(C(CC(CC)C)=O)CCC(F)(F)C(CNC(=O)C2=CCCCC2)C1 20172,C12(CNC(C3C(C)C3C)=O)CCCCC1N(C(=O)COc1ccsn1)CC2 20173,C1(C(=O)NC2CCN(C(C3CN(CC)C(=O)N3)=O)CC2)C2CCCCCC12 20174,c1(OC)cnc(Cl)cc1C(=O)NC1CCC(C)(CNC(=O)C=CC(=O)N(C)C)C1 20175,c1(CCCC(=O)NCCN(C(=O)CSCC(N)=O)C)n[nH]c2ccccc12 20176,C=CC(C)(CCOC)C(=O)NC(C1CCN(C(c2cc(N)cc(N)c2)=O)CC1)C 20177,N1(C(C(CC)COC)=O)CCC2CCC(C1)N2C(=O)COCOC 20178,c1(CC(=O)NC(C(C)NC(CC(=O)NC)=O)CO)cc(F)cc([N+](=O)[O-])c1 20179,CC1C(=O)N(CC(N2CCCCC2C2(NC(c3ccns3)=O)CC2)=O)C(=O)C1C 20180,C1(COC)N(C(=O)Cn2cc(-c3ccc(CO)s3)nn2)CC1(C)C 20181,n1(CCCOCC)c(N(C)CCOC(C)(C)C)nnc1-c1ccon1 20182,Cc1[nH]nc(C(=O)NC(C)(CNc2cc(O)ncn2)C2CC2)c1C 20183,C=CC1(CC(=O)N(CC[Si](C)(C)C)C)CN(C(=O)C(C)CC2CC2)C1 20184,C1(n2cc(CN(C(C)(C)C)C)nn2)CCCN(C(c2cnn(CCO)c2)=O)C1 20185,C1(C(=O)NC2CN(C(COCC#C)=O)CC2(C)C)C(O)C(=O)N(C)C1C 20186,C(=O)(C1=CCCC1)N(C)CCOCCCN(C)C(C1(c2ncco2)CCC1)=O 20187,c1(CNC(=O)OC(C)(C)C)cc(F)c(NC2C=CC(CO)C2)c(F)c1 20188,CC(N=c1nc(N(CCC(F)(F)F)C)c2c([nH]1)CSC2)c1cc(Br)cs1 20189,C(=O)(C1=NOC2(CCCN(C(=O)OC(C)(C)C)C2)C1)NC1(C)CCCCC1 20190,c1(C(=O)NC(CCC)CNC(c2cc(CO)ccn2)=O)nnn2c1COCC2 20191,Cn1cc(C#N)cc1C(=O)NC12CCC1CN(C(C1CSCCS1)=O)C2 20192,c1(OC)ccc(C=CC(N2CC(NC(C3CCCN3N=O)=O)C(C)(C)C2)=O)nc1 20193,N1(C(C(C(CC)C)C)=O)CCCC(C2CCN(C(C3(C#N)CC3(C)C)=O)C2)C1 20194,C1(NC(C(c2ccc(Cl)cc2)CC)=O)CN(C(=O)C(C)=C2CCC2)CCC1(C)C 20195,CN1CCCCCC1C(=O)NCC#CCNC(=O)CCC1(C)CC1 20196,c1(C(N2C(C(C)NC(CNS(NC)(=O)=O)=O)CCC2)=O)cc(O)c2ccoc2c1 20197,c1(C(=O)NCCOC)cccc(NC(=O)C(=O)Nc2ccc(=O)oc2)c1 20198,C(CO)(C(=O)NC1(CN(C(=O)Cc2ccc(C)s2)C)CC1)OC 20199,c1(CC(=O)NCC=CCNC(C(C)C=Cc2ccccc2)=O)c(F)cccc1F 20200,N1(C(c2c[nH]c(=NC)o2)=O)CCN(C(c2cc(Cl)ns2)=O)C(C)C1C 20201,Cn1cc([N+](=O)[O-])cc1C(=O)NCC1(F)CCN(C(c2cnn(CCF)c2)=O)C1 20202,C1(CNC=O)CC2CN(C(=O)COCCF)CC12.C1(CCC=O)(OCC)CCCC1 20203,C(CN=c1[nH]cc([N+](=O)[O-])cc1C#N)N1CC(NC(C(C)OC2CCCCCC2)=O)C1 20204,c1(C(=O)Nc2cccc(NC(CN(C)CC)=O)c2)cc2oc(Br)cc2s1 20205,C1(CC)CCCC1(C)C(=O)NCCC(=O)N(CC(C)(C)N(C)C)C 20206,N1(C(C=CCOC(C)(C)C)=O)CCOCC(CNC(C2CCCCC2O)=O)C1 20207,c1(C(=O)NC(C2CCCC2)CNC(C2CC(OC)C2)=O)cnc2cc(C)nn2c1 20208,N1(C(=O)OC(C)(C)C)CCC(C(O)C(N2CCC(ON3CCCCC3)C2)=O)C1 20209,N1(C(C(C)Sc2ccccn2)=O)CCC(CO)(CNC(c2cscn2)=O)C1 20210,c1(OC)ncc(C)cc1C(N1CCC(CC(=O)NC2(c3ncccn3)CC2)C1)=O 20211,CN1C(=O)NC(C2CCN(C(=O)NC3(C)CC3c3ccccc3)CC2)C1=O 20212,N1(C(C2CC(SC)C2)=O)CC(O)CC1CNC(=O)CNS(=O)(=O)N(C)C 20213,N1(CC=C)CCC(NC(=O)CN(C(=O)C(O)CC2CC2=C)C2CCC2)C1=O 20214,CCCCN=C(NCC(O)Cc1ccccc1)NCCc1ccc(Cl)cc1Cl 20215,c1(C(=O)NCCCN(CCCNC(CSC)=O)C)cc(C(F)F)ccc1F 20216,c1(OC)ccc(NC(c2cc(-c3ccccc3)nc(O)c2)=O)c(F)c1 20217,c1(C(=O)NC(C2CCCN(C(c3ncccc3O)=O)C2)C)ncnc2sccc12 20218,N1(Cc2ccc(C(CNC(C3C(C)C3)=O)NC(N)=O)cc2)Cc2ccccc2C1 20219,N1(C(=O)NC2CC(COCC)C2)CCC2(CCS(=O)(=O)C2)C1 20220,c1(C(=O)OC)ccc(S(=O)(=O)N2CCC(F)(c3ccc(F)cc3)C2)cc1 20221,C(=O)(C(C)(O)Cn1cc(Br)cn1)NCC(C)CN1CCCC1=O 20222,c1(C(=O)NCC(CC)NC(c2c[nH]nc2C)=O)ccc(SC)cc1 20223,C(C(C)(CC(C)C)NC(C1CCC(C)(F)CC1)=O)NC(C(COC)NC(C)=O)=O 20224,C1(N(C(=O)C(F)CC2CCOC2)C)CN(C(c2cc(N)ccc2F)=O)CC1(C)C 20225,C1(C(N2CCCCC2c2nccs2)=O)CC2CCN(C3CCCNC3)CC12 20226,C=C=CCCC(=O)N1CCC(N(C)C(c2noc(Cc3ccc(Cl)cc3)n2)=O)C1 20227,C(=O)(C1=CC2CC(C1)CC2O)NC(CNC(C1(c2c(C)c(F)ccc2)CC1)=O)C 20228,N1(C(=O)NC(c2cccnn2)CC)CCN(C2CCCN(C(C)=O)C2)CC1 20229,N1(CCC(=O)NCC(CC(C)C)NC(c2ccon2)=O)C(C)CCCC1C 20230,N1(C(C2N(C)C(=O)CC2)=O)CC2(CCCC(CNC(C3CC(F)C(=O)N3)=O)O2)C1 20231,c1(C(N2CCC(OCC=C)C2)=O)cc(Br)c(C)c([N+](=O)[O-])c1 20232,CCCC(C#N)C(=O)N1CC(CC(=O)N(C(C)C(C)CC)C2CC2)C2(CC2)C1 20233,C#CC1(O)CCCN(C(C2C3CN(C(=O)Cc4ccccc4F)CC23)=O)C1 20234,C1(C(C)(C)C)(CNC(COCC(=C)C)=O)CCN(C(C2OCCC2C)=O)C1 20235,c1(NC(C2CC23CNC3)=O)cccc2c1CCS2(=O)=O 20236,c1(C(C)C)ncc(Cl)c(C(=O)NC(CNC(=O)C(F)CC2CC2)C2CCC2)n1 20237,Cc1noc(C)c1NC(c1c(CNC(C2CCC(C)(CC)O2)=O)nnn1C)=O 20238,C1(C(=O)NCC(=O)NCC(=O)NC2(CC=C)CC2)CCCC1 20239,C1(NCC(CN2CC(C)OC(C)C2)O)COC2(CCCCC2)C1 20240,c1(C(CC)O)nc(-c2csc(-c3csc(C)n3)c2)n(CC)n1 20241,S(=O)(=O)(c1ccc2c(c1)COC2)N(c1ccsc1)CC1(O)CC(N)C1 20242,n1(CCOC)c(N2CCN(C(=O)N(C)C)CC2)nnc1C1CC(O)CN1C 20243,c1(C(N2CCCC(Nc3cc(C)nc(C)n3)CC2)=O)ccc2sccc2c1 20244,C1(C(=O)NC2C(C(=O)NCCCn3ncc(C)c3)C2(C)C)CCCCCN1C 20245,C1(OC)CC(NC(=O)C(C)C)CN(C(C2CCCCN2Cc2ccccc2)=O)C1 20246,C#CC1(C(N2CCC(CNC(c3conc3COC)=O)CC2)=O)CCCC1 20247,N1(C(C2CC=C(C)CC2)=O)C2CC(F)C(C2)C1C(=O)NCCc1cccc(F)c1 20248,CC1(CNC(C2CC2(F)F)=O)CCc2ccccc21 20249,CCCCC(C)CCC(=O)NC1CC(NC(=O)C(c2cncn2C)O)C1 20250,N1(C(C2C(C(=O)OC)C=C2)=O)CC2(CCCN(C(=O)C=C3CCC(C)C3)C2)C1 20251,N1(C(CC=CC)=O)CCC2C(CCN2C(=O)Cc2cnccc2OC)C1 20252,C1(NC(CCC(C)(C)c2ccccc2)=O)CN(C(=O)CO)CC12CCOCC2 20253,C#CC1(O)CN(C(=O)C(C)CNC(C2CCOCC2)=O)C1 20254,c1(-c2n(C)cnc2)cnc2ncc(C(=O)Nc3cc4ccccc4cn3)n2c1 20255,C(=O)(C1=C(Cl)CCOC1)N(C)CC1CCCN(C(C2CCC3CC23)=O)C1 20256,Cn1ncc(C(=O)NC2CCCC(NC(c3ccncc3)=O)CC2)c1C#N 20257,C(CC(CC)C(=O)NC1(CNC(c2cnn(CC(F)F)c2C)=O)CCCC1)=CC 20258,c1(C(=O)NC(CO)C(=O)NCC2CCC(F)(F)C2)n[nH]c2c1CCC2 20259,N1(C(C2CCC(=O)OCC2)=O)CCC2(CC1)CCN(C(C1CC13CC(O)C3)=O)C2 20260,C(=O)(C#CC1CCCO1)N(C1CN(C(c2ccc[nH]2)=O)CC12CC2)C 20261,c1(C(=O)NCCOCCNC(CN2CCC(C)C2)=O)cc2cccc(O)c2[nH]1 20262,c1(C(N(C2CCN(C(C3CC3(C)C(C)C)=O)CC2)CC#C)=O)cccc(CC)c1 20263,c1(C(N(CCC(C(C)C)NC(=O)Cn2ncccc2=O)C)=O)c(Cl)cncc1Cl 20264,C1(NC(c2nccc(C)c2)=O)COC2(CCN(C(=O)Cn3c(C)csc3=O)C2)C1 20265,C(=O)(C(C)(F)C(=O)NCC(C)NC(c1ccccc1C(C)(F)F)=O)OC 20266,Cc1nc(C)c(CNC(C2CC=CCN2C(=O)CSC(F)F)=O)o1 20267,CC1CCc2nc(C(N3CC(CO)(NC(c4cc(F)cc(Cl)c4)=O)C3)=O)cn2C1 20268,Cn1cc(Cl)cc1C(N1CCCCC1C1CCCCC1)C(=O)NCC1CCOCC1 20269,CCC1=C(C(=O)NC23CCC(C2)N(C(=O)C=NOC)C3)SCCO1 20270,C1(NC(C2C(C)=C2)=O)CCN(C(=O)Cn2nnnc2C2CC2)CC1C 20271,N1(C(c2c(NC(c3c(C)cnnc3)=O)ccs2)=O)Cc2ccccc2C(F)(F)C1 20272,CCC(O)(C(=O)N(CCCNC(C1(CC)CCNC1=O)=O)CC)c1ccccc1 20273,C1(NC(C=CCC)=O)CN(C(c2ccc(C(N)=O)[nH]2)=O)C2(CCCCC2)C1 20274,C(=O)(C#CC1CCOCC1)NC1(C(N2CCC(C)CC2C)=O)CCCC1C 20275,C(CC1=CCN(C(C2(C3CCOCC3)CC2)=O)CC1)NC(C(C)(C)C(N)=O)=O 20276,c1(C(=O)NCCC2CN(C(C=CSC)=O)C2)ccccc1[N+](=O)[O-] 20277,c1(CC)onc(C(=O)NCC2CN(C(C3CCN(C)C3=O)=O)CC2C)c1C 20278,n1(CC)ncc(C(N2CC(C)(OCC(=O)NC(c3nccc(C)n3)C)C2)=O)c1C 20279,C1(CC)CN(C)c2ccccc2CN1C(=O)C(N1CCN(CCOC)CC1)=O 20280,C(=O)(C1CSc2ccccc21)NCC1(CNC(C(F)=CCC)=O)CC12CCC2 20281,CN1CC(NC(N2CCCC(CCO)CC2)=O)C(F)(F)C1 20282,C1(C(N2CCCC2)=O)CC2(C1)CC(CN=c1ccn(-c3nccs3)[nH]1)C2.n12nnnc1C1CC21 20283,C(=O)(CC(F)(F)F)NCC(C)(CC)NC(c1ccn(CCC)n1)=O 20284,C1(C(=O)NCc2ccc(-c3cccc(C)c3)cc2)COCC(=O)N1C(C)C 20285,n1(CC)ncc(C(=O)N(CCCN(C)CC2CCOCC2)C)n1 20286,Cc1cccc(CNC(=O)CC(C(C)C)NC(C2CC(N(C)C)C2)=O)c1C 20287,C12(COC)CC(NC(=O)C(Cc3ccco3)NC(=O)Cn3cc(CO)nn3)(CO1)C2 20288,c1(CNC(C2CCC2)=O)cccc(N2CCC(NC(=O)C(O)C3CC3)C2)n1 20289,S(=O)(=O)(c1ccc(Cl)c(C(F)(F)F)c1)NC1CCC(NC(C2(F)CC2)=O)C1 20290,C1(COC)(NC(=O)C(C)OCCOC)CCN(C(=O)C(c2ccccc2)C)CC1 20291,CN1CCN(C(c2cnc(C3CC3)nc2)=O)C(CNC(C2CCC3CC3C2)=O)C1 20292,Cc1nc2c(NC(c3ncccc3NCc3cnn(C(C)C)c3)=O)cccn2n1 20293,Cc1ccccc1OCC(=O)NCCN(C1CC1)CC1(C)CC1 20294,N12CC(C3(CC3)C1)C2=O.N1(C(COCCOCC)=O)CC(C)C1.N(C)C 20295,C1(C(N(C)CCOCC2CC2)=O)CC(C)(C)CCN1C(c1cnccc1C#N)=O 20296,C(C(C)(C)CC(=O)NC1(C(=O)NCCC(O)C(=O)OC)CCCCC1)OC 20297,C(C(=O)N(CCCCO)C)(C(C)OC)NC(CCOCC#C)=O 20298,c1(C(N2CC(NS(C)(=O)=O)C2)=O)csc(Cl)n1 20299,C1(NC(c2cc(C(C)C)ncc2)=O)CN(C(C2CCCCO2)=O)CC1(F)F 20300,O=C(C1=C2CCCN=C2NN1)N1CCC2(CC1)CN(C(C1CC(F)C1)=O)C2 20301,CCC(CC(=O)NCC(CC(=O)Nc1ccc(C(C)C)nc1)C1CCC1)OC 20302,C1(C(N(C(C(C)C)CO)C)=O)C2CC3C(C2NC(c2c[nH]c(=N)o2)=O)C13 20303,c1(C(=O)NCCN(C(=O)C(CO)OC)CCOC)ccc(C#N)cc1O 20304,c1(CC(=O)N(C(C)C)CCNC(C2(CCF)CC2)=O)ccco1 20305,c1(NCC(C)CO)nc(NC(CCC(F)(F)F)c2ccccc2)nc2sccc12 20306,c1(C(=O)OC)cc(=NC2CCCC(NC(=O)CCCC(C)=O)C2)[nH]c(Cl)n1 20307,Cc1cc2cc(C(=O)NCC3CCCN3C(=O)C=C3CCN(C)C3)oc2cc1C 20308,c1(C(=O)NC(c2cccc(Cl)c2)CNC(C2(CC)CC2)=O)cnc2scnc2c1 20309,c1(C(=O)NCC2CN(C(CC(CC)OC)=O)C2)cc(Br)c(C)cc1C 20310,c1(C(c2n(CCC)nnn2)NCc2nc(C)n(C)n2)ccc2c(c1)OCC(=O)N2 20311,c1(NC)ccccc1C(=O)NCC1(CN(C)C(c2ccn(CC(C)C)n2)=O)CC1 20312,c1(C(=O)NC2CCC(CNC(c3cnc(C(C)=O)s3)=O)C2)cc(C)c(Cl)cc1C 20313,C(C(O)CS(C)(=O)=O)N(C=O)Cc1c(C)nn(Cc2ccccc2)c1 20314,CCCCC(C(=O)NCCCOC)NC(c1cn(CC)nc1C)=O 20315,Cc1cccc(C(N2CCC(F)CC2C(=O)NCCN2CCCC2)=O)c1O 20316,N(C1CCC(Nc2ncccc2C#N)c2ccccc21)C(C(C)N1CCC1)=O 20317,c1(C(=O)NC2C=CCN(C(Cc3c(C)scc3)=O)C2)cccc(Cl)c1C 20318,Cc1nc[nH]c1CC(=O)N(C1CCC(NC(=O)Cc2cnc[nH]2)C1)C 20319,CON=CC(=O)NCc1nc(C(=O)NCCCC(C)O)co1 20320,C(CNC(=O)Cn1nccc1C(F)F)(CCCC)NC(CCCNC(C)=O)=O 20321,C12(CNC(c3c(C)noc3)=O)CCCC1CN(C(c1cnc(N(C)C)o1)=O)C2 20322,C#CC1(C(=O)NC(CC)CCCCC)CCN(C(C2C3CCC(C3)C2C)=O)CC1 20323,C1(NC(c2c(C)coc2C2CC2)=O)CC(F)CN(C(C2CCCOC2)=O)C1 20324,Cc1nc2nccc(NC3CC(F)(F)CC3C(=O)OC(C)(C)C)n2n1 20325,C1(NC(=O)C=Cc2ccc(Cl)cc2F)COC2(CCN(C(=O)CC3(O)CC3)C2)C1 20326,C1(CNC(C2CCC(C)(CC)O2)=O)CN(C(=O)CSc2nncn2C)CCN1C 20327,c1(C(=O)NC2C(CO)CCN(C(c3c(CC)ccs3)=O)C2)cc(S(C)(=O)=O)co1 20328,Cc1cccc2c1CC(C(=O)NC1CC(CNC(C3(C)CCC(=O)NC3)=O)C1)O2 20329,N1(C(CC(n2ccc(C)n2)C)=O)CCCCC12CC(NC(=O)CC(C)CF)C2 20330,CCC(CC)CC(=O)NC(CNC(=O)CC1CCCN1C)C(C)C 20331,N1(C(=O)OC(C)(C)C)CC2(C1)CC1(CC(NC(=O)Nc3ccc(I)cc3)C1)C2 20332,N1(C(C(CC)=CC)=O)CC2(NC(=O)CCCC(F)(F)F)CCC1CC2 20333,CC1(CNC(=O)CCOCC(F)(F)F)CCN(C(C2CCCC(F)C2)=O)C1 20334,Cc1cc(C(=O)NCC2CN(C(=O)CN3CCCS3(=O)=O)C2)ccc1Cl 20335,N1(C(Cc2n(C)ccc2)=O)CC2(CCCC(CNC(C3CCCCS3)=O)O2)C1 20336,C=CCCC(C(=O)NCC1(C)CCCO1)NC(c1ccccc1Cl)=O 20337,c1(CC)ccc(C(=O)NC2(CNC(=O)CC3CC34CC4)CCCC2)cn1 20338,C1(N(C2CC(CC(=O)O)(CO)C2)C(C2(c3cn(C)nc3)CC2)=O)CCC(F)(F)C1 20339,CS(C)(=O)=NC(=O)C(=O)NC12CC(CNC(=O)CCc3cn[nH]c3)(C1)C2 20340,C1(CCNC(c2cnn(CC3CC3)c2)=O)CC(F)(F)CN1C(=O)Cc1ccno1 20341,N1(C(c2c(N)ccc(C)c2)=O)CC(NC(=O)CC2OCCCO2)C2CCCCC12 20342,CCCCC(C(=O)N(C)CC1CCC(CNC(=O)Cn2ccnn2)CC1)N(C)C 20343,c1(C(N(CC(C)NC(C2CC(C(C)C)C2)=O)C)=O)ccc2cc(O)ccc2c1 20344,C(C(C(C)C(C)C)NC(=O)Cc1ccc(C)cc1)NC(c1ccc(CCC)[nH]1)=O 20345,CC1(Cn2cc(CCN3CCSCC3)nn2)CCCCC1(F)F 20346,C#Cc1ccc(C(N2CCC(C(=O)NCC(O)COC)(CC)C2)=O)o1 20347,N1(C(c2cc(F)cc(Br)c2)C(=O)NC)CCC2CCCCC12 20348,c1(C(N2CCCCC(NC(c3ccc(C)s3)=O)C2)=O)cc(Cl)c(N)cc1F 20349,c1(-c2n(CC=C)c(N(CC(C)C)CC)nn2)ccc(S(C)(=O)=O)cc1 20350,C(=O)(C#Cc1ccccc1)NC1CC(CC(=O)NC2CCN(C(C)=O)CC2)C1 20351,c1(C(C)C)ccccc1C(=O)NC1CC1CNC(=O)C=C1CC1 20352,C1(NC(C(CSC)(C)NC(=O)Cn2cnnc2)=O)CCN(OC)CC1 20353,N1(C(CCCOCC)=O)CCCC(NC(C2(n3ccnn3)CC2)=O)C1 20354,N1(C(CN(C2CC2)CC)=O)CC2CC(C(=O)NCc3cnc(C)cc3C)(C2)C1 20355,CN=c1nc(N2CCC(C)(CC#N)C2)[nH]c(=NCC2(c3ccccc3C)CC2)[nH]1 20356,c1(C(N2CC(C)C(CCNC(=O)CCS(C)=O)C2)=O)cc(F)c(F)c(C#N)c1 20357,c1(CN(CCN)CC2CC2)cc(Cl)cc(Cl)c1Oc1ccc(Cl)cc1 20358,C1(CNC(CSCC(=O)OC)=O)CC2CCC1N(C(=O)C(C)C1CCOC1)C2 20359,C(=O)(CCCC(F)(F)C(F)(F)F)N1CCCC(CC)(NC(=O)CCC2CCCO2)C1 20360,n1(CC)cnc2c(NC(C)(C)CF)nc(N3CCC(CC(C)C)C3)nc12 20361,C1(NC(c2cc(COC)[nH]n2)=O)CCCCC1CNC(=O)Cc1ccns1 20362,CN1CC(CC(=O)NCCOCCN(C(=O)CC=C(Cl)Cl)C)C(O)C1 20363,c1(C(N2CCC(N(C)C(C3(C)CCCC3)=O)C2)=O)cc(F)c2cn[nH]c2c1 20364,N1(C(Cc2cc(C)nn2C)=O)CCCC(C)(C(=O)Nc2cccnc2C(C)C)C1 20365,C1(CCCC)CCCN1C(=O)C(C1CCC1)NC(=O)C=CCC1CCCC1 20366,c1(CC)cc(N2CCCC(NC(C3CCC(=O)N(C)C3)=O)C2C)nc(CC)n1 20367,CCC(CC(=O)N1CC(C2CC2C(=O)N(CC(C)C)C)C1)C(C)(C)C 20368,C1(NC(C(C)OCC)=O)CCCCN(C(C2(C)CCN(C)CC2)=O)CC1 20369,C(=O)(C1CCCc2nc[nH]c21)N1CCC(NC(=O)C=Cc2ccsc2)C12CC2 20370,Cc1nc[nH]c(=NCC2(C)CCN(C(=O)CC(C(F)F)c3ccccc3)C2)c1Br 20371,CCCCCCCCCCCC(=O)N(CC(CC)NC(C1(OC)CCSC1)=O)C 20372,C1(NC(c2cc(CC)c(OC)cc2)=O)C2CC(CN(C(C3(O)CC3)=O)C2)C1CO 20373,Cc1cccc2c(CC(=O)NC3CCCC3NC(C3CC4(CCC4)C3)=O)c[nH]c12 20374,C1(COC)CCCN1C(=O)C(n1nnnc1C1CCC1)C 20375,N1(C(CC2CC(OCC)C2)=O)CC2CC2(CNC(c2cnc(C3CC3)s2)=O)C1 20376,C(CC1=CCN(C(C2CC(=O)OC2(C)C)=O)CC1)NC(CC(C)CN(C)C)=O 20377,C1(CC(=O)NC(c2nc(C)cs2)CC)CN(Cc2ccc(C(=O)O)s2)CCO1 20378,Cc1cc(CC(=O)NC23CC2CN(C(=O)CSc2cn[nH]c2)C3)nn1C 20379,N1(C(C(CC)C#N)=O)CC2CCOC2(C(=O)OC)C1 20380,C1(C(F)(F)F)CCN(C(=NCc2ccc3c(c2F)CCCC3)NC2CC2)CC1 20381,CC1CCCN(C(c2c[nH]c(=O)cn2)=O)C1CNC(=O)C(O)Cc1cnc[nH]1 20382,Cc1ccc(C(F)(F)C(=O)NC2CCC(NC(C3CC(=O)N(O)C3)=O)CC2)cc1 20383,c1(C(N2CCC(C)(O)C2)C(=O)NCCCC)cc(Br)c(OC)nc1C 20384,C=CCCCC(C(=O)N1CC(=O)N(C)C(=O)C1)NC(c1nc(C)ccc1C)=O 20385,O=C1NCCCCC1NC(c1ccc(I)cc1)c1nnnn1CCCF 20386,N1(C(C(CN(C)C)O)=O)CCC(N=[N+]=[N-])(C(=O)N(C)Cc2ccccc2)C1 20387,Cc1cc(NCC2CC2)ncc1S(=O)(=O)NC1CCC2C(CC1)C2(F)F 20388,O=C(CC1=CSC2=NCCN12)N1CCC(O)(CF)CC1 20389,c1(OC)ccc(C(N2CC(O)(C(C)NC(=O)C(O)Cc3[nH]cnc3C)C2)=O)o1 20390,CCC(C(=O)N1CC2CC1(C(=O)NCCC1(COC)CCC1)C2)C(F)(F)F 20391,c1(CC)occ(C)c1C(=O)NCC1CCCC(NC(C2(N=[N+]=[N-])CC2)=O)C1 20392,c1(C(=O)NCC(C2CC2)NC(=O)Cc2cnsc2)cn2cnnc2cn1 20393,CN1CCN(C(=O)Cc2n[nH]c(=N)s2)CC1CNC(C1CCCCC1CO)=O 20394,C(CC(=O)N1CCC(OC2CCC2)C1)(C(F)(F)F)NC(C(F)=CCC)=O 20395,C1(NC(c2c(C)n[nH]c2)=O)C2CCN(C(=O)C=CC(=O)NC3CC3)CC12 20396,Cc1ccnc(N2CCCC2(C)CC2CCCC2)c1Br 20397,Cc1cccc(CC(=O)NCCC2CCCCN2C(=O)Cc2cccnc2)c1 20398,c1(C(=O)NC(c2ccc(C)cc2)c2ccccn2)ccc(F)c(C)c1Cl 20399,N1(C(C2(CC=C)CC2)=O)CC2(CO)CC1(C(N1CCOC(C3CC3)C1)=O)C2 20400,CC1CN(C(C2(CO)CCCC2)=O)CC(C)C1NC(c1cc(C2CC2)cs1)=O 20401,N1(C(C(CC=CC)C)=O)CC2CCC(NC(c3ccn(CC(C)C)n3)=O)(C2)C1 20402,c1(C(=O)OC)no[nH]c1=NC(=O)c1nc(C(=O)Nc2csc(C)n2)cs1 20403,C1(NC(CC(C)SC)=O)CCCC(NC(c2cn(C(C)C)cc2C)=O)C1 20404,c1(SCC)ncc(Br)cn1.C1C(C(=O)N(C)CC)n2cc(nn2)CCCO1 20405,c1(C(N2CC3(OCC(NC(c4ccco4)=O)C3)C2)=O)c(F)ccc2occc12 20406,O=C(C#Cc1c(F)cccc1F)Oc1nnc(CC2CC2)s1 20407,S(=O)(=O)(C1CC1)NCC(=O)NC(CN(C(=O)CC(C)C1CC1)CC)C 20408,C1(C(=O)NC2CCCC(C(N(CCCC(C)C)CCO)=O)C2)CC2(C1)CC(O)C2 20409,C1(C(N(CCCC(=O)NC)C)=O)C(C2CC2)CCN1C(C1CCCC1)=O 20410,C1(CNC(CS(C)(=O)=O)=O)CC2(CCN(C(c3cccc(C#N)c3F)=O)CC2)C1 20411,C1(C(=O)NC2CCN(C(C)=O)C2)CC(N=[N+]=[N-])CN1C(=O)Cc1cn[nH]c1 20412,C1(NC(c2ccon2)=O)CN(C(c2cnc3ccnn3c2)=O)C2(CCOC2)C1 20413,c1(CC2CCN(C(c3cc(Cl)ccn3)C(=O)NCC(C)C)C2)ccc(F)c(F)c1 20414,N1(C(c2c(CC)nc[nH]2)=O)CCC2(C1)CN(C(=O)CCc1ccncn1)C2 20415,N#Cc1ccc(C(=O)NC2CC2CNC(C2CCS(=O)(=O)C2)=O)o1 20416,CC(CN(C)C)CCC(=O)NCC(O)CNC(C12CCC(CC1O)C2)=O 20417,c1(C(N(CC(CC)NC(c2nccc(OC)c2N)=O)CC)=O)cnn2c1CCC2 20418,C#CCCCC(C)C(=O)NCc1ccc(CNC(=O)C(C)(C)OC(F)(F)F)cc1 20419,c1(C(N2CC(OCCC(=O)NC(CCC)CC)C2)=O)cc2occc2[nH]1 20420,N1(C(CN2CC(C)C2)=O)CCOC2(CCN(C(=O)C3=CCCCCC3)C2)C1 20421,c1(OCC)cnc(C(=O)NC2CCC2NC(c2ccon2)=O)cn1 20422,C#Cc1ccc(C(=O)NC2CCCCN(C(c3scnc3CC)=O)C2)cn1 20423,c1(OC)cc2cc[nH]c(=O)c2s1.c12ccccc1-c1cn(nn1)CC(=O)N1CC2C1 20424,CC1C(NC(=O)C(C)NC(N)=O)CCCN1C(C1CC12CCCC2)=O 20425,C1(NC(CCN(C(C(CC)CCOC)=O)C2CC2)=O)CCN(C)CC1(C)C 20426,c1(C(C)C)ccc(C=CC(=O)N(C)CCN(C)C(C2CSCCS2)=O)cc1 20427,N(C1CCCc2cccc(F)c21)S(c1ccc(C(C)(C)C)cc1)(=O)=O 20428,N1(CCC)CC(NCC2(C)CC2(F)F)CC1=O 20429,N1(C(C(=O)NCCOC)=O)CCCC(C(=O)NCC23CC(C2)C(C)O3)C1 20430,c1(CN(C)CC2CCCN(C(c3ccc(F)cc3Cl)=O)C2)ccc(C#N)cc1 20431,C=CCC(C)(C)CC(=O)NCc1ccccc1CNC(C1NC(=O)CC1C)=O 20432,N1(C(C2C(=C)C2C(=O)OC)=O)CCC(CO)C(O)C1.C1C(=O)N1CCC 20433,O=C(N=c1nc(-c2ccsc2)[nH]s1)c1cncc(OC2CCOCC2)c1 20434,C1(CC)CCCC1(C)C(=O)NC(C1CCN(Cc2ccsc2)CC1)C 20435,C12(NC(c3cccc4nonc34)=O)CCCN(C(C3CC(F)(F)C3)=O)CC1C2 20436,Cc1cc(C(N2CCC(CCNC(c3csc(Cl)n3)=O)CC2C)=O)nc(C)n1 20437,N1(C(CC2CC(C)(C)C2)=O)CC2(CC(NC(C3(C)CNC(=O)C3)=O)CO2)C1 20438,Cc1cc(F)c(NC(CNC(CC2CC2(F)F)C(=O)OC(C)(C)C)=O)nc1Br 20439,c1(OC)cc(Br)c(CN(c2ccnc(F)c2F)C2CC3CNC2C3)cc1O 20440,c1[nH]ccc1C(=O)NCCC(C)OCC.C1(C(=O)N)CCCN1C(=O)C1CC1 20441,Cc1ccc(N2CCOC2=O)cc1NC(=O)CC(c1cccs1)n1cccc1 20442,C1(NC(C(C)C(F)F)=O)(CNC(c2cnn(C3CC3)c2)=O)Cc2ccccc2C1 20443,c1(-c2cn(CCC)nc2)nc(C(=O)N(Cc2ccccc2Cl)CC2CC2)c(C)s1 20444,CC(C)C(C(=O)N(C)CCOCCN(C(=O)CC1CCCC(=O)C1)C)NC=O 20445,N1(C(C2(OC)CCN(C(c3scnc3Cl)=O)C2)=O)CC(C)(C2CCC2)C1 20446,C1(CNC(c2ccc(SC)s2)=O)CC(NC(=O)Cc2cncnc2)C12CCC2 20447,C1(O)(CN(C)C(c2ccc(C(C)(F)F)cc2)=O)CCN(C(C2CC2F)=O)C1 20448,N1(C(c2c(C)ncn2O)=O)C2CCC1CN(C(c1cc(CO)ccc1Cl)=O)C2 20449,c12cccc(c1)OC2=O.c1(COC)nc(C(=O)NC(c2nn[nH]n2)C)cs1 20450,N1(C(C=C(CCC)C)=O)CC(NC(c2ccc(O)cc2)=O)CC1(C)C 20451,C1(NC(C(C)c2cccs2)=O)CN(C(c2cncn2C2CC2)=O)CC1C1CC1 20452,c1(OC)ccc(-n2nnc(NC(c3cnnn3C(C)C)=O)c2C)cc1 20453,c1(C(=O)NC2(C)CCCN(c3cnc(C#N)cn3)C2)cc2n(n1)CC1(CC1)C2 20454,c1(C(c2nnnn2C)Nc2ccc(OCCC)cc2C)ccc2c(c1)CCC2 20455,C1(C(N2CCC(C(=O)NCCOCCC=C)(CF)C2)=O)CCCC2(CC2)C1 20456,CCCC(O)C(=O)NC1CN(C(=O)C(CC)OC)C1 20457,C1(N(C(=O)CCCc2sccc2C)CC)CCCN(C(C2CCCCC2)=O)C1 20458,C#Cc1cccc(CNC(C2CCCCN(C(=O)CC3CCCC(C)O3)C2)=O)c1 20459,C1(CNC(C2C(C)OCCC2)=O)CC2(CO1)CN(C(c1nnc(S)n1C)=O)C2 20460,N1(C(c2n(CC)ccn2)=O)C2CCC1CC(C(=O)Nc1cnn(CC(N)=O)c1)C2 20461,c1(C(=O)NC(C(=O)NCCOC)C2CCCO2)cnc(O)c(F)c1 20462,O=C1CC(C(=O)N2CCCOCC23CCC3)c2ccccc21 20463,C1(CC)CCN(C(=O)C(C)C2CCCC2)C(CNC(=O)CCC(F)(F)F)C1 20464,c1(C(=O)NC2CC(NC(CCCc3onc(C)n3)=O)C2)ccc2c(c1)COCO2 20465,c1(CC)cc(F)ccc1C(=O)NCC(=C)CCNC(=O)C(C)(C)F 20466,c1(OCC(=O)N(CC(C)CNC(=O)CNS(C)(=O)=O)C)ccc(C#N)cc1Cl 20467,C1(CC(=O)NCC2CC(C(N3C(CCC#C)CCC3)=O)C2)CC(O)C1(C)C 20468,NS(=O)(=O)CCC(=O)NCCC1CCN(C(=O)CN2CCN(C3CC3)C2=O)CC1 20469,CCCC(CC(C)C)C(=O)NC1CCN(CCCNC(=O)C#CC(C)C)C1 20470,c1(C(C)(F)F)ccccc1NC(C1CC1c1ccc(Cl)cc1)=O 20471,N1(C(C(=O)NCCC(=O)OCC)CC(O)CC)C2CCC1CC(CCCF)C2 20472,N1(C(C2(CNC(C(C)N(C)C)=O)CC=CC2)=O)CCCNC(=O)C1 20473,c1(OC)ccc(C(=O)NCC2(NC(=O)CC3CCC(=O)C3)CCCC2)cn1 20474,C=C=C(C)CC(=O)NCCC(C)NC(=O)C(c1ccc(OC)cc1)CC 20475,c1(C(=O)NCC2CN(C(C3C4CCCC34)=O)CC2(F)F)scc2c1CCCC2 20476,c1(OC)cc(C)c(NC(=O)C(=O)NCCN2CCNC(=O)C2)cc1F 20477,N1(C(CC(C)F)=O)CCCCC12CN(C(=O)C(F)(F)c1csc(=N)[nH]1)C2 20478,C1(C(=O)NCC2(OC)CN(C(=O)CC3(O)CCCCC3)C2)CCCC(C)(C)O1 20479,C(=O)(C1=CCc2ccccc21)NC(C)CC(C)NC(c1sccc1S(N)(=O)=O)=O 20480,C1(NC(CSc2ccc(OC)cc2)=O)CCN(C(=O)CCCCCBr)CC1F 20481,c1(C(=O)NC2CC3CN(C(c4c(Cl)nc(OC)s4)=O)CC32)cncc2nc[nH]c12 20482,Nc1cc(C(=O)NCC2COCC2NC(C2(O)CCC2)=O)c(F)c(F)c1F 20483,C1(NC(C2(C)CCN(C)C2)=O)CC2CC(NC(c3occc3C3CC3)=O)C2C1 20484,c1(C(=O)NCC2(O)CCCN(C(C(C(C)O)(C)C)=O)C2)cccn2nccc12 20485,C(c1ccc2c(c1)OCO2)=CC(=O)NC1(CNC(C(CCCC)C)=O)CCOC1 20486,C1(OC)CC(CC(N2CC(CN(C(=O)CCN3CCC(C)CC3)C)C2)=O)C1(C)C 20487,c1(C(=O)OC)ccc(OC)c(F)c1NC(C1CSC(c2ccccc2F)C(=O)N1)=O 20488,c1(C(N2CC(F)(CNC(C3CCC(CC)C3)=O)C2)=O)ccc(OC)c(Cl)c1OC 20489,c1(OC)c(C(=O)NCCC2CN(C(C3CCCC(F)C3)=O)C2)c(C)nn1C 20490,C12(C(=O)NCc3ccc(C)nc3O)CCC(CN(C(=O)C(F)CCC(C)C)C1)C2 20491,c1(C(N2C3C(NC(C4C(CC)C4)=O)C(C3)C2)=O)ccc(S(=O)(=O)CC(N)=O)cc1 20492,c1(C(=O)NCC(C(C)C)NC(Cn2c(C)nnn2)=O)ccc(N=S(C)(C)=O)s1 20493,C(CNc1ccc(-c2ccc(Cl)cc2)cc1F)(CS(C)(=O)=O)OC 20494,C1(CCC(=O)NCCOCC#C)CCN(C(=O)Cc2cncnc2)C1(C)C 20495,C1(CNC(=O)C=Cc2cc[nH]c2)CC2CCC1N2C(C1(CO)CCOCC1)=O 20496,C(=O)(C(O)C(F)(F)F)N(CCNC(C1CCC(=C)CC1)=O)CC1CC1 20497,c1(C(N(C2CCN(C(CCCC#C)=O)CC2C)C)=O)ccc2cccnc2c1 20498,c1(C(=O)NCC2(O)CCCN(C(c3c(C)cnnc3)=O)C2)cc2ncccc2o1 20499,Cc1c([N+](=O)[O-])c(C(=O)NC(C)Cn2cccn2)nn1C 20500,CCCC(C(O)C(=O)N1CCOC(C)(C)CC1)NC(c1ccc(CO)cc1)=O 20501,C(C)(CO)(C(=O)NC1CCOC(C(=O)NCC(C)CC2CCCC2)C1)OC 20502,c1(N2C(CCCNC(C)=O)CCC2)ccc(C#N)nc1.C12CCCN1CC(=O)N2 20503,CCCC(O)C(=O)N1CCC(OC2CN(C(C3COCCN3C)=O)C2)CC1 20504,C12(C(=O)NC3(C)CCSC3)CC(CO)(CN1C(C1(C#N)CC3CC3C1)=O)C2 20505,C1(C(=O)NCC2CC(F)(CNC(=O)C(O)CSC)C2)(OC)CCOCC1 20506,c1(C(=O)NCCN(CCOC)C(c2c[nH]cc2Br)=O)scc(C)c1Cl 20507,CN1C(=O)CN(CC(=O)NCCCNC(=O)CCc2cc(Cl)no2)C1=O 20508,N1(C(C(=O)NCC(=C)C)C2CC2c2ccsc2)CC2CC2(C(N)=O)C1 20509,N1(C(C(C)OCCC=C)=O)CC(CNC(=O)C(C)OC2CCCC2)(SCC)C1 20510,n1(CCCC(=O)NC2CC(F)(CNC(COCCCC#C)=O)C2)c(C)csc1=O 20511,N1(C(c2nnc(C(C)(C)C)s2)=O)CC2(CCN(C(=O)C=CI)CC2)C1 20512,C(CCSC)(C(=O)NCC(CO)NC(=O)C=Cc1scnc1C)OC 20513,n1(CCCC(=O)NCCN(C(C2CCCC2)=O)C2CC2)cnc2ccccc12 20514,Cc1c(NCc2cc(C(C)(C)C)n[nH]2)ncnc1N1CCCC(N2CCC2)C1 20515,N1(C(c2cnc(C)n2C)=O)CCC(n2cccn2)(C(N2CCSC2(C)C)=O)CC1 20516,CC1CC(C(N2CCC(CN(C(=O)Cc3cn(C)nn3)C)CC2)=O)CCO1 20517,C1(NC(C=CC)=O)CCN(C(=O)C(c2ccccc2Cl)(C)C)CC1F 20518,N1(C(c2c(C)n(-c3cccc(Cl)c3)nn2)=O)CCCC2C1CCN2C(=O)C1CC1 20519,c1(C(N2CC(c3cnc4ccc(F)cn34)C2)=O)ccc(=O)n2c1CCC2 20520,C1(OC)C(NC(=O)CNC(=O)CN2CCC(C)CC2)CC1(C)C 20521,C(=O)(CC1CCCc2cc(OC)ccc21)NC1CN(C(C=CC)=O)CC1(C)C 20522,c1cn(C)nc1C1CC1.c12nnnn1CCC2NC(C)CCC1CC1.C(C)(C)C 20523,CCC(C(=O)NCC(C)(C)CN(C)C(C1CC12CC2)=O)n1ccnc1 20524,N1(C(C2(CC#C)CCC2)=O)CCC(NC(=O)CNS(N)(=O)=O)C2(CCC2)C1 20525,CC(C)CCCCC(=O)NC1CN(C(C2CC(c3cccc(F)c3)C2)=O)CC1O 20526,c1(C(=O)NC2(CN(C(CCn3c(C)ncc3)=O)C)CC2)cnn(C)c1C 20527,C1(C(N2C(CN(C(C3CC(=C)C3)=O)C)COCC2)=O)OCCCC1(C)C 20528,C=C=C(C)C(=O)NC(c1cn(C2C(N(C)C)CCC2)nn1)C(C)C 20529,C(C(=O)NCCC1CCCN(C(c2cn(C)nc2Cl)=O)C1)(C(F)(F)F)OC(C)=O 20530,C1(C)(CNC(CC2OCC(C)(C)C2)=O)CCC(O)CC1.C12(CCC1)C(=O)N2C1CC1 20531,N1(C(C2(CC#C)CC2)=O)CC(NC(=O)CN2CCC(C(N)=O)CC2)C(F)C1 20532,Cc1cc(F)ccc1N1CCCC(NC(N2CCC3CC23)=O)C1 20533,N1(C(C2=CC(C)C2)=O)CCC(CNC(c2cnco2)=O)C1(C)C 20534,C1(NC(=O)CCSc2ccccc2)CCCC12CCN(C(=O)CCOC1CC1)C2 20535,CC1(C)CN(C(=O)C2=COCC2)CC1NC(C1C2CCCC12)=O 20536,N1(C(C(C)NC(=O)NC)=O)CCC2(CC1)CC(NC(=O)CC1(O)CC1)C2 20537,C=CCC(F)(F)C(=O)N1CCC(F)(CNC(C2(C)CC(F)C2)=O)CC1 20538,C(=O)(C(C)(F)C(F)(F)F)N1C(CNC(c2c(SC)cccc2F)=O)CCCC1 20539,Cc1ccc(CN2CC3C(C2)N3C(=O)C(c2ccccc2)C)c(C)c1 20540,c1ccc(Cl)cc1O.C(c1ccncn1)=CC(=O)NCC12CCN(C1)C2=O.C 20541,CCC(CC(=O)NC(CCO)C(F)F)N(C)C(C1CC(C)(CC)C1)=O 20542,C1(CCNC(c2ccnc(OC(F)(F)F)c2)=O)CN(C(C2(F)CC2)=O)CCS1(=O)=O 20543,c1(C(=O)NCC(CC=C)NC(=O)C=Cc2ncc(C)[nH]2)ccc(Br)cc1N 20544,C(=O)(C(O)CC(F)(F)F)NC(C(=O)N(CCOCC#C)C)CCSC 20545,c1(OCCC(=O)NCC(CO)NC(CC(C)N2CCCC2)=O)ccc(F)cc1 20546,C1(C(=O)NCC2C(CC(=O)N(C(CC)CC)CCO)C2)CNC(=O)O1 20547,c1(CCNC(C(CC2CC2)NC(C(COC)C)=O)=O)ccccc1F 20548,c1(NCc2cc(C(N(CCOC)CCO)=O)ncc2)cc2cccnn2n1 20549,C1(C(N(C2CCC(NC(C3(CO)CCCO3)=O)CC2)C)=O)C2CC3C(C2=O)C13 20550,C(=O)(C1=C(Cl)CCOC1)NCCCCNC(=O)CCCn1cccn1 20551,C1(NC(c2ccc(C)nc2O)=O)COC2(CCN(C(C3COC(=O)C3)=O)CC2)C1 20552,N1(C(C2OCCC(NC(C(C)(C3(C)CC3)OC)=O)C2)=O)CC2CC=CCC2C1 20553,c1(NC(C(C)OC(c2cccc(C#N)c2)=O)=O)ccc(C(F)(F)F)c(Cl)c1Cl 20554,CC1CN(C(c2csc(C3CC3)n2)=O)CC1CNC(C1(n2cccn2)CCC1)=O 20555,C(=O)(C#CC1CCC1)NCCCC(=O)NCC1CCC(C)C1 20556,C1(C(N2CC3C(C)C3C2)=O)CC12CCN(C(C13CCCC(CO1)C3)=O)CC2 20557,c1ccc(C2SCCS2)cc1.C1(C(=O)NC(C)CNC(C2CC2)=O)(OCC)CCC1 20558,c1(C(=O)OC)cc(C)c(C(=O)NC(C)CN(C(=O)C(C)(C)c2ccnn2C)C)o1 20559,CCC(C)CCCCC(=O)NCCC1CSCCN1C(=O)C1=CCC(C)CC1 20560,N1(C(c2sc3ccn(C)c3c2)=O)CCC2(CCN(C(c3cc(F)c[nH]3)=O)C2)C1 20561,C1(CNC(C(COC)OC)=O)CCC(N(C(=O)CN2CCCC2=O)C)CC1 20562,C12(C)CCCN(C1)C2=O.C1(NC(COC)=O)CCN(C(=O)C(C)C)CC1 20563,CCCC(CCC)NC(=O)C(O)C1CN(C(=O)CCCC2CC2C)C1 20564,C12(C(=O)OC)CCC(C(=O)NC3CCN(C(=O)C(COC)OC)CC3C)(CC1)C2 20565,N1(C(C(C=CC)O)=O)CCC(C)(C(=O)NCC2CC23CCOCC3)CC1 20566,c1(CC(=O)NC2C3(NC(CCOC)=O)CCC(C2)C3)c(C)nc(O)nc1C 20567,C1(CNC(C2(C)ON=C(C)C2)=O)CC2(CO1)CN(c1cc(O)nc(O)n1)C2 20568,CC1CN(C(C2(NC(c3ccc(Cl)s3)=O)CCSC2)=O)CC(C)(C)O1 20569,c1(C(=O)NC2C(NC(C(C(C)C)OCC)=O)C2)sc(Cl)c(Cl)c1OC 20570,C1(NC(c2nc(C)oc2C)=O)CC(C)CN(C(=O)CC2(C)CCC2)C1 20571,S(=O)(=O)(c1ccc(C(=O)NCC2CCC2NC(C2(C)COCCO2)=O)cn1)NC 20572,C1(CNC(=O)C(C2CC2)C2CC2)CC2COCC2N1C(=O)CCCCCO 20573,C(=O)(CCC1=CCCCC1)NC1(CO)CCCN(C(CCN(CCC)C)=O)C1 20574,N1(C(=O)CN2CCCC2=O)CCCC2CN(c3cc4nncn4cn3)CC12 20575,C1(C(=O)NCCc2onc(C)n2)CC2CC1CC2NC(=O)C(C)CN(C)C 20576,C1(C(=O)OCC2C(CC)C2)CCCCN1CC(F)F 20577,C1(CC(=O)NC2(CC)CCN(C(COCCC)=O)CC2)COCC2(CCC2)O1 20578,C1(C(N2CC(CNC(COC)=O)C(C)C2)=O)CCCCC1C1CC1 20579,C1(C(N(CC#C)C2CC2)=O)CSCN1C(C1CCCC1O)=O 20580,c1(CC)ccc(C(=O)NC2CCC2NC(c2cccnn2)=O)cc1CC 20581,c1(CN=C(NC2(C(F)(F)F)CC(C)(C)C2)NC2CC2)ccc(O)cc1Cl 20582,Cn1nc(O)cc1C(=O)NCc1ccccc1CNC(=O)C=Cc1nccs1 20583,CCCCCCCC(=O)N1C2CCC(C2)C1CNC(c1ncccc1C(C)=O)=O 20584,C1(CCOC)(NC(=O)C(F)=CC2CC2)CCN(C(c2cnc(C)n2C)=O)C1 20585,c1(COC)noc(Cn2cc(CCn3cncn3)nn2)n1.C1C(=O)N(C)C1 20586,CCS(=O)(=O)CCCNC(c1nnnn1-c1ccc(F)cc1)c1cnco1 20587,C1(C(=O)NCCCC(C)NC(=O)C(c2ccc(F)cc2)=O)CC(=O)NC(=O)N1 20588,O=C(CC1CC12CC2)Nn1cnnc1 20589,N1(C(C2(COC)CC2)=O)CC(CCNC(=O)C=Cc2ncc[nH]2)C(C)C1 20590,C1(NC2(C(N)=O)CCN(C(=O)OC(C)(C)C)CC2)CCC12CCOCC2 20591,N1(C(C(N2CCCCC2CF)=O)=O)CCC(O)(c2cccc(Br)c2)C1 20592,c1(CC)nc(CC(=O)NC2(C(C)NC(=O)C=CCF)CC2)cs1 20593,C1(C#CC(=O)N2CCC(F)(CNC(c3n[nH]c(C)n3)=O)CC2)(CC)CC1 20594,N1(C(C(=O)NC2CCC(N3CCCCC3)C2)=O)CCc2nccn2CC1 20595,C(=O)(C(CNC(C1CCCCO1)=O)CC1CC1)N(CC(CCC)O)C 20596,N1(C(C(CC)NC(N)=O)=O)CCC(CC)CC1C(=O)NCC(C)(C)COC 20597,C1(NC(C=Cc2n(C)ncc2)=O)CC2(C1)CN(C(C1CC3(C1)CC3(F)F)=O)C2 20598,c1(C(C(=O)NCC=CBr)NC(=O)CN2CC=CC2)cccnc1 20599,N1(C(CC2(C)CC2)=O)CCCCC(C2CN(C(C3CCS(=O)(=O)C3)=O)C2)C1 20600,c1(OC2(CC(=O)NC(CC)CNC(=O)CSCC(=O)OC)CCC2)ccccc1 20601,C(C(O)CCNC(c1cc(F)c[nH]1)=O)NC(c1cc(-c2ccccc2)cs1)=O 20602,N1(C(C2C(C(=O)OC)C2(C)C)=O)CC2CCC(CNC(=O)C=CC3CCC3)C2C1 20603,C(CC(=O)NC(C)CCCNC(c1nnn(C)n1)=O)(C1=CCCC1)OCC 20604,C(=O)(C1=C(C#N)CCC1)N1CC(CC(=O)NC2CC(O)C(O)C2)(OC)C1 20605,C1(N(C(C2(CC)COC2)=O)C)CCCC(NC(c2cc(CC(C)(C)C)on2)=O)C1 20606,Cc1cc(NC(c2ncc(Cc3cccc(F)c3)s2)=O)n2ncc(Br)c2n1 20607,C1(C(=O)NCCc2ncn(CC)c2)CC(N=[N+]=[N-])CN1C(=O)C(C)SC 20608,C(C(CCNC(C1(NC(=O)Cc2ccsn2)CC(O)C1)=O)OC)OC 20609,c1(C(N2CCC(CNC(c3c(OC)nccc3)=O)C2)=O)cc2cccc(C)c2s1 20610,c1(CNC(CC2OCCN(C(C(C=C)C)=O)C2)=O)ccc(C#N)cn1 20611,C1(C(N(C2CCN(C(c3cccn3C)=O)C2)CC)=O)CC(=O)N(O)C1 20612,c1(C(=O)NC2C(NC(c3c(Cl)cn(CCC)n3)=O)CC2)c[nH]c2cnccc12 20613,c1(C(N2CC3CCN(Cc4ncc(C)c(Br)c4)C3C2)=O)cccc2ccncc12 20614,N1(C(c2ccsc2Cl)=O)CC2CC(C1)N2C(C1(Br)CC1)=O 20615,n1(CC)cnc2c(N3CC4CC4(CC)C3)nc(N3CCC(CF)CC3)nc12 20616,CCC(C(=O)OC)C(=O)NC(CC1CCC1)C(=O)NCC1CC1C(=O)OC 20617,C1(CNC(COCCCC(C)C)=O)CN(c2ccn3nccc3n2)CCC1(C)C 20618,Cc1ccc(C(F)(F)F)cc1C(=O)NC1(C(F)F)CCCC1 20619,c1(OC)ccccc1C(F)(F)C(=O)NCC1CCN1C(c1nc(Cl)c(Cl)s1)=O 20620,C(=O)(C=C1SCC(=O)N1C)N(C(C(=O)OC)Cc1ccsc1)C1CC1 20621,CC1CC(CO)N1C(=O)C(C1(C)CC1)NC(=O)C(=O)C1CCCC1 20622,S(=O)(=O)(c1cccc(O)c1)N1CCC(OCC)CC1.N12CCOCC1C1(CC1)C2=O 20623,C(C(C)S(C)(=O)=O)NC(C(C1CCC1)NC(C1C(=C)C1)=O)=O.C(C)(=O)O 20624,c1(C(C(C)NC(=O)NC(c2cccs2)C)OC)cc(Cl)cc(Cl)c1 20625,Cc1cc(C(=O)NC(C2CCN(C(=O)C(F)OC(F)(F)F)CC2)C)cc(=O)n1C 20626,N1(C(C2C(C)CCCC2)=O)CCC12CN(C(c1nc[nH]n1)=O)C2 20627,C1(C(=O)NCC2(COC)N(C(C(CCCC)C)=O)CCC2)CCc2c[nH]nc2C1 20628,c1(C(N2C(C)(CCC(=O)NC(c3cnc(C)s3)C)CCC2)=O)cc2n(n1)CCO2 20629,CN1CCC2(C(=O)O)CN(CC(N3CCN(c4ccncc4Cl)CC3)=O)CC2C1 20630,c1(C(N2CCN(C(CC=C=C)=O)CC2c2cccnc2)=O)cncc2sccc12 20631,N1(C(c2c(C)cccc2)=O)CC2(CC(CNC(=O)CC3(N(C)C)COC3)C2)C1 20632,O=C1CCc2cc(C(N3CC(F)CC3CNC(=O)CC3CC3C3CC3)=O)ccc21 20633,CC1CN(C(=O)CNS(N)(=O)=O)CC1(C)C(N1CCC(C)C1(C)C)=O 20634,CC(C)(C)CC(O)C(=O)NCC1(C(=O)NCC(N)=O)CC12CCC2 20635,CC(CC(F)F)C(=O)NCC1(NC(=O)Cc2cc(F)cc(F)c2)CCOC1 20636,n1(CC)cccc1C(c1nnnn1CC1CCCO1)NCCn1ncnn1 20637,C(=O)(C(C)(O)C1CC1)NCCC(C)NC(C1(C2CC2)CC1)=O 20638,N1(C(=O)Cn2cnnc2O)CCN(C(C2CCC23CCOCC3)=O)C2(CCC2)C1 20639,c1(C(N2C(C)CC(NC(=O)C=C3CCN(C)CC3)C2)=O)cc(C(F)F)cc(F)c1 20640,N1(C(C(COC)O)=O)CCN(C(=O)COCc2cccc(C)c2)CC1CCO 20641,c1(CC)onc(C)c1C(=O)NCCC1CC(NC(=O)C(c2cccnc2)C)C1 20642,Cc1c[nH]c2ncc(C(N3CC4CCC3CN4C(=O)CCCC(C)(F)F)=O)cc12 20643,CC(C)CCC(=O)C(=O)NCC1(C)CCCN(C(C2CCCN(C)C2)=O)C1 20644,N1(C(CC(C)n2cc(Br)cn2)=O)CCCN(C(=O)C=CC2CCCO2)CC1 20645,CC(C)CC(C)(C(N)=O)NC(=O)CCCCNC(=O)C(c1ccccc1)C 20646,CC1CC(NC(C2CC2(C)C)=O)CN(C(c2nccc(Cl)c2F)=O)C1 20647,N1(C(C=CC(CC)C)=O)CC2(CC)CC1(CNC(c1ccncc1N)=O)C2.C1CC1 20648,C(CC(CC)C(=O)NCCCCC1CCN(C(C2CCOCC2)=O)CC1)=CC 20649,c1(C(N2C(C)CCC(CC(=O)NCCN(CC)CC)C2)=O)cc2ccncc2[nH]1 20650,CC1CN(C(c2snc(Cl)c2Cl)=O)CC2(CCN(C(=O)CCc3nccs3)C2)O1 20651,c1(CC(C)NC(c2c(CC)csc2)=O)ccc(CNC(=O)C(CC)N(C)C)cc1 20652,C1(NC(CN(CCOC)C(C2CCC(F)(F)C2)=O)=O)CCCC(F)C1 20653,C12(C(=O)NCCCN(C(C)C)Cc3nc(C(C)C)sc3)CCC(C1)C(C)O2 20654,c1(C(N2CC=CC(NC(c3cc(OC)ncc3)=O)C2)=O)ccc(C)c2c1CCC2 20655,c1(CCOC)nc(=NC2CN(C(=O)C(F)(F)C3CC3)CC23CCC3)s[nH]1 20656,C1(CC)CN(C(c2ccc(OC(C)=O)s2)=O)CCN1C(=O)C(F)=C(C)C1CC1 20657,C1(NC(C2CN(C(C)C)C2)=O)COCCN(C(=O)CCCn2cccc2)C1 20658,O=C(CS(=O)(=O)CCO)NC1CCN(C(=O)Cc2ccc3c(c2)CCC3)C1 20659,CCCC(C)CCCC(=O)NC(C1CCN(C(=O)CC(C)C)C1)(C)C 20660,N1(C(COCCCOC)=O)CCC(O)(C2(NC(=O)C(C3CC3)SC)CC2)CC1 20661,N1(C(c2c(C)nc(CC(C)C)o2)=O)CCCC(O)(CNC(c2ncoc2C)=O)C1 20662,C1(NC(C(C)O)=O)CCC2(CC1)CN(C(c1ccc(Br)c(Cl)c1)=O)CCO2 20663,C1(Cl)(C(=O)NC2C3CN(C(C4C(C)(C)COC4)=O)C2C3)CC12CCOCC2 20664,c1(CC(=O)NCCC(C)NC(c2cnc(CCC)s2)=O)csc2ccccc12 20665,C12(C(N)=O)CC(CNC3CCS(=O)(=O)N3)(C1)OC21CN(c2nnc(O)s2)C1 20666,C1(O)(CNC(c2c(OCC)cccc2)C)CCc2ccccc2C1 20667,C(N=c1cc(F)nc[nH]1)C1CCC(NC(=O)CC2CCC(C(F)(F)F)O2)CC1 20668,C12(NC(C3CCC(CN(C)C)C3)=O)CCC(CC1n1cc(CO)nn1)C2 20669,Cc1cn2c(n1)C(C)CC(C(=O)NC1CC(F)CN(C(c3cnco3)=O)C1)C2 20670,n1(CC)cc(CC(=O)NCC(C)(C2CCC2)NC(c2cc(C)on2)=O)c(C)n1 20671,NC12CCCC1CN(C(c1c[nH]nc1OCc1ccccc1)=O)C2 20672,C(=O)(CCC(CF)CF)N1CCC(NC(c2c(C(C)C)ncnc2)=O)C(C)C1 20673,CC(F)(F)C(F)C(=O)NC(C(=O)NCCC1=CCOCC1)c1ccco1 20674,Cc1cc(C(N2CC(F)(C(N3CCC(O)C3C)=O)C2)=O)c(C)n1C 20675,c1(COC)csc(C(=O)NC2CCC(N(C(=O)C=Cc3cncs3)C)C2)c1 20676,C#Cc1cc(COC(C2CC2C2CCCC2)=O)ccc1Cl 20677,n1(CC(=O)NC2CCN(C(c3noc(CC)c3C)=O)C2)c(C)cc(O)cc1=O 20678,C(N=c1nc2c(ncn2C)c(NCc2cn(C)nc2C)[nH]1)C1(S(CC)(=O)=O)CC1 20679,c1(C(N(CC(=O)NCCC(CC)O)C)=O)cnnc(C)c1 20680,CC1=C(C(=O)NC(C2(O)CCN(C(C3(F)C(C)(C)C3(C)C)=O)CC2)C)SCCO1 20681,N1(C(=O)Nc2c(C(C)=O)cccc2)CC(C)N(C(c2ccccc2)=O)C(C)C1C 20682,C1(C(=O)NC(CC)(CC)c2nn[nH]n2)CCc2ccc(F)cc2C1 20683,C#CCCCC(=O)NCC1(C(N2CCC(CCCC=C)C2)=O)CCCO1 20684,c1(CCC(=O)NCC2(CC)CC(NC(C3(C#C)CC3)=O)C2)ccc(F)cc1 20685,C1(NCc2cccc(Cl)c2)CCCC12CCCO2 20686,Cn1nc([N+](=O)[O-])c(Cl)c1C(=O)NCC1C=CCN1C(=O)CCC1CCC(=O)N1 20687,c1(NC(C)=O)cc(C(N2CC(CO)(CNC(=O)C(C#N)C3CC3)C2)=O)ccc1C 20688,c1(C(=O)NCC2C3CN(C(C4N(C)CCCC4)=O)C2C3)ccc2cnoc2c1 20689,C#Cc1ccc(C(N2CC=CC2CNC(c2ccc[n+]([O-])c2)=O)=O)c(C)c1 20690,CC1(C(N2CCN(CC(=O)NCC3(C)CC3(C)C)CC2)=O)CCCCCC1 20691,c1(SCC)cnc(O)c(C(=O)NCC(CNC(C2CN(C)CCO2)=O)CO)c1 20692,N1(C(CC2C(CN(C=O)Cc3ncc(F)cn3)CCC2)=O)CC(F)(F)C1C1CC1 20693,C1(CC(=O)NC2C3(CC(OCC)C3)C2)CC2(C1)CN(C(=O)CC1CC3CC3C1)C2 20694,c1(NCC2CC(=C)C2)cc(N(C)CC2(CCCOC)CC2)nc(COC)n1 20695,c1(C(N2C(CC(N3CCC(C)(O)C3)=O)CCC2)=O)ccc(Cl)cc1F 20696,C12(C(N3C(C)CC(CNC(c4c(CC)noc4)=O)C3)=O)CCC(CC1)C2(C)C 20697,c1(NCCS(C)=O)[nH]c(=NC2CC3OCCCC23)nc2c1cnn2C 20698,C(=O)(C(C#N)C(C)(C)C)N1CCC(NC(c2c(C)ccc(CC)c2)=O)C1C 20699,C(CCSC)(CN=c1cccc(S(=O)(=O)N(C)c2nc3ccccc3s2)[nH]1)OC 20700,Cc1c(C(=O)NC2CC(N(C(=O)CCC3CCCC(O)C3)C)C2)nnn1C(C)C 20701,N1(C(C(C)S(N)(=O)=O)=O)CCCC(C2CN(C(C3(c4ccncc4)CC3)=O)C2)C1 20702,C(=O)(CC(C)C(C)(C)NC(c1sccc1F)=O)N(CCn1c(C)ncc1)C 20703,N1(C(CC2C(=O)OCC2)=O)CCCOC(CNC(=O)CC2CCCOCC2)C1 20704,CC1OC2CCC1(C(=O)NC1CCCC(CC(=O)NCC3NC(=O)NC3=O)C1)C2 20705,CC(C)CC(=O)NCC1CC1CNC(=O)C(N1CCNC1=O)C 20706,C1(C(N(CC(C)C)CCc2c(C)ocn2)=O)CCN(CCSc2ccco2)CC1 20707,c1(C(C)=O)ccc2oc(NC(=O)C=Cc3cncc(F)c3)nc2c1 20708,N1(C(C)C)CCCC(NC(=O)C(C)N(C(=O)C(C)(C)CF)C2CC2)C1 20709,Cn1nc2ccccc2c1C(=O)NCCN(C(c1c[nH]c(=O)cn1)=O)C1CC1 20710,N1(C(C(C(=O)OC)C)=O)CC2(CCC(C(=O)Nc3nc(-c4cccnc4)cs3)O2)C1 20711,CC(C)CC(C)C(=O)NCC=C1CCN(C(C2(C#N)CCC2)=O)CC1 20712,C1(NC(c2c(C)nc(CNC(=O)CCN=[N+]=[N-])o2)=O)CC(F)(F)C1(C)C 20713,N1(C(C(c2ccccc2F)OC)=O)CCC(CNC(=O)CCCC(N)=O)C1(C)C 20714,c1(CC)ncc(C(=O)NC2CCCCC2NC(=O)C(n2nccc2C)C)cn1 20715,N1(C(c2cc(C)n(CC)c2C)=O)CCCC2(NC(=O)C(C)CC(N)=O)CC2C1 20716,N1(C(CC2CCC(C)O2)=O)CCC2(CCN(C(c3coc(C(F)F)n3)=O)CC2)C1 20717,CC1CN(C(C2CC3(CCC3=O)C2)=O)CCC1NC(=O)C=C(Cl)Cl 20718,N1(C(Cn2ccc(C)n2)=O)CCC(O)(C(C)NC(c2ccnc(O)c2)=O)C1 20719,c1(NCC(CCCC)NC(=O)CC(C)CN(C)C)cc(C)nc(OC)n1 20720,C(=O)(CCC(C)(C)C)NC1C(CNC(CCc2n(C)cnc2)=O)CC1 20721,Cc1ccc(N(C(=O)CN(C)CCO)Cc2cccnc2)cc1F 20722,c1(CC(=O)NCCCNC(CC(C)(C)SC)=O)noc2ccc(Br)cc12 20723,C1(NC(CSSC)=O)CCCCC12CCN(C(=O)C(=O)N(C)C)C2 20724,Cn1cccc(C(=O)Nc2ncnc(Cl)c2F)c1=O 20725,CC(Cc1cnn(C)c1)C(=O)N(CCCCNC(=O)C(C)Cc1ccncc1)C 20726,C1(CC(=O)NC(CC)C(C)C)CN(C(c2c(C)noc2N)=O)CCO1 20727,C1(C(N2CC3N(C(CC4CC(=C)C4)=O)CC(C3)C2)=O)COc2ccc(F)cc2C1 20728,C#CCC(C)(CC)C(=O)N1CCCC(N(C)C(c2nccc(Br)c2C)=O)C1 20729,N1(CC(=O)NC(C2CCCC2C(=O)OC)C)CC2C(CNC(=O)C3CC3)C2C1 20730,N1(C(c2c(C(C)C)c[nH]n2)=O)CC2CCC1C(CNC(=O)C1=C(Cl)CCCC1)C2 20731,c1(NC(C2N(C(C3(OC)CCSC3)=O)CCCC2)C)c(C)c(C)nc2ncnn12 20732,Cc1cc(C)c(NC(=O)Cn2cc(CN(C(C)C)C3CC3)nn2)cc1Cl 20733,N1(C(C2(CC=C)CC2)=O)CC2CCC1CN2C(C12CCCC1CCC2)=O 20734,N1(C(c2cc(C)oc2)=O)CC2(CCCN(C(c3ccnc(Cl)c3N)=O)C2)C1 20735,C(=O)(C(C)CC(F)F)NCC(C)NC(c1ccc(C2(C(F)(F)F)CC2)cc1)=O 20736,c1(C(=O)NCCn2cncn2)cn(CCNC(C2CC2C(F)(F)F)=O)cn1 20737,c1(C(N2CC(CCOC)N(C(=O)C3=CCCS3)CC2)=O)cnc2[nH]ccc2n1 20738,C1(CC)CN(C(c2ccsn2)=O)CCC1NC(c1nc(CC)sc1N)=O 20739,CC(C)CC(C(=O)N(C)CC1CCCC1NC(=O)Cc1cnnn1C)C(C)C 20740,C1(C(N2C(C(N(C)CC3C(C)C3)=O)CC2)=O)CCCCNC1=O 20741,CCC(C)C(C(=O)NCCC1CN(C(c2sccc2SC)=O)C1)OC 20742,c1(C2CCC(NC(=NC)NCCc3ccn(C(C)C)n3)C2)ccc(F)c(F)c1 20743,C1(C(N(C)CC2N(C(C3CN(C(C)=O)C3)=O)CCOC2)=O)CCn2nncc2C1 20744,CCC(C)(Cc1nc2ccccc2s1)CC(=O)Nc1ccc(CC(=O)OC)cc1 20745,c1(CCC(=O)N(CC(C)NC(C(F)CCOC)=O)C)ccc(OCC(C)C)cc1 20746,C12CCN(C1)C2=O.C1(CNC(=O)CCNC(C2CCCO2)=O)CC(Cl)(Cl)C1 20747,N1(C(C2N(C)CCN(C(c3scc(C)c3)=O)C2)=O)CCN2C(=O)OCC2C1 20748,CCC(CC(=O)NC1CC(CO)N(C(=O)Cc2cccc(C)c2F)C1)C(C)C 20749,C1(C)(C(=O)NCc2cc(COC)on2)CCN(C(C2CC(=O)CS2)=O)C1 20750,C1(CC=C)(NC(=O)COCCCC)CCCN(C(C2CCC(F)C2)=O)C1 20751,C1(C(=O)NCC=CCNC(C(COC)NC(C)=O)=O)CCN(CC(F)(F)F)C1=O 20752,N1(C(=O)OC(C)(C)C)CCCC12CCNC2.c1(CN2CC2(C)C2CC2)ccccc1 20753,Cc1cc(F)ccc1-c1noc(C23CCC(C(F)(F)F)(CC2)C3)n1 20754,c1(C(=O)NC(C2CN(C(C3(F)CCCC3)=O)C2)C)ccc2c(c1)NC(=O)CN2C 20755,C1(C(=O)OCC)CCC2CCC1N2C(=O)NC1CCN(CC)CC1C 20756,Cc1n[nH]c(C)c1C1CCCN1C(c1cccc(C(=O)O)c1)=O 20757,N1(C(c2ccc(C)nc2)=O)CCC2CN(C(=O)CN3CCCC3C)C2C1 20758,Cc1ccc(C=CC(=O)N(CCC(C)NC(=O)CCc2cccnc2C)C)nc1 20759,Cc1cc(C2(C(=O)NC3CC3CNC(c3cc(Cl)ccn3)=O)CCC2)cc(C)c1 20760,c1(C(=O)NC(=O)C2CC2)cc(C(F)(F)F)ccc1O.c12noc(n1)C1CC1C2 20761,C(=O)(C(C)CCC(C)(C)C)N(N(C(CC(CC)NC1(CC(=O)OC)CC1)=O)C)C 20762,c1(OC)cccc(Cl)c1C(=O)NCC1COCCN1C(c1cnncc1C)=O 20763,CCC(C)(F)C(=O)N1CC2CC2(NC(c2ccc(F)cc2)=O)C1 20764,C1(C(=O)NCC2(O)CCN(C(C=CCCC)=O)CC2)C2CCC(C2)C1(C)C 20765,N1(C(C(C(C)C)NC(N)=O)=O)CCC(C)C(NC(=O)CCC23CCC(CC2)C3)C1 20766,c1(C(N2CCC(n3ccc(C(F)(F)F)n3)CC2)C(=O)NC)cc(C)nn1C 20767,C1(C(N2C(CC(=O)NCCC(C)C(F)F)COCC2)=O)CCOC(C)(C)C1 20768,CCCCCC(=O)NCCOCCNC(=O)CCNC(C1CCOCC1)=O 20769,c1(C(N(C2CCN(C)CC2)CCCOC)=O)cccc(O)c1F 20770,C(CCC[Si](C)(C)C)N(C(Cn1cncn1)C(=O)O)C 20771,C1(C(=O)NCCCCC2N(C(C3CCC4CC4C3)=O)CCC2)C2CC3C(C2=O)C13 20772,c1(OC)nccc(C(=O)N(CC(O)CN(C(=O)CC2CC3CCC2C3)C)C)n1 20773,CCCC(O)(CCC)CC(=O)N(CCNC(C1CCCC1)=O)Cc1ccccc1 20774,c1(C(=O)NCC2C(C)CCN(C(c3cccc(C)c3)=O)C2)cnn2c1NCCC2 20775,c1(CNC(C2CN(C(C)=O)C2)=O)nc2c(s1)CCN(C(=O)CC1COC(=O)C1)C2 20776,c1(C(=O)NCC2C3CN(C(C(CC=CC)C)=O)CC32)ccc2c(c1)CC(C)(C)C2 20777,CP(C)(=O)c1cccc(C(=O)NCC2CN(C(C3CCNC(=O)C3)=O)CC2O)c1 20778,c1(CN2CCC(C(=O)Nc3c(OC)cccc3O)C2)c[nH]c2ncccc12 20779,C1(NCC(=O)NC2(CCC(N3CC(C)(OCC)C3)=O)CCCC2)CCN(C)C1C 20780,C12(C(N(CC(C3CCC3)OC)C)=O)CCC(CC1)N(C(c1cn[nH]c1)=O)C2 20781,c1(CC(=O)NCC(C)N(C(C(CC)C2CCOCC2)=O)C)ccccc1N 20782,c1(NC(N(C(C)CCc2ccccc2C(F)(F)F)CC)=O)ccc(C(F)(F)F)cc1 20783,n1(CC(=O)NC2CN(C(CCCC(=C)C)=O)C(C)C2)ncn2nccc2c1=O 20784,C1(C(=O)NCC(C2CCCCC2)O)(CNC(c2ccc(Cl)o2)=O)CC12CCC2 20785,N1(C(C(CC)c2cccnc2)=O)CCCN(C(=O)C=Cc2cnccn2)CC1C 20786,c1(C(N2CCN(C(COCC(=C)C)=O)C(CO)C2)=O)ccsc1S(C)(=O)=O 20787,CN1CC(NC(C2CCOCCN2C(c2cn(C3CC3)nn2)=O)=O)C(F)(F)C1 20788,CN=c1[nH]cc(C(N2CCCC(C3CCCCN3C(=O)CSCC(N)=O)C2)=O)o1 20789,c1(C(=O)NC2C(NC(C(C(C)(C)C)SC)=O)CCCCC2)nc2ncccn2n1 20790,c1(C(N(C)CC2(O)CN(C(CSC)=O)C2)=O)ccn(CC(F)(F)F)c(=O)c1 20791,C1(C(CNC(c2c(C)nsc2)=O)O)CCN(C(=O)C(C)C2CCOC2)CC1 20792,C(CCCCC(=O)NC(CCC1CCC1)C(=O)NCc1cccc(C)c1O)OC 20793,c1(OC)ccc(Cn2cc(CNCCn3ccnc3C)nn2)cc1[N+](=O)[O-] 20794,N1(C(CC=CC)=O)CCC(NC(C2CCCC(NC(=O)OC(C)(C)C)C2)=O)CC1 20795,C=C=CCCC(=O)NCCCN(C(=O)CC1(N(C)C)COC1)C 20796,c1(N2CCC(CCOC)C2)nc(C)cc(=NCc2ccc(O)nc2)[nH]1 20797,C#CC1CCCN(C(=O)C(C2CC2)NC(=O)CC2CCCN(C)C2)CC1 20798,C12(C(=O)NC3(CNC(C(C)(C)C)=O)CCCC3)CCCCC1C2 20799,N1(C(C=CCNC(C2CCCC(CF)C2)=O)=O)CCC(O)(CO)CC1 20800,Cc1cc(Cl)c(C(=O)NCC2CN(C(c3cc4occc4[nH]3)=O)CCO2)cc1N 20801,N1(CC)CCOC(CNC(C2CCCN2C(=O)C(C)C2CCCC2)=O)C1 20802,C(=O)(C(C(C)C)n1cnnc1)N(C1CC1)CC1N(C(C(COC)OC)=O)CCC1 20803,N1(C(C(=O)NC2CCC(SCC(=O)OC(C)(C)C)CC2)=O)CCc2ccccc21 20804,N1(c2nc(C)cc(CC)n2)CC(C2CCCN(C(c3ccsc3OC)=O)C2)C1 20805,N1(C(C2C(C)CC2)=O)Cc2ccccc2C(NC(c2cc(C(N)=O)n(C)n2)=O)C1 20806,C1(NC(c2ccc(C)o2)=O)CC(O)CN(C(C2(C)C(C)(C)C2(C)C)=O)C1 20807,c1(CC)[nH]ccc1C(=O)NC(C1CC=CCC1)C(=O)NCCc1ccco1 20808,c1(CCC(=O)NCCC2(NC(C3CC(=C)C3)=O)CC2)cccc(F)c1 20809,N1(C(C2(COC)COC2)=O)CC(n2cc(CNc3nccs3)nn2)C(O)C1 20810,c1(OC)ccc(NC(=O)CCn2cncn2)cc1.C1C(=O)N1CC(O)C1CCC1 20811,CC1CCN(CC(=O)N(C)CCNC(=O)COC2CCCCCC2)CC1 20812,c1(C(C2CC2)OC)nc(-c2nc(Cl)oc2C)n(C(c2ccccc2)C)n1 20813,C1(NC(C=COCC)=O)COC2(CCN(C(c3cc(C)c4n[nH]cc4c3)=O)C2)C1 20814,N1(C(C(C)=C2CC2)=O)CCC(CO)(CNC(C2CCC2(F)F)=O)C1 20815,c1(C(=O)NCC(=C)CCNC(=O)CC(C)(C)O)ccc([N+](=O)[O-])cc1C 20816,Cn1cc(C(=O)NCC2CCC2NC(c2ccccc2C(N)=O)=O)ccc1=O 20817,c1(C(N2CC(CNC(c3c(C)con3)=O)C3(C2)CC3)=O)cc2c(C)cccc2o1 20818,C1(C(N(CCC(=O)N2CC(N3CC(F)C3)C2)CC)=O)C2CCC(=O)C12 20819,N1(C(=O)COC(F)F)CCC2CN(C(c3ccc(Cl)nc3)=O)CC2C1 20820,C1(CNC(C(C)OCCN(C)C)=O)CCCN(C(=O)CN2CCS(=O)CC2)CC1 20821,N1(C(COCCC=C)=O)CC2(C1)SCCC2NC(=O)Cc1cccc(Cl)c1OC 20822,C1(CC(=O)N(CC(=O)OC)CC)CN(C(=O)CCCN(C)C(C)C)CC1C 20823,C1(C#N)(C(=O)NC23CCC(CNC(CC(CC)CC)=O)(OC2)C3)CC12CCCC2 20824,C(=O)(CC(C)(C)C)NCCc1c(CNC(C(C)C2CC2)=O)nco1 20825,C(C(C)(C)C)N(CC(=O)NCCCN(C(C1C(C(N2CCCC2)=O)C1)=O)C)C 20826,C(=O)(C(C)(C)CC(C)(C)C)N1CC2C(NC(CCNC(=O)NC)=O)C(C2)C1 20827,c1(CC)ccc(C(=O)NC2CC(C)N(C(=O)Cn3ncc(Br)n3)C2)c(N)c1 20828,c1(C(C)NC(c2nc(O)nc(O)c2F)=O)cccc(C2=Cc3ccccc3C2)c1 20829,c1(OCC)c(C(=O)NCCN(C)C(C2(C)CC(O)CN2C)=O)cccc1F 20830,c1(OC)cccnc1C(=O)NCC1COCC1NC(=O)C=Cc1ccc(C)o1 20831,c1(OC)ccc2c(c1)C(C(=O)NCC=CCNC(=O)CC1CCC(C)C1(C)C)CC2 20832,c1(Cn2cc(NC(CC(N3CCC(C)C3)=O)=O)nn2)ccc(N)cc1 20833,c1(C(N2CCCC(CN(C(C(C(C)C)F)=O)C)C2)=O)cccc2nc(O)ccc12 20834,CP(C)(=O)c1cncc(C(=O)NC2CCCC(F)(F)CC2)c1 20835,CN1CCC(CC(=O)NC2CC(NC(c3conc3C3CCCO3)=O)C2)CC1 20836,C1(NC(C=CC(=O)OCC)C)CCCC2(CCC2)C1 20837,CC(F)(F)C(F)C(=O)N1CCC(C(=O)NCc2cccc(CO)n2)(CF)C1 20838,CCC(C)(CCNC(=NCCF)NC1CC(c2cccc(C#N)c2)C1)C(N)=O 20839,c1(NC)ccc(CNCCN2CCN(CCCC#N)CC2)cc1 20840,c1(C(N(C(CCNC(c2c(C)ccn2C)=O)C)C)=O)ccc2[nH]ccc2n1 20841,c1(CC)noc(CC)c1CC(N1CC(CNC(C2(C)CC3CC3C2)=O)C(C)C1)=O 20842,C1(OC)CCC(C(=O)N(C)CCN(C(=O)CCCNC(=O)C(C)(C)C)C)C1 20843,C1(O)(C(C(=O)Nc2ncn(CC)c2)O)CCOCC1 20844,c1(CC)ccccc1C(=O)N(C(C)C(=O)NCC1CC(C)(C)CO1)C 20845,C1(C(N(CCC(=O)N2CC(N3CCCC3)C2)CC#C)=O)CNC(=O)CC1C 20846,c1(C(N(C2CCN(C(c3ccc(OC(C)C)cn3)=O)C2)C)=O)cc(Cl)ccc1N 20847,c1(CC(N2CC(NC(C(CCC)C)=O)C3(C2)CCC3)=O)cn2cc(F)ccc2n1 20848,C1(CNC(C(CC)O)=O)CN(C(c2cnn(CCO)c2)=O)CCCO1 20849,N1(C(C2CN(C(C)C)C2)=O)CCC(CCNC(C2CCSC2)=O)CC1 20850,c1(C(=O)NC(C2CCN(C(C3COC3)=O)CC2)C)ccc2c(F)cc(F)cc2n1 20851,C(=O)(C(Cc1ccccc1)N(C)C)NCC(C)CN(C(=O)CC1COC(=O)C1)C 20852,c1(C(N2CC(CC(C)NC(C3CC(=O)N3)=O)C2)=O)coc(C(C)(C)C)n1 20853,C1(CN(C(=O)CC2(O)CCCCC2)CC)CCCCN1C(=O)C#CC1CC1 20854,c1(OC)cccc(OCC(=O)NC(C)C(C)NC(=O)NC2(CF)CCOCC2)c1 20855,CN1CCC(C(C)NCc2nncs2)C1 20856,N1(C(c2cscc2C)C(=O)NCC=C)CCCCC(N(C)C)C1 20857,Nc1c(C(=O)NCC(C2CCCC2)NC(=O)C(c2ccccc2)F)cccc1F 20858,CCC(C#N)C(=O)N1CCC(O)(C(C)NC(C2CCC(C)CC2)=O)C1 20859,N1(C(CN(C(=O)C(SC)SC)CC)=O)CCSCC1C 20860,N1(C(C(=O)NC(c2ccc(C#N)cc2)CF)=O)CC(S(=O)(=O)C2COC2)C1 20861,C1(CC)C(NC(c2cncn2C)=O)CCCN1C(=O)C(=O)NOC 20862,C(C)(C(C(=O)NC1CCCC(CNC(C2CC2c2cccs2)=O)C1)N(C)C)OC 20863,CC#CCCC(=O)NC(C1CCCN(C(C2CN(C)C2)=O)C1)C 20864,C1(NCCc2cccc(OC)c2)CCCCC(O)CNCC1 20865,C1(C(=O)NCC(C)N(C(=O)CCCCc2cnn[nH]2)CC)CCCCN1N=O 20866,C(=O)(C1=CCC2(COC2)OC1)NCC1C(NC(c2c(C)nccn2)=O)CCC1 20867,C(=O)(C1CCc2cccnc21)N1CC(N(C)C(c2ccc(F)cc2C2CC2)=O)C1 20868,C1(C(=O)NCCC(=O)N(C2CCCCCC2)CC)CCCCC1OC 20869,C1(CCNC(c2cnc(C(C)C)o2)=O)CSCCN1C(c1cccn1C)=O 20870,Cc1cc(C(=O)NCCC2CN(C(C3(Br)CC3(F)F)=O)C2)nn1C 20871,Cc1ccc(C=CC(=O)NCC2CCCN2C(=O)C(C)Cn2ccc(C)n2)cc1 20872,N1(C(C(N2CC(F)=C(C)CC2)=O)=O)CCc2c(ccc(C)c2Br)C1 20873,C12(C(=O)NC3C(NC(C4N(S(C)(=O)=O)CCCC4)=O)CC3)CCC(CC1)CO2 20874,C(=O)(C(=O)CCc1ccccc1)NCC(C(C)C)NC(C1N(C(C)=O)CCC1)=O 20875,N1(C(CCOC(C)=O)=O)CC=CC(C(N2CCC(O)C2C(C)(C)C)=O)C1 20876,CC(CCC(=O)N(C)CCN(C)C(N)=O)NC(C1(Cl)CC1(F)F)=O 20877,N1(C(C(C)(C)CO)=O)CCC2(CCC2)C(NC(C2CC(F)(F)C2)=O)C1 20878,C1(C(N2CCC(COC)(NC(=O)CCCF)C2)=O)OC(C)(C)OC1(C)C 20879,c1(C(=O)CN2CCC23CC(Cn2cnnc2)C3)c(Br)cncc1Br 20880,C1(C(=O)NCCN2CCOC2=O)CC2(CC2)CN1C(c1cccc(Cl)c1)=O 20881,c1(C=O)oc(CC2(CNC(C=CC)=O)CCC2)nc1C.C1(C)C(=O)N1.C1CC1.N 20882,c1(C(=O)NC2C(C)N(C(c3cccnc3N)=O)CC2)ccc2c(c1)COC2 20883,c1(N2CC(CC=C)(NC(c3csc(C(F)(F)F)c3)=O)C2)ccc([N+](=O)[O-])cc1Br 20884,C1(OCC(=O)NCCN(CC(C)=O)C(C2(CCC)CC2)=O)CCCCC1C 20885,C1(NC(C2C(C)C2C)=O)CN(C(=O)CCc2cn(C)cn2)C2(CCOCC2)C1 20886,c1(NCCCOC(c2ccc3cnnn3c2)=O)ccc([N+](=O)[O-])cc1Cl 20887,C1(CN(C(C2(C)C(C(=O)OC)C2)=O)C)CCCN1C(=O)CC1(CO)CCCC1 20888,C(=O)(C#CC1CCOCC1)N1C(CNC(C(C)OCCN(C)C)=O)CC(O)C1 20889,CCCCCS(=O)(=O)CC(=O)Nc1cc(N2CC(C)OC(C)C2C)ccc1F 20890,C1(C)(N(C)C)CCN(C(C2(CNC(=O)CC3(O)CCCCC3)CC23CCC3)=O)C1 20891,N1(C(C=C(C)C(F)F)=O)CCC(C(CO)NC(=O)Cc2cc(C)cs2)CC1 20892,N1(C(C(=C(C)C2CC2)F)=O)CC(C)CN(C(=O)CC2CCC(F)(F)CC2)CC1C 20893,C1(NC(C2(C)CC=CCO2)=O)CCC12CN(C(c1cccc(C#N)c1)=O)C2 20894,N1(C(C2C(OC)CC2)=O)CCC2(CC2NC(=O)C(C)COC)C1 20895,CC(C)(O)C(F)C(=O)N1CCC(CC(=O)NC2CC23CC(O)C3)CC1 20896,c1(C(C)(C)C)ccc(C(=O)NCC2CC2CNC(=O)C=Cc2ccccn2)cn1 20897,CC1(C)COCC(C(=O)NCC2(NC(=O)C(O)CN3CCOCC3)CCCC2)O1 20898,c1(OC)nc(C(N2CCN(C)C(c3nc(C)no3)C2)=O)ncc1F 20899,c1(C(=O)NCC(C2CCOC2)NC(c2scc(C(=O)OC)c2)=O)ncccc1F 20900,C1(C(=O)NCC2C(F)(F)CCN(C(C3CC(=C)C3)=O)C2)CCCCN1S(N)(=O)=O 20901,C1(C(N2CC(CC(N)=O)C2)=O)CC2(CC(NC(C3CC4CCC3O4)=O)C2)C1 20902,c1(C(=O)NCC2(C)CCC(OC)CC2)nc2ccccc2n1C1CCCNC1 20903,c1(C(C)C)cccc(F)c1C(=O)NC1CC(O)CN(C(=O)Cn2cncn2)C1 20904,C(C)(CCC(=O)NCc1cccc(C(=O)NC2CCN(C3CC3)C2)n1)OCC 20905,c1(C(N2CC(CNC(c3scc(C)c3C)=O)C3(C2)CC3)=O)snc2ccccc12 20906,Cc1ccc(CC(=O)N(CC(C)NC(=O)C(O)CC2CCCC2)C)c(F)c1 20907,CC1(C)CN(C(=O)Cc2cccnc2Cl)C(CNC(C2(C)CC2C(F)(F)F)=O)CO1 20908,c1(CC)cc(C)c(C(=O)N(C)CCNC(c2cn(C3CCOC3)nn2)=O)o1 20909,c1(C(N2CCC(CC(N3CC(C)C(=O)CC3)=O)CC2)=O)c(F)cccc1C#N 20910,CCCCCC(=O)N1CC(O)CC1C(=O)N(CC(C)(CO)CO)C 20911,c1(OC)ccc(N)c(C(N2CCC3(NC(=O)C(N)=O)CC3C2)=O)c1 20912,Cc1cc(F)cnc1-c1cn(C2CCN2C(c2n[nH]c(O)n2)=O)nn1 20913,C(=O)(CC(C)CC(C)C)NCc1cccc(NC(c2c(OC)n(C)nc2C)=O)c1 20914,c1(CNC(CN(C(=O)C(C)CC2CC2)CC)=O)cncn1C(C)C 20915,c1(C(=O)NCC(CN(C(C2(OC)CCOC2)=O)C)(C)C)ccc(CO)cc1.C(N)=O 20916,C(c1ccccc1NC1CC1)=C(C=C(CC)CN1CC(OC(C)C)CC1CCF)C 20917,O=C1CC(C(=O)NCC2CCCN2C(C2(O)CCSCC2)=O)NC(=O)N1 20918,c1(C(N2CCC(C(C(N3CC(C)(CSC)C3)=O)F)C2)=O)cnc(C)cc1C 20919,C1(CC=C)(C(N2CCC(C(F)F)C2)=O)CCN(C(=O)COC2CCC2)C1 20920,N1(C(C2CCCN(C(=O)C(O)C3CCC3)C2)=O)CCOCCC1C1CC1 20921,Cc1c(Cl)ccc(C(=O)NC(C2CCN(C(c3ccc(=O)oc3)=O)CC2)C)c1N 20922,C1(NC(C(C)SCC)=O)CC(C)(C(=O)NC(C)Cc2cc(C)[nH]n2)C1 20923,c1(C(=O)NC(C(C(=O)NCCOCC(C)C)C)C)cc(F)ccc1F 20924,C1(CNC(CCn2c(C)ccc2C)=O)CC2(CC(NC(C3CCNC3=O)=O)C2)C1 20925,Cn1cc(C(=O)NC2CCCC(NC(=O)Cc3ccccc3)C2)c(O)nc1=O 20926,Cc1cc(C(=O)NC2CCC2CNC(=O)CNS(N)(=O)=O)cc(F)c1 20927,c1(CC(=O)NC(CNC(c2nc(C(C)=O)sc2)=O)C)ccc(C(F)F)cc1 20928,C1(NC(c2cc(SCC)ncc2)=O)CCCN(C(c2c(N)cccc2F)=O)CC1 20929,c1(C(N(CC(CC)NC(c2oc(C)nc2C(F)(F)F)=O)C)=O)cnc(O)cc1C 20930,c1(CC(=O)NCCCC(C)NC(=O)CCCC(=O)N(C)C)nnc2n1CCOC2 20931,c1(-n2ccc(C(N3CC(c4cn(CC(F)(F)F)nn4)C3)=O)n2)ccccc1C 20932,C(=O)(C(C)(C)C(C)O)N1CC(NC(c2ccc(C(C)C)cn2)=O)C(F)C1 20933,C12(CNC(CCC#C)=O)CC(CN1C(=O)CC1CCCCC1)C2 20934,c1(-c2c(OC)cnc(OC)n2)c(C(F)(F)F)cccc1C1CCc2ccccc21 20935,c1(OC)ncc(C)cc1C(N1CC(N(C(=O)CN2CCCC2C)C)C(O)C1)=O 20936,c1(CC(=O)NCCCNC(c2ccc(F)s2)=O)nsc2ccccc12 20937,c1(C(=O)NCC(CC)NC(C2(C)CC2Br)=O)ncc(C)cc1C(F)(F)F 20938,N1(C(c2n(CCC)ccc2)=O)CCC(C)C1CNC(=O)CCOC1CCC1 20939,c1(C(N(C2CCN(C(C34CC(C(F)(F)F)(CO3)C4)=O)C2)C)=O)cnccc1Cl 20940,N1(C(C(C)c2cccs2)=O)CCC2(CC1)CC2NC(n1nnc2ccccc12)=O 20941,C1(C(=O)NCC(C(C)(C)C)NC(c2coc(C(C)(C)C)n2)=O)(CC)CCCCC1 20942,C(=O)(CCCCC1CC1)NCCCN(C(C(C)N(C(C)=O)C)=O)C(C)C 20943,N1(C(CCC#C)=O)CC2CN(C(c3ccc(C#N)c(F)c3)=O)CCC2(CO)C1 20944,n1(CC(N2CCCSCC2)=O)nc(-c2ccccc2)ccc1=O 20945,CC1(C(=O)NC2CCC(NC(c3ccnc(O)c3)=O)C2)CC2CC2C1 20946,C(C(C)(C)CNC(C12CCC1C2)=O)NC(C1(CC=C)CC1)=O 20947,C(c1ccccn1)=CC(=O)NC1(CC)CN(C(=O)C(C)=C2CC2)C1 20948,c1(C(N2CCCN(C(C(C(C)O)(F)F)=O)CC2)=O)nccc2[nH]ccc12 20949,C(=O)(C1=C(C)C(C)(C)OC1=O)NCC12OCC(CNC(Cn3nnc(C)n3)=O)(C1)C2 20950,n1(CC(=O)NC2C3CC(NC(C4(C)CCC4)=O)CC32)cccc(O)c1=O 20951,C1(NC(c2nc(SC)sc2)=O)CCN(C(=O)C(C)OCC(C)C)C12CC2 20952,c1(CNC(=O)CC2COCCN2CCNS(C)(=O)=O)cnc(Cl)c(F)c1 20953,c1(CC)ccc(C(=O)NCC2OCCC2C(=O)NCCC(=O)NC2CC2)cn1 20954,c1(NC(c2c(CO)cn(C(C)C)n2)=O)cccc([N+](=O)[O-])c1Cl 20955,C(CCCC(=O)NCCCN1CCC(NC(=O)CCOC(C)=O)C1)OC 20956,CC1CN2CCN1CC2C(N1CCN(C(c2cc(O)cc(N)c2)=O)C(C)C1)=O 20957,N1(C(c2c(C)scn2)=O)CCC(NC(C2(c3ccc(F)cc3)CC2)=O)CC1 20958,N1(C(c2c(C)occ2)=O)CCN(C(=O)Cc2ccon2)C(c2ccnn2C)C1 20959,C(C)(CCC(=O)N1CCC(C)(CNC(c2cncc(CO)c2)=O)C1)SC 20960,C(=O)(CCCCC(F)(F)F)N1CCC(CNC(C2CCN(CC)C2)=O)C(F)(F)C1 20961,c1(OC)cccc(Cl)c1CC(=O)NC(C)CCNC(c1ccnn1CC#N)=O 20962,N1(C(C(CC=C)(C)C)=O)C2CCC1CC(NC(=O)C=Cc1nc(C)c(C)[nH]1)C2 20963,C1(NC(C2(C(C)(F)F)CCOCC2)=O)COC2(C1)CN(C(C1(Br)CC1)=O)C2 20964,C(=O)(C(CC(F)F)NC(=O)Cn1cc(C#N)cn1)N(CC#C)CC 20965,Cc1cccc([N+](=O)[O-])c1NC(C)CCNC(C1(CF)CCC1)=O 20966,c1(OC)c(C)ccc(C(=O)NCC(CNC(c2cc(C)[nH]n2)=O)OC)c1F 20967,C=CC(C)(CC)C(=O)NC1CN(C(c2coc(OCC)n2)=O)C(C)(C)C1 20968,C(=O)(C(C)CCC(C)(C)C)N1CCCC(CCNC(C(C)c2cccs2)=O)C1 20969,c1(C(=O)NC2C(CNC(c3ccc(C(=O)OC)s3)=O)C2)ncc(F)cn1 20970,c1(C(N(C)CC2N(C(C=C)=O)CCOC2)=O)c(Cl)cncc1Cl 20971,c1(NCC2(O)CCN(C(Cc3cccc(C)c3F)=O)CC2)cc2nncn2cn1 20972,Cc1ccc(CNC(c2ccc(-c3n[nH]c4c3CCC4)cc2)=O)c2ccccc12 20973,c1(N(C)C)ncc(C(N2CCOC(CNC(=O)CC3(C(F)F)CC3)C2)=O)cn1 20974,CC(C(=O)N1CCC(C)(CNC(=O)CCC(C)CN(C)C)CC1)C(F)(F)C(F)F 20975,C(C(C(C)(C)C)NC(=O)CCC(F)F)NC(C(C1CCC(=O)N1)C)=O 20976,N1(C(C(C(C(CC)C)O)C)=O)CCC2(CC1)CCN(C(C13CC(F)(C1)C3)=O)CC2 20977,C1(C(C)Nc2cc(C(F)(F)F)cc(N)c2)CC2(CCCCC2)C1 20978,N1(C(c2cnc(OCC)nc2)=O)CCN(C(c2nc(C)no2)=O)C2(CC2)C1 20979,c1(C(=O)Nc2scc(C)n2)ccc(OC(F)(F)F)cc1 20980,c1(OC)cc(C(N2CCC(F)(C(=O)Nc3cnc(C(C)(C)C)nc3)C2)=O)nn1C 20981,Cc1cc(C(C(=O)NC2CC2)N(CCCc2cnn(CCO)c2)C)on1 20982,C1(CCC(=O)OCC)CCN(C(c2csc(C3CCCNC3)n2)=O)CC1 20983,c1(CC(C)C(=O)NCC2CN(C(=O)CN(C)C)CC2O)ccc(Br)cc1F 20984,N1(C(CC(C)(C)C2CC2)=O)CCC2(CCCCN(C(C3(CF)CC3)=O)C2)C1 20985,C1(C(=O)NC2C(NC(C3(C)CC=CC3)=O)COC2)CCC2(CCOCC2)O1 20986,C1(C(=O)NCC2C(CNC(COCC=C)=O)C2)CCC(C(=O)OC)O1 20987,C1(C)(NC(C2C(C)C2C)=O)CCN(C(=O)CC2CCNC(=O)C2)CC1 20988,C1(NC(C2(CC)COC2)=O)CCC2CN(C(c3cc(C)cnc3F)=O)CC2C1 20989,c1(N(C(C)=O)C)ccccc1C(=O)NCC1CC1NC(=O)CCc1ccon1 20990,C=CCCN=C(NCCc1ncc(C)cc1C)NCC1CN(C(=O)OC)C1 20991,CCCCCCCCC(=O)N1CCN(C)C(CNC(C2C3CCC(F)(F)C23)=O)C1 20992,C1(C(N2CCC(N(C)C)C2)=O)CC2C=CC1N(C(=O)C(C)(C)C(=O)N(C)C)C2 20993,Cc1cc(Cl)c2ccc(C(N3CCC(C(C)NC(=O)CC(C)C)CC3)=O)cc2n1 20994,C(=O)(CCC1CCc2ccccc21)N1CCC(CNC(CCCCC)=O)C1 20995,C(=O)(C1CC(=O)c2c(F)cccc21)N1C2CN(C(C3(C=C)CC3)=O)C(CC2)C1 20996,c1(C(N(CC(C)NC(=O)C(F)n2ccnc2)C)=O)cccnc1N(C)C 20997,C(=O)(CC(C1CC1)NC(=O)CCCn1cncn1)NCCC=CC=C 20998,C=C(C)CCC(=O)N1CCC(N2CCN(C(C3(c4ccncc4)CC3)=O)CC2)C1 20999,CCC(C(=O)NCC1CN(C(c2cnn(C(C)C)c2)=O)C(C)(C)C1)C(C)(F)F 21000,C(CC(C)C(F)(F)F)NC(c1n(CC)nnn1)CCC1OCCO1 21001,C1(NC(=O)C=CCF)CN(C(c2[nH]ccc2C2CC2)=O)CC1CC1CC1 21002,c1(C(C(=O)OC)C2(CS(C)(=O)=O)CC2)ccccc1.C1(=O)CON1C 21003,N1(C(C(C)(C)NS(C)(=O)=O)=O)CCC(NC(C2CCOC2)=O)C1C(C)(C)C 21004,N1(C(Cc2c(C)noc2)=O)CCC(C)(C)C1CNC(c1cc(F)cc(F)c1)=O 21005,c1(N2CCCCC(SC)C2)ccncc1S(=O)(=O)NC(c1cccc(SC)c1)C 21006,c1(CN2C(C(N3CCC(NC(C(CC)SC)=O)CC3)=O)CCC2)cc(F)ccc1C 21007,n1(CONC(C2(CC)CCCCC2)=O)ccc(C(=O)NC2CCCCC2)c1C 21008,CC1(C)CCC(O)(C(=O)NCC(O)CNC(C2CCC=CO2)=O)CC1 21009,N1(C(Cc2c(C)ocn2)=O)CCC2(CC1)CC(C)N(C(=O)CCS(C)(=O)=O)C2 21010,c1(COC)ncc(C(=O)NC(C)(C)C(C)NC(C2C(C)C2C)=O)c(=N)[nH]1 21011,c1(C(=O)NCCN(C)C(c2cc3n(n2)CC(F)C3)=O)nn(C)cc1S(C)(=O)=O 21012,c1(C(=O)OCC)cn(CC(=O)NC(C2CCN(C(=O)C3=CCC3)C2)(C)C)nn1 21013,C1(CNC(C2CC(C(C)(C)C)C2)=O)CCCCCN1C(C1CC12CC2)=O 21014,c1(C(=O)NCCC(C)N(C)C(C2CC(O)C2)=O)c[nH]c2cc(Br)ccc12 21015,c1(NCCC(C)NC(C2CCCC(O)C2)=O)snc(Cl)c1C#N 21016,Cc1nncc(C(N2CC3CCC3(CCNC(c3cnsn3)=O)C2)=O)c1C 21017,c1(C(=O)NCCN(CC(C)O)C(C2CC23CC3)=O)cn2ccnc2s1 21018,C(C)(C)(CCC(=O)N1CCCC(NC(c2nn(C)nc2Br)=O)C1)OC 21019,C#CC1(O)CC(C(=O)NCC2OCCC2C(=O)Nc2ccccc2C)C1 21020,CCCCCC(C(=O)NC1CC1NC(=O)CN1CCCCC1=O)C(C)C 21021,c1(C(C(N2CC(C)C(NC(=O)C3=CCCC3C)C2)=O)=O)ccc(F)cc1F 21022,c1(OC)ccc(F)c(C(N2CCCC(NC(=O)CCCC(C)=O)C2)=O)c1 21023,c1(-n2c(C(C)(CNC(=O)CCBr)NCc3nc(C)on3)nnn2)ccccc1C 21024,c1(C(N(C)CC2(CNC(C3(O)CCOC3)=O)CC2)=O)ccc(C2=CCCC2)cc1 21025,C1(NC(c2c(CC)cno2)=O)CCC2(CC1)CN(c1nc(C3CC3)ns1)C2 21026,N1(C(c2cc(C(F)(F)F)cs2)=O)CC2CCC1CN2C(C1CC1Br)=O 21027,c1(C2(C(N3CC(CNC(CC=CC)=O)C(N(C)C)C3)=O)CC2)ccc(Cl)cc1F 21028,C(CCOCC)(C(=O)NCC(CSCCC)OC)NC(C(C=C)N(C)C)=O 21029,c1(-n2ccc(C)n2)ccc(C(=O)NC2CC(NC(c3[nH]c(O)nc3C)=O)C2)cc1 21030,C1(C(N2CCN(C(C(=O)NCC(F)F)=O)CC2CO)=O)CCc2ccnn2C1 21031,Cc1ccc2c(c1)c(CCNC(c1cc3c(Br)cnn3cn1)=O)cn2C 21032,C(=O)(C1CCc2ccccc21)NC1CC2(CN(C(C3=CCCN(CC)C3)=O)C2)C1 21033,C(CS(=O)(=O)c1ccc(CC)cc1)N(C(C(C=CCCC)O)=O)c1ccccc1 21034,C1(C(=O)NCC#CC)C=CC(NC(=O)CC(=O)OCC)C1 21035,c1(NC(COC(C2C(CCOC)C2)=O)=O)cc(OC)cc(O)c1 21036,FC1CCCCCC1N=c1[nH]c(=NCc2cc(C(N)=O)co2)[nH]c2c1CCC2 21037,N12CCC(C1)C2=O.C(CN(C)C)(C(C)C)NC(CNC(C(C)NC(C)=O)=O)=O 21038,C1(NC(CN(CCOC)C)=O)C(C)CN(C(c2cc(COC)cs2)=O)CC1C 21039,C=CCN=C(NCc1cnn(CC(C)C)c1C)NC(c1ccc(OC)cc1)C 21040,N1(C(C(CC)C2CCOCC2)=O)CCC(NC(c2cnoc2C)=O)C1C(C)(C)C 21041,CC1Cc2cc(CC(N3CCCC(CNC(=O)C=C4CCC4)CC3)=O)ccc2O1 21042,C1(C(=O)NCC2(OC)CCOC2)CC2CCC(C1)N2C(=O)CN1CCCC1 21043,Cc1nn(C)c(C(=O)NC2CC3(C2)CC3NC(=O)C(C)(C)C(=O)N(C)C)c1Br 21044,C1(NC(c2occ(C)c2)=O)CCCCC1NC(C1CCC(C(N)=O)O1)=O 21045,c1(OC)ccc2nc(C(=O)N(CCC#N)CCNC(=O)CN(C)C)ccc2c1 21046,C1(NC(C2CC(C(C)C)C2)=O)COC2(C1)CN(C(c1coc(C(N)=O)c1)=O)C2 21047,N1(C(C2N(C(C)=O)CC(O)C2)=O)CC2(CC(NC(c3cccc(F)c3O)=O)C2)C1 21048,CCCCC(CCCC)NC(C1CC(F)CCN1C(C1CCCC(=O)N1)=O)=O 21049,CC1(C)CCCC1C1CCN(C(=O)C(N2CCCC3CC(O)CCC23)=O)C1 21050,C1(C(=O)NC23CC(CNC(CSCC)=O)(C2)OC3C)CCc2nnnn2C1 21051,c1(C(N2C(CNC(CC(C)O)=O)COCC2)=O)cc(Cl)cnc1Br 21052,c1(OCC)ccc(C(=O)NC(C)(C)CNC(c2nccc(C(F)F)n2)=O)cn1 21053,C1(NC(=O)C(F)C2CCC2)CCCCN(C(c2cnc(C(F)F)cn2)=O)C1 21054,CC1(F)CC(N=c2[nH]c(N3C4CCC3CNC4)nc3c(F)cccc23)C1 21055,C(N=c1nc(N2CC(=O)NC3(CCCC3)C2)c2c([nH]1)CCCC2)C1(C)C(C)(C)C1 21056,C1(C(=O)NC2CC(CC)OCC2)CCN(C(c2cn(C)nn2)=O)C12CC2 21057,c1(CC)nc(=NC(C)C)[nH]c(=Nc2cc(OC)ccc2C)[nH]1 21058,CC1(C)NC(=O)CCC1NC(C1CNC(=O)CN1C(=O)CP(C)(C)=O)=O 21059,c1(OC)cc(F)c(C(=O)NCCC(C)NC(=O)CCC2C(=O)NN=C2C)c(Cl)c1 21060,c1(C(C)C)nc2ccccc2nc1SC1CCN(C)CC1 21061,c1(OC)cc(F)c(Cl)cc1C(N1CCC(NC(C2CN3CCN2C(C)C3)=O)C1)=O 21062,C1(C2CCN(C(=O)C3=CCCSC3)CC2)(NC(C2CCCN2C(=O)C2CC2)=O)CC1 21063,c1(OC)ccc(F)cc1NC(C1CC1C(=O)Nc1ccc(Br)c(F)c1)=O 21064,C#CCC(CC(=O)N(C)CCOC)NC(=O)CCc1cnccn1.C(C)(=O)O 21065,c1(SCCN(C(Cn2c(C)cnc2)=O)C2CC2)ccccc1N(S(C)(=O)=O)C 21066,c1(OCC)cccc(C(=O)NCCC2CCN(C(=O)Cc3conc3C)CC2)c1 21067,c1(C(=O)NC2(COC)CN(C(=O)Cc3ccsc3C)C2)cnc2c[nH]nc2c1 21068,CC(CC(=O)NCC1CN(C(c2ccc(F)c(F)c2)=O)CC1O)P(C)(C)=O 21069,C1(NC(C2CC(O)CN2C(=O)CN2CCC(O)CC2)=O)CCCN(O)C1=O 21070,c1(C(N2CCC(F)(CNC(C3CCC3F)=O)CC2)=O)ccc2c(c1)CNC2=O 21071,N#Cc1ccc(C(N2CCCC2C2CCN(C(c3cnc(Cl)cn3)=O)C2)=O)cn1 21072,N1(C(CN(CC(C)C)C(c2cn[nH]c2)=O)=O)CC(CO)OCC1C 21073,C(CCCCCCCO)=CC(N1C(CCNC(CCCC#C)=O)CSCC1)=O 21074,N1(C(C2CCN(CC#C)CC2)=O)CC(O)C(O)C1CNC(=O)CCCCCO 21075,C1(NC(CNC(CC)=O)=O)CN(C(C2(c3ccc(F)cn3)CC2)=O)CCC1CO 21076,CCC(C)CC(=O)NCCCCN(CCCNC(=O)CCCCC1CC1)C 21077,C(=O)(CC(O)C1CCCC1)NCCOCCN(C)C(c1csc(CC2CC2)n1)=O 21078,CC1CCC(F)(C(=O)NCC2(C)CCCN2C(c2ccc(CCF)cc2)=O)CC1 21079,Cc1cc(OCCCN2CCCC2)ccc1N1CCCC1=O 21080,C=CCC(C)(C)CCO.C(=O)(C(C)(C)Cc1cn(CC=C)nn1)NC1CCOCC1OC 21081,N1(C(C2C(C)(C)C2)=O)CCN(C(=O)COc2ccc(CO)cc2)CC1CCO 21082,C(=O)(C1CCCn2cncc21)NC(CNC(c1sc(C)c(O)n1)=O)C 21083,C(=O)(C(O)CC(C)C)NCC1CCC(NC(CCSCCCC)=O)CC1 21084,S(=O)(=O)(c1cccc(N2CCCC(CCO)CC2)n1)NCC(CC)C(C)C 21085,C1(C(=O)NCC(N(C)C(C2CC(F)C2)=O)C2CC2)CCOC(C)(C)C1 21086,N1(C(CCNC(=O)OC)=O)CCN(C(=O)C=CBr)C(CO)C1 21087,C(=O)(C(C)(C)C(=O)NCC1CC1NC(=O)C1=CCCCO1)N(C)C 21088,C1(C(N2CCC(C(CNC(=O)CCc3cn[nH]c3)F)CC2)=O)CCC(F)(F)CC1 21089,c1(NCC2CCCN(C(C3(CC#C)CCCCO3)=O)C2)cc(C)nc2ncnn12 21090,n1(C(C)C)ncnc1CNC(=O)C=CC(c1cnn(C)c1)=O 21091,N1(C(C2CN(S(CC)(=O)=O)C2)=O)CC2CCCC2(NC(=O)C=C(C)C2CC2)C1 21092,CC1=C(C(=O)NCC2CCCCN2C(=O)CCc2cncnc2)CCO1 21093,CC(C)CCCC(=O)NC1(CF)CCN(C(c2coc3c2CSC3)=O)C1 21094,CC(C(=O)N1CC2CC2(NC(=O)CC(=O)NC2CC2)C1)C(C)(F)F 21095,C(=O)(C(C)(F)F)N(CCN(C(C)=O)CC)CC 21096,C1(CNC(c2[nH]cc(CC)c2)=O)CN(C(c2n[nH]c(CC)n2)=O)CCN1C 21097,C(=O)(CCCCCCS(N)(=O)=O)NC(CNC(C(C)OC(c1cn[nH]c1)C)=O)C 21098,C1(C(N2CC(OC)C(C(N3CCC(N(C)C)C3C)=O)C2)=O)CCC2(CC1)CC2 21099,c1(N(C)C)ccc2nc(CC(=O)NC3CC4CC3N(C(C3CCC3)=O)C4)[nH]c2n1 21100,C#CCC(O)C(=O)NCC1CCCCN1C(=O)CCCSCc1ccc(C)cc1 21101,S(C(F)(F)F)CC(=O)NC1CC(N(C(CNC(C)=O)=O)C)C1 21102,c1(N(CC(C2CC2)C2CC2)C)nc(=N)[nH]c(=NCCCCCCCCO)[nH]1 21103,N(C1CC(C)Sc2ccccc21)C(=O)Nc1cc2nc(C(C)C)oc2cc1 21104,C(CC(N)=O)(C(=O)NC1CC1NC(C1(Br)CC1)=O)NC(CC(C)C)=O 21105,C1(O)(C(CNC(COCC(C)C)=O)C)CCN(C(=O)Cc2nc(=N)[nH][nH]2)C1 21106,c1(C(=O)OC)ncccc1NC(=O)CNc1[nH]c(C)nc1Cl 21107,C1(C(=O)NCCCC)CCCN(C(c2cn(CC)nn2)=O)C1CC 21108,C1(CCCNC(COCCOCC#C)=O)CN(C(=O)Cc2ccno2)CCO1 21109,c1(CC2CCCC2C(N2CC(C#N)(c3nn[nH]n3)C2)=O)nc2ccccc2s1 21110,N1(CC)CCC1C(=O)NCC(C)=CC(=O)NC(c1cnn[nH]1)C 21111,c1(C(CC(=O)NCCCNC(c2cn(CCOC)nn2)=O)C)ccc(F)cc1F 21112,C1(C(N)=O)CN(C(c2csc(C(N)=O)n2)=O)CCC1NC(C1(C)CCC(=O)C1)=O 21113,c1(C(N2CCC(F)(C(=O)OC(C)(C)C)CC2)=O)cc2n(n1)CCCN2 21114,Cn1nc(C2CC2)cc1C(=O)NC(C1CCOC1)CNC(C1CC(O)C1)=O 21115,c1(C(C)NC(COCC)CO)cc(C(=O)OC)c2n1CCOC2 21116,N1(C(CCSCC)=O)CCC(C2CCC2)(CNC(c2cc(=O)n(C)o2)=O)CC1 21117,CC(C)C(C(=O)N(CCCCN1CCCC1)C)NC(=O)C(C)Oc1ccccc1 21118,CN1CCCC(O)(CC(=O)NCCC2(O)CN(C(c3cc(Cl)ncc3O)=O)C2)C1 21119,c1(CC(=O)NC2CC(NC(CC3(C)CC3F)=O)C2)ncncc1Cl 21120,Cc1ccc(F)cc1C(N1CC(C)(C(=O)NC(C)(C(N)=O)C(C)C)C1)=O 21121,CC(C)C(C(=O)NC1(CNC(=O)CSc2cccc(Cl)c2)CC1)c1ccn(C)n1 21122,CC(C)CC(O)C(=O)NC1CCN(C(=O)CN2CCN(C)CC2)C1C(C)(C)C 21123,C1(CNC(c2ccc(C)cc2)=O)CC2COCC2N1C(c1c[nH]c(C)cc1=O)=O 21124,N1(C(C)=O)CCC(NC(=O)C(C(C)C)NC(C2CCCC2)=O)CC1 21125,C1(NC(C(C)NS(C)(=O)=O)=O)C=CCN(C(c2cc(-c3ccoc3)on2)=O)C1 21126,N1(C(C(CC#C)O)=O)CCn2nc(CNC(C3(O)CCCC(C)(C)C3)=O)cc2C1 21127,C1(NC2CC(C(F)(F)F)(OC)C2)CNC2(CCC2)C1 21128,N1(C(C2CCN(C(C)=O)CC2)=O)CC(C)CN(C(=O)COc2ccsn2)CC1C 21129,Cn1c(C(=O)NC2CCCN(C(c3ccc(S(C)(=O)=O)s3)=O)C2)ccc1[N+](=O)[O-] 21130,N1(C(C(C2CCC2)OCC)=O)CCC(C)(CCNC(c2c(Cl)nsc2Cl)=O)C1 21131,C1(NC(c2c(OC)nsc2)=O)CC(C(=O)NC2CCNC(=O)C2)C1(C)C 21132,C1(O)(CNC(C(C=C)(F)F)=O)CCCN(C(C2CCN(S(C)(=O)=O)C2)=O)C1 21133,c1(NC(=O)Nc2ocnc2-c2cn(CC3CCCOC3)nn2)ncc(Br)cc1F 21134,CC1CCCCC1CNC(=O)CN1CCC(NC(=O)CC2CCC(C3CC3)O2)CC1 21135,CC1CCN(C2CCNC2)C(NC(=O)CSc2nnnn2-c2ccccc2)C1 21136,c1(C(=O)NC2(CCNC(c3ncccc3Cl)=O)CC2)c(O)nnc2c1COCC2 21137,C1(C(C)C)(C(=O)NC(C)CNC(C2CCC2n2ccnc2)=O)CCC1 21138,C(CNC(=O)CCCC1(NC(c2ccc(CO)o2)=O)CCC1)(C(F)(F)F)OC 21139,Cc1sc(O)nc1C(=O)N(CC(C)NC(c1cnc(-c2ccsc2)s1)=O)C 21140,c1(C(=O)NC2CC2NC(c2ccc(Br)c(F)n2)=O)cccc([N+](=O)[O-])c1 21141,CCCCCCCC(=O)NCC1(F)CC(NC(=O)CCc2cnco2)C1 21142,C(c1ccncn1)=CC(=O)NCC1CC(NC(C2C3COCC23)=O)C1 21143,N1(Cc2cn[nH]c2)CCN(Cc2ccnc(Cl)c2)CC1.C123CC(C1)(C2)NC3=O 21144,c1(OCC)ncc(C(=O)NCCC(O)CNC(=O)CCC2CCCOC2)s1 21145,N1(C(C(n2c(C)ccn2)C)=O)CCC(CCN(C(=O)Cc2ccsc2)C)CC1 21146,CCS(=O)(=O)CC(=O)NC1CCN(C(=O)CSc2ccc(OC)cc2)CC1C 21147,C1(C(=O)NC2(CO)CN(C(C3(COC)CC3(F)F)=O)C2)Cc2ccccc2S1 21148,c1(C(=O)NCc2ccsc2-n2cnnn2)ncsc1-c1ccccn1 21149,C(=O)(C1CCCc2scnc21)NC1C2N(C(c3ncc(C)cc3F)=O)C(CC2)C1 21150,C(=O)(CC(O)CC(C)C)N1CC(C(NOCC2CC(=C)C2)=O)C(F)(F)C1 21151,N1(C(c2cnc(CC)s2)=O)CCCC(CN(C(=O)CC2CC3CC3C2)CC)C1 21152,CC1(C)NC(=O)OC12CCN(C(=O)C(C1(O)CCCCC1)(C)C)C2 21153,N1(C(c2cncc(C)c2C)=O)CCC2CN(C(=O)C(O)C3CC3)CC12 21154,c1(C(N2C(CNC(C3CCCS3(=O)=O)=O)CC2)=O)ccc2[nH]c(=O)c(=O)[nH]c2c1 21155,C1(NC(C(CCC)N(C)C)=O)CC2CCC1CC2NC(=O)CN(C)CC 21156,N1(C(CCc2ccc(C)o2)=O)CCOCC1CNC(c1ncoc1C(C)C)=O 21157,CCC(CC(=O)N1CCC(NC(=O)Cc2ccon2)C(O)C1)C(C)C 21158,C12(CNC(C(C)OCC)=O)CC(NC(=O)C=Cc3ccncn3)(CO1)C2 21159,N1(C(C2C(C(C)=O)C2)=O)CC(CNC(c2ccc(=O)n(CCO)c2)=O)CC(C)(C)C1 21160,C1(CC(=O)NCC2CC2c2ccc(Cl)cc2)CCN(C(C2(CO)CCC2)=O)CC1 21161,c1(CNC(c2cccc(C(=O)OC)c2)c2nnnn2C)ccn2cnnc2c1 21162,c1(CC)ccc(C=CC(N2CCN(CCNC(C3CCCC3C)=O)CC2)=O)cc1 21163,N1(C(=O)CCCCn2ccnn2)CCCN(C(C2(c3ccc(Cl)cc3)CC2)=O)CC1 21164,C1(CNC(C2C(C)C2C)=O)CN(C(=O)COc2ccc(CO)cc2)C2(CCC2)C1 21165,c1(CC(N2CC(NC(CC(C(=O)OC)C)=O)C(C)(C)C2)=O)ccn2cncc2c1 21166,CN1CCOC2CN(C(=O)C3=CCN(C(C4CCOCC4(C)C)=O)C3)CC12 21167,C=CC1CCC1C(=O)N(C1CN(C(=O)C=CC(CC)=CC)C1)C 21168,c1(C(=O)NCCN(C(c2oc3ccccc3c2Cl)=O)CC)ccc2nncn2c1 21169,Cc1noc(C)c1CSCC(N1CC(NC(c2cc(C3CC3)no2)=O)C(C)C1)=O 21170,c1(NC(C(=O)N(CC(C)(C)S(C)(=O)=O)C)=O)cccc2c1CCOC2 21171,c1(C(C(=O)NC2CCCC2)N(CC(COC)C)C)ccncc1F 21172,N1(C(C(=O)N(CCCCNC(C2(OC(C)C)CCOC2)=O)C)C)CCN(C)CC1 21173,c1(C(C)O)ccc(C(=O)NCC2CCCCN2C(=O)C(F)=CC2CC2)cc1 21174,C(=O)(CCCC(=O)NCC(CO)NC(c1cccc(C2CCC2)c1)=O)N(C)C 21175,N1(C(CCSC)=O)CC2CCC(CNC(=O)C(C)(C)c3ccno3)C2C1 21176,C1(CNC(c2cscn2)=O)CN(C(c2ccc(F)cc2F)=O)C2CCN1C2 21177,Cn1[nH]c(=NC(=O)C(C)(C)c2cnn(C(C)(C)C)c2)cc1C(F)(F)F 21178,C(C(=O)Nn1cccn1)C1CCC(NC(C=CCCC)=O)C1 21179,C1(CCC)(NC(=O)Cc2ccc(OC)c(Cl)c2)CCN(C(=O)C2=COCC2)CC1 21180,c1(CC)n[nH]cc1CNC(=O)C=CC(C)(C)NC(=O)C(F)=C(C)C 21181,C1(O)(CNC(C2CC3C=CC2C3)=O)CCN(C(c2ccn(CC(F)F)n2)=O)CC1 21182,C(CC(C)C(F)(F)F)NC(CC1(OC)CN(C(C2(CC#C)CCCO2)=O)C1)=O 21183,C1(C(=O)NCCC(C)N(C)C(c2cc(O)nc(Cl)c2)=O)CC1C1(C)CCOCC1 21184,C(C(CC(C)C)C(=O)N(C)CC=CC(=O)NCC(C)(O)C1CCCC1)OC 21185,c1(C(=O)NC2CC3(C(NC(c4c(C)onc4)=O)C3)C2)cc2c(o1)CCCC2 21186,C1(NC(=O)NCC(CSC)(C)C)CCC2(CC1)CC2C#N 21187,C1(COC)(CNC(C2CCC2(C)C)=O)CCN(C(c2cc(Cl)nnc2O)=O)CC1 21188,C(CC(F)F)(C(=O)N=c1ccn(C2CC2)[nH]1)NC(c1scc(C(N)=O)c1)=O 21189,c1(C(CNC(CC2(N)CC2)=O)F)cccc(Br)c1 21190,c1(C(=O)NC(CN(C(C2CC(F)C(=O)N2)=O)CC)C)cc(OC)c(O)c(Cl)c1 21191,C1(NC(C2CN(CCOC)C(=O)C2)=O)CN(C(C2(C)CCCCC2)=O)CC12CC2 21192,C1(NC(C2C(NC(C(=O)N(C)C)=O)C2)=O)CCCC1C(C)(C)C 21193,c1(C(=O)NC2COCCN(C(C(COC)(C)C)=O)C2)ccc2ccccc2c1F 21194,Cc1ccnc(C(=O)NC2CCC(C(=O)NCC(c3ccccc3)O)C2)c1 21195,N1(C(C=Cc2ccc(C)s2)=O)C(C)CC2CN(C(=O)C(C)C(O)C(C)C)CC12 21196,C1(c2cccs2)(C(=O)NC2C(CNC(C(C=CC)O)=O)C2)CCCCC1 21197,c1(C(N2CCC3(CC2)CC3)C(=O)NC(CC)C)ccc(C)c2c1CCC2 21198,N1(C(CCC(CC)C)=O)CC2CCC(C(=O)NC(C)CC3CC3)(C2)C1 21199,CS(=O)(=O)C1CN(C(C2(F)CCC2)=O)CC1NC(c1cn2cc[nH]c(=O)c2n1)=O 21200,N1(C(C2C(c3n(C)ncc3)C2)=O)CCC2(CCCO2)CC1 21201,C(=O)(CCC(C)(C)NC(=O)CCCNC(=O)CCOC1COC1)OC 21202,c1(C(COC)NC(C2CC(O)(CO)C2)=O)ccc(F)cc1 21203,c1(SCC)cnccc1C(=O)NCCC(C(C)C)NC(=O)C=CC1CCCN1C 21204,Cc1cc(C)c(CC(=O)NC2C=CCN(C(c3n[nH]cc3C)=O)C2)c(C)c1 21205,C1(NC(CNC(=O)OCC=C)=O)C2CC1CN(C(C1(OC)CCC1)=O)C2 21206,N1(C(c2ccn(C)n2)=O)CC(CNC(=O)COc2ccccc2)C2CC12 21207,N1(C(C=C(CCC)C)=O)CCC(C)(C(=O)NC(c2cnn(C)c2)CO)C1 21208,CC12CC(NC(C3CCC3(C)C)=O)(C1)C1(CCN(c3ncnc(Cl)c3Br)CC1)O2 21209,c1(C(=O)NC(C)CNC(=O)C(F)(F)c2csc(Cl)c2)cnc(N)cn1 21210,N1(C(c2cccc(CCC)c2)=O)CC(C)C(NC(=O)CNS(=O)(=O)NC)C(C)C1 21211,CCC(C)(CCO)NC(=O)CCCn1cc(-c2cnc(C)s2)nn1 21212,C1(O)(CC(=O)NCc2ccc[nH]2)CN(C(c2ccsc2)=O)C1 21213,N1(C(CCC)C(=O)NCCCC(=O)OCC)CC(C)CCC12CC2 21214,C(=O)(C1CCCc2nnn(C)c21)NC(CNC(CCCCC)=O)CC(F)(F)F 21215,CCCCC(O)C(=O)N1CCC(OCCNC(C2(C)CCCN2C)=O)C1 21216,C1(NC(COCCCCC)=O)CCN(C(=O)COCc2cc(C)on2)CC1(C)C 21217,C1(CC)CN(C(C2CC(C)(N)C2)=O)CC(C)S1=O 21218,N1(C(C2C(CC)CCN2C(c2ccnc(C)n2)=O)=O)CCc2ccsc2C1 21219,c1(C(=O)NC2CCN(C(C(CC)NC(N)=O)=O)C2(C)C)ccc2c(n1)CCCN2 21220,C12(C(=O)NC(c3ccc(N4CCOC4=O)cc3)C)CC(C1)C(C(F)(F)F)N2 21221,CCCC(CC)CCC(=O)NC1C(C)(C)C(NC(c2cc(OC)cs2)=O)C1(C)C 21222,Cc1ccc2c(c1)CC(NC(c1occc1-c1ccc(F)c(F)c1)=O)C2 21223,C(=O)(CC(C)CC(F)(F)F)N(C1CCN(C(=O)C=C2CCC2)C1)CC#C 21224,N1(C(C2(C)CCCO2)=O)CCOC2CCN(C(=O)Cn3cnc([N+](=O)[O-])c3)CC12 21225,N1(C(c2c(COCC)nn[nH]2)=O)CC2CC1CN2C(C1CC1OC(C)(C)C)=O 21226,C(C(=O)N1CCC(CO)(NC(=O)CS(C)(=O)=O)C1)(C(C)(C)C)SC 21227,C1(CC(=O)NCCC(=C)CNC(C2CC(=O)N(CC)C2)=O)CCC(C)(C)C1 21228,N1(CC(=O)NCc2c(C)occ2)CC(NC(c2coc(O)n2)=O)CCC1C 21229,N1(C(C(CN(C)C)(C)C)=O)CC2(CCC(CNC(=O)CSCc3cscn3)O2)C1 21230,c1(C(N2C(C(C)NC(CCSCCCC)=O)CCC2)=O)cn(C)nc1OC 21231,C(CC(C)(C)C(=O)N1CCC(C)(CNC(=O)CCC(C)(F)F)C1)SC 21232,c1(C(N2CCN(C(c3ccc(CC)s3)=O)CC2CF)=O)ccc2cccnc2c1 21233,c1(C(N2CC(C)(NC(C3C(SC)CCC3)=O)C2)=O)nn(C)c(C(F)(F)F)c1Cl 21234,C1(NC(=O)Nc2c(C(C)C)csc2)CCCN(c2cnn(C)c2)C1=O 21235,C1(NC(C(F)=C(C)C)=O)CN(C(=O)Cc2cccc(OCC(C)C)c2)CC1C 21236,n1(CC)cc(CC(=O)N(C(C)CN(C(=O)Cc2cnc(C)s2)C)C)cn1 21237,C(C)(C)(CC(=O)NC(CCNC(=O)C1CC1)=O)N(C(CCCOC(C)C)=O)C 21238,C(=O)(CC(C)(C)N(C(=O)CC1CCC=CCC1)C)N(CCCCCO)C 21239,c1(C(N(C(CC(=O)NC(COC)COC)(C)C)C)=O)cnn2c1OCC2 21240,C1(C)(CNC(Cc2nc(CC)sc2)=O)CC(F)(F)CN1C(c1scnc1C)=O 21241,N1(C(C(CC)OC)=O)CCC(C)C(CNC(c2nccc(Cl)c2F)=O)C1 21242,c1(C2(C(=O)NC(CC=C)C3CCC3)CCC2)ccc(F)cn1 21243,C1(OC)CC(CNC(C2CC2c2cnnn2C)=O)N(C(c2nc(C)n(C)n2)=O)C1 21244,C=CC1(NC(C23CC2CCN3C(c2sccc2F)=O)=O)CCCC1 21245,Cc1occc1CC(=O)NC1CCN(C(c2cn(C3CCCC3)nn2)=O)C1 21246,C#Cc1ccc(F)c(C(N2CCC(C)(NC(C3CCC(C)(C)OC3)=O)C2)=O)c1 21247,c1(C(C)NCc2cnc(C)nc2O)ccc(S(C)=O)cc1 21248,N1(C(C(C)Cc2ccccc2)=O)CC2CN(C(c3coc(O)n3)=O)CC2C1 21249,c1(C(N(C2CC(NC(c3ccc(Cl)cn3)=O)C2)C)=O)cnc2[nH]c(O)nc2c1 21250,c1(C(=O)NC(C(C)NC(C2CCCN2C=O)=O)CO)ccc(Cl)c(N)c1Cl 21251,c1(OC)ccc(CNC2CN(C(c3csc(C)c3C)=O)CC2C)c(C#N)c1 21252,C(CCN(C)C)(C(=O)NCc1cn(C)cn1)NC(COCCC)=O 21253,C=CC1CN(C(=O)C(C)(C)n2ccc(C)n2)CC1NC(=O)CC1C(=O)NN=C1C 21254,C(C)(CCCC(=O)N1CC(N2CCNC2=O)C1)NC(c1[nH]cc(C)c1C)=O 21255,C(=O)(C(CC(F)F)NC(c1ccc[n+]([O-])c1)=O)NC(CCC)CCO 21256,CCC(C)C(O)C(C)C(=O)NC1C2CCN(C(=O)C(O)C(C)(C)C)CC12 21257,C1(CNC(CCN(CCC)C)=O)C2CCCC1N(C(c1cccc(O)c1F)=O)C2 21258,C1(CNC(C2CC(O)(N(C)C(=O)OC(C)(C)C)C2)=O)CC2CC(C1)CC(F)(F)C2 21259,CC1CN(C(c2cnn3ccsc23)=O)CCC1NC(C1CN2CCN1CC2)=O 21260,c1(C(=O)NCC(CC=C)NC(=O)CC23CCC(CC2)C3)ccc2[nH]ccc2c1F 21261,c1(C(N2CCCC(C(=O)NC(C)CC#N)C2)=O)ccc(Cl)nc1Cl 21262,C(c1ccc(C(C)(C)C)cc1)=CC(N1C(CNC(CCOCC#C)=O)CCC1)=O 21263,C#CCC(O)C(=O)NC(CCOCC)C(=O)NCCC1CCCCO1 21264,CC1(C)C(C)(NC(=O)C(F)CC2CN(C(=O)C(F)F)C2)C1(C)C 21265,CCC(CCOC)C(=O)NC1(Cc2cccc(C)n2)CC1 21266,Cc1c(NC(=O)CC2CCN(C(=O)Cc3cccnc3)CC2)cnn1C1CC1 21267,c1(C(N2CCC(COC)(NC(c3cncs3)=O)C2)=O)c(C)oc2nc(Cl)ccc12 21268,C(=O)(CC1=CCCC1)NC1CCCN(C(c2c(C)nsc2Br)=O)C1 21269,C1(C)(C(=O)NC2CC3(CC(NC(CNC(C)=O)=O)C3)C2)CCc2ccccc2C1 21270,C1(CNC(c2c(C)nc(CO)o2)=O)C2CCC(C2)N1C(=O)CCn1cccn1 21271,C1(C(=O)NCCC2CC(C)(C)C2)(NC(C(CCOC)C)=O)CCC(C)(C)C1 21272,C1(NC(CC(C)OC)=O)CCC(C)N(C(=O)C(CO)c2ccccc2)C1 21273,c1(C(N(C2CCN(C(Cc3ccc(C)cc3C)=O)C2)C)=O)ccc2sncc2c1 21274,c1(C(=O)OC)ccc(Br)c(NNC(=O)C2Cc3c(F)cccc32)c1 21275,C(O)(CC(=O)NCC1(CC2CC2)CC1)(C(F)(F)F)c1ncc(C)o1 21276,c1(-n2cc(C(C)NC(C3CC3(Br)Br)=O)nn2)cccc(Br)c1 21277,C1(NC(C(CC)C)=O)CC(NC(c2sccc2CO)=O)C(O)C1 21278,N1(C(C2C(C)(C(F)F)C2)=O)CCCCCC(NC(=O)C2=CCCS2)C1 21279,CCCCC(C)CCC(=O)NCCCN(C(=O)CC#N)C1CCCC1 21280,c1(C(CNC(c2cnn(CCC)c2)=O)NC(CCCCC)=O)cc(F)cc(Cl)c1 21281,Cc1cncc(-c2cn(C(C)C(=O)NCc3csc(Br)n3)nn2)n1 21282,N1(CC)CCCCC1C(=O)NCCOc1nnn(C)c1C(N1CCOC(C)C1)=O 21283,CC1CN(c2nnc(-c3sccc3CO)n2Cc2ccc(F)cc2)CCS1 21284,CC(C)(O)C(F)C(=O)N1CCOC(CNC(C2CCCCO2)=O)C1 21285,C(=O)(CC(C)(C)n1cc(C2COCC2O)nn1)N(C(=O)C(C)(F)CC1CCCC1)C 21286,c1(OC)cccc(-c2cc(C(=O)NCC=CCNC(c3sccc3SC)=O)on2)c1 21287,c1(C(=O)NC2CC(C(C(=O)N(CC(O)CO)CC)F)C2)csnc1Cl 21288,C1(NC(C2(COC)CCCNC2)=O)CCC(F)(F)CC1(C)C 21289,S(=O)(=O)(c1cnn(C)c1)N(CC(N1CCC(CNC(C2COCCN2C)=O)C1)=O)C 21290,C1(C(=O)NC2CCC(CC(=O)NC3(C)CC(O)C3)C2)CC2C(C1)C2(C)C 21291,CC1(C)OCc2c1n[nH]c2C(=O)NCC1CC(NC(=O)C(F)CC2CCCC2)C1 21292,c1(C(=O)NC2C(NC(COCCCCC)=O)CCC2)c2ccccc2nn1C 21293,c1(OCC(=O)NC(C)C(CO)NC(=O)CC(C)(C)CC(N)=O)ccc(Cl)nc1 21294,CC(CNC(=O)C=Cc1ccsc1)(CO)NC(C1C(c2cccnc2)C1(C)C)=O 21295,c1(-c2nc(CC(C)CCO)on2)c(Cl)cccc1Cl.C(CCCCCSSC)NC(=O)CO 21296,C(=O)(C1CCOc2ccccc21)NCC(C1CCCN1C(C1C=CCC1)=O)(C)C 21297,C(CC(=O)NC(C)CCCCO)(C(C)C)NC(C1(OCC)CCCC1)=O 21298,c1(C(N2CCC(COC)(NC(C3(C)CCC(=O)N3)=O)C2)=O)ccnc(Cl)c1O 21299,C1(NC(C2(CNC(=O)CC3CCCC3)CCCO2)=O)CCCCCC1F 21300,c1(C(N2CC(C)OCC2C)=O)nc2ccccn2c1C1=CCOCC1 21301,c1(CNC(CSCC#C)=O)cc(C(=O)N(C)CC2(C#N)CC2)no1 21302,c1(C(N2CCN(C(CC=C=C)=O)CC2C)=O)cc(Cl)cc2nc(C)[nH]c12 21303,N1(c2snc(CC)n2)CC(C2CCCCN(C(=O)CC3(C)CCCO3)C2)C1 21304,S(=O)(=O)(c1[nH]c(=NC2CCCC(C(C)(C)C)C2)ccc1Br)NCCCOC(C)C 21305,c1(C(=O)NCC2(CCNC(COC(C)C)=O)CC2)cncc2c(O)nccc12 21306,CCC(CC)CC(F)C(=O)NC(C12CCC(CC1)C2)CNC(=O)C(C)(C)O 21307,N1(CCc2c(C)cccc2Cl)CC2CCCCC12c1ccccc1 21308,C#CCC(O)C(=O)NC(c1ccccc1)CNC(=O)C(O)(C1CC1)C1CC1 21309,N1(C(C(CCC)CC)=O)CCCCCC(NC(=O)CN2CCC(=O)CC2)C1 21310,Cc1cncnc1N1CCC(C(C)(C)NC(=O)Cn2cc(Cl)cn2)CC1 21311,C1(C(=O)NC(CC)C2CCC2)CC(F)CN1C(=O)CC1COCCO1 21312,C1(CNC(C2CC(SC)C2)=O)CC(C)CN(C(c2cn(CCO)nc2C)=O)C1 21313,NS(=O)(=O)C1(C(=O)NCC2(O)CCN(C(C3(n4cnnn4)CC3)=O)CC2)CCC1 21314,Cc1nc2ccc(C(=O)NCC3C4CN(C(c5csc(C)c5)=O)CC34)cc2s1 21315,N1(C(CN(C)C(c2c[nH]c3nccc-3c2)=O)=O)CCC2(CC1)CC2C#N 21316,O=S(=O)(c1ccc(NOCCC(F)(F)F)cc1)Nc1ccc(F)cc1 21317,C1(CC(=O)N(CCOC)CCNC(c2cncc(C(C)(F)F)c2)=O)CCCCC1O 21318,C1(O)(CC=C)CCN(C(=O)C(CCCOC)NC(=O)C(C)NC(=O)NC)CC1 21319,c1(NC(N2CCC(CC(=O)OC)C2)=O)nc2ccccc2n1CC#N 21320,CC1CCC(CNC(c2scc(Cl)c2Cl)=O)N(C(=O)C2=COCCO2)C1 21321,Cn1nc(C(F)(F)F)c(Br)c1CN1CCCCC1C(c1ccccc1)O 21322,C1(NC(CC2(C=C)CC2)=O)CC(=O)N(C2CN(C(=O)Cc3c[nH]ccc3=O)C2)C1 21323,C1(C)(CNC(CCOC)=O)CCC(NC(C2(F)CCCC2)=O)C1 21324,C12CCOC1C(=O)N2.C1(NC(C(C)OCC)=O)CCCC1C(=O)OC 21325,C1(C(N2C(C(=O)NCC3CCOC3)CC=CC2)=O)CC2(C1)CC2(F)F 21326,C1(NC(=O)CCC2CC2)CCC2(CCN(C(c3csc(Cl)c3Cl)=O)CC2)C1 21327,c1(OC)cccc2scc(C(N3CC4C(NC(=O)C(C)N(C)C)C4C3)=O)c12 21328,c1(OC)[nH]c(=N)ccc1C(=O)NCC1CC2CN(C(=O)Cc3nnc(C)o3)CC12 21329,C1(C2CCN(C(C3CCC(F)CC3)=O)CC2)(NC(C(CC)C(C)C)=O)CCC1 21330,C(CNC(=O)C(=O)NCc1nc(C)no1)(C(F)(F)F)NC(CN(CC(=C)C)C)=O 21331,c1(NC(C)=O)ccc(C(N2CCC(O)C(N(C(C)CCO)C)C2)=O)cc1Cl 21332,C1(CNC(=O)NC2(c3ccccc3)CC2)CC2N(C1)C2=O.C1(COC)CCC1 21333,C1(NC(C23C(C(=O)OC)(CCC2)C3)=O)CN(C(=O)C(C)(C)C(N)=O)CCC1F 21334,CC(C(=O)N(CCNC(=O)COc1cn[nH]c1)C(C)C)C(C)(F)F 21335,c1(C(N2C(CNC(=O)C(F)CC3CCC3)CCCC2)=O)cccc(C#CCO)c1 21336,C1(C(N2C3(CNC(C=CCC#N)=O)CCC3CC2)=O)CCC2(CC1)OCCO2 21337,C1(CNC(C=C(CC)CC)=O)(COC)CCCN1C(C1(CCF)CC1)=O 21338,C1(C)(C(N(CC(C)N(C)C(C2CCN(C)S2(=O)=O)=O)C)=O)CCC(F)(F)CC1 21339,C(=O)(CC(=O)N(CC(C)CNC(c1cocc1C)=O)C)OCC 21340,N1(C(C2(NC(CC3C(C)CCC3)=O)CCOCC2)=O)CCN(C)CC(O)C1 21341,N1(C(C(C)(C)C(F)F)=O)CCCC(O)(CNC(C23CCC(C)(CO2)C3)=O)CC1 21342,c1(C(N2CCCCC2C(=O)NCC(F)(F)F)C(=O)NC)cc2cccnc2s1 21343,c12nccc(n1)N2.N1(C(CCC)=O)CCC(C(=O)OC(C)(C)C)C1 21344,O=C(CCCC1(NC(c2ccn(C3CC3)n2)=O)CCC1)NCC(F)(F)Cl 21345,c1(C(N2CC(C)N(C(C3CCCC34CC4)=O)CC2)=O)cc2c(cn1)CCCC2 21346,c1(CNC(C2CCCN(C3CCC3)C2)C)ccc(I)c(F)c1 21347,C1(NC(C(CC)Oc2ccccc2)=O)CN(C(=O)CCC#N)CCC1(C)C 21348,C(=O)(CC(C)(C)CC(F)(F)F)N1CCCC(C(=O)NCc2cc(C)no2)C1 21349,C1(NC(CCCc2cc(C)no2)=O)CCN(C(=O)C(C)SC(F)(F)F)CC1O 21350,C(=O)(C1CCCc2cncn21)NCC1C2CN(C(c3c(C)cc(N)cc3)=O)CC21 21351,c1(C(=O)NC(C2CCN(C(C(C)=C3CC3)=O)CC2)C)ccc2c(C)nn(C)c2n1 21352,c1(-c2cc(C(N3CCC(C)(O)C3)=O)c(Cl)nc2)ccc(S(=O)(=O)NC2CC2)cc1 21353,C1(NC(CC2(C=C)CCC2)=O)CN(C(=O)C#CC(C)C)C(C)(COC)C1 21354,N#CC1CN(C(c2cncs2)=O)CC1NC(c1cccnc1Cl)=O 21355,C1(C(=O)NCC(C2CCC2)NC(CCCNC(C)=O)=O)CCC=CCCC1 21356,Cn1[nH]c(=NC(=O)C2CCCN2C(C2(C(F)(F)F)CCC2)=O)cc1Cl 21357,C1(C(N2CC(C)C(F)C2)=O)N(C(c2cc(C(N)=O)c[nH]2)=O)CC12CCCC2 21358,N1(C(c2c(C)nc(CC)o2)=O)CCOC(C)(CNC(=O)CCOC2CC2)C1 21359,N1(C(Cc2c(C)n[nH]c2)=O)CC2CC(NC(c3nnn(C)c3N)=O)C(C2)C1 21360,N1(C(C(N2CCC(Cc3nccc(=N)[nH]3)CC2)C)=O)CC(S(=O)(=O)N(C)C)C1 21361,C(=O)(CCC(N)=O)NC(C1(C(N2CCC(c3nc[nH]n3)C2)=O)CC1)C 21362,C(C)(c1cccc(C(F)(F)F)c1)=CC(=O)NC(CCC)(C)C(=O)O 21363,C1(c2c(OC)cc(Br)c(F)c2)NC(=O)N(CCC2CC2)C2=C1C(=O)NC(C)C2 21364,C(=O)(CCc1ncc[nH]1)NCCNC(CNC(=O)OC)=O 21365,C1(CC=C)CCCN(C(=O)NCCNC(C2CCCCC2)=O)C1 21366,C1(NC(CCC2CCN(C(c3c(C)nc(C)o3)=O)C2)=O)CC2(CCCC2)C1 21367,C1(CN(C(=O)Cc2cncs2)C)CCCCN1C(=O)Cn1ncccc1=O 21368,c1(C(=O)NCC(c2ccccc2)NCC)cc(C(=O)O)oc1C 21369,N1(C(C2C(CC)CN(C(C3CCN(C)C3=O)=O)C2)=O)CCc2nc[nH]c2C1 21370,c1(C(=O)NC(C)CCNC(=O)C=CC2CCCC2)cnc2ncnn2c1O 21371,N1(C(C#CC(=O)N(C)C)=O)CCN(C(=O)CC2C=CCCC2)CC1CCO 21372,CCC(C(=O)N1CC(OCC(N)=O)C1)NC(c1cc(CO)[nH]n1)=O 21373,C1(NC(CC(CCC)C)=O)CCC2CN(C(=O)CCC(C)=O)CCC2C1 21374,n1(SCC(N2CC(CC(C)NC(=O)C(F)C3CCCC3)C2)=O)nnnc1C1CC1 21375,CC(C)(C)C(C#N)C(=O)NCCC1(C)CCN(C(C2CC3(CCC3)C2)=O)C1 21376,c1(CC)cnn(CC(=O)NC2CC(CNC(=O)C(C)O)C2)c1 21377,N1(C(C(C)OC)=O)CCC2CN(C(=O)CN3CCP(C)(=O)CC3)C2C1 21378,CCC(C)(O)CCNC(N1CC(N2CCOCC2)C(C)C1)=O 21379,N1(C(CCc2cc(C)no2)=O)CC(N(C(=O)C(F)OC(F)(F)F)C)C(O)C1 21380,C1(F)(CNC(c2c(C)snn2)=O)CCN(C(c2cc(C(C)(C)C)[nH]c2C)=O)C1 21381,Cn1nc(C2CC2)cc1C(C1(C(C)(F)F)CC1)=O 21382,c1(OC)cccc(F)c1C1CCCN1C(=O)CCNc1ccnc(Cl)n1 21383,CC(C)CCCCC(=O)N1CC(C(=O)NCC2CC23CC3)CCC1(C)C 21384,Cc1cc(C(C)NC(=O)N(C2CC=CCC2)CCO)no1 21385,CN1CCN(C)C(C(N2CCOCC2C(=O)NC2CCCC2O)=O)C1 21386,n1(C(C)C(C)(C)C)nc(-c2cccc(Cl)c2)nc1C1CC2CC2C1 21387,C=C=CC(C)C(=O)NC1(C)CCN(C(C2CC(=C3CCC3)C2)=O)C1 21388,Cc1csc2ccc(C(N3CCCC3(C)CNC(c3nn(C)cc3C)=O)=O)cc12 21389,N1(C(c2cnn3c2OCC3)=O)CC2CCC(C1)N2C(c1cnc2n1CCC2)=O 21390,C12(CNC(C3CC(SC)C3)=O)CCC(CC1)N(C(c1cncn(C)c1=O)=O)C2 21391,C(=O)(NNc1ccc(C(=O)OC)cn1)c1c(CCC)[nH]cc1 21392,c1(N2CCC(C)(CC)C2)ccc(S(=O)(=O)NCC(c2ncccc2F)(C)C)cn1 21393,CCC(C)(C)C(O)C(=O)NCC1CC(C)CCN1C(c1cc2c(nn1)CCC2)=O 21394,c1(CC(=O)NCCNC(c2cc(F)cc(N)c2F)=O)ccc(S(=O)C2CC2)cc1 21395,Cc1ccc(C)c(C(N2CC(CNC(=O)CC=CC(C)(C)C)C(O)C2)=O)c1 21396,C1(OCCC)CCN(C(=O)CC2CC(C)N(C(c3cccc(CO)n3)=O)C2)CC1 21397,c1(C(C)(C)C)cc(C(=O)NC2CC(CNC(C3(C)C=CCCC3)=O)C2)ccn1 21398,C1(C(=O)OC)CCN(C(=O)C(C)NC(c2c[nH]nc2C(C)C)=O)CC1 21399,c1(CNC(NC(COC)C(C)C=C(C)C)=NCCCF)cc2c(cc1Cl)OCCO2 21400,C1(NC(CCC=CCC=C)=O)CCCN(C(c2ccn(C3CC3(F)F)n2)=O)C1C 21401,CN1CCCC(C(N2CCCC(n3cc(COCCO)nn3)C2)=O)C1 21402,c1(CC(=O)NCC2CC(NC(c3ccsn3)=O)C2)ccc(OC(F)F)cc1 21403,C1(C(=O)NC(C(C)CN(C2CCCC2)C(CNC(CC)=O)=O)(C)C)CCCN1N=O 21404,C1(OC(C)=O)C2CCN(C(=O)C(=O)NCc3n[nH]c4c3CCCC4)C2C1(C)C 21405,c1(C(N2CC3C(CNCc4c(OCC)nccc4)(C3)C2)=O)ccc(F)cc1C#N 21406,C(CCC(C)(C)C(=O)NC(c1nccn1C)CC)NC(C(CCCC)O)=O 21407,C1(CNC(=O)CCOC2CCOC2)CCCN(C(c2cc[nH]c2)=O)CC1 21408,c1(NC(c2ccc(-n3ncc(C)c3)cc2)=O)ccc(Cl)c(Br)c1Cl 21409,N1(C(c2c(SCC)cc(C(F)(F)F)cc2)=O)C2CCC1CN(C(C1CC1C)=O)C2 21410,C1(C(=O)NC(C)CN2CCN(C(C3CC4(CSC4)C3)=O)CC2)CCC(=O)C(C)C1 21411,N#CC1CCN(C(=O)CC2(CNC(=O)CC3CCOC3)CC2)C1 21412,c1(C(N2CCC(NC(CCCN(C)C)=O)(CO)CC2)=O)ccc2nonc2c1 21413,CC1CC(NC(c2ccoc2Cl)=O)CN1C(c1c[nH]c(C(F)(F)F)c1)=O 21414,O(N1C(=O)c2ccccc2C1=O)CC(=O)NC(C)CNC(C1(F)CCCCC1)=O 21415,c1(CC)nc(CC(=O)N(C(C)CN(C)C(C2CC2(C)C)=O)C)cs1 21416,N1(C(C2N(N=O)CCCC2)=O)CC(NC(=O)C(F)(F)C(F)(F)F)CC2(CC2)C1 21417,N1(C(C(C)(C)SC)=O)CCC(C=CC(=O)NOCCN(C)C)CC1 21418,c1(OC)cc(C(=O)NC2CN(C(=O)CC3CC3C3CC3)CC2F)c(Cl)cc1Cl 21419,C1(NC(C=C(CC)C)=O)CC2(C1)CC(NC(C1CCC(C)(CC)O1)=O)C2 21420,C1(NC(Cc2cccc(OC)c2)=O)CCCN(C(=O)CS(C)(=O)=O)CC1 21421,N1(C(C(=O)N(CCOCC2CC2)C2CC2)CC2CCCC2)CCCC(F)CC1 21422,C(=O)(C(C)(F)C(C)(C)F)NC(CCC)C(=O)Nc1ccc(F)c(C(=O)O)c1 21423,CC1=CC(NC(=O)CCC2CC(NC(=O)Cc3ccns3)C2)CCC1 21424,N1(C(c2ccc(OCCC)cc2)=O)CCOCC(NC(=O)CC2CCC(=O)O2)C1 21425,C1(N(C(C2(CC)CC2)=O)C)CCCN(C(=O)Cc2nccc(OC)n2)C1 21426,CC(CCNC(C1(S(C)(=O)=O)CC1)=O)CCNC(=O)CSC1CC1 21427,c1(C(N2CCC3CN(C(C(CC=C)CC=C)=O)C3C2)=O)cccc2oc(O)nc12 21428,c1(OC)cc(OC)cc(C(N2CC3(NC(=O)Cc4cnc[nH]4)CC2C3)=O)c1 21429,C(C(C(=O)N1CC(NC(N)=O)C1)C(C)(C)C)NC(Cn1ncc(C#C)c1)=O 21430,c1(C(=O)NCCCC=C)ccc(S(=O)(=O)NCCSC2CC2)cc1Cl 21431,c1(C(c2n(CCC)nnn2)NCC(c2ccccc2F)C)noc2c1CCC2 21432,N1(C(CCCCC=CC)=O)CC(NC(=O)C(=C2CCCCC2)F)CC(C)(C)C1 21433,c1(C(=O)NCC(C)N(C(c2cnc(O)n2C)=O)CC)c(C)cncc1C 21434,N1(C(c2c(C)cn(C)c2)=O)Cc2[nH]nc(C(N3CC(O)(C(N)=O)C3)=O)c2C1 21435,C(=O)(CCCC(=O)NOC(C)(C)C)NC(C(C)NC(CC=C)=O)C 21436,C1(NC(c2cnnn2C2CC2)=O)CC2CC(C1)N(C(C1SC3C=CC1CC3)=O)C2 21437,c1(C(N(CC2N(C(c3cn(CCC=C)nn3)=O)CCC2)CC)=O)cc(Cl)cn1C 21438,N1(CCCC(C)(F)F)CCC2C(O)CC2C1 21439,N1(C(CC2CC(NC(C=CC=CC)=O)C2(C)C)=O)CCCC2(CC(O)C2)C1 21440,C(C(F)(C(=O)N1CCCCC1C(C)C)C(C)C)NC(c1nc(CC)oc1)=O 21441,N1(c2cc(SC)nc(SC)n2)CCC(CNC(C2CC(C)(C)C2)=O)C(F)(F)CC1 21442,N1(C(C2(C)COC2)=O)CC2(CCCCN2C(=O)CN2CCNC2=O)C1 21443,c1(OC)cnccc1C(=O)NC1CCCCC1NC(=O)COCCSC 21444,C1(NC(CCC2(C(=O)OC)CCCC2)=O)CN(C(C2CCOC2C)=O)CC1C 21445,C12(C(N(C3CCC(n4cc(CN(C)C)nn4)CC3)C)=O)CCC(CF)(CC1)CC2 21446,N1(C(c2ccn(CC)n2)=O)CCN(C(=O)CNC(c2ccccc2)=O)CC1 21447,c1(N2CC(O)C2)nc(N2CCC(OC)CC2)nc2cc[nH]c12.O=S1(=O)CCCN1 21448,C=CCC(CNC(=O)CC(CC)C1CCC1)C(=O)NC(c1ncc[nH]1)C 21449,c1(C(=O)NC(CC)CNC(=O)CC(C)C2CCCCC2)nccc2cccnc12 21450,C1(NC(c2c(OC(C)C)nccc2)=O)CN(C(C2CCC3CC23)=O)CC2(CC2)C1 21451,C1(NC(COCC(C)(C)C)=O)CN(C(c2cnco2)=O)CC2CC12 21452,O(NC(=O)C(CC#CC)n1ccnc1)CCCC#C.C(c1ccncc1)=CC(=O)NC 21453,c1(C(=O)NCC(CC)NC(c2cccc(N)c2C)=O)cccc2[nH]cc(Cl)c12 21454,c1(C(N2CCCC(CC(=O)NC3CCC(C)CC3)C2)=O)c(F)cc(O)cc1F 21455,c1(C(C)C)noc(CCC(=O)N2CCC2CNC(=O)C(F)(F)c2nccs2)n1 21456,c1(C(=O)NC2C(C)N(C(=O)C(C)S(C)(=O)=O)CCC2)cnc2cc[nH]c2c1 21457,N1(C(C(=Cc2cnc[nH]2)C)=O)CCN(C)C(CNC(=O)C(C2CCC(=O)N2)C)C1 21458,Cc1cc(CN(C(=O)C(C2(C)CC2)NC(c2nccn2C)=O)C)n(C)n1 21459,C(=O)(C(CCOCCO)NC(C1(n2cccc2)CC1)=O)NC(C1CCN(C)C1)C 21460,c1(C(N(C(C)CCNC(c2cn(C3CCCC3)nn2)=O)C)=O)cccc(=O)n1C 21461,c1(C(C)NC(=O)NCC(=O)NCC2CCOC2)ccncc1F 21462,C(=O)(C1CCCc2cncn21)NC(C)CCNC(=O)C(c1cc(F)cc(F)c1)O 21463,C1(C(=O)NC2(CO)CN(C(C=CC(=O)OCC)=O)C2)CC(O)CN1C(N)=O 21464,c1(CCC(=O)N(C)Cc2ccccc2Br)cccc(OC(F)(F)C(F)F)c1 21465,C1(CC(=O)NCCC2(OC)CN(C(=O)COCCCF)C2)CCCC(C)(C)C1 21466,C(=O)(C1=CCCCC1)N1C(CN(C(CCC2COC(C)(C)O2)=O)C2CC2)CCC1 21467,C(C)(C)(CCC(=O)N1CCC(c2ccccc2)(CNC(=O)CC2CC2)CC1)OC 21468,C1(C(=O)NCC(CNC(=O)CC(F)(F)Cl)F)COc2ccccc2C1 21469,C1(O)(C(C)NC(c2csc(Cl)n2)=O)CCN(C(C2CCN(C)C2=O)=O)CC1 21470,N=c1cc[nH]cc1CN1CCC(NS(C)(=O)=O)C1.N12CCN(CC1)CC2=O 21471,C1(C)(CNC(CC)=O)CN(C(C23CCCC2CCC3)=O)CC1C 21472,c1(C(N2CC3(CN(C(CN(C)CC)=O)C3)C2)=O)cccc2[nH]nc(O)c12 21473,N(C1CCCc2n[nH]cc21)C(c1c(C(=O)OC)c(F)ccc1Br)=O 21474,c1(OC)cccc2c(Br)cnc(N3CCOC(CS(C)(=O)=O)C3)c12 21475,C1(NC(CCc2c(C)ncs2)=O)CN(C(c2ncc(F)cc2F)=O)CCC1C 21476,c1(C(=O)NC2CCN(C(C(C(C)C)NC=O)=O)C2)cccc2nc(O)oc12 21477,C1(CCCNC(C=CC=CCC)=O)CCCN1C(c1cc(C)c[nH]1)=O 21478,C1(C(=O)NC2CCN(C(CCNC(=O)OC)=O)CC2O)CC(C)(C)OC1(C)C 21479,C(=O)(C#CC1(C)CCCO1)NCCOC1CCN(C(C(C2CCOCC2)C)=O)C1 21480,C1(NC(CN2CCC(C)CC2)=O)CC2CC1CC2C(=O)NCCCc1cccs1 21481,C1(C)(C(=O)NC(C=C)C2CC2)CCN(C(=O)COC2(C)CCC2)C1 21482,N1(C(CS(=O)(=O)NCC)=O)CCN(C(c2scc(C)c2C)=O)CC1CC 21483,Cc1cc(Cl)ccc1NC(C1CSCCN1C(c1ccc(CCO)cc1)=O)=O 21484,N1(CCNC(CCNC(C2(CO)CCCC2)=O)=O)CC(CO)(CF)C1 21485,c1(CN2CCC(C)(NC(C3CN(CCC)C(=O)C3)=O)C2)n[nH]c2ccccc12 21486,c1(OC)cccc(S(=O)(=O)NNC(=O)c2ncccn2)c1 21487,C1(C(=O)NC2(C)CCCCC2)CCC2(CCN(C(C3CCNC(=O)C3)=O)CC2)O1 21488,N1(C(COCCC(C)C)=O)CCC2CN(C(C34CCCC3C4(F)F)=O)CC2CC1 21489,c1(C(=O)NCC2OCCN(C(C3CC(C#N)(O)C3)=O)C2)ccnc2[nH]nnc12 21490,CC1(C)NC(=O)CC1C(N1CC(NC(C23CCOC(C)(C2)C3)=O)C1)=O 21491,c1(OC)ccc2c(c1)OCC(CN1CCCC(CCO)CC1)=C2 21492,C12(C(=O)NC3CCN(C(C)=O)C3c3ccccc3)C3C4C1C1C2C3C41C#N 21493,C1(N(C(=O)CC(C)COC)CC)CCCN(C(c2occc2C)=O)CC1 21494,C(=O)(C#CC1(C)CCCO1)NCC(C)CNC(c1ccccc1C1CC1)=O 21495,C1(F)(C(=O)NC2CC(CCNC(C=CC(C)C)=O)C2)CCCOC1 21496,N1(c2snc(CCC)n2)CCC2(CCCCC2NC(=O)CCc2nnc(C)o2)C1 21497,CCC1=C(C(=O)N2CCN(C(c3ccnn3CC)=O)C(CCSC)C2)SCCO1 21498,C=CCC(CC(C)C)C(=O)N1CCN(C(=O)Cc2ncoc2C)CC12CCC2 21499,c1(CC(=O)NC(C)CC(C)NC(c2ncoc2C2CC2)=O)ccc(F)c(Cl)c1F 21500,N1(C(CCC(=O)NCC)=O)CC(C)C(C)(C(=O)NCc2[nH]cnc2C)C1 21501,C(C(C)(C)CCNC(=O)CC1CC=CCC1)NC(C1C(C(=O)OC)COC1)=O 21502,c1(C(=O)NC(c2cccnc2)C(N2CCC(CO)C(O)C2)=O)cnn2ccccc12 21503,N1(CCC(=O)NCCNC(c2ncccc2O)=O)CCCCC1=O 21504,Brc1c[nH]c2c(NCc3cc(COc4ccccc4)c4n3CCCC4)ncnc12 21505,C(C(COC)CC(=O)NCCn1cc(Cl)c(C(F)(F)F)n1)OC 21506,C1(NC(C2C(=C)CC2)=O)CCN(c2cc(C)nc(CC3CC3)n2)CC1O 21507,C1(C(=O)NCCC(C(N2C(CN(C)C)COCC2)=O)O)CC(=O)CC(=O)N1 21508,C1(NC(C(=Cc2cccnc2)C)=O)C2CCC1CN(C(c1ccns1)=O)C2 21509,O=C(C#CC1CCCCO1)NC1CN(C(=O)CCC2CCCC2)CC1C(F)F 21510,Cn1ncc(Cl)c1-c1cc(C(=O)NC2CC2CNC(=O)Cc2cnsc2)on1 21511,C(=O)(C1CCCc2nn[nH]c21)NCC(CNC(=O)COC1CCCOC1)O 21512,C1(C(=O)NCc2ccc(C(=O)OCC)o2)C(Cl)(Cl)C12CC2 21513,C1(C2CC2)(CNC(C(c2cccc(C)c2)C)=O)CCN(C(=O)CCN2CCC2)C1 21514,N1(C(CCC2CCN(C(C3(Cl)C(C(C)=O)C3)=O)C2)=O)CCC(C2CCC2)C1 21515,c1(C(=O)NC(C2CCOCC2)(C)C)cc(CNC(C2CCCOCC2)=O)ccn1 21516,Cc1cccc2c1CCCN2C(C12CCNCCC1C2)=O 21517,c1(CC(=O)N(C(C(=O)N(CC(O)CF)CC)C)C2CC2)ccc(C)nc1 21518,c1(C(=O)OC)ccc(CC(N2CC3C(NC(C4CC4C)=O)C3C2)=O)cn1 21519,C1(c2cn(Cc3cccc(N(C)Cc4ccncc4)c3)nn2)CC2CCC1CC2 21520,c1(C(=O)NC(CCNC(C(C(CC)C)O)=O)C)c[nH]c2cccnc2c1=O 21521,N1(C(CC(=O)N(C)C)=O)CCCC2C(NC(c3[nH]nnc3C3CC3)=O)C(C)(C)C12 21522,N#Cc1ccc2c(c1)C(=Cc1cnc(CO)cn1)CC2 21523,C=CCC(O)(CC=C)C(C)NC(C1CCC(N)CC1)=O.c12cc3c1cccc3[nH]2 21524,C(=O)(C1=NOCC1)N1CC(C(=O)NOC(C)CC)(CC)C1 21525,C(=O)(CCCCCN1CCOCC1)NC(c1cn(CCO)nn1)CCC 21526,C1(C(C)NC(C23CCC2C3)=O)CCN(C(=O)C(F)(F)C2CC2)CC1 21527,N1(C(C2(OC)CC2)=O)CC=CC(NC(c2c[nH]nc2C2CC2)=O)C1 21528,CC(C)C(CNC(C1CCC2(CCC2)O1)=O)C(=O)NCc1cccc(F)c1 21529,C1(O)(CNC(CN(C(C=C=C(C)C)=O)CCO)=O)CC2C=CC1C2 21530,c1(C(=O)NC23CCC(CC2)CC3)coc2c1CN(C(C1CC(O)C1)=O)C2 21531,C1(C)(C(=O)NC(C2CCCO2)CC)CN(C(=O)CCCCNC(C)=O)C(C)(C)C1 21532,N1(C(C(CC)F)=O)CCN(C(C2(C)CCC(=O)C2)=O)CCC1C 21533,C=CCCC(F)(F)C(=O)NC(CO)CCCCNC(c1cnsn1)=O 21534,c1(C(C(=O)N(CCN(C(CC2(C=C)CC2)=O)C(C)C)C)(C)OC)ccccc1F 21535,CCCCCCC(C)C(=O)NC1CC1NC(c1cc(C)cc(F)c1N)=O 21536,c1(C(=O)NC(CNC(Cc2c(C)non2)=O)CO)ncc[nH]c1=O 21537,c1(-c2cn(CC(N3CCCC3CN3CCCC3)=O)nn2)cccc(OC(F)F)n1 21538,C1(CNC(CC(CC)OC)=O)CN(C(=O)CCc2nc(C)no2)CCC1(F)F 21539,N1(C(c2ccc(CN(CC)CC)o2)=O)CC(CCNC(c2ccsc2)=O)C(C)C1 21540,c1(C(=O)Nc2c(C)ncc([N+](=O)[O-])c2)ccc2ncc(Br)cc2c1 21541,c1(C(N2CCC3CCC(NC(=O)C4=CCC4)C2C3)=O)cc2c(c([N+](=O)[O-])c1)OCO2 21542,n1(CC)nc(C)c2cc(C(=O)NCC(C)(CO)NC(C3CC4CCC4C3)=O)sc12 21543,N1(CC)CC(NCc2cnc(Cl)c(F)c2)CC(C)C1 21544,N#Cc1ccnc(N2CC3CN(Cc4ccncc4C(F)(F)F)C3C2)n1 21545,C1(COC)CN(C(=O)C=Cc2cccs2)CCN1C(=O)CC(C)(C)F 21546,C=CCC(C)(C)CC(=O)NCCNC(=O)C(c1ccc(OC)cc1)NC(C)=O 21547,C1(CCNC(C2C(C(=O)OC)CCC2)=O)CCN(C(c2nc(O)c(C)s2)=O)CC1 21548,C1(C2CCN(C(=O)CCCCC(F)F)C2)(NC(=O)Cn2ccc(O)nc2=O)CC1 21549,N1(C(COCCCOC)=O)CCC2(CC1)CCN(C(C1CCCC1OC)=O)C2 21550,c1(CC(C(=O)NCC(CNC(Cc2nc(C)[nH]n2)=O)CO)C)ccccc1F 21551,c1(C(=O)NC2C(C)(C)N(C(C3CN4CCN3CC4)=O)CC2)cnc2nccn2c1 21552,CC1C(C)N(C(=O)C2=CCOC2)CCN1C(=O)CCCCN1C(=O)CCC1=O 21553,c1(CC(=O)NCC2(O)CN(C(c3oc(C)c(CO)c3)=O)C2)cccc([N+](=O)[O-])c1 21554,CC(C)C(C(=O)NCC(n1cc(-c2cccc(C(F)(F)F)c2)nn1)C)C(C)C 21555,S(=O)(=O)(c1ccc(Cl)nc1C)NC(C1CCN(C(CCCC)=O)CC1)C 21556,N1(C(COC2CN(C(c3snc(C)c3N)=O)C2)=O)CC2CC(C)(C)C2C1 21557,C(C(CC(C)C)C(=O)NCc1c(C)noc1C)NC(C=CCN(CC)CC)=O 21558,c1(OC)ccc(C(=O)NCC(CNC(=O)CCc2cccnc2F)CO)c(C)c1 21559,CC1(C)COCCC1C(=O)NC1CCC(NC(C2COC2)=O)C1 21560,c1(C(=O)NC)ccc(F)c(-c2ccc(NC(C3CCC(O)CC3)=O)c(OC)n2)c1 21561,C1(CC=C)(NC(=O)CCc2ccc(C)s2)CCN(C(C2CCO2)=O)C1 21562,c1(C(N2C(CN(C)C(c3ccon3)=O)COCC2)=O)noc2c1CCCCC2 21563,C1(C(=O)NCCOC2CN(C(C(C)(C)C)=O)C2)Cc2ccccc2O1 21564,Cc1scnc1C(=O)N(CC(C)C(=O)NCCN1CC2CC2C1)C 21565,C=C(Br)CC(=O)NCCC1CCN(C(C2CCCC2)=O)C1 21566,N1(C(=O)Cc2cncc(F)c2)CC2CC(C1)N(C(=O)COc1cccnc1)C2 21567,OC1(CNC2CCN(Cc3ccccc3)C2)CC(O)C1 21568,Cc1cc(C(=O)NC2(CNC(=O)CC3CCOC3=O)CC2)c2ccccc2n1 21569,CCC(CC(=O)NCCCOCCC(=O)NC1C(CO)CC1O)C(C)C 21570,CC1=CC(NC(=O)COC(C)(C)CNC(C2(C)CCCC2)=O)CCC1 21571,CN1CCN(C(C2COCC2NC(=O)C=Cc2cocn2)=O)CC1=O 21572,c1(C(N2CCN(C(C3(C(=O)NC)CCC3)=O)CC2)=O)cncc(Br)c1C 21573,N1(C(c2cscc2C)C(=O)NCc2ccc(OC)cc2)CCn2ncc(Cl)c2C1 21574,C(CCC(=O)NC(c1ccccc1)CNC(=O)CCc1ncccn1)=CC(C)C 21575,Cc1[nH]c(C)c(NC(N2CCC(c3ccccc3)(C(F)(F)F)C2)=O)c1C 21576,CN1CCc2ccc(C(N3CC4CC4(NC(=O)CCn4cncn4)C3)=O)cc21 21577,C1(NC(=O)CCc2cscn2)CCOCC1NC(=O)CCC(=O)N1CCCCC1 21578,CC1(C(=O)NC2CC(CNC(=O)CC3CCCC34CC4)C2)CC(C#N)C1 21579,CC1CN(C(c2cnc(CNC(=O)C3=CCCCO3)nc2)=O)CC(C)(C)O1 21580,c1(OC)nn(C)cc1C(N1CCC(C(=O)Nc2cc(C(C)(C)C)no2)CC1)=O 21581,C(CCC(CO)NC(=O)CC1CC(O)C1(C)C)NC(c1nc(COC)oc1)=O 21582,N1(C(Cn2c3cccc(C)c3cc2)=O)CCC2(NC(=O)CCF)CCCCCC12 21583,C(=O)(C1=CCCSC1)NC1(C)CN(C(C2CCN(C3CC3)CC2)=O)C1 21584,C1(C(=O)NCC(COC)C)COCC1NC(c1cnn(CCO)c1)=O 21585,c1(C(=O)NC2(CNC(c3nocc3Cl)=O)CC(OC)C2)cc(C)c2n[nH]cc2c1 21586,Nc1cc(C(N2CC(NC(=O)CCNC(c3ccsc3)=O)C2)=O)cc(F)c1 21587,CC(C(=O)NCCN(C)C(c1ccns1)=O)C(F)F 21588,c1(CC(C(=O)N(C(CNC(COC)=O)C(C)C)CC)N2CCCC2)ccc(Cl)cc1 21589,N1(Cc2scc(C)n2)CCOCC(NC(c2ccc(C#N)s2)=O)C1 21590,N1(C(c2cccc(CNC(C(C)(C3(C)CC3)OC)=O)n2)=O)CCOCCC1C 21591,c1(C(N2CCC(NC(CCS(C)=O)=O)(CO)CC2)=O)ccc2c(c1)CC(=O)N2 21592,C1(SC)CCC(NC(=O)C(C)OC(C)=O)C1.C1(=CC=O)CCOCC1 21593,CCC1=C(C(=O)N2CC(OCCNC(c3cc(OC)cnc3F)=O)C2)CCCO1 21594,N1(C(CN(C(=O)OC)C)=O)CCCC(NC(=O)CCC2CC(C)C2)CC1 21595,CC1C2CCC(C2)C1C(N1CCCC(C)(C(=O)NC2CC23CCOCC3)C1)=O 21596,C1(CCNC(C(C)OC(C)=O)=O)CCN(C(c2cn(C)cn2)=O)C1 21597,C(C(CC(F)(F)F)NC(C1(C)CC1(Cl)Cl)=O)NC(c1c(CC)oc(C)c1)=O 21598,O(NC(=O)CCC1CCC(NC(=O)Cn2cc(CC3CCNC3=O)nn2)C1)CC 21599,Cn1ncc2cc(C(N3CC(NC(=O)CC4CCCOC4)C(F)C3)=O)cnc12 21600,N1(C(c2cc(CC)ncc2)=O)CCC2CCCC12C(=O)NC1CCCC(C)(C)C1 21601,C1(C(=O)NC2CCC(OC)CC2)CCN(C(C2CCCCC(=O)C2)=O)C12CCC2 21602,N1(C(CC(CCC)(C)O)=O)CCOC2(CCN(c3cc(OC)ncn3)CC2)C1 21603,c1(C(=O)NC(CNC(c2cc(C)no2)=O)CO)ccn2ncc(Br)c2c1 21604,c1(C(=O)NCC23C(CN(C(CC)=O)C2)C3)ccc(S(=O)(=O)CC)cc1 21605,C(C(=O)NCC1CC2(CCC2)CN1C(=O)CC(C)CF)(c1ccccc1)=C(C)C 21606,N1(C(C(C)NC2(CO)CCCC2)=O)CCC(N(C(=O)C(C)(O)C2CC2)C)CC1 21607,C(=O)(C(C)(C)CCCC(C)=O)NC(CCCC)CCC 21608,c1(C(N2CCN(C(C(COC)O)=O)CC2CF)=O)ccc2c(c1)CCCC2=O 21609,c1(CNC(N2CCCN(CCN(C)C)CC2)=O)cccc2cccn12 21610,c1(N2CCCC(N(C(=O)C(C)(C)C(F)(F)F)C)CC2)nc2ccc(F)cc2s1 21611,c1(-c2nc(CCOC)nn2-c2ccn(C(C)C)n2)c[nH]c2cccnc2c1=O 21612,C1(C(=O)NC2C3CCN(C(=O)Cn4cccn4)C23)C2C3CC4C1C1C2CC3C41 21613,Cc1cc(Oc2ccc(-c3noc(-c4c[nH]cc4Br)n3)nc2)ccc1F 21614,N1(C(c2ncc(C)nc2)=O)CCC2(CC1)CC2NC(c1nccc(C)c1F)=O 21615,O=C(CC1CCOc2ccccc21)NC1C=CCN(C(c2c[nH]nc2F)=O)C1 21616,c1(C(=O)NC2CN(C(c3cocn3)=O)C3CC23)ccc(-n2cccn2)cc1Cl 21617,N1(C(CCn2ccc(C)n2)=O)CCCCC(CNC(=O)CC2COCCN2C)C1 21618,c1(CCC(=O)NCC(C)(C)NC(c2nonc2N)=O)csc2nc(C3CC3)cn12 21619,c1(C(=O)NC2CN(C(c3cccs3)=O)CC2F)ccc2nnc(C(F)F)n2c1 21620,C1(CNC(C2C(C=C)C2)=O)CN(C(=O)CCC(=O)OCC)CC12CC2 21621,C1(C)(C(N2CCC(N(C(=O)COCCSC)CC)C2)=O)CNC(=O)C1 21622,N(C1CCc2cc(Cl)ccc21)c1ccc(NC(C)=O)c(C(F)(F)F)c1 21623,N1(C(C(CC)CCOC)=O)CCC2(CC2)CC1C(=O)NCC(C)(O)CO 21624,CC(C)CCNCC(C)NC(=O)C(C1CCCC1)NC(=O)OC(C)(C)C 21625,c1(OC)ncccc1C(=O)N(CC(C)NC(c1ccc(-c2ccccn2)o1)=O)C 21626,c1(OC)cc(Cl)c(CNC(c2cc(C(C)C)nc(O)c2)=O)cc1Cl 21627,C1(C)(C(=O)NCC(C)CN(C(=O)CN2CC(C)(C)C2)C)CCC(=O)N(C)C1 21628,C1(COC)(NC(C2CC3CC3C2)=O)CCN(C(c2ccnc(C)c2)=O)CC1 21629,NCC(Cc1ccc(F)cc1)C(=O)N1CCC(CC#N)CC1 21630,c1(C(=O)NCC(C2CCCOC2)OCC)cnc2ccccn12 21631,C1(CNC(CCC(=O)NC)=O)CN(C(=O)CC(C)(F)F)CC12CCC2 21632,C1(C(=O)NCCc2scc(C(C)C)n2)CCCC1S(C)(=O)=O 21633,c1(OC)cc(C(N2CCCC2C2CCN(c3nnc(CO)s3)C2)=O)on1 21634,C=Cc1cc(C(=O)O)cc(F)c1.c12csc(n1)CCC2.C12(CC1)NC(=O)NC2 21635,n1(C2CCC(C)C2)nc(CCCN(C)C)nc1-c1cnc(C(F)F)s1 21636,C(c1ccccc1F)=CC(=O)NC1CC(CCNC(C2CC3(C2)CC3F)=O)C1 21637,c1(CC(=O)N(C2CCC(CNC(=O)COC(C)=O)CC2)CC)sc(C)nc1C 21638,C1(C(=O)NCCCCCOC)CCN(C(=O)C2=C(C)CC2)C1C(C)C 21639,CC1(C(N2CCCC(CNC(=O)COc3ccccc3F)C2)=O)CCC(F)(F)C1 21640,C1(CNC(C2(C)CSC2)=O)CCCCN1C(C1CC(C(N)=O)C1)=O 21641,N1(C(CSCCOC)=O)CCOC(c2cn(CCCC3CCOC3)nn2)C1 21642,c1(-c2nc(C3CCCC(=O)O3)n(C3CCCSC3)n2)cc(F)cc(F)c1 21643,N1(C(c2ccn(CC#N)n2)=O)CCC(CNC(c2cccc(C(F)F)c2)=O)CC1 21644,c1(C(N2C(CC)CN(C(c3cc(Br)cn3C)=O)CC2)=O)ccc2n[nH]cc2c1 21645,C1(CCCCNC(C(C=CC)O)=O)CCN(C(=O)CCSC)CC1 21646,C1(C(=O)NC(C)Cc2cccs2)C=CCN1C(C1(C)CCCO1)=O 21647,CC1=NOC(CC(=O)NCc2ccsc2C(=O)NCC(C)OCCO)C1 21648,C(=O)(C(F)(F)CCn1cccn1)NCC(C)CN(C)C(c1cc(=O)cc[nH]1)=O 21649,c1(C(N2CC(CCNC(C=CC(C)C)=O)OCC2)=O)cccc2c1C(C#N)C2 21650,O=C(C1CCCc2scnc21)N1CCCNC1=O 21651,CC1CCN(C(C2C(C(F)F)C2(C)C)=O)CCN1C(=O)CSc1ccccc1Cl 21652,C(=O)(C(C)CC(N)=O)NCCCN(CCCCNC(C(C(C)O)N(C)C)=O)C 21653,C1(C(=O)NC2(CC=C)CN(C(=O)Cc3csc(Br)n3)C2)CC=C(C)CC1 21654,C(=O)(C1=CCCC1P(C)(C)=O)N(CCN(C(C(CCCC)CC)=O)C(C)C)C 21655,c1(OC)ccc(Br)cc1CC(=O)NC1CC2(C1)CC2NC(=O)CCCC#N 21656,CC1C2CC(C2NC(=O)CN(C)C(c2ccccc2F)=O)N1C(C1CC12CC2)=O 21657,C(=O)(CS(=O)(=O)CC(F)(F)F)NC(C1CCN(C(c2c(OC)nn(C)c2)=O)C1)C 21658,c1(CNC(C2CCC(CC)C2)=O)nc(CNC(=O)C(F)(F)CC2CC2)cc(O)n1 21659,C1(CNC(C2(CCC)CCNC2=O)=O)CN(C(C2(Cl)CC2)=O)CC12CCC2 21660,N(C1c2ccccc2OCC1C)C(c1ncnn1C)CC 21661,C(=O)(C(C)S(C)(=O)=O)NCc1oc(C(N(C(c2ccccc2)CC)CC)=O)c(C)c1 21662,C1(C)(CC)C=C(C(=O)N2CC3CC(NC(c4cccc(=O)n4O)=O)C3C2)C1 21663,CCC(CC(=O)NCc1cn(C2CC2)nn1)NC(=O)C(O)Cn1cncn1 21664,CC1CC(NC(C2CCCN(CCNS(C)(=O)=O)C2)=O)CCS1 21665,N1(C(C(C(=O)OCC)(C)C)=O)Cc2cccc(CNC(C3CC(CF)C3)=O)c2C1 21666,C1(C(=O)NC(C(C)C)(C)C)CC(=O)CN1C(=O)CCc1ccncc1 21667,C1(NC(COCC(C)C)=O)CCC2CN(C(=O)CSC(F)F)CCC2C1 21668,c12cccc(c1)CO2.C(=O)(CP(C)(C)=O)NC(CCNC(c1nc(C)[nH]n1)=O)C 21669,N1(C(=O)CCc2nnc(SCCl)o2)CCCC(C)C1.N1CCCC1 21670,c1(C(N2C(C)CC(CNC(=O)CSC(F)F)C2)=O)cc(Cl)ccc1OC(C)C 21671,c1(CC)ccc(CC(N2CCN(Cc3cc(-c4ccccc4)n[nH]3)CC2)=O)cc1 21672,C(C(C(=O)N1CCN(C(=O)C=C2CCSCC2)CC1)C(C)(C)C)OCC=C 21673,Cc1nn(C2CCC2)cc1C(=O)NC(C(C)NC(c1ccc(Cl)[nH]1)=O)C(C)C 21674,O=C1CCCC(C(=O)NCCCNC(c2csc(C3CCCCC3)c2)=O)O1 21675,Cc1cc(C(C)C)nc(N2CCCOC(CNC(=O)C3=CCOCC3)C2)n1 21676,CC1(C)CC(C(=O)NC2CCCCC2CNC(C2CCCN2S(C)(=O)=O)=O)=NO1 21677,N1(C(C(c2cnn(C)c2)NC(C=CCC)=O)=O)CCC(C)(O)C(O)C1 21678,c1(NC(CCC(CC)NC(=O)C(CC)C(F)(F)F)=O)cnn2cccnc12 21679,C1(CNC(CCC=C(C)C)=O)CCC2CN(C(c3[nH]nnc3C)=O)CC12 21680,N#CC12CC(C(=O)NC3CC(CC(N4CCCC4CN4CCSCC4)=O)C3)(C1)C2 21681,c1(C(N2CC(C)C(NC(=O)CCC(C)(C)O)C2)=O)cc([N+](=O)[O-])n[nH]1 21682,Cc1ncc([N+](=O)[O-])cc1C(=O)NCCNC(C1CC(C2CCCC2)C1)=O 21683,N1(C(C2C(CCC)CCC2)=O)CCSCC1CCNC(=O)Cn1nnnc1C 21684,C1(n2cnnn2)(C(=O)NCC(CC)NC(c2c(OCC)ccs2)=O)CCOCC1 21685,N1(C(Cc2cn(CC)nn2)=O)CCC(NC(=O)CC(F)F)C1c1ccccc1 21686,n1(CCOC)nc(C(N2CCC(C(C)NC(C3(CCO)CC3)=O)C2)=O)ccc1=O 21687,C=CCC(Cc1ccccc1)C(=O)NC(c1cc(OC)ns1)C(=O)OC 21688,C1(CS(C)(=O)=O)CCCC1(c1nnnn1Cc1ccccc1)NCCSC1CC1 21689,C1(CCC(=O)N(CC(C)(C)NC(C=C(C)C(C)(C)C)=O)C)CCCCN1C 21690,N1(C(C2(C#C)CC2)=O)CC(CNC(=O)CCCN(C)C(C)C)OC2COCC12 21691,c1(C(=O)NC2CCC(CNC(C3NC(=O)OC3)=O)C2)cccc(Cl)c1Br 21692,n1(C(C)C)cnc2c(N3CCC(C)=C(C)C3)[nH]c(=NCc3ccncc3N)nc12 21693,c1(C(N2CCN(C(c3c(OC)nsc3)=O)C(CCO)C2)=O)nc(O)nc(O)c1N 21694,c1(C(=O)OC)ccc(Cl)c(C(F)F)c1.c12nc(no1)CNC2=O 21695,N1(C(c2n(CC)ncc2)=O)CC2CCCC1(CNC(c1conc1C1CC1)=O)C2 21696,C(c1ccccc1)=CCC(=O)NC(C)(C)CNC(=O)Cc1csnn1 21697,Cc1cc(CN2CC(NC(=O)COc3ccccc3F)C2)ccc1Br 21698,C1(C(=O)NCC2CC(NC(C(n3ccc(C)n3)C)=O)C2)CCOC(C)(C)C1 21699,N1(C(c2ccncc2)=O)CC2CCN(C(c3nc(Cl)c(Cl)s3)=O)C2C1 21700,C1(C(=O)NCC(CC)(C)NC(c2cn[nH]c2)=O)CC(C)CCO1 21701,Cc1nc(Br)oc1C(=O)N(C1CCCC(NC(C2(CCF)CC2)=O)C1)C 21702,N1(CC)CC2(CN(C(=O)C(c3ccnn3C)NC(=O)C(O)CN(C)C)C2)C1 21703,c1(OC)cc(C)c(C(=O)NC2CC3(C2)CC3NC(=O)CC2CCCN2C)cc1Cl 21704,C1(C(N(C)CCOCCNC(=O)C=CC2CCCC2)=O)CCCCC1C(F)(F)F 21705,Cc1ccnc(C(=O)NC2CC2CNC(c2snc(O)c2Cl)=O)c1N 21706,C(=O)(CC1OCCc2ccsc21)N(C1CCN(C(C(C2CC2)OC)=O)CC1)C 21707,c1(C(=O)NCC2C(NC(C(COC)OC)=O)CC2)cc(=O)n(C)cc1Br 21708,CCC(C(=O)NCC1CCN(C(c2cnn(CCF)c2)=O)C1)C(C)(C)CC 21709,N1(C(C(CC=C)NC(C)=O)=O)CCOCC(NC(C2CC(O)CN2C)=O)C1 21710,C(=O)(C(C)(F)C(C)(C)F)NCCCOCCN(C(c1cnc(C(C)C)nc1)=O)C 21711,C1(NC(N(C(c2ncccn2)C)C)=O)Cc2n[nH]cc2CC1C 21712,CCC(CNC(=O)CCS(N)(=O)=O)(CC)C(=O)NCC1CCOC(C)(C)C1 21713,Cc1ccc(C(=O)NC(C)CN(C(=O)CC2COC(=O)N2)C)c2c1CCC2 21714,c1(NC(C2NCCN(C(C(C)O)=O)C2)=O)cc(F)c(Cl)c(Cl)c1 21715,c1(CC(=O)NC(C2CN(C(=O)C#CC3(C)CC3)C2)C)c(Br)ccc(F)c1F 21716,CCC(CC(F)F)C(=O)NC1CCN(C(=O)CCC2CC2)C1 21717,C=C(C)CCC(C)NC(c1cccc(Cn2cc(CN(S(C)(=O)=O)CC)nn2)c1)=O 21718,c1(C(=O)NCC2C(C)(C)C(NC(C34CSC(C3)C4)=O)C2)ccc2c(c1)OCCO2 21719,N1(C(CCN(C(C)=O)C)=O)CC2CC(C1)CN(S(=O)(=O)c1ccc(F)cc1)C2 21720,C(CCNC(=O)C(C)CO)(C(=O)NCCCN1CC=CC1)OC 21721,c1(C(=O)OCC)c[nH]c(=NCC2CCN(c3cnccn3)CC2)c(C)c1.C=O 21722,c1(CNCc2c(OC)nc(C)cc2)[nH]c2ccccc2c1Cl 21723,CCC(C)C(C(=O)N1CCC(C(=O)NC2(CN(C)C)CC2)C1)N(C)C 21724,Cc1ccc(CNC(C2CSCCN2C(=O)CC2NC(=O)NC2=O)=O)nc1 21725,Cc1csc(=O)n1CC(=O)NC(C1CCCC1)CNC(=O)C(C)N=[N+]=[N-] 21726,C1(C2CCOCC2)(C(N(C2CCN(C(C34CCCC3C4Br)=O)C2)CC)=O)CC1 21727,c1(C(=O)NC(CC(C)NC(C2CCC(=O)N2)=O)C)ncccc1OC(F)F 21728,c1(OC)cc(F)cc(C(N2CCC(N(C)C(C3CC(CC(F)F)C3)=O)C2)=O)c1N 21729,C1(NC(C=CC(C)(C)SC)=O)CCCN(C(C2CCCCCO2)=O)C1 21730,S(=O)(=O)(c1ccc(C(N2C3CN(C(=O)C(C)(C)C)CC23)=O)cc1)N(C)C 21731,C(CO)(CCCCNC(c1ccc(=O)n(CCO)c1)=O)NC(C(C)OCC#C)=O 21732,C1(NC(C)=O)CCN(C(=O)OC(C)(C)C)CC1CSc1ccncc1Cl 21733,n1(CC)cc(S(=O)(=O)N2CCOCC(C(N3CCOCC(CO)C3)=O)C2)c(C)n1 21734,n1(CC(N2C(C=CC(=O)NCn3c(C)ccc3C)CC2)=O)cnc2c1CCCC2 21735,N1(C(c2c(=N)cc[nH]c2)=O)CCCC(NC(c2ccsc2Br)=O)C(F)C1 21736,c1(C(N(C2CCCCC2c2ccc(O)cc2)C)=O)csc2c1CCNC2 21737,CC(CC(F)(F)F)C(=O)NC(CC(=O)N(CC(O)C(C)(C)C)C)C(F)(F)F 21738,c1(C(=O)NCC(CC)(CC)NC(=O)CCC(C)(C)C)ccc(C#N)cn1 21739,c1(C(N(C(CN(C(Cc2c(C)nn(C)c2)=O)C)C)C)=O)ccc2c(c1)CN(C)C2 21740,C=CCCCC(=O)NCC1(OC)CN(C(=O)C(C)NC(C2CCC2)=O)C1 21741,C1(NC(=O)Cc2ccc(C(F)F)cc2)CC2CN(C(C3C4COCC34)=O)CC2C1 21742,C1(CNC(C2N(CC)CCC2)=O)C2CCC1CN(C(C1CCC1)=O)C2 21743,c1(CC(=O)OC)ccc(C(=O)NC(C)CC(C)NC(=O)Cc2cccs2)c(C)c1 21744,N1(C(CCC=CC)=O)CCC(F)(CNC(C2CCC3(CCC3)O2)=O)CC1 21745,N1(CCCC(=O)Nc2c(OC)ccc(OC)c2)CC(C)C(P(C)(C)=O)C1 21746,c1(C(C(C)NC(c2ccsc2Br)=O)NC(C=C(C)C)=O)ccccc1 21747,C(=O)(CC(C(=O)OC(C)(C)C)C(C)=O)NCC1CCN(C(C2C(CC)C2)=O)C1 21748,S(=O)(=O)(c1cccs1)NCC(=O)NC1CC(F)(CNC(c2ccco2)=O)C1 21749,c1(C(N2CCC(NC(C(C#C)(C)C)=O)C(C)C2)=O)nc2ccccn2n1 21750,c1(OC)nccc2c(C(N3CC(C)CN(C(c4cn[nH]c4)=O)C(C)C3)=O)c[nH]c12 21751,C1(NC(C(F)=CCC)=O)CC2CC(C1)N(C(C1CC1[N+](=O)[O-])=O)C2 21752,C(=O)(CC(CC1CC1)NC(C1C2CCC(F)C12)=O)N(CCC#C)C 21753,N1(C(C(C)(C)F)=O)CCC2(CNC(=O)CCCc3ccc(Cl)cc3)CCCCC12 21754,c1(OC)nc(C(N2CCN(C(c3cc[n+]([O-])cc3)=O)CC2C)=O)ccc1Br 21755,C(C)(C(=O)N(CCNC(C1CCC1n1ccnc1)=O)CC)OCC=C 21756,CN1CC(C)(C)CC1C(N1CC2CC(C1)C2NC(=O)C(C)(C)C#N)=O 21757,Cc1ccc(C(=O)NC2CCN(C(=O)CCc3cnn(C)n3)C(C)C2)c(O)c1 21758,c1(C(C(=O)NC2C(NC(C(C)C)=O)CCC2)OC(C)C)ccc(O)cc1 21759,Cc1c(C(=O)NCC2CCCC(NC(C34CCC(C3)C4)=O)C2)cnc2ccnn12 21760,C1(C(C)NC(=O)C(c2ccn(C)c2)C)CCCN(C(C2CCCC2O)=O)C1 21761,N1(CC(=O)NC2C=CC(CC(=O)NC3COC(C4CC4)C3)C2)C(=O)CNC1=O 21762,N1(C(C(C)OCCCCCC)=O)CCC(CNC(=O)OC(C)(C)C)C(O)C1 21763,c1(CNC(=O)NCCN2CCCC2C=Cc2ccccc2)cc(I)c(F)cc1Cl 21764,CC1CC(NC(c2ccc(C3CC3)nc2)=O)CN(C(c2cnc(S)n2C)=O)C1 21765,CCC(CC)C(C)C(=O)NCC1(F)CC(NC(=O)CC2=CCOCC2)C1 21766,c1(C(C)C)ccc(C(N2CCC(CF)(NC(=O)CC3CCCC3(F)F)C2)=O)cc1 21767,Cc1nc(CC(C)C)sc1C(=O)NCC1CN(C(C2OC(C)CC2C)=O)CCO1 21768,CC(C(O)C(=O)NC1CC(CCNC(=O)Cn2cnnn2)C1)c1ccccc1F 21769,CC1CC(NC(C2CCC2)=O)CCN1C(=O)C(=C1CCCCC1)F 21770,Cc1cc(C)n(-c2ccc(-c3noc(-c4ccc(F)cn4)n3)cn2)n1 21771,C12(CNC(=O)CN3CCNC3=O)CCC1CCN2C(c1ccccc1Cl)=O 21772,C(C)(CC(C)C(F)F)(c1n(CCOC)nnn1)NCCSc1ccc(OC)cc1 21773,N1(C(C2=CCC(NC(c3nc(C(C)C)oc3)=O)C2)=O)CCCC(C)(C#N)C1 21774,C(C(C)CN=c1[nH]c(=NC(C)c2cnn(C)c2)[nH]c2ccsc12)OC 21775,N1(C(CCN(C(=O)C(C(C)O)N(C)C)CC)=O)CCCC(C)C1CO 21776,c1(C(=O)OCC)cc2cc(NCC3CCCC3N)ccc2s1 21777,c1(C(N2CC(CC)C(NC(=O)CN=S(C)(C)=O)CC2)=O)nccc2cc[nH]c12 21778,CC(C)CC(CNC(=O)CC(C)NC(c1ccccc1)=O)NC(C1CC(F)C1)=O 21779,N1(C(C(C=C)C)=O)CCOCC1CC(=O)N(C1CCNC1=O)C 21780,Cc1cc(N)ccc1C(=O)NC(C)(C)CCCCNC(=O)CC1CCCOC1 21781,N1(C(CCCC#C)=O)CCC(O)(CCNC(c2csc(COC)c2)=O)CC1 21782,CC1CN(C(c2ccc(C3CCC3)nc2)=O)CC1NC(C1(F)CCOC1)=O 21783,Cc1ccc(S(=O)(=O)N(CC(N2CC(NC(=O)CC3CCC3)C(O)C2)=O)C)cc1 21784,C(C(CC(F)(F)F)NC(=O)CN1C(=O)CCC1=O)NC(C(C)(C)c1cnco1)=O 21785,c1(NCC(=O)NC(c2nncs2)C2C(C(=O)OC)C2)cc2scc(Cl)c2[nH]1 21786,c1(C(=O)NCCC2CC(NC(C3ON=C(C(C)C)C3)=O)C2)cncc2c[nH]nc12 21787,S(=O)(=O)(c1cccnc1NCCc1nncs1)NC1C(C)CCCC1 21788,C=CCCCCC(=O)N(C(C)CNC(=O)C(N1C(=O)CCC1=O)CC)C 21789,C1(C)(CNC(C=C(C)Cl)=O)CCCC1NC(c1cnc(C(C)C)nc1)=O 21790,C=CCC(C(=O)NCCCCN1CCN(C(=O)C(O)CCSC)CC1)NC(C)=O 21791,c1(-n2ncc(C(N3CC(C)(NC(CCOC)=O)C3)=O)c2)ccc(F)cc1 21792,c1(SCC(=O)NC2CC(Nc3cc(OC)nc(SC)n3)C2)nc2ccccc2s1 21793,CCC(C)(C)C(=O)C(=O)NC1CC(C)N(C(=O)CN2CCC2)C1 21794,Cc1ncc(N)cc1C(N1CC(CNC(C2CCCCCN2C)=O)C(F)(F)C1)=O 21795,c1(SC)ccc([N+](=O)[O-])cc1C(=O)NCCCC(C)(C)NC(=O)CC1(CO)CC1 21796,CCCCC(CNC(c1c(C)nsc1N)=O)NC(=O)CCN(CC)CC 21797,c1(OC)ccc(OC)c(C(=O)NCC2CN(C(c3sncc3C)=O)CCO2)n1 21798,c1(C(N(C2CCOC2)CC)=O)cccc(CNC(=O)CC(C2CC2)SC)c1 21799,CC(C)S(=O)(=O)CC(=O)N1CC(CN(C(=O)C(C)N(C)C)C)C2(CC2)C1 21800,c1(C(=O)NCCN=[N+]=[N-])cc(CNC(C2CC(CF)C2)=O)ccn1 21801,C(=O)(C(C(F)(F)F)C(F)(F)F)NC1(C2CN(C(c3ncc(CC)cn3)=O)C2)CC1 21802,N1(C(CCSCC)=O)CCN(C)CC1C(=O)NCc1nnn(C)n1 21803,c1(C(C)C)cc(N2CCCC2CNC(=O)C(C)C2CC2)n2ncnc2n1 21804,CC1CC(NCC2CCN(C(C)(C)C)CC2CO)CC(C)O1 21805,C(=O)(CC(C)(C)CC(F)(F)F)NCCCNC(c1cnc(OC)nc1)=O 21806,C1(c2cccs2)(CSC2CC23CC3)CCCC1 21807,N1(C(C(C)OC2CCOC2)=O)CCCC1C(C)NC(c1ccc(F)s1)=O 21808,c1(C(N(CC)CC2CCCN2C(C2(C)CN(C(C)=O)C2)=O)=O)ccc(CF)cc1 21809,C1(CNC(C(C(C)C)NC(C)=O)=O)CCC2(CN(C(=O)C(C)C(C)(F)F)C2)O1 21810,c1(C(=O)NCC2C(CNC(C3C(C)(C(F)(F)F)C3)=O)C2)ccn2nccc2c1 21811,C=CCCC(CO)NC(c1nc(CNC(c2ccncc2)=O)oc1C)=O 21812,C1(NC(C2(CNC(C(C)N(C)C)=O)CCCO2)=O)CC2(C1)CC(O)C2 21813,c1(C(=O)NC2CN(C(CC=C=C)=O)C(C)C2)ccc(SC)c(Br)c1 21814,CCC(C(=O)NC(C(=O)NCC1C2COCC12)C1(O)CCC1)n1ccnc1 21815,C1(CN(C)CC2C=CCCC2)C2CN(C(=O)COCC(F)F)CC12 21816,C1(CNC(C2Cc3nccnc3C2)=O)CC2(CCC2)CN1C(=O)Cn1ccnn1 21817,C(=O)(C#CC1CCCOC1)NCC1=CCN(C(Cc2cc(C)no2)=O)CC1 21818,C1(NC(c2cc(Cl)ccn2)=O)CC2CC1N(C(=O)C(C1(O)CCCC1)F)C2 21819,C1(CC(=O)NCc2cnns2)CC2(C1)CN(C(=O)Cc1cccc(F)c1)C2 21820,C1(C(=O)OC(C(=O)OCC)Cc2ccc(F)cc2)CC(=O)N(CC(F)(F)F)C1 21821,c1(C(=O)NCC2N(C(CCOCCOC)=O)CCCC2)c2c(c[nH]c1=N)CCC2 21822,N1(C(c2n(C)cc(Cl)c2)=O)CC2CN(C(C3CN=C4N=CNN4C3)=O)CC2(C)C1 21823,C(c1cc2c(cc1OC)CC(C)O2)=CC(=O)NCC(CC)NC(C1CC1F)=O 21824,c1(C(N(CCCNC(=O)CC(C)C(F)F)CC)=O)cn2cc(C)c(C)cc2n1 21825,C=CCC(C)(C)CC(=O)N1CCC(C)(C)C1C(=O)NC1CCNC(=O)C1 21826,C1(C(=O)NCC2(C(N3CCC3(CO)CO)=O)CC2)COc2ccccc2O1 21827,C1(C(=O)NC2(CCCC(=O)NC3CC4CCC3C4)CCC2)OC2CCC1C2 21828,C12(C(=O)NC(CC=C)(C)C)CCCC1N(C(=O)COCC1CCCOC1)CC2 21829,N1(C(c2c(CNC(C(C)CO)=O)noc2)=O)CCC(C)C1c1ccccc1 21830,c1(NC(C(N2CCC(C(=O)OC)C2(C)C)=O)=O)ccc(N=[N+]=[N-])cc1 21831,CCCCC(O)CC(=O)NC1CCC(CNC(c2ccc3c(c2)C(C)CO3)=O)C1 21832,N1(C(C(CC(C)C)=O)=O)CCC2(CCCN2C(=O)CCC(=O)c2ccncc2)C1 21833,C1(C(=O)NCC2C(NC(Cc3c(C)ncs3)=O)C2)CC(=O)N(C)C1c1cccs1 21834,C1(C(=O)NCc2c(C)cn(C)n2)CN(C(=O)C(CO)C(C)(C)C)CC1C1CC1 21835,n1(C(C)C(N2CC=CC(NC(=O)C(C)(F)F)C2)=O)c(S)nc2ccccc2c1=O 21836,c1(NC(C2N(C(c3ccc(N(C)C)cc3)=O)C(C)CC2)=O)nc(Br)cnc1Cl 21837,c1(C(N2CCC3(CNC(=O)O3)C2)C(=O)NCCC#N)cn2cc(Cl)ccc2n1 21838,c1(C(=O)NCCCN(C(C(C2CCOCC2)OC)=O)CCO)cn(C)[nH]c1=N 21839,c1(OC)cc(F)c(C(=O)N(CCCNC(c2cccc3c2COC3)=O)C)cc1N 21840,C1(C(=O)NC(CNC(c2sc(CC)c(C)c2)=O)(C)C2CC2)CC2CSCC(C1)C2 21841,C(=O)(CCN=c1[nH]c(=NCCC(C)C(F)F)c2sccc2[nH]1)NCC(C)C 21842,C(=O)(C1CCCn2ccnc21)N1CC2(C(NC(C(CC)OC)=O)CCC2)C1 21843,N1(C(CN(C(=O)CCc2cc(Cl)no2)C)=O)CCN(C(c2ccoc2)=O)C2CC12 21844,CCCC(C(=O)N(CC(CC)NC(c1ocnc1C(C)C)=O)C)C(C)C 21845,N1(C(=O)NC2CC(Cl)(Cl)C2)CCC(n2ncnn2)CC1.C12CCN(C1)C2 21846,O=C(CS(=O)(=O)C1CCCC1)NC1CCCN(C(c2ccc(F)c(Br)c2)=O)C1 21847,N1(C(CC(COC)COC)=O)CCCCC12CN(C(c1cc(O)ncn1)=O)C2 21848,c1(NC2(CF)CCN(C(C(C(C)C)C3CCC3)=O)C2)ccc(C#N)nc1 21849,N(C(=NCCCCC1(C)OCCO1)N1CC=C(c2ccccc2C)CC1)C(C)C 21850,Cc1nn(C)cc1CNC(C1CSCCN1Cc1sc(Br)nc1Br)=O 21851,N1(C(C2C(C)(C)C2C#N)=O)CCC(NC(=O)CSCc2cccnc2)C(CO)C1 21852,C1(C(N(C)CC2(C)CCCO2)=O)C2CC1N(C(C1CCOCC1)=O)C2 21853,c1(C(=O)NCCC2(O)CCN(C(CSCC)=O)CC2)cc2c(cc1Cl)NC(=O)C2 21854,C1(n2cc(CC=C)nn2)CCN(C(=O)Cc2csc(CCCC3CC3)n2)CC1 21855,C(=O)(C(C)(C(=O)OC(C)(C)C)OC)N.N1(C(C=CC)=O)CCCC(CN(CC)CC)C1 21856,C(=O)(C(c1cccs1)NC(=O)C(C)n1cccn1)N(CCF)CC 21857,c1(SC)nc(Cl)c(CN2CC(C(N3CCCCC3C)=O)CC(F)C2)c(Cl)n1 21858,N1(C(C(C)OCC)=O)CCCC(N(C(c2cc(SC)oc2C)=O)CC)C1 21859,N1(C(C2(OCC)CCOCC2)=O)CC(NC(c2cnccc2C)=O)CC(O)C1 21860,c1(C(N(C)CC2N(C(C(F)=C(C)C)=O)CCCC2)=O)ccc2c(c1)C(=O)C(=O)N2 21861,c1(C(N(CCCN(C(C2C(CC)OCC2)=O)C)C)=O)ccccc1C(C)=O 21862,C(C(CNC(=O)C=C1CC1)C(F)(F)F)NC(C(CC)(C)OC)=O 21863,N1(C(C(c2ccn(C)n2)C)=O)CCCCCC1C(=O)N(C)Cc1nccs1 21864,CC(C)CC(O)C(=O)N1CCCC(C(C)C(=O)NCCC#CCO)C1 21865,C(=O)(C(C)(O)CC(C)C)NCC1C(NC(c2c(C)nc(Br)o2)=O)C1 21866,N1(C(=O)NCC(=O)Nc2oc(C)c(C(=O)OC)c2C#N)CCS(=O)(=O)CC(C)C1 21867,c1(C(=O)NC(C)CCCCNC(C2CC3(CSC3)C2)=O)ccc([N+](=O)[O-])s1 21868,N1(C(C(C)CC2CCCC2)=O)CCCC(O)C1.C12(CC1)C(=O)N2 21869,C(=O)(CCC(=O)NC1(C)CCN(C(=O)C(C)OCc2ccncc2)C1)OCC 21870,c1(CNC(CCCSC)=O)nnc2n1CCN(C(=O)Cc1cnc(C3CC3)[nH]1)C2 21871,c1(C(N(C(C)(C)C)CCC)=O)oc(C)nc1C.C12CC3CC3N1C(=O)O2 21872,c1(CC#N)ccccc1CC(=O)NC1C=CCN(C(c2ccc(Br)cn2)=O)C1 21873,CC(C(=O)NC1CC(NC(=O)C(C)N2CCC2)C1)S(C)(=O)=O 21874,c1(C(=O)NCC(CNC(C2(CCC)CC2)=O)C)cnc(C(C)(C)C)[nH]1 21875,C=CCCCCCCCC(=O)NCCOCCNC(=O)C(c1c(C)n[nH]c1C)C 21876,C=CC(C)(CC)C(=O)NCC1(F)CC(NC(=O)C=CC)C1 21877,CCC(CC(=O)NCCC1(O)CCN(C(=O)C(C(C)C)NC(C)=O)C1)OC 21878,c1(C(N2CC(CNC(c3cocn3)=O)C3C2C3)=O)ncc2ccccn12 21879,N1(C(CCNC(COC)=O)=O)CCCN(C(C2CC2[N+](=O)[O-])=O)CC1C 21880,C1(NC(=O)CC2CCOC2=O)(CNC(=O)CC2CC3(CC3)C2)CC(F)(F)C1 21881,O=C(O)CC1(CNC(N2CCC(c3ccc(O)nc3)C2)=O)CCCc2ccccc21 21882,C(CCCC(=O)NCC1(OC)CCN(C(=O)Cn2cccn2)C1)NC(=O)OC 21883,CC1=C(C(=O)O)N(C(=O)OC2CCOCC2)CC1 21884,c1(CCNC(C(c2scnc2Br)N(c2ccsc2)C)=O)cccc(F)c1 21885,c1(CCC(=O)NCC(C2CCC2)NC(c2cc(C)sc2)=O)ccc(Br)cn1 21886,c1(C(N2CC(CNC(c3cncc(F)c3)=O)C(O)C2)=O)coc2c1C(O)CCC2 21887,N1(C(CNC(=O)C=CC2CCC2)=O)CC2(CC2)CC1CO 21888,c1(C(N2CC(C(=O)Nc3cnc(Cl)cc3I)SCC2)=O)c(F)ccc(Cl)c1Cl 21889,c1(C(N2CC(NC(CNC(c3ccc(C)cc3)=O)=O)C2)=O)cc(Br)c(C)cc1F 21890,C(=O)(CCCN=[N+]=[N-])N(CCC(C(C)C)NC(C1(C)CC=CCO1)=O)C 21891,Cc1cc(NCCCCC(C)NC(=O)C(F)(F)CN(C)C)n2nc(C)nc2n1 21892,N1(C(C2(CC)CC2)=O)CCCC2C1CCN2C(c1cn(CC(F)(F)F)cn1)=O 21893,Cc1cc(C(=O)N(C)CC2CCN(C(=O)C(F)C(C)C)CC2)ccn1 21894,c1(OCC)ccc(C(=O)NCC2CC2CNC(C23CCCN2CCC3)=O)c(O)c1 21895,C(=O)(C(C(C)C)n1cccc1)NCCC1CCN(C(c2cc(OCC)no2)=O)C1 21896,c1(NCC(N2CCC=C(Br)C2)=O)ccc(-c2nn[nH]n2)cn1 21897,CCS(=O)c1ccccc1C(=O)NC1CC(NC(C2CC2C)=O)C1 21898,N1(c2snc(C(=O)OC)n2)CC(C)(C)CC1CNC(c1cccc(F)c1)=O 21899,CCC(C)C(C)C(=O)N1CC2(CC(CNC(=O)COCc3ccccn3)C2)C1 21900,c1(CC)nc(C(=O)NC(C2CN(C(=O)C(C)NC(C)=O)CCO2)C)c(N)s1 21901,c1(C(=O)NCC(CNC(CCCC=C)=O)C)ccn2ncccc12 21902,C(CCC(C)(C)C(=O)N1CCC12CCCC2)NC(c1cnn(C(C)C)n1)=O 21903,c1(CN2CC3(N(C(c4ccc(O)cc4)=O)CC3)C2)c[nH]c2ncccc12 21904,CS(=O)(=NC(=O)C12CCC(CC1F)C2)N1CCOCC1 21905,C(CS(C)(=N)=O)NC(C(n1cc(CCC2CCOC2)nn1)C)=O 21906,O=C(C1=CCCOC1)N(C1C2CN(Cc3ccc(=O)oc3)CC12)Cc1ccccc1 21907,C1(CNC(c2ccc(NC)cc2)=O)CC(C(=O)N(C2CC3CC3C2)C)=NO1 21908,c1(CC)oc(C(=O)N(CC(C)NC(=O)C=Cc2ccsc2)CC)cc1C 21909,c1(Cc2[nH]nc(SCC(=O)NCCNC(C)=O)n2)c(F)ccc(F)c1F 21910,Cc1cc(C(N2CCC(C(C)(C)NC(=O)CSCC(N)=O)C2)=O)cc(C)c1F 21911,c1(CN2C(C(N3CC(C(=O)NCCOC)C3)=O)CC(C)C2)c(Cl)ccc(Cl)c1Cl 21912,CC(C)C(C(C)NC(c1cn(C(C)C)cn1)=O)NC(=O)CCC1CCC1 21913,CCC(C)(C)C(C)CC(=O)N(CC(O)CNC(=O)CCc1ccccc1O)C 21914,C12(NC(c3c(F)ccc(OC)c3)=O)CCCC1N(C(=O)COc1ccsn1)CC2 21915,Cc1ccnc(C(=O)N(C2CCN(C(=O)CC3CCC4CC34)CC2)C)c1O 21916,CC1CCN(C(=O)C(N2CCC3CC23)=O)CCN1 21917,N1(C(C(C2(O)CCCCC2)NC(COCC(=O)NC)=O)=O)CCOC(CF)C1 21918,C1(F)(CC(=O)NCC2(CC)CCCCC2)CCCN(C(C23CC(CO)(C2)C3)=O)C1 21919,N1(CCCC(C)C#N)CCC(S(C)(=N)=O)C1 21920,N1(C(CC2(CCCC)CC2)=O)CCC(Cn2cc(C3(OC)CCCC3)nn2)CC1 21921,CP(C)(=O)CC(=O)N1CCOC(CCNC(=O)CC2CCC(=O)O2)C1 21922,c1(C(=O)NC2(CCNC(Cc3c(C)occ3)=O)CCC2)cnc(S)nc1 21923,N1(C(C(CCC)CC)=O)C2CCCC1CN(C(C1(OC)CCCCC1)=O)C2 21924,c1(CN(CC(C(C)(C)C)=O)C(=O)CN2CCC(CO)CC2)ncn2ccccc12 21925,N1(C(C(CCN(C)C)NC(C2C(C)=CCS2)=O)=O)CCCC2(CCCC2)C1 21926,c1(CC(N2C(CCNC(CC3CC(OC)C3)=O)CCC2)=O)cncc(C)c1 21927,C1(NC(C(F)OC)=O)COC2(C1)CN(C(=O)CN(C)C)C2 21928,c1(OC)cc(F)c(CN=c2[nH]c(C(=O)Nc3ncnc(Cl)c3Br)cs2)cc1OC 21929,C12(NC(=O)Cc3cnccn3)CCCN(C(C3CCC=CO3)=O)CC1C2 21930,c1(CC(N2CCC(O)(CNC(c3ccc(CC)[nH]3)=O)C2)=O)cccc2sccc12 21931,c1(C(=O)NCCc2nc(CC)[nH]n2)oc(CNC(C2(OC)CC2)=O)nc1C 21932,c1(C(=O)NC2C(NC(COCCC=C)=O)CCC2)cc(F)c(C)cc1N 21933,C1(CNC(=O)COCC(F)F)CN(C(c2ccc(Cl)cn2)=O)C2CCN1C2 21934,c1(SC)cc(N2CCSCC2CCNC(=O)CC2CCCN2C)nc(SC)n1 21935,N1(CC)CCN(CC(N2CCC(OC(=O)Nc3ccc(F)cc3)C2)=O)C(=O)C1=O 21936,CC1CC(C(=O)NCC2(F)CN(C(c3c(F)cccc3Br)=O)C2)=NO1 21937,C1(NC(C(C)N(C(C(CC)n2ccnc2)=O)CC)=O)CN(C)C2(CCC2)C1 21938,C1(CC(=O)NC(C(C)NC(CN(CCOC)C)=O)CO)CCC(=O)N1C 21939,C(C(=O)Nn1cnn(C)c1=S)C1N(C(COCC)=O)CCCC1 21940,C1(NC(C2CC(C)C2(C)C)=O)CC2(C1)CN(C(c1cc(C(F)(F)F)nn1C)=O)C2 21941,N1(C(C(C)C)=O)CC2CC1CN2CC(N1CCNC(=O)C1)=O 21942,C(C)(C(CC(=O)N1CC(C)(F)C1)NC(c1c[nH]nc1OC)=O)OC 21943,c1(C(N2CCC(NC(C)C)C(C)C2)=O)ccc2c(c1)CCC(C)(C)O2 21944,N1(C(CCC=C(C)C)=O)Cc2[nH]nc(C(=O)NC3CN(C4CCC4)C3)c2C1 21945,c1(C(=O)NCC2(O)CCN(C(c3c(C(C)C)nn(C)c3)=O)C2)cc2n(n1)CCC2 21946,C1(CNC(c2c(CCCC)ocn2)=O)CC(F)(F)CN1c1nnc(C(=O)OC)s1 21947,C(=O)(CC(C)(C)COC)N(CC(C)(C)NC(C1C(CC)CCC1)=O)C 21948,c1(CN(CCOC)C(c2coc(Br)c2)=O)cccc(CNC(C2(CO)CC2)=O)c1 21949,N1(C(CC2(OC)CCCC2)=O)CC(NC(C2CCN(C3CC3)C2=O)=O)CCC1C 21950,N1(C(Cc2cc(C)nn2C)=O)CC(NC(C2(n3cc(Cl)cn3)CC2)=O)CC(C)C1 21951,c1(OC(C)C)cccc(C(N2CCCCC2CCNC(C2CCCCO2)=O)=O)c1 21952,C(=O)(NNc1nc(C)nc2sc(CC)cc12)c1cccc(SC(CC)C(=O)O)c1 21953,c1(C(=O)NCC(C)(C)O)n[nH]c2c1CCN(C(c1cccc(F)c1O)=O)C2 21954,C1(C)(NC(C(CCC)O)=O)CCN(C(=O)CCC2CC2(F)F)CC1 21955,c1(C(N2CCC(CNC(C(C)N(CC)CC)=O)(OC)C2)=O)c(C)ccc(F)c1N 21956,Cc1cc(N(C)C)nc(NC(c2ccccc2)CN(N2CCCC2)C)n1 21957,c1(C(=O)NCC2CCC(NC(c3cnnc(Cl)c3)=O)C2)ccc2nn[nH]c2n1 21958,C(=O)(CC(Cl)Cl)N(C)CC=CC(=O)N1CCC1 21959,N1(C(C2CC(C)C2)=O)CC2CCC1(CNC(C1CCC=CCC1)=O)CC2 21960,N1(C(c2c(CC)cccc2)=O)CCC2(CCCN2C(C2CCC(C)C2)=O)C1 21961,N1(C(C(CC)C#N)=O)CCC2(C(=O)NC3(C)CC4CCC3C4)CCCC12 21962,N1(C(C(N2CCC(OCCOCCOC)C2)=O)=O)CCC(F)(COC)C1 21963,C1(C(=O)NC2CC(N(C(CCNC(C)=O)=O)C)C2)Cc2ccccc2S1 21964,N1(C(COCP(C)(C)=O)=O)CCN(C(c2ccc(Cl)s2)=O)CC(CO)C1 21965,Cc1c(Cl)ccc2c(CC(=O)NCCCC3CCCN3C(=O)CC(C)F)coc12 21966,CC1CC(NC(=O)CN2CC3CC3C2)CN(C(c2cc3sccc3[nH]2)=O)C1 21967,c1(C(CC)NCC(c2ccccn2)N(C)C)ccc(Br)cc1 21968,C1(NC(COc2cn(C)nc2)=O)(CF)CCN(C(=O)C(C2CCCCC2)O)C1 21969,CN1CCC2(CCN(C(CCC3CC(F)(F)C3)C(=O)NC3CCCCC3)C2)C1 21970,N1(C(C=CC(C)C)=O)CCC2CC(NC(C3CC(=O)N3)=O)CCC2C1 21971,O=C(CCCCCNC(=O)CC1COCCO1)NCC12CCC(CC1)O2 21972,C(=O)(n1nccc1NC(=O)Nc1ccc(F)c(C(F)F)c1)OC(C)(C)C 21973,C(=O)(C(O)CC(C)C)NCC1(COC)CN(C(=O)CCC2(C#N)CCC2)C1 21974,c1(C(N2CCC(N3CCN(C(C4(O)CC4)=O)CC3)CC2)=O)cccc(Cl)c1 21975,c1(Oc2nccc(N(C(CN(CCC)CCC)=O)C(C)=O)n2)cc(Cl)cc(Cl)c1 21976,C1(NC(c2cc(C(C)C)ncc2)=O)CN(C(c2cnco2)=O)CC1C#N 21977,C1(C(=O)NCC2(OCC)CN(C(=O)C(C)Oc3ccccc3)C2)CCC(C)(C)O1 21978,C(CC(C(C)(C)C)NC(c1coc(Cl)c1)=O)N(C(=O)CC1CCOCC1)C 21979,C(=O)(C1=CC2(CCOCC2)C1)NCC1CCC(CNC(C2C(C)CCC2)=O)CC1 21980,N1(C(c2c(OC)cc(OC)nc2)=O)CC2CC(C1)N(C(C1CCC3(CC3)C1)=O)C2 21981,CC1C(C(N2CCC(C3OCCCC3NC(=O)C3=NOCC3)CC2)=O)CCN1C 21982,N1(C(CC2COCC(C)O2)=O)CCN(C(c2cccc(C(C)C)c2)=O)C(CO)C1 21983,c1(CNC(C2(OC)CCSC2)=O)cnn2c1CN(c1ccnc(C(C)C)n1)CC2 21984,C(=O)(C1=CC2C=CC(C1)C2)NCCC(C(=O)NC1(CC(C)(C)C)CC1)OC 21985,CC1(C)CCCC(C(=O)NCc2ccc(C(=O)NCCc3cccnc3F)s2)C1 21986,C(=O)(C(C(C)C)C1CCC1)NCC(NOCCCC=C)=O 21987,C1(NC(C(C)NS(CCC)(=O)=O)=O)CCCCC1C(=O)OCCC(=O)NC1CC1 21988,c1(CN(CCC)C(=O)NC2CCC2C)ccc(F)cc1 21989,CN1C(=O)C2CN(C(C3CC4C=CC3CC4)C(=O)NC3COC3)CC2C1=O 21990,c1(CNC(CC2C(C)(C)C2CN=[N+]=[N-])=O)ccc2c(c1)S(=O)(=O)C=C2 21991,c1(CCC(=O)N(CC(C)NC(C2CC(CF)C2)=O)C)ccccc1OC(F)F 21992,C1(CC=C)(NC(=O)CC(C)OC)CCN(C(=O)CSC(F)(F)F)C1 21993,Cc1nc(C)c(C(=O)NCC(C2CCCN(C(c3[nH]cnc3C#N)=O)C2)(C)O)s1 21994,c1(-c2cn(C)nc2)ccc(NC2CCOC(c3ccc(F)cc3)C2)cc1Cl 21995,N1(C(=O)CCC2CCC2)CCC2(CC1)CCN(C(C1CC1CF)=O)C2 21996,C(=O)(N=c1cc(C)n(C(C)C)[nH]1)C1(OC)CCN(C(=O)CC2CC=CCC2)C1 21997,N1(C(=O)NCCCOc2ccc(F)cc2)CCS(=O)CC1c1ccccc1 21998,C(=O)(CC(C)C(F)(F)F)NC(CC)CCC(=O)NCC1CC12CCCCC2 21999,CS(=O)(=O)c1cscc1C(N1CC(NC(C23CC2C3)=O)C(c2ccccc2)C1)=O 22000,c1(C2C(C(N3CC(CCC=C)(C(=O)OC)C3)=O)C2)ccc(-c2ccc(C)s2)cc1 22001,C(C(C)C)(C(O)C(=O)NC(C)(CNC(c1cccc(C)n1)=O)CC(C)C)OC 22002,C1(O)(CC(N2CC(C(=O)NCC(C)OC)(Sc3ccccc3)C2)=O)CCOCC1 22003,N1(C(C(C)c2ccsn2)=O)CCC(CCNC(C2CCCC2)=O)C(F)(F)CC1 22004,C(=O)(C(CCNC(=O)C(C)c1cc[nH]n1)OC)NCC(C#C)CC 22005,C1(C(N(CC(C)(C)NC(C(C)SC)=O)C)=O)CCNC(=O)C1 22006,CN=c1nc(N(C)Cc2cncn2C)[nH]c(=NC2Cc3ccc(Cl)cc3C2)[nH]1 22007,C1(C(=O)NC(CN(CCOCCC(C)C)C)C)CN(C)CCO1 22008,c1(OC)ccc(C(F)(F)F)c(CNC(c2cncc(OC)c2)=O)c1 22009,C1(NC(c2ccn(CCF)n2)=O)CCOC(CNC(C2(n3cnnn3)CC2)=O)C1 22010,N1(C(=O)OCC)c2ccccc2CCC1C(=O)NCC(C1CCC(C)CC1)(C)O 22011,C1(NC(C2C(C=C)C2)=O)CCC(C)N(C(c2cc(-c3ccccc3F)[nH]n2)=O)C1 22012,Cc1cc(C(=O)NC(C)CCNC(c2c(C)noc2N)=O)nc(O)c1 22013,C1(NC(C2C3C(NC(c4cnc(CC)o4)=O)C4C(C3)C42)=O)C(C)(C)C(O)C1(C)C 22014,C(CC(=O)N(CCNC(C1(n2ccnn2)CC1)=O)C1CC1)=CCC 22015,c1(N(C)C(C2(C)CCC(COc3ccc(F)cc3)CC2)=O)c[nH]c2cc(Br)ccc12 22016,FCCN=C(NCC=CC1CC1)NCCc1ccccc1 22017,N1(Cc2ccn(CC)c(=O)c2)CCC2(CCN(C(=O)CC(C)C(=O)OC)C2)C1 22018,c1(OC)cc(C2(C(=O)NCC#CCNC(=O)CCCSC)CCCC2)ccc1C 22019,c1(-c2c(OC)cccc2)c(NC(N2CC(C)C2)=O)nc2c(C(F)(F)F)cccn12 22020,c1(C(N2CC(F)CC2CO)=O)cc2ccc(-c3ccc4n[nH]cc4c3)cn2c1 22021,N1(C(C2C(C)(C)C2)=O)CC2CCC(NC(c3ncoc3C3CC3)=O)C2C1 22022,c1(C(N2C(CN(C(=O)C(C)(C)CF)C)COCC2)=O)noc2c1COCC2 22023,C12(O)CCN(C1)C2=O.c1(OC)ccc(C(=O)N(CC(C)C(=O)OC(C)(C)C)C)s1 22024,C1(C(N(CCN(C(c2occc2C)=O)CC)CC)=O)CCc2ccccc2C1 22025,C1(CNC(C(COC)(C)O)=O)CC2CCC1N2C(=O)Cc1ccc(OC)c(O)c1 22026,c1(C(C)NC(C(c2conc2C)N(CCC)CC2CC(F)(F)C2)=O)ccccc1 22027,c1(CC(=O)NCCN(C(=O)CC2CC2(Cl)Cl)CCC)ccnc(Cl)c1F 22028,C1(CCC)CCCN(c2nnc(-c3ccccc3Cl)n2CCC(=O)N(C)C)C1 22029,N1(C(C(C)(C)OC)=O)CCN(C(c2ccc(F)cc2Cl)=O)C(C(C)C)C1 22030,Cc1ccc(C(=O)NCC2(NC(C3CC(F)(F)C3)=O)CCOC2)nc1O 22031,N1(C(CC(=O)NCC)=O)CCN(C(c2c[nH]c(=N)o2)=O)C(CC(F)F)C1 22032,CCC(CCC(=O)NC1(CNC(c2ccc(CC)c(O)c2)=O)CCC1)OC(C)=O 22033,N1(Cc2cc([N+](=O)[O-])cc(Cl)c2)Cc2ccccc2C(CO)C1 22034,N1(CC(=O)NCC(C)N(C(c2ccc(Cl)cc2)C(N)=O)C)CCCCCC1 22035,N1(C(C2C(C(=O)O)C23CC3(F)F)=O)CCc2c(I)n[nH]c2C1 22036,N1(C(CCCCOC)=O)C2CCC1CC(CNC(=O)CC1CC(C)=NO1)C2 22037,CCC(C)C(C(=O)OCC)N(C)C.C(=O)(C(=O)N(C)C)NCC 22038,C1(CNC(C)=O)CCN(C(=NCCSC2CC2)NC(C)C)C1 22039,c1(C(=O)OCC(=O)NCC2C(C(=O)OC)CCC2)cc(C)cc(C)c1 22040,C(C(C)N=c1[nH]c(=NCC2CC(=O)N(CC(C)C)C2)c2[nH]ccc2[nH]1)OCC 22041,CC(C)C(C)(CNC(c1n[nH]cc1CNC(C1C=CC=CC=C1)=O)=O)C(C)C 22042,CN1CCC2(CC1)CN(C(C1CCN(C(C3(C)CC=CC3)=O)CC1(C)C)=O)C2 22043,c1(C(N2CC(NC(c3cc(-c4ccccc4)on3)=O)C2)=O)csc(O)n1 22044,c1(-c2ccc(C)o2)ccc(=NC(=O)C2CCC2)[nH]n1 22045,c1(OC)cc(Br)cc(C(N2CCN(C(C3CC3F)=O)C(C(C)C)C2)=O)c1OC 22046,N1(C(C(C)Cc2ccc(Cl)cc2)=O)CC2CCC(C1)N2Cc1ccc(F)nc1 22047,c1(NC(CNC(C2(SC)CC2)=O)C(C)C(C)C)ncc(Cl)cc1[N+](=O)[O-] 22048,CS(=O)(=O)c1ccc(S(=O)(=O)N2CCOC3(CCC(NC(=O)CN)CC3)C2)cc1 22049,N1(C(c2cccc(Br)c2)=O)CCC(C2CN(Cc3c[nH]c4ccncc34)C2)CC1 22050,CCN=C(NCCC1CCCCO1)NC1CC(=O)N(C(C)(C)C)C1 22051,N1(C(CCOC(CC(C)C)C)=O)CCC(C2(NC(=O)CN(C)C(N)=O)CC2)C1 22052,c12cnn3c1CN(CC3)C2=O.c1(-c2cc(C=O)on2)cccc(C)c1.CN 22053,C1(CNC(CCN(C(CC(OCC)OCC)=O)C)=O)CC(=O)N(C2CC2)C1 22054,c1(C(=O)NCCC(C)NC(c2ccc(C)c(F)c2)=O)ccc2c(n1)OCCO2 22055,c1(CC(=O)NCC(C)NC(C2(CC)CCC(O)CC2)=O)c(C)nc2ccccn12 22056,C1(C(=O)NCCCN(C(c2c(C)cc(C)cc2C)=O)CC)CCCCC12CCC2 22057,C1(C(=O)NC(CC)C)CC(=O)CN1C(=O)C(c1ccccc1)F 22058,C(CCCCC(=O)N(C1CCC(NC(C2CCCC(C#N)C2)=O)CC1)C)OCC 22059,c1(CCNC(C(C2CCC2)NC(c2cc(Cl)n[nH]2)=O)=O)ccncc1F 22060,C(=O)(C(F)CCC(C)C)N1CCCC(C(N(CC=C)CCOC)=O)(CC)C1 22061,Cc1ccc(OCC(=O)N(C(C)CCNC(=O)C(O)C2CCCC2)C)cc1 22062,c1(C(=O)NCCN(C)C(c2cc(F)c(N)cc2F)=O)cnc2[nH]cncc1-2 22063,C1(C(C)(C)O)CCCN(C(=O)C(N2CCNCC2)C2CC2)C1 22064,C(=O)(CC(C)(C)C(C)(F)F)NC(C)C(N1CCC(c2coc(=N)[nH]2)CC1)=O 22065,c1(C(=O)NCC(C)NC(c2c(C)nn(C)c2C)=O)cc(Br)c2ccccc2c1 22066,c1(C(c2n(CC)nnn2)NC2CCCCC2SC)ccc(Cl)c(Cl)c1C 22067,Cc1cc(C)c(C(=O)NCC2CCCCN2C(=O)Cn2ncn(C)c2=O)c(C)c1 22068,N1(C(CC2N(C(C=C(CCC)C)=O)CCOC2)=O)CCC2CCC(C1)N2C 22069,CCCC(C)(C)C(=O)NC(C1CCN(C(=O)CNS(=O)(=O)N(C)C)C1)C 22070,C1(Cc2nc(C)sc2)CCN(N2CCOCC3(CC3)C2)C1 22071,N#CC12CCC(NC(C3CSCCN3Cc3cnc(Cl)cn3)=O)(CC1)CC2 22072,N1(C(CN2CC(CC)C2)=O)CC2CC2(NC(=O)Cc2cncc(O)c2)C1 22073,c1(C(=O)NCC(F)=C(C)C)ccc2oc(=N)[nH]c2c1 22074,Cc1cnccc1C(=O)NCC1CCC(NC(=O)C(C)C(F)F)CC1 22075,c1(C(=O)NCC23C(CN(C(C(CSC)C)=O)C2)C3)cccc(=O)n1C 22076,C1(CNC(C2CC3CCC2O3)=O)C2CN(C(c3ccc(-c4cccs4)o3)=O)CC12 22077,Cc1cc(C(=O)NC(C)(CNC(=O)C2=CCC2)C2CC2)nn1C(C)C 22078,CCC1=NOC(C(=O)NC(CCC2CC2)C(=O)Nc2ccccc2OC)C1 22079,C1(CNC(C(C)c2cccs2)=O)CCN(C(=O)CCS(N)(=O)=O)C1(C)C 22080,Cc1ccc2c(N3CC4CC3C4)nc(=NC3CCCCCC3C)[nH]c2c1 22081,C1(CC(=O)N(CCNC(c2c(C)cco2)=O)C)CCCCN1C 22082,C(=O)(C(C(C)C)n1cnnn1)NCC1CCN(C(CN(C(C)=O)C)=O)C1 22083,CC(C)(C(=O)N1CC(C2CN(C(=O)Cc3ccon3)C2)C1)C1=CCSCC1 22084,C#CCC(C(=O)N(CCCO)CC#C)NC(c1cccnc1)=O 22085,C1(CC(=O)NCCC#CCC)CCN(C(c2c[nH]c(C#N)c2C)=O)C1(C)C 22086,C1(C)(C(=O)NCC23N(C(C(=O)NC(C)C)=O)C(CC2)CC3)CC(C(C)(C)C)=NO1 22087,Cc1cccc(C(=O)N(CC(O)CNC(=O)C(C)SCc2ccccc2)C)n1 22088,N1(C(C23C(CCN(C(C4(C)CCC(=O)C4)=O)CC2)C3)=O)CCCC2(CCCC2)C1 22089,C(=O)(C1=CNS(=O)(=O)N=C1C)N1C2CC(NC(C(CC)F)=O)C(C)C1CC2 22090,Cc1ccc(C(N2CCN(C(=O)CSCC(C)C)CC2C(C)C)=O)c(C2CC2)n1 22091,C1(N(C(CC)CO)C(C2(CN)CCC2)=O)CCN(Sc2cccc(F)c2)CC1 22092,Cc1cncc(C)c1C(=O)NC1C=CC(CC(N2CC3CC3(CO)C2)=O)C1 22093,C(=O)(C(CCOC)NC(=O)CCc1ccc[nH]1)NCC(CCC)O 22094,N1(C(C(CNC(CSCC)=O)CC(C)C)=O)CC(C)OC(C)(C)C1C 22095,c1(NC2CC=C(C)CC2)ccc(S(=O)(=O)N2CCCCC2C(C)C)cn1 22096,N1(C(COC)=O)CC2CC(NC(c3ccc(NC(c4cccs4)=O)cc3)=O)C1C2 22097,N1(C(c2c(C)c(F)ccc2Cl)=O)CC2CC3CC2C1C3NC(c1ccccc1)=O 22098,Cc1ccn2ncc(C(=O)NC3CC(C)N(C(=O)CCCc4ccsc4)C3)c2c1 22099,c1(CCNC(c2cccc(NC(=O)NC)c2)=O)c[nH]c2cc(F)c(Cl)cc12 22100,CCC(C)(CNC(c1ccnc(C)c1C)=O)C(=O)NC1(CCF)CCC1 22101,N1(C(=O)NC)CCN(C(C2CC(NC(c3ccc(F)s3)=O)C(O)C2)=O)CC1 22102,CC1CC2(CCN(C(=O)CC3CCCC3)CC2)CN1C(=O)CCCCC(C)(C)C 22103,Cc1cnn(C(C)C(=O)NC2CCC2NC(c2ccn(C3CC3)n2)=O)c1 22104,C1(O)(CC=C)CCN(C(c2conc2CNC(C2CC(=O)C2)=O)=O)CC1 22105,c1(CN2CCC(O)(C(=O)Nc3cc(O)nc(O)n3)C2)ccc([N+](=O)[O-])cc1O 22106,n1(C(C)C)cnc(C(=O)NC(c2ccnn2C)C(=O)NCC2(C)CC2(C)C)n1 22107,c1(C(N2CC(O)(C(C)NC(C3CCOC3)=O)C2)=O)coc2c1CCCC2 22108,C1(C(C)C(=O)Nc2cnns2)CCN(Cc2scnc2Cl)CC1 22109,CN1CCC2CN(C(C3(NC(C4CN(C(N)=O)C4)=O)CCOCC3)=O)CC2C1 22110,C(=O)(CCCC(=O)N1CCN(C(=O)CC2CCCSC2)C(C2CCC2)C1)N(C)C 22111,C1(c2cn(CC(=O)Nc3ccn(CC(C)C)n3)nn2)COCCC1C(=O)O 22112,c1(CSCCC)ccc(C(=O)NC2(CNC(C3CCOC3)=O)CCOC2)o1 22113,c1(CC(=O)NCC(CNC(COC(CC)C)=O)O)ccc(F)c(Br)c1 22114,Cc1oc(C(C)(C)C)cc1C(N1CC(CNC(=O)C(O)CC2CCCCC2)C1)=O 22115,c1(N2CCC(C(=O)OCC)(NC(=O)OC(C)(C)C)C2)c(Cl)cc(SC)cc1Cl 22116,C1(CSC)C(=O)Nc2noc1n2.c1(OC)ccccc1 22117,C(=O)(CCS(=O)(=O)N1CCOCC1)NC1CC(CNC(C2C(C)(CC)C2)=O)C1 22118,C(CNC(C1CC(N(C)C)C1)=O)(CCNC(=O)CCc1nccn1C)OC 22119,c1(C(=O)NC2CCC(C)N(C(c3cccnn3)=O)C2)cccc2c1CCCCC2 22120,C(c1c(C)coc1C)=CC(N1CC(O)(CNC(C=C(C)C2CC2)=O)C1)=O 22121,Cc1ncccc1C=CC(=O)NC1(CN(C)C(c2nccn2C)=O)CC1 22122,c1(NCC(C)(C)C2CCC2)[nH]c(=NCCc2ccn(C(F)F)n2)nc2scnc12 22123,N1(C(CCCOC)=O)CC2CCC1C1CN(C(c3c(CO)noc3C)=O)CC21 22124,C(C(C(=O)NC1CCCCC1)N1CCC2CCC12)(C1CCCC1)OCC 22125,c1(OCC)c(C(N2CCC(NC(=O)Cc3ccc(C)c(Cl)c3)C2)=O)cccc1F 22126,C1(NC(C2CCC(CC)CC2)=O)CCN(C(=O)C(C)(C)COC(C)C)CC1CO 22127,CC(=O)C(C)CC(C)C(=O)N1CCC(C)(C)CC1C(=O)N(CC(C)C)C 22128,c1(C(N2CCC(C(N(CC(O)C(F)(F)F)C)=O)C(O)C2)=O)cccc2ccnn12 22129,C1(CNC(=O)CCN2CCC2)CCN(C(C23CC(C(F)F)(C2)C3)=O)CC1 22130,C12(C(=O)NCc3snc(CC)n3)C(NC(=O)CC3CCOC3(C)C)C3CC1C2C3 22131,Cc1cccc(C)c1C(N1CCC(C)C(CC(N2CCC2(C)C)=O)C1)=O 22132,c1(CCOC)nc(=NCC2CN(C(=O)CC(O)CN(C)C)CCO2)s[nH]1 22133,C(C(C)(C)CCNC(=O)C(O)C1CC1)NC(c1cc(CN(C)C)on1)=O 22134,c1(OC)cc(Br)c(CN2CC(C)CC2C(=O)NCc2cccc(Cl)c2Cl)cc1O 22135,C1(CC=C)(NC(c2cnc(C(F)F)s2)=O)CN(C(c2cc(C(F)F)cs2)=O)C1 22136,Cc1cc(C)c(CN2CCC(N(C(=O)C(F)(F)Cl)C)C2)cc1C 22137,c1(CC)ncc(C(=O)NC2CCCN(C(=O)CCC(F)(F)F)C2CC)c(C)n1 22138,c1(CCC)onc(CN(C)Cc2cccs2)c1CC 22139,C1(NC(=O)CC(F)F)CC2CC1CN(C(c1cnnc(O)c1)=O)C2 22140,Cc1cccc2c1CCC2NC(c1cnc2n1C(C)CCC2)=O 22141,N1(C(C(C)C)=O)CC2CCC(C1)N(C(c1cc(C(F)(F)F)ccc1N(C)C)=O)C2 22142,CC(C)CC(CNC(=O)CC1CCC(=O)C1C)C(=O)NCC(C1CC1)N(C)C 22143,Cc1cc(C(=O)NCCc2ccn(C)n2)nn1CC(F)(F)F 22144,c1(C(N2CC(CNC(C3CN(CC(C)C)C3)=O)C2)=O)ccc2c(O)ncnc2c1 22145,N1(C(C23C(C)(C)OCC2C3)=O)CCN(C(C23C4CC(CC24)C3(F)F)=O)CC(O)C1 22146,c1(C(=O)NCCCCC2CN(C(C(C(C)O)(F)F)=O)C2)cc2ccsc2n1C 22147,c1(CNC(C(C)N(CC)CC)=O)ncoc1C1CN(C(C2CCCS2)=O)C1 22148,N1(C(c2nc(C)[nH]n2)=O)CCC2(CCN(C(C3CCC(C4CCCO4)O3)=O)C2)C1 22149,C=C(Cl)CCC(=O)NCC1CCN1C(c1ccnn1C(CC)CC)=O 22150,C(=O)(C1CCc2nccn21)NC(C)C(=O)NOC1CCCCCC1 22151,C(CC(C(=O)NCC(C)(C)N(C)C)NC(=O)C(C1CC1)OC)OCC 22152,C1(CC)CN(C(c2ccc(C#N)cc2)C(=O)NCC(F)F)CC2(CCCOC2)O1 22153,C12(NC(C(C)=CC3CC3)=O)CCC1CN(C(c1ccsc1C)=O)C2 22154,Cc1cc(NCCCCC(C)NC(c2c(F)cccc2F)=O)n2nc(C)nc2n1 22155,C(=O)(CS(=O)(=O)N1CCOCC1)NCC(C)CNC(C1(F)CCCC1)=O 22156,c1(N2CCOCC(C(N3CC4CC3CO4)=O)C2)ncc2[nH]ncc2n1 22157,c1(C(CC)N(C(=O)C(=O)Nc2cnn(-c3ncccn3)c2)C)ccc(Cl)cc1 22158,CC1CCC(NC(=O)Cc2cn[nH]c2)CN1C(c1ccc(O)nc1Cl)=O 22159,Cc1cc(NC(C23CC2CN(C(c2ccno2)=O)C3)=O)c(F)c(Br)c1 22160,C1(NC(C2C(=C)C2)=O)COC2(C1)CN(C(c1cccc3nncn13)=O)C2 22161,N1CCC(OC2CCC2)C(CC)C1.c1(OCC)cc(C=O)oc(=O)c1 22162,C1(C(=O)NCC(CNC(c2cnn(C(C)C)n2)=O)(C)F)CCCCC(=O)N1 22163,c1(CC(N2C(Cn3cc(CN(C(C)C)C)nn3)CC2)=O)c(Br)ccc2c1OCO2 22164,N1(Cc2cc(Cl)c(Br)nc2)CCC2(CCSCC2)C1 22165,c1(C(=O)NC2(C(=O)OC)CC2(C)C)cc(Br)ccc1Cl 22166,C(=O)(CS(=O)CCC(F)(F)F)N1C2(CNC(CC=CCC)=O)CCC1CC2 22167,c1(C2C(C(=O)NCC(C)(C)C(C)(C)C)C2)c(F)cccc1F.C(=O)(CCC(=O)O)N 22168,N1(C(C(CCCC)C)=O)CCC2CCCC12C(=O)NCC1CC2(CCC2)C1 22169,c1(C(=O)NC2CN(C(C(C=C)(C)CC)=O)CC2(C)C)cnc2onc(C)c2c1 22170,C1(C(N(CCCNC(c2c(OC)nsc2)=O)C2CC2)=O)CCSC(C)C1 22171,Cc1cnc(C(N2CCCC(CN(C)CCc3cnn(C)c3)C2)=O)cn1 22172,c1(C(N(C)C2CC2)=O)ccc(NC(C2CCCN2C(=O)C2CC2)=O)cc1 22173,C(C)(C(=O)N1CCC(N(CCO)C(C2CC(C)C2)=O)CC1)(C(C)C)OC 22174,C(CCN=c1cccc(S(=O)(=O)N(C)Cc2cccc(F)c2F)[nH]1)OC(C)C 22175,C(=O)(CCCCC(=O)NOC(C)(C)C)N1CCC(C(=O)OC)(NC2(C)CSC2)C1 22176,C(=O)(C1=CCCOCC1)N1CC(CC)N(C(c2cc(C)c(C)nn2)=O)CC1 22177,Cc1cc(C)c(CNC(=O)C(c2ccoc2)NC(c2cccc(O)n2)=O)cn1 22178,c1(C(N2CC(CNC(c3c(CCC)n[nH]c3)=O)(COC)C2)=O)c(C)nnn1CC 22179,C1(N(C(C2(SCC)CC(O)C2)=O)C)CC2CCC(C1)N2C(=O)CCCCN(C)C 22180,N1(C(CCC2C(=O)NC(=O)N2)=O)CCC(NC(c2cnccn2)=O)C2CC12 22181,C1(C(=O)NC(C(C)NC(c2cc(C)n(C)c2C)=O)C)CN(C)CCN(C)C1 22182,N1(C(c2c(C)snc2)=O)CCC(NC(=O)CC(C)c2cccnc2)C(F)(F)CC1 22183,C1(C(=O)NCc2ccc(C)cn2)CCCCC1(C)NC(=O)C(C)OCCN(C)C 22184,c1(CNS(CCCC)(=O)=O)cc(NC(=O)CC(C)C(=O)OC)ccc1C 22185,C#Cc1ccc(C(N2CCCC(CF)C2)C(=O)NCC(=C)C)cc1NCC 22186,c1(C(C)C)conc1CC(=O)NC1CC(Cc2nn[nH]n2)C1 22187,N1(C(C2C3CN(C(CCC(C)OCC)=O)CC32)=O)CCCC12CCCC2 22188,Cc1ccc(C2C(=O)N2)cc1.C(=O)(CCCC1CC1)NCC(O)COCC1CC1 22189,c1(SCC(C)C(=O)NCC2CCN(C3CCCC3)CC2)ccc2nonc2c1 22190,N1(C(C2C=C(C)CS2)=O)CC(F)CC1C(=O)NOCCCO 22191,C1(N(CCOC)C(c2ccncc2)=O)CCN(C(=O)C(F)n2cccn2)CC1 22192,c1(N(C)C)cccc(CNC(=O)CN2CCN(c3nc(=N)[nH]s3)CC2)c1 22193,C1(C(=O)NCCCNC(CN(c2ccccc2)S(C)(=O)=O)=O)CCC(F)C1 22194,C1(Nc2ccc(COC(C3CCOCC3)=O)cc2)CCC2CC1CN2 22195,c1(CC(=O)NC2CCN(C(=O)C(=O)NCC3CC3)CC2)ccc2c(c1)CC2 22196,c1(C(N(C2CCN(C(=O)Cc3cnn(C4CC4)c3)C2)CC)=O)cc(OC)ncn1 22197,c1(C(N2C(C)C(N(C)C)CC2)C(=O)NCCCF)cccc2c1CCO2 22198,c1(C(=O)NC2(C(N3CC(C)(CC=C)C3)=O)CCCCC2)cnc(C)c(C#N)c1 22199,N1(C(CCc2ccc(C)s2)=O)CCN(C(=O)C=Cc2cocn2)C(C)C1C 22200,C(=O)(C(CC)C(=O)N(C)CC1CCCN1C(c1cnc(C)cn1)=O)OCC 22201,C(=O)(C(C)CCCC(C)C)N1C(CCNC(=O)C=C(C)C)CC(OC)C1 22202,c1(C(=O)NC2(C3(C)OCCO3)CC2)cc(=NC(=O)CCc2c[nH]nc2C#N)[nH][nH]1 22203,C1(NC(c2ccnc(C)c2N)=O)CN(C(=O)CCCF)C2(CCCCCC2)C1 22204,c1(C(=O)NC(C(C)C)CCNC(=O)CC2NC(=O)NC2=O)ccc2[nH]ccc2n1 22205,N1(C(C(CC)N(CC)CC)=O)CC2(C1)CN(C(C1(C(F)F)CCCC1)=O)C2 22206,C1(C(=O)NCC(O)CNC(=O)Cn2ccnc2)(SC)CCOCC1 22207,c1(C(N2CCCC(c3cn(-c4ccc(Cl)cc4)nn3)C2)=O)cc2scc(Cl)c2[nH]1 22208,C1(NC(COCC)=O)CCN(C(c2cc(C)n(-c3nccs3)c2C)=O)C(C)C1 22209,c1(NC)cnc(C(N2CC3C(C(=O)NCCn4ccnc4)C3C2)=O)cn1 22210,N1(C(C2CCN(C)C2=O)=O)C2CCC1CN(C(=O)CC(C)(C)c1ccccc1)C2 22211,C12(CNC(C(CC)n3nccc3C)=O)CC(NC(c3ccccc3)=O)(CO1)C2 22212,CCCCCC(C)CC(=O)NCC1C2CN(C(=O)C(c3ccc(C)o3)C)CC12 22213,CN1CCOc2cc(C(N3CCCC3C(N3CC4CCC3CO4)=O)=O)ccc21 22214,N1(C(CC2CN(C(C)=O)C2)=O)CCC2(CC(NC(=O)Cc3ccn(C)n3)C2)C1 22215,CC1OCCCC1C(=O)NC(C)CNC(c1cccc(OC(C)(C)C)c1)=O 22216,C1(O)(CNC(NC(C)C)=NCc2ccnn2CC2CCCO2)CCC(C)CC1 22217,C1(C)(C(=O)NC2CCC(N(C)C)C2)CCN(C(c2csc(F)c2)=O)CC1 22218,N1(C(CC2(C=C)CCC2)=O)CC(CNC(C2CCC(=O)NC2)=O)CC(C)(C)C1 22219,C(C(CNC(C1C(C)C1C)=O)CO)NC(CC1(OC)CC1)=O 22220,CC1c2cc(C(=O)NCCNc3ncnc4c3CCCC4)ccc2OC1C 22221,C(=O)(C(C)(C)CC(=O)NC(C)C(C)NC(c1cc(=O)cc(Cl)[nH]1)=O)OCC 22222,C1(NC(CCC(=C)C)=O)CC(NC(c2ccc(S(C)(=O)=O)o2)=O)C12CCOCC2 22223,c1(CN2CC(F)(C(=O)NCCc3ccc(OC)cc3)C2)cc(F)cc(Br)c1Cl 22224,C(=O)(CC(F)(F)C(F)F)N1CCC(CNC(C2(C)CCNC(=O)C2)=O)(CO)CC1 22225,N1(C(c2c(SC)csc2)=O)CC2CCCC2(NC(C2OCCC2(C)C)=O)C1 22226,N1(C(c2ccc(SCC)nc2)=O)CCC(OC)C(C)C1 22227,Cc1cn(C(C)(C)C(=O)NCC(=C2CN(C(c3cc(C(N)=O)[nH]n3)=O)C2)F)cn1 22228,C(C(=O)NC1CCC(NC(C2(N3CCCC3)CC2)=O)CC1)(C(C)(C)C)NC(C)=O 22229,C1(CNC(C(CCC)OC)=O)CC2(CCOCC2)CN1C(=O)CSSC 22230,S(=O)(=O)(CC(=O)NC1(C)CC(C(=O)NC2CC23CCC3)C1)NCC 22231,N1(C(C(C)NC(=O)NC)=O)CCN(C(=O)C(C)=C(C)C)CC1CC1CC1 22232,Cc1cc(NC(=O)C(C)O)ccc1NC(c1ncsc1Br)=O 22233,N1(C(c2c(CC)oc(C)c2)=O)CC(Nc2ncncc2Br)CC(F)C1 22234,C(=O)(C(C)S(C)(=O)=O)NCCN1CCN(C(c2c(OCC#C)nccc2)=O)CC1 22235,c1(C(N2CCN(C(C3C(C)(CC)C3)=O)CC2)=O)c(F)ccnc1Cl 22236,C1(S(N)(=O)=O)(C(=O)NCC(C)N(C)C(c2cc(Cl)cn2C)=O)CCC1 22237,c1(C(=O)NCC2CC(F)CN2C(C2CCCC23CC3)=O)cnn2cnnc2c1 22238,Cc1nc(CCNC(c2cccnc2-n2nccn2)=O)c(C)o1 22239,c1(CCC)c(C(N2CCN(CCOCCC(C)C)CC2)=O)nnn1CC 22240,C1(N(C)C(C2CCOC2)=O)CCCN(C(c2cc(O)ccc2Br)=O)CC1 22241,C(=O)(C(O)CCC(F)(F)F)N1C(CN(C(=O)Cc2ncc(C)s2)CC)CCC1 22242,C1(NC(C2OCCC(C)(C)C2)=O)CN(C(=O)CC2CCC(C)(C)C2)CC12CCC2 22243,N(C1CCCc2ccoc21)C(CC1C(NC(C(C)(C)CCC#N)=O)CCC1)=O 22244,CC(C)C(CC(=O)N1CC(N(C)C)C1)NC(C1CCC2(CCC2)O1)=O 22245,C1(NC(CC(CCC)O)=O)CCCCN(C(c2cccc3cnsc23)=O)CC1 22246,c1(-c2nn(C(C)C3CC3)c(C(OC(F)(F)F)F)n2)ccc(F)c(Cl)c1 22247,C1(CCNC(Cn2ccc(C)n2)=O)CCN(C(C2CC2C(C)(F)F)=O)CC1 22248,C1(C(=O)NC(c2cc[nH]n2)C)CC2CCCC2N1C(C1CC12CCCC2)=O 22249,N1(C(c2cc(CCC)on2)=O)CC2CCN(C(c3cncc(O)c3)=O)CC(C2)C1 22250,C1(NC(CCC(N)=O)=O)CC2(CCN(C(c3cncc(OC(F)F)c3)=O)CC2)C1 22251,c1(CC(=O)NCC(C)CNC(=O)Cn2cnc(C#N)n2)cc(F)ccc1F 22252,c1(N2CCC(C)C(CO)C2)nc2cc[nH]c2c(=NCC2CSC2)[nH]1 22253,N1(CC(=O)NCC2CCN(C(C3C4CCC3CC4)=O)C2)CCN(C2CC2)C1=O 22254,CC#CC1CCN(C(=O)CC2CCCC2NC(=O)C(O)C(C)(C)C)CC1 22255,C1(CNc2ccccc2)CCN(c2ccnc(NCc3ccc(Cl)o3)n2)CC1 22256,N1(C(C(C2CC2)OCC)=O)CCC(C)(NC(=O)Cc2ccn(C3CCCC3)n2)C1 22257,c1(OC)cccc(F)c1C(=O)NCC1CN(C(=O)Cc2csc(C)n2)CCC1C 22258,C(=O)(C(O)CC(F)(F)F)NCC1N(C(CSc2nc(C)[nH]n2)=O)CCCC1 22259,C1(CCCNC(c2c(CC)noc2)=O)CCCCN1C(=O)C=CC1CCOCC1 22260,n1(CC)nnc(C(=O)NC2CC(CNC(c3cc[nH]c3)=O)C2(C)C)c1C 22261,C1(C(N2CCCC(CC3CC3)C2)=O)(CC)CCN(C(C2CCCS(=O)(=O)C2)=O)CC1 22262,Cc1c(C(N2CCOC(C(=O)NCCC3OCCC3C)C2)=O)cnn1C 22263,C1(NC(C(C)n2cnnn2)=O)CCCCCN(C(c2cn3ccnc3cn2)=O)C1 22264,c1(OC)ccc(C=CC(=O)NC2CCCCC2CNC(C2CC2C)=O)c(OC)c1 22265,Cc1cc(NC(=O)NC2CC2(F)F)cc(F)c1Br 22266,Clc1cc2c(cc1-c1cc[nH]n1)CCCC2 22267,c1(Nc2ccc(OC)cc2CS(C)(=O)=O)cccc2c(Cl)c(Cl)oc12 22268,c1(C(C(=O)NCC(=C)C)N(CCC(C)(C)C)CCCC)ccnc(Br)c1 22269,N1(C(C2C(=C)CC2)=O)CC(CNC(c2ncccc2C(=O)OC)=O)C(O)C1 22270,C1(CC=C)(NC(C2CCCN2C(C)C)=O)CCCN(C(c2cc(OC)cs2)=O)C1 22271,C12(CNC(CN(C)C(c3ccccc3)=O)=O)CC1CN(C(C1CC1C(N)=O)=O)C2 22272,Nc1cc(C(=O)NCC(c2cccc(Cl)c2)NC(c2csnc2Cl)=O)cc(F)c1 22273,N1(C(c2c(CC)c[nH]n2)=O)CCN(C(c2cnc(C)cn2)=O)CC1CCOC 22274,CCC(CCC(=O)N(C(C)CC(N)=O)C)NC(C1(C)CCCCC1)=O 22275,C#Cc1cccc(C(=O)NCC2COC(CNC(=O)C(C)(C)c3ccsc3)C2)c1 22276,C1(C(=O)NC(C(N2CCC(O)(CC(N)=O)C2)=O)CCOCCO)CCC(N=[N+]=[N-])C1 22277,CCCCC(CNC(=O)C(C)(C)NC(=O)C1CC1)OC.C12=CC(=O)N(CC1)CC2 22278,c1(OC)cc(C(N2CCN(C(C3CCCCN3C(C)=O)=O)CC2C)=O)cnc1C 22279,c1(CNC(C2(C(C)NC(CCOC(C)=O)=O)CC2)=O)n[nH]cc1C 22280,N1(C(COC(C)C)=O)CCC(C(C)(C)C)(CNC(=O)C(C)Cc2ccncc2)C1 22281,c1(-c2c(F)cc(C)cc2F)ccc2c(C(=O)NCC(C)(C)C(N)=O)nn(C)c2c1 22282,c1(C(N(C(CNC(c2ccc(C(OC)OC)o2)=O)C)C)=O)occ2c1CCOC2 22283,COn1cnc(C)c1C(=O)NCC1CCC1C(=O)NCC1CCCC2(CC2)C1 22284,c1(C(N(CC(C)NC(CN(CCC)C)=O)C)=O)cn2cccc(Br)c2n1 22285,c1(C(N2C(CN(C(CCCC)=O)C)CCCC2)=O)cnc(C2CC2)[nH]c1=N 22286,Cc1cc(C(=O)NC2CC(C(=O)NCCC(C)(C)CO)C2(C)C)c(C)s1 22287,CC(CN(C)C)C(=O)NCCn1ccc(C(=O)NCC(C)CN(C)C)c1 22288,C(=O)(CS(=O)(=O)C(C)C)N1CCC(N(C(=O)CCn2ccnc2C)CC#C)CC1 22289,c1(NCC2(C(C)C)CC2)[nH]c(=NC2CC3(C2)CC3(C)C)nc2c1cnn2C 22290,N1(C(c2ccn(C3CC3)n2)C(=O)NCC)CCc2c(cc(C#N)n2C)C1 22291,C1(CC(=O)NCC(C)(CO)NC(=O)C=CC2CCCO2)CCCCCCC1 22292,CC(c1ccc(F)cc1)=CC(N1CC(NC(c2c[nH]nc2[N+](=O)[O-])=O)C(C)C1)=O 22293,N1(C(COC(C)=O)=O)CCCC2CN(C(c3cc([N+](=O)[O-])oc3C)=O)CCC12 22294,C(=O)(C1=CC2CCCC12)NC1CCC(NC(CSCCC(C)C)=O)C1 22295,C1(C(N(C)CCOCCN(C(=O)C(F)(F)c2cscn2)C)=O)CCCC(F)C1 22296,CC1CC(C2CN(C(C3CCC3NC(c3ccnnc3)=O)=O)C2)=NO1 22297,C1(n2ccc(C)n2)CCC(N=c2cc[nH]cc2S(=O)(=O)NCC=CCl)C1 22298,N1(C(C(CC)=O)=O)CCC2CN(S(=O)(=O)c3ccccc3F)CC2CC1 22299,CC1(c2cccc(CNC(=O)NCc3ncccn3)c2)NC(=O)NC1=O 22300,c1(OC)nc(Cl)ccc1C(=O)NCC1CN(C(c2cc3sccc3s2)=O)CC1O 22301,c1(OC)c[nH]nc1C(=O)NC(CN(C(=O)CC1C=CCC1)C)Cc1ccccc1 22302,N1(C(C(C2CCCCC2)NC(c2cn(C)c(=O)cc2)=O)=O)CC2(C)CC1CCO2 22303,Cc1cnccc1C(C)C(N1CC(NC(=O)CCc2cncnc2)CC1C)=O 22304,CC1(F)CN(C(C2CCCSC2)=O)CCN(c2nc3cc(Br)ccc3o2)C1 22305,N1(C(C(C)C2CCCO2)=O)C(CNC(c2n[nH]cc2Cl)=O)CC2COCC12 22306,c1(C(=O)NC(CC=C)(C)C(C)C)n[nH]c2c1CN(C(c1nnn(C)c1CC)=O)C2 22307,N1(C(CN(C(C)C)C)=O)CCC2(CC2NC(=O)COC2CCCCCC2)C1 22308,CC1(C)CC(O)CCN(C(C2C3CC(O)C(C3)N2C(=O)CSC(F)(F)F)=O)C1 22309,c1(C(C(=O)NCCN(C(=O)C=C(C)C(F)F)C)NC(COC)=O)ccccc1 22310,c1(OCC(=O)NC2CN(C(=O)C(F)F)CC2C(F)F)ccc(C2CCC2)cc1 22311,CC1CCN(C(=O)CC23COC(CF)(C2)C3)CCN1C(=O)Cc1ccc(Cl)nc1 22312,N1(C(C(C)N(C(=O)CC2OCCO2)C2CC2)=O)CC(CO)C(O)C1 22313,C1(CC)CN(C(=O)Cn2ccsc2=N)CCC1NC(c1ccnc(O)c1)=O 22314,n1(CC)c(C(=O)NCC2CC3CCC2N3C(C2(SC)CC2)=O)cc2ccccc12 22315,Cc1c(C(N2CC3CN(C(=O)CCC(C)(C)C)C3C2)=O)cccc1O 22316,c1(C(=O)NC2C(C)CN(C(=O)C(F)(F)CC3CCCO3)C2)c(N)cccc1Cl 22317,CCCCC(C(=O)NCC1CC(C)=NO1)NC(=O)Cc1cnns1 22318,C1(C(c2ccccc2)NC(C)C(=O)NCc2ccccc2)(OC)CC(C)(C)C1 22319,CCC(C)CC(C)C(=O)N(C)CCN(C(c1nn(C(F)F)cc1Cl)=O)C(C)C 22320,N1(C(Cc2cccc(OC)n2)=O)CCC(C)(C)C(NC(c2ccc(F)cn2)=O)C1 22321,c1(CN(C2COC(C)(C)O2)C(c2ccc(CO)o2)=O)ccc(Cl)cc1F 22322,Cc1ccc(C)c(CNC(C2CC(O)(CNC(=O)C(O)Cc3cnc[nH]3)C2)=O)n1 22323,CC(C(C)C(=O)N1CCOCC1C(C)O)NC(=O)C(C)CC1CCCC1 22324,Cc1cc(C(=O)NC(CNC(C2(S(C)(=O)=O)CCCC2)=O)C2CC2)ncc1C#N 22325,c1(C(c2n(C)nnn2)NC2CCCN(O)C2=O)nc2c([nH]1)CCCC2 22326,Cc1cc(NC(=O)C(C2CCOCC2)O)ccc1NC(=O)C(C1CC1)N(C)C 22327,C1(C(=O)NCC(C)(C)OCCNC(C(C)Cn2ccnc2)=O)NC(=O)OC1C 22328,N1(C(Cn2cc(C(C)O)nn2)=O)CC(NC(c2cccn2C)=O)C2CCCC12 22329,C=CCC(CNC(=O)C(C)OCC1CC1)C(=O)NC1(CO)CC2CCCC12 22330,N1(C(C2CCN(CC)CC2)=O)CCC2(CC1)CC(N1CCC(F)(F)CC1)C2 22331,c1(C(=O)OC)cc(C(=O)NC2CC(C)(NC(c3sc(CO)nc3C)=O)C2)c(C)o1 22332,C(C(F)(F)CNC(=O)CCCNC(=O)CC1(C)CC1)OC 22333,c1(C(N(CCC(C)NC(=O)C(=Cc2c[nH]cn2)F)C)=O)cc2scc(Cl)c2[nH]1 22334,CC(C)C(C)C(CNC(c1cccc(C2(F)COC2)c1)=O)NC(=O)C1=COCC1 22335,OC1(F)CCN(N2CCOC3(CCSCC3)C2)C1c1ccccc1 22336,C1(NC(C2CSC2)=O)COCCN(C(c2ccnc(C(F)(F)F)c2F)=O)C1 22337,c1(OC)cc(C)c(C(=O)NC(CNC(=O)Cc2cnccc2C)C2CC2)c(C)c1 22338,Cc1nn(C)c(C)c1C(N1CCCC(C(=O)NC2CC(=O)N(C)C2)CC1)=O 22339,Cc1cc(CC(=O)NCC(C)(CO)NC(=O)CNC(=O)CCCCl)n[nH]1 22340,N1(C(C=C(C)C)=O)Cc2occ(C(N3CCC3CC3CC3)=O)c2C1 22341,c1(N2CC(C)(NC(C(C(C)O)C)=O)C2)nc2cc(Cl)cc(Cl)c2o1 22342,CC(C)(CO)C(=O)N1CCC(CCC(N2CCC(O)C2)=O)C1 22343,N1(C(=O)CCc2sccc2Br)CCN(c2ccc(-c3ccsc3CO)cc2)CC1 22344,CC1CN(C(c2ccc(OCC(N)=O)cc2)=O)CC1NC(=O)CCC1CC1(Cl)Cl 22345,Cc1ncnc(O)c1CCC(=O)NC(C1CN(C(C2CCCN2C(N)=O)=O)C1)C 22346,c1(NC(c2c(Cl)ccc(OC)c2)=O)ccc(S(C)(=O)=O)cc1Cl 22347,n1(CC(=O)NCC2CC2CNC(c2c[nH]c(C(F)(F)F)c2)=O)cccnc1=O 22348,C12(C(=O)NCC(CCC)NC(C3C4CN(C)CC34)=O)CC(C#N)(C1)C2 22349,c1(CC=CCNC(c2nnn(C)n2)=O)ccc(O)c(Cl)n1.C(CCN)NC=O 22350,C(=O)(C(C(C)C)C(C)C)N(C)CC1(C)C(NC(C(C(CC)O)C)=O)CCC1 22351,N1(C(c2cncc(COC)c2)=O)CC2CC(NC(c3c(C)nn(C)c3C)=O)C2C1 22352,c1(C(=O)NCC(C2CC2)NC(C(OC)OC)=O)ccc2cccnn12 22353,C1(C(=O)NC2(CO)CCCN(C(=O)CCCC3CC3)C2)(OC)CCS(=O)(=O)C1 22354,N1(C(CCC(C)O)=O)CC(NC(c2coc(C3CCOCC3)n2)=O)CC2(CC2)C1 22355,N1(C(c2cn(CC)nc2C)=O)CC(NC(=O)Cc2ccns2)C(N=[N+]=[N-])C1 22356,Cc1ncnc(N2CC3CC3(CNC(c3cc(F)ccc3Cl)=O)C2)c1Br 22357,C(c1cnc(C)s1)=CC(=O)NCC1(CNC(C(C=CCCC)O)=O)CC1(F)F 22358,CC(=Cn1ccnn1)C(=O)N1CC(C)N(C(c2ccn3ccsc23)=O)CC1C 22359,c1(NC(c2ccsc2)CC)ccc(S(=O)(=O)NC2(C)CC2)cc1Br 22360,Cc1nn(C)c(C)c1C(=O)NCCC(C)NC(=O)C(=O)C(C)(C)C 22361,C1(NC(CCCNC)=O)CCCC(NC(c2ncncc2OC)=O)CC1 22362,N1(C(C(CC=C)(F)F)=O)CCC2C(COC2CC(=O)N(CC(F)F)C)C1 22363,C1(O)(CNC(C2(C(=O)NC)CC2)=O)CCN(C(=O)CN2CC3CC3C2)CC1 22364,CC1OC2(C(=O)NCC3CC4CC4N3C(=O)Cn3cnnc3O)CC1C2 22365,c1(CC)nnc(N(CCCNC(c2ccc3c(c2)COC3)=O)C)c(C#N)c1CC 22366,N1(C(C=C(C)Cl)=O)CC2C(NC(=O)CCSc3ccccn3)C2C1 22367,C=CC(C)(C)CC(=O)N(C1CCCN(C(=O)CC2CCC(C3CC3)O2)C1)C 22368,Cc1c(C(N2CC3CC2C3C(=O)NCC2(O)CCN(C)C2)=O)cccc1F 22369,N1(C(c2c(C)nc(C(C)C)s2)=O)CC(NC(c2ccnc(CO)c2)=O)C2CC2C1 22370,C=CCC(CC(=O)NC(CCC)c1nn[nH]n1)NC(=O)CCCF 22371,C(=O)(CS(=O)(=O)N(C)C)NCCOCCN(C(=O)C(F)(F)c1cncs1)C 22372,N1(C(CCN(C(Cn2cnc(C#N)n2)=O)CC2CC2)=O)CCC(O)C(F)(F)C1 22373,c1(C(=O)NCC2CC(NC(c3cccnn3)=O)C2)cnc(S)nc1 22374,C12(CNC(COCC#C)=O)CCC(CC1)N2C(C1(C)CNC(=O)C1)=O 22375,n1(CCC)c(C)cc(C=CC(=O)Nc2c(CC#N)cc(CO)cc2I)c1C 22376,N1(C(=O)C=CC=Cc2ccccc2)CCC(CNC(C2COC(=O)C2)=O)C(O)C1 22377,c1(C(=O)NC2CC(NC(=O)CNC(c3ccsc3)=O)C2)ccc2c[nH]nc2c1 22378,N1(CCN2CC(OC(C)(C)C)CC(OC)C2)CC2C(C(F)(F)F)(C1)CS2(=O)=O 22379,N1(C(C)=O)CCC(CC(=O)NCCCCN(C(=O)CC2CCN(C)C2)C)CC1 22380,N1(C(C(F)=CC)=O)CCC(NC(=O)CC2CCCN2CC)C1 22381,c1(CC(=O)NCC2C(NC(c3cnc(C)[nH]3)=O)C2)ccc2c(c1)OCCO2 22382,C1(C(N2C(C(N)=O)CC2)=O)C=CCN(C(=O)CC2OCCCO2)C1 22383,C(=O)(C(C(C)(C)O)NC(c1cccn(C)c1=O)=O)NC(C(=O)OC)CO 22384,c1(N2CCCC3(CC(NC(=O)C4CCCc5n[nH]cc54)C3)C2)nc2ncc(Cl)cc2s1 22385,N#Cc1cc(F)ccc1C(N1CCN(C(C2CCSCC2)=O)C2CC12)=O 22386,Cc1ccc(CC(N2CCCC(O)(CNC(=O)C(C(C)O)N(C)C)C2)=O)cc1C 22387,N1(C(c2c(C)ccnn2)=O)CCN(C(=O)C(C)(F)C(C)(C)F)CC12CCC2 22388,C(=O)(CCC(CC)OC)NC(CC#C)C(=O)NCCC1CCOCC1 22389,n1(CC)cc(CC(=O)NC(C(=O)NC(C)CC2CCC2)C2CCOC2)cn1 22390,CC(C1CCCCC1)=CC(=O)NC1CN(C(=O)CCOC2CC2)CCC1C 22391,c1(C(=O)NC2CCC(CNC(C(n3ccc(C)n3)(C)C)=O)C2)cccn(C)c1=O 22392,C(=O)(C(C(=O)NC1CC2(C(=O)NC3CCOCC3C)COC1C2)C(C)C)OCC 22393,n1(CC(=O)NC2CCC(NC(C(CC)O)=O)C2)nc(-c2ccccc2)oc1=O 22394,c1(CNC(c2cnc(S)nc2)=O)ccc(C(=O)NCCC(O)CCO)cc1 22395,c1(C(=O)NC2CC(C(=O)NC3(CCC)CCNC3=O)OCC2)ccc2n[nH]cc2c1 22396,N1(C(C(CC#C)(C)NC(=O)CCC#CC)=O)CC2(CNC(=O)C2)C1 22397,N1(C(C=C(C)C(C)C)=O)CCC(O)(C(C)NC(=O)CCOC(C)CC(C)C)CC1 22398,C1(C(=O)NC(CC)C(C)(F)F)CN(C(=O)C(C)O)CC1C1CC1 22399,c1(C(=O)NC2(C)CC(NC(=O)CC3COC4CC3C4)C2)cc([N+](=O)[O-])ccc1Cl 22400,C(C(C)(C)C(=O)NCCC(C)CCNC(=O)C=C1CCCC1)OCC 22401,CC1(C)CN(C(=O)C=CC=CCO)CC(CNC(=O)CC2CC3(CCC3)C2)O1 22402,Cc1ncc(Cl)c(C(N2CC3C(CNC(=O)C(C)(C)O)C3C2)=O)n1 22403,N1(C(C2(F)CCN(C(C(CC=C)N(C(C)=O)CC)=O)CC2)=O)CC(C)N(C)CC1C 22404,c1(C(N2CC(C(=O)NCCc3ccc(OC)nc3)SCC2)=O)cccc(C#N)c1 22405,c12cc(c(C)o1)S(=O)(=O)NC2=O.N1(CCC)C(=O)CCC1C(=O)NC 22406,C(=O)(C1=NN2CCCN=C2N1)NCC1CN(C(CSC(C)C)=O)CC1(C)C 22407,C1(CNC(C(CC)(C)C)=O)C(O)C(O)CN1C(=O)C=Cc1ccnn1C 22408,c1(CC)nn(C)c(NC(C2C3CN(C(=O)CCS(=O)(=O)N(C)C)CC23)=O)c1Cl 22409,c1(C(=O)NC2C3CN(C(C4(CF)CC4(F)F)=O)CC23)cccc2cnccc12 22410,C1(C2CC2)(C(=O)NC2C(C=C)COC2)CN(C(=O)CC23CCC(CC2)C3)C1 22411,C1(CC)CCc2nnc(NC(c3ccccc3C(F)(F)F)c3nnnn3C)n2C1 22412,N1(C(CNC(C(C)(C)C)=O)=O)CCC2CCCC12C(N1CCCC(C)(CO)C1)=O 22413,Cc1nsc(C(=O)NC2(CF)CN(C(=O)CCc3ccccc3)C2)c1N 22414,C1(CCCNC(=O)CSc2cccnc2)CCCCN1C(c1cccnc1)=O 22415,c1(CC(N2CCC(N(C(CC(CC)OC)=O)C)C2)=O)c(F)cccc1Cl 22416,C1(C(C(=O)N(C)CCN2CC=CC2)(C)C)CCCN(C(=O)C=CC2CCC2)C1 22417,CC1CN(C(C2(c3ccccc3Br)CCC2)=O)CCN1C(=O)CC1C=CCCC1 22418,C1(C)(C(=O)NCC(C)(C2CCC2)NC(Cn2ncc(C)c2)=O)COCCO1 22419,C(CNC(C1(CC2CC2)CCC1)=O)(CC(=O)N1CCC1(C)C(C)C)OC 22420,N1(C(C(CC)OC)=O)CCOC(C(=O)NCC2(F)CC(CO)C2)CC1 22421,CCC(C(=O)OC)C(=O)NC1CC=C(C(=O)NCCc2nc(C)no2)C1 22422,c1(NC(CC(=O)N2CCOCC2)c2ccccc2)ncnc2[nH]cc(Cl)c12 22423,Cc1ccc2c(C(=O)NCC3CC3NC(c3cc(N(C)C)ccn3)=O)n[nH]c2c1 22424,C1(COC)(CNC(=O)CC(C)O)CCN(C(=O)Cc2ncccc2C)C1 22425,c1(C(=O)NCCC2(O)CN(C(C34CCCC3CC4)=O)C2)cnc2n1CCOC2 22426,S(=O)(=O)(CCN=c1ccnc(NCC(c2nc(C)cs2)(C)C)[nH]1)NCC 22427,N1(C(C(C)C)=O)CCCC(NC(=O)CC(c2ccc(C(F)(F)F)cc2)C)C1 22428,C(=O)(C1=C2CCCN=C2NN1)N1C2C(NC(c3n[nH]c(C)c3C)=O)CC(CC2)C1 22429,c1(OCOC)cccc(C(=O)NC(C)CNC(=O)C(F)C(C)C)c1 22430,Cn1cc(C(N2CCC(CNC(=O)Cc3cscn3)C2)=O)nc1C(F)F 22431,N1(C(CCOCCOC)=O)CCCC1C1(CNC(=O)C(N2CCC(C)C2)=O)CC1 22432,c1(C(=O)NC(CNC(C(C(CC)C)O)=O)CC(F)(F)F)ccc2cccnc2c1 22433,C(=O)(C1=C(Cl)CCC(C)C1)N1CCC(CC(=O)NC2(C(=O)NC)CC2)C1 22434,C1(NC(CC2CN(C)C2)=O)CCCC(NC(=O)C=Cc2cccc(F)c2)CC1 22435,c1(CC)nc(=N)[nH]c(=NC2C3CC2CN(C(=O)C(C)(C)CC2CCOCC2)C3)[nH]1 22436,CC(C(=O)N1CCC(C(CO)NC(=O)C(C)(F)c2ccon2)CC1)S(N)(=O)=O 22437,N1(C(c2cn(CC)nn2)=O)CC2(CCC2NC(=O)CC2CC3(CC3)CO2)C1 22438,Cc1ccc(C2(C(N3CCC(NC(C4CC4C#N)=O)C3)=O)CCOCC2)cc1 22439,C(=O)(C(CC(F)F)c1ccccc1)NC(C(C)NC(c1n(CC)ncc1)=O)(C)C 22440,CC1=C(C(=O)N(CC(=O)NC2N(C)CCCC2(C)C)C(C)(C)C)C(=O)OC1(C)C 22441,CC1CC(NC(C2COCCN2CC(F)F)=O)CCN1C(=O)Cn1cncn1 22442,C1(NC(CCOCC)=O)CN(C(=O)C=CC2CCOC2)CC12CC2 22443,c1(CC)c(C(=O)NC(CNC(=O)CC(C)C(F)F)CO)cccc1C 22444,c1(C(=O)NC2CC3CC(NC(CCCOC)=O)CC3C2)ccc2c(c1)ncn2C 22445,CC1OC2(C(=O)NCC3CN(C(=O)CCNC(N)=O)CC(C)(C)O3)CCC1CC2 22446,c1(C(N(C(CNC(C2C(OC)C2)=O)C)C)=O)ccc(-c2ccccc2)[nH]1 22447,N1(CC)CCC(N(C2CCOCC2OC)C(=O)NC2CC2C)C1=O 22448,C12(NC(COC(C)=O)=O)CCCC(NC(=O)Cc3nccn3C)(C1)C2 22449,C(C)(C(O)C(=O)NCC(C)(C)NC(=O)CNS(=O)(=O)Cc1ccon1)OC 22450,C(=O)(C#CC(C)(C)C)NCCNC(CC(C)c1ccncc1)=O 22451,N1(C(CSC)=O)CCC2(NC(=O)CC3CCCC3C)CCCC12 22452,N1(C(C2(C)CC(C)C2)=O)CCC(C2(O)CN(C(C3C4COCC34)=O)C2)CC1 22453,c1(CC)cc(F)ccc1CC(=O)NC(C)C(C)(C)NC(c1sccc1C#N)=O 22454,C1(NC(=O)CC2=CCCC2)CCC2(CCCN2C(C2COC2)=O)CC1 22455,c1(CSc2nc3ccc(C(=O)OC)cc3o2)nc2ccc(Br)cc2n1C 22456,C1(F)(C(=O)NCC2C(NC(=O)Cc3sc(O)nc3O)C2)CS(=O)(=O)CC12CCC2 22457,c1(C(=O)NCCCN(C(c2c(SC)scc2)=O)C2CC2)cn(C)nc1C(N)=O 22458,c1(OC)cccc(CC(C)(C)NCc2c[nH]nc2C(C)(F)F)c1 22459,n1(C(C)C)ccc(C(N2CCC2CNC(c2nc(Cl)cs2)=O)=O)n1 22460,N1(C(CCC#C)=O)CC(CCNC(c2ccnc(Cn3cnnc3)c2)=O)OC(C)C1 22461,C1(C(N2CC(C)(CO)C2)=O)C2CCC(C2)N1C(C1(C)CC(C#N)C1)=O 22462,N1(CCC)CCCCC1C(=O)NCC(CNC(c1cn(C2COC2)nn1)=O)CO 22463,Cc1[nH]ccc1C(=O)NCc1cn(CC(N2CCC2CN(C)C)=O)nn1 22464,N1(C(C2N(CC)CC2)=O)CCC(NC(c2cnn(C3CC3)c2Cl)=O)C(F)C1 22465,C1(OC)CCN(C(c2n[nH]cc2CNC(=O)C(C)OC2CCCC2)=O)C(C)C1 22466,c1(C(=O)NCC2(F)CC(CNC(C3CCN(CC)CC3)=O)C2)nccc(C)c1F 22467,Cc1cc(C)[nH]c(=NCC2(N(C)C(c3cccn4c(O)nnc34)=O)CC2)n1 22468,C1(CC(=O)NC(C(C)(C)NC(c2cncc(COC)c2)=O)C)NC(=O)CNC1=O 22469,CC(N=c1cc(C(C)(C)C)nc(Cl)[nH]1)C1CCCN(C(=O)C=Cc2nccs2)C1 22470,CCCCC(O)CC(=O)NCC1(Cc2cn(C(C)C(=O)O)nn2)CC(OC)C1 22471,n1(CC)cc(Cl)cc1C(=O)NC1(CNC(C23COCC(C2)C3)=O)CCCC1 22472,c1(C(N2CC3C(NC(c4c(OC)n[nH]c4)=O)C3C2)=O)cc(Br)cc2cc[nH]c12 22473,c1(CC(c2ccccc2)N2CCOCC2)cc(Cl)cs1.C12(COC1)CNC(=O)N2 22474,CCS(=O)c1ccccc1C(N1CCN(C(c2cc(C)cs2)=O)CC1)=O 22475,C(C)(C(C(=O)NCCN(C)C1CC1)NC(c1nc(C)oc1C)=O)OC 22476,N1(C(C)C)CCC(C(=O)NC2C3CC(NC(=O)C4=C(Cl)CC4)CC23)CC1 22477,Cc1ccc2c(c1)C(C(=O)N(CCCN(C)C(C1CCCSC1)=O)C)C2 22478,N1(C(C2CC(C)(C)C2)=O)CC(CNC(=O)CC2=CCCCC2)C2(CCOCC2)C1 22479,c1(OCC)ccc(NC(C2=CCSC2)c2nnnn2CC2CCCO2)cc1CO 22480,N1(C(C(CC)(C)C)=O)CCC(NC(=O)Cc2cc(Cl)ccc2O)C(C)C1 22481,c1(C(=O)NCC(C)NC(c2c(C)nn(C3CC3)c2)=O)cnn2c(N)ccnc12 22482,C(=O)(C(=O)C(C)(C)C)N(C(C(=O)Nc1ccsc1)C1CC1c1cccc(I)c1)C 22483,N1(C(=O)CN2CCOCC2)CCCC(CCC(=O)NCC23CC(CO)(CO2)C3)C1 22484,c1(CCC(=O)NCC2(OC)CN(C(=O)C(C)CO)C2)ccc(C#N)cc1 22485,C(C(CC(C)C)C(=O)N(C(C)CN(C)C(c1cnc(Cl)n1C)=O)C)OC 22486,Cc1cc(N2CCC(C(C)NC(C3CCCC(O)C3)=O)C2)c(Br)cc1[N+](=O)[O-] 22487,c1(C(=O)NC2CCC(NC(=O)C3=CCSC3)C2)c(Cl)ccc(Br)c1F 22488,C12(NC(CN(C)C)=O)CCCCCC1N(C(c1coc(Br)n1)=O)CC2 22489,Cc1cnn(C)c1C(=O)N(C(C)(C(=O)N1CCC(C(N)=O)C1)C1CC1)C 22490,C1(CN(C(C(C2CC2)OC)=O)C)CCCN(C(=O)CCCOC(C)(C)C)C1 22491,CC1(C)CC(NC(=O)C2=NOCC2)CN(C(c2ccnn2CC#N)=O)C1 22492,c1(OC)cc(CN(CC(C)(C)C2(O)CNC2)C=O)cc(F)c1 22493,c1(-c2c(C)c(N3CCn4c(C)cnc4C3)ncn2)cccc2c1OCCO2 22494,CC(C)(O)CC(=O)NCCn1ccc(C(=O)NCC2(CC3CC3)CCC2)c1 22495,Cc1cc2nc[nH]c(=NCCOCCNC(c3cscc3Cl)=O)c2[nH]1 22496,N1(C(c2cccc(OC)n2)=O)CCC(F)CC1C(=O)NCC1CC(C)(C)CCO1 22497,C1(NC(C(=O)NC(c2ccccc2)CC=C)=O)CCCCC1N1CCOCC1 22498,N1(C(C2CC3(CC(NC(C(CC(C)(C)C)OC)=O)C3)C2)=O)CCC2(CCC(O)C2)C1 22499,C1(NC(C(c2ccc(F)cc2)C)=O)C2CC(CN(C(=O)C=C3CCC3)C2)C1CO 22500,N1(C(c2ccc(NC(C)=O)cn2)=O)CCCC(NC(=O)C(F)(F)CC2CC2)C1C 22501,C(=O)(C(C)CC(F)F)N1CC(CCNC(c2c(C)[nH]c(=N)s2)=O)C1 22502,C(=O)(C(C)CC(C)(F)F)NC(CCNC(CCc1ccc(OC)cc1)=O)C(C)C 22503,C(CCCC(C)C)N(C(CCC1N(C(c2c(C)scn2)=O)CCC1)=O)C 22504,C1(C(N2CCC(OCCO)C2)=O)(CNC(C2N(C)CCC2)=O)CCCCC1 22505,c1(CC(C)NC(=O)Nc2cncc(C(C)(C)C)c2)nc2ccccc2s1 22506,N1(C(c2c(C)cc(SC)o2)=O)CC(NC(=O)Cc2coc(C)n2)CC1(C)C 22507,C1(COC)(NC(C2CCC(C(F)(F)F)C2)=O)CN(C(=O)Cn2cnnn2)C1 22508,c1(CNC(C(C2CCN(C(=O)CCOCC(F)F)CC2)C)=O)ccc(O)c(O)c1 22509,c1(C(=O)NCC=C)cccc(C(=O)NCC(CC(C)C)NC(=O)C(=O)NCC)c1 22510,N=c1ncn(CC(=O)NC(CC2CC2)C(=O)NCCC2CC(F)C2)[nH]1 22511,C1(NC(C2(N(C)C)CCCC2)=O)CN(C(=O)CC2CCC23CCC3)CC1C(F)F 22512,c1(N2CCOCC(C)C2)ncnc2c1ncn2CC1CCC2(COC2)OC1 22513,CCC(CC)(CC)C(=O)N1CC(O)(c2cn(-c3ccc(C(C)(C)C)cc3)nn2)C1 22514,CCC(CC)CC(=O)NCC12CC1CN(C(=O)CC1(C)CC1(F)F)C2 22515,C12(C(N3CCC(C)(NC(C=C(C)Cl)=O)CC3)=O)CCOC1CC(=O)NC2 22516,C(=O)(C(COC)OCc1ccccc1)NC(CNC(C=CC(CC)=CC)=O)C 22517,c1(N2CCCC(C(C)C)C2)nc(=NC2CCCc3n[nH]cc32)[nH]c2c1COCC2 22518,c1(C(C)C)ncncc1C(=O)NCC1CC(NC(=O)CC(C)C2CC2)C1 22519,N1(C(CC2(N(C)C)CCC2)=O)CCOCC(NC(c2cc(Br)no2)=O)C1 22520,c1(C(N2C(C(=O)NCC3CCC(O)CC3)CC(O)C2)=O)ccc([N+](=O)[O-])o1 22521,C1(N(C(=O)C=CBr)C)CCCCN(C(=O)C(C)(C)c2ccno2)C1 22522,C1(CNC(C)=O)CCCN(C(C2(n3cc(CC(C)O)nn3)CC2)=O)C1 22523,c1(C(=O)NCC(C2CC2)NC(c2ccc(CC)[nH]2)=O)ccc(=O)n(CC(C)O)c1 22524,c1(CCC(=O)NCC2(C(=O)OC)CC2(F)F)cccc(F)c1Br 22525,C1(NC(C(=CC2CCCC2)C)=O)CN(C(=O)C(F)=CCCF)CCC12CCC2 22526,N1(C(Cc2c(C)n[nH]c2)=O)CC(CNC(=O)CCC2CCCO2)C(C)(C)C1 22527,C(=O)(CC(C)(C)C(=O)N1CC2C(CNC(C3CCS(=O)CC3)=O)C2C1)OCC 22528,O(NC(=O)C(CC(=C)C)NC(C1CCC2CC1CO2)=O)CC#C 22529,c1(NCC)ncc(C(=O)NC23CC(CNC(=O)C#CC(C)C)(C2)C3)cc1Cl 22530,c1(CC(=O)NCC23CC(NC(C(COC)N(C)C)=O)(C2)C3)c(O)ncnc1O 22531,c1(C(=O)NC2CN(C(CNC(=O)OCC)=O)CC(F)C2)csc2ccc(F)cc12 22532,CCCC(C)CC(=O)NC(C)C(C)NC(c1onc(OC)c1Br)=O 22533,c1(OCC)cccnc1C(=O)NCCC(C)N(C(=O)C=Cc1ccc[nH]1)C 22534,C1(C)(CNC(C(CC)O)=O)COCCN(C(c2cc(F)c(O)c(Cl)c2)=O)C1 22535,C(C(=O)N1CCCC1CC(=O)O)(C(C)C)N(C(=O)OC)C 22536,N1(C(CC2CC(C)C2)=O)CC2(CNC(c3cnn(C)c3Cl)=O)CC1CO2 22537,C=C(C)C(C)(C)C(=O)NCC1CCC1NC(=O)C(CO)N(C)C 22538,c1(C(=O)NCC(CO)NC(C(C2CC2)OC)=O)c[nH]c(=N)nc1C 22539,c1(C(=O)NC2(C)CC(C(N3CCCN(C(C)=O)CC3)=O)C2)cc2ccccn2c1 22540,CC(C)CC(O)C(=O)NC1(C(=O)NC2CCCCCC2C)CC1(C)C 22541,CC(CC(C)(C)C)C(F)C(=O)NCC1C2CN(C(=O)CCCn3ccnn3)CC12 22542,N=c1[nH]c2ccc(C(=O)NCC3(O)CN(C(=O)CC4CCCCC4F)C3)cc2[nH]1 22543,C=C(Cl)C(C)(C)C(=O)NC(C1CCCCN1C(=O)CN1CCC(C)(C)C1)C 22544,CCCCCC(O)C(=O)N1CC=CC1CNC(=O)CNC(C1CCC1)=O 22545,c1(C(C)OC(C2CC(CCC)C2)=O)ccc(Cl)nc1 22546,C(=O)(C1=CCCOC1)NCC1CCC(NC(CC(CC)c2ccccc2)=O)C1 22547,c1(C(C)(C)C)cncc(NC(C2CN(C(=O)C3CC3)CCN2)=O)c1 22548,C1(C(=O)NCC=CCCC)N(C(=O)Cn2nnc(C)n2)CCCC1(C)C 22549,c1(C(N2CC(C(Cn3cc(CNC)nn3)F)C2)=O)ccc2nc(Cl)nn2c1 22550,c1(C(=O)NC2(CCNC(C(CC)C(C)C)=O)CC2)ncnc2c1CCC2 22551,c1(-n2c(C(CC#C)C)nc(C(C)CCC)n2)ccc(S(=O)(=O)N(C)CC)cc1 22552,N1(C(CC2CCCC(OC)C2)=O)CC2CC3CC2C1C3NC(C1CC1C(N)=O)=O 22553,N1(C(c2n[nH]c(C)c2O)=O)CCC(C2CC2)(CNC(=O)COc2ccccc2)C1 22554,C1(C(=O)NC(COC)(C)C)CC(C)CN(C(c2cnc(SC)nc2)=O)C1 22555,N1(C(c2cnc(-c3cccs3)nc2)=O)CC2COC(C1)C2O 22556,N1(C(C(C2CCCN(C(C(CC#C)C3CC3)=O)C2)(C)C)=O)CCCSCC1C 22557,c1(C(N2CCC(O)(CCNC(CSCC=C)=O)C2)=O)cccc(C(N)=O)c1F 22558,c1(C(C)SCC)nc(-c2ccc(C(C)C)cn2)n(CC2CCSC2)n1 22559,C1(C)(CNC(CC2CC(SC)C2)=O)CCCN(C(=O)CC2CCCC2(F)F)C1 22560,N1(C(c2cnc(SC)s2)=O)CCC2CN(C(=O)CC(C)CF)C2C1 22561,C1(C(=O)Nc2cnc(I)cn2)CCN(Cc2ccc(OCCO)cc2)CC1O 22562,C(C(O)(C(F)(F)F)c1nccn1C)NC(=O)NC(C(C)F)C(=O)O 22563,N1(C(c2c(CCC)n[nH]c2)=O)CC=CC(NC(c2cnco2)=O)C1 22564,Cc1cc(C)n2ncc(C(N3CC(F)(C(N4CC5CCC(C4)N5C)=O)C3)=O)c2n1 22565,C(=O)(CS(=O)(=O)CC1CCCO1)NCC(C(C)(C)C)NC(=O)C=C1CCCC1 22566,c1(NC(=O)NCC2(C=C)CCOCC2)cncc2sccc12 22567,C(CCC)(C(=O)NC1(COC)CCN(C(=O)CCCc2ccncc2)C1)=CCC 22568,c1(-n2cc(OCC3CCCN(C(C(COCC)O)=O)C3)nn2)ccc(C)c(Cl)c1 22569,Cc1cc(C)n(CC(=O)NCCNC(c2cccc(CS(C)(=O)=O)c2)=O)n1 22570,C1(NC(c2ccc(NC(C)=O)s2)=O)CN(C(=O)COC2CCNCC2)CCC1O 22571,N1(C(CCc2ccc(OC)c(C)c2)=O)CC(C)N(C(C2(C)COC2)=O)CC1C 22572,O=C(C1=CCCCO1)Nc1cccc(CNC(C2CCN(C3COC3)C2)=O)c1 22573,N1(C(CC=CC)=O)CCC(C)(CC(=O)N(C(C2CCC2)C)CC)C1 22574,N1(C(c2ccn(CCNC(C3(CC)CCC3)=O)c2)=O)CC(S(N)(=O)=O)C1 22575,CC1(C(=O)NC2CCOC(CNC(=O)CCc3cccnc3Cl)C2)COCCO1 22576,N1(C(c2nn(CC)c(O)c2)=O)CC2CCCC2(CNC(=O)C2=NOC(C)C2)C1 22577,c1(NC(=O)NC(c2ccccn2)Cc2cccc(C)c2)cc(F)c(I)c(F)c1 22578,N1(C(C(C)(C)CC(F)F)=O)CC(NC(c2nccc(N)c2Cl)=O)CC2(CCC2)C1 22579,C(CN=c1[nH]cc2ccnc-2[nH]1)=CCNC(c1cc2sccc2[nH]1)=O 22580,C1(NC(C(CC)N(C)C)=O)CCN(C(C2CC(=O)NC2(C)C)=O)C12CCC2 22581,C1(N(C)C(C2C=CCS2)=O)CN(C(c2cc(Cl)c[nH]2)=O)CCC1O 22582,C1(N(C(=O)C(O)C2CN(C(C3CCCC3F)=O)C2)CC)CCCCC1 22583,CC(C)CCCC(C)CCNC(=O)N(C(C)(C)C)Cc1ccc(Cl)cc1 22584,c1(C(=O)NCCC2(O)CCN(C(=O)CSC(F)F)C2)cnn2ncccc12 22585,C(=O)(C(C)(O)COC)NCCC1(NC(c2ccc(CC)[nH]2)=O)CC1 22586,c1(C(N(CCCNC(=O)C(C)C(F)F)CC)=O)cc2c(cc1N)CCCC2 22587,C1(C(N(CC(O)C2CCC2)C)=O)CCC(NC(=O)C(C2(O)CCCC2)F)C1 22588,Cc1cc(NC(=O)C(C)CNC(=O)Cc2cnccc2C)c(C)c(C)c1 22589,N1(C(C2(C)CCCO2)=O)CCOC2(CCN(C(c3cc(C4(C)CC4)n[nH]3)=O)C2)C1 22590,C1(C(=O)NCC=C2CCSCC2)(NC(C(c2cncnc2)C)=O)CC(O)C1 22591,O=C(CC(F)(F)F)NCC1(CNC(=O)CCCOCCc2ccccc2)CC1 22592,c1(C(N2C(C(=O)Nc3nnc(C)o3)CC2)=O)c(C)[nH]c2ccccc12 22593,c1(C(N(CC(C)CNC(C23CCCC(CO2)C3)=O)C)=O)cc(O)c(O)c(O)c1 22594,C1(C(N2CC(NC(CN(C(C)=O)C)=O)(CO)C2)=O)CCC(=O)N1C 22595,c1(C(=O)NC2(CCNC(=O)Cc3csc(-c4cccs4)n3)CC2)ncc[nH]c1=O 22596,C1(NC(c2nccc(CC)c2)=O)CC2CC1N(C(c1ccc(F)c(N)c1)=O)C2 22597,c1(C(=O)NCc2sc(Cl)nc2Cl)ccc(=O)n(Cc2ccccc2Cl)c1 22598,C=CCC(CNC(=O)CC1(C#N)CC1)C(=O)NC(C)Cc1nncn1C 22599,C(=O)(C1=CC2(CCOCC2)C1)NCC(C)CN(C(=O)C(CO)C(C)(C)C)C 22600,C(C(C)(C(=O)N(CC(O)CNC(c1n[nH]cc1I)=O)C)OC)OC 22601,N1(C(C(C2CCC2)NC(c2c(OC)ccnc2)=O)=O)CCC(C)C(F)(F)C1 22602,N1(S(=O)(=O)c2cnccc2N2C3CCC2CC3)Cc2ccccc2CC1CO 22603,N1(C(C(CC)(C)O)=O)C2CCC1CN(C(c1cc(O)ccc1Br)=O)C2 22604,C1(C)(C(N2CC(C)CC(NC(CCNC(=O)OCC)=O)C2)=O)CCC(=O)N(C)C1 22605,CN1CCCC1(C)C(=O)NCC(c1cccc(Cl)c1)NC(C1(C2CC2)CC1)=O 22606,N1(C(c2ncc(NC)nc2)=O)CC(C)C(C)(CNC(=O)COC(C)C)C1 22607,Cc1ccc(NC(C2C=CC(NCc3c(F)cccc3F)C2)=O)c(C(C)C)n1 22608,Cc1cc(C(N2CCCCC2CNC(=O)CNC(=O)C(C)C)=O)cc(C(F)F)c1 22609,Cc1oc([N+](=O)[O-])cc1C(=O)NCCC(C)(C)NC(=O)C=CC1CCCO1 22610,C(=O)(C1=C(C)S(=O)(=O)CC1)NC1CN(C(c2c(C#C)c[nH]n2)=O)C(C)(CC)C1 22611,C1(C)(CC(=O)N(CCC(C)NC(COCC(C)C)=O)C)CCCC1 22612,c1(C(=O)NC2(CCOC)CCC2)ccc(O)c(CO)c1.C123CC(C1)(C2)C(=O)NC3 22613,N1(C(c2cnnc(C)c2C)=O)CCOC2CN(C(C3CCN(C)C3)=O)CC12 22614,c1(NC(C2N(C(c3c(C)nn[nH]3)=O)CC(O)C2)=O)ncc(Br)cc1F 22615,Cc1cc(C(N2CCCC(C)C2CNC(=O)C2=C(Cl)CC2)=O)cc(=O)n1C 22616,c1(C(=O)NC2CC(NC(CCCOC)=O)C2)cc(C)c(Br)cc1C 22617,N1(C(c2[nH]cc(C)c2)=O)CCN(C(=O)C=Cc2cnc[nH]2)CC1C#N 22618,C#CCC(C(=O)NCC1(CNC(=O)C(=Cc2cccnc2)F)CC1)C1CC1 22619,C1(NC(C2CC(C)CC(C)(C)C2)=O)CCC2(CC1)CN(C(=O)CSS(C)(=O)=O)C2 22620,CCC(CC)(CC)C(=O)NC1CN(C(=O)CS(=O)(=O)CC)CC1O 22621,C1(S(C)(=O)=O)(C(=O)NC2CC(NC(c3nc(OC)nc(O)c3)=O)C2)CC(O)C1 22622,C#CC1CCN(C(=O)C(Cc2cn[nH]c2)NC(=O)CCCN(C)C(C)=O)C1 22623,Cc1cn2c(C)c(C(=O)NC(C)(C)CN(C(=O)CCCNC(N)=O)C)nc2s1 22624,C1(C(=O)NCC(=O)NC2CCC2)CCC(O)CN1C(=O)Cc1cccc(O)c1 22625,S(=O)(=O)(c1ccccc1Br)N1CCC(C(N2CCCC(C#C)CC2)=O)CC1 22626,c1(NC(=O)NC(C)C(=O)NC2CC3CC3C2)ccccc1 22627,CC1COC2(C1)CN(C(C1CN(C)CCN1C(C1CCOCC1(C)C)=O)=O)C2 22628,C1(NC(C(C)NC(C)=O)=O)CC1C1CCCN(C(C2(NC(C)C)CC2)=O)C1 22629,N1(C(C(C(CC)O)C)=O)CCc2nc[nH]c2C12CCN(C(c1csc(C)n1)=O)C2 22630,C1(COCC(=O)NCC2CC2C(=O)NCC2(Br)CC2)CCCO1 22631,Cc1nc(N(C2CC3CNC2C3)C(c2cc(C(C)C)[nH]n2)=O)cc(C(F)(F)F)n1 22632,C1(O)(CNC(C2CCC(=C)CC2)=O)CC(N=c2[nH]c3c(C)cccc3o2)C1 22633,C1(NC(c2cc(Cl)nnc2O)=O)CN(C(=O)CSCC(F)(F)F)CC1C1CC1 22634,CC(C)(CC(=O)NCC1CCCCN(C(C2CCC(N=[N+]=[N-])C2)=O)C1)CC(F)F 22635,C1(F)(C(=O)NCC2N(C(C)=O)CCC2)CCN(C(C2(C)CCN(C)C2)=O)C1 22636,N1(C(C2(CCC)CC2)=O)CCC(F)(F)C(CNC(C2(N(C)C)CC2)=O)C1 22637,CC1=CC(C)CN(c2cc(NCc3cc(C)nc(C)c3)ncn2)C1 22638,c1(C(N2CC(NC(Cc3c(OC)ccnc3)=O)C2)=O)cncc2c(O)nccc12 22639,C(CC(C(=O)NC1(CCCCNC(c2csc(Cl)c2)=O)CC1)OC)OC 22640,C1(CNC(=O)C=CC2CCCC2)CCCCN(C(=O)CC2CC3(CCC3)CO2)C1 22641,c1(C(N(C)CC2N(C(C(C=C)C)=O)CCCC2)=O)cc(CC)ccc1F 22642,CCC(C)(C)CCCC(=O)NC(CC)CCCC(=O)NC1(C2CC2)CC1 22643,c1(C(N2CC(N(C)Cc3cc(OC)ns3)C2)=O)cc(F)c2ncccc2c1 22644,C1(C(=O)NCC(C)CN(C)C(c2nccnc2O)=O)CS(=O)(=O)CC12CC2 22645,C1(CN(C)C(C2(N(C)C)CC(O)C2)=O)CCN(C(=O)Cn2ncccc2=O)CC1 22646,C(C(C)C(C)(C)C)NC(C1CCCN(Cc2ccccc2)C1)C 22647,C1(NC(C2(OC)CCN(C(C(CC)N(C)C)=O)C2)=O)CCCOC12CCC2 22648,c1(C(=O)NCCCCN(C)C(C2CC(=O)N(O)C2)=O)coc2c(F)cccc12 22649,C1(C(=O)NCC2N(C(C=Cc3ccc(CC)o3)=O)CCC2C)CC(S(C)(=O)=O)C1 22650,CCC(CO)CCNC(=O)C(C)CN(C(=O)CCC1CC(C)C1)C 22651,C=CCC(CC)C(=O)N1C2CCC1C(CNC(=O)C=C(C)Cl)C2 22652,c1(C(=O)NCCCN(C(CCNC(N)=O)=O)C2CCCC2)nocc1Cl 22653,c1(OC)ccc(CN2CCCC(CNC(=O)C(N3CCC(OC)C3)=O)C2)cc1 22654,c1(CC)c(NC(C2CC2C(=O)NCc2cnc(C)[nH]2)=O)cnn1C 22655,c1(OC)ccc(C(=O)NCC(C(C)C)NC(=O)Cc2cnn(C)c2)c(C)c1OC 22656,c1(C(N2C3C(NC(C(c4ccccc4)SC)=O)C(C3)C2)=O)ccc(=O)n(C)c1 22657,c1(C(N2C(C)CC(C(=O)OC(C)(C)C)CC2)=O)ccccc1S(C)(=O)=O 22658,C1(O)(C(C)NC(C2(CO)CCCCC2)=O)CCN(C(c2nccnc2N)=O)CC1 22659,c1(C(N2CCCC(N(C)C(c3cn(C)nn3)=O)C2)=O)ccnc(Cl)c1O 22660,CC1=C(C(=O)NC(C2CCN(C(c3ncccc3N(C)C)=O)C2)C)CCO1 22661,Cc1cccc(C(N2CC(CC(=O)N(CC(C)C(F)(F)F)C)C(C)C2)=O)c1O 22662,c1(C(=O)NC(C)(C)CCNC(c2cc(CCO)on2)=O)ccnc(F)c1O 22663,N1(C(c2cncc(NC)c2)=O)CCC2(COC(CNC(=O)C(F)CC(C)C)C2)C1 22664,C(CN=C(NCC1CCCO1)N1CC(C(F)F)C2(CCC2)C1)c1c(C)ocn1 22665,N(C(=S)NC1CCCn2c(C)nnc21)CC#C 22666,C(C)(C(C(=O)NCc1nccn1C1CC1)C(C)C)NC(C#CC(C)C)=O 22667,c1(C(N2CC(NC(c3[nH]n(C)c(=O)n3)=O)C(O)C2)=O)occ2c1CCOC2 22668,C(CNC(c1cc(CN(C)C)c[nH]1)=O)(CC(C)C)NC(c1c(CCC)occ1)=O 22669,c1(N(CCC(=O)NC)C)nc(=NCC(CO)C2CCC2)[nH]c2cccnc12 22670,c1(NC(=O)OC)cccc(CNC(=O)NCc2nnc(-c3ccco3)s2)c1 22671,N1(C(CC(=C)Br)=O)CCC(NC(=O)COCCCC)C(F)C1 22672,c12ccccc1CS(=O)C2.N#CCCCN 22673,N1(C(c2cncc(C)c2)=O)CC2CC1CN2C(=O)C(C)Cc1cccc(Br)c1 22674,C1(CNC(C(C)N(C(=O)CCC2CC2)CC)=O)CCCC1CC1CC1 22675,C(=O)(C1=CCCOCC1)N1CCC(N(C(C2C3CC4C(C3)C24)=O)CC2CC2)CC1 22676,C=CCC(CC)C(=O)NC1CN(C(c2cn(C(C)C)nn2)=O)CC1(C)C 22677,C1(C2CCN(C(c3ccc(C#N)nc3O)=O)CC2)(NC(COCC)=O)CCC1 22678,c1(C(=O)NC2CC(C)(NC(CNC(CC)=O)=O)C2)cc(F)c2c(c1)CCC2 22679,C(C(=O)NCC1CC(O)CN1C(=O)C=Cc1cnccn1)(C(C)C)OC 22680,c1(CC(=O)NCCN(C(CCC(N)=O)=O)C2CCCCC2)ccc(F)c(F)c1F 22681,C(CO)(CCCNC(=O)C(c1cnn(C)c1)=O)NC(C(C)C1CCCC1)=O 22682,c1(C(=O)NC(CCNC(c2n(CC)nnc2)=O)C)cc2c(s1)CCOC2 22683,N1(C(c2ccc(C#C)cn2)=O)CCC2(CC(NC(=O)C3=NOCC3)CO2)C1 22684,c1(OCC(=O)OCC2CCN(C(=O)OC(C)(C)C)C2)nc2cc(F)ccc2s1 22685,c1(C(N2CCC(C(F)(F)CO)CC2)C(=O)NC)ccc(Br)cc1OC 22686,N1(C(=O)CCCC2CC2)CC2CCC(C(N3CCc4c[nH]nc4C3)=O)(C2)C1 22687,c1(C(=O)NC2CN(C(C=CCCC)=O)C3C2C3)ccc(NC(=O)OC)cc1 22688,C1(C(=O)NCCC2CCN(C(=O)CCc3ncc[nH]3)C2)CCCC(CF)C1 22689,C(CCCC(CO)NC(c1cc(C)nnc1O)=O)NC(c1cccc(CC)c1)=O 22690,C1(CC)(CC)COCCN1C(=O)CCCN1CCC(O)C1.c1(C)ccccc1 22691,C1(C(=O)NCCC2(O)CN(C(c3c(C)cnn3C)=O)C2)CCC2(C1)CC2(F)F 22692,N1(C(CCP(C)(C)=O)=O)CCOC2CN(C(=O)C=C(C3CC3)C3CC3)CC12 22693,N1(C(C(C)OCc2ccccc2)=O)CCC2(CCCN2C(C2CCC(=O)N2)=O)C1 22694,Cc1cnsc1C(=O)NC1(C(=O)NOCC2CC(=C)C2)CCC1 22695,C1(CC(C)NC(C2C(F)(C(=O)OC)C2)=O)CCN(C(c2ccon2)=O)CC1 22696,N1(C(C(C)OCCC=C)=O)CC(O)CC1C(=O)NCCN=S(C)(C)=O 22697,c1(OC)ccc(C(C(F)(F)F)NC(c2coc(C(C)OC)n2)=O)cc1 22698,c1(C(=O)NCC2C(C)CCN(C(C)=O)C2)cc2c(c(S(N)(=O)=O)c1)CCC2 22699,C1(NC(C(C=C)(C)C)=O)CCC2(CC1)CN(C(C1(CC(F)(F)F)CC1)=O)C2 22700,c1(C(=O)OC)nc(C(=O)Nc2nc(C)c(NCCC3COCCO3)s2)oc1C 22701,N1(CC)CCC(C(N2CC(C(O)C(=O)NC(CC3CCC3)CO)C2)=O)C1 22702,C1(CN(C(c2n(CC#C)ccc2)=O)C)CCCCN1C(c1cnsc1)=O 22703,c1(C(=O)NCCCN(C(C)C)C(C2CCC(=O)C2)=O)cnc(C2CCC2)nc1O 22704,C1(C(N(CC(O)CF)C)=O)C(C)CCN1C(=O)C(C(C)C)SC 22705,C1(C(=O)NC(C#C)CC(C)C)CCN(C(=O)CC2(O)CCCCC2)C12CC2 22706,CC(CS(=O)(=O)N=c1ccn(C2CCOC2)[nH]1)C1CC1 22707,c1(NC(c2nccs2)C)cc(-c2cccs2)n2nccc2n1 22708,C(=O)(CCC(CF)CF)NC(C(C(=O)NC(C)CC1CC1)(C)C)C 22709,Cc1cc(=NC(=O)C(C)(C2CC2)N(C)C(c2ccon2)=O)[nH]n1C 22710,c1(C(N2CC3C(NC(C(CCC)O)=O)(C3)C2)=O)cc(OC)ccc1C 22711,C12(C(N3CCC(OCCNC(C(C)n4cnnn4)=O)C3)=O)CCCCC1C2(F)F 22712,c1(C(=O)NC2CC3CN(C(CCOCCC)=O)C2C3)c(F)cc(C)cc1Br 22713,Cc1nnc2cnc(C(=O)NC(C)CN(C(=O)C(C)(O)CC(C)C)C)cn12 22714,Cc1oc(C)c(C(=O)NC2CC(CNC(=O)CCc3ccc(O)c(F)c3)C2)c1C 22715,C1(NC(CCN(C)C)=O)COCC1C(=O)NCC(F)CO 22716,c1(C(=O)NCC(C)CNC(C2CCCN2C(=O)C2CC2)=O)cncc2[nH]ccc12 22717,N1(C(Cc2ncc(C)o2)=O)CCC(CNC(C2CCC(C)(C)O2)=O)C(F)(F)C1 22718,C1(CNC(CCCCNC(N)=O)=O)CCN(C(=O)CC2CCCOC2)CC1(F)F 22719,N1(C(Cc2c(C)scc2)=O)CCCC(C)C1CCNC(c1cccc(Cl)c1)=O 22720,Cc1nc(NC2CN(C(c3nc(N(C)C)nc(=N)[nH]3)=O)CC2C)cc(O)n1 22721,N1(C(CC2CC(C)C2)=O)CCC(C)(C)C(C(=O)NCC2(C)CC(C)(C)C2)C1 22722,c1(C(C)NC(=O)CC(c2cccc(C(F)(F)F)c2)N)ccc(F)cc1F 22723,N1(C2C(NC(C(CC)F)=O)CCC2)CCN(C(C2CC(O)C2)=O)CC1 22724,C(=O)(C1c2ccccc2CCCN1CC(c1cc(Cl)ccc1Br)=O)OC 22725,C=C(C)CC(C(=O)NC(CCC1CCC1)C(=O)N1CC(C(C)OC)C1)OC 22726,CC1CN2CCN1C(C(N1CCCC1C1CCN(C(=O)CC3CC3(Cl)Cl)C1)=O)C2 22727,N1(C(COCCN(C)C)=O)CC(O)CCC1C(=O)NCCCc1ncn(C)n1 22728,Cc1cc(=NCc2ccsc2)[nH]c(=NCCn2cccn2)[nH]1 22729,N1(C(c2ccc(C)c(Cl)c2Cl)=O)CCCC2CCN(C(c3ccncn3)=O)CC12 22730,c1(OCC)ccc(C)nc1C(=O)NCC1CN(C(=O)CC2COC(=O)C2)C1 22731,N1(C(CN(CCC)C)=O)CC2CCC1CN2C(=O)Cc1c[nH]c2ncccc12 22732,CCCC(CC)CC(=O)NC1CN(C(C2OCC3COCCC23)=O)C1 22733,c1(C(=O)NC2(CC=C)CN(C(=O)C(C)CC3CCCO3)C2)cc2scc(C)c2[nH]1 22734,C=CC1(C(=O)N(CCOCC)CC)CCN(C(=O)CCCn2cccc2)C1 22735,c1(C(=O)NCC2(C)CCC(NC(c3ncn(C)c3)=O)C2)ccnc2ncccc12 22736,C12(C(N3C(CNC(c4cccc(COC)n4)=O)COCC3)=O)CC1CCC2(F)F 22737,N1(C(C2=C(C)CC2)=O)CC2COCC2(C(=O)N(C2CCCC(O)C2)C)C1 22738,O=C1CCC2(CCCN(C(C34CC5CC(CC(C5)C3)C4)=O)C2)N1 22739,c1(CC=C)cccc(C(=O)NCCN(C(=O)C=C(C)C)CC2CC2)c1 22740,c1(CC)nc[nH]c1C(N1CCCC1CN(C(=O)C=Cc1ccsc1)C)=O 22741,c1(C(N2CC(C(=O)NCC(C)(C)C3CC3)(COC)C2)=O)ccc2cccnn12 22742,Cc1coc(C2CC2)c1C(=O)NCC1CC(NC(c2coc(CF)n2)=O)C1(C)C 22743,C#Cc1ccc(C(N2CCC(CO)(NC(c3cc(O)ncc3Br)=O)C2)=O)nc1 22744,CC1CCn2c(C(N3CC4C(NC(C56CC(CO5)C6)=O)C4C3)=O)cnc2C1 22745,Cc1ccc2occ(C(=O)NC3CCC(CNC(c4cscc4C)=O)CC3)c2c1 22746,C1(NC(CC(C)C2CCCCC2)=O)CC2(CCCN(C(C3CC(=O)C3)=O)C2)C1 22747,c1(C(C)C)ccccc1CC(=O)NC(C)(C)CCNC(=O)C(C)NS(C)(=O)=O 22748,C1(C(N2CC3C(NC(C4(C)CCOCC4)=O)(C3)C2)=O)CN2CCN1CC2 22749,c1(CC(N2CC(O)(C(C)NC(COC(C)C)=O)C2)=O)noc2cc(F)ccc12 22750,n1(CC(=O)NCCNC(C23CNC(CO2)C3)=O)cc([N+](=O)[O-])cn1 22751,N1(C(c2c3ccc(C)cc3no2)=O)CC2CCCC(C1)N(C(=O)C=C(Cl)Cl)C2 22752,CCCCCC(F)C(=O)N1CC2CC1C2C(N1CCC2CC12C)=O 22753,N1(C(CCC2(NC(c3c(CC)cno3)=O)CCC2)=O)CC(C)SC(C)C1 22754,C1(CNC(C(C)OCCN(C)C)=O)CCN(C(c2c[nH]cc2C2CC2)=O)CC1F 22755,N1(C(=O)NC2CCC(N(OC)C)CC2)CCOC2(CCC(F)(F)CC2)C1 22756,N1(c2scc(CC(=O)N(C3CN(C(C4(CO)COC4)=O)C3)C)n2)CCCNC1=O 22757,c1(CCC)ccc(C(C(=O)NC(C)CC)N(CCCCO)C)cc1 22758,CCCC(C(=O)NCC1(c2nn[nH]n2)CCCCC1)OCC 22759,c1(C(CCNC(=O)NC(c2ccc(C)o2)CCC)NC(=O)NC)ccccc1C 22760,CC(C)C(O)C(=O)NC1CC12CC(NC(=O)C=Cc1ccsc1Br)C2 22761,O=C(CC1=CCN(C(C2(O)CCOC2)=O)CC1)Nc1cncc(C2CC2)c1 22762,c1(C(=O)NCc2occc2C(=O)NC2CN(c3ccncc3)C2)ncc(F)cc1F 22763,c1(C(N2CCN(C(CCSC)=O)C(C3CC3)C2)=O)ccc2c(c1)nc(CO)n2C 22764,C1(N(C)Cc2ccc(C(N(CCC)Cc3ncc[nH]3)=O)cc2)CC(C)(C)OC1(C)C 22765,CC1=C(C)CC(C(=O)N(C)CC2(CNC(C3(O)CCC(C)CC3)=O)CC2)CC1 22766,c1(OC)cc(C(=O)NCC#CCNC(=O)CCc2ccc(Cl)nc2)ncn1 22767,C1(C(N(C)Cc2ccc(Br)s2)=O)CCCN(CCC(=O)Nc2ccccc2Cl)C1 22768,CCC(CC(=O)N1CCC(CNC(=O)C(C)(CC)OC)C1)C1CCC1 22769,CC1(C)Cc2cccc(C(=O)NCC3CC(NC(C4(C)CC4)=O)C3)c2O1 22770,Cc1ccn2cnc(C(N3CCN(C(C4CC(F)(F)C4)=O)C(C)CC3C)=O)c2c1 22771,C(=O)(CC(C)(C)CC(=O)N(C1CN(C(=O)C(O)c2ccco2)CC1(C)C)C)OC 22772,N1(C(C(n2ncc(C)c2)C)=O)CCC(CNC(=O)CC(C)C(F)F)C(F)(F)CC1 22773,c1(C(N(C2CCN(C(=O)C=CS(C)=O)C2)CC)=O)ccccc1Cl 22774,C1(CNC(COCC(C)C)=O)CC2(CCC2)CN1C(=O)CC(C)n1cccn1 22775,O=C(C(F)C(F)(F)F)NC1CCC(c2ccccc2)(NCc2cscn2)CC1 22776,C1(C(N2CCCC2Cn2cc(C(c3nccn3C)O)nn2)=O)(CC)CCCC1O 22777,C1(NC(C2CC(CCC)C2)=O)CCN(C(c2ccnn2CC(F)(F)F)=O)C(C)C1 22778,c1(C(N(CCCN(C(C(C=C)O)=O)C)C)=O)nc2ncccc2cc1C 22779,CCCC(O)CC(=O)N(C1CCCN(C(=O)Cc2nccn2C)C1)C 22780,C1(CC=C)(C(N2CC(O)(C(F)C(=O)NC(C)C(F)F)C2)=O)CCOC1 22781,C1(CNC(=O)Cc2ccco2)CC2(CO1)CN(C(=O)Cc1ccc(F)cc1F)C2 22782,N1(C(CCCCC(=O)NC)=O)CCC2(C1)CN(C(=O)C(F)n1ccnc1)CCO2 22783,N1(CC(C)NC(=O)Nc2noc(C)c2C)CCSC(C)(C)C1 22784,S(=O)(=O)(c1ccc(=NCc2csc3cc(Cl)ccc23)[nH]c1)NC1C(C)CN(C)C1 22785,CCC(CO)(C(=O)N1CC=CC(C(=O)NOC(C)C)C1)OC 22786,Cc1cc(NC(C23CC2CCN3C(c2ccc(C)nc2O)=O)=O)c(=O)n(C)c1 22787,c1(OC2CN(C(C(=O)NC(CC)C)CC3(C)CC3)C2)ccc(F)cc1 22788,C1(CC(=O)NC(CNC(C2(COC)CCC2)=O)(C)C2CC2)C=NN(C)C1=O 22789,c1(CC=C)ccccc1C(=O)NC(C)(CSC)C(=O)NCCOC(F)F 22790,C(C(C(C)(C)C)NC(=O)Cn1c(C)csc1=O)NC(C1C(CC)C1)=O 22791,C(=O)(C(O)C(C)(C)C)N1C(C(=O)NC(COC)COC)CC2CC21 22792,C1(NC(C2(CC#C)CCOC2)=O)CCN(C(=O)C=C(C)C)CC1CC 22793,N1(C(C(C)OCC)=O)CC2CCC(N=c3[nH]nc(C(F)(F)F)s3)CC2C1 22794,C1(CC(=O)OC)CCN(C(=O)N(C2CCN2)CCCO)CC1 22795,C1(N(c2ncncc2F)C(c2csnn2)=O)CNCC(F)(F)C1 22796,c1(CC(=O)NCC2CC(NC(c3c(=N)cc[nH]c3)=O)C2)cc(O)nc(O)n1 22797,c1(CNC(c2c(C)c(C3CC3)on2)=O)cnn2c1CN(C(=O)CCC1CC1)CC2 22798,C(C)(C(=O)NC1(CN(C)C)CC1)(N(C(C(C)C1CCCC1)=O)C)C1CC1 22799,C1(NC(C=C(C)C)=O)COC2(CCN(C(=O)CCc3ccc(=N)[nH]c3)CC2)C1 22800,C1(C(=O)NC(COC)C(C)(C)C)CCCCCCN1C(=O)C(F)CCC(C)C 22801,c1(C(N(C2CCCC2)CC(=O)OC)=O)cc(OC)ncc1C1=CCCCC1C 22802,C1(OC)CC(NC(c2cn(C(C)(C)C)nn2)=O)CN(C(=O)CC2C=CCCC2)C1 22803,C(=O)(C(CCF)NC(=O)OC(C)(C)C)NCC(N(C(CC=C)=O)C1CC1)C1CC1 22804,C1(CNC(c2cn(CC)nc2)=O)CCC(NC(=O)CN2CCSCC2)CC1 22805,C1(NC(C2CCC(C)(C)OC2)=O)CC1C1CCN(C(c2ccoc2Cl)=O)CC1 22806,c1(NCC2(C)N(C(=O)OC(C)(C)C)CC(OC)C2)oc2ccccc2c1Cl.OC 22807,O=C(CC(Cc1cccs1)Sc1cc[nH]c1)N1CC(Cn2ccnn2)C1 22808,c1(N2C(C(=O)Nc3c(C(=O)OC)nsc3)COCC2)ncc(C)c(C)n1 22809,c1(OC)cncc(NC(CC2(NC(=O)COCC3CCC3)CCC2)=O)n1 22810,CCCC(C(=O)NCC1CCC(NC(=O)C=Cc2nc(C)cs2)CC1)NC(C)=O 22811,N1(C(C(C)(C)CO)=O)CC2CC1CCC2NC(c1cn(-c2ccccc2)cn1)=O 22812,c1(OCC)ccc(-c2ccc(NC(=O)Nc3cc(C)cc(C)c3)nc2)c(C)c1 22813,N1(C(c2c(C)cccc2C)=O)CC2CCC(C1)C(NC(C1CC(F)(F)CS1)=O)C2 22814,N1(C(C2(C)CC(C)C2)=O)CCOC2(CCN(C(=O)C3=COCC3)CC2)C1 22815,C1(NC(C=C(CC)C)=O)CCN(C(=O)COc2ccc(C)cc2)CC1C 22816,Cc1c(C(=O)NC(c2cn(C)nn2)C(N2CC3C=CC2CC3)=O)cccc1C#N 22817,CC1CC=C(C(=O)NC(CC2CC2)C(=O)NCCn2cncn2)CC1 22818,C1(C)(C(N2CC(C(C)OC)C2)=O)CCCN(C(=O)CC(F)(F)F)C1 22819,c1(C(=O)NCC(C2CC2)NC(C(COC)N(C)C)=O)sc(C)c(Br)c1OC 22820,C1(NC(c2c(C)nc(C(C)(C)C)s2)=O)CCCN(C(C2CCCC(C)C2)=O)C1C 22821,c1(NC(CCCCc2cccc(OC)c2)=O)cccc(CC#N)c1F 22822,Cc1c(C(=O)NC(C)(C)C(=O)NCc2ccccc2)nc(O)c2ccccc12 22823,N1(C(CC2OCC(C)(C)C2)=O)CC2(C1)CN(C(C1(O)CCC1)=O)CCO2 22824,c1(OCC=C)ccccc1C(N1CCCC1(C)C(=O)NCc1ccccn1)=O 22825,C1(CNC(C=CC(C)=O)=O)CC2CCC(C1)N2C(=O)CCCc1cccnc1 22826,Cc1ccc(C(F)C(N2CCCCC2CCNC(=O)CSCCC#N)=O)cc1 22827,C1(CNC(=O)C(O)CN2CCCC2)C2CN(C(=O)CC3(n4cncn4)CC3)CC12 22828,C1(C(=O)NC)CCN(C(C2(COC)CN(C(c3ccn(C4CC4)n3)=O)C2)=O)C1 22829,N#Cc1c(Cl)nsc1NCC(C1CCCC1)NC(C1COC(=O)C1)=O 22830,C1(NC(C=CC=CCC)=O)CCC(O)CN(C(=O)CCC2CCN(C)C2)C1 22831,c1(C(=O)NCC(CNC(Cc2c(C)n(C)cn2)=O)C)ccc(S(N)(=O)=O)nc1 22832,CC(CC(C)(C)C)C(=O)NCc1ncc(C(=O)NCC2(O)CCN(C)C2)cn1 22833,C(CNC(=O)NCc1cc(C)c(F)c(C)c1)(CCS(C)(=O)=O)OC 22834,N1(C(c2cnn(CC)n2)=O)CCCC(NC(c2cccc(C)c2Cl)=O)CC1 22835,C1(CC)CN(C(=O)CN2CCCCCC2)CCC1NC(c1c(C)nn(C)c1N)=O 22836,c1(C(N(CC(CC)NC(C=CC)=O)CC)=O)cnn2cccc(Br)c12 22837,N1(CC(=O)NC2C(NCC(=O)NC3CC(C(F)F)C3)CCC2)CCOCC1 22838,C1(CN(C(=O)CCCNC(C)=O)CC)CCN(C(c2cc(C)cs2)=O)CC1 22839,CC1CCc2sc(C(N3CCC(N(C(=O)CNS(C)(=O)=O)C)C3)=O)cc2C1 22840,c1(NC(C(c2cc(C(=O)OC)ccn2)N(CC=C)CC#N)=O)ccc(F)cc1C 22841,C(=O)(CC(O)C(C)C)NC(CC=CC)C(=O)NCc1ncccc1F 22842,C1(CN(C)Cc2cnn(C)c2)CCN(C(=O)C(C2CCOCC2)=O)CC1 22843,C(=O)(C1=CNC2=NCCCN12)N1CCCCC(NC(C2CC(C)N(C)C2)=O)C1 22844,C1(CNC(c2cnn(CC(C)C)c2C(F)F)=O)CN(C(C)C)CCC1(C)C 22845,c1(C(N2CCC(C3N(CC#C)CCC3)CC2)=O)cc(C#N)[nH]c1C 22846,C1(C(N(C)CC2(CC(C)C)CC2)=O)CC2(CCN(C(C3CCCCS3)=O)C2)C1 22847,C(=O)(C(C)CC(=O)NCCCc1cncc(C(=O)OC)c1)OC 22848,c1(C(=O)NC2CN(C(c3c(OC(F)F)cccc3Cl)=O)C2)cccc2c1CCC2 22849,c1(C(C)(C)C)nc(=NCC2CCCCN2C(=O)Cn2cncn2)s[nH]1 22850,C1(NC(c2cc(C)ncc2)=O)CCN(C(C2OCCCO2)=O)CC1F 22851,c1(NC(CSCC(=O)OC)=O)c(Cl)cc(OC)cc1Cl.c1nnc(C)o1 22852,CCC(C)C(C)C(=O)N(C)CC1CCCCN1C(=O)C(C)CC1CC1 22853,CC(C)(C(=O)NCCC1CN(C(C2CCS2(=O)=O)=O)C1)c1ccccc1 22854,Cc1cc(N2CCC(NC3CCSC(c4cnn(C)c4)C3)CC2)ccn1 22855,n1(CC)ncc(C(=O)NC(CO)C(C)NC(=O)CCC2CCCCC2)c1C 22856,Cc1cc(Cl)c(C(=O)NC2CC3CC(NC(C4C5(CC5)C45CC5)=O)C3C2)cc1C 22857,Cc1ccc(C(N2CCCC(C)C2C)C(=O)NC2CCOC2)cc1[N+](=O)[O-] 22858,c1(C(=O)NCC(C)(C)NC(CC(=C)Br)=O)ccc(CC)nc1C 22859,Cc1nc2nccc(C(=O)NC3CCCC(CNC(C4CN(C)C4)=O)C3)n2n1 22860,N1(C(=O)C2=C(Cl)CCC2)CCC2(CCCN2C(C2CC3(C2)CC3F)=O)C1 22861,c1(-c2nc(C(C)O)nn2C2CCOC(C)(C)C2)cccc2ccsc12 22862,Cc1ccncc1C=CC(=O)NC1CC(NC(=O)C(=C2CCCCC2)F)CC1O 22863,CC(CCCCNC(C1CCOC1C1CC1)=O)NC(c1ccc(F)nc1)=O 22864,C(=O)(C1=C(C)C(C)(C)OC1=O)N1C(COC)CN(C(=O)Cc2ccc(C)s2)CC1 22865,C1(C)(c2cn(CCC=C(C)C)nn2)COCCN1C(c1cc(Cl)c(Br)s1)=O 22866,C1(C(N(CCN(C(=O)CC2CCC(=O)N2)C(C)C)C)=O)CCNC(=O)C1 22867,N1(C(CCC(C)C)=O)CCC2(CCCCN(C(C3(N4CCCC4)CCC3)=O)C2)C1 22868,C1(C(=O)NCC(C)(C)NC(C(C)NC(c2ccco2)=O)=O)C(C)(C)OC1(C)C 22869,CCCC(CC(C)C)C(=O)N1CC=CC1C(=O)NCC(=O)OC 22870,c1(N2CC(CC)C(C)C2)ccc(S(=O)(=O)N(C)Cc2cscc2Br)cn1 22871,C1(C(=O)NCCC2COCCN2C(c2cnc(SC)n2C)=O)(CC)CC(C)(C)C1 22872,Cc1nc2cncc(C(=O)NCC3CN(C(C4C(Cl)(Cl)C45CC5)=O)CCO3)c2[nH]1 22873,C(=O)(C1=NOC(C)(C)C1)NCC1(NC(C2C(c3c(C)cccc3)C2)=O)CC1 22874,C(=O)(CCCc1ccncc1)N(CC(CC)NC(=O)C(C)(C)C1CC1)C 22875,N1(C(C(C)(C)CF)=O)CCC2(CCCC2CNC(c2ccnc(O)c2)=O)CC1 22876,S(=O)(=O)(c1c[nH]c(NCC2CC(C)N(C(C3C4CC5C(C4)C35)=O)C2)c1)NC 22877,CC1CCN(C(c2cn(CCNC(c3cnc(Cl)s3)=O)nn2)=O)C(C)C1 22878,N1(C(CC2ON=C(C)C2)=O)CCCC(C)(CNC(=O)CCCc2ccc(C)s2)C1 22879,c1(C(=O)NCC23N(C(COCCOC)=O)CCC2CC3)nccn2nccc12 22880,C(=O)(C1=Cc2ccccc2OC1)N(CC(C)NC(=O)C(N1CCCCC1=O)C)C 22881,c1(OCCCC)ccc(C(=O)NCCCc2cn(CCC(F)(F)Cl)nn2)cc1 22882,c1(CC(=O)NC2C(C(N)=O)CN(C(C3(C)CC3F)=O)CC2)ccc2c(c1)OCO2 22883,c1(C(C)=O)cc(O)cc(O)c1C(=O)N(C)C.C123C4CC1C1C(C4C21)NC3=O 22884,c1(OC)cc(CN2CCC(C(=O)NCc3ccncc3Cl)C(O)C2)c(Br)cn1 22885,c1(C(=O)NC2C(NC(C3(CCCC)CCCC3)=O)CC2)cnc2[nH]cnc2c1 22886,C(CNC(C1(C(F)F)CC1)=O)(C(C)C(C)C)NC(c1cc(C)c(C)[nH]1)=O 22887,N1(C(C2CCC(C)O2)=O)CC=C(CCNC(c2cc(Br)n[nH]2)=O)CC1 22888,C1(C(=O)OCC)CC(F)CN1C(=O)CCCCc1cn(C2CCOC2)nn1 22889,N1(C(c2cn(CC)nc2)=O)CCC(C)(C)C1CC(N1CC(C)(C#N)C1)=O 22890,S(=O)(=O)(c1cccc(-c2nnc(CC(=O)O)o2)c1)C1(CS(C)(=O)=O)CC1 22891,C1(NC(Cc2c(C)cco2)=O)CN(C(=O)CC2CCCOC2)CC2(CC2)C1 22892,C(C1C(C(=O)N(C)CCOCCNC(c2sc(CO)nc2C)=O)C1(C)C)=C(C)C 22893,O=S(c1ccc(NC2CCc3c(O)cccc32)cc1)C(F)(F)F 22894,c1(C(=O)NC2CC3(CN(C(C4(SC)CC4)=O)C3)C2)cc2nc[nH]c2cn1 22895,CCC(CC)CC(=O)NCc1nnn(C)n1 22896,C1(C(=O)NC(C)C(=O)N(C)CCN(C)C(C2CC(O)C2)=O)CCCCC1 22897,Cc1ccc([N+](=O)[O-])c(C(=O)NC2CCCN(C(c3c(C)nsc3C)=O)C2)c1C 22898,CCC(CC)CCCC(=O)NC(C1(O)CCN(C(c2noc(CC)c2C)=O)C1)C 22899,C1(NC(c2csc(Cl)n2)=O)CC(O)CN(C(c2ccc(OCC3CC3)nc2)=O)C1 22900,C12(CNC(C(CC=CC)C)=O)CCCC(CN1C(=O)Cc1cnoc1)C2 22901,N1(C(C(C)O)=O)CC(NC(=O)CN2CSCC2=O)CC2(CC2)C1 22902,C1(NC(=O)Cc2cccnc2)CCCN(C(C2CC(=C3CCC3)C2)=O)C1 22903,C=CCC(C)(C)CC(=O)NCCC1CCC(NC(c2cc3ncccc3s2)=O)C1 22904,C1(NC(c2nc(C)sc2)=O)CN(C(C2C=CCC2)=O)CC12CCS(=O)(=O)CC2 22905,C(=O)(C(O)C1=CCCCC1)N1CC(C)(OCC(N2CC3CCCC2C3)=O)C1 22906,C1(C(=O)NC2CC(CN=c3nc(C)[nH]s3)C2)CCc2ccccc2O1 22907,C1(C(C)NC(=O)Cc2cn[nH]c2)CCN(C(c2cnnn2C2CCCC2)=O)CC1 22908,N1(C(C(CO)OC)=O)CCC2(CC1)CC(NC(=O)CCCn1ccnc1)CO2 22909,c1(OC)c(CNC(=O)N(CCCN(C2CCCC2)C)C)cccc1Br 22910,C(CC(=O)N1CCN(CC(C)(C)NC(C2CC3CC2C3)=O)CC1)(C(F)(F)F)OC 22911,c1(CNC(=O)CC2CCC(NC(C3C=CCCCC3)=O)C2)ccc(C2CC2)nc1 22912,C(C)(N=c1cc(C)nc(N2CCC(CC(C)C)C2)[nH]1)c1[nH]nc(N(CC)CC)n1 22913,N1(C(c2ccc(CN(C)C)o2)=O)CCC(CO)(CNC(C2CCS(=O)(=O)C2)=O)C1 22914,c1(CC)cc(CNC(=O)C(C)=CCNC(c2cc(OC)n[nH]2)=O)on1 22915,CCC(C)(C)C(C)NC(C1CCN1C(=O)C(C)NC=O)=O 22916,C=CC1OCCC1C(=O)NCCC1CC(NC(=O)CCC2CC2C)C1 22917,c1(OCC)cc(Cl)ccc1C(N1CCN(C(=O)CCC=CBr)CC1CF)=O 22918,Cc1cn(C)nc1C(=O)NC(CC1CCCC1)C(=O)NC1CCOCC1F 22919,C(=O)(C1COc2ccccc21)N1C(CNC(c2n[nH]c(C)c2O)=O)CC(F)(F)C1 22920,CC(C)C(O)C(C)C(=O)NCC1CCOC1C(N1CC2CC(O)CC1C2)=O 22921,N1(C(=O)OC(C)(C)C)CCC2CN(C(c3ncc(F)cn3)=O)C2C1 22922,C(=O)(CC(O)CC(C)C)NC(C(C)(C)NC(CCCN(C(=O)OC)C)=O)C 22923,c1(C(N2CC(CNC(CC=C=C)=O)C(O)C2)=O)c(-n2cccn2)cccc1F 22924,c1(C(=O)NC2C(NC(=O)CC3CC4(CC4)CO3)CCC2)ccc2c(c1)CNC2=O 22925,C#CCCC(O)C(=O)N1CC(F)CC1CNC(C1(S(N)(=O)=O)CC1)=O 22926,c1(C(=O)NC2C(F)CCN(C(C3CC(=C)C3)=O)C2)ccc2nc(C(F)F)[nH]c2c1 22927,C1(C(=O)NC(CC#C)CC#C)CCCCCN1C(C1CC(C)=NO1)=O 22928,c1(C(=O)NCC(C(C)(C)C)NC(C(C)OCC#C)=O)ccc(C#N)c(O)c1 22929,N1(C(c2nn(CC)c(O)c2)=O)CCCC(C)(C)C1CNC(=O)C(C)(C)OC 22930,c1(C(=O)NCC2(F)CN(C(C3C4CCOCC34)=O)C2)ccc2ncnc(O)c2c1 22931,CCCCCCCCCCCCCCCOC(C1CC(=O)NC2(CCC2)C1)=O 22932,c1(CNC(C2CCC(F)C2)=O)ncc(Cl)cc1Cl 22933,c1(-n2cnc(C(N3CCC(NC(CCC=C)=O)C3)=O)n2)ncccc1F 22934,N1(C(c2cc(Cl)nc(Cl)c2)C(=O)NC)CCc2[nH]nc(CO)c2C1 22935,c1(CNC(=O)COCC2CCCC2)cc(C(F)(F)F)on1.C12CC(C1)NC(=O)C2 22936,Cc1oc(CNC(C2CN(C)C2)=O)nc1C(=O)N(C)CCC1CCC1 22937,c1(C(=O)NCC2(CN(C)C)CCC2)ccccc1-n1cc(CCS(N)(=O)=O)nn1 22938,C12(C(N(CC(CCC)C)C)=O)C(NC(c3cocn3)=O)C3CC1C2C3 22939,N1(C(CO[Si](C)(C)C)=O)CC(O)CC1CNC(C1(C(F)(F)F)CC=CC1)=O 22940,C12(COC)CC(C(=O)NCC3CCC(F)(CNC(=O)CC(C)(C)C)C3)(CO1)C2 22941,C1(CC(=O)NCC(O)C2(Cl)CC2)CCCN1C(c1cnsn1)=O 22942,c1(OCC#C)cc(CNCc2noc(C3CCOCC3)n2)cc(F)c1 22943,Cc1nnn(CC(=O)NC(C)C(=O)NCc2ccn(C3CC3)n2)n1 22944,N1(C(C(C)(C)NC)=O)CCC2(CC1)CC2NC(c1cnn(CCCOC)c1)=O 22945,c1(CC)nc[nH]c1C(=O)OCCCn1cc(CCC2CCCCO2)nn1 22946,Cc1csc(Cl)c1C(=O)NCC1CN(C(=O)CC(c2cccc(F)c2)O)CC1C 22947,c1(C(=O)NC2CCC(CC(=O)NC3(CC)CC=CC3)CC2)cc2ccccn2n1 22948,c1(C(=O)NC2C(C)(C)CN(C(=O)C#CC3CCCO3)C2)nccc2ccncc12 22949,c1(C(=O)NC(CN(C(C(CCC)O)=O)C)(C)C)nn(C)c2ccc(Br)cc12 22950,CC(C)CC(C(=O)N1CCCC(CNc2ncccc2C#N)C1)C(N)=O 22951,N1(C(c2occ(C)c2)=O)CC2OCCN(C(C3CCCCS3(=O)=O)=O)C2C1 22952,N1(S(C)(=O)=O)CCc2c(NCc3cc(C4CC4)ccc3F)cccc21 22953,N1(C(CCCCC)=O)CC2(C1)CN(C(C1CCCC1)=O)CC2CO 22954,C(=O)(C(CCCC)C(C)C)N1CCN(C(CCC=CC)=O)C(C)CC1 22955,C1(C2(NC(c3c(CCCC)ocn3)=O)CC2)CCCCN1C(=O)C=CC(F)(F)F 22956,Cc1cn2c(C(=O)NCC3CC3CNC(=O)C=C3CCOCC3)c(Cl)nc2s1 22957,CC1(C)C(NC(=O)CC(=O)NCC2CC2)CCN1C(=O)C(O)Cc1ccc(Cl)cc1 22958,N1(C(C=CCCC(C)C)=O)CC(C)CN(C(=O)Cc2n[nH]cc2Br)C(C)C1 22959,c1(C(=O)NC2C(NC(C3=CCCC3C)=O)CCC2)cc2c(s1)CCCCCC2 22960,N#Cc1ccc(NC(C2CN(C(=O)CCc3ccccc3F)CCS2)=O)cc1Cl 22961,N1(C(c2c(CC)occ2)=O)CCC(C(C)C(=O)NCC2CC3C=CC2O3)CC1 22962,C(=O)(C(CCC(C)C)NC(C1CN2CCN1CC2)=O)N(CC(=O)OC)CC 22963,CC(O)CCC(=O)NC1CCC(N(C(=O)CCc2ccccc2C(N)=O)C)CC1 22964,C1(CC#C)(C(=O)NC2CCC2NC(C2CN(c3nncs3)C2)=O)CCCCO1 22965,C1(C)(COC)CC(NC(c2cc(N)ccc2Cl)=O)CN1C(=O)CCC(N)=O 22966,c1(CNC(C(CC2CC2)NC(CN2CC(CC)C2)=O)=O)ccc(F)cc1C 22967,CC(C)CC(C(=O)NC(COC(C)C)C(=O)NC1CC(C)(C)OC1(C)C)C(N)=O 22968,C(=O)(CC(C)c1ccncc1)N(C(C)C)CCNC(=O)CCSC(F)(F)F 22969,Cc1ccc(CCC(=O)NC2CN(C(C3CC4(CC4)CO3)=O)CCC2O)cc1Cl 22970,c1(C(=O)NC(CNC(C(CCC)C)=O)C(C)C)c(NC(=O)C2CC2)sc(C)c1C 22971,c1(C(=O)NCCN(C(C23COCC2C3)=O)CC2CC2)sc2sccc2c1Cl 22972,CCCCC(CNC(c1cc(C#N)c[nH]1)=O)NC(=O)COCC1CCOC1 22973,c1(C(N2C(C(C)C(=O)O)CCC2)=O)cc(C(F)F)ccc1Br 22974,CC1=C(C)CC(C(N2CCCC(N(C)C(C34COC(CF)(C3)C4)=O)C2)=O)CC1 22975,N1(C(C(COCC)C)=O)CC(N(C)C(c2cnc(SC)nc2O)=O)C2(CC2)C1 22976,c1(OC)cc(NC(c2cnc(F)c(C)c2)=O)c(OC)cc1Br 22977,c1(C(c2n(CCCOC)nnn2)NCC(c2cccs2)(C)C)nc(C)c(C)[nH]1 22978,CC1CCN(C(=O)CN(C)C(=O)C2CC2)CCN1C(C1C2CCN1CC2)=O 22979,c1(CNc2c(C(=O)NCC)nccc2)oc2ccccc2c1C 22980,C(c1ccc2c(c1)COCC2)=CC(N1CC2CCN(C(CCC=C)=O)CC2C1)=O 22981,N1(CC(N2CCCCCC2)=O)CCC2CC(NC(c3ccc(C)s3)=O)C2C1 22982,C1(C2CCC2)(C(N2CCC(C(F)F)(CNC(c3cc(C4CC4)[nH]n3)=O)C2)=O)CC1 22983,N1(C(c2c(C(C)C)nn(C)c2)=O)C(CNC(=O)COCC2CC2)CC2COCC12 22984,c1(C(N(C(C)CNC(=O)CC2CCC2)C)=O)ccc2c(c1)CCN2C(C)(C)C 22985,CC12CC(C(N3CCC(F)(CNC(=O)C4=CCCOC4)C3)=O)(CCO1)C2 22986,C1(NC(C2(CCOC)CC2)=O)CCN(C(=O)CCC=C(C)C)CC1O 22987,N#CC1(C(N2CCC3(CC(NC(c4ncccc4Cl)=O)C3)C2)=O)CC2(CCC2)C1 22988,C(C)(C)(CCC(=O)N1CCCC(COC)(NC(=O)Cc2ccco2)C1)OC 22989,C12(C(=O)NCC3CN(C(C4CCCC45CCC5)=O)CCO3)C3CC(CC13)C2(F)F 22990,c1(C(=O)NCCN(CCCN(C)C)C(C2C(C)C2C)=O)csc(Cl)c1 22991,N1(C(c2ccc(SC)o2)=O)CCCC2CN(Cc3noc4c3COCC4)CCC12 22992,C=CC(C(=O)NC(C1CCCN1C(C1CC1(C)C)=O)C)OC 22993,CC(C(=O)N1CC(CCNC(C2(C(F)(F)F)CC(O)C2)=O)C(C)C1)C(F)F 22994,C(C1c2ccccc2CCN1C(=O)COC1CC1)NC(C1CCCS(=O)(=O)C1)=O 22995,Cc1ccc(F)cc1CC(=O)NCCCC1CCCN1C(C1C2CCC1CC2)=O 22996,C(=O)(C(C)(O)CCN(C)C)N1C2C(C(=O)NCCC=CCCC)C(C2)C1 22997,C1(C(N2C(CN(C(c3c(CC)non3)=O)C)CCCC2)=O)Cc2ccncc2C1 22998,c1(OC)cc(C(N2CCC(N(C)C)C(F)C2)=O)ncc1-c1ccn(C(C)C)n1 22999,S(=O)(=O)(c1ccc(F)c(F)c1)N1CCC(NC(c2ccc(C(N)=O)nc2)=O)C1 23000,Cc1cc(O)ncc1C(=O)NCC1C(C(=O)NCCC(F)(F)F)CC1 23001,CC1(C#N)CCN(C(=NC2CCC2)NC2CC3(CCCCC3)C2)CC1 23002,CCC(C)C(O)C(C)C(=O)NCC(C)=CC(N1CCC(O)(CO)C1)=O 23003,c1(C(N2CCC(C3(NC(C4CC4(F)F)=O)CC3)C2)=O)ccc2ncccc2n1 23004,N1(C(c2n[nH]c(CC)c2Cl)=O)CCCC(O)(CNC(C2CC23CCCC3)=O)CC1 23005,N1(C(c2c(CC)cno2)=O)CC(CNC(=O)C(F)C2CCCC2)C2(CC2)C1 23006,N1(C(C=CC(=O)OCC)=O)CCN(C(c2coc(Br)c2)=O)C(CF)C1 23007,c1(NC(CNC(CNC(C(CC=C)C)=O)=O)=O)ccc2ccncc2c1 23008,CCCC(C)(O)CNC(C1(CNC(=O)C(n2ccc(C)n2)C)CC2(CC2)C1)=O 23009,C1(C(C(=O)O)NC(c2nc(CCP(C)(C)=O)sc2)=O)CC2C=CC1C2 23010,C1(N(C(=O)CN(C)C2CC2)C)CCN(Cc2ncccn2)CC1 23011,c1(SC)ccc(CN(C(c2cc(C)ns2)C(=O)NCC(F)F)C2CC2)cc1 23012,C=C(CNC(=O)C(C)(C)C1CCCC1)CCNC(=O)CSCCOC 23013,C(C(=O)NC1CCN(C(C2(OC)CCCC2)=O)C1)(C(C)C)N(CC)CC 23014,C1(CNC(C(CC=CC)C)=O)CN(C(c2cc(Cl)cs2)=O)CC1(F)F 23015,c1(C(=O)NCCC2CN(C(C3CCCS3)=O)CCO2)coc2c1COC2 23016,N1(C(c2cn(CCCOC)nc2)=O)CC(O)CC1CNC(=O)COC1CC1 23017,Cc1nc2[nH]c(C(N3CC4CCC(NC(=O)CCNC(N)=O)(C4)C3)=O)cc2s1 23018,N1(C(C(C)OCC(F)(F)F)=O)CCC2(CC1)CC2CNC(=O)CN1CC(C)(C)C1 23019,Cc1cc(N2CCC3CC3C2)ncc1S(=O)(=O)NCc1csc(Cl)c1 23020,C1(NC(C2C(NC(Cc3n(C)ccn3)=O)COC2)=O)CCCCC12CC2 23021,N1(C(c2cc(OC)nc(F)c2)=O)CCN(C(c2c[nH]nc2C(C)C)=O)CC(O)C1 23022,c1(OC)ccc(F)c(C(c2nnnn2C2(C)CC2)NCCn2cncn2)c1F 23023,C1(CNC(=O)CC2=CCCC2)CC2CCC1N(C(=O)CC1CCC3CC13)C2 23024,N1(C(c2c(-c3cn(C)nc3)onc2)=O)CC=C(CCNC(c2ccsc2)=O)CC1 23025,C1(O)(C(C)NC(C(C)OCC=C)=O)CN(C(=O)C=Cc2ccc[nH]2)C1 23026,c1(COC)ccccc1NC(=O)CCC(=O)NC(c1cccc(C(F)(F)F)c1)C 23027,c1(C(N2CCCC(CCNC(C(CN(CC)CC)F)=O)C2)=O)cnc(O)cc1O 23028,c1(CC(=O)NC2C(C)N(c3ccnc(Cl)n3)CCC2)nsc2ccccc12 23029,c1(NC(C2CC2C(=O)Nc2ccc(C3CC3)cc2)=O)cncc(C2CC2)c1 23030,c1(C(=O)NCCNC(c2cc(-c3c(F)cccc3F)on2)=O)cc2c(s1)CCC2 23031,CC1CCC(C)N1CC(=O)NCCc1ccc(C(=O)N(C)C)cc1 23032,c1(OC)ccc(C(N2CC3CC3(NC(c3cc(C4CCC4)[nH]n3)=O)C2)=O)c(N)c1 23033,N1(CCC(=O)NC2CC(C)(NC(C3C=CCCC3)=O)C2)CCCS1(=O)=O 23034,c1(C(=O)NC2(CCCCNC(c3c(C)nns3)=O)CC2)cc2ccccc2n1C 23035,c1(OC)cccc(CC(C)CC(=O)NCC2(NC(=O)C(C)C3CCC3)CCC2)c1 23036,c1(C(=O)NC2(C)CC(NC(C(C)(C)NC(=O)OC)=O)C2)cc(OC)cc(Cl)c1F 23037,C1(NC(C(C)OC(C(C2CC(F)(F)C2)OC)=O)=O)CCC(F)(F)CC1 23038,CC(C)CC(F)C(=O)NCC1C2CCC(C2)N1C(C1CCN(C(=O)N(C)C)CC1)=O 23039,c1(OC)cc(F)cc(C=CC(=O)NC2CCC2NC(=O)C2=CCCCCC2)c1 23040,CCC(C)(CCNC(c1nocc1C)=O)NC(=O)COC1(C)CCCC1 23041,N1(C(C(=O)N(C)CC2CC3CC3C2)=O)CCCC(N2CCCC2)C1 23042,c1(C(=O)NCCN(CC(C)O)C(=O)CC2CN(C)CC2O)ncc[nH]c1=O 23043,C(=O)(C(C(C)(C)S(C)(=O)=O)NC(=O)OC(C)(C)C)N(C1CCC(C)CC1)CCO 23044,N1(C(C(C)(C)NC(C2C(C)C2)=O)=O)CCc2ncccc2C1 23045,N1(C(CC2CCC(=O)NC2)=O)CC2CC3CC2C1C3NC(C1CCC2(CC2)C1)=O 23046,CC(C)(O)C(C(=O)NOC1CC1)NC(c1ccc(=O)n(C)c1)=O 23047,C(=O)(C(O)CCCC)N(C)CC1OCCN(C(C2(C=C)CC2)=O)C1 23048,N1(C(C(F)=CC)=O)CCC2CN(C(C3CCN(c4ccccc4)C3)=O)C2C1 23049,C1(C(N(C(C)CNC(C2(CCF)CC2)=O)C)=O)CCC(NS(C)(=O)=O)C1 23050,c1(NCc2cc(C)cc(N)c2)cc(Br)ccc1S(=O)(=O)N1CCCNC(=O)CC1 23051,N1(C(c2n[nH]cc2Br)C(=O)NCc2cccc(OC)c2)CCNC(=O)C1C(C)C 23052,C12(C(C)NC(C3(C)CC3)=O)CC(NC(C3CN(CC(F)F)C3)=O)(C1)C(C)O2 23053,c1(C(CF)NC(=O)Nc2ccc(CCC(=O)OC)cc2)ccc2c(c1)OCCO2 23054,C1(OC)CN2CCCC2(C(=O)NC2CC(NC(c3c(Cl)cccc3Cl)=O)C2)C1 23055,N1(C(c2n[nH]c(C)c2C)=O)CC2CN(C(C3CCC([N+](=O)[O-])CC3)=O)CCC12 23056,N1(C(C=C(CC)CC)=O)CC(CNC(C2(CO)CCOCC2)=O)C2(CCC2)C1 23057,N1(C(C2C(CNC(C3CCCS3)=O)CC2)=O)CC(F)(F)C(F)(F)C1 23058,C#Cc1ccc(C(=O)NC2CN(C(=O)Cc3sc(O)nc3O)CC23CC3)cc1F 23059,CC1CCC=C1C(=O)NCC1(O)CN(C(C2CCCC(C#N)C2)=O)C1 23060,Cc1ncnc(C(N2CCC(NC(=O)CC3C=CCCC3)C2(C)C)=O)c1C 23061,C1(NC(CC)=O)(CNC(C2CCN2S(C)(=O)=O)=O)CCC(C)(C)CC1 23062,C1(O)(CC(N)=O)CCN(C(c2ccc(O)nc2)C(=O)Nc2ccccc2Cl)CC1 23063,c1(C(N2C(CNC(C3N(C)CCCC3)=O)CC(O)C2)=O)ccc(N)c(Cl)n1 23064,C1(CN(C(CC(=O)OCC)=O)C)CN(C(C2(C)CCN(C)C2)=O)CCO1 23065,c1(OC)cccc(C(=O)NCC23CC2CN(C(=O)C(CC2CC2)OC)C3)c1C 23066,Cc1cc(N2CC(F)(F)CC2CNC(=O)C(c2cccnc2)O)n2ncnc2n1 23067,S(=O)(=O)(c1ccccc1Cl)NCCC(=O)N(C)CCNC(c1ccns1)=O 23068,c1(CC(N2CCN(CC3CCCN(C(COC)=O)C3)CC2)=O)csc2nccn12 23069,S(=O)(=O)(c1cccc(=NCC(C)c2cccs2)[nH]1)NCCCCCC(=O)NC 23070,N1(S(CCOC)(=O)=O)CCC(N=c2nc[nH]n3cc(Br)cc23)C1 23071,C1(NC(c2ccn(C(C)C)n2)=O)CC(CNC(c2cc(C(N)=O)cs2)=O)C1(C)C 23072,C1(CNC(c2cccc(C)n2)=O)CN(C(=O)C(C)(C)C2CCCO2)CCN1C 23073,C1(C(C)C)CCC(NC(c2nc(NS(=O)(=O)CC#N)cn2C)=O)CC1 23074,C1(NC(CCCCCC)=O)CC2CN(C(c3cc(C)n(C(C)(C)C)n3)=O)CC2C1 23075,c1(C(=O)NCC2OCCCN(C(C(C(C)C)F)=O)C2)ccc2c(c1)C(C)(C)CO2 23076,C1(S(N)(=O)=O)(C(=O)NCCCOCCCNC(C2(SC)CC2)=O)CC1 23077,C(=O)(CC(C)C(C)(C)C)NCCN(C(C(CC)CC)=O)CC1CC1 23078,C(CO)(C(F)(F)F)NC(C(CC1CCCC1)NC(=O)CCC1CC1)=O 23079,N1(C(C=C(C)c2cccs2)=O)CCN(C(c2ccc3cc[nH]c3n2)=O)CCC1C 23080,C1(C(N2C(CNC(c3ncoc3C(F)(F)F)=O)CCC2)=O)CCC2(CCC2)C1 23081,c1(OC)cccc(C(N2CCC(CF)(NC(=O)Cn3cccn3)C2)=O)c1 23082,c1(NC(C2CN(C(c3cnc(Cl)cc3I)=O)C2)=O)nc(Br)ccc1Cl 23083,N1(C(CC(C(C)C)O)=O)CC(C)(CNC(=O)COCCCN(C)C)CC1(C)C 23084,C#CCCCCC(=O)NCC(CC(=O)NCC(=O)OC(C)C)C1CCC1 23085,N1(C(CC)=O)CCN(C(c2[nH]ccc2-c2ccccc2)=O)CC1CC1CC1 23086,Nc1ccc(C(N2CC(CC(=O)C(=O)O)C2)=O)cc1Cl 23087,CN1CCCC1C=CC(N1CCOC(CNC(=O)CC(C)(C)c2cccs2)C1)=O 23088,C1(C(=O)NCCC2CCN(C(=O)C(C3CCC3)C3CCC3)C2)CC(F)C(=O)N1 23089,c1(CNC(c2cc(CC)on2)=O)ccc(CNC(C2(C)COC2)=O)cc1F 23090,C1(C(C(=O)N(CC(C)NC(c2nnc(C(C)(C)C)o2)=O)C)C)CCOCC1 23091,c1(SC)cc(F)ccc1C(=O)NCCOCCNC(=O)COCC(F)F 23092,C1(N(C(CN(C)C(C)C)=O)CCO)CCN(C(c2cc(CC3CCC3)c[nH]2)=O)C1 23093,N1(C(C(CC)O)=O)CCN(C)CC1C(=O)NOCC(F)F 23094,CN1CC(NCCc2c[nH]c3cc(F)ccc23)CCc2ccccc21 23095,c1(C(C(N2CC(N(C(CCC#C)=O)C)C2)=O)C)cccc(Br)c1 23096,c1(C(N2CCC(N(C(c3coc(O)n3)=O)CC)C2)=O)cc(F)c2ncccc2c1 23097,c1(C(=O)NCCC(=O)NC(C(C)NC(c2ccsc2Cl)=O)(C)C)ncc(F)cn1 23098,Cc1ccc(C2CC2NC(C2CC(C)CCN2C(=O)C(O)C(F)(F)F)=O)c(Cl)n1 23099,c1(C(N2CC(NC(C3C(C(C)C)C3)=O)C3(C2)CC3)=O)cc(Cl)cc2ccncc12 23100,N1(C(CCCOC(C)C)=O)CC2(CC(NC(c3csc4cncn34)=O)C2)C1 23101,C1(N(C(C2C(OCC)C2)=O)CC)CCN(C(=O)Cc2cccc(F)c2)CC1 23102,N1(C(COC(C)C)=O)CCC(O)(CN(C)C(c2cn3ccsc3n2)=O)CC1 23103,CN1CC2C3CCN2C(=O)N2CC1=C3C2.C1(OC(C)(C)C)CCC2(C1)CC2(F)F 23104,C(CN=c1nc2scnc2c(NCC2CC2C2CCCC2)[nH]1)N(C(=O)OC)C 23105,Cc1ccc(C(O)C(=O)N(c2cnncc2C)C2CC3(CNC3)C2)nc1 23106,c1(C(=O)NCC2C(C)CCN(C(C34CC(C3)C4)=O)C2)ccc2nn[nH]c2n1 23107,c1(C(N2CCCN(C(C3CC4CCC3O4)=O)CC2)=O)ncc(F)cc1F 23108,n1(C(C)C)cc(C(=O)NC(C2CCOC2)CNC(c2cc(C(F)F)no2)=O)nn1 23109,N1(C(c2n(CCCC)ncc2)=O)CCCN(C(=O)CCCSC(C)(C)C)C(C)C1 23110,C1(NC(c2c(CC)c[nH]c2)=O)CC2CCC1CN(C(=O)CC(C)C(C)C)C2 23111,c1(N2CCCC(SCC(=O)Nc3ccc(C)cc3)C2)cc(C(=O)O)c(Br)cn1 23112,C1(NC(CC2(N(C(Cn3ccc(C)c3)=O)C)CC2)=O)CCC2(CC2)C1 23113,C1(OCC)CC2(C1)CC2NC(C1C=CCN1C(C1CCC1COC)=O)=O 23114,N1(C(C2COC(=O)O2)=O)C(CNC(C2(C(F)F)CC2)=O)CC2COCC12 23115,C1(CC(=O)Nc2cccc(Oc3nccs3)c2)CCC2(CCCC2)CC1 23116,N1(C(c2cnc(C(C)(C)C)nc2)=O)CC(NC(C2CCCC2)=O)CC(C)(C)C1 23117,N1(C(c2c(C)ccnn2)=O)C2CCCC1CN(C(c1cnc(O)cc1O)=O)C2 23118,CCS(=O)CC(=O)NCC(CCOC)NC(C1COCCOC1)=O 23119,c1(CC)c(C(=O)NCC2CCC(C(=O)NC3(CCO)CCC3)O2)nnn1C 23120,C(=O)(C(CNC(c1cnsc1C)=O)CC(C)C)NCc1c(C)nc(C)[nH]1 23121,Cc1cc(C(=O)NC(C)CCNC(=O)C=Cc2cnccc2C)ccc1C#N 23122,c1(-c2cnc3c(c2)N(C(C=CC=CC)=O)CC3)ccc2c(c1)n(C)c(=O)n2C 23123,c1(CNC(c2occc2CNC(C2C=CCCC2)=O)=O)ccc2n[nH]cc2c1 23124,c1(C(N(CCC(C)NC(c2csnn2)=O)C)=O)ncccc1C1CC1 23125,n1(CC)c(C)cc(C(=O)N(C2CC(NC(=O)C(F)C(C)C)C2)C)c1C 23126,C1(CNC(=O)NC(C)CN2CCOCC2)CCCS1(=O)=O 23127,c1(N(C)Cc2nccc(C)c2)nc(=NC2CCN(C)C2C)[nH]c2cc[nH]c12 23128,CC(C)C(CC(=O)N(CC(C)CNC(=O)CC(C)(C)C)C)c1ccccc1 23129,C1(F)(C(=O)NCC23CC(CNC(C(CC)COC)=O)(OC2)C3)CCC(F)(F)CC1 23130,c1(C(=O)NC(CC)CN(C(=O)C(C)(C)C(C)C)C)[nH]c(C2CC2)c(C(=O)OC)c1C 23131,C(=O)(C#CC1CCCCO1)NCCN(C(C(CSC)C)=O)C 23132,C1(C(C)CNC(C2CCC(=O)C2)=O)CCN(C(=O)Cc2cccc(Cl)c2)CC1 23133,C#CCC(C)(CC)C(=O)NCCN(CCOC)C(c1cc(C)[nH]n1)=O 23134,CCC(CCOC)C(=O)NC12CCC(C1)N(C(c1sccc1-n1ccnn1)=O)C2 23135,CC1CN(C(C2CC3C=CC2C3)=O)CC1NC(c1cnn(C)c1N)=O 23136,N1(c2c(S(=O)(=O)NC3CCOC4(CCC4)C3)cccn2)CCOCC2(CCCC2)C1 23137,N1(C(c2ncc(C)c(C)c2)=O)CC(NC(=O)CC2CCCCN2C)C2(CCC2)C1 23138,N1(C(C(C)NC(c2ccc(Cl)cc2)=O)=O)CC2(C(=O)ON)CC1CCO2 23139,C1(N(C(c2c(C)ocn2)=O)C)CCCC(N(C)C(c2ccon2)=O)C1 23140,C1(C(N(C)Cc2ncc(C)o2)C)CCCCCC1 23141,Cc1cccc(C(N2CCOCC2CCNC(=O)CC2CCC23CCC3)=O)c1F 23142,C1(C(N2C(CC(NOCCOCCOC)=O)CC2)=O)CC2(CCC2)C1 23143,Cc1onc(Cl)c1NC(=O)C(=O)NCc1nccn1CC(C)C 23144,C1(NC(COC(C)C)=O)C2CC1N(C(c1ccnc(CN(C)C)c1)=O)C2 23145,C1(CC(NOCCCCC)=O)CN(C(=O)CC2CCOC2C)CC1C 23146,C1(n2cc(CNC)nn2)CCCN(C(=O)C(C)(C)c2ccc(Cl)s2)C1 23147,C1(C(=O)NCC2C(C)CCN2C(=O)Cc2cnco2)CC2CC1C1CC21 23148,C1(CC)CN(C(c2sccc2Cl)=O)CCN1C(=O)Cc1ccc(Cl)nc1 23149,c1(C(N2CC(CNC(C(c3c(C)cncc3)C)=O)C2)=O)cc2c(s1)CCSC2 23150,c1(CC(N2CCCC(NC(C3C(C=C)C3)=O)CCC2)=O)ccc2c(c1)CCCO2 23151,c1(C(C(=O)N(C(CNC(Cc2c(OC)cccc2)=O)C)C)C)cc(C)cc(F)c1 23152,N1(C(CC2(C)CCOC2)C(=O)NCCN2CCOCC2)Cc2ccccc2CC1 23153,C1(CC)C(NC(=O)C=C2CCC(C)C2)CCN1C(c1oc(C(F)(F)F)nc1C)=O 23154,C1(CC=C)(NC(=O)CCOCC2CCCO2)CCN(C(=O)C(C)=C2CCC2)CC1 23155,c1(NC(c2ccc(Cc3nc(C)sc3)cc2)=O)ccc2nn(C(F)F)cc2c1 23156,Cc1cc(C(N)=O)cc(C(=O)N(C)CCN(C)C(c2c(C)cccc2Cl)=O)c1 23157,C(C(=O)N1CCC(CO)(NC(=O)Cn2nnc(C3CC3)n2)C1)(C(C)C)OCC 23158,C(C(C)(CCO)NC(C1CCC2(CC2)C1)c1nnnn1C1CC(F)(F)C1)OC 23159,CC(C)CCC(O)C(=O)NC1CCN(C(=O)CC2(O)CCCCC2)CC1F 23160,N1(C(C(C(C(CC)C)O)C)=O)CC=C(C(C)(C)C(=O)N(CCC(N)=O)C)C1 23161,c1(C(C)NC(c2ccc(OC)c(Cl)c2N)=O)cc2c(cc1Br)OCCO2 23162,c1(C(N2CC3C(C(=O)NCc4cn(C(C)C)nc4)(C3)C2)=O)cc(I)ccc1O 23163,c1(C(=O)NCCCC2CCCC2O)ccc(S)nc1 23164,C(=O)(C1CSc2ccccc21)NCCC1CC(NC(c2c(CC)nn(C)c2)=O)C1 23165,N1(C(C(c2cnn(C)c2)C)=O)CCOC(C(=O)NC2COCC2CN(C)C)C1 23166,C(=O)(C(F)(F)CC(C)C)NC1CC2(C(NC(c3c(C)n(C)nn3)=O)C2)C1 23167,C1(C2CC2)(NC(c2c(C)cc(CC)o2)=O)CCN(C(C2CCCNS2(=O)=O)=O)C1 23168,CC1(NC(C2(NC(=O)Cc3ccsc3)CC(F)C2)=O)CCCC1O 23169,c1(C(=O)NCC2C(NC(C=Cc3c(C)cncc3)=O)C2)c(Cl)cccc1[N+](=O)[O-] 23170,c1(N2CC(C(C)C)C(O)CC2)nc(=NCC(C(C)C)N(C)C)[nH]c2c1COCC2 23171,C1(CNC(c2ncncc2Cl)=O)CCCCN1C(=O)CCc1cccc(Br)c1 23172,c1(NC)cnncc1C(N1CCC(C(=O)NCC(C)C#N)(CO)C1)=O 23173,c1(N(CCOCCN(C(c2ccc(SC)cc2)=O)C)C)cc(Cl)nc(SC)n1 23174,C1(NC(c2cc(OCC)ncc2)=O)CN(C(=O)C(O)CC(N)=O)CC1(C)C 23175,N1(C(c2cncs2)=O)CC2CCC1C1CN(C(C3(CO)CCC3)=O)CC21 23176,c1(CN(C(=O)C(C)(C(C)C)OC)CC)nc2ccccc2[nH]1 23177,c1(C(N(CC(CNC(C2C(C)OCCC2)=O)(C)C)C)=O)nccc2cccnc12 23178,C(CNC(=O)C=Cc1ncc[nH]1)(CCCC)NC(C1(CC#C)CCCO1)=O 23179,C1(C(C=O)F)CCNCC1.c1(C(C)N(CC(c2ccccc2)F)CC)ccccc1 23180,CC1=C(C(=O)N2CCN(C(C3CC4C=CC3C4)=O)C(CF)C2)CCS1(=O)=O 23181,C#CCCCCC(=O)NC1CC2(C1)CC2NC(c1ccc(-c2ccc(=N)[nH]c2)o1)=O 23182,CCCC(CC(C)C)C(=O)N1CCC(N(C(c2nocc2Br)=O)CC)CC1 23183,N1(C(c2ccc(C(=O)OC)o2)=O)CC(NC(c2cscc2Br)=O)C(F)C1 23184,CC1=C(C)C(OC(c2cnc(C3CC3)nc2)=O)CCC1 23185,c1(NC(C(C)F)C)[nH]c(=NCCC(C)(C)S(C)(=O)=O)nc2c1ncn2C 23186,C12(C(N3CCC(N(C(c4c(C)cc(SC)o4)=O)C)C3)=O)CCC(CC1)C2(C)C 23187,C1(C2CCCO2)(C(=O)NCC(C(=O)OCC)C)CCCCC1 23188,c1(COC(C(COCC)NC(c2cnn(CC3CC3)c2)=O)=O)c(C)[nH]c(C)c1C 23189,c1(SCC)ccc(C(N2CCCC(CCNC(c3ccc(Cl)nn3)=O)C2)=O)cc1 23190,C(=O)(C1=CC2(CCN(C(=O)C(O)Cn3cncn3)C2)C1)NCCC(CC)C 23191,N1(C(C2(CC)CCC2)=O)CCN(C(=O)Cc2coc(-c3cccs3)n2)CC(O)C1 23192,c12c(cccc1F)C(c1nnnn1C)N2.C1(C)CCC(=O)S1.C(C)(C)(C)OCC 23193,Cc1ccc([N+](=O)[O-])c(NC(C2CCCN(Cc3ccc(Br)o3)C2)=O)n1 23194,C1(NC(C=C2CCC(C)C2)=O)CN(C(c2nc(=O)n(C)[nH]2)=O)CC1C(F)F 23195,C1(C)(CNC(CCc2c(C)cccn2)=O)CCCN(C(=O)CC2CC2)C1 23196,C1(CNC(c2c(Cl)nc(OC)s2)=O)CCCCN(C(=O)C(C)C2CC2)CC1 23197,C1(CCC(=O)NC2(C3N(C(C4(C#C)CC4)=O)CCC3)CC2)CCCC(=O)N1 23198,CCC(C)C(C(=O)NC(C)CNC(c1cccc(NC(N)=O)c1)=O)NC(=O)OC 23199,C(C(F)(F)CCC(=O)NC(C)CCc1ccc(C)cc1)n1cc(CCOC)nn1 23200,c1(C(=O)NCCC2(NC(COCCCC#C)=O)CC2)cc2c(s1)CC(C)CC2C 23201,C(=O)(CCC#Cc1ccccc1)NC(C)CCNC(c1ccn2ncnc2c1)=O 23202,C1(CNC(CC2CC(C)(C)C2)=O)CCCCN(C(=O)CC2CCCO2)CC1 23203,C1(C(=O)NCC(F)CNC(c2sccc2SC)=O)(COC)CC=CCC1 23204,CC1Oc2c(C(=O)NCC3(NC(=O)CC4CCCCC4)CC3)cccc2C1C 23205,N1(C(c2cnnn2C)C(=O)NC)CCN(C(C)=O)CC1.c1(C(C)=O)ncc[nH]1 23206,Cc1c(C(=O)NCCCCCCNC(=O)CC2CCCC(C)C2)cccc1O 23207,CCCCCC=CCC(=O)NC(C)CC(C)NC(=O)CSC(F)F 23208,N1(c2c(C)nccn2)CCC(O)C(C(=O)NCC2CCCC(=O)N2C)C1 23209,C#Cc1ccc(NC(=O)C(CNC(=O)C(C)C(C)CC)CCC)cn1 23210,N1(C(C(=O)NC(c2ccc3c(c2)OCCO3)C)=O)CC(=O)NCCNC(=O)C1 23211,C(=O)(C(O)CNC(=O)CCC1CCCCC1)N1CC(CCOC)C1 23212,N1(C(CCSc2nc(C)sc2)=O)CC2(CCN2C(=O)CCCCNC(N)=O)C1 23213,CCCCC(O)CCC(=O)NC(CNC(c1ccc2nc[nH]c2c1)=O)C(C)C 23214,C1(C(=O)NC2CN(C(C3CCCN(C(C(C)C)=O)C3)=O)C2)CC2CC1CC2(F)F 23215,N(C1CCc2c(Br)cccc21)C(C1CC1C(=O)Nc1cccc2nc(O)oc12)=O 23216,C1(C(N2CCC(C(=O)Nc3ccc(CC)c(Br)c3)CC2)=O)Cc2ccccc2C1 23217,c1(CNC(Cn2ncc(CC)c2)=O)cccc(C(=O)NCc2[nH]nnc2C)c1 23218,C1(C(N(CCCN2CCNCC2)C)=O)CC2(CCO1)CC(F)(F)C2 23219,c1(C(=O)NC2(CCNC(c3ccncc3-n3cccn3)=O)CC2)ccc(F)cc1 23220,c1(OCCC(=O)NCC2CCCN2C(c2nn[nH]c2Cl)=O)ccccc1F 23221,CC1CCCC(C(=O)NCC2(CNC(c3cn[nH]c3)=O)CC(F)(F)C2)C1 23222,N1(C(=O)NCCc2ccon2)CCC2(CC1)CC2c1cccnc1 23223,Cc1ncnc(C(=O)N(CC(C)N(C(=O)CN2CCN(C(C)C)CC2)C)C)c1C 23224,C1(NC(c2cnn(CC)n2)=O)CCC2(CC1)CC2NC(=O)CCC1CCCCO1 23225,c1(C(=O)NC(C(C)NC(c2nn(C)cc2N)=O)C)cnc2cccnn12 23226,S(=O)(=O)(c1c(C)sc(C)c1Br)NCCOc1ccc(OC)cc1C(=O)O 23227,C1(CC(=O)NCCCN(C(C)C)C(C2CCC2)=O)CCCC(C)(C)O1 23228,N1(CC)CCC(NC(=O)C(CC2CCC2)NC(=O)CSc2cn[nH]c2)C(C)C1 23229,O=C1CC(C(N2CC(CC(F)C(N3C4CCC3CC4)=O)C2)=O)CCN1 23230,O=C(C1=CCCCCC1)NCC12CCC1CN(C(c1nncs1)=O)C2 23231,CC(CC(=O)NCC1(F)CCN(C(c2cnc(Cl)cc2N)=O)C1)C(C)(C)C 23232,C1(NC(c2cnc(Cl)s2)=O)CC(O)CN(C(C2CC2c2ccccn2)=O)C1 23233,c1(C(=O)OC)cnn2c1CC(Nc1nn3cc(CC(C)C)nc3s1)CC2 23234,C(=O)(C(CC)CCCCC)N1CC(NC(c2cn(CC=C)nc2)=O)C(F)CC1 23235,Cc1ccccc1C=CC(N1CCC(NC(C2CC2[N+](=O)[O-])=O)C(O)C1)=O 23236,c1(C(=O)NC2(CNC(CSSC)=O)CCC2)c(Cl)nsc1Cl 23237,C12(NC(c3ccc(CC)c(C)c3)=O)CCCC1N(C(c1cncn1C)=O)CC2 23238,c1(C(N2CCN(C(C3C(C)(C)NC(=O)C3)=O)C(CO)C2)=O)cnn2ncccc12 23239,C(=O)(C1Cc2ccc(F)cc21)N1CC(CCNC(CS(CC(=O)OC)(=O)=O)=O)C1 23240,N1(Cc2ccn(CC)n2)C=CCCC2CC1C2(C)C 23241,Cc1cc(NC(=O)NC2(C(=O)Nc3ccccc3)CCCCC2)cnc1Br 23242,C12(NC(Cc3c(C)occ3)=O)CCCN(C(c3ccc(Cl)c(F)c3F)=O)CC1C2 23243,C(=O)(C1=NOC(C(C)(C)C)C1)N1CCCC(N(C(C2C3CCC(F)C23)=O)CC)C1 23244,N1(C(C(COCC)n2cc(C3CCCC4CC34)nn2)=O)CCN(C)C(C(F)F)C1 23245,c1(C(=O)NCCOCCNC(COCCOC)=O)c(Br)sc2nnsc12 23246,C(=O)(C1=CC2C=CC1C2)N1CCC(C)(CNC(C2=CCCC2C)=O)C1 23247,CCCC(C(=O)N1CC(CCNC(C2CCCC(O)C2)=O)(OC)C1)N(C)C 23248,Cc1ncncc1C(N1CC(NC(C2CCCCC2)=O)C(C)C1)=O 23249,C1(C(N(CCN2CCN(C(C(=O)NCC)C)CC2)C)=O)CC2CCC1CC2 23250,c1(CCNC(CN2CCCC(CNC(CC)=O)C2)=O)ccc2cnccc2c1 23251,C1(C(=O)OC(CC#C)CC)CC(=O)N(C)C1c1ccc(F)cc1 23252,Cc1ccc2c(c1)C(NC(C1CCC1)=O)CCCN2Cc1cccc(Br)n1 23253,N1(C(c2cccc3c([N+](=O)[O-])c[nH]c23)=O)CC=C(c2cccc3ccccc23)CC1 23254,C(CN=c1cc(C)nc(-c2ccccn2)[nH]1)N(C(=O)Cc1csnn1)CCN.CO 23255,c1(CC(=O)N(CC(Cn2cc(C3(C)CCCO3)nn2)OC)C)c(F)cccc1Br 23256,N1(C(C(C)OCCC(C)C)=O)C(C(=O)Nc2cnccc2C(C)C)CC2CC12 23257,CC(C)C(C(=O)NCCn1ccc(C(=O)O)c1)S(=O)(=O)C1CCCCC1 23258,C(=O)(C(F)CC(C)(C)NC(=O)C(c1ccc(C)cc1)C1CC2CCC1C2)OCC 23259,c1(C(N2CCC3(CCCN3C(=O)C(F)C3CC3)C2)=O)ccc([N+](=O)[O-])cc1O 23260,C(C1COCc2ccccc21)NC(=O)NC1CCCC(C)(C)O1 23261,C1(COC(=O)NCC(=O)OCC(C=C)O)CC(=O)N(c2ccccc2)C1 23262,CC1ON=C(C(=O)N2CC(NC(c3c(Cl)cnn3C(C)C)=O)C(C3CC3)C2)C1C 23263,c1(OCOC)ccc(F)c(F)c1-c1ccc(CNC(c2ccc(F)cn2)=O)nc1 23264,N1(CC)CC(C)N(c2nc(C)nc(N3CCOCC3)n2)CC1C 23265,C1(NC(C)=O)CCC(C(N2CCC(NC(c3cn(C(C)C)cc3C)=O)C2C)=O)CC1 23266,N1(C(c2c(C)n[nH]c2)=O)CC2CC1(CNC(=O)C(C)(O)Cc1ccccc1)C2 23267,c1(CC)nnc(=NCC2CCCC2NC(c2sc(C)nc2C)=O)[nH]c1CC 23268,N1(C(C=CC=CC)=O)CCc2ccccc2C1CNC(=O)CCc1scnc1C 23269,N1(C(c2cncc(C(C)(C)C)c2)=O)CCN(C(c2csc(Cl)c2Cl)=O)C(CO)C1 23270,c1(SCC)ccccc1NC(=O)C(C)Oc1cccnc1F 23271,c1(NC(C(CC)(C)CNC(=O)C(C)CN(C)C)=O)cnc2ccnn2c1 23272,C(=O)(C1=CC2CCCC12)N(C)CC1N(C(c2cccc(CC)c2N)=O)CCCC1 23273,N1(C(C(CC(C)C)C(C)C)=O)CCCC2(CCCN2C(=O)COCP(C)(C)=O)C1 23274,N1(C(C2(CNC(C(C)=NOCC#N)=O)CCCO2)=O)CC[Si](C)(C)CC1 23275,c1(C(=O)NCCCCOCC)c(-c2cncc(OC)c2)ncn1C 23276,Cc1cccc(C)c1CC(N1CCCC(NC(C2(O)CCC2)=O)C1)=O 23277,CC1=C(C(=O)NCC2CCCN(C(=O)CCCc3nccs3)C2)CCC(C)(C)C1 23278,c1(C(=O)NCC2CCC(NC(C=CC=CCC)=O)C2)ccc(P(C)(C)=O)s1 23279,C1(CCCCNC(c2c(CC)cno2)=O)CCN(C(=O)C(C)=CC2CC2)CC1 23280,S(=O)(=O)(c1cccnc1NCC(CO)C(F)(F)F)NCC1CCC(=O)NC1 23281,N1(C(COCc2c(C)cccc2)=O)CC2CC(NC(c3ccncn3)=O)C1C2 23282,c1(C2(C(=O)NC(CNC(CCSC)=O)C3CCC3)CC2)cc(C)no1 23283,Cn1nc(CN2CCC(Nc3ncccc3C(F)(F)F)C2)c2c1CCCC2 23284,c1(N2CCC(NC(c3nc(Cl)ccc3F)=O)(CF)C2)ncc([N+](=O)[O-])cc1Br 23285,C(=O)(C1=CS(=O)CCC1)N1CC(NC(=O)CCCn2cccn2)C(O)C1 23286,N1(C(COCCSC)=O)CCC2(NC(C3CCN(C)C(=O)C3)=O)CCCCCC12 23287,C(=O)(CC(C)CN(C=O)Cc1nc(C2CCOC2)n[nH]1)NC 23288,N1(C(CC(CCC)NC(c2oc(C)nc2C)=O)=O)CCC2(CCCCC2)C1 23289,CCC(CC(F)(F)F)C(=O)N1CC2(CNC(C3CCC(C)CC3)=O)CC1CO2 23290,c1(C(=O)NCCN(C(=O)CC2CCCC23CC3)C(C)C)ccc(C(F)(F)F)cn1 23291,c1(C(=O)NCC(CN(C(c2ccsc2Cl)=O)CC)(C)C)cc2sc(C)cc2[nH]1 23292,N1(C(c2cccc(OC)c2F)=O)CC2CCC1CN2C(c1ncccc1Cl)=O 23293,CC1(C)CCC(CNC(C2(C)CCCS2(=O)=O)=O)N(CC(N2CCOCC2)=O)C1 23294,N1(C(c2nc(C(C)C)oc2)=O)CCn2nc(C(=O)N(c3ccccn3)C)cc2C1 23295,c1(C(=O)NC(C2CC2C(=O)Nc2cncc(Cl)c2)C)ccnc(O)c1 23296,O=C(C1CCCn2c(Br)cnc21)NC12CC(C1)N(C(C1CC1F)=O)C2 23297,C1(C(=O)NC2(C)CCN(C(c3n(CC)cc(Cl)c3)=O)C2)CCc2ncnn2C1 23298,C(C(=O)N=S(C)(=O)c1cnn(C)c1CN)c1c(OCC(C)C)c2c([nH]1)cccc2 23299,C#CCCCC(=O)NC1CCOC(C2CCN(C(=O)Cn3ccsc3=N)CC2)C1 23300,CCS(=O)(=O)CC(=O)N1CCC(N(C(c2ccncc2)=O)C)C1.C1(N(C)CC)CC1 23301,N1(Cc2cc(C)ncc2)CC2CN(C(c3cccc(C)c3I)=O)CC12 23302,c1(C(=O)NC2C(NC(C3(C)CC4CC4C3)=O)CCOC2)cc2nn[nH]c2cc1F 23303,C1(C(N2CCCC(NC(c3c(C)nc(C)s3)=O)C2C)=O)CCOC2(CCCC2)C1 23304,Cc1ncnc(C(N2CCC3CC23C(N2CC=CCC2)=O)=O)c1C 23305,c1(Cn2cc(CC3N(C(CC4CN(C)C4)=O)CCC3)nn2)ccc(F)cc1 23306,C1(CN(C(=O)CC2C=CCC2)C)COCCN1C(=O)Cn1cnnc1O 23307,N1(C(C2(C#C)CC2)=O)CCC(C(=O)Nc2cnccc2C)C(C)(C)C1 23308,C(=O)(C(O)CC(N)=O)N(CCCNC(=O)C=C1CCN(C)C1)CC 23309,C(=O)(CCC(C)N(CC(O)COCC1CC2(CC2)C1)C)OC 23310,Cc1cc(C(=O)NCC2CCC2NC(C2(CF)CCC2)=O)sc1Br 23311,c1(N2CC(O)(CNC(c3nn(C(CC)CC)c(C)c3)=O)C2)cc(O)nc(=O)n1C 23312,N1(C(C(c2ccc(C)o2)C)=O)CC(NC(c2onc(C)c2C)=O)CC(F)C1 23313,C1(CC)(CO)CCCN(C(=O)CC2COCCN2C(c2ccc(C(N)=O)o2)=O)C1 23314,CC(C)CCC(C(=O)NCCCc1ncn(C)n1)NC(C1CC1(F)Cl)=O 23315,N1(C(CC(C)C)=O)CCN(C(=O)C(C)NC(=O)OC(C)(C)C)CC2(C)CCCC12 23316,C1(NC(c2cccc(C(=O)NC)n2)=O)CN(Cc2noc(C)n2)CC1(C)C 23317,C1(NC(c2ccc(CCCCCC)s2)=O)CCN(C(=O)C(C)CCOC)CC1C 23318,N1(C(c2n(CC)nnc2)=O)CCC(CNC(=O)CCN(CC(C)(C)O)C)(OC)C1 23319,CC1CCN2N=C(C(=O)NC(C3CN(C(c4ccnn4C(F)F)=O)C3)C)NC2=N1 23320,N1(C(=O)OC(C)(C)C)CC(CNCC2CC(C)(C)CO2)C(F)C1 23321,c1(C(C(=O)NCC=C)N(c2cc(Br)ccc2OC)C)cn2c(Br)cnc2s1 23322,N1(C(C(CC)N(C)C)=O)CCCC(C)(CNC(=O)CCc2cnco2)C1 23323,N(C1CCCc2ccc(F)cc21)C(C(CC)C1COC1)=O 23324,c1(NCc2[nH]nc(CSC)n2)nccc(=NCc2ccnc(C#N)c2)[nH]1 23325,CC1OC2(C(=O)OCC3CC(C#N)(Oc4ccccc4)C3)CCC1CC2 23326,C(C1CN(C(=O)Cn2cc([N+](=O)[O-])cn2)Cc2ccccc21)NC(C(=O)NC)=O 23327,N#CC1CN(C(=O)C=Cc2ccc(O)cc2Cl)CCN1C(=O)C=Cc1ccoc1 23328,C1(CC)CN(C(C2CCCC2F)=O)CC1C(=O)NC1CCCC1CN(C)C 23329,C1(C(=O)NCCN(C(CC(CC=C)(C)C)=O)CCC)CC12CCC1(CC1)CC2 23330,N1(C(=O)Nc2ccc(CC)cc2)CC(CO)OCC12CC2 23331,C(=O)(C1=CS(=O)(=O)CCC1)NC1C2(CN(C(c3cn(CC=C)nn3)=O)C2)CCC1 23332,C1(CNC(C(=O)NC(c2ccccc2)C)=O)(COC2CCOCC2)C=CCCC1 23333,c1(C(N2C3CN(Cc4c(OC)cccn4)CC2C3)=O)ccc(C#N)cc1Cl 23334,CC1(C)NC(=O)CC1C(=O)NCC1(F)CC(CNC(c2scnc2C(F)F)=O)C1 23335,c1(OC)ccc(C(=O)OC(C(=O)NCc2sc(Br)nc2C)C)c(OC)c1 23336,C1(F)(C(N(CC(C)N(C(C(c2cc(F)cc(F)c2)C)=O)C)C)=O)CCN(C)CC1 23337,N1(C(CCOCC)=O)CC2CC1C2NC(c1nn(CC)cc1Br)=O 23338,N1(Cc2cn(C(C)CNC(c3conc3C(F)(F)F)=O)nn2)C(=O)CNC1=O 23339,Cc1nccc(C(=O)NCCC2(C(=O)N(C3CC3C)C)CC2)c1N 23340,C#CCCCCC(=O)NC1(CN(C(=O)C=Cc2cc(Br)cs2)C)CC1 23341,C(=O)(C(F)C(=O)N1CC(F)CC1CC(=O)NC(CO)C(F)(F)F)OCC 23342,CC1CN(C(=O)C=Cc2ccco2)CC2(CCN(C(C3CCC(C)(C)O3)=O)C2)O1 23343,O=C(C#CC1CCCCC1)NCC1CN(C(=O)COCC(F)(F)F)CC12CC2 23344,O=C(N=c1[nH]nc2n1CCCC2)N1CCC(Cc2cccnc2)C1 23345,CCCS(=O)(=O)CC(=O)N1CCN(C(=O)CCOc2ccccc2F)C2CC12 23346,Cc1cc(=NCc2cc(NC(=O)C(C)C)on2)[nH]c(N2CCc3ncncc3C2)n1 23347,c1(C(=O)NCCc2ccc(C(N(C)C)=O)cc2)c(F)ccc2n[nH]cc12 23348,N1(C(c2ccc(C#C)o2)=O)CCC(C2CCCN(C(=O)C(C)C(C)(C)C)C2)CC1 23349,N1(C(CC(CCC)C)=O)CC2CCC(N(C)C(c3ncc(F)cc3C)=O)C2C1 23350,N=C1NC(=O)C(CC(=O)NCCC2(O)CN(C(c3coc(C(F)(F)F)n3)=O)C2)S1 23351,C1(CNC(c2c(CC)ncs2)=O)C(O)C(O)CN1C(=O)CN1CCCC1=O 23352,CC12CC(C(=O)NC3CC(O)CN(C(c4cnco4)=O)C3)(C1)C(C)(C)O2 23353,C(=O)(C#CC1CCOCC1)NC(C1CCCN1C(c1cc(C(F)(F)F)n[nH]1)=O)C 23354,C1(C)(C(=O)NCCN(C(CC=CC=C)=O)Cc2ccccc2)CC(OC)CN1C 23355,c1(CC(N2CC(NC(C3CC(C)(C)OC3)=O)C3(C2)CC3)=O)ncn2c1COCC2 23356,C1(CNC(CCC=C(C)C)=O)CC2(CC2)CN1C(C1CC(C2CC2)=NO1)=O 23357,c1(C(N(CC(C)NC(C(CSC)C)=O)C)=O)cc2ccc(Cl)cc2c(O)n1 23358,N1(C(C(c2ccc(C)cn2)(F)F)=O)CCCC(NC(c2cccs2)=O)C1C 23359,C1(CNC(c2c(C)[nH]cc2)=O)CN2CCCCC2CN1C(c1ccn(C)n1)=O 23360,c1(C(N2CC3C(NC(=O)COCc4cccc(Cl)c4)C3C2)=O)cc(O)nc(O)n1 23361,c1(C(=O)NC2CCN(C(C(CC)NC(C)=O)=O)CC2F)cc2n(n1)CCNC2=O 23362,N1(C(C(=O)NCCCC)C2CCC2C(F)(F)F)CCCC(C2CCC2)C1 23363,c1(C(=O)NCC2(F)CC(NC(C3CCSC3)=O)C2)cccc(CC(F)(F)F)c1 23364,CC1=NNC(=O)C1CC(=O)NCC1(CN(C)C(c2ccn(CC(C)C)n2)=O)CC1 23365,CCCC(CNC(=O)CC1CCN(C(=O)CC2(COC)CC2)C1(C)C)CCO 23366,C(=O)(CS(=O)(=O)CC(C)C)NC1(CCNC(c2ccnc(C)n2)=O)CC1 23367,C(CCCCCCCO)=CC(N1CC(CCNC(=O)OC(C)(C)C)C1)=O 23368,C1(CNC(c2ncn(C)n2)=O)CN(C(=O)Cc2n[nH]c(=N)s2)C(C)(C)C1 23369,CC1CCCN1C(=O)CCn1cc(CCC2CCCCC2)nn1 23370,C=CC1(CC(=O)NC(CO)(CO)CO)CN(C(c2csc(CC)n2)=O)C1 23371,N(C(=NCCc1csc(C)n1)NC1CC(c2ccccc2Br)C1)C(C=C)C 23372,n1(CC)cc2ccc(C(=O)N(C)CCNC(=O)CNC(C3CC3C)=O)cc2n1 23373,c1(N2CC(C(C)NC(C3(C)CCC(=O)N3)=O)C2)nc(Cl)nc2[nH]c(O)nc12 23374,C1(NC(CCC=C=C)=O)CC2CC1CC2C(N1CC(N2CCC2)C1)=O 23375,c1(C(N2CC(Cn3ncc(C)c3)OCC2)=O)c(O)ncc2c1CCC2 23376,N1(C(c2cc(CC)ncc2)=O)CC2ON=C(CNC(=O)C=CBr)C2C1 23377,c1(N2CC(CC)C3(C2)CC3)ncc(C)cc1S(=O)(=O)NCc1cc(Cl)nc(Cl)c1 23378,Cc1nscc1CC(=O)N(C1CCC(NC(=O)COC(C)C)C1)C 23379,c1(N2C(C)C(NC(=O)CC3(C)CC3)CCC2)ncc2ccnc-2[nH]1 23380,N1(C(C(N2CCN(C)CC2)C)=O)CC2CN(C(C3(Br)CC3)=O)CC(C1)O2 23381,c1(SCCC)cccc(C(=O)NC2(C)CCN(C(c3nnc(S)n3C)=O)C2)c1 23382,CC(C(O)C(F)F)NC(=O)C(c1ccco1)NC(=O)CC1(C)CCOC1 23383,C(C)(CN=c1[nH]c(=NC(C)CCCO)[nH]c2c1COC2)(c1ccccc1)OC 23384,C1(OC)CCN(C(=O)C(CN)C2CCCCC2)CC1(C)C 23385,N1(C(COCCC(C)C)=O)CCC(C)(C)C1CNC(=O)CSc1cccnc1 23386,N1(C(COC)=O)CC2CCCC(NC(C3CCC=CCC3)=O)(C2)C1 23387,N1(C(C(CC=C)C(C)C)=O)CC2(CCN(C(c3cc(C)ns3)=O)CC2)CC1C 23388,N1(C(C=C(C)C(=O)O)=O)CC2CCN(C(=O)Nc3cc(C)ccc3F)CC2C1 23389,c1(NC(N(C)Cc2coc(Br)n2)=O)cccc2c1OCC2 23390,C(CC(C)(C)CC(=O)NC(CC(C)C)C(=O)Nc1ccc(O)c(Cl)c1)OC 23391,C1(NC(=O)CC(O)C2CC2)CCCOC12CCN(C(=O)CCC1(O)CCC1)CC2 23392,CC1(C)CC(C(=O)NCC(CNC(C2(C)CCCO2)=O)S(C)(=O)=O)CCO1 23393,c1(OCCOC)ccc(Cl)cc1C(=O)NCC1CN(C(=O)C(C)CF)CCO1 23394,CC(C)C(C)CC(=O)N1CC(C)CCC1C(=O)Nc1cc(Cl)cnc1O 23395,c1(OC)nccc(Br)c1C(=O)N(CCCNC(C1CCSC1)=O)C 23396,N1(C(c2nc(C)oc2)=O)Cc2[nH][nH]c(=NC(=O)c3cc(Br)ccc3Cl)c2C1 23397,c1(C(N2CCC(OCCNC(CCC#CC)=O)C2)=O)cc(C)c(O)c(C)c1 23398,c1(SCC(=O)Oc2c(C(CC)=O)cccc2)[nH]c(=N)c(C#N)cc1C#N 23399,CCCCC(CNC(=O)CCSc1ccccc1)NC(=O)CCC1CCCN1C 23400,C(=O)(C1=NNC(=O)CC1)NCC1N(C(c2cc(CN(C)C)on2)=O)CCN(C)C1 23401,C1(O)(CC(=O)N(C)CC)CCN(C(=O)C(O)Cn2cncn2)CC1 23402,C1(C(=O)NC(C)CCNC(=O)C(C(C)O)N(C)C)(COC)CCCCO1 23403,CC1=C(C(=O)N2CCCC(NC(c3cc(F)ccc3Cl)=O)C2C)CCC1 23404,c1(NC)cccc(C(=O)NC(C)C(c2ccccc2)NC(=O)C(C)SC)n1 23405,c1(OCC#C)ncccc1C(=O)NCC1CC(NC(c2cnn(CC=C)c2)=O)C1 23406,C(CO)(CCCNC(c1n[nH]cc1Cl)=O)NC(CN1CCC(OC)C1)=O 23407,C(C(CC1CCCC1)C(=O)NOCCN(C)C)NC(C1OCCC(C)C1)=O 23408,c1(C(=O)NC23C(CN(C(c4n[nH]c(CC)c4Cl)=O)C2)CC3)cc(F)cc(F)c1O 23409,CC1(NC(=O)C(C2CCOCC2)O)CCCN(C(=O)CSCc2ccccc2)C1 23410,c1(C(=O)NCC2(O)CN(C(C(C)NC(CC)(C)C)=O)C2)cc(Br)cn1C 23411,CC1(C)CC(NC(c2ccco2)=O)CN(C(C2CC2(F)F)=O)C1 23412,c1(CCC(=O)NCCN(C(C=CC(C)(C)C)=O)Cc2ccccc2)cnc(O)[nH]1 23413,c1(OC)cccc(NCC2(NC(=O)CCNC(=O)OC)CCOCC2)c1[N+](=O)[O-] 23414,C=C1CC2(C1)CC(C(=O)NCC(C)CNC(=O)C(O)C(F)(F)F)C2 23415,C(=O)(CC(C1CC(F)(F)C1)NC(c1ncoc1C(F)F)=O)OCC 23416,c1(C(=O)OCCC(=O)Nc2ccc(OCC)cc2C)cnc2ccccn12 23417,N1(C(C(C(C)C)CNC(C2(C)CCC3CC3C2)=O)=O)CCCOC(C)(C)C1 23418,C1(CC)CCC(C)CN1C(c1c[nH]nc1CNC(c1cnc(Cl)s1)=O)=O 23419,C1(N(C(=O)CCC2CCOC2)C)CCCN(C(=O)C(C)(C)c2ccccn2)CC1 23420,C1(O)(CNC(c2c(C)csc2)=O)CCCN(C(c2cc(Cl)nnc2O)=O)C1 23421,N1(C(C2CCCN(CCC)C2)=O)CCC(NC(=O)CN2C(C)CCC2C)C(F)C1 23422,CC1CCN(C(=O)CC=CC(C)(C)C)C1CNC(c1cncc(F)c1)=O 23423,c1(C(=O)OC)cc(CC(=O)NC(C)CNC(c2[nH]ccc2C2CC2)=O)cs1 23424,c1(C(C)=O)cncc(C(=O)NC2COCC2n2cc(-c3csc(C)n3)nn2)c1 23425,C1(C(=O)NC(C(C)NC(C2CC3(CC(=C)C3)C2)=O)CO)CCC2(CCCC2)CC1 23426,N1(C(C(C)NC(COC)=O)=O)CC2CC1C2CNC(C1(C)CC1(F)F)=O 23427,c1(C(C)NC(c2ccc(C)nc2)c2nnnn2C2COC2)ccc2nc[nH]c2c1 23428,c1(C(N2CCN(C(Cn3ccc(C)n3)=O)CC2CF)=O)ccc(O)c(C)c1C 23429,C1(NC(CC2CCCC(C)C2)=O)COc2ccccc2N(C)C1=O 23430,n1(CCCNC(COCCCOC)=O)cc(C(=O)NCC2CCOC2)nn1 23431,C(=O)(C1=NOC2COCC12)NCC1C(C)(C)C1C(N1CC2CCC=CC12)=O 23432,CC1(C)C(CC(=O)NCC2(N3CCNC3=O)CC2)CCN1C(=O)CCSC1CC1 23433,C1(CC2(O)CCN(C3CC(=O)N(CC)C3=O)CC2)COC2(CCCC2)O1 23434,C1(C(N(CCCC)CC)=O)CN(C(C2CCCOC2)=O)C(C)(C)C1 23435,C12(OC)CCC(C(N3CCC4C(NC(c5cc(C)cs5)=O)CC34)=O)(CC1)CC2 23436,c1(C(=O)NC2CC3CC(NC(C(C(C)(C)O)F)=O)C2C3)ccn2cccc2c1 23437,C(=O)(C(O)(C(C)C)C(F)(F)F)N1CCCCC(NC(C=CC=CC)=O)C1 23438,N1(C(=O)NC)CCN(C(=O)CC2CC2CNC(c2ncco2)=O)CC1 23439,c1(CNC(C(CC)OCC)=O)ccc(CNC(=O)C(N2CCCCC2)C)c(F)c1 23440,C(=O)(C(CC(F)F)NC(=O)Nc1cc(C)cnn1)OC 23441,N1(C(C(C)C)=O)CCN(C2CCC(NC(=O)C(N3CCC(C)(O)C3)=O)C2)CC1 23442,c1(C(C(=O)NC(CCOC)CNC(c2cc(C)sn2)=O)C)cccc([N+](=O)[O-])c1 23443,N1(C(c2ccc(C#N)cn2)=O)CCC(NC(=O)CCF)C12CCC2 23444,C1(NC(C2N(CCC(C)C)CCC2)=O)CN(C(=O)Cn2nccn2)CC1CO 23445,N1(C(C(C(C)O)C)=O)CCC(C2(NC(c3ccccc3)=O)CC2)C1 23446,C1(COC(CC(C)(CN)c2ccccc2)=O)CC2(C1)CC(C#N)C2 23447,C(=O)(CC(F)(F)C(F)F)N1CCC(NC(c2cc(COC)sc2)=O)C(F)C1 23448,C(=O)(C(O)(C(C)C)C(F)(F)F)NCC(C)NC(Cc1c(C)ccnc1)=O 23449,C1(C(C)NC(=O)C(O)C2CC2)CN(C(C2(C(N)=O)CC2)=O)C1 23450,CC1CC(NC(c2cccn2C)=O)CN1C(C1CC1C)=O 23451,C1(N(CC(=O)Oc2cccc(C)c2)C)CCC12CCN(C(=O)OC(C)(C)C)CC2 23452,c1(NC(C2CCCN2C(=O)CN2CCOC2=O)=O)cnc2ccccc2c1Cl 23453,Nc1cncc(C(=O)NCC2CCCCN2C(c2cc(C(F)(F)F)ccn2)=O)n1 23454,C1(C(=O)NCCN(C)C(c2ccc(-c3nccs3)cc2)=O)CS(=O)(=O)CC12CC2 23455,Cc1c[nH]cc1C(=O)NC1CCCC1CNC(=O)C(C)c1cccs1 23456,C1(NC(COCc2onc(C)n2)=O)CN(C(C2CCN2C2CCCC2)=O)CC1F 23457,Cc1cc(C(N2CCN(C(c3ccc(Br)c(O)n3)=O)C3CC23)=O)nc(C)c1 23458,Cc1cnc2n1CC(C(N1CCCOC(CNC(C3CCSCC3)=O)C1)=O)CC2 23459,N1(C(C(CCOC)C)=O)CCC(NC(C23CC2COC3(C)C)=O)C(C)(C)C1 23460,c1(C(=O)NC2CN(C(C(c3cccc(C)c3)(C)C)=O)C2)ccc(F)c2[nH]ccc12 23461,c1(C(=O)NC(C)CC(N)=O)cccnc1CNC(c1nn(C)cc1Cl)=O 23462,C=CCC(C(=O)NCC1(O)CCCC1)NC(c1sccc1Cl)=O 23463,C1(CCC(=O)NC(CNC(C2CC(OC)C2)=O)(C)C)CCCCO1 23464,c1(OC)cc(OC)nc(N2CC(C(=O)NCC(=O)N(C)C)CC(F)C2)n1 23465,c1(C(N2CCCC2(C)c2ccccc2)C(=O)NC)cccc(C(F)(F)F)n1 23466,N1(C(C2CC(OC)(OC)C2)=O)CCC(C)C(CC(=O)NC(C)(C)CN2CCC2)C1 23467,N1(Cc2cnn(C)c(=O)c2)CC(n2cc(-c3cccc(Cl)n3)nn2)CCC1(C)C 23468,CCCCC(C(=O)NC(C)CCCCNC(C)=O)N1CCCS1(=O)=O 23469,CC(F)(F)CCCC(=O)NC(CNC(C1OCC1(C)C)=O)CO 23470,C1(CN(C(=O)C(F)=C2CCC2)C)CCCN(C(=O)CCOCC2CC2)C1 23471,C(=O)(CCCCCc1ccc(O)cc1)NC1C(NC(C(C)CN(C)C)=O)COC1 23472,NC(=O)CCC(=O)NC(c1ccccc1)C1CC(NC(c2cn[nH]c2)=O)C1 23473,CC1(C)CCC(C(=O)NC2(CNC(=O)CSc3ccccc3Cl)CC2)CO1 23474,CC(C)CCCC(=O)N1CCCCC1CCN(C)C(c1cc(CC(C)C)c[nH]1)=O 23475,CC(C)(F)CCC(=O)NCC(F)CNC(c1cccc(Cl)c1O)=O 23476,N#Cc1ccccc1C=CC(=O)NCC1(NC(c2n[nH]cc2F)=O)CCOC1 23477,Cc1cc(C#N)nc(N2CCC(N(C)C(c3ccn4ccnc4n3)=O)C2)n1 23478,C1(N(C(=O)C(C)NC(C)=O)CCC)CCN(C(=O)CCC(=O)OC)CC1 23479,CCC(CC(F)F)C(=O)NC1CCC1NC(=O)C(C(C)C)NC(=O)CCCOC 23480,C1(NC(C(C)=C2CC2)=O)CN(C(c2ccc([N+](=O)[O-])c(C)c2)=O)C2CCCCC12 23481,c1(C(=O)NC2C(NC(CCCC(C)C)=O)CCCC2)cc(F)cc2c1CCC2 23482,Cc1ccc(Cl)c(C(N2CC3(CCC3NC(C3CC(F)C3)=O)C2)=O)c1N 23483,c1(OC)cnc(Cl)cc1C(=O)NC1(CO)CN(C(C2CCCC(=O)N2C)=O)C1 23484,C(=O)(C(C)(C)c1sccc1Cl)N(CC(C)NC(=O)CCNC(=O)C=CCl)CC 23485,N1(C(COCCSC)=O)CCOCC(NC(=O)C(n2cnc(C#N)n2)C)C1 23486,c1(C(=O)NCC(c2ccc(OC)cc2)NC(C2(C#C)CC2)=O)nc(O)sc1C 23487,C1(C(N(C2CCN(C(c3nccnc3Cl)=O)C2)CC)=O)CCC(C)(CC)O1 23488,c1(N2CC3N(C(C4(O)CC4)=O)C(CC3)CC2)nc2ccc(F)cc2s1 23489,C1(CNC(COC(CC)C)=O)CCCN(C(c2cn[nH]c2)=O)C1 23490,CC(CC#N)C(=O)N1CC(n2cc(C(C)N(C)C)nn2)C1 23491,C(=O)(CC1=CCN(C)CC1)NCC(N1C(C)CS(=O)(=O)CC1)=O 23492,N1(C2(c3cn(C(C)C)nn3)CCC2)CCCN(C(c2ccc[nH]2)=O)CC1 23493,C1(CCC(=O)OC)CN(C(C)=O)CCO1.c12ccc(cc1)-c1nsc(n1)S2 23494,c1(CN(C(C)C)C(=O)NCC2CC(O)C2)ccccc1.C1(C)CCCO1 23495,C#CC1CN(C(C2CCCCCCN2C(C2CS(=O)(=O)C2)=O)=O)CCN1C 23496,Cc1nc2cncc(C(=O)NC3CCN(C(=O)C(C)(F)C(C)(C)F)CC3)c2[nH]1 23497,C=CC(C)(C)C(=O)Nc1cccc(CNC(=O)C(c2ccnn2C)C)c1 23498,c1(OC)c(C)cc(C(=O)NC2CCCC(N(C(=O)CSC3CC3)C)C2)cc1Cl 23499,N1(C(C(C(=O)OC)C)=O)C2CCCC1CC(NC(C1CCC(O)CC1)=O)C2 23500,c1(CNC(C(C2CC(NC(C(C)SC)=O)C2)F)=O)cc(C)ccc1C 23501,N1(C(Cc2cn(CC)nc2)=O)C2CC1CN(C(C1CCCN1C(C)C)=O)C2 23502,c1(C(N(CCNC(C2C(COC)C2)=O)C)=O)cccc(Cl)c1O 23503,c1(C(=O)NCC2CCCN(C(c3ccon3)=O)CC2)c[nH]c2ccc(Br)cc12 23504,c1(COC)ccccc1CC(=O)NC(C)CNC(=O)Cc1cc(C)nn1C 23505,c1(C(=O)O)cccn(O)c1=O.CC(C)COC(C)(C)C1(CO)CC1 23506,c1(C(N2CC(SC)C(NC(=O)C(O)C(C)C)C2)=O)cc(S(N)(=O)=O)cnc1C 23507,N1(C(C(C(CC)C)OC)=O)C2CCC1CN(c1ncnc(Cl)c1OC)CC2 23508,C(=O)(C(C)(C)C(C)NC(N(C)C(=O)CSC(C)(C)C)=O)NC1(C(C)C)COC1 23509,C(=O)(CC1OCCc2ccsc21)N(CCCNC(C1CC2C(C1)C2(C)C)=O)C 23510,Cc1csc(C(C)CNC(=O)C=Cc2ncc[nH]2)n1 23511,c1(NC(c2nc(C)[nH]c2Br)c2nnnn2CC(F)F)cccc(CO)c1C 23512,N1(C(COCCNC(Cc2n(C)nnc2)=O)=O)CC2CC2C2CC12 23513,n1(CC(=O)NC(=O)NCC2CCN(CCCC(=O)OCC)C2)ncn(C)c1=O 23514,C(=O)(CCC(CF)CF)NCCn1ccc(C(N2CCC(N(C)CC)C2)=O)c1 23515,N1(C(COC)=O)CC2C3CCC(C2C1)N(C(c1occc1-c1ccccc1)=O)C3 23516,N1(C(C2C(OC)CCC2)=O)CCC2(CCN(C(=O)CN3CCCCC3)CC2)C1 23517,c1(C(N2CCC(C3N(C(C(C)C4CCCO4)=O)CCC3)C2)=O)ccc(F)cc1Cl 23518,Cc1cc(Cl)cc(C(N2CCCOC(CNC(C3CC4(CCC4)C3)=O)C2)=O)c1C 23519,c1(C(=O)NCCN(C(=O)CC23COC(C2)C3)CC)ccc(C(C)C)s1 23520,C1(CNC(CCCc2c(C)ccc(C)c2)=O)(NC(=O)COC)CCC(F)(F)CC1 23521,N1(C(C(C)(C)SC)=O)CC2CS(=O)(=O)CC2(NC(c2ccc3cccnn23)=O)C1 23522,N1(C(C(COC)O)=O)CCOCC(F)(CNC(=O)CCc2ccccn2)C1 23523,CCS(=O)(=O)CC(=O)N1CCN(C(=O)CC2C=CS(=O)(=O)C2)C(CO)C1 23524,c1(CC)ccc(C(=O)NCC2COCC2NC(c2c(C)cncc2C)=O)cc1Cl 23525,C(=O)(CC(F)(F)CC)N1CC(C(=O)NCC2N(CC)CCC2)C(F)C1 23526,C1(CC)CN(C(=O)CCC(F)F)CCC1NC(c1nc(-c2cncn2C)no1)=O 23527,C1(NC(c2c(C)nn(C(C)(C)C)c2)=O)CC2CCC1N(c1ncncc1C#N)C2 23528,C1(O)(C(=O)NCC(C)CNC(=O)C(n2ccc(C(F)(F)F)n2)C)CCCCCC1 23529,C1(CNC(C(C2(O)CCOCC2)C)=O)CN(C(c2cc(Br)c[nH]2)=O)C(C)(C)C1 23530,c1(CNC(=O)NC2C(C(=O)OC)CNC2)ccc(O)cc1Cl 23531,CCCC(C(C)(C)C)NC(=O)CC(C)(C)NC(C1CCCN1C(C)=O)=O 23532,c1(C(=O)NCC2(O)CN(C(C3(CSC)CC3)=O)C2)cccc(C(C)C)c1 23533,CCCC(C(F)(F)F)NC(C1CCCC(NC(=O)C(C)=C2CC2)CC1)=O 23534,C1(OCCCNC(CC2CC(CC)C2)=O)CCN(C(=O)CC2CCOC2C)CC1 23535,c1(C(=O)NC(CNC(c2ccc(CCC)[nH]2)=O)CC)ccc(NC)cc1Cl 23536,N1(C(C(C(C)C)O)=O)CC2=C(C1)CN(C(c1cccnc1-n1cncn1)=O)C2 23537,C1(CNC(CC)=O)CC(NC(c2ccc(=NC)[nH]c2)=O)C12CCC2 23538,c1(C(N2CC(C=C)C(NC(=O)CSC)C2)=O)n[nH]c2cccc(OC)c12 23539,Cc1cc(C(=O)N(CCC(C(C)C)NC(=O)CC2CCCO2)C)c(C)nc1C 23540,O=C(CC1CCc2ccccc21)NC1CC2CN(C(=O)CC3(CO)CCC3)CC12 23541,CC1CCN(C(=O)C(F)CC2CC2)CCN1C(=O)CC1NC(=O)NC1=O 23542,c1(C(=O)NCC2CC(NC(C3CC(C(C)C)OCC3)=O)C2)cc(F)cc(F)c1N 23543,c1(NC(c2ccc(CC)s2)=O)cccc(NC(=O)CCc2cncn2C)c1 23544,Cc1cccc(C(N2CC(C)(CNC(=O)Nc3ccccn3)C2)=O)c1O 23545,c1(C(c2n(CC=C)nnn2)NC2CCCC=C2Br)cn2cc(C)ccc2n1 23546,CC1CN(C(c2cccc(=O)n2C)=O)CC(C)C1NC(=O)Cc1cccs1 23547,C=CCC(F)(F)C(=O)N(CC(CC)NC(c1ccc(Cl)cc1Cl)=O)C 23548,C(=O)(C#CC1CCOC1)N1C(CC)CN(C(c2cc(N)cnc2C)=O)CC1 23549,CCCC(C(=O)NC(CC)C(c1ccc(OCC)cc1)=O)N(C)C 23550,N1(C(C2(N(C)C)CCC2)=O)CCCC(CNC(=O)CCc2cnco2)C1 23551,c1(NC(C2CCCCO2)C)ncc(Cl)cn1.c12ncoc1CNC2=O 23552,C1(N(C(CCN(C(=O)C(C)NC=O)CC)=O)C)CCCC(C)(C)C1 23553,c1(N(CCCCN(C(Cc2cnc(C)s2)=O)C)C)snc(Cl)c1C#N 23554,O=S(=O)(c1ccc(NCC2=CCCC2)cc1Br)NCc1cscc1Br 23555,N1(C(CN(C(=O)OC)C)=O)CCC2(COC(CNC(c3ccccc3)=O)C2)C1 23556,c1(CNC(C2(N(C(C3CC(C)OCC3)=O)C3CC3)CCC2)=O)cc(F)ccc1O 23557,c1(C(=O)NCC2(NC(C(C(CC)C)C)=O)CC(OC)C2)cc2cccnc2[nH]1 23558,CCCC(C)(C)C(=O)NCCC1(C)CCN(C(c2cn(C(C)C)nn2)=O)C1 23559,CN1CCCN(C(c2cscc2Br)C(=O)NC2CC2)CCC1 23560,C12CCCC(C1)NC(=O)CN2C(C1(N(C)C)CC1)=O.c1(CSC)ccccc1 23561,Cc1oc(Br)cc1C(N1CCC(O)C1c1cccc(F)c1)=O 23562,C(C)(C(C(C)C)NC(c1cc(C)sn1)=O)NC(c1ccn(CC)n1)=O 23563,c1(N(C)Cc2cc(C)on2)nc(N2CC3CCC(CC3)C2)nc2ncn(C)c12 23564,S(=O)(=O)(c1cnc(N(C)Cc2conc2C2CC2)cc1C)N(CCF)CC 23565,c1(CC(C(=O)CC2(C(F)(F)F)CC2)=O)cn[nH]c1.C(C(C)N)NCC 23566,O=C(NNC(=O)C1CCOC1)c1nn(-c2cccc(Cl)c2)cc1Br 23567,N1(C(C2N(CC)CC2)=O)CC(C2(NC(c3cccc(CO)c3)=O)CC2)C1 23568,c1(C(=O)Nc2ccc(C3(NC(COC)=O)CCC3)cn2)ccc2occc2c1 23569,c1(N(C(C(=O)OCC)C)C(=O)Cn2cnnn2)cc(CC2CCCO2)cnc1O 23570,N1(C(=O)NC(C)CN2CCCCC2)CCC(c2nc(-c3ccccc3)no2)CC1 23571,N1(C(CC2CCCC(C)C2)=O)CC2CC(NC(=O)Cc3ccc(F)cc3F)C2C1 23572,C1(NC(c2cnc(-n3cccn3)cn2)=O)CCN(C(C2CC3CC3C2)=O)CC1O 23573,CC(N=c1[nH]c(=NCC(F)(F)Br)[nH]c2c1CSC2)c1cc(F)ccc1F 23574,CC(C)(O)C(F)C(=O)N1CCOC(CNC(c2ccc(-c3ccco3)[nH]2)=O)C1 23575,c1(OC)nc(=NCC(C2CCCCC2)NC(=O)C=C(C)C(C)C)[nH]c2[nH]cnc12 23576,N1(C(c2cnc(C)o2)=O)CC2CCCC2C1C(=O)NCC(O)CF 23577,C(CCSC)(C(=O)N(C)CC1(NC(=O)CC2CSCCS2)CC1)OC 23578,c1(C(=O)NCC2C(NC(C(OC)OC)=O)CCCC2)ccc2c(n1)CCC2 23579,c1(C(N2CCN(C(=O)CCN3CCCC3)C(C3CC3)C2)=O)ccn2nccc2n1 23580,CC1(C)C(NC(c2cnn(CCN)n2)=O)CC1CCC1CCC1 23581,C1(C(=O)NCC#CCOC)(CNC(C2CCC(C)(C)C2)=O)CC12CCC2 23582,C(=O)(C1=NOC(CNC(c2cccc(CO)c2)=O)C1)NC(C(=O)N(C)CC)C 23583,N1(C(CC2(COC)CC2)=O)CCCC(C)(C)C1CNC(c1ccc(C)c(F)c1)=O 23584,N1(C(C(CC#C)O)=O)CC2CCC(C1)N2C(=O)CC(C)(C)COC 23585,c1(C(N2C(C)CC(CNC(c3occc3F)=O)C2)=O)cc2n(n1)CCC2 23586,C(=O)(C1=CCC(F)(F)CC1)N(CCCNC(C1(COC)CCCOC1)=O)C(C)C 23587,c1(C(=O)NC2CC(C)N(C(=O)C(C)(C)CCC#N)C2)ccc2nc(CO)[nH]c2c1 23588,C1(C(N2CCC(F)(CNC(c3ncn(C)n3)=O)CC2)=O)CC2CCCCN2C1 23589,C(=O)(C(CCC(N)=O)n1cc(CCC(C)O)nn1)NC(C12CC(CO1)C2)C 23590,Cc1ccc(CCC(=O)NC2CCCC2NC(C2(O)CCOC2)=O)c(Br)c1 23591,c1(C(=O)NC(C2CCOC2)C)ccc(-n2cccn2)cc1 23592,C1(OC(C)C(=O)NC(C2CCCN2C(C2CC(C(F)F)C2)=O)C)CCCCCC1 23593,C(=O)(C(C(=O)N1CCC(C(C)(C)NC(C2CCCC2C(C)C)=O)CC1)OC)OC 23594,N1(C(CCCOCCOCC)=O)CC2ON=C(CNC(c3cnn(C)c3)=O)C2C1 23595,C1(NC(C(n2cc(C)nc2)(C)C)=O)CN(C(c2ccncc2)=O)CCC1CO 23596,Cc1nn(C)c(C)c1C(N1C(C(=O)N(C2CCC(=O)N(C)C2)C)CC2CC12)=O 23597,C(=O)(C(CC(C)C)N(C(=O)CN1CC(=O)NC1=O)C)NCc1c(C)non1 23598,CCC(C)C(C)C(=O)NCCCN(C(=O)CCc1csc(C)n1)C 23599,N(C1CC(C)(C)Oc2ccc(F)cc21)C1CC(S(=O)(=O)N)C1.CCC 23600,n1(CC)cnc(C(=O)NCc2occc2C(=O)NC2CC2(C)C)n1 23601,CCC(C)(C)C(=O)C(=O)N1CCCC1CC(=O)NCc1noc(C(C)C)n1 23602,N1(C(CC(OCC)OCC)=O)CC(NC(c2ccc(Br)nc2Br)=O)C(C#N)C1 23603,S(=O)(=O)(c1c[nH]c(=NCCN2CCS(=O)(=O)CC2)cc1C)N1CC(C)=C(C)CC1 23604,CC(C)S(=O)(=O)CC(=O)N1CCCC(N(C(=O)CSCCC(F)(F)F)C)C1 23605,C1(C(N2CCC(NC(CC=CC)=O)C23CC3)=O)CC(c2ccccc2F)=NO1 23606,N1(C(c2n[nH]cc2-c2ccccc2)=O)CCN2C(=O)OCC2C1 23607,Cc1cnccc1CN(C(=O)C(C)CNC(=O)Cn1nnnc1C)C 23608,C1(C(N2CCC(C(C)(C)NC(c3[nH]c(=N)sc3)=O)CC2)=O)CCC(=C(F)F)CC1 23609,c1(CC)ccc(N)c(C(N2CC3C(CNC(=O)CC4C(C)C4(F)F)C3C2)=O)c1 23610,N1(C(CC=CC=C)=O)CCC(F)CC1C(=O)NCC(C)C(F)F 23611,C1(C)(C(N(C(c2ccccc2)CNC(=O)C(O)CC2CCCC2)C)=O)CCCN1C 23612,N1(C(CNS(CC)(=O)=O)=O)CCC(NC(C2CCC(=O)N2C2CC2)=O)C1(C)C 23613,C(=O)(CC(C)(C)CC(=O)NC1CCN(C2CCN(C)CC2)C1=O)OCC.C1C(=O)O1 23614,c1(C(=O)NCC(CNC(C2CCC(CC)O2)=O)(C)O)c(CC)ncnc1CC 23615,C1(NC(=O)CCn2ccnn2)CCC(NC(=O)C(C2CC(F)(F)C2)O)C1 23616,C1(NC(C2CCS(=O)(=O)N2)=O)C2CC3CN(C(c4cnsn4)=O)C1C3C2 23617,c1(C(C(=O)NC2CCN(C(=O)CSC(F)(F)F)C2)=O)cnn(C(F)F)c1 23618,c1(NC(C2CC23CN(C(c2ccc(O)nc2)=O)C3)=O)cc2ccccn2n1 23619,Cc1ccc(C(c2nnnn2-c2ccccc2C)NC(C)(C)C)c(Br)c1 23620,N1(C(C2CCN(C(=O)OC)CC2)=O)CCC(C)(C)C1CNC(=O)C(C)N1CCC1 23621,CCCC(CC)CC(=O)NCC(O)CN(C)C(c1ccoc1CC)=O 23622,CC(c1ccccc1)=CC(N1CCC(C)(NC(C2(C3CCCCO3)CC2)=O)C1)=O 23623,N1(C(C(C)NC(N)=O)=O)CCC(N(C(=O)CN(C2CCCC2)C)C)C1 23624,N1(Cc2cnc(C)[nH]2)CCCC2(CCN(C(c3ncc(OCF)cn3)=O)C2)C1 23625,N1(S(CC=C)(=O)=O)CCc2[nH]nc(C(=O)Nc3c(F)ccc(F)c3Cl)c2C1 23626,C#CCCC(C(=O)NCC1CCSCC1)NC(c1cc(C(N)=O)[nH]n1)=O 23627,CCC(C)(COC)C(=O)NCc1ncoc1C1CN(C(C2CCN(C)C2=O)=O)C1 23628,N1(C(c2c(C(C3ON=C(C(C)C)C3)=O)cccc2)=O)CC(C)(C)OCC1CN 23629,Cc1cccc(CCC(=O)NCC(CNC(=O)CCc2cnoc2)CO)c1Br 23630,N1(C(CN(C(C=Cc2n(C)cnc2)=O)C2CC2)=O)CCC(N=[N+]=[N-])C(O)C1 23631,N1(C(C=CCC)=O)CCN(C(C2CCCCN2N=O)=O)C(CCC)C1 23632,c1(C(=O)NC(C2CCN(C(c3cnco3)=O)C2)C)ccn2nccc2n1 23633,S(=O)(=O)(c1cc(C(N)=O)ccc1F)N(C)Cc1c[nH]nc1C(F)F 23634,C12(NC(=O)Cc3coc4ccccc34)CCCCC1CN(C(C1(O)CC1)=O)C2 23635,CCCC(C)(C)CN=c1[nH]c2c(c(=NC3CCC(C(C)C)(OC)CC3)[nH]1)SCC2 23636,N1(C(C2CC(CCC)C2)=O)CCN(C(=O)C(N)=O)C(C2CCC2)C1 23637,C1(C#CC(=O)NC2CCC(C)N(C(=O)CCc3cc(C)cs3)C2)(CC)COC1 23638,c1(C(C)C)cccc(C(N2CCC(F)(C(=O)NC(c3ccccc3)C#N)C2)=O)c1 23639,O(C1CCOc2cc(Cl)cc(Cl)c21)C(=O)CCCCc1cnn[nH]1 23640,Cc1cc(C(=O)N(CCNC(c2cnc[nH]2)=O)CCN2CCCC2)c(O)nn1 23641,c1(CC)ncccc1C(=O)N(C)Cc1cncc(Br)c1 23642,N1(C(c2c(Cl)cn(CCC)n2)=O)CC(NC(=O)COCC(C)C)CC1(C)CC 23643,C=CCC(CC(F)F)NC(=O)CC1CCCCC1NC(C1CCC(C)(C)C1)=O 23644,c1(C(=O)N(C2CCCCC2)CCNC(C2(F)CCCC2)=O)cc(F)cc(F)c1 23645,C#Cc1cccc(C(N2CCN(CCNC(=O)CC3CCC(O)C3)CC2)=O)c1C 23646,C1(c2ccccc2)(C(N(CCCCNC(C2C(C(C)C)C2)=O)C)=O)CC(O)C1 23647,C(=O)(CCCCCC(C)(C)C)NC1CC2(C(NC(c3c(C)cc(N)cc3)=O)C2)C1 23648,C12(CNC(C(CC)F)=O)CCCC1N(C(c1cc(C)c(C)o1)=O)CCC2 23649,CC(C)C(C)CCNC(=O)C(C(C)O)NC(=O)CN1CCC(F)CC1 23650,Cc1ccc(Cl)c(O)c1C(N1CC(NC(c2ccc(F)cn2)=O)CC(C)C1)=O 23651,N1(C(C(CC(=C)C)C)=O)CCC2(CC1)CN(C(c1ccc3scnc3c1)=O)C2 23652,C1(C(=O)N(C)CCNC(=O)C(C)Cc2ccco2)(OC)CCC(F)(F)CC1 23653,c1(C(N2C(C(C)(C)NC(C(F)=C(C)C)=O)CCC2)=O)cc2cc(Br)cn2cn1 23654,C(=O)(C(C)C(CC)CC)NC1(CC=C)CCN(c2nc(CC)nc(C)c2F)CC1 23655,Cc1cc(C(=O)N(C(C)CNC(=O)CC2CCCOCC2)C)cnc1O 23656,C1(NC(C(N2CCOCC2)C)=O)CC2(CCCN(C(C3C(C)C3C)=O)C2)C1 23657,C12(CNC(COCCCC)=O)CCC(CC1NC(c1ncccc1CSC)=O)C2 23658,N1(C(CC2CC(C)(C)OC2=O)=O)CC2CC(C1)CN(C(=O)C=Cc1cnc[nH]1)C2 23659,C1(NC(c2c(C(C)=O)cccc2)=O)COC2CNCC12 23660,C12(C(=O)NC(c3ccc(C#N)cc3)C)CC(C)(C1)OC21CCC1 23661,Cc1cccc(Cl)c1CN1CC(O)(CNC(=O)CC2CCOC(C(C)C)C2)C1 23662,N1(C(C)=O)CCC(C)(C(=O)NCC2(CNC(=O)C#CC3CC3)CC2)CC1 23663,CCCCC(C)C(=O)N(CC(CC)NC(=O)C(C)(C)CO)C 23664,N1(C(C2C(C)CC2C)=O)CCCCC(NC(=O)CC2CC3CCC2CC3)C1 23665,C#Cc1ccc(CC(=O)NC(C2CN(c3cc(C(F)F)ncn3)C2)C)cc1 23666,C1(NC(CNC(CC)=O)=O)CC2CN(C(c3cc(C)ccc3C)=O)CC12 23667,c1(OC)cccc(C(N2CCC(C(C)(C)NC(=O)CSC(F)(F)F)C2)=O)c1 23668,Cc1cc(NC(C2(CNC(=O)Cn3c(O)nnc3O)CC23CCC3)=O)c(C)cc1O 23669,CN(C)NC(=O)CCC(=O)N1CCC(NC(C2CCS2(=O)=O)=O)C1C1CC1 23670,c1(C(N2CCC(O)(CNC(c3n(C)ccn3)=O)C2)=O)c(O)ccc2ccccc12 23671,C(=O)(C1CCCc2sc(=N)[nH]c21)N1CC(NC(C2OCC(C)C2)=O)CC2(C1)CC2 23672,c1(NC(CCC2N(C(C(CC(C)C)O)=O)CCC2)=O)c(O)ccc(Br)c1O 23673,CC(C(=O)N1CC(N(C)C(c2nc3cccnc3s2)=O)C1)C(C)S(C)(=O)=O 23674,c12cccc(c1)N2.c1(CC(COC)(C)C)nc(-c2nccs2)nn1C(C)COC 23675,c1(C(=O)NC2(C)CN(C(C34CCC(F)(CC3)C4)=O)C2)noc2ncccc12 23676,Cc1cc(CNC(c2coc(CNC(=O)CC3CCN(C)C3)n2)=O)sn1 23677,Cc1c(C(N2CCOCC(NC(=O)C(=O)NC(C)C)C2)=O)oc2ccccc12 23678,CC1CN(C(=O)CC2(O)CCOCC2)CC1CNC(c1ccn(C)n1)=O 23679,CC(C(F)(F)C(F)(F)F)=CC(=O)N(CCCN(C)C(c1cc(C)ccc1Cl)=O)C 23680,N1(C(C2C(C)C2)=O)CCCC(O)(CNC(=O)C=Cc2ccsc2C(F)(F)F)CC1 23681,c1(C(N(C2CN(C(c3cc(Br)no3)=O)C2)C)=O)cc(Cl)no1 23682,Cc1oc(CO)cc1C(N1CCN(C(C2CNC(=O)C2)=O)CC1)=O 23683,N1(C(Cc2cnc(C)[nH]2)=O)CC2CCC1C1CN(C(=O)C=CC3CC3)CC21 23684,C1(CCNC(CN(C)C2CC2)=O)CCN(C(C2CC3C(C2)C3(F)F)=O)CC1(F)F 23685,C(CS(=O)(=O)CC(=O)N1CCCCCC1CNC(c1ccc(=O)oc1)=O)OC 23686,C1(C(N2CCC(n3cc(C(C)N(C)C)nn3)CC2)=O)CCC2(CCC2)C1 23687,C12(CNC(CCOCCCOC)=O)CCN(C(=O)CC(C)(C)C)CC1C2 23688,c1(OC)ncnc(C)c1C(=O)NCC1CCCCN1C(C1CC(F)(F)C1(F)F)=O 23689,c1(C(N(C)CC2(O)CN(C(c3noc(CC)c3C)=O)C2)=O)ccc(C)c(C)c1O 23690,c1(C(=O)NCC=CCC(=O)Nc2cnn(CC3CC3)c2)cc(C(F)F)no1.C 23691,C1(C(N2CC(C(C)NC(c3cc(C(C)(C)C)n[nH]3)=O)C2)=O)CCC2(CCOC2)O1 23692,c1(OC)cc(C(=O)NCC2CN(C(=O)C(O)c3ccsc3)CC2(C)C)cc(Cl)n1 23693,C1(O)(C(CNC(CCN(C)CC)=O)C)CCN(C(c2cc(CO)n(C)n2)=O)C1 23694,Cc1oc(S(C)(=O)=O)cc1C(N1CCC1CNC(c1cc2c(s1)CCC2)=O)=O 23695,c1(CNC(C2CCN2C(c2ccsn2)=O)=O)nnc(O)o1 23696,N1(C(c2ccc(OC)nc2F)=O)CCCC2(CCCN2C(C2C=CCC2)=O)C1 23697,N1(C(c2cc(C)nc(C)c2)=O)CC(C)CN(C(c2nc(Cl)sc2Cl)=O)C(C)C1 23698,N1(C(c2cnc(OC)s2)=O)CC2CCC1C(CNC(=O)CCCC(N)=O)C2 23699,Cc1cc(Br)ccc1C(=O)NC1CCC(NC(=O)C(C)Cn2cccn2)C1 23700,c1(C(=O)NCCN(C(=O)CC(O)c2ccccc2)CCOC)nocc1C 23701,C1(CC(N2CCC(CCNC(C3(C)CC=CC3)=O)C2)=O)CCCC1(F)F 23702,C1(NC(C#CCNC(c2c(C)occ2)=O)=O)CCC12CCCC2 23703,N1(C(C2(C3N(C(C4CCCCCC4)=O)CCC3)CC2)=O)CCN2CCCCC1C2 23704,c1(C(N(c2cc(C)c(Cl)cc2)C)=O)ccc2c(c1)COC2 23705,N1(C(c2ccc(C)o2)=O)CCCC(C)(C(N2CCCC2c2ccc(Br)cc2)=O)C1 23706,c1(N2CC3CC(NC(c4cccc(C(C)C)n4)=O)C3C2)ncnc2c1CCO2 23707,N1(C(C(C)(C)c2cc[nH]n2)=O)CCC(NC(c2cscc2Br)=O)C(O)C1 23708,N1(C(C(CC)n2cccn2)=O)CCC(O)(Cn2cc(CO)nn2)C1.C12(CC1)C(=O)N2 23709,N1(C(=O)Nc2n(C)nc(C)c2Br)CCCc2ncccc2C1 23710,C(C(=O)NOCCN(C)C)N(C(=O)CC1(C)OCCO1)C(C)C 23711,c1(OC)cc(F)c(S(=O)(=O)NC2CCCC2P(C)(C)=O)cc1OC 23712,c1(CC(=O)NC2CC(NC(C(n3cc(C)nc3)(C)C)=O)C2)cccc2nonc12 23713,S(=O)(=O)(c1c[nH]c(C(=O)NC2CCN(C(=O)C(C)(C)C#N)C2)c1)NCC 23714,N1(C(C(C)c2ccsc2)=O)CCCC(O)(CCNC(=O)C(C)(Cl)Cl)C1 23715,C(=O)(C(O)CC(F)F)NC(C1CCN(C(Cn2nc(C)c(Cl)c2)=O)CC1)(C)C 23716,C(=O)(C1=CCC(NC(c2cnn(C)c2Cl)=O)C1)NC(C1CC(F)(F)C1)C 23717,CC(C)(C)C(CN=c1ccn2c(Br)cnc2[nH]1)NC(C1CC2CCCC12)=O 23718,N1(C(Cc2scc(C)c2)=O)CC2(CNC(=O)C(F)=CC3CC3)CC1CO2 23719,C12(CNC(C(C)C3CCC3)=O)CC1CN(C(c1nccn1C)=O)C2 23720,C1(NC2CCC(CN(C)C)C2)CCNC(C2CC2)C1 23721,N1(C(Cc2ccc(C)nc2)=O)CC(C)(C)C(NC(c2cnc(Cl)s2)=O)C(C)(C)C1 23722,C(CSC)(C(=O)NCCCOCCCNC(=O)C=CCc1ccccc1)OC 23723,N1(C(=O)OC(C)(C)C)CC2COCC2(C(=O)NC(C)(C)CN2CCOCC2)C1 23724,c1(C(=O)NC2C(CNC(C34CCC(OC)C3C4)=O)C2)[nH]c2ccccc2c1C 23725,c1(C(N2CC(NC(C3(CN(C)C)CC3)=O)C2)=O)ccc(C2CC2(F)F)cc1 23726,c1(CC(N2CCC3C(NC(C4CC(CCO)C4)=O)C32)=O)ccc(F)cc1[N+](=O)[O-] 23727,C1(OCC)CCCN(C(c2nc(CNC(C3CC(C)=NO3)=O)cs2)=O)C1 23728,C(=O)(C(C)(C)CC(C)=O)NCC(=O)NCC(=O)NCC(C(CC)C)(C)O 23729,C1(CC(=O)NCC2(F)CN(C(CC3(C)CCCO3)=O)C2)CN2CCN1CC2 23730,CC1(C)CN(C(=O)CCc2nccs2)CC1CNC(c1cc(CO)[nH]n1)=O 23731,N1(C(C(C)OCCCC)=O)CC(C(N2CC(C(C)(C)O)C2)=O)CC(C)C1 23732,C(=O)(C#CC1CCCCO1)NCCN(C(C)C)C(c1ccc(OCCF)cc1)=O 23733,c1(C(N2C(C(C)NC(C3CC(C#N)C3)=O)CCCC2)=O)cc2cc(F)ccc2o1 23734,CCCCC(F)C(=O)N1CCCCC1C1CCN(C(c2ccc(F)cn2)=O)C1 23735,NS(=O)(=O)c1ccnc(C(=O)NCC2C(CNC(=O)CC3CC=CC3)C2(F)F)c1 23736,Cc1ccc(C(=O)NC(CNC(=O)C2=CCC2)CC(C)C)cc1OC(F)(F)F 23737,C1(C(N2CCC(CC=C)(NC(c3cnc(Cl)[nH]3)=O)C2)=O)CCC(N=[N+]=[N-])CC1 23738,N1(C(COCCCC(C)C)=O)CCC2(C1)CN(C(C1CC1C(F)F)=O)C2 23739,CCC(O)CCN=c1[nH]c(N2CCN(C)C(C)(C)C2)nc2cccnc12 23740,c1(CCC)nc(C(N2CCC(C(C)NC(c3cncs3)=O)C2)=O)co1 23741,c1(C(=O)NC(CC(C)NC(=O)Cn2ccnn2)C)ccc(-c2csnn2)cc1 23742,N1(C(c2ccc(C)nc2)=O)CCC2C(C1)CN2C(=O)CCn1ccc(O)nc1=O 23743,C(CC(C)C(=O)NCC(CO)NC(c1c(C)ncn1O)=O)OC 23744,C12(NC(C=CC(=O)OCC)=O)CC1CN(Cc1cccc(CO)n1)C2 23745,C1(CC(=O)NCc2cccc(O)c2)CCCCN1C(=O)CN1C(=O)CNC1=O 23746,C1(NC(CC2C(=O)NCC2)=O)CC2CC(C1)N(C(=O)Cc1cnsc1)C2 23747,C12(C(N(C3C4CN(C(c5cc(O)ccc5Cl)=O)CC34)C)=O)CC3CC1C2C3O 23748,N1(C(C2(OC)CCSC2)=O)CCOC(Cc2cn(CCC=C(C)C)nn2)C1 23749,c1(C(N(CC(C)N(C(=O)CC2CC3C=CC2C3)C)C)=O)c(Cl)csc1Cl 23750,CC1CN(C(C2CC3CC3C2)=O)CC1NC(=O)Cc1ccccc1C(F)(F)F 23751,C(=O)(C(CCC)N(C)C)NCC(C)(C)NC(COCCOCC#C)=O 23752,N1(C(C(C(CC)C)O)=O)CC2(CC(NC(C3CCCCN3N=O)=O)CO2)C1 23753,N1(C(=O)NCc2c(CC)noc2)CCC(CNc2nccnc2CC2CC2)CC1 23754,c1(CC(=O)N(C(C)C(C)(C)O)C)ccc(NC(=O)OC(C)(C)C)nc1 23755,C1(NC(CN(C)CC)=O)CN(C(c2nscc2Br)=O)CC1C 23756,c1(C(=O)NC(C(C)NC(C2C=C(C)CS2)=O)C)cn2cccnc2n1 23757,c1(C(N2C(CNC(C3N(CC)C(=O)CC3)=O)C=CC2)=O)noc2ccccc12 23758,c1(CC(N2CC3(CCN(C(CC(CC)C)=O)C3)C2)=O)ccc(Cl)c2cccnc12 23759,c1(OC)ccccc1OCC(=O)NC(C)CN(C(=O)Cc1cn(C)nc1C)C 23760,CC(CC(=O)N1CCC(CNC(=O)C(c2cc(F)cc(F)c2)O)C1)C(F)(F)F 23761,c1(C(N2CC(C#CC(=O)N3CCCC3)C2)=O)cnc2ncnc(O)c2c1 23762,Cc1ccc(C2(C(=O)NCc3c[nH]c(C#N)c3)CC2)cc1.C12CCCN1C(=O)N2 23763,C(C(C)(C)C(F)(F)F)C(N1CC(C(C(N2CC(CC(=O)OC)C2)=O)OC)C1)=O 23764,CC1=C(C(=O)NC2CC3CC(NC(=O)C(O)CN(C)C)CC23)SCCO1 23765,N1(C(c2nn(CC)c(O)c2)=O)CCC2(CC1)CC2CNC(=O)CC(O)CC(C)C 23766,C1(C(=O)NCC2C3CN(C(C4(C)CCCCC4)=O)C2C3)CS(=O)(=O)CC(=O)N1 23767,O=C1CCN(C(C23CC(CO2)N(C(=O)C(C)(C)C2CCCO2)C3)=O)CCN1 23768,N1(C(c2c(C)nc(O)[nH]2)=O)CCC(NC(c2cc(C(F)(F)F)no2)=O)CC1C 23769,CC1CC(C(N2CCOC(CN(C(=O)C=Cc3cocn3)C)C2)=O)CC(C)C1 23770,N1(C(C2(OC)CC(C)C2)=O)C2CCC(C(=O)NCc3cnns3)C1CC2 23771,C(CCCCC(=O)NC1CCC(C)N(C(c2[nH]nnc2C2CC2)=O)C1)NC(C)=O 23772,Cc1nn(CC(=O)NCCCC(=O)NCCC2CCCO2)c(=O)o1 23773,C1(CNC(C2C(=O)NCC2)=O)CC2CC2N1C(c1ccn(CC(F)F)n1)=O 23774,n1(CC(=O)NCC(CNC(C2CC3CCC(C2)O3)=O)OC)nc(C)c(C)c1C 23775,C1(NC(C2(C)CC(NC(c3c(C)noc3)=O)C2)=O)CCOC2(CCC2)C1 23776,C1(O)(CN(C(=O)C(F)=CC2CC2)C)CCN(C(c2ccc(C(F)(F)F)[nH]2)=O)C1 23777,c1(C(=O)NCC2CCC(NC(C3C(C)CCC3)=O)C2)cc2c(F)c(F)ccc2[nH]1 23778,c1(N(C)C)ccc(C(=O)NC(CNC2CCC(=O)N2)C2CC2)cc1[N+](=O)[O-] 23779,c1(C(N(C2CCN(C(c3conc3C(C)C)=O)C2)CC)=O)cc(C(F)(F)F)co1 23780,C1(F)(CNC(c2ccc(C#C)cc2OC)=O)CC2CCC(C1)N2C(=O)C=C(C)C 23781,Cc1cc(C)n(-c2ccc(-c3nc(-c4ccn(C)c4)n(CCC(C)C)n3)nc2)n1 23782,c1(C(=O)NC2(C)CCN(C(C3C(C)C3)=O)C2)cnc2c(c1)CNC(=O)N2 23783,C(=O)(C(O)CCNC(=O)C(O)C1CCCC1)NC(C1CCCC1O)C 23784,C1(CNC(COCCN(C)C)=O)COCCN1C(C1(c2nccn2C)CC1)=O 23785,N1(C(C(CSC)C)=O)CC(NC(=O)C(CO)NC(=O)C(F)(F)F)CC(F)C1 23786,c1(SC(C(=O)NC2CC(CNC(Cn3nnc(C)n3)=O)C2)C)ccc(C#N)cc1 23787,N1(C(C=CC=CCC)=O)CC(NC(c2cnc(C)nc2CC)=O)CCC1C 23788,CC(C)CC(F)C(=O)NCC1(C)CN(C(c2cc([N+](=O)[O-])c[nH]2)=O)CC1C 23789,N1(C(C(C)C(C)(F)F)=O)CCCC2(CCCN2C(c2cnc3ccccn23)=O)C1 23790,C1(C(N)=O)(CNC(C23CC4CC2C3C4)=O)CCN(C(=O)Cc2cccnc2Cl)C1 23791,N1(C(c2c(C)scc2)=O)CC2(CC(NC(C3CC(=C4CCC4)C3)=O)C2)C1 23792,c1(OC)cc(Br)c(C(=O)COC(c2cc3c(s2)CCC3N)=O)cc1OC 23793,N1(C(c2c(CC)nc(C)[nH]2)=O)CC(NC(C2(C)CCN(C)C2)=O)CC12CCC2 23794,c1(CC)cc(C(=O)NC2(C)CCN(C(C3(c4ccnn4C)CC3)=O)C2)ccc1C 23795,c1(C(N(CCCOCCNC(=O)CCC2CCCO2)C)=O)ccc2ncsc2c1 23796,C1(CN2CCC(C=C)C2)CN(C)CCN1C(c1cc(OC)cc(F)c1)=O 23797,N1(C(CC(C=C)CC)=O)CC(C)CN(C(=O)CCCc2cnn[nH]2)C(C)C1 23798,N1(C(Cc2ccc(C)s2)=O)CCC(C2CC2)C1CNC(=O)COc1ccsn1 23799,c1(C(=O)NC(C)CC(C)NC(=O)C(C)(C)c2ncco2)ccc([N+](=O)[O-])c(N)n1 23800,CCC(CC)CCCC(=O)N(CC(N1CC(O)CC1C(C)C)=O)C 23801,CC(C(=O)NC1C=CC(C(=O)NC(C)C(=O)NCCF)C1)C(F)F 23802,C1(OC)CC(CNC(c2csnc2C)=O)N(C(C2CC(N(C)C)C2)=O)C1 23803,c1(-c2nc(NC(CC3(C#N)CNC3)=O)sn2)ccccc1OC(F)F 23804,C(C)(CN=c1[nH]c(N(C)Cc2cccc(CO)n2)nc2ccccc12)OCC 23805,CCCC(C(O)C(=O)NCC1(O)CCN(C)C1)NC(c1ccccc1CC)=O 23806,N1(C(C2C(COC)C2)=O)C2CCC1CC(NC(c1cc(-c3cccs3)on1)=O)C2 23807,C#CCCCC(=O)N1CCC(C(F)C(=O)Nc2cnn(CCC)c2)C1 23808,c1(C(=O)OC)cnc(C(C)C)[nH]c1=NCCCC(C)(C)NC(=O)CC(C)SC 23809,C(CCCC(=O)N1CC(NC(c2sc(CC(C)C)nc2C)=O)C(C)C1)OC 23810,C(C(C)(C(=O)NC(C(=O)NC1CCOCC1O)C(C)C)OC)OC 23811,c1(CC(N2C(CCN(C(CC(CC)SC)=O)C)CCCC2)=O)ccc(C)c(C)c1 23812,Cc1c(C(=O)NCCCC(C)NC(C2CCCS2)=O)ccc(Br)c1F 23813,C1(CC=C)(C(=O)NC2CC(C(C)NC(c3cscc3Cl)=O)C2)CCOC1 23814,N1(C(C2(C)CCOC2)=O)CCC(C(F)F)(CNC(c2ncc(F)cn2)=O)C1 23815,C(=O)(C(C)CSC)N(CC(=O)NC(C)CCSC)CCOC 23816,C1(C(=O)NCC2(O)CCN(C(c3c(C)cc(F)s3)=O)C2)SC2C=CC1CC2 23817,C#CC1(O)CCN(C(c2conc2CNC(=O)C(C)(C)C=C)=O)CC1 23818,c1(-c2ncc(C(=O)OCc3ccnn3C3CC3)s2)ccccc1Cl 23819,c1(C(=O)NC(C)C(C)(C)NC(=O)CC2COCCN2C)cccc(C(C)(F)F)n1 23820,N1(CC(=O)NCC2(CC(=O)N(CCOC)CC3CC3)CC2)C(=O)CCCC1=O 23821,Cc1cncc(C=CC(=O)NCCN(C(=O)C(c2cc(Cl)ccc2Cl)(F)F)C)c1 23822,Cn1cnc2nc(N3CCC4(C3)CC4(F)F)nc(NCCCc3nc[nH]n3)c12 23823,Cc1nc2cccc(C(N3CC(CNC(C4(CCO)CC4)=O)C4(CC4)C3)=O)c2s1 23824,C(=O)(C(C)=CCNC(=O)C(F)C1CCC1)NCC(C)NC(C)=O 23825,N1(C(C2CCC(C)(CC)O2)=O)CCCC(N(C)C(c2cccc(O)n2)=O)CC1 23826,Cc1cc(NC2(F)CC2)ccc1C(=O)NCCCC(C)NC(=O)C1=CCCC1 23827,C(=O)(C(C)(CC1CCC1)OC)NCC1C(NC(CCNS(CC)(=O)=O)=O)CC1 23828,Cc1nnc2ccc(C(N3CCC(NC(=O)CC4(C)CC4(Cl)Cl)C3(C)C)=O)cn12 23829,c1(C(N2CCC(C(C)NC(C=C=C(C)C)=O)C2)=O)cccc2c[nH]nc12 23830,C(=O)(CC(O)CC(C)(C)C)NCCN(CC(C(C)C)OC)C(=O)COCC(C)(C)C 23831,C1(CC(=O)N(CCOCC)C)CN(C(=O)CC2(COC)CCOCC2)CCO1 23832,Cc1nn(CC(=O)NC2CC3C(NC(=O)C(c4cnccn4)C)C3C2)c(=O)o1 23833,c1(C(C(N2C(CN(C(C(F)=CCC)=O)C)CCC2)=O)O)ccccc1F 23834,N1(C(C(C(C)O)(C)C)=O)CC2COCC2(C(=O)NCc2ccc(Cl)cc2)C1 23835,c1(C(C(=O)NCCCN(C(=O)C(O)c2ccsc2)CC)C)c(F)cccc1F 23836,C1(C)(C(N2CCN(CCCNC(C(C(C)C)F)=O)CC2)=O)CCCCC1(F)F 23837,C1(C(=O)NCCOC2CCN(C(CCNC(C)=O)=O)CC2)CC(C(C)C)=NO1 23838,C(C(CCC)C(=O)N1CCC1(C)CC)NC(C(C=C)(C)C)=O 23839,c1(C(N2CCN(C(CC(C=C)C)=O)CC2C2CC2)=O)ccn2ncc(C)c2n1 23840,N1(C(C2C(CCC)C2)=O)CC2(C)CC1C2NC(c1ccc(=O)n(C(C)C)c1)=O 23841,C(C)(C)(C(=O)N1CCC(C(F)C(=O)N(C)Cc2nc[nH]n2)C1)SC 23842,c1(C(=O)NC2CC(C)N(C(=O)CC3COCCO3)C2)ncc(Cl)cc1Cl 23843,c1(C2C(=O)N(C3CCOCC3)CC2)ccc(F)c2cccnc12 23844,c1(CC)ncsc1C(=O)NC1(CN(C(=O)CC(F)F)C)CC1 23845,CCCCC(CNC(c1cnccc1Cl)=O)NC(=O)CC1CC(F)(F)C1 23846,C1(C(N2CC(C(C(=O)NC3C=CC(CO)C3)OC)C2)=O)CC(C)(CO)C1 23847,N1(C(C(CC=C)(F)F)=O)CCC2CN(C(=O)CC3CCCN3CC)CC2CC1 23848,C1(C(=O)NC(C)(C)CCNC(=O)CC2CC=CC2)CC2COCCN2C1 23849,Cc1c(C(=O)NS(=O)(=O)c2cc(Br)ccc2Cl)cc([N+](=O)[O-])cc1I 23850,CCC(C)C(O)C(=O)N1CCCC(CN2CCN(C(=O)C3=COCCC3)CC2)C1 23851,c1(C(=O)NC(C(CO)NC(c2cccc(C(C)=O)c2)=O)C)onc2c1CCCC2 23852,N1(CC2CCC(C(=O)OCC(C)C)CC2)CCC(CO)C(F)(F)C1 23853,C=CC(C)CC(=O)NCC1(OCC)CN(C(c2ncn(C)n2)=O)C1 23854,c1(C(=O)NC(CNC(CN(C)CC)=O)C)ccc(C(=O)NC(C)(C)C)cc1 23855,c1(OCC)nc(Cl)cc(=NC(=O)C2CC(F)CN2Cc2cccc(I)c2F)[nH]1 23856,c1(C(N(CC(O)CNC(=O)C=CS(C)=O)C)=O)cnn2cccnc12 23857,c1(C(N2CC(C)(CNC(c3c(C)c[nH]n3)=O)OCC2)=O)cc2c(s1)CCCC2 23858,c1(C(N2CCN(Cc3c(C)n[nH]c3C)CC2)=O)ccc(O)c(C(=O)C(C)C)c1 23859,S(=O)(=O)(c1cccnc1[N+](=O)[O-])NS(NC)(=O)=O 23860,c1(C(=O)NC2C(NC(=O)Cn3nccn3)C2)ccc(SC(F)(F)F)s1 23861,N1(C(CN(CC)CC)=O)CC(NC(=O)C(N2CCSCC2)C)CC(C)(C)C1 23862,C1(O)(C(C)NC(Cc2c(C)scc2)=O)CCN(C(c2n[nH]c(C3CC3)c2C)=O)C1 23863,C1(C(N(CC(CNC(C2(CCOC)CC2)=O)C)C)=O)Cc2cc(F)ccc2O1 23864,C1(C)(CNC(CCNC(Cc2c(C)noc2C)=O)=O)CC2CCC1C2 23865,N1(C(C=CC(CC)=CC)=O)CC2CCC1C2NC(C1C(C)C1C)=O 23866,C1(N(C(c2c(C)nsc2C)=O)C)CCC2CN(C(C3CC(F)CN3C)=O)CC12 23867,S(=O)(=O)(c1cnccc1N1CCS(=O)(=O)C(CO)C1)NC(c1ccc(Br)cc1)C 23868,C1(NC(CC=C)=O)CN(C(C)=O)Cc2nccn2C1 23869,c1(C(N2C(CNC(C3(C)CC=CCC3)=O)CC2)=O)c(N)cc(F)c(Br)c1F 23870,c1(NC(CC)CO)cc(Br)ccc1S(=O)(=O)NC1CCCN(C)C1 23871,CCCC(CCCO)C(=O)N1CCCC(C)(CNC(C2CCCC2(C)C)=O)C1 23872,C1(C2CCOCC2)(Nc2cccc(Cn3c(C)csc3=O)c2)CC1 23873,N1(C(c2ccc(-c3ccco3)[nH]2)=O)CCC(NC(C2(CC(F)F)CC2)=O)C(O)C1 23874,CCC(c1cccc(Cl)c1)=CC(=O)NCCCCN(C)C(C1CCCN1CC)=O 23875,C(=O)(C(O)CCCC)NC(C1(O)CCN(C(CN(CCC#C)C)=O)C1)C 23876,N1(C(C(C2CCCC2)OCC)=O)CCC(CNC(c2cnc(O)o2)=O)CC1C 23877,N1(C(C=CC=CC)=O)CCN(C(=O)Cn2c(C)c(C)sc2=O)C(c2ncc[nH]2)C1 23878,Cc1cc(C(=O)NCC(C)(CC(C)C)NC(=O)C(C)Cn2ccnc2)c(C)cn1 23879,Cc1cc(C(C)C(=O)NCCCC2CN(CC(C3CCC3)N(C)C)C2)cc(F)c1 23880,N1(C(CSc2nc(C)[nH]n2)=O)CC(C)OC2(CCN(C(=O)C(C)NC(N)=O)C2)C1 23881,N1(C(=O)NCC23CC(C(F)F)(CO2)C3)CC=CC12CCCC2 23882,C(=O)(CS(=O)CCC(F)(F)F)N1CCC(NC(C(CC)=CCCC)=O)CC1C 23883,c1(C(=O)NCC(CC)NC(c2cn(CCF)nn2)=O)c(OC(F)F)cccc1F 23884,c1(C(=O)NCC2(NC(CCC=C)=O)CCC2)sc2nc(C)nc(C)c2c1C 23885,Cc1ccc(-n2ccnc2)c(C(=O)NC2C=CCN(C(C3CC3C)=O)C2)c1 23886,c1(OCC(N2CC(C3CCN(C(=O)C(F)=CCCF)CC3)C2)=O)cccc(O)c1 23887,Cc1cc(=N)[nH]cc1C(=O)NC1CC(C)N(C(c2cn(CCO)nn2)=O)C1 23888,CC1=CC2CCCC(C1)N2C(=O)NCCCNC1CCC1 23889,CC#CCC(C(=O)Nc1ccc(O)cc1C)NC(=O)C(C)NC(N)=O 23890,C1(NC(CCC(C)OC)=O)CC2CCC(C1)N2C(=O)C(=Cc1cnn(C)c1)C 23891,c1(C(N(CCN(C(C(CCCOC)C)=O)C)C)=O)cccc2c1C1CCC2CC1 23892,N1(C(C2(CCNC(C(CC)C)=O)CCCC2)=O)CC2C=CCC(C2)C1 23893,c1(OC)c(Cl)nc[nH]c1=NCC1(CNC(c2cc(C(F)F)ncn2)=O)CCCC1 23894,C12(C(=O)NCc3ccc(C)c(Cl)c3)CCC(CC1)N(C(=O)C(O)CC(F)(F)F)C2 23895,c1(NC(C(C)C)CCNC(=O)CC2CCCC2)cnc2ccccc2n1 23896,S(=O)(=O)(c1ccc(N2CCC(O)C2)cc1Br)N(CC(CC)NCC)CC.C(C)(C)(C)O 23897,c1(ONC(C(CCO)OC)=O)ccc(Cl)c(OC)c1 23898,N1(C(=O)NCCCCCC)CC(Cc2cc(-c3ccccc3)n[nH]2)C(C)C1 23899,CCS(=O)(=O)CCNC(C1(C(C)NC(c2cnnc(O)c2)=O)CC1)=O 23900,c1(OC)ccccc1C(CNC(C1CCC(C)(C)C1)=O)NC(c1ccoc1)=O 23901,c1(N(CCNC(c2c(OC)cccc2OC)=O)C2CC2)ncc2c(ncn2C)n1 23902,N1(C(C(CCCC)C)=O)CCCC2CN(C(=O)C(=O)Nc3ccc(Cl)cc3)CC12 23903,C1(C(=O)NC(c2ccn(C)n2)C)(NC(Cc2c(C)ccs2)=O)CCN(C)C1 23904,C(C)(CNC(=O)C(n1nc(C)cc1C)C)(C(C)C)NC(Cn1ncc(CC)c1)=O 23905,N1(S(c2c(NC(CCC)C)nccc2)(=O)=O)CCc2cc(C)cc(C)c2C1 23906,C1(CNC(c2n(CC)ncc2)=O)CC(OC)CN1C(c1cn(C2CC2)nn1)=O 23907,C(=O)(C1=CCCOC1)NC12C(CN(C(C(C)(C)CC3CC3)=O)C1)C2 23908,c1(C(=O)NCC2N(C(C(C(CC)C)O)=O)CC(F)C2)c2n(c(=O)n1C)CCCC2 23909,Cc1ccc(C(F)C(=O)NCC(=O)NCC2CCOCC2)cc1 23910,Cc1nccc(CCC(=O)NCC2CCCCN(C(C3(C)CCCCO3)=O)C2)n1 23911,CCCCC(C(=O)NC)NC(C12CC1CN(C(c1cc(C)ccc1O)=O)C2)=O 23912,c1(C(=O)OC)ncc(NC(C2CC2Cc2cnco2)=O)cc1C 23913,n1(C(CC)C)ccc(=NC(=O)c2ccc(C3CCCN3)s2)[nH]1 23914,C1(CCCNC(=O)CCc2ccccc2)CN(C(=O)CC2CC3CC3C2)CCO1 23915,C(=O)(CCCCC(F)F)N(C1CC(NC(C2CCN2Cc2ccccc2)=O)C1)C 23916,C(=O)(C#CC(C)(C)C)N1C(C)(C(=O)NC(CCCC)C)C=CC1 23917,CC(CN=C(NCC1(N2CCCC2)CCCC1)NC1CCCC1)CC(F)(F)F 23918,N1(C(C2CC(SC)C2)=O)CCC(NC(C2CCN(CC(F)(F)F)C2)=O)C1C 23919,C(=O)(CCC(F)(F)F)NC(C1(O)CCN(C(c2nn(C)cc2Cl)=O)C1)C 23920,C1(C)(NC(COc2ccc(C)cc2)=O)CCN(C(C2CC(C)OC2C)=O)CC1 23921,c1(OC)cc(CCNC(=O)C(F)(F)c2ccncc2)ccc1I 23922,N1(C(COC(C)=O)=O)CC2CCC2(CC(=O)NC(C)(CO)C2CCC2)C1 23923,N1(C(C(C2CCOC2)OC)=O)CC(C)(NC(=O)COC2CCCCC2)C1 23924,C(=O)(C(F)C(C)CNC(c1cncc(OC)n1)=O)NCc1n(CC)cnn1 23925,c1(C(=O)NC(CC(C)NC(=O)Cc2ccon2)C)ccc2cccnc2c1 23926,N1(C(CCC(=O)OC(C)(C)C)=O)CC2(C1)CN(C(c1cnn(CCF)c1)=O)C2 23927,N1(C(c2c(C)nn(C)c2C)=O)CC(NC(=O)Cc2nncs2)CC2(CC2)C1 23928,C1(CNC(C2CC(=C)C2)=O)C2CCCC1N(C(=O)Cc1cc[nH]c(=N)c1)C2 23929,CCCCCCCC(F)C(=O)N1CC(O)(CNC(C2CC3CCC2O3)=O)C1 23930,Cc1c(C(N2CCCC2C(C)NC(C2CCCN2C)=O)=O)cnn1CCO 23931,S(=O)(=O)(c1cccc(S(N)(=O)=O)c1)NC(c1ccc(C)c(S(N)(=O)=O)c1)=O 23932,N1(C(C(C)N(C(=O)C2=NOCC2)C)=O)CC(F)CC1C 23933,C1(OC)CN(C(=O)COCc2ccccc2)CC1NC(=O)C(C)CF 23934,C(CNC(=O)Cc1c(Cl)cnn1C)(CCCC)NC(CSCC=C)=O 23935,C(c1ccc(F)cc1F)=CC(=O)NCCC1(NC(C(CCSC)OC)=O)CCC1 23936,C(=O)(CCCCC(=O)OC=[IH])N1C(C)CC(CNc2csc(CO)n2)C1.C(C)(C)C 23937,C(=O)(C1=CC2CCC(C1)C2)N(CC(CC)NC(C1CCC([N+](=O)[O-])CC1)=O)C 23938,C(C)(C)(CCN=c1nc(C#N)cc(C)[nH]1)NC(c1ccc(OC)cn1)=O 23939,C1(CC)CN(C(c2nc(C3CC(N)CN3)cs2)=O)CCN1 23940,C1(C(=O)NC2CC(NC(Cn3c(C)ccc3C)=O)C2)CC(S(C)(=O)=O)C1 23941,Fc1ccccc1CN=C(NC(C1CC1)C1CC1)NC1CCOC(c2ccccc2)C1 23942,c1(C(=O)NCC(CNC(COCC)=O)C)c(Br)c(C)nn1C 23943,CC1SCCCC1C(=O)NC1CCN(C(=O)C=Cc2cnccn2)CC1 23944,N1(C(C(C)(C)O)=O)CCC(C2CCN(C(C3(CCCF)CC3)=O)CC2)C1 23945,N1(C(CCCOCC=C)=O)C2CCC1C(C(N1CCC(C(C)CO)CC1)=O)C2 23946,N1(C(CCSCCC)=O)CCN(C(=O)Cc2nocc2C(C)C)CCC1C 23947,C=CC(CC)CC(=O)NCC1(O)CCN(C(c2cnc(C)c(OC)c2)=O)C1 23948,CCC(C)CCC(=O)N1CCC(CNC(c2cncnc2C)=O)C1(C)C 23949,C(C)(C(=O)N(CCNC(=O)CN1CCC1C)CC)OCCC#C 23950,C#Cc1cc(NC(C(CNC(C2CC2CC(C)C)=O)N(C)C)=O)ccc1C 23951,Cc1nsc(NC(=O)NCC=CCF)c1Cl 23952,C1(C(=O)NCCC(=O)NCC#C)CCCC(NC(=O)CN(CC)CC)CC1 23953,C1(NC(C(C)C2CC2)=O)CN(C(c2cc3scnc3[nH]2)=O)CC12CCOCC2 23954,c1(C(=O)NC2CCN(C(C3(OC)CCC3)=O)CC2)cnc2nc(C)ccc2c1O 23955,N1(C(C2C(C(=O)OC)CCCC2)=O)CCOC2(C1)CN(C(C1(O)CCC1)=O)C2 23956,c1(C(=O)NCC2CCCN2C(c2ccc(O)cc2)=O)cc(Br)cc2c1OCC2 23957,C1(NC(c2ccn(CC)n2)=O)CC(C(N2CC(O)(C(N)=O)C2)=O)C12CCC2 23958,c1(C(=O)OC)cc(Br)cc(C)c1NC(C1CN(C(=O)C(F)(F)Cl)CC12CC2)=O 23959,Cc1ncnc(C(N2CCCC(NC(C3(F)CCCOC3)=O)C2)=O)c1C 23960,Cc1noc(C)c1CC(=O)NCC(C1CC1)N(C)C(C1CC2C=CC1C2)=O 23961,N1(C(c2cc(C)c(C)o2)=O)CCC(C)(CNC(=O)CCNC(C2CC2C)=O)CC1 23962,C1(C(=O)OCC)(C(=O)N(C2CCN(C(C3CC=CCO3)=O)C2)CCO)CC=CC1 23963,C(N=c1[nH]c2ccc(Cl)cc2[nH]1)C1(CCO)CCCCC1 23964,CCC(C)(C)CC(=O)NCC1OCCC1C(=O)Nc1cc(OC)ccc1O 23965,n1(CC(=O)NC2C(CNC(C(C)C)=O)COC2)cc(C(N)=O)c2ccccc12 23966,C1(=O)CCCCCn2cc(nn2)-c2ccccc2O1.CC1(CO)COC1 23967,c1(NC(CNC(C2CC(=C)C2)=O)=O)ccc(CCCC)nc1 23968,C(=O)(NNC(=O)N1CCCC1C(F)(F)F)c1n(C)ncc1 23969,c1(CCC)cccc(C(=O)NC(C)CCCNC(=O)CC2CC3(CC3)C2)c1 23970,C1(COC)(NC(=O)CNC(N)=O)CCN(C(c2ncncc2Br)=O)CC1 23971,c1(C(=O)NC2C(C)CCN(C(=O)CCn3cncn3)C2)cccc2c1OCC2 23972,CC(C)C(C)(C)C(=O)NCc1cc(C(=O)NC(C2(CO)CC2)C)n[nH]1 23973,O=S(=O)(c1ccc(NCC2(CO)CCCC2)cc1Br)NCCc1cc(F)ccc1F 23974,C1(C2C(C#N)CC2)CCC2(CC1)CC(NC(=NCCN=[N+]=[N-])NC1CCOCC1)C2 23975,c1(SCC(=O)NCC2(OC)CCN(C(C(CC)N(C)C)=O)C2)nc2ccccc2s1 23976,c1(C(N2CCN(C(C3C(COC)C3)=O)C(C)C2)=O)sc2ccccc2c1Cl 23977,CC1(C)CCCC(CC(=O)NCC(C)(O)CNC(C2CC(O)C2)=O)C1 23978,CC1CC(C(N2CCN(C(=O)COc3ccc(Cl)cn3)CC2C)=O)CCC1C 23979,N12CC(C(F)C1)n1cc(nn1)CNc1sccc1C2=O.N1(CC)CCSCC1 23980,c1(C(N2CC(C(C(=O)NC3CCC(=O)NC3)OC)C2)=O)nccc(C)c1N 23981,C1(NC(COCCOC)=O)CC(NC(c2sccc2C#N)=O)C12CCC2 23982,C1(NC(CC(C)O)=O)CN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CC1(C)C 23983,C(c1cccc(F)c1)=CCC(=O)NC(c1cn(CC(C(=O)OC)(F)F)nn1)C 23984,C1(C(=O)NC(C(=O)NCCCC)C)OCCOC1C 23985,CCS(=O)(=O)CC(=O)NC(C)(CNC(c1c(C2CC2)noc1C)=O)c1ccccc1 23986,c1(NS(C)=O)ccc(C2C(C(=O)NC(=O)CN(C)C(N)=O)C2)cc1 23987,Cc1c(CC(=O)NCC2CC2CNC(=O)CC2CCOCC2)cccc1[N+](=O)[O-] 23988,N1(C(C2(CCC=C)CC2)=O)CCC(NC(=O)CC2CC(C)=NO2)C2(CCC2)C1 23989,N1(C(CCCCN(C(=O)CCC2CCOC2)C)=O)CCn2nc(C)cc2C1 23990,C1(N)(C(=O)NCC(c2cnn(C)c2)N(C)C)CC(C(C)(C)C)C1 23991,N1(C(C2(C=C)CCC2)=O)CC2C(NC(=O)CCCc3ccc(O)cc3)C2C1 23992,Cn1nnc2ccc(CN3CCCC3c3ccc[nH]3)cc12 23993,Cn1cnc(C#N)c1C(=O)NC(c1cccc(Cl)c1)CNC(=O)CS(C)(=O)=O 23994,CCC(C)C(C(=O)NCCCC(C)(C)NC(C1C2CCC1CC2)=O)OC 23995,c1(C(N2CC=CC(NC(C3=CCN(C)C3)=O)C2)=O)nccc2occc12 23996,C(CC1CC1)(C(=O)NOC1CCC(O)C1O)NC(CC(COC)C)=O 23997,N1(C(C2C(C)N(C)CC2)=O)CCC2CN(C(=O)CNS(N)(=O)=O)C(C)C12 23998,c1(C(=O)NCC2N(C(CC#N)=O)CCOC2)cccc2c1OCC2 23999,C(C(=O)N1CC(NC(=O)Cc2c(F)cncc2Cl)CC(O)C1)(C(C)(C)C)N(C)C 24000,c1(OC)cc(NCc2cc(O)nc(O)n2)nc(OCCOC)n1 24001,c1(-c2c(OC(F)(F)F)ccnc2)ccc2c(c1)CN(Cc1cnc(O)c(Br)c1)C2 24002,C1(N(C(C2(CC)CCC2)=O)C)CN(C(=O)C=CCO)CCC1O 24003,C12(CC(=O)N(C)CC3CCC(CNC(C(=O)NCC)=O)CC3)CCC(CC1)OC2 24004,CCC(CC)C(C(=O)N1CCC(F)(F)C(CNC(C2C3CCCCC23)=O)C1)OC 24005,N1(C(CC2(C(=C)F)CCC2)=O)CCS(=O)(=O)C(CCNC(C2CC2C)=O)C1 24006,c1(C(=O)NC2(C(=O)OC)CC23CCC3)cc(O)ccc1O 24007,c1(C(=O)NCC2CN(C(COCCC)=O)C2)c[nH]nc1-c1cnn(C)c1 24008,c1(OC)ccc(C(=O)NC2CC(C)CN(C(c3c(C)cnn3C)=O)C2)c(F)c1Cl 24009,O1NC(=O)C(CCSC)NC(=O)CCC1.C1(C(=O)OC)CC1(F)F 24010,C1(NC(C(C)SC)=O)CCN(C(C2CC(n3cnnc3)C2)=O)CCC1(F)F 24011,c1(C(=O)NCC2C3CN(C(C4=CC(C)(C)C4)=O)CC32)[nH]cc2c1CCC2 24012,C(=O)(C(F)C(=O)NC(=O)Cc1ccc(O)cc1)NCCCOCCCOCCOC 24013,c1(CCOC(c2cnn(CC)c2C(F)(F)F)=O)ccc(Br)cc1OC 24014,C1(CN(CC(=O)NC(C)C)C)CCCCN1C(=O)CC1CCC=CCC1 24015,C1(CC(c2nnnn2C2CCCCC2)(C)NCCN2CC=CC2)CCCC(=O)N1 24016,CCC(C)CCCCC(=O)N(C1CCCN(C(c2cnc(S)n2C)=O)C1)C 24017,Cn1ncc2c(NC3CC4CN(C(C5C6CC7C(C6=O)C57)=O)CC34)ncnc12 24018,C(=O)(CCCCN(C)C(c1ccn(CC)n1)=O)NC(C#C)CC1CCCC1 24019,CCC(C)CC(C)C(=O)N(C)CC1CC(F)CN1C(=O)COC(C)(C)CC 24020,CS(C)(=O)=Nc1ccc(C(N2CCN(C(c3ccc[nH]3)=O)C3CCC23)=O)s1 24021,C1(C(=O)NOCC2CCOCC2)(C(C)C)CCCN1C(=O)CC1CCCO1 24022,c1(C(N(CC(CNC(C(C)=C(C)C)=O)C)C)=O)c(C)c[nH]c1CC(N)=O 24023,c12cc3c(cccc3[nH]1)C2=O.c1(C(N(CCC)CCN)C)ncc(C)o1 24024,C#Cc1ccc(C(=O)NCC(C)(C2CC2)NC(=O)C(C(C)(C)C)NC(N)=O)cc1 24025,Cc1cc(Cl)cnc1-c1cn(CCCC(=O)N(CC(C)(C)S(C)(=O)=O)C)nn1 24026,c1(OC)ccc(C2(C(=O)N(CCCCNC(=O)CN(C)C3CC3)C)CCC2)cn1 24027,C1(C(N2CC(C3(NC(C(c4ccnn4C)C)=O)CC3)C2)=O)CS(=O)(=O)CC(=O)N1 24028,N=c1cc(C(N2CCN(C(=O)C=CC3CCOC3)CC2CCO)=O)[nH]c(=N)[nH]1 24029,Cc1nc(-c2ccccc2)sc1C(=O)NC1(CCNC(C2(C)CC2(F)F)=O)CC1 24030,C1(NC(c2ccc(F)c(Cl)c2F)=O)CN(C(C2SCCS2)=O)CC12CCOCC2 24031,c1(C(=O)OC)sccc1S(=O)(=O)NCC1C2CC1N(C(=O)C(C)CC(C)C)C2 24032,c1(Nc2n(CC)nnn2)ncccc1OC(c1nnn(C)c1C(F)(F)F)C 24033,c1(OCC)ccnc(C(N2CC(CCNC(C3(OC)CCOC3)=O)C(C)C2)=O)c1 24034,C1(NC(c2ccc(N(C)C)c(F)c2)=O)CN(C(C2(C)C=CCC2)=O)CC1C1CC1 24035,CCCC(CCC)C(=O)N1CCC(C(=O)N(C2CC(C)CC(C)C2)C)(OC)C1 24036,C1(C(C(=O)N(C(COC)C)C)C)CCN(C(c2ccns2)=O)C1 24037,n1(CCCOC)c(N(CCC(=O)OC)C2CC2)nnc1-c1coc(C)n1 24038,c1(OCC(N2CCN(C(c3ccc(C(F)F)o3)=O)C3CC23)=O)ccc(Cl)c(F)c1 24039,c1(C(=O)NC(CC)(CNC(C2(C)CSC2)=O)CC)ccc2occc2c1 24040,c1(OC)cnccc1CNC(C1(NC(=O)CC2CSC2)CCC1)=O 24041,N1(C(C(CCC)C)=O)CCN(C(c2cc(C(N)=O)c[nH]2)=O)C2CCC12 24042,C(=O)(C1=C(C)CCC1)NC1CCN(CCCNC(C(CC)O)=O)C1 24043,c1(C(N2CC3C(CC(=O)NCCC(CCC)C)C3C2)=O)ncc2ccccn12 24044,N1(C(C(Cc2ncn(C)c2)O)=O)CCCC2(CCN(C(=O)CNS(N)(=O)=O)C2)C1 24045,CP(C)(=O)c1cncc(CNC(=O)NC(c2ncccc2F)c2ccccc2)c1 24046,C#CCC(CC(=O)N(C(C)C(=O)NC)C)NC(c1cnc(CC)o1)=O 24047,C=CC(C)(C)CC(=O)NC12COC(C1)C(NC(C1CCCC1(F)F)=O)C2 24048,C(CCCC(=O)NCCCC(=O)N(C)C)NC(Cc1n(C)nnc1)=O 24049,c1(C(N2CC3(CN(C(C4=C(C)OCCS4)=O)C3)C2)=O)ccc2c(c1)OC(C)(C)C2 24050,C1(C(=O)OCC2CC(=O)N(C(=O)CCC3CCC3)C2)CCCN(C2CCCC2O)C1 24051,n1(CC(=O)NC2CN(C(c3ccc(NC(C)=O)nc3)=O)C2)c(C)cc(C)nc1=O 24052,c1(OCCNC(=O)C(c2ccc(I)cc2)F)c(F)cc(Cl)cc1F 24053,c1(C(=O)NCC(CNC(=O)CCc2cncc(C)c2)OC)cnn2c1NCCC2 24054,N1(C(C(C)Sc2ccccc2)=O)CCCC12CN(C(=O)C(c1ccccc1)O)C2 24055,N1(C(C(C)=C2CCC2)=O)CCCC(C)(NC(=O)C(=Cc2cnn(C)c2)C)C1 24056,C(=O)(CCC(=O)C(C)(C)C)NCC1C(C)CCCN1C(C1CCCCC1(C)C)=O 24057,c1(C(N2CC(CNC(C=CC=CCC)=O)C(F)(F)C2)=O)c(S(C)(=O)=O)cnn1C 24058,C1(CC(=O)NC(CC=C)CNC(=O)C=CCC)COC(C)(C)CO1 24059,N1(C(CCC(C)=O)=O)CCC2(CCCN2C(c2nn(C)c(C)c2Br)=O)CC1 24060,N1(C(CCNC(=O)NC)=O)CC(CO)CC1CNC(=O)CC1CCCC12CC2 24061,C1(OCCNC(C(C)SC)=O)CCN(C(=O)CCOC(C)=O)C1 24062,C1(NC(c2cc(C)sc2C)=O)CC12CCN(C(c1nccnc1N)=O)C2 24063,N1(C(=O)CC2CC=CCC2)CCC2CC(CNC(=O)CC3(O)CCC3)CCC2C1 24064,N1(C(c2ccnc(C)n2)=O)CC2CC(NC(c3csc(C(C)(C)C)n3)=O)CC2C1 24065,C1(NC(c2c(SC)csc2)=O)CC2CCC1(NC(=O)CC(C)(C)C#N)C2 24066,C(=O)(C(C)CC(F)(F)F)NCCCCCNC(c1ccc(OCC(C)C)nc1)=O 24067,c1(CC(=O)NCCC(CNC(C(CC)C)=O)O)cccc2cnccc12 24068,CCCCC(C)CCC(=O)NCC(CC)NC(C1CCN(C)C1CC)=O 24069,c1(NC(=O)CC2CC(O)CN2C(C2CCCSC2)=O)cc(O)cc(F)c1 24070,CC1CN(C(=O)CNC(N)=O)C(C)CN1C(c1cc(N)cnc1Br)=O 24071,Cc1c(NC2CC(C)NC(C)C2)ncnc1N(C)CC1CCOCC1 24072,N1(C(c2n(C)c(Cl)c(Cl)c2)=O)CCC2(CCCCC2NC(=O)Cc2cnc[nH]2)C1 24073,CCC(CC(=O)NC1CCC(C)N(C(c2nc(C)sc2C)=O)C1)CC(C)C 24074,c1(C(=O)NCCN(C(c2cc(C)ccc2N)=O)CC)coc2c(Cl)cccc12 24075,c1(OCCNC(C(C)C(C)S(C)(=O)=O)=O)c(Cl)cc(Cl)cc1C#N 24076,N1(C(CCC2(C)CCC(=O)N2)=O)CC2CCC(C1)C(NC(=O)CC1CC1)C2 24077,C12(C(=O)NCC(CCOC)NC(c3ccsc3)=O)CCC(OC)C1C2 24078,C1(CNC(C2(NC(C)=O)CCCC2)=O)CN(C(c2ncncc2Cl)=O)CC1C 24079,Cc1ccc2c(C(=O)NC3C4CN(C(C5(CC(F)F)CCC5)=O)CC34)onc2c1 24080,C=CCCC(C(=O)NCCC(O)C(F)F)NC(=O)C(=O)NC1CC1 24081,c1(C(=O)NC2C(NC(CC3(C=C)CCC3)=O)CCCC2)cc(F)c2[nH]nnc2c1 24082,c1(OC)cc(C(N2CCCC2CNC(C2C(C#N)C2(C)C)=O)=O)cc(Cl)c1 24083,c1(C(N2C(CNC(C(C)CC(N)=O)=O)(CO)CCC2)=O)cnn2cccnc12 24084,c1(C(N2CCC(N3CCN(C(C)=O)CC3)C2)=O)n[nH]c2ccc(Cl)cc12 24085,Cc1ncc(C=CC(N2CC(F)(F)CC2CCNC(=O)C(C)C(F)F)=O)c(O)n1 24086,c1(C(=O)NCC(CNC(c2sc(CC)c(C)c2)=O)CO)ccc2cccnc2n1 24087,C1(NC(CN(C)CC)=O)C2CC3CN(C(=O)CC4CCCC(C)(C)CC4)C1C3C2 24088,c1(COC)nc(CC(=O)NCC2CC2N)cs1.C1(=O)CC12CC2.CSC 24089,C1(C(C(=O)NCC(C)C)N(C(CCCC)C)C)CCC2(CC1)CC2 24090,C#CC1CN(C(C2(NC(c3cnc(Cl)n3C)=O)CCCC2)=O)CCN1C 24091,N1(C(CC(=C)C)=O)CCC(OCCCNC(=O)CC2CC3CC3C2)CC1 24092,Cc1ccc(C=CC(=O)NCCCC2CCCN2C(=O)CN(C)C)nc1 24093,C1(CNC(CC(C)C)=O)CCCCN(C(c2cc(=N)[nH]c(=N)[nH]2)=O)C1 24094,C(=O)(CCC(C)SC)N1C(CNC(C=CC=CCC)=O)C=CC1 24095,c1(N2CCN(C(CCCCSC)=O)CC2C)nc(Cl)nc2[nH]ccc12 24096,C(CC(COC)N=c1[nH]c(=NCc2cnc(OC)n2C)[nH]c2c1SCC2)OC 24097,N1(C(C(CC#C)O)=O)CC2CCCC(C1)N2C(=O)CCN1CCCC(C(N)=O)C1 24098,CC(C)(C#N)C(=O)NCCc1ocnc1CNC(=O)CCc1nncs1 24099,C1(C(=O)NCCCOCCNC(CSS(C)(=O)=O)=O)CC2(CCOCC2)CO1 24100,N1(C(C2CC(C)(C(=O)OC)C2)=O)CC(NC(=O)Cc2cc(C)on2)C(O)C1 24101,CC1C(NC(c2c[nH]ccc2=O)=O)CC2CCC1N2C(c1ccc(F)s1)=O 24102,c1(C(N(C2CCN(C(=O)OC)C2)CC)=O)ccc(NC(=O)CC2(C)CCCO2)cc1 24103,C(=O)(C(C)CC(C)(C)C)N(C(C)C(=O)NCCCC(N)=O)CC 24104,C1(NC(C2(CC=C)CC2)=O)CS(=O)(=O)C2CN(C(C3CC(OC)C3)=O)CC12 24105,N1(C(CCC=C=C)=O)CC2(C1)CN(C(c1cc(C)nc(C)n1)=O)C2 24106,c1(OC)ccc(C2CN(C(C3CC34CC(O)C4)=O)CC2NC(C2(C)CC2)=O)cc1 24107,C1(C(N2CCN(C(CC(c3c(C)noc3C)C)=O)CC2)=O)CC(C2CC2)=NO1 24108,C12(CNC(c3c(C)cccc3)=O)CCCC1CCN2C(=O)Cc1cnn(C)c1C 24109,c1(OC)cc(OC)cc(CN2CCC(O)C(C(=O)Nc3ccc(C)cc3C)C2)c1 24110,C1(C(=O)NCC2(C)N=C(C)SC2)CC(C)(C)CN1C(=O)CCC1CCCCC1 24111,c1(SC)ccc(C#N)c(SC(C(F)F)C2CC2)n1 24112,C(=O)(C(C#N)C(C)C)NCC1(C(=O)NCCc2ncc[nH]2)CC(=C)C1 24113,C1(C(=O)NC2CCCC2)(CC)CN(C(=O)C(CO)OC)C1 24114,Cc1nc2sccn2c1C(=O)NC1CN(C(c2cccc3ccoc23)=O)C1 24115,C12CN(CC1(F)F)C(=O)OC2.C1(N(C)C(=O)NC(C)(C)C)CCN(C)C1(C)C 24116,C(=O)(C1=Cc2ccc(Cl)cc2OC1)NCCOCCCNC(C=CC(C)C)=O 24117,C(CC(O)C(=O)NC1CC(NC(=O)CCSc2ccccc2)C1)SC 24118,c1(C(C(=O)N(CCN(C(=O)C(O)CF)CC)CC)O)ccccc1OC(F)(F)F 24119,c1(N(CCCC(F)(F)F)C)nc2c(c(=NCCc3n[nH]c(C4CC4)n3)[nH]1)CCC2 24120,c1(COC(C2CC(=C(F)F)C2)=O)cccc2ncccc12 24121,C1(CC(N2CC(C(C)NC(CC(C)C3CCCC3)=O)C2)=O)Cc2ccccc2O1 24122,c1(C(=O)NCC(COC)O)n[nH]cc1CNC(=O)CN1CCCC1C 24123,C1(C)(CNC(C2N(CC)CC2)=O)CC(F)(F)CN1C(C1CC(C)C1)=O 24124,c1(C(N2CCC(O)(CN(C(C3C(OCC)C3)=O)C)C2)=O)cnc2cnccc2c1 24125,C(=O)(N1CC(O)CCO1)C1(CC)CCN(C(=O)C(O)CC(F)(F)F)CC1 24126,C1(C)(C(=O)NC2CC(NC(c3c(COC)scc3)=O)C2)CCC2(CC1)OCCO2 24127,C1(C)(C(=O)NC2CCC(CNC(c3cc(CC)oc3C)=O)C2)CC(C(C)C)=NO1 24128,C1(NC(c2ccc(O)nc2Cl)=O)CC(F)CN(Cc2cc(B(O)O)co2)C1 24129,CC1CCCC(CCNC(=O)CC2CC(O)CN2C(c2cnn(CCO)c2)=O)C1 24130,N1(C(CCCCOC)=O)CC(CNC(=O)C2=NOC(C(C)(C)C)C2)C(F)(F)C1 24131,N1(C(C(CCCCC)C)=O)CCCC2(CCCN2C(=O)Cc2nnc(C)s2)CC1 24132,Cc1nn(-c2ccccc2)cc1C(=O)NCC1C2CC1N(C(=O)C=CBr)C2 24133,Cc1cc(C)c(CC(=O)NCC(F)CNC(=O)C(c2ccccc2)=O)s1 24134,C(CC(O)C(=O)N1CC=CC1CNC(=O)CSC(C)C)SC 24135,C12(NC(C3CC4CCC3C4)=O)CCC(CC1)N(C(c1cnc3occc3c1)=O)C2 24136,n1(CC)nnc(C(=O)NCc2csc(CNC(c3cc[nH]n3)=O)n2)c1C 24137,c1(C(=O)NC2C(NC(CC3CC(=O)NC3)=O)CCC2)cccc2nccnc12 24138,Cc1nc(C2CC2)ncc1C(=O)NC(CCNC(=O)C(C)NS(C)(=O)=O)C(C)C 24139,CC(C)(C)CCCC(=O)NC1CCN(C(=O)CC2(CCCO)CCCC2)C1 24140,c1(CNC2(c3n(CCCF)nnn3)COC3(CCC3)C2)nc2c(s1)CCCCC2 24141,CC1CCCN(C(C2(N(C)C)CCC2)=O)C1CNC(=O)CC1CC1 24142,N1(C(C2(C(F)(F)F)CC2)=O)CCC2CN(C(=O)C(F)(F)Cl)CC2C1 24143,Cc1cc(O)c(F)cc1NC(C1CCN(C(c2cscc2Cl)=O)C1C(C)C)=O 24144,N1(C(CCCC=C)=O)CC(C(N2CCCC2CSC)=O)C2(CC2)C1 24145,CC(CCC(=O)N1CCOC(CCO)C1)NC(=O)C=C1CCC1 24146,N1(C(CNC(C)=O)=O)CC(C(N)=O)(CNC(C2(c3ccno3)CCC2)=O)C1 24147,Cc1coc(C)c1C=CC(N1CC(O)(CCNC(C2COC(C)C2)=O)C1)=O 24148,C1(N(C(C=CC)=O)C)CN(C(=O)C(C)N(CC(F)(F)F)C)CC1(C)C 24149,c1(C(=O)NC(CN(C(c2nscc2C)=O)CC)C)cnn(C(C)(C)C)c1 24150,c1(CC)[nH]nc(C(=O)NCC2(OC)CN(C(=O)C(C)OC(C)(C)C)C2)c1[N+](=O)[O-] 24151,C1(C(N(C2CCN(C(=O)OC(C)(C)C)CC2)C2CC2)=O)SC2C=CC1CC2 24152,CC(C)C(C)CC(=O)NCC1CCCC(CNC(=O)C=Cc2ccncn2)C1 24153,C1(C(=O)NC(c2ccc(Cl)s2)C)CC2(CC(=O)C2)C1.C12CCN(C1)CCNC2=O 24154,Cc1c(C(N2CCN(C(c3c(Cl)cnn3C)=O)C3CC23)=O)cccc1O 24155,c1(COC)ccc(C(=O)NCC2CC(CNC(=O)CCc3cncn3C)CO2)o1 24156,N1(C(c2c(CC)ccc(Br)c2)=O)CCCN(C(=O)CC2CC(C)C2)CC1C 24157,c1(C(=O)NCC2(Cn3cc(C(C4CCCC4)OC)nn3)CC2)nnc(O)nc1O 24158,C1(=O)CC(C2CC2)N1.C1(C(C)C)CCCN1C(=O)CCCn1cccc1 24159,S(=O)(=O)(c1cnc(NCCN2CCC(C)(C)C2)c(Cl)c1)N(C(C(OC)OC)C)C 24160,C1(C)(C(=O)NCCCNC(C2(C)CC(C(F)(F)F)C2)=O)CC2CC2C1 24161,C(=O)(C(O)CC(F)F)N1CC(O)(CCNC(CCC2C(C)=NOC2=O)=O)C1 24162,C1(CC)CCCCC1NC(C1(CC)CN(C(=O)COCC2CCCO2)C1)=O 24163,C1(NC(=O)OC(C)(C)C)CC2CCC1CC2NC(=O)Nc1cc(F)cnc1Cl 24164,N1(C(C(C)CC(F)(F)F)=O)CC2N(C(c3cccc4nc[nH]c34)=O)CCC2(C)C1 24165,c1(C(N2CC(C)C(NC(C3CC4CC4CC3C)=O)C2)=O)ccc(F)c2c1CCC2 24166,c1(C(=O)OCC)c[nH]c(=NCC2(C)CCN(C(=O)CCc3nc[nH]n3)C2)cn1 24167,C1(C(=O)NC2(C)CCN(C(c3cc(Cl)cc(Cl)c3N)=O)C2)OCC2COCCC12 24168,N1(C(COCCOCC#C)=O)CCCC12CCCN(C(=O)C=CC)C2 24169,CC1(C)C2CCC(C2)C1(C)C(=O)NCc1ccccc1CNC(c1csnn1)=O 24170,C1(CNC(COCCC#C)=O)CCCC(CNC(c2cnccc2C(F)F)=O)C1 24171,c1(CC(=O)NCC(C)NC(=O)CC2CCCC2)ccc2c(c1)CC2 24172,c1(C(=O)NCC(C)NC(C=CCOC)=O)cc(C)ccc1S(N)(=O)=O 24173,c1(CNC(C2CC=CCO2)=O)ccncc1OC1CCN(Cc2ccsc2)C1 24174,c1(CC(N2C(C(C)(C)NC(C3CC4C=CC3C4)=O)CCC2)=O)cccc(Cl)c1Cl 24175,N1(C(C2(CC)COC2)=O)CCC(C2CCCN(C(=O)C=CCO)C2)CC1 24176,N1(C(c2c(C#C)c[nH]n2)=O)CCC(C2CC2)C1CNC(C1C=C(C)CS1)=O 24177,CC1CN=C(NC(C2CCCN2C(=O)OCc2ccccc2)=O)S1 24178,c1(C(C)C)ccc(C=CC(=O)NC23CCC2CN(C(=O)CC2CC(F)C2)C3)cc1 24179,Cc1nc2cnn(C)c2cc1-c1ccc(C2CCC(C#N)(C(=O)O)CC2)cc1 24180,c1(C(=O)NCCC(CNC(c2ccnn(C)c2=O)=O)O)c2c(nn1C)CCSC2 24181,CC1CC(NC(C2CN(C)C(=O)N2)=O)CCN1C(=O)Cc1nnc(O)s1 24182,c1(-c2ncc(C(C)NC3CCOC(C(=O)O)C3)s2)ccccc1F 24183,C1(O)(C(N(CCCNC(=O)CNC(c2ccc(C)cc2)=O)CC)=O)CC2CCC1C2 24184,C(=O)(C1=C(C#N)CCC1)NC(CC(=C)Cl)C(=O)N1CCCC(F)(CO)C1 24185,c1(C(N2CCCC(CNC(C3C(CC)CCO3)=O)C2)=O)cc2cc[nH]c(=O)c2s1 24186,C1(C(=O)NC2(C(=O)NCC3(OC)CCCC3)CC2C)CCC(=O)N(C)C1 24187,c1(C(N(CCCCCNC(C(CC)N(CC)CC)=O)C)=O)cc(C)ccc1F 24188,C1(NC(CC2(C)CCN(C(C(CO)OC)=O)C2)=O)Cc2cscc2C1 24189,CCC(CC(=O)NC(C)(CO)C(=O)NC1(CC(=O)OC)CC1)SC 24190,c1(C(=O)NC2CN(Cc3c(Br)ccc(OCC)c3)C2)ccc(O)c2ccccc12 24191,C12(C(=O)NC(CN(C(Cc3cc(OC)cc(Cl)c3)=O)C)C)CCC(C1)C(C)(C)O2 24192,C(=O)(CCCCCF)NCc1c(C(=O)NCC2(OCC)CCOC2)nco1 24193,C1(C(=O)OCc2nnc(C)o2)CC(F)(F)CS1 24194,C1(C)(C(=O)NCCCOC(C)C)CCCN(C(=O)CC2CCOCC2)C1 24195,C1(O)(C(=O)NCc2ccccc2)CCN(C(=O)C(N2CCC(C3CC3)C2)=O)CC1 24196,CC1(C)CCCC1CCNC(=O)C(=O)Nc1ccc(CN2CCCCC2)cc1 24197,S(=O)(=O)(c1ccc(NC(C)CCC)cc1Br)N(C)CC1C(SCC)C1 24198,O=S1CCC(N=c2nc3sccc3c(NCC3(n4ccnn4)CC3)[nH]2)C1 24199,C(=O)(CCS(N)(=O)=O)NCC(CCNC(=O)C(c1cccc(C)c1)F)OC 24200,N1(C(C(COCC)N=[N+]=[N-])=O)CCC2CN(C(C3CN(C4CCC4)C3)=O)CCC12 24201,Cc1ccn(CC(=O)NCC2(NC(c3cn(C)c(=O)cn3)=O)CCCC2)c(=O)c1 24202,c1(NC(c2ccc(Cl)nc2)C)[nH]c(=NCc2cc(N)ccc2F)nc2scnc12 24203,CCC(C)(CO)C(=O)NC1CCCCCC1NC(=O)Cn1cc(C(=O)NC)nn1 24204,N1(C(CCOC(C)C)=O)CCN(C(C2CCC(=O)NC2)=O)C2(CCC2)C1 24205,N1(C(C(C)OCCC#C)=O)Cc2nccn2CC(NC(=O)C2=CCC(C)(C)C2)C1 24206,c1(C(=O)NC(CCC)C)cccc(-n2cc(-c3cnccn3)nn2)c1 24207,N1(CCC)CCCC(C(=O)NCCC2CN(C(c3ccc(C)nc3)=O)CCO2)C1 24208,c1(C(=O)NC23C(CN(C(CC(=O)OCC)=O)C2)C3)c(OCC2CC2)cccc1Cl 24209,C(=O)(CCC(C(=O)NCC1CCN(C(=O)C(O)C(C)(C)C)CC1)N(C)C)OC 24210,c1(NC(C(COC(C)(C)C)N(C)C)=O)ccc(N=Nc2ccc(N)cc2)cc1 24211,CC1CN(C(=O)Cc2cscn2)CCC1NC(c1ccc(C(C)(C)C)cc1N)=O 24212,C1(C(=O)NC2CCC(NC(CC3(COC)CCCC3)=O)CC2)OCC2CCCC12 24213,c1(NC(C2CC2C(=O)NC2C3COCC23)=O)ncc(Cl)nc1Cl 24214,N1(C(C)=O)CCCC2C1CCCN2C(=O)CC(F)(F)CS(C)(=O)=O 24215,C1(C(=O)NC2C(O)CCN(C(c3n(CCC)ncc3)=O)C2)CCn2cnnc2C1 24216,c1(OC2CC(F)(F)C2)ccc(C(CO)NC(=O)OCC)cc1.C1(=O)CO1 24217,C1(C)(CNC(C2C(OCC)CC2)=O)CCCN(C(c2ccc(C(F)(F)F)[nH]2)=O)C1 24218,c1(CNC(N2CCC(c3ccncn3)C2)=O)cc(O)ccc1F 24219,N1(C(C(C)SC(F)(F)F)=O)CC2OCCN(C(c3cc(CCO)on3)=O)C2C1 24220,C1(N(C)C(C2CC(C)(O)C2)=O)CCCN(C(C2CC23CC(F)(F)C3)=O)CC1 24221,c1(CNC(C(COC)OC)=O)ccc(CCNC(c2c[nH]c(C#N)c2)=O)cc1 24222,C(=O)(C(O)C(C)(C)C)N1CCC(CC=C)(C(=O)NCc2cncnc2)C1 24223,C12(NC(=O)Cn3cncn3)CC(CNC(C3(N4CCOCC4)CCCC3)=O)(C1)C2 24224,CC1CCn2cc(C(=O)NCCC3=CCN(C(=O)Cc4nc[nH]n4)CC3)nc2C1 24225,c1(C(=O)NC(CCOC)CNC(C2(C)CCCCC2)=O)cc(=O)n2nccc2[nH]1 24226,N1(C(CCC)=O)CCCC(CO)(NC(c2nn(C)cc2SCC)=O)C1 24227,C=CC(C)(C)CCN=C(NC1CN(C(=O)OC(C)(C)C)C1)N(C)Cc1cnn(C)c1 24228,c1(C(N2C(CNC(=O)C#CC3CCC3)CC2)=O)cc2cccnc2s1 24229,C12CCCN(C1)C(=O)OCCNC2=O.C1(N(C)C)CNC1=O.C(N)(=O)N(C)C 24230,Cc1ccccc1C(C)(C)CNC1CCOC(c2ccc(F)cc2)C1 24231,c1(C2(C(=O)NC(C)CC3CN(C(=O)CC4CSC4)C3)CC2)ccncc1 24232,C(CC(O)CNC(C1(c2ccccc2)CC1(F)F)=O)NC(c1coc(Cl)n1)=O 24233,C1(CNC(C=Cc2n(CC)ncc2)=O)CCC12CCN(C(=O)C(F)OC)CC2 24234,CCCCC(C)CCC(=O)NCCC1(OC)CN(C(=O)C(C)COC)C1 24235,c1(C(N2CC(O)(C(C)NC(c3cc(Br)no3)=O)C2)=O)ccc2c(c1)CCC2=O 24236,Cc1cc(C(=O)NCC2(NC(=O)C(C)OCCC(C)C)CCC2)c(O)c(C)n1 24237,c1(CCC(=O)NC2CN(C(c3c(C)n[nH]c3)=O)C(C)CC2)n[nH]c2c1CCCC2 24238,CS(=O)(=O)CCC(=O)NC1C2CC1CN(C(=O)CCc1cccc(O)n1)C2 24239,S(=O)(=O)(c1cc(Br)ccc1Br)N(C)CC1CN(C(c2ccnc(Cl)c2F)=O)C1 24240,c1(C(c2n(CCOC)nnn2)NCC2(OC(C)C)CCOCC2)cncc(F)c1 24241,C(=O)(CC1=CCN(C(=O)CCC(=O)NCC)CC1)NC(CCCC)C(=O)OC 24242,C1(NC(c2cn(CCC)nc2)=O)(CF)CCN(C(c2cccc(O)n2)=O)C1 24243,O=C1NCCC2CCN(C(c3cc4occc4s3)C(=O)NCc3ccco3)C12 24244,c1(CC(N2CCC(NC(=O)Cc3cnoc3)(CO)CC2)=O)cccc2c1OCO2 24245,c1(OC)cc(F)c(COC(C2CCC2c2ccc(Cl)c(Cl)c2)=O)cc1OC 24246,c1(OC)ccc(C(=O)NC2CC(NC(c3ccn(CCSC)n3)=O)C2)c(F)c1F 24247,C1(O)(CCNC(C(C)OC)=O)CCN(C(c2cccc(CF)c2)=O)C1 24248,Cc1c(C(=O)NC(C2CCCN2C(=O)Cn2cnc(=N)[nH]2)(C)C)ccn1C1CC1 24249,C1(COC)(CNC(=O)CCc2conc2C)CCN(C(c2sccc2C)=O)CC1 24250,N1(CCCCNC(COCCSC)=O)CCCN(C(C2C(C)(C)C2(F)F)=O)CC1 24251,n1(CC)ncn(NC(=O)Cn2cc(CNC(=O)CC3COCCO3)nn2)c1=O 24252,C1(CNC(=O)C=CC2CC2)CC2CN(C(=O)C(c3ccccc3F)O)CC12 24253,c1(C(=O)OC)csc(S(=O)(=O)NC(=O)NNC(=O)C2CCCOC2)c1 24254,C1(CNC(C2C(C)SCCC2)=O)CC(C(=O)NCc2ccc(Cl)cn2)=NO1 24255,C1(C(=O)NCCC(C)NC(C2(CO)CC(F)(F)C2)=O)COC2(CCC2)CO1 24256,C1(OCC(N2CC(C(C)NC(C(C3CCC3)OC)=O)C2)=O)CCC(C)CC1 24257,C(=O)(CCCCC(=O)NCC1CN(C(C2CCCN2c2ccncn2)=O)C1)NC 24258,C(=O)(CCCCCNC(C)=O)NCC1CN(C(c2n(CC)nc(C)c2)=O)C(C)C1 24259,c1(C(N(CC(C)Cc2ccc(C(C)(C)C)cc2)C)=O)cc(F)cc([N+](=O)[O-])c1N 24260,C1(C(=O)OC)CCN(C(=O)C2CN(C(=O)CN3CC4CCC3C4)CC23CC3)O1 24261,C1(CNC(=O)CCc2nc[nH]n2)COC(CNC(C2CC(O)C2)=O)C1 24262,N(C(=NCCCCl)NCC1CC12CCSCC2)CC(Cc1ccc(OC)cc1)C 24263,C1(CC(N2C(CC(=O)NCC3CCC(O)C3)CC2)=O)CN2CCC1CC2 24264,C(C(=O)NCCc1cccc(F)c1)(C(C)C1CCCCC1)N(C)CC1COC(=O)O1 24265,c1(C(N(CCOC)CCNC(=O)CNS(=O)(=O)CC)=O)nc(C)nn1C 24266,C1(OC)(CNC(=O)CCc2ncnn2C)CN(C(c2ccc(C(C)C)s2)=O)C1 24267,c1(OC)c(Cl)nc(NC(c2csc(NC(c3nc(Br)ccc3F)=O)n2)=O)nc1Cl 24268,C1(C(=O)NCCSCC=C)CCCCN(C(c2c[nH]c(=N)o2)=O)C1 24269,c1(SCC=C)ccccc1C(=O)NCC(CO)NC(c1occc1C(C)C)=O 24270,c1(C(=O)NC2C(N(C(COCCC)=O)C)CCCC2)cc(C)c(O)c(N)c1 24271,N1(C(c2c(N)non2)=O)CCC(NC(c2ccn(C3CC3(F)F)n2)=O)C(CO)C1 24272,C(=O)(C(F)C(C)(F)F)N1CC(C)(OCC(=O)N(C)CC2CC2(F)F)C1 24273,C(C1=CCN(C(=O)Cc2ccc(Br)cc2F)CC1)NC(Cn1c(C)cnc1)=O 24274,C(=O)(CC(C)C(F)F)NCCCCC1CCN(C(C2(CC)CC(F)(F)C2)=O)CC1 24275,c1(C(=O)NC(CC2CCOCC2)C(=O)N2CCC2CO)ncnc(O)c1F 24276,c1(C(=O)NC2CC(NC(c3cnc(OCC)s3)=O)C2)nccc(OC)c1N 24277,CC(C)C(C)(O)C(=O)NC(c1ccccc1)CNC(c1ccns1)=O 24278,c1(C(CC)NCC2CCC(C)O2)ccc(O)c(Br)c1 24279,c1(C(N(CCC)CCNC(=O)C(C)C2CCOC2)=O)c(F)ccc2nc[nH]c12 24280,C(CC(C(C)C)(c1nnnn1CC(F)F)Nc1ccc(CO)c(F)c1)OC 24281,C(CCC(=O)N1CCC(CN(C)C)C1)(C(C)C)NC(C=Cc1cc(C)no1)=O 24282,c1(C(=O)NCCC2(C)CCN(C(=O)CCC3CC3)C2)ccn2ccnc2c1 24283,Cc1cc(C(=O)NCC2(CNC(=O)C=Cc3cncs3)CC2(F)F)ccc1O 24284,CC1C2CC(C2NC(C2(C3CC3)CC2)=O)N1C(=O)CC1CCC1 24285,C1(CC)CN(C(=O)C(C2CCCCC2)O)CCN1C(c1cc(C)n(C)c1)=O 24286,N1(C(c2ccn(C3CCOCC3)n2)=O)CCN(C(C2CSCCS2)=O)C2CCC12 24287,C1(C(N2CC(C)C(N=[N+]=[N-])C2)=O)CC(F)(F)C12CCCC2 24288,c1(C(=O)NC2C3(CC(NC(=O)COCC(F)F)C3)C2)ccc2cnnn2c1 24289,C1(NC(C2CCCC(NC(CC3(C#N)CC3)=O)C2)=O)CC2(CNC(=O)O2)C1 24290,CC1CCN(C(=O)CCc2c(F)cccc2F)CC1NC(=O)C=C1CCCCC1 24291,N1(CC(=O)NCC2(O)CN(C(c3c(N)cc(Cl)nc3)=O)C2)CCCCCCC1=O 24292,C1(NC(c2c(Cl)cn(CC)n2)=O)COCCN(C(=O)C(C)Cn2ccnc2)C1 24293,c1(C(=O)NC(C(=O)NC(CCOCC)C)c2cccs2)cc2ccccc2o1 24294,C(C)(C(=O)NCC1CC(C(C)NC(=O)CCNC(N)=O)C1)OCCOC 24295,N1(C(C2CC(=C)C2)=O)CCC(CF)(NC(c2cnc(C3OCCO3)s2)=O)C1 24296,c1(N2CC(C)(C)SCC2)nc(N2CCOC(C)(C3CC3)C2)nc2c1SCC2 24297,C1(CC)CCCCC1C(N1CCC1(C)C)C(=O)Nc1ccccc1Cl 24298,c1(CC(=O)NCC2C(NC(CNC(C3C(C)C3)=O)=O)CC2)ccc(C2CC2)cc1 24299,Cc1c(CC(=O)NCC2(CCNC(=O)CC3CC=CC3)CC2)ncn1C 24300,N1(C(CNS(C)(=O)=O)=O)CC2COCCC2(NC(c2ccn3cncc3c2)=O)C1 24301,Cc1cccc(C(=O)N(C2CCC(NC(C3CN(C)CCO3)=O)CC2)C)n1 24302,N1(C(c2ccccc2S)=O)CCC2(CCC(C(N3CCC3)=O)O2)CC1 24303,c1(NC(COC(C)(C)C)CO)ccc(S(=O)(=O)NCC2CC2(Cl)Cl)cc1Br 24304,C1(C(N2CCC(OCCNC(C(C=C)O)=O)C2)=O)CCC2C(CC1)C2(F)F 24305,N1(C(c2c(C)ccs2)=O)CCC(NC(=O)C(c2ccc(F)cc2F)C)C(F)C1 24306,C=CC(CC(=O)NC(C1CCN(C(=O)CC(F)(F)F)CC1)(C)C)c1ccccc1 24307,C(=O)(C1=C(Cl)CCC1)N(C1CCN(C(=O)C(c2cccnc2)OC)CC1)CCC 24308,c1(OC)ccc(Cl)c(C(N2CCCC2CCNC(C2CC(C)(C)CN2C)=O)=O)n1 24309,c1(CC(=O)NC2CC2CNC(C2CS(=O)(=O)C2)=O)cc(F)c(F)cc1F 24310,C(CN=C(NCc1c(F)cncc1F)NC1CC1C)c1ccc(C(=O)OC)cc1 24311,C1(C(=O)NCC2(C)CCN(C(c3nccc(CC)c3)=O)C2)CCCCS1(=O)=O 24312,c1(C(=O)OC)cnc(NCC2CC(C)N(C(=O)CN(S(C)(=O)=O)C)C2)nc1 24313,c1(C(C(N2CCC(O)(C(C)C)C2)=O)(F)F)ccc2c(c1)OCO2 24314,Cc1cncc(C(=O)NCC2CCN(C(c3ccc(=N)[nH]c3Cl)=O)C2)c1Cl 24315,N1(C(c2cc(C)nn2C)=O)CCN(C(c2c(C)coc2C)=O)CC12CC2 24316,c1(OC)ccc2nc(N3CC(NC(C4(C)C=CCC4)=O)C(C)(C)C3)sc2n1 24317,N1(C(C2CCC(C(C)C)CC2)=O)CCCN(C(=O)C(CO)NC(N)=O)CC1 24318,Cc1cc(C)nc(SCC(=O)N(C2CCCN(C(=O)C(C)C(C)(C)C)C2)C)n1 24319,Cc1ccc(Br)c(F)c1C(N1CC2CC1C2C(N1CC2CC1CC2(F)F)=O)=O 24320,C(=O)(CC(O)C(C)C)NC(CCOC)C(=O)NCC12CC(CN1C)C2 24321,N1(C(CN(C(=O)C(O)C(C)CC)CCC)=O)CC2(COCC(=O)N2)C1 24322,c1(C(=O)NCC(CCNC(CC2CCCC(C)(C)C2)=O)O)cnn2c1CCCC2 24323,N1(C(=O)NCc2c(CC)ccc(F)c2)CCc2cc(OC)ccc2C1C 24324,c1(C(N2CCC(N(C(C3CC=CC3)=O)CC)C2)=O)nc(OC(C)C)ccc1Cl 24325,c1(SCC(=O)NCC2CC2CNC(c2cccnc2C(F)F)=O)ccc(O)cc1 24326,C(C(=O)N1CC(NC(=O)CC2(CO)CCC2)C(C)C1)(C(C)(C)C)NC(C)=O 24327,c1(C(N2CCC(N(C(=O)CC3CCCS3(=O)=O)CCO)C2)=O)cccc2nsnc12 24328,C1(C(=O)NCCCN(C(C(C)SCC)=O)CCO)CCCC1n1ccnn1 24329,C(C(CC(C)C)C(=O)N(C)Cc1c(C)cnn1C)NC(CC(C=C)C)=O 24330,C1(NC(C(CC)N(CC)CC)=O)COCCC1NC(c1cnc(C2CC2)s1)=O 24331,N1(C(C(CC)C)=O)CCN(C(=O)CNC(c2ccccc2C)=O)CC1 24332,c1(CC)cccc(C(=O)NCC2CCCN(C(=O)CN(C)C(C)=O)C2)c1N 24333,c1(OC)ccccc1C(C)=CC(=O)NCCCN(C)C(c1ccc(Cl)c(O)c1)=O 24334,C1(C(=O)NCC(C2CCOCC2)CC)CCC(C2CCC2)CC1 24335,c1(CC)ccc(C(=O)NCCC2(C)CCN(C(c3ocnc3C3CC3)=O)C2)cc1 24336,N1(C(c2c(OC)nsc2)=O)CC2CC(NC(=O)C(C)CCO)C2C1 24337,c1(C(=O)NC2CCC(CNC(C3C(=C)C3C(=O)OC)=O)C2)c(F)cc(Cl)cc1F 24338,N1(C(c2cnn(CC)c2C)=O)CC2(CC2)CC1C(=O)NCC(C)(F)F 24339,C(=O)(CCCCCN=[N+]=[N-])N1CC(CC)N(C(=O)CC(C)c2cnn(C)c2)CC1 24340,CCC(C)C(O)CC(=O)NCC(CC(=O)N1CCOCC1CC)OC 24341,c1(C(=O)NCC(CN(C(C(C)SCC)=O)C)O)ccn(CCN(C)C)n1 24342,c1(C(C)C)cccc(C(=O)NC2CC(NC(=O)CC3CCC(C)(C)C3)CC2O)c1 24343,c1(OCC)ccc(CNC(=O)C(=O)NCC2CCC(O)C2)c(O)c1 24344,c1(C(=O)NCC(C2CC2)NC(C2C(COC)C2)=O)cc2cc(Cl)cnc2[nH]1 24345,CC1(C)CCCOC1CC(N1CCOC(CNC(C2CC(=O)N(O)C2)=O)C1)=O 24346,N1(C(C(C2CCC2)OC)=O)CC(CNC(C2CCCCC2O)=O)C(C)C1 24347,Cc1cc(C(N2CCC(CNC(c3ncccc3C)=O)C(C)C2)=O)[nH]c1C#N 24348,C1(C(N2CCC(N(C(C(c3ccccc3F)C)=O)CCO)C2)=O)C(C)(C)C1(F)F 24349,Nc1ccc(CCCC(=O)NC2CN(C(C3CCOC(C(=O)O)C3)=O)C2)cc1 24350,Cc1ccc(S(=O)(=O)N2CCN(CC(=O)NC3CCCC3)CC2)nc1 24351,Cc1ncnc(C(N2CC3(C(=O)NOCCC(C)C)CC2CO3)=O)c1C 24352,C=CC1CCCCN1C(=O)Cn1cc(CNC(c2cc(C(C)=O)c[nH]2)=O)nn1 24353,c1(C(=O)NCC(C2CCCC2)NC(C2(COCC)CCC2)=O)ccc(C)cc1 24354,c1(C(N(C(C)C(=O)NC2CCOCC2OC)CC)=O)cnn2ccccc12 24355,N1(C(c2c(CC)con2)=O)CC(NC(C2CCC(C(F)(F)F)CC2)=O)C2(CC2)C1 24356,c1(N2CCC(NC)C2)nc(N(C)Cc2ccc(F)c(Cl)c2)c2cnn(C)c2n1 24357,n1(CCOC)cc(C(=O)NCC(C2CC2)NC(=O)CC2CCCCCC2)c(C)n1 24358,Cc1ccc2c(C(=O)NC3CCN(C(=O)C#CC4CC4)C(C)C3)n[nH]c2c1 24359,c1(C(N(C)CC2(CNC(c3cc(COC)on3)=O)CC2)=O)ccc(C)nc1OC 24360,c1(C(=O)NC2C(NC(C3(C#N)CCCO3)=O)C2)ccc(S(N)(=O)=O)s1 24361,N1(C(c2c(C)ncc(Cl)c2)=O)CC2(CCN(C(=O)C3=CCCCC3)CC2)CC1C 24362,N1(C(C(C)OCCC(C)C)=O)CCCN(C(c2cnc3c[nH]nc3c2)=O)C(C)C1 24363,C1(CC)CCOC1C(=O)NC1CC(NC(=O)CC2(O)CCCC2)C1 24364,N1(C(CC(C(C)C)O)=O)CCCCC12CC(NC(=O)COC1CCCOC1)C2 24365,C1(CC(=O)NC2CCN(C(=O)CC3CC4CC4C3)C23CC3)CCS(=O)(=O)CC1 24366,Cn1cc(C(=O)NC2C3(CC(NC(=O)CC45CCC(CC4)C5)C3)C2)ncc1=O 24367,C(=O)(CC(F)(F)F)OC.c12nsc(n1)CCN(C)CCOCCN(C)C2=O 24368,CC(N=c1[nH]c(N(C)CCC2CN(C)C2)nc2c1CCC2)c1nnc2n1CCC2 24369,C(=O)(C1OCCc2ccccc21)NCC1(CNC(c2cnns2)=O)CC12CCC2 24370,C1(CNC(c2cnc(CC(C)C)[nH]2)=O)CCC(CNC(C2CCN(C)C2)=O)CC1 24371,FC1(F)CCC1c1noc(C(C2=NOC3CC23)Cc2ccccc2Cl)n1 24372,C(=O)(C1CCc2c[nH]nc21)NC(C(NOCCCC#C)=O)c1cnn(C)c1 24373,C(C)(CCC(=O)NC1CC1CNC(c1cnc(-c2ccccc2)[nH]1)=O)OC 24374,C1(CNC(C2CC(C)OC2)=O)CC2(CCN(C(C3CC4CCC3CC4)=O)C2)CO1 24375,c1(NC(CC=C)CC=C)ccc(N(C)C)c(C#N)c1 24376,c1(C(N2C(CC)CN(C(C3(C)CC3)=O)CC2)=O)c(F)ccc(Br)c1Cl 24377,C1(NC(CN(C)C(N)=O)=O)CC2CN(C(=O)C(c3ccccc3)C3CC3)CC2C1 24378,C1(CNC(Cc2cc(C)[nH]n2)=O)(CO)CCN(C(c2sccc2C#N)=O)C1 24379,c1(C(N2CC3(CN(C(c4c(C)coc4C)=O)C3)C2)=O)cc(N)c(O)c(F)c1 24380,n1(COC)ncc2c(NC3CC(Cn4ccnc4)C3)ncnc12 24381,C(=O)(C1=NOC(C)C1)N1CCCC(C(C(=O)NCC(=C)Cl)C)C1 24382,C1(C(=O)NC(C)C(C)NC(c2cnoc2-c2ccoc2)=O)CCCC2(CC2)C1 24383,C=CC(CC)CC(=O)NCCOCCNC(=O)C=Cc1ccc(C)cc1 24384,n1(C(CC)C)ccc(=NC(=O)CC(CC(C)C)NC(C2C=CCCC2)=O)[nH]1 24385,N1(C(C(C)Cc2ccco2)=O)CCC(OC2(C(C3CC3)NC(N)=O)CC2)CC1 24386,N1(C(c2c(COC)cc[nH]2)=O)CC2CC(NC(c3cc(OC)no3)=O)CC(C2)C1 24387,N1(CCCNC(C(C)OC)=O)CCC(NC(=O)C(C)(F)F)C1 24388,C(=O)(C1CCCc2c[nH]nc21)NC1CCN(C(Cn2ncn(C)c2=O)=O)C1 24389,C(C)(CN=c1cc(COC)nc[nH]1)(C(C)C)NC(c1ccc(CC)cc1)=O 24390,C(C)(CSC)(C(=O)NC(c1cccnc1O)C)NC(C1CC(=C)C1)=O 24391,C12CCC(F)(C1)CNC2=O.c1(C2C(N(C(=O)C(C)C)CC)C2)ccc(Br)s1 24392,C(=O)(C(CC)(CC)c1ccccc1)NC(CCCC)CNC(=O)CCN(C)CC 24393,C1(C(=O)NCCN(C(=O)CN(C)Cc2ccccc2)C(C)C)CN(C)CC(C)O1 24394,C1(C(c2c(NCC(=O)NC(=O)NC(C)C)cccc2)=O)COC2(CCCCC2)O1 24395,Nc1cccc(C(N2CCN(C(c3ccn4ccsc34)=O)CC2C2CC2)=O)c1O 24396,C(=O)(C(F)CCCC)N1CC(C2N(C(CCC=CCC=C)=O)CCC2)(O)C1 24397,N1(C(C2C(C)(C)C2(F)F)=O)CCC(NC(c2ccnc(N(C)C)c2)=O)C12CCC2 24398,N(C(=NCCF)NC(C)CCN1CCCCCC1)CC1(CC)COC1 24399,C#CCCCCCCCNC(=O)C(CC#C)NC(=O)CNC(=O)CC 24400,C12(C(N(CCCN(C(C(C3CCCC3)OCC)=O)C)C)=O)CC(C3CC3)(C1)C2 24401,C1(C(NOC(C(C)C)CO)=O)COC(=O)N1C.C1(=O)C(Cn2ccnn2)N1 24402,C1(C(=O)NC2C(C=C)CN(C(=O)CC(C)(C)O)C2)CC2(C1)CC(F)(F)C2 24403,N1(C(CCC(C)OCC)=O)CCC(C2CCCN(C(=O)C(=O)C(C)CC)C2)CC1 24404,C12(C(=O)OCC)CC(CC3CCC3)(C1)OC2c1ccccc1.c12cnn(c1)C2 24405,c1(C(=O)NC2(CO)CN(C(CCc3scc(C)c3)=O)C2)ccc(Br)nc1C 24406,N1(C(c2n(C(C)C)cnc2)=O)CCCCC(N=c2ccc(C(F)(F)F)n[nH]2)C1 24407,C1(NC(c2cnc(CC)[nH]2)=O)(CNC(c2cc3c(s2)CCC3)=O)CC2CCC1C2 24408,c1(C(=O)NCCC2N(C(C(N3CCOCC3)C)=O)CCC2)cc2ccccn2n1 24409,C1(C(=O)NCC(C2CCC2)OCC)CC(O)CN1C(c1ncccc1Cl)=O 24410,C(=O)(C(CO)C(C)(C)C)N1CC(CCNC(=O)Cn2ccc(O)nc2=O)(OC)C1 24411,N1(C(CCCC#C)=O)CCC(C(=O)NCC2(O)CCC(C)C2)C12CCC2 24412,c1(CC(=O)NC(C2CCCN2C(=O)CCC2CC2)C)cn(C2CC2)cn1 24413,c1(NC(=O)CN2CCCC2C(F)(F)F)cc(Cl)ccc1Cl.C1(=O)NCCN1 24414,N1(C(C(COC)OC)=O)CC(CNC(c2cccc(-n3cccc3)c2)=O)CC1C 24415,Cn1cc(C=CC(=O)NC(c2cccnc2)C(=O)NC2CC3CC3C2)cn1 24416,N1(C(c2cnc(C)c(N)c2)=O)CCC2(CCCC2CNC(C2(Cl)CC2)=O)CC1 24417,c1(C(=O)NCC2C(CNC(C(C)(C)OC(C)C)=O)C2)cn2c(n1)CCCC2 24418,Cc1c(F)ccc(F)c1CN1CCN(C(c2csnn2)=O)CC1 24419,c1(OC)ccc2ccnc(C(C)NC(=O)C(=O)NC(c3c(C)noc3C)C)c2c1 24420,C(N=c1nc2c(ncn2C)c(NC2CC2c2c(Cl)cccc2Cl)[nH]1)c1c(C)occ1 24421,Fc1cc(CNCC2CCCC(C(F)(F)F)C2)ccc1Cl 24422,N1(C(c2ncc(CC3CC3)s2)C(=O)NCCOCC)CCOC(c2cccs2)C1 24423,C1(CNC(c2ccc(OCC)cc2)=O)CCC(C)CN1C(c1cccc(O)n1)=O 24424,C1(CCNC(c2c(C)ocn2)=O)CCCN(C(C2CCCOCC2)=O)C1 24425,c1(CSC)cccc(C(N2CCC2CNC(=O)C(C(C)C)NS(C)(=O)=O)=O)c1 24426,C1(C(N2CCOCC2CO)=O)CC12CCN(c1nccc(C(F)F)n1)C2 24427,C1(CC)(CC)CC(NC(C2CC2C2CC2)=O)CN1C(=O)CCCF 24428,C(C(=O)N1CCC(NC(=O)CCc2ccccn2)C1C)(C(C)C)SC 24429,c1(C(=O)NC(C)CCCNC(c2cn(C3CC3)cn2)=O)cccc2nc[nH]c12 24430,N1(C(C)(C)C)CC(C(N2CCC2CNC(C2(c3ccsc3)CC2)=O)=O)CC1=O 24431,Cc1ccc(C(N2CCC(NC(=O)CN3CSCCSC3)C2)=O)cc1OC(F)F 24432,N(C(=NCC(C)OC(C)(C)C)NCc1cccc(N2CCOCC2)c1)C1C(C)C1 24433,CCC(CC(=O)NC1CC=C(C(=O)NCCCC2CCC2)C1)C(F)F 24434,C1(CNC(CCC=C)=O)(NC(=O)C(O)Cc2cccc(Cl)c2)CCCCC1 24435,c1(C(N2CCC(NC(C(C=C)O)=O)C(O)C2)=O)c(C)cc(O)cc1C 24436,Cc1cc(C(N2CC3(NC(c4nnc(S)n4C)=O)CCC2CC3)=O)cc(N)c1O 24437,C1(C(N2CC(N(C(CCSCC)=O)C)C3(C2)CC3)=O)CCC2(CC1)CC(O)C2 24438,C(=O)(C1=NNC(=O)CC1)NC1C(NC(c2c(C)ccnc2O)=O)CCCC1 24439,CC1(C)CN(C(=O)C2=CCCCO2)CC1C(=O)NC1CC2C=CC1C2 24440,c1(OC)cccc(C(=O)NCC(C)CNC(c2cnc(CC(C)C)s2)=O)c1N 24441,c1(C(c2n(CC=C)nnn2)NCC2(OC)CCCC2)cncc(C(=C)C)c1 24442,C#Cc1ccc(C(=O)NC2CCN(C(C)=O)C2)nc1 24443,C(=O)(CC(C)C(C)(C)C)NCC1N(C(C(CC(=O)OC(C)(C)C)O)=O)CCC1 24444,c1(NC(C2C(C(N(CC#C)C)=O)C2)=O)cc(Br)cc(F)c1OC 24445,c1(C(=O)NCC2C(CNC(C(C)SCC)=O)C2)c[nH]c2c(C)c(C)ccc2c1=O 24446,Cc1c(C(=O)NCC2(CNC(=O)C(C)CS(C)=O)CCC2)ccc2c1CCC2 24447,c1(C(=O)NCC(C)NC(c2c(CC)scn2)=O)cccc(COC)c1 24448,c1(SC)nc(OC)cc(OC)n1.C1(N(C(=O)CN2CCCC2)CC)CC2CNC1C2 24449,CC1COCCCN1C(C1CC(O)CN1C(=O)Cn1cnnc1)=O 24450,c1(C(=O)NC2CN(C(C(C)SCC)=O)CC2C2CC2)c(C)[nH]cc([N+](=O)[O-])c1=O 24451,N1(C(C2C(NC(=O)Cc3ccccc3[N+](=O)[O-])C2)=O)CCc2cc(O)ccc2C1 24452,C1(C(=O)OC)C(F)(F)C12CC(C(=O)NC(C)(C)CNC(C1CCSC1)=O)C2 24453,c1(CC(=O)N(CC(CC)NC(C(C)SCC)=O)C)cccc2ncccc12 24454,Cc1n[nH]c(C)c1C(C)CC(=O)N1CCCC1CN(C)C 24455,C(=O)(N=S1(=O)CCNC(CNC(=O)OC(C)(C)C)C1)c1c(C)c2n(n1)CCCO2 24456,N1(C(COC(C)=O)=O)CC=C(C(C)(C)C(=O)N(C)CC2OCCC2(C)C)C1 24457,C1(CNC(c2cn(-c3nccs3)nn2)=O)CCN(C(c2ccoc2)=O)CC1 24458,C1(C(=O)OCCC2(CC3CC3)OCCO2)Cc2ccncc2C1 24459,C(CC(C(=O)NCCc1cccnc1C)NC(C1CCN(C)C1)=O)=CC 24460,C12(NC(C3OCCC(C)C3)=O)CC(CNc3cc(CC4CC4)ncn3)(C1)OC2C 24461,Cc1ccnc(C(N2CC3CC2(C(=O)NCC2CC(=O)NC(C)C2)C3)=O)c1F 24462,c1(OC)cc(CC(N2CCCC2NCCN2CCOCC2)=O)cc(F)c1OC 24463,c1(CNC(=N)NC(c2cccc(Cl)c2)C(F)F)ccccc1Br 24464,N1(C(C(C)NC(c2nc(C)oc2C)=O)=O)CCCC12CCCOC2 24465,c1(Nc2nc(C)c(C(=O)NCc3cncs3)s2)ncnc2c1ncn2C 24466,c1(CCCOC)cn(CC(N2CC(SC)C2)=O)nn1 24467,CC1CC(c2nnnn2CSc2ccccc2)(NCC2(SC)COC2)CS1 24468,N1(C(C2CC(C)(CC)C2)=O)CC=C(CC(=O)N2CC(F)(F)CC2CO)CC1 24469,N1(C(C(c2ccccc2F)C)=O)CCN(C(=O)CC=C(Cl)Cl)C2(CC2)C1 24470,N1(C(CC2CCC(=O)C2)=O)CC2CCC1CN2C(C1C2C=CSC12)=O 24471,C1(C(=O)NC(CNC(c2nc(C)sc2)=O)(C)Cn2cccn2)CCC(O)CN1C 24472,Cc1nc2ccc(-c3cncnc3C(=O)NCc3cccnc3Br)cc2[nH]1 24473,N1(CCNC(C2(F)CN(CC)CC23CCC3)=O)CCc2ccccc2C1 24474,C1(CNC(C)C(=O)Nc2cccc([N+](=O)[O-])c2)NCCC12CCCCC2 24475,Cc1csc2c(NC3CCC(NC(=O)CC4CCC(C(N)=O)O4)CC3)ncnc12 24476,c1(C(CNC(c2ccnc(C)n2)=O)NC(C2CCCN2C)=O)cc(F)cc(Cl)c1 24477,c1(SC)ccc(-c2nc(C3(c4cncc(F)c4)CC3)no2)cc1 24478,C(=O)(CC(C)(C)C(F)F)N(C1CCN(C(c2cnn(C3CCC3)c2)=O)C1)C 24479,C(CC(CC)C(=O)N1CCCC(OCC(=O)N(CCC(C)C)CCO)C1)=CC 24480,N=c1[nH]n(CC(=O)NC2CC(NC(C3C4CNC(=O)C34)=O)C(O)C2)cc1Br 24481,c1(C(N2CCC(NC(C3(COC)CC3)=O)C2)=O)c(C)nc2sc(C)cn12 24482,C1(NC(c2sc(C)c(O)n2)=O)CCCC2CN(C(=O)C=Cc3cccs3)CC12 24483,C1(c2ccccc2)(C(=O)NCC(C)NC(c2cc(C(=O)C(C)C)c[nH]2)=O)CCCO1 24484,c1(C(N(CCNC(c2cncc(CO)c2)=O)CC2CC2)=O)cnc2n1CCS2 24485,CC(C)C(C(=O)N1CCCC(C(=O)N(CCC(=O)O)CCO)C1)c1ccncc1 24486,CC1COc2c(C(=O)NC3CN(C(c4ccc5c(c4)nnn5C)=O)C3)cnn2C1 24487,Cc1cc(C(=O)N(CCNC(=O)CCC2CCCN(C)C2)C2CC2)cn(C)c1=O 24488,n1(CCC)nc(C)cc1C(=O)N(CC(C)CNC(C1(c2oncc2C)CC1)=O)C 24489,c1(C(=O)NC(C2CCCCN(C(=O)C(F)=CC3CC3)C2)C)cnc(N)c(Cl)c1 24490,Cc1ccc(-c2ocnc2C(=O)Nc2cncs2)s1 24491,C1(CC(=O)NC(C(C)NC(CNS(CC)(=O)=O)=O)(C)C)COCCN1C 24492,CN=c1[nH]ccc(C(N2CCC(C)(C)C2CNC(C2CCC(C)CC2)=O)=O)c1N 24493,c1(COC)ccc(C(=O)NC2CN(C(C3CC(N4CCCCC4)C3)=O)C2)s1 24494,CCCCC(CNC(=O)Cn1cc(CN(C)C)nn1)NC(C1CC(F)(CO)C1)=O 24495,C#CC1CCCC(NC(C)C(N)=O)C1 24496,c1(C(N(CCNC(C2C(C)C2(F)F)=O)C2CC2)=O)cccc(C2CNC(=O)C2)c1 24497,c1(C(=O)NC2(C)CN(C(C3CCN(CC#C)CC3)=O)C2)cnc2nncn2c1C 24498,N1(C(C2CCCC(OC)C2)=O)CC2(CCN(C(=O)C(C)NC=O)C2)C1 24499,N1(C(C2CC(C#C)(O)C2)=O)CCC2(CC1)CN(C(=O)Cc1ccco1)CC(C)O2 24500,c1(NC2CCN(CC=C)C2=O)ccc(OCCN(C)C)c(Br)c1.C(COC)O 24501,C1(C(=O)NC2CC(CC)(CC)C2)CN(C(=O)CC(C)SC)CC1N=[N+]=[N-] 24502,c1(NC(c2cn(C3CCSC3)nn2)=O)ccc2c(O)ncnc2c1 24503,C(=O)(C(C)C(F)(F)C(F)F)NC1(CCCNC(c2cc(CC)c(F)cc2)=O)CC1 24504,Cn1c(C(=O)NCC2CCCC(NC(=O)C=C3CCC3)C2)cc2ccsc12 24505,c1(C(N2CCC(N(C(CCC=C)=O)CCO)C2)=O)cc2n(n1)CC1(CC1)C2 24506,n1(CC(=O)NCC(C)(CO)NC(C2CSCC(=O)N2)=O)sc2ccccc2c1=O 24507,CC1CN(C)CC1NC(C1CCN(C(c2ccoc2Cl)=O)C1C)=O 24508,c1(C(N2C(C(=O)O)C3(C2)CCC3)=O)ccc2nnn(C(C)(C)C)c2c1 24509,CC1CCNC(=O)C1NC(c1c(CNC(c2cc(CO)ccn2)=O)nnn1C)=O 24510,C(CC)(CCCC(=O)NCc1ccc(O)cc1)NC(C1(OCC)CCCC1)=O 24511,CCCCC(CO)NC(=O)CC1CC(NC(=O)CN2CCNC(=O)C2)C1(C)C 24512,C1(C(=O)NCCCN(CC)CC)(NC(=O)CCSC)CCOC1 24513,Cc1cc(Cl)c(C(=O)NCC2(C)CCCN2C(=O)CSCc2ccncc2)cn1 24514,c1(CC(C)NC(C(N2CC(CC)C(C(F)(F)F)C2)=O)=O)cc(C(F)(F)F)ncn1 24515,c1(NC(CC)CCOCC)[nH]c(=NCC(C2CCC2)N(C)C)nc2c1ncn2C 24516,CC1CCCC(N=c2nc(N3Cc4ccc(F)cc4C3)c3c([nH]2)CCOC3)C1 24517,C1(COC)(NC(c2cocc2C)=O)CCN(C(=O)C(C#N)C(C)C)CC1 24518,c1(C(=O)NC(CC(C)NC(CCOCC(C)C)=O)C)ccc(F)cn1 24519,c1(-n2c(C(C3CCCCCC3)SCC)nnn2)csc2c1N2.C1(CC)(SC)CC1 24520,CCC(C)C(C(=O)NC(C)CCSC)N(C)C(c1cccc(C)c1C)=O 24521,C1(C(N2C(CNC(=O)CN3CSCC3=O)CCCC2)=O)CCC=CCCC1 24522,N1(C(c2cccc(CC)c2)C(=O)NC)Cc2nccn2CC(C(=O)OC)C1 24523,C(=O)(CCC(CF)CF)N1CC(CC(C(=O)NCCC2CC(O)C2)F)C1 24524,C1(NC(c2c(C)scc2)=O)CN(C(C2CCC2C(C)(C)C)=O)C2(CCC2)C1 24525,C(CS(=O)(=O)CC(=O)NC(C)(C)CC(F)C(=O)NCc1nnnn1C)OC 24526,C1(C(=O)NC2COCC2F)(COC)CCCNCC1 24527,c1(CC(=O)NC2(C(=O)OC)CCC2COC)ccc(OC(C)C)cc1Cl 24528,Cc1c[nH]c(C#N)nc1=NC(CO)c1cccc(F)c1 24529,Cc1ncc2n1CCC(C(=O)NCCN(C(=O)CCc1ccc(CO)cc1)C)C2 24530,C1(NC(C(CCCCC)O)=O)CCN(C(c2cccnc2OC)=O)CC12CCC2 24531,c1(C(C(=O)NC(C)CN(C(=O)CSC(=N)N)C)C)cccc(O)c1 24532,C(C(CC(C)C)C(=O)N(C)Cc1ccncc1)NC(C(CCC)CC)=O 24533,Cc1cccc(Br)c1CN1CCCN(c2cc(C#N)ncn2)CC1 24534,N1(C(C(CCF)NC(C2CCC(=O)OCC2)=O)=O)CCC2(CCC2)CC1 24535,c1(CCCC(=O)NC(CNC(C2CCOC2)=O)C2CCC2)ccccc1Cl 24536,C(=O)(C1=C(F)CN(C(=O)CN2CCC(OC)C2)CC1)N1CC(CC)OCCC1 24537,C(=O)(CC(C)(C)C1CCCCC1)NCC(CCOC)NC(=O)C(F)OC 24538,C1(C(=O)NCCC2CCC(CO)C2)CC(c2cccc(Cl)c2F)=NO1 24539,N1(C(CC(C(C)C)NC(CC(=O)OCC)=O)=O)CCn2ccnc2C1C 24540,c1(C(=O)NCC(C2CCC2)NC(CC2C(C)(C)C2)=O)cocc1Br 24541,N1(C(c2ccc(C)cc2)=O)CCC(NC(C2CCC(CO)CC2)=O)C(F)C1 24542,C=CC1(CC(=O)NCC(C2CCN(C(C3CCC(=O)O3)=O)CC2)F)CCCCC1 24543,n1(C(C=C)C)nc(-c2ccoc2)nc1-c1cccc(-c2ccncc2)n1 24544,C(=O)(C(F)C(C)CNC(c1ccc(F)c(O)c1)=O)N1C(COC)C=CC1 24545,C(=O)(C(C)(C)C(=O)Nc1cc(F)cc(F)c1)NCC1(O)CCN(C(C=CC)=O)C1 24546,Cc1ccc(F)cc1C(N1CC2CC1C2NC(=O)CC1(O)CCCCCC1)=O 24547,C(=O)(C(F)C(F)(F)F)NCCCCNC(c1cccc(SC(F)(F)F)c1)=O 24548,Cc1c(Br)cnn1CC(=O)N(CC(C)NC(=O)C(F)=C1CCC1)C 24549,CC(C)CS(=O)(=O)CCC(=O)NCC(C)CN(C(=O)CP(C)(C)=O)C 24550,CC1(C)CC(CC(N2CC(CC(F)F)C2)=O)N(C(=O)OC(C)(C)C)C1 24551,C1(C(=O)NC(C)COCC2CC2)CC(F)(F)CN1C(=O)CCC1CC1 24552,CCCCCC(CC)C(=O)NC1C2CCC1N(C(=O)C=Cc1cccc(Cl)c1)C2 24553,c1(NC2CCCN(C(C(CCC)(C)C)=O)CC2)ncc([N+](=O)[O-])cn1 24554,N1(C(C=C(C)CNC(=O)CC2C=CC(N(C)C)C2)=O)CC=CC12CCCCC2 24555,N1(C(c2cc(F)cc(C)c2N)=O)CCOC2(C1)CN(C(=O)OC(C)(C)C)C2 24556,Cc1cc(CN2CCCC(C(N(CCC#N)C(C)C)=O)C2)nn1C 24557,N1(CC(=O)N(C)CCO)CCCC(N(C)C(c2coc(Cn3cccn3)c2)=O)C1 24558,N1(C(C(n2cc(CNC(=O)OC)nn2)C)=O)Cc2ccc(F)cc2CC1C 24559,C1(C(=O)NCCN(C(C(CC=C)C(C)C)=O)C)CCOC2(CCOCC2)C1 24560,c1(C(=O)NC2CC(CNC(Cc3nnc(C)n3C)=O)CC2O)c(C)ncnc1O 24561,c1(-c2c(C(=O)Nc3ccc(F)cc3O)n[nH]c2)ccc(S(=O)(=O)N2CCCC2)cc1 24562,C1(NS(CC=C)(=O)=O)CC2(C1)CN(C(c1cc(I)ccc1O)=O)C2 24563,C1(CC(=O)NCCCC(C)NC(Cc2cccc(OC)c2)=O)CCCC(C#N)C1 24564,CC1(C)CN(C(=O)CCn2ccnc2)CC(C)(C)C1NC(c1ccc[nH]1)=O 24565,C1(NC(=O)CN2CCOCC2)CCN(C(=O)CCc2cn[nH]c2)CC1F 24566,C(=O)(CC(O)CC(C)C)N1C(CCC)CN(C(=O)CCC(C)(F)F)CC1 24567,c1(OC)cc(F)c(C(N2CCC3(C2)CN(C(C2C=CCCC2)=O)C3)=O)cc1F 24568,C1(c2c(C)cc(C(F)(F)F)s2)NC(=S)N(c2cccc(F)c2)C2=C1C(=O)NC2C 24569,C(C(=O)N1OC2CCC1CC2)N(C(=O)C(F)C1CCCC1)CCOC 24570,C1(N2C(c3nc(C)nc(=N)[nH]3)CCC2)CCC2(CC1)OCCO2 24571,C(C)(CCCNC(=O)C(C)Sc1nncn1C)NC(C1(CCC=C)CC1)=O 24572,c1(C(c2nnnn2C2COC2)NCC2(CCC)CC2)ccc(CC)cc1F 24573,Cc1ccc(C(F)(F)C(N2CC(NC(c3cnc(C)o3)=O)C(C)C2)=O)cc1 24574,C1(CNC(c2c(CC)nc(C)o2)=O)CN(C(=O)C(CCSC)OC)C2(CCC2)C1 24575,C=C=C(C)CC(=O)N1CCC(O)(C(C)NC(=O)Cc2cnn(C)c2C)C1 24576,CCCC(C)CC(=O)N1CC(NC(=O)CCCc2ccccc2)C(O)C1 24577,N1(C(c2cccc(CC)c2)=O)CCN2C(=O)C(NC(=O)Cc3cncs3)CC2C1 24578,c1(C(C(C)NC(=O)C(F)(F)CO)NCC2=CCN(C(C=NOC)=O)CC2)ccc(=O)oc1 24579,N1(c2nnc(C(C)(C)OC)o2)CCC(NC(c2ccnc(SC)c2)=O)C(C)(C)C1 24580,C(=O)(C(O)C(C)CC)NCC1(CCNC(CNS(CCCC)(=O)=O)=O)CC1 24581,N1(C(C(CC)NC(N)=O)=O)CC2CC2C1C(=O)NCc1nccn1C(C)C 24582,c1(NC(CC(C)F)=O)sc2c(c1C(=O)Nc1ccccc1)CCCC2 24583,c1(OC2(C(=O)NCC(c3cccc(F)c3)C)CC2)ccc(Cl)cc1 24584,N1(C(=O)Cc2cnc3cccnn23)CCc2c(Cl)ccc(Br)c2C1 24585,N#Cc1c(N2CCC(F)(CNC(C34CC=CCN3CCC4)=O)CC2)cccc1F 24586,c1(C(N2CCC(O)(CCNC(C(C)C)=O)C2)=O)nc(N(C)C)nc(=N)[nH]1 24587,Fc1cc(Cl)cnc1-c1nnc(N2CC3CN(CC(F)(F)F)C3C2)n1C 24588,C(=O)(C(C)(CNC(=O)CCc1nc(O)n[nH]1)CC)NCC(N(OCC)C)=O 24589,C(=O)(C(C)C(C)CC)N(CC(CNC(c1nc(C(=O)NCC=C)sc1)=O)(C)C)C 24590,c1(C(=O)NCC2OCCCN(C(COCCC#C)=O)C2)cccc2nc(O)[nH]c12 24591,N1(C(CC(=O)NC)=O)CCC2(CC1)CCN(C(c1ccc(CC(C)C)cc1)=O)C2 24592,c1(C(=O)NC23CCN(C(=O)Cc4nc[nH]n4)CC2C3)ccc2ccsc2c1 24593,N1(C(CCCOC)=O)CC2CCCC(N(C(=O)CC3CCCC34CC4)C)C2C1 24594,CC#CCCCC(=O)NCCOCCCN(C(=O)C(c1ccn(C)n1)C)C 24595,C(=O)(C(CCC(C)C)NC(c1ccnn1CCC)=O)NC(C=C)C1CCC1 24596,CCC(O)C(C)C(=O)N1CCCC1CN(C)C(C1CN(C2CCOC2)C1)=O 24597,c1(OC)ccc2nc(N3CC(CO)(NC(c4c[nH]nc4C)=O)C3)sc2c1 24598,N1(C(c2c(SC)cn(C)n2)=O)CC(C)(CNC(=O)C(F)(F)C2CC2)CC1(C)C 24599,N1(C(C2=CC(C)(C)C2)=O)CC2(C1)CN(C(c1cccc(CCO)c1)=O)CC2CO 24600,CCC(C)(CO)C(=O)NC1CC(CNC(=O)C(C(C)C)n2cnc(C)c2)C1 24601,C1(CNC(=O)CCC2CCN(C(c3ccc(CO)o3)=O)C2)CCC=CCCC1 24602,c1(OC)cccnc1C(=O)N(C(CNC(=O)CCSc1nnnn1C)C1CC1)C 24603,N1(C(C2CCN(C)C2=O)=O)C(CC(=O)NC(c2ccsc2)(C)C)C2CCCC12 24604,C(C(C)(O)CC)NC(C1(CCNC(CC2CC(=C)C2)=O)CCC1)=O 24605,CC1CCSCCN1C(c1cn(CC(F)F)cn1)C(=O)NC1CC(F)(F)C1 24606,C(=O)(C(C)(C)C(C)(C)C)NCC1(C(=O)NCc2cccc(C)c2O)CC1 24607,Cc1ncnc(C)c1CC(N1CCC(F)C(NC(C2CCC3CC2CO3)=O)C1)=O 24608,C1(C(=O)NC(CN(C)C)CCO)(CC)CCN(C(c2ccon2)=O)C1 24609,N1(C(C2C(C)CCN2C(=O)CCC(N)=O)=O)CC2(CCCCCC2)C1 24610,c1(C(N(c2cc3ncnn3cn2)C23CC(N)(C2)C3)=O)[nH]nc2ncccc12 24611,c1(-c2c(C)ccs2)ccc2c(c1NC(=O)Cn1cccn1)OCO2 24612,C1(NC(C(CC2CC2)OC)=O)CC2CC(C1)CN(C(=O)Cc1ccc(O)cc1)C2 24613,N1(C(C2CC(n3cc(C4(C5CC5)CCCCC4)nn3)C2)=O)CC2CCCC(C2)C1 24614,CCC(F)(F)C(=O)N1CCOC(CCNC(c2cnnn2C2CCOCC2)=O)C1 24615,N1(C(C(C)n2cnnn2)=O)CCOC2(CCCN(C(c3cc(Cl)ncn3)=O)C2)C1 24616,c1(OC(C(=O)N(CCN(C(=O)CC2CC3CC3C2)C(C)C)C)C)cccnc1 24617,N1(C(COCCCOC)=O)CCC(NC(c2cc3c[nH]nc3s2)=O)C(O)C1 24618,Cc1ccccc1C(C)C(N1CCC(CN(c2ncc[nH]2)C)CC1)=O 24619,C(=O)(C1=NNC(C(F)(F)F)C1)N(CCCNC(C(C)SCCCC)=O)CCO 24620,N1(C(C=C(C)Cl)=O)CC(CNC(C23CCC(C)(CC2)CO3)=O)CC12CCOCC2 24621,CCC(CN(C)C)C(=O)NC(C)CCCNC(=O)C(C)(C)N(C)C 24622,C1(C(N2CC(OC)(CNC(=O)C(C)(C)c3ccccn3)C2)=O)CC1C1CCCC1 24623,C(CCC(=O)N1CC2(CCC2O)C1)(C(C)C)NC(c1cccc(CC)n1)=O 24624,c1(C(=O)NCC(CC)(CC)NC(=O)C(O)CN(C)C)nc2n(c1Cl)CCCC2 24625,N1(CC(N2CCC(CNC(C(c3ccccn3)C)=O)C2)=O)CCC(=O)CC1 24626,CC1CC(CC(N2CCC(C3(C)N=N3)C2)=O)CN1C(=O)C=CC(=O)NC1CC1 24627,c1(C(N2CCC(N(C(=O)CC3CCOC3)CCC)C2)=O)cccc2c1OCCO2 24628,c1(CN(C(=O)Cc2ccnn2C2CCOCC2)C)cccc2c1OC(F)(F)O2 24629,N1(C(c2c(CC)c[nH]n2)=O)CC2CCCN(C(=O)C(C)O)C2C1 24630,N1(C(CN(C)C)=O)CCn2ncc(C(=O)NCc3ccc4cc[nH]c4n3)c2C1 24631,C1(CC2(NC(COCCC#C)=O)CC2)CCN(C(=O)CC(C)C)CC1 24632,c1(C(C(=O)NCC(C)NC(C2CC2[N+](=O)[O-])=O)C)cncc(F)c1 24633,Cc1cc(C(=O)NC(c2ccccc2)C(C)NC(=O)CCC2CC2)nc(O)n1 24634,N1(CC(=O)N(S(CC2CCC(C)O2)(=O)=O)CCO)CC2(CCCC2)C1 24635,N1(C(C(C)(C2(C)CC2)OC)=O)CCCC(F)(C(=O)Nc2cn(C)nc2C#N)C1 24636,C1(C(=O)N(CC)CC)(OC)CCN(C(c2ccc(C)o2)C)CC1.CCO 24637,N1(C(C(C)c2ccco2)=O)CCCN(C(c2ccc(Br)s2)=O)CC1CO 24638,C1(NC(CCC=C(C)C)=O)CC2CC(NC(=O)CSC(F)(F)F)CC2C1 24639,Cc1cc(C(=O)NCCC2(C)CCN(C(c3nnn(C)c3N)=O)CC2)ncc1Cl 24640,C(C1CCN(C(C2CCCC(=O)N2C)=O)CC1)=CC(=O)NCc1c(CC)nccn1 24641,C1(N(C)C)CCC(N=c2ccnc(NCc3ccc(C#N)cc3)[nH]2)CC1 24642,Cc1nc(-c2ccn(C)n2)sc1CC(N1CC(NC(=O)C(C)C(C)C)C1)=O 24643,C(=O)(C(CCF)NC(=O)CCOC1COC1)NC(CCC)CO.O.O=CC 24644,C1(CC(=O)NC(C)(CNC(C2(O)CC(F)(F)C2)=O)C2CC2)CCCOCC1 24645,c1(C(=O)NCC2CCC(NC(c3cc(C)on3)=O)C2)cc2c(C)cc(F)cc2[nH]1 24646,N1(CC)CCOC(C(N2CCOC(CNC(=O)CC(F)(F)Br)C2)=O)C1 24647,CCN=C(NCC(CO)C(C)(C)C)N1CCC(COc2cccc(C)n2)CC1 24648,C(=O)(CC(C(F)F)c1ccccc1)OCc1ncc(N(C)C)nc1 24649,Cc1oc(C)c(C(=O)NCCC(O)CNC(c2cnn(C(C)(C)C)c2C)=O)c1C 24650,Cc1ccc(F)c(CC(C)NC(c2cccc3[nH]ncc23)=O)c1F 24651,N1(C(C2CC(N(C)C)C2)=O)CCC(NC(C2CCC(F)(F)CC2)=O)C(O)C1 24652,N1(C(CN(CCC)C)=O)CC(C(=O)NCc2ccnc(Cl)c2)C2(CCC2)C1 24653,C1(C(=O)NC2CC(CNC(c3c(OC)nccc3)=O)CC2O)CCCC(=O)N1C 24654,C(C)(C)(CCC(=O)N(C)Cc1ccon1)NC(C(CC)NC(N)=O)=O 24655,Cc1nccc(C(=O)NCCOC2CCN(C(C3CCC(C)NC3=O)=O)C2)c1C 24656,c1(C(=O)NCC2C(C)CN(C(c3cccc(C(N)=O)c3)=O)C2)c(F)ccnc1F 24657,N1(C(C(CC)NC(c2cc(C)ns2)=O)=O)CCOC(C)CC1 24658,C1(CNC(CSCC)=O)CCC(C)CN1C(c1ccnn1CC(C)C)=O 24659,C1(C(C)(C)NC(=O)C=C2CC2)CCCN(C(c2ccc(C(N)=O)cn2)=O)C1 24660,C1(NC(=O)C(O)C2CCCC2)CC2CN(C(c3occc3C3CC3)=O)CC2C1 24661,C(C)(C(=O)NC1(C(=O)NCCC(C)N(C)C)CCC1)OCCC#C 24662,c1(C(=O)NCC(CC)NC(=O)C(Cc2ccccc2)n2cccc2)cscc1C 24663,C(C1CC(=O)Nc2ccccc21)NC(=NCC)NCC1COC(C)(C)O1 24664,Cc1ccc(C(=O)NC2CCN(C(=O)CC3(C)OCCO3)C2)cc1[N+](=O)[O-] 24665,C12(C(N(CC(CN(C(=O)C(=O)Cc3ccccc3)C)O)C)=O)CCOC(C)(C1)C2 24666,Cc1c(NCC2CC(Oc3ccc(F)cc3)C2)ncnc1N(C)CCC(C)(C)C 24667,N1(C(CC=C=C)=O)Cc2ccnn2CC(NC(=O)C(C)CCOC)C1 24668,C(=O)(C(C)(C(F)(F)F)c1ccccc1)N(CC(C)NC(=O)CC(C)(F)F)CC 24669,N1(c2n(CC(C)(C)C(F)F)nnn2)Cc2ccccc2C(c2cccs2)C1 24670,CC(C)C(C)(C)C(=O)NCC(CC1CCCC1)C(=O)N(C1CCCN(C)C1)C 24671,c1(C(=O)NC2(c3cn(C(CC=C)CC=C)nn3)CCC2)ccc2occc2c1 24672,c1(N2CC(CC(C)C)OCC2)nc(=NCC2CCC2)[nH]c2ccc(Cl)cc12 24673,N1(C(C(C(C)C)NC(=O)OC)=O)CCCC(O)(CNC(C2SCCS2)=O)CC1 24674,C1(CC2(OC(=O)C3CC3)CCC2)CCCN(C(=O)CN2CCCC2=O)C1 24675,Cc1occc1C(=O)NC1CC(C)(NC(c2ccon2)=O)C1 24676,CC1(C)CN(C(c2cnc(Br)s2)C(=O)NCc2ccccc2Cl)C1C1CC1 24677,C1(CCN(C(CC(C)F)=O)C)CCN(C(=O)CC2CCC23CCC3)CC1 24678,c1(NC(C2N(C(c3cnc(C)nc3C)=O)C3C(C2)C3)=O)ccc(O)c([N+](=O)[O-])c1 24679,c1(C(=O)NCCC(C)NC(c2cc[nH]n2)=O)cc2c(s1)CCCNC2=O 24680,c1(C(N(C(C)CNC(=O)C(C)(O)CC)CC)=O)ccnc(CO)c1 24681,c1(NC(C)C)ccc(C(=O)N(C)CC2CCCN2C(c2ncc(Cl)n2C)=O)cc1 24682,c1(C(=O)NCC2C(NC(=O)Cc3ccc(F)c(F)c3)CC2)cc2c(s1)CCCC2 24683,C1(F)(c2cn(CCC(C)C)nn2)CCN(C(C2CC3(CC3)CO2)=O)C1 24684,C1(C(N2CC(SCC)C2)=O)C(NC(=O)COCC2CCCO2)C1(C)C 24685,N(C(=NCCC(C)=O)NCc1ccc(Cl)cc1F)C1CCC(C#C)CC1 24686,Cc1cn2c(n1)CC(C(N1CC(C)(NC(C3CC34CCOCC4)=O)C1)=O)C2 24687,C(=O)(CCCC(F)(F)F)NCC1CN(C(C2C(C)(C)C(F)(F)C2)=O)CC12CC2 24688,c1(N(CC2(CCC=C)CC2)CC2CCC2)nnn(C)c1N 24689,N1(C(c2nc(C(C)N)sc2)=O)CCOCC1CN(C)C(c1cnn(C)n1)=O 24690,C1(C(N2CCCCC2CNC(=O)C(C)NC(=O)NC2CC2)=O)(SC)CCCCC1 24691,N1(C(C=CC)=O)CC2CC1CN2C(=O)CC1NC(=O)CNC1=O 24692,Cn1cc2c(n1)C(O)CC1(CCN(C(N3CCC4(CCC4(CCOC)C)C3)=O)CC1)O2 24693,c1(C(=O)NC2CCCN(C(C3C(C)C3)=O)C2)ccc2c(c1)CC2 24694,c1(C(=O)NCc2ccc(CNC(C3(C)C=CCCC3)=O)cc2)ccc2c(c1)CC2 24695,C1(NC(C(C)NC(CC)=O)=O)CC2(C1)CN(C(c1cc3ccsc3s1)=O)C2 24696,C1(CC(C(=O)NCCOC)N2CCCC2CCOC(C)=O)CCC(C)(C)CC1 24697,N1(C(CC(COC)C)=O)CCCC2CN(C(c3ncc(C)cc3C)=O)CCC12 24698,N1(C(c2c(C)nc(CC)s2)=O)CCC2(NC(C3(NC(C)=O)CCCC3)=O)CC2C1 24699,c1(CC)cccc(C(=O)NC(C2CCN(C(=O)CS(=O)(=O)N(C)C)C2)C)c1O 24700,N1(C(Cc2c(C)cco2)=O)CCCC12CCN(C(C1(CC(F)(F)F)CC1)=O)C2 24701,c1(CC(=O)NCCN(C(c2cnn(-c3ccccn3)c2)=O)CC)ncncc1Cl 24702,N1(CC(C)O)CCC(NC(=O)CCCc2ccc(Cl)cc2)C(C)C1 24703,C1(C(N2CC(OCC)(CNC(=O)CCS(C)=O)C2)=O)CCCCC1(F)F 24704,c1(-c2cn(C3CC(NC(=O)Cn4cccnc4=O)C3)nn2)cccc(Cl)c1Cl 24705,C#CCCC(O)C(=O)N(C1CCN(C(=O)COc2ccsc2)C1)CCC 24706,N1(C(C(CC)N(CC)CC)=O)CCCN(C(=O)C(COC)C(F)(F)F)CC1C 24707,N1(C(CC(C)(F)F)=O)CC2CC(NC(c3ccnc(C(F)F)c3)=O)CC1C2 24708,C1(NC(C(C)=C2CC2)=O)CC2(C1)CN(C(C1(C(C)C)CC1)=O)C2 24709,CC(C)CC(C)C(=O)NCCN1CCN(C(c2csnn2)C)CC1 24710,C1(C)(C(N(CC(CC)NC(c2ccc(CN(C)CC)o2)=O)CC)=O)CCNC1=O 24711,N1(C(C2C(CC)CCO2)=O)CCN(C(c2c(C)cc(C)nc2S)=O)CC(O)C1 24712,N1(CCOc2ccc(OC)cc2)C=NC2=NC(C(c3ncsc3Br)C)C(=O)N12 24713,CCC(CC(=O)NCCN(C(C1CCC=CCC1)=O)C1CC1)C1CC1 24714,N1(C(CCSC)=O)CC(CNC(c2cc(I)c[nH]2)=O)C2CC12 24715,N1(C(C(C2CC2)SC)=O)CC(NC(c2ccc(F)c(Br)c2)=O)CC(F)C1 24716,C(=O)(C1=CCS(=O)(=O)C1)N1CCC(NC(=O)COCC2CCOC2)C1 24717,Cc1c(C(=O)NCCC2(O)CN(C(=O)C(c3ccccn3)C)C2)cccc1N 24718,N1(Cc2cc(C)ncn2)CCC2(CC1)CN(C(c1sccc1F)=O)CCO2 24719,C1(CCC(C(=O)NC)N2CCC(OCC(N)=O)CC2)CCC(F)(F)CC1 24720,CCC(CC(=O)NCC=CC(N1CCC(OC(C)C)CC1)=O)SC 24721,n1(C(C)(C)C)ncc(C(=O)NC2(CNC(=O)CC3C=CCC3)CCC2)c1N 24722,C1(CC(=O)NCCC(C)N(C(C(CCSC)O)=O)C)CCCCCCC1 24723,c1(C(=O)NCC)ccc(C(N2CC(OCCNC(c3cnc(Cl)s3)=O)C2)=O)s1 24724,c1(N(CCN(C(CC2(CC)CC2)=O)C)C2CC2)cc(C(F)(F)F)nc(Cl)n1 24725,N1(C(C(C)NC(N)=O)=O)CCN(C(=O)Cc2csnn2)CC12CC2 24726,c1(CC)nccnc1C(=O)NC(C)CCNC(c1ccccn1)=O 24727,C(=O)(CC(CC=C)NC(=O)CC1(O)CCC1)NC1(CC=C)CC=CC1 24728,c1(C(=O)NCCCCC2(NC(C(C)n3ccnc3)=O)CC2)cc2cccnc2[nH]1 24729,C1(CS(C)(=O)=O)CCN(S(=O)(=O)CC2CCC(C3CC3)O2)C1 24730,N12CCC(C)(CC1)NC2=O.c12nocc1C2C.n1(C2(C(=O)NF)CC2)ccnn1 24731,C12(C(N3C(C)(CC)CC3)=O)CC(C)(CN1C(=O)CCCn1cccc1)C2 24732,CC(F)(F)CCC(=O)NN1CCCC1C(=O)NCC1(CF)CCC1 24733,c1(C(N2CCCC(NC(C3CS(=O)(=O)C3)=O)CC2)=O)cc(O)c2ccccc2c1 24734,C1(C(=O)NC2CCC(OC)C2)CCN(C(=O)CCc2cnco2)C1C 24735,C1(C(N(CCCC)CCOC)=O)C=CCN(C(C2(OC)CCOCC2)=O)C1 24736,C1(C(=O)NCC(C)N(C2CCN(CC(F)(F)F)C2=O)C)CC(=O)N(C)C1 24737,O=S(=O)(c1cccc(F)c1)NCC1CCCN(Cc2cccc(I)c2F)C1 24738,c1(OCC(=O)NC2C(NC(CC=C=C)=O)C2)ccc(-n2nc(C)cc2C)nc1 24739,CC1CCC(CC(=O)NCC#CC(=O)NCc2ncccc2F)CC1 24740,c1(C(N2CCN(C(CC(C=C)C)=O)C(CCOC)C2)=O)c[nH]c2nc(F)ccc12 24741,c1(C(=O)NC2CCN(C(c3cccc4nccn34)=O)C2)ccc2c(c1)COCO2 24742,C1(C(=O)NC(CN(C(CS(=O)(=O)NC)=O)C)C)CCCC(=O)N1C 24743,C12(CNC(C(C=C=C)C)=O)CN(C(=O)COCCCCC)CC1CS(=O)(=O)C2 24744,Cc1c(-c2ncc(Cl)cc2CN2CCCC3CCCCC23)cccc1S(C)(=O)=O 24745,N1(C(C#CC)=O)CCC(CN(C(=O)CC(c2ccc(C(C)C)cc2)C)C)CC1 24746,C(C(=O)NCC1CC(C)N(C(=O)CCn2cnnn2)C1)(C(C)C)OCC 24747,Cc1ccc(CC(=O)NC2(C)CCN(C(C3COCCC3(F)F)=O)CC2)c(C)c1 24748,c1(C(N2CC(O)(C(C(=O)N(CC(F)F)CCC)F)C2)=O)ccn(CC)c1C 24749,C(CCC(C(=O)Nc1ccccc1)N1CCC(c2nnc(C)s2)CC1)OCC=C 24750,c1(OC)ccccc1C(N1CC2CC1C2NC(c1cnn(C2CCC2)c1)=O)=O 24751,c1(C(N(CCCNC(C2CC3(CC3)CO2)=O)CC)=O)cc(Cl)c(N)cc1F 24752,n1(CCC(N2CC(C(N(CC#N)CC#N)=O)C(O)CC2)=O)ccc2ccccc12 24753,N1(C(C2(C)CC2)=O)CC2(CC(NC(=O)C(c3ccc(Br)cc3)(C)C)C2)C1 24754,N1(C(CSC)=O)CCCCC1C1CCCN(Cc2nc(C(C)(C)C)no2)C1 24755,C1(C2CCN(C)CC2)(C(=O)NC2C(OC)CN(C(C3CCCC3(F)F)=O)C2)CC1 24756,C(=O)(C(C)N(OC)C(=O)CCCCCN(C(=O)CC1CCCC1)C)OC 24757,CC(C)CCN=C(NCc1cccc(Cl)c1Cl)N1CCC(OC2CCCC2)CC1 24758,CCS(=O)(=O)C=CC(=O)N1CCC(CCNC(c2cncc(N)c2)=O)C1 24759,N1(C(c2n(CC)cnc2)C(=O)NC2CCOC2)CCn2nc(C)c(Br)c2C1 24760,c1(C(C(N2C(CNC(COCCCOC)=O)C=CC2)=O)OC)cc(F)cc(F)c1 24761,c1(C(=O)NC2CC(NC(C3C(COC)(COC)C3)=O)C2)cc(C)nnc1O 24762,N(C(=NCc1ccco1)NCC1(O)CCSC1)CC(C1CCCCC1)(C)C 24763,C#CC(CNC(C1C=CCCN1C(=O)COCC(=C)C)=O)CC(C)(C)C 24764,N1(C(C(CCC)OCC)=O)CCN(C(c2ccc3nncn3c2)=O)C2CCC12 24765,N1(c2n(CCC#C)c(C3CCc4c[nH]nc4C3)nn2)CCCC2(CCCC2)C1 24766,c1(NC)cnncc1C(N1CCC(O)(CN(C)C(C2CC=CCC2C)=O)C1)=O 24767,c1(CCS(=O)(=O)NCC)nc(CC(C)(C)C)nn1-c1nccn1C 24768,N1(C(C2CCN(C)C2)=O)CCC12CCCN(C(c1ccnc(OCCO)c1)=O)C2 24769,N1(C(C(C=C=C)C)=O)CC2COCCC2(NC(c2ccc([N+](=O)[O-])[nH]2)=O)C1 24770,N1(C(c2n[nH]c(CC)c2[N+](=O)[O-])=O)CC(C2CCCN(C(=O)C#CC3CC3)C2)C1 24771,N1(C(C(C)OCCC=C)=O)CCCCCC1C(=O)NCC1(OC)CC1 24772,c1(C(N2C(CC(=O)NCCC(=O)NC)CCC2)=O)cc(Br)ccc1O 24773,CCC(CO)C(=O)NCCCCCn1cc(COCCN(C)C)nn1 24774,C(=O)(CCCCC(=O)NCC1(C(C)NC(c2cnc(N)cn2)=O)CC1)NC 24775,Cn1cc(N)c(C(=O)N(C2CCN(C(c3ccc(Cl)s3)=O)C2)CCO)n1 24776,S(=O)(=O)(c1ccnc(NC(c2cncc(CN)c2)=O)c1)NC 24777,c1(C(N2CC(O)(CCNC(C(C=C=C)C)=O)C2)=O)cc(Br)c2ncccc2c1 24778,c1(SCCC(C)NC(=O)C(=O)NCCC2(C)CC2c2ccccc2)ccccc1 24779,C1(CC(=O)NC(C2CCCC2)CNC(CCc2n(C)cnc2)=O)CCC=CCC1 24780,Cc1ccc(F)c(OCC(=O)N(CC(C)NC(c2ncn3c2CCC3)=O)C)c1 24781,C1(C#N)(C(=O)NCC(C(C)(C)C)NC(c2cnn(C(F)F)c2)=O)CC2CC2C1 24782,n1(CC)cc(CN2C3CN2C3)nn1.C(=O)(C(C1CC1)OC)N(N1CCCC1)C.C(C)=O 24783,Cc1cc(Br)cc(C(N2CCC3C(NC(C4CC=CCC4)=O)C23)=O)c1N 24784,c1(C(=O)NC2C(C)CCN(C(c3cnc(C)o3)=O)C2)cc2c([nH]1)CCCC2 24785,N1(C(CSCC)=O)CCC2CCN(C(=O)Cc3c(C)nn(CC)c3C)CC2C1 24786,c1(N2CC(NC(c3cccc(C#C)c3)=O)C(C#N)C2)ncnc2sc(Br)cc12 24787,Cc1c(C(=O)NCCCOCCNC(=O)CC(C)c2ccco2)ccn1C(C)C 24788,CCCC(C(=O)N1CC(NC(C2COCCOC2)=O)CC1CO)OC 24789,c1(OC)cc(NC2CC2)ccc1C(=O)NC(C)CCCCNC(=O)C(=O)C(C)(C)C 24790,CC1(C)COc2cc(CNC(N3CCCC3c3nncs3)=O)ccc21 24791,c1(-c2nc(N(C(C)=O)C(c3nccnc3Br)=O)sc2)cn(C)nc1C(F)(F)F 24792,N1(C(C(C=CC)O)=O)CC(C)(CNC(C2CC3CCC2CC3OC)=O)CC1(C)C 24793,C1(C(=O)NCC(CNC(C(C)Cc2ccncc2)=O)F)C2CC3C(C2=O)C13 24794,N1(C(C(CC#C)NC(=O)CCC(F)(F)F)=O)CC(C)(C)CCC1C 24795,C1(NC(C2CCC(N(CCOC)C)CC2)=O)CC(=O)CN(C(=O)OC(C)(C)C)C1 24796,Cc1ncc(N)cc1C(=O)N(C1CCCN(C(C2CC3CCC2CC3)=O)CC1)C 24797,CN1CCN(C(=O)C(C)(C)CC2CC2)CC1C(=O)NCC1C2CCCC12 24798,c1(C(N(C(C)CNC(=O)CSC(C)C)CC)=O)cccc(CCO)c1 24799,C1(NC(c2c(CC)cncc2)=O)COC2(CCN(C(c3cn(C)c(C)n3)=O)C2)C1 24800,C1(C(=O)NC(CC=C)CO)CN(C(c2ccns2)=O)CC1C(C)C 24801,C1(C(=O)NC2CCCCN(C(c3ccco3)=O)C2)CCC2C(CC1)C2(F)F 24802,c1(C(=O)NC2CCC(C)N(C(c3cncc(Cl)c3Cl)=O)C2)cnc2ccnn2c1 24803,C(=O)(C1Cc2ccccc21)NC(C(=O)NCCc1ccc(C)nc1)CCC1CC1 24804,N1(C(C2(CC)COC2)=O)CC(C)CC1C(=O)Nc1cccc(F)n1 24805,C1(C(=O)NC(CNC(c2n(C)cnn2)=O)C(C)(C)C)CCCCN1N=O 24806,N1(C(C(C2CN(C(c3cc(C)sn3)=O)C2)O)=O)CC(O)CC(O)C1 24807,c1(OC)cc(Cl)ccc1NC(=O)NCC(N1CC(=O)NC(C)C1)(C)C 24808,N1(C(C(C)(C)C2CC2)=O)CCOCC(C(=O)NCC2(CC3CC3)CCC2)C1 24809,N1(C(C(C)(CSC)NC(C(CC#C)C2CC2)=O)=O)CCOCC(=C)C1 24810,C=CCCCC(C(=O)NOC(CC)CC)NC(c1csc(C)c1)=O 24811,Cc1cc(CN(C(C)CCNC(=O)CC2CCOC(C(C)C)C2)C)c(C)o1 24812,c1(C(C(=O)NCc2ccccc2)N(c2nnn(C)n2)C)c(Cl)nc2sccn12 24813,N1(C(C2=CCC(NC(C(CCC)=CCC)=O)C2)=O)CC2CCCCC12C 24814,C1(C(=O)NC(C2CCCC2)CNC(C2NC(=O)OC2)=O)CCS(=O)CC1 24815,CC1(C)CC2(CO1)CN(C(C1CN(C(C3(C)CCCCO3)=O)CCO1)=O)C2 24816,c1(C(N(C(CNC(Cc2cncc(C)c2)=O)C)C)C)cccc2ccccc12 24817,N1(C(c2n(CCCC)ncc2)=O)CC(NC(c2cc(O)ncn2)=O)CC(O)C1 24818,N1(C(C2CCN(C(C(CC)COC)=O)C2C)=O)CCC(O)C(O)C1 24819,CC1CCc2nc(C(N3CCC(N(C)C(c4cccs4)=O)C3)=O)ccc2C1 24820,CCCC(CCC)CCCC(=O)NC(C)(C)CN(C(=O)C(C)n1cncn1)C 24821,n1(CC(=O)NC2C(NC(C(C)C(F)(F)F)=O)CCCC2)ccc(=O)n(C)c1=O 24822,N1(C(C(C)CC(C)(C)C)=O)CCC2(CC1)CCN(C(C1COC(=O)N1)=O)CC2 24823,c1(C(N2CCC(CN(C(Cc3ccc(C)s3)=O)C)CC2)=O)cc2c(ncn2C)s1 24824,N1(C(c2csc(-c3ccccn3)n2)=O)CCC2C(CCCN2C(=O)C2CC2)C1 24825,N1(C(C2(NC(C(CCC)O)=O)CC2(C)C)=O)CC(OC)CC(C)C1 24826,CC1CCN2N=C(C(=O)NCC3CCN3C(c3ncccn3)=O)NC2=N1 24827,C1(c2cc(C)no2)CCCCCN1C(=O)CC1CCN(C(=O)C2CC2)C1 24828,CCC(CC)C(C)C(=O)NC1CCC(C)(CNc2nc(C(=O)OC)ns2)CC1 24829,c1(CNC(CC2(C)CCN(C(=O)C(F)(F)C3CCCC3)C2)=O)cnc(O)c(F)c1 24830,C1(CCOC)CCCN(C(c2ccc(NCC(N)=O)cc2)=O)C1.C1(C)CC(=O)N1 24831,N1(C(C(N(C)C)C2CC2)=O)CCC2C(C1)NC(=O)CN2C(=O)Cc1cncn1C 24832,c1(-c2c(C)ccnc2)cccc2c(C(=O)NCCCO)n[nH]c12 24833,C1(C(=O)NC(C(C)NC(c2ccn(C3CCCC3)n2)=O)CO)CCOC(C)(C)C1 24834,c1(C(=O)NCCC2N(C(CN(C(C)=O)C)=O)CCCC2)ncc(Cl)cc1O 24835,C1(C(=O)NCC(CO)NC(c2ccc(C(=O)OC)cc2)=O)CC(C)(C)CN1C 24836,C1(CC(N2CCC(OCC=C)CC2)=O)CN(C(=O)CN2CCOC2=O)CCC1C 24837,N1(C(c2ccc(C#C)cc2OC)=O)CCCC12CCCN(C(C1CCOC1)=O)C2 24838,O=C(CCCC(F)F)NCCC12CCC1CN(C(=O)Cn1cc(Cl)cn1)C2 24839,C1(NC(CCCNC(N)=O)=O)CCC2(CCN(C(c3ccnnc3O)=O)C2)C1 24840,N1(C(CCOCC#C)=O)CC=CC1CNC(=O)C(C)OCCN(C)C 24841,Cc1ccn2ncc(C(=O)NC(CNC(=O)COC3COC3)CC(C)C)c2c1 24842,N1(C(CCc2c(C)ncs2)=O)CCN(C(=O)CCn2cc(Cl)cn2)C(C)CC1C 24843,C12(CC(=O)NC(CC)CNC(c3cnc(NC4CC4)s3)=O)CCC(CC1)C2(C)C 24844,Cc1c[nH]c(=NC(=O)c2cc(C)c(NC(c3ccccc3)=O)c(Cl)c2)cn1 24845,c1(C(=O)NCC(=O)NCC(=O)NC2CCCC(OC)C2)ccc(P(C)(C)=O)o1 24846,c1(C(=O)OC)ccc(C(=O)NCC(C)NC(=O)CCC(C)SC)cc1Cl 24847,c1(C(=O)NCC(CC)NC(=O)Cc2cc(F)ccc2Cl)cc(F)c2cn[nH]c2c1 24848,c1(C(N(CCN(C(=O)CC2C=CS(=O)(=O)C2)C)C)=O)cccc2c1OCC2 24849,C1(NC(=O)COCC2CCC2)CC(F)(CNC(c2cc(Cl)no2)=O)C1 24850,c1(C(=O)NC(C)CCNC(=O)C(C2CCCCC2)C)nnn(C)c1N 24851,c1(SC)nc(N2CCC(C(=O)NCc3c(F)cccc3F)C(O)C2)cc(C)n1 24852,c12cc(C(C)(C)C)cc(C(C)(C)C)c1N2.c1(C2C(OC)CC2)ccc(C)cc1 24853,Cc1cnncc1C(=O)NC1(CC=CC(=O)NCC2CN3CCC2C3)CCC1 24854,C1(NC(c2ccncc2Br)=O)CN(C(C2CCCCO2)=O)CC(F)(F)C1 24855,C(=O)(CC(C)(O)C(F)(F)F)N1CC(C(C)NC(c2c(C)cc(C)[nH]2)=O)OCC1 24856,c1(CNC(CCSCCC)=O)ccc(CN(C)C(c2ccncc2F)=O)cc1 24857,CS(=O)(=O)C1(C(=O)NC2CC(CNC(C34CCCN3CCC4)=O)C2)CCC1 24858,CC1CN(C(=O)C(F)(F)c2cscn2)CCC1N(C(=O)CSC(F)F)C 24859,c1(NC(=O)CC(c2ccc(F)cc2)NC(=O)CN2CCCC2)c(Br)ccnc1Cl 24860,Cc1n[nH]cc1CC(=O)NC(CO)C(C)NC(=O)CC(C)n1cccn1 24861,Cc1ncnc(C)c1C(N1CCC(C(C)NC(c2cnn3c2CCC3)=O)CC1)=O 24862,C1(F)(C(=O)NCC2(NC(Cc3ccc(C(N)=O)cc3)=O)CC2)CC12CCCCC2 24863,C1(C(N2C(CC)CN(C(=O)C(F)(F)CC3CC3)CC2)=O)CCC(=O)C(C)C1(C)C 24864,C(=O)(CC(C)C(F)F)N1CCC(N(CCOCCOC)Cc2cccnc2)CC1 24865,CCC(C)(C#N)C(=O)NCc1ccc(C(=O)NC2(CO)CC(F)(F)C2)cn1 24866,c1(C(=O)NC(CNC(=O)C(F)OC(F)(F)F)C2CC2)cc2c([nH]1)CCOC2 24867,S(=O)(=O)(c1ccc(CC(=O)NCC#CCNC(=O)CC#N)cc1)NCC 24868,Cc1c(CC(N2CC(O)CC2CNC(c2cnc(Cl)s2)=O)=O)ncn1C 24869,C1(NC(=O)CCC2CCCCN2C(C2CCCCCCC2)=O)C2CCC(F)(F)C12 24870,CON=CC(=O)N1CCC(C(=O)NCC2CC2c2ccco2)O1 24871,N1(Cc2c(C)cc(Cl)cc2)CC2C3CCC(C2C1)N(C(c1ocnc1C)=O)C3 24872,c1(C(N2CC(NC(c3csc(Cl)c3Cl)=O)CC(C)C2)=O)ccc2c(c1)CCCC2 24873,CCCCC(O)CC(=O)NCC1CCCN1C(c1cnc(C(C)C)s1)=O 24874,N1(C(C(c2ccccc2)=O)=O)CC(NC(C2CCCSS2)=O)CC2(CCC2)C1 24875,CCC(C)(CO)C(=O)N1CCCOC(CCNC(=O)CCC(=O)N(C)C(C)C)C1 24876,Cc1cccc(-n2nnc(CC3CC(F)CN3C(=O)OC(C)(C)C)c2C(C)C)c1 24877,c1(N2CCC3(CN(C)C3)C2)ccc(Br)c(S(=O)(=O)NC2C(CO)CCC23CCC3)n1 24878,CC(C)C(C)(C(N)=O)NC(C1CC2CC2N1C(C1CC2C=CC1O2)=O)=O 24879,c1(N2CCC(NC(N3CCCCC3c3ncc[nH]3)=O)C2)ccc(Br)nc1 24880,c1(OC)ccccc1C(=O)NCC(=O)NC1CC1NC(C1CC(C(F)(F)F)C1)=O 24881,c1(C(=O)NC2C(NC(C3C(c4n(CC)cnn4)C3)=O)COC2)cc(N)ccn1 24882,c1(N(C(CC)C)CCOCCn2nc(C(C)C)cc2C)ccc(C=O)cc1 24883,c1(CC)nn(C)cc1C(=O)N(CC(CC)NC(=O)C(C)Cc1cccc(F)c1)C 24884,c1(C(N2C(CC)CCCC2)C(=O)NC2CCOC2)cc(=O)n2ccccc2n1 24885,C(c1ccc2cc(OC)ccc2c1)=CC(=O)NCCNC(CCC(=C)C)=O 24886,c1(C(=O)NCC2CCN(C(C(C)=C3CCCC3)=O)C2)cccn2c(C)nnc12 24887,Cc1csc(=NCC(=O)N2CCC3C(C2)CN3C(=O)CC(C)CN(C)C)[nH]1 24888,C(=O)(C1CCCc2nc[nH]c21)NCC(CNC(c1nc(OCC)sn1)=O)OC 24889,C1(C(=O)NCC2C(NC(c3nc(OC)c(C)s3)=O)C2)CCc2ncnn2C1 24890,c1(OC)cc(N2CC3CN(C(c4ccco4)=O)C3C2)nc(C)n1 24891,CC1(CNC(c2cn(CCO)nn2)=O)CCN(C(C2(OC)CCC2)=O)CC1 24892,C=CCC(CNC(=O)C(C1CCOCC1)F)C(=O)N(C1CC=CCC1)CCF 24893,c1(C(N2C(C3CCN(C(CCC(C)C)=O)CC3)CCC2)=O)ccc2n[nH]cc2c1 24894,N1(C(c2c(C)[nH]nc2C(F)F)=O)CC(NC(=O)C=Cc2cnc[nH]2)CC(O)C1 24895,C1(=O)C(O)CC(=O)NCCN1CCCC1CC(O)C1.c1(S)ccccc1.CCO 24896,C(CNC(=O)CCCNCCO)(C(C)(C)C)NC(CCNC(C)=O)=O 24897,Cc1nn(C)cc1C(=O)NCC(C1CCCCC1)NC(=O)C(F)n1ccnc1 24898,C(=O)(CS(=O)(=O)CC(F)(F)F)NCC(C1CC1)NC(C1(CC#C)CCOCC1)=O 24899,Cc1n[nH]c(C)c1C(C)C(=O)N(CC)CC1CCCN1C(=O)CC1CCOCC1 24900,c1(N(C2C3CCC2CNC3)C(C(c2n(C)ccc2)=O)=O)nc(Cl)c(Br)cc1O 24901,N1(C(C(OC)OC)=O)CCCC(NC(c2ccc(OC)cc2C(F)(F)F)=O)CC1 24902,C(=O)(C(CN(C)C)CC(C)C)NCC1C(C(=O)NC2(CC=C)CCCCC2)C1 24903,C1(CNC(C(C)n2cccn2)=O)CC2CC2N1C(=O)C=CCN1CCOCC1 24904,Cc1cccnc1CC(=O)NC1CC(C(=O)N(CCC#N)C2CC2)C1(C)C 24905,c1(OC)cc(F)c(CC(=O)NCCNC(c2cnc(C(F)(F)F)s2)=O)c(Cl)c1 24906,c1(C(C(=O)NCC2(F)CN(C(C3CC(OC)C3)=O)C2)(C)F)ccc(F)cc1 24907,c1(C(=O)NCC2CN(S(=O)(=O)C3CC3)CCO2)c(C(F)(F)F)cccc1Br 24908,c1(C(=O)NC2CC(C)(CNC(CC=C)=O)C2)cccc(OC)c1 24909,Cc1ccc(C(c2ccccc2)N(C(=O)NCCN2CCC(O)C2)CC#N)c(C)c1 24910,c1(OCC)cc(C(=O)NC(C(=O)OCc2ccccc2)C2CC2)ccn1 24911,C#CCC(C)(C(=O)NCC(CCC)OCC)NC(=O)C(CC)C(=O)OC 24912,O=C(C1=NOCC1)N1CCC(C2CCCCN2C(c2n[nH]cc2Cl)=O)C1 24913,C(CCCCCN)N(C(=O)C(N)CC1CCS(=O)(=O)C1)C 24914,C1(NC(C(=O)NC2CC2)=O)CCCOC12CCN(C(C1(C3CC3)CCC1)=O)CC2 24915,c1(-c2cn(C3(C(=O)OC)CN(C(C4(C)CNC(=O)C4)=O)C3)nn2)cc(OC)nn1C 24916,c1(C(=O)NCC(CNC(C2CN(C)C(=O)CC2)=O)(C)O)c(F)ccc2[nH]ccc12 24917,c1(C(C)NC(C2CC(F)(F)C2)C)cccc(NC(c2ccccc2)=O)c1 24918,c1(C(=O)NCC(CC)NC(C2C3CC(=O)CC23)=O)nc(C)oc1C 24919,C(C(=O)N(CC(=O)NCc1nonc1C)CC(C)C)(C(C)C)SCC 24920,c1(OC)ccccc1OC(C)C(=O)NCCC(C)N(C)C(c1c[nH]c(C#N)c1)=O 24921,C1(OCC(=O)OC)CCN(C(C2CN(C(c3ocnc3C)=O)CCS2)=O)CC1 24922,C#CC1(O)CC(C(N2CC(F)CC2C(=O)N(CC=C)CCC)=O)C1 24923,C12(C(N3CC(CC)(CC)C3)=O)CCCC1CCN2C(=O)CCC1OCCO1 24924,CN1CCC(CC(=O)NC(CC2CCC2)C(=O)NCCN(CC(F)F)C)CC1 24925,N1(C(C2CC23CCCC3)=O)CC2CCC1C(CNc1cc(F)ncn1)C2 24926,C1(NC(c2cc(C(C)C)[nH]n2)=O)CC2CC1N(C(C1(C(F)F)CCC1)=O)C2 24927,CCC(C(=O)N1CC(CCNC(c2ccn(C)c2C)=O)C(C)C1)C(C)C 24928,Cc1cc(C(N2C3CC2CN(C(c2c(O)cccc2O)=O)C3)=O)cc(Br)c1 24929,Cc1ccc2cc(C(=O)N(CCNC(=O)Cc3ccc(C)s3)C(C)C)cnc2c1 24930,c1(C(=O)NC2(C)CCC(NC(c3ccn(C)n3)=O)CC2)ccc2c(c1F)CCC2 24931,Cc1ccc(NNC(=O)c2csc3cc(Br)ccc23)cn1 24932,c1(OC)cc(C=CC(N2CCC(NC(=O)C(F)CC3CCCC3)C2)=O)sn1 24933,c1(C(=O)NC2CCN(Cc3cc(F)ccc3Br)CC2)ccc2c(c1)CNC2 24934,N#Cc1ccc(Cl)c(C(=O)NCCNC(C2CCOC2c2ccccc2)=O)c1 24935,c1(COC)n[nH]c(=NC2(CNC(=O)CCc3c(N)cnn3C)CCCCC2)s1 24936,O=C(CN1C(=O)Cc2cc(F)ccc21)NC1CN(C(=O)CC2CC=CCC2)C1 24937,C1(NC(CCCSC)=O)CCC2CCN(C(=O)C=Cc3cncn3C)C1C2 24938,c1(C(=O)NCC2C3CN(Cc4cccc(C)c4Br)CC32)ccc2scnc2c1 24939,C1(NC(c2ccc(C(=O)OCC)o2)C)CCC(CC(C)(C)C)C1 24940,Cn1nc(C(N2CC(CCNC(c3cnoc3C3CCC3)=O)C2)=O)cc1Cl 24941,CC1CC2(C(N3CC(SC(C)(C)C)C3)=O)CC12 24942,C1(C(=O)NC2(CC(=O)NCC(CNC(N)=O)O)CC2)CC=CCO1 24943,c1(C(=O)NC(CN(C(c2ccc(F)c(O)c2)=O)CC)C)ccc(C)cc1OC 24944,N1(C(c2ccc(C(C)C)s2)=O)CCC(NC(=O)CCN2CCCC2=O)C1(C)C 24945,CC(CC(=O)N1CCC(N(CC(C)C)C(C2CCC(O)C2)=O)CC1)C(F)(F)F 24946,C=CC(CC(=O)N1CC(O)(CNC(c2oc(CC)nc2C)=O)C1)c1ccccc1 24947,c1(C(N2CC(O)(C(C)NC(CCC(=C)C)=O)C2)=O)nc(Cl)ccc1Cl 24948,c1(OCC)ccc(CN(C2CCC2(F)F)Cc2ccccn2)c(C)c1 24949,N1(C(CC2CCN(C(CNC(N)=O)=O)CC2)=O)CCCC(C2CCC2)C1 24950,c1(CN2CCC(NC(C(c3ccnn3C)C)=O)C(O)C2)ccc(F)c(C#N)c1 24951,C12(C(N(C3CCCC(NC(c4coc(C5CC5)n4)=O)C3)C)=O)CCC(CC1)C2 24952,C(C(=O)NCCCC(C)NC(=O)CCNC(c1ccco1)=O)(C(C)(C)C)SC 24953,Nc1nc(NC(=O)NCCS(=O)(=O)Nc2c(Cl)nsc2Cl)ccc1O 24954,C=CC(C)(O)CC(=O)N1CCC(C(C)(C)C(=O)N(C2CCOC2)C)C1 24955,N1(C(c2c(C)non2)=O)CCC(C)(C(N2CCC(CN(C)C)C2)=O)C1 24956,CC(O)C(C)C(=O)NC1(CNC(=O)CCCc2cccs2)CC1 24957,N1(C(C2N(CCC)C(=O)CC2)=O)C2CCC1CN(C(C1C(C)(C)C1(F)F)=O)C2 24958,C(=O)(CCCCC#N)NCC1CN(C(C=CCOC)=O)C(C)C1 24959,C1(NC(C(CC)OCC)=O)CC2CC(C1)N(C(c1ccnc(Cl)c1N)=O)C2 24960,c1(OC)nc(Cl)ccc1C(N1CCCCC(NC(C2CCN(C)C(C)C2)=O)C1)=O 24961,C(=O)(C1=CCC(C)(C)CC1)NC1(CCCCNC(c2cc(C)sc2C)=O)CC1 24962,C(=O)(CCCC(N)=O)N1CCC(NC(C2C(C)C2(F)F)=O)C1C1CC1 24963,CCN=c1[nH]cc(C(=O)NCC2CCN2C(c2cn(C3CCOC3)nn2)=O)s1 24964,CCC(C)(COC)C(=O)NC1C=CCC(C(=O)NCC(C)C(C)O)C1 24965,C1(C)(C(N(C(CCNC(C(C(C)C)n2cnnc2)=O)C)C)=O)CC2CCC(C1)S2 24966,N1(C(C2CCN(c3ccccc3)C2)=O)CCc2sccc2C1c1ccc(Cl)cc1 24967,c1(C(=O)NCC2CCCN2C(=O)C2=CCS(=O)(=O)C2)ncnc2ccccc12 24968,Cc1cnc(C(N2CC3CC2C3C(=O)N(C)Cc2cnn(C)c2C)=O)c(F)c1 24969,c1(OC)ccc(C)cc1C(=O)NC1CCC1C(=O)NCCN(C)CC(=O)C(C)C 24970,c1(C(CN(C)Cc2snc(C)n2)O)ccc(Cl)c(Cl)c1 24971,N1(C(c2nc(OCC)oc2)=O)CCC(C)(C)C1CNC(=O)C(C)(C)CO 24972,c1(CC(N2CCSC3CCC23)C(=O)NCC=C)ccc(OC)c(OC2CC2)c1 24973,Cc1cccc(CO)c1C(=O)Nc1ncc(CNC(=O)C(C)(C)C(=O)N(C)C)s1 24974,N1(C(c2n[nH]c(C)c2C)=O)CC(C)(C(=O)NCC(c2ccccc2)O)CC1(C)C 24975,C1(C(=O)NC(C2CCCN2C(=O)CC2CCC(=O)O2)(C)C)CCc2cncn2C1 24976,C=C=CC(C)C(=O)NC1(C(F)F)CC(NC(=O)CCCOCCOC)C1 24977,N1(C(c2scc(COC)c2)=O)CC2CCCC(N=c3[nH]nc(C(C)(C)C)o3)C2C1 24978,CCC(CCCC(=O)N1CC2COCC2O1)NC(C1(F)C(C)(C)C1(C)C)=O 24979,N1(C(CCC(C)OCC)=O)CCN(C(c2cnc(C)s2)=O)CC1CC(F)(F)F 24980,CC1CCN(C(c2cc(Cl)c(Cl)[nH]2)=O)CC1NC(=O)Cn1ccc([N+](=O)[O-])n1 24981,N1(C(C(=O)NC(C(=O)OC)C)c2ccoc2)CC(c2cccc(Cl)c2)OCC1C 24982,CCCCC(C)C(=O)NCCn1cc(CNC(=O)CSc2ccc(Cl)cc2)nn1 24983,c1(C(N(C(CCNC(C=NOC)=O)C)C)=O)cccc2c(C)coc12 24984,C=CC(CCC)CC(=O)NCc1ccoc1C(=O)NC1(C)CC1(C)C 24985,C1(NC(C2CC(=C)C2)=O)CC2CCC1CN(C(c1cn(C3CCOC3)cn1)=O)C2 24986,C(=O)(CCC(C)(C)O)N(C)CCn1cc(-c2ccc(CO)cc2)nn1 24987,C1(COC)(NC(=O)CCNC(N)=O)CCN(C(C2CC3(CSC3)C2)=O)C1 24988,N1(CC2CCC(C)O2)CCN(C(=O)CC2CCCC2)CC1 24989,c1(C(=O)NC2CCC(N(C(CCN(CCC)C)=O)C)C2)cc(C)ccc1C1CC1 24990,C1(C(=O)NC(C(=O)NCC(C)(C)SC)(C)C2CCC2)Cc2ccccc2C1 24991,c1(C(N(C2CCN(C(=O)CCc3ncco3)CC2)C)=O)ccc(F)c2c1OCC2 24992,O=C(CC1CCOc2ccccc21)NC1CN(C(c2nccc(Br)c2)=O)C1 24993,Cc1cc(-c2cncc(C(N3CCN(CCCO)CC3)=O)n2)c(C)cc1O 24994,C1(SCC)CCCCC1NC(=O)C(n1cc(C(C)(C)S(C)(=O)=O)nn1)C 24995,CCC(CN)(CC)NC(C1CCCN1C(=O)C(C(=O)C(C)(C)c1cnc[nH]1)=O)=O 24996,C1(CC)CN(C)CCCN1C(=O)C(CC(N)=O)NC(=O)C(C(C)OC)N(C)C 24997,c1(CC)ccc2c(c1)C(CC(=O)Nc1cc(S(C)(=O)=O)ccn1)C(=O)N2 24998,c1(OCC)ccc(CN(C(=O)C(CC)n2cccn2)CCCC(=O)O)cc1 24999,C1(OC(c2ccccc2)C(C)C)CC(C(=O)NC2CC3CNC2C3)CCC1O 25000,Cc1cc(CNC(=O)C(CC2CCCC2)NC(=O)C(C)C#N)no1 25001,c1(CN2C(CCP(C)(C)=O)CCCC2)ccc(Cl)c(Br)c1 25002,c1(C(=O)NCC23CC(NC(CCC(=C)Cl)=O)(C2)C3)c(C)cccc1[N+](=O)[O-] 25003,C=CC1(C(=O)NCC(C(C)C)NC(c2cncc(OCC)c2)=O)CCOCC1 25004,c1(C(N(CC(C)CNC(=O)CCCn2ccccc2=O)C)=O)cc(Cl)ccc1N 25005,CCCC(C)C(=O)NC1CC(F)(C(=O)NC2(O)CN(C(=O)OC(C)(C)C)C2)C1 25006,C1(C(N2CC(CO)(CO)C2)=O)CCC(CNC(c2n[nH]cc2C(F)(F)F)=O)CC1 25007,n1(CC)cnnc1CNC(=O)C(C1CC1)N(C(=O)Cc1nonc1C)C 25008,N1(CCC)CC(C(=O)NC(C)(C)C(C)NC(=O)C(c2ccc(F)cc2)=O)CC1=O 25009,C1(NC(CCCCCOC)=O)CC2(CCN(C(c3cc4sccc4s3)=O)CC2)C1 25010,c1(CCC)ccc(N)c(C(=O)NCC=CCNC(=O)C=CC2CCC2)c1 25011,C1(C(=O)OCC)CN(C(=O)C(Br)=C(C)C)CC1C1CC1 25012,N1(C(c2ncn(C)n2)=O)CCCC2CN(c3nc4ccc(Br)cc4s3)CCC12 25013,C=CCC(CC=C)C(=O)NC(CN(C)C)C(=O)NCC(=O)NCC1CCC1 25014,C1(CNC(C=C(CC)C)=O)CN(C(c2cc(C)[nH]n2)=O)CC12CCC2 25015,C(CC(O)CCc1ccccc1)c1cn(COCCCC(=C)Br)nn1 25016,C=CCCCCC(=O)N(C1CCCN(C(=O)C(c2cccnc2F)(C)C)C1)CC 25017,N1(C(c2cc(C)n(C3CC3)n2)=O)CC(CNC(=O)C=CCO)C2(CC2)C1 25018,N1(C(C(COC(C)(C)C)(C)C)=O)CC2CC(NC(=O)CCC3CCOC3)C1C2 25019,c1(C(=O)NC(C2CC2C(N2CCCC(O)C2)=O)C)ccccc1O 25020,N1(C(c2cc(CC)sn2)=O)CC2CCN(C(C3CCc4nc[nH]c4C3)=O)C2C1C 25021,C1(NC(c2cn(CCC)nc2)=O)CS(=O)(=O)CC1NC(=O)C=Cc1csc(C)n1 25022,c1(C(N2CCC(NC(c3c(CC)cno3)=O)C23CC3)=O)noc2c(F)cccc12 25023,C(=O)(C(C)(C)CN1CCN(C)CC1)NCC1CC(NC(C(C)OC)=O)C1 25024,Cc1ccnc2sc(C(=O)NCC3CC3NC(=O)Cc3ccc(O)c(F)c3)c(C)c12 25025,CC1CN(c2nnnn2CCCC(C)(C)C)C(C)C1C 25026,C(=O)(CCOCC)OCC.C(=O)(C(c1cnsc1)N(CCCN(C)C)C1CC1)C1CC1 25027,C12(C(=O)NCC3C(NC(CN(CC)CC)=O)CCCC3)CCCN(CC1)C2 25028,CC(C)CC(CNC(C1OCCC1C(C)C)=O)C(=O)Nc1ccccc1N=[N+]=[N-] 25029,c1(CC)onc(C(N2CCOC(C(=O)N(CC(C)CO)C)C2)=O)c1C 25030,C1(NC(c2n(C)c(S)nc2)=O)CN(C(c2noc3c2CCCC3)=O)CCC1(C)C 25031,C(C(O)CC(=O)NC1(CCCCO)CC1)NC(CCCNC(C)=O)=O 25032,CN1CCC(N=c2[nH]c(=NCC3CC4CCC3N(C)C4)[nH]c3cccnc23)CC1 25033,C(c1c(C)nn(C)c1Cl)=CC(=O)NC1C(OC)CN(C(c2cc(=O)cc[nH]2)=O)C1 25034,C1(NC(C(C2CC2)OC)=O)CCN(C(c2cn(CC(=O)N(C)C)nn2)=O)C1C1CC1 25035,C(C(c1ccccc1)NC(=O)CCF)(C(C)C)NC(c1c(OC)nsc1)=O 25036,C(C(=O)NCC1CC(NC(c2csc(CO)n2)=O)C1)(C(C)O)NC(C)=O 25037,C1(NC(CC2(C=C)CC2)=O)C2CC3CN(C(c4n[nH]c5c4CCCC5)=O)C1C3C2 25038,c1(N(C2CNCC2F)C(c2ccc(OC)nc2OC)=O)ncnc2c1ccn2C 25039,C(=O)(C1=Cc2cc(Br)ccc2OC1)NC1CCN(C(C)=O)CCC1(F)F 25040,c1(C(N2CCC3(C(C(=O)Nc4ncc(Br)s4)C3)CC2)=O)c(F)c(F)cc(F)c1F 25041,c1(OC)ccc(C2CC2C(=O)NCCCCNC(=O)C(F)(F)c2cscn2)cc1 25042,CCC(C)(CC)NC(C1CC(CCNC(=O)CC(=O)N(C)C)C1)=O 25043,C1(N(C(=O)CCCC2CCC2)C)CCCCN(C(=O)C(c2ccccc2)O)C1 25044,C1(C(=O)NCCCCN(C)C(C2(C(F)(F)F)CC=CCO2)=O)CC12CC(C)(C)C2 25045,C(=O)(C(C)CS(=O)(=O)NC1CCC(CC(C)(C)C)C1)OC 25046,CCC(c1ccccc1)=CC(N1CCC(C)C1CNC(c1c(C)coc1C)=O)=O 25047,C1(CNC(CCN(CC#C)C(C2CC(C)CO2)=O)=O)CCCOCC1 25048,c1(C(N2CCCCC2C=Cc2ccccc2)C(=O)NCC)cc(C)c(Br)cc1F 25049,N1(C(C2C(OC)CCC2)=O)CCCCC(C(=O)NCCC2(CO)CCC2)C1 25050,N1(C(Cc2cc(C)[nH]n2)=O)CCC2(CCN(C(c3cc(Cl)c(N)c(Cl)c3)=O)C2)C1 25051,C1(C(=O)NCCN(C(c2c(N)cc(F)cc2Cl)=O)CC)CCn2c(cnc2C)C1 25052,C(N=c1cc[nH]cc1)C1CCN(C(=O)Nc2c(C)n(-c3ccccc3)nn2)CC1 25053,C=CC(O)C(=O)N1CCC(n2cc(CNC(=O)C(=O)NCC(F)(F)F)nn2)C1 25054,C1(NC(c2ccsn2)=O)COCCN(C(=O)CCc2ccsc2)C1 25055,c1(C(N2CCOC(CN(C)C)C2)C(=O)NCCCCCC)cc(F)cc(Br)c1 25056,C(=O)(C1SCc2cccnc21)NCC=CCNC(c1cc(CCC)[nH]n1)=O 25057,C(=O)(C1CCc2c(F)cccc21)NCc1cc(OC)ns1 25058,C1(C(=O)NC2C(C(N(C(C=C)C3CC3)C)=O)OCC2)CCOC(C)C1 25059,C(=O)(C(C)(C)Cc1ccccc1)NCCCN(C(C1CCN(C(C)C)C1)=O)CC 25060,c1(OC)cccc(CC(=O)OCC2CC(C)N(C(=O)C=Cc3cocn3)C2)n1 25061,c1(OC)cc(I)c(C(N2C3COCC2C3)=O)cc1OC 25062,c1(CCNC(=O)CN(C(=O)CCc2cnco2)C(C2CC2Cl)=O)nncs1 25063,N1(C(CN2CC(C)(C)C2)=O)CCC(CNC(=O)Cn2ncc(O)nc2=O)C(O)C1 25064,N1(CCC(=O)NC(CN(C(c2ccncc2)=O)CC)C)CCCCCC1 25065,c1(CC(=O)NC2C(C)(C)N(C(=O)CCCC(N)=O)CC2)ccc([N+](=O)[O-])cc1Cl 25066,C=CCC(C(=O)NCC(CCOC)NC(c1[nH]nc2ncccc12)=O)C(C)C 25067,c1(C(=O)NC2CC(NC(CS(CC)=O)=O)C2)cc(O)nc2cc(F)ccc12 25068,C1(NC(CN(C(=O)CN2CCCC2C)C(C)C)=O)COCCOC1 25069,C(C(=O)OCC)(C(C)C)NC(N1CCCC(c2c(C(=O)OCC)cn(C)n2)C1)=O 25070,C1(O)(CCNC(C(C)c2ccco2)=O)CN(C(=O)CCSCC(N)=O)C1 25071,c1(C(N2CC(O)(CNC(c3ncn(C(C)(C)C)c3)=O)C2)=O)ccc2c(c1)COC2 25072,C1(OCC)CS(=O)(=O)C2CN(C(=O)C(C)(C)Cc3ccc(C(F)(F)F)cc3)CC12 25073,CC1(CO)CCCN1C(C1CCC(NC(=O)CCC2CC2(F)F)C1)=O 25074,C1(n2cnnn2)(C(=O)NCCC(C)NC(=O)C(C)(C)NS(C)(=O)=O)CCOCC1 25075,Cc1cc[nH]c(=N)c1C(=O)NC(CNC(=O)C(C)c1cccs1)C1CC1 25076,c1(OC)ccc([N+](=O)[O-])c(C(N2CC(F)CC2C(=O)NCC2CCOC2)=O)c1 25077,C1(C(=O)NC(C(=O)N(C)CC)C)COCCN(C(c2c(C)nn(C)c2N)=O)C1 25078,S(=O)(=O)(c1cc(C)ccc1C)N(CC(CC)CC(C)C)C1CCNCC12CC2 25079,c1(OC)ncc(C(N2CCCCC2C2CCN(C(=O)C(C)SC)CC2)=O)cc1F 25080,c1(OC)cc(OC)cc(CC(N2CCN(CCOCc3ncc(C)o3)CC2)=O)c1 25081,c1(C(=O)NC(CNC(C(C(C)C)(C)O)=O)CO)coc(S(N)(=O)=O)c1 25082,CCCCC(CC)C(=O)N1CCCC(C)(C(=O)NC(c2ccc(C)cn2)C)C1 25083,C1(OCC)CN(C(=O)C(=Cc2c[nH]cn2)F)CC1CNC(c1cn(C)nc1Cl)=O 25084,c1(C(N2CCCC(NC(C3CC3(F)F)=O)C2)=O)c(OC(F)F)cccc1Br 25085,c1(CCC(N2CC(C)(NC(c3c(OCC)scc3)=O)C2)=O)n[nH]c2ccccc12 25086,Cc1cc(C(=O)NCC2CCCC2C(N2CCCC(C#N)C2)=O)cc(O)n1 25087,c1(NC(CCCC)=O)ccc2c(c1)CCN(Cc1cccc3c1CCCC3)C2 25088,CC(C)(C)C(C(=O)N1CCC(NC(=O)CC2CCC3CC23)CC1)N1CCOC1=O 25089,Cc1cccn(CC(N2CCN(C(=O)CCCCCN(C)C)CC2C)=O)c1=O 25090,N1(C(C(CCC)=CCC)=O)CCC2CC(C1)CN(C(=O)CCc1cnoc1)C2 25091,c1(N(c2ccc(F)cc2)CCC#N)ccc2ccccc2c1O 25092,c1(CC)cc(C(N2CCCC2CCCNC(c2sccc2F)=O)=O)cn(C)c1=O 25093,N1(C(C2(C3CC3)CN(C(CC3N(C)CCCC3)=O)C2)=O)CCCC2C(O)CC12 25094,N1(C(C2CC(CCNC(C(C)n3ccnn3)=O)C2)=O)CC(C)(C)C12CCC2 25095,c1(C(=O)NC(C2CC2C(N2CC(O)CC(O)C2)=O)C)ccc(C#N)c(C)c1 25096,C1(NC(C(C)C(C)O)=O)CC2CCCC(C1)C2NC(=O)Cn1ccc(O)nc1=O 25097,C(CCCC(C)(C)C(=O)NNC(=O)C1CSC1)NC(c1cc(C)c(F)c(C)c1)=O 25098,Cc1nc(=N)[nH]c(C)c1C(N1CC(NC(c2ccc(C(C)C)cn2)=O)C(C)C1)=O 25099,c1(C(=O)NC2C(NC(C3(C(C)(C)C)CCCC3)=O)C2)cccc(C(F)F)c1 25100,C(=O)(CC(C)C(F)(F)F)N1C(C(N2C(COC)COCC2)=O)CC2CC21 25101,C1(F)(CNC(C(C2CCC(=O)N2)C)=O)CCN(C(=O)CC2SC(=N)NC2=O)CC1 25102,N1(C(C2CCCC(C(N)=O)C2)=O)CCCC(C)(CNC(c2ccc(CO)o2)=O)C1 25103,N1(C(CSCCN(C)C)=O)CCCCC(N=c2ccc(C(F)(F)F)n[nH]2)C1 25104,NS(=O)(=O)CC(=O)NC1CN(C(C2CC(Cc3ccc(F)cc3)C2)=O)CC1O 25105,c1(C(=O)NC2(CNC(C(C)OCCOCC)=O)CCCC2)ccc(C)cc1 25106,N1(C(C(C=C)O)=O)CC(C2CCCN(C(=O)Cc3ccc([N+](=O)[O-])cc3F)C2)C1 25107,Cc1ccc(C)c(C(C)N(C)C(c2cc(-c3ccccc3)[nH]n2)=O)c1 25108,c1(C(=O)NCC(C(C)C)NC(C2CCc3c[nH]nc3C2)=O)cncc2ccsc12 25109,C1(NC(c2cnn(-c3ccncc3)c2)=O)CN(C(=O)C=CBr)C2(CCC2)C1 25110,C(=O)(CC(C)(C)CC(=O)N1CCCC1CNC(C1(C2CC2)CCOCC1)=O)OC 25111,C(=O)(C1=NOC2(CCC2)C1)N1C(CNC(c2occc2Cl)=O)CC(O)C1 25112,C(=O)(CC(F)(F)CC(=O)NCCCOCCNC(=O)CC1CCCOC1)OC 25113,N1(C(c2n(C)cnc2)=O)CCCC(C(=O)N(C(C)(C)C)CCO)C1 25114,C(=O)(C1CCCc2nccn21)N(CCCNC(Cc1cn(C(C)C)nn1)=O)C 25115,c1(C(=O)NCCCCC2CN(C(C3N(CC)CC3)=O)C2)cc(N2CCCC2)ccn1 25116,NS(=O)(=O)CC(=O)NCC1CCCN1C(=O)CC(F)(F)F 25117,c1(C(=O)NC(CC)CNC(=O)Cn2cnnc2)ccc2nc(CO)[nH]c2c1 25118,c1(CC)[nH]nc(C(=O)NC(CCC2CCC2)C(=O)NC(c2cnc(C)s2)C)c1C 25119,N1(C(C=CCOC)=O)CC2OCC(NC(=O)CCOCCc3ccccc3)C2C1 25120,CC(c1cccnc1)=CC(=O)NCC1CC2CCC1N2C(=O)Cc1ccco1 25121,c1(C(=O)NCC(CCOC)NC(=O)C(=O)NOC)ccnc(OC(C)C)c1 25122,c1(N(C(=O)Cn2ccc(CN(C)C)n2)C(C)C)cc(O)nc(C2CC2)n1 25123,CC(CC(=O)NCC1C(C(=O)NC(CC(N)=O)C2CC2)C1(C)C)C(F)F 25124,CCCC(CC1CCCC1)C(=O)NC(C)CCCCNC(=O)CC1CCCCC1 25125,c1(OC)cc(F)c(F)cc1C(N1CCCN(C(C)C)CC1)=O 25126,c1(OC)ccc(C(=O)N(C)CCNC2CC2)cc1S(=O)(=O)NC(=O)C(C)S(N)(=O)=O 25127,C(=O)(C(C(C)(C)C)NC(=O)C(C)C)NCCC1(NC(CCC(C)OC)=O)CCC1 25128,C(=O)(C(C)(C)C(O)CC)N1C2C(NC(c3cccc(CC)c3)=O)CC(C2)C1 25129,c1(C(=O)NCCN(C(c2cc3ccccn3n2)=O)CC)ccc([N+](=O)[O-])cc1Cl 25130,C1(CNC(C2(C(C)(F)F)CCC2)=O)CCCN(C(=O)C=CC2CCOCC2)CC1 25131,CCCC(C(=O)NC1CCCN(C(c2ccc(F)c(C(F)F)c2)=O)C1C)C(C)C 25132,Cc1nn(C2CC2)c(C)c1C(=O)NCC(C)(C)OCCNC(=O)CCC1(C)CC1 25133,CC1CCC(NC(c2ccc(C#N)n2C)=O)CN1C(c1cnc(C(F)(F)F)s1)=O 25134,C1(C(N2C(CNC(c3c(C)ccc(OC)n3)=O)C=CC2)=O)CC2(CCOCC2)C1 25135,N1(C(CCC(=C)C)=O)CCCC(CO)(NC(=O)CCSc2ccc(C#N)cc2)C1 25136,C12(CNC(C3CC(CC)C3)=O)CC(C1)C(NC(=O)C=Cc1nccn1CC)CO2 25137,CC1(C)C(C(N2CC(CNC(=O)C(c3ccccc3)O)C2)=O)CCS1(=O)=O 25138,c1(C(C2(OC)CCOC2)NC(CCC)C2CCCC2)nnnn1CCC1CC1 25139,CC1CN(C(C)C(C)O)CC(c2ccc(F)cc2)O1 25140,C1(C(=O)NC23CC(C(N4C(CN(C)C)CCCC4)=O)(C2)C3)CC2CC1CC2O 25141,c1(C(N2CCCC(CCNC(C(COC)O)=O)C2)=O)cc(C)cc(Cl)c1 25142,C1=C(CNc2nc(C3CC3)co2)CCC1 25143,C1(C(=O)NC(C2CCN(C(CC(C)C)=O)C2)C)Cc2ccccc2N1C 25144,c1(OCC)ccc(C2(C(=O)NCC3C=CCN3C(=O)CC(C)OC)CCC2)cc1 25145,c1(OC)csc(C(N2CCOC(CNC(C3CCCC3C)=O)C2)=O)c1OC 25146,c1(C(=O)NC(C(C)NC(c2ccn(C3CC3)n2)=O)C)c(F)cccc1Cl 25147,c1(OC)cnc(F)c(C(=O)N(C(C)CNC(c2cncc(C(=O)N(C)C)c2)=O)C)c1 25148,S(=O)(=O)(c1cnn(C)c1)N1CC(C(=O)NCC(C)CN(C(=O)C(C)C(F)F)C)C1 25149,CCC(C)CC(=O)C(=O)N(CCC(=O)NC(C1CSC1)C)C 25150,CC1(C)CCCOC1CC(=O)NC1(C)CN(C(=O)C(c2ccccc2F)O)C1 25151,N1(C2CC(C(=O)OC)C2)CCCCC(NCC(N2CCN(C)CC2)C)C1 25152,C123CCN(CCC1C2)C3=O.C1(C)(CC=C)CNC1.C12(CC=O)CCCC1C2 25153,C1(CCNC(CCCOCCOC)=O)CCCN(C(=O)Cn2cnnc2)CC1 25154,CC(C(=O)NC1CC(C(F)(F)F)CN(c2ncccn2)C1)S(N)(=O)=O 25155,N1(C(CCOC(C)C)=O)CC2CCC1C1CN(C(c3ccnc(CO)c3)=O)CC21 25156,CCCCCCCC(=O)NC1C(C)CCN(C(=O)COc2ccc(O)cc2)C1C 25157,CC1CCN2N=C(C(=O)N3CCCC(CNC(=O)COCCCF)CC3)NC2=N1 25158,c1(C(=O)NCCCCNC(c2cncc(OC)c2)=O)cc(C)c2c(c1)CCCN2 25159,c1(OCC)ccc(C2(CNC(c3n(CC)nnn3)c3ccon3)CC2)cc1 25160,N1(C(CN(C(=O)CCC2CC(C)C2)CC)=O)CC(CO)OCC1C 25161,C1(CNC(CC=C(C)C)=O)CN(C(=O)C(C2CCCCCC2)C)CC12CCC2 25162,C(=O)(CC(C)CC(C)(C)C)NCC1=CCN(C(c2c(NC(C)=O)cccn2)=O)CC1 25163,N1(C(C(C)OCCC=C)=O)CCCC1C=CC(=O)NCc1ccc(C)cc1 25164,Cc1noc(C(C)C)c1C(=O)NC1CCCC1CNC(=O)CC1CCC=CCC1 25165,N1(C(CC(C)NC(CCC)=O)=O)CCCC(C(C)C)CC1 25166,c1(C(C)NC(CCN(C(C(COC)OC)=O)CCO)=O)ccncc1F 25167,N1(C(C(C)n2cnnn2)=O)CC2CCCC(C1)N2C(c1cnc(F)c(F)c1)=O 25168,c1(CC(=O)N(N2CC(C)CC(C)C2)CCOC)ccc2ccccc2c1 25169,c1(CN2CCC(CC(=O)N(c3ccsc3)C)CC2)ccc(Cl)cc1 25170,C1(=CC(=O)NC(C)C(C)NC(=O)CCC23CCC(CC2)C3)CN2CCC1CC2 25171,CC1CCN(C(C2(O)CC2)=O)CC1NC(c1coc(-c2ccccc2)n1)=O 25172,C#CCCC(O)C(=O)NCC(c1ccccc1)N(C(=O)Cc1sc(C)nc1C)C 25173,Cc1scc(CNC(=O)C(C2(O)CN(C(c3ccn(C)c3)=O)C2)F)c1C 25174,c1(OC)ncc(C(=O)N(C(C)CN(C(=O)C(O)C2CC2)C)C)c(C)n1 25175,O=S(=O)(c1cnn2ccc(=NCCN3CC4CC4C3)[nH]c12)N1CC(CF)C1 25176,C(=O)(N=c1[nH]nc(SCC(=O)OC)s1)NCCOCCOC 25177,c1(CNC(c2nc(C)oc2)=O)cc2n(n1)CCN(C(=O)C(C)CC1CCC1)C2 25178,CCCC(C(=O)N1CC(O)(CCNC(=O)C(=O)N=S(C)(C)=O)C1)S(N)(=O)=O 25179,CC(CC(F)(F)F)C(=O)NCC#CC(N1CCC(C)(CCO)C1)=O 25180,CC1CC(C(C)(C)C)CCN1C(=O)NCCNC(=O)CCCCO 25181,CCC(C(=O)N1CC(CNC(=O)CC2CCOC2=O)C1)N(C)C 25182,N1(C(c2c(C)cco2)=O)CC(CNC(C2CCC(C(N)=O)C2)=O)OC(C)(C)C1 25183,N1(C(C(C2(OC)CCCC2)(F)F)=O)C2CCCC1CC(NC(=O)CSC(F)F)C2 25184,Cc1[nH]nc2cc(C(N3CC4CC3CN4C(C3CC(=O)N(OC)C3)=O)=O)ccc12 25185,C1(C2CC2)(C(N2C(CC=C)CCCC2)=O)CN(C(C2C(C)(C)C2(C)C)=O)C1 25186,CC1CCN(CC2CCN(C(=O)OC(C)(C)C)C(C)C2)CC1C 25187,C1(C)(C(=O)NCC(C)CN(C)C(C2CC(C)(C)C2)=O)CC(F)(F)C1(F)F 25188,C=CC(C)(C)CC(=O)N1CC(F)CC1CNC.C1(=O)CN1.C(=O)(NC1CC1)NC 25189,N1(C(C(C(=O)OCC)OC)=O)CC2CCCC2C1C(=O)NC1(C(=O)N(C)OC)CC1 25190,C1(CC(=O)NC2CN(C(c3ccc(C)o3)=O)C2)COCCOC1 25191,C(=O)(C(C)CC(N)=O)N1CCC(C(=O)N(C)CCc2nccs2)(CC)C1 25192,c1(C(C)(C)C)ccc(SCC(=O)NCC(O)CNC(C2(C)C=CCC2)=O)cc1 25193,C(N=c1[nH]c(=NC2CCSC2C)c2cc(OC)ccc2[nH]1)c1c(CC)nn[nH]1 25194,C(CC(C)N=c1[nH]c(N2CCC(Cn3ccnc3)CC2)nc2c1CC(C)CC2)SC 25195,C=C(C)C1CN(C(C2CCC3(CC3)N2C(=O)C(O)C(C)(C)CC)=O)CCO1 25196,N#Cc1cc(-c2cnn3c2OCC2(CC2)C3)cc(S(N)(=O)=O)c1 25197,C(c1ccc(F)c(F)c1)=CC(=O)NCCCCC(C)NC(=O)C(C)CC1CCC1 25198,Cc1nc(C(=O)NCC(O)CNC(=O)C(C)(C)C(N)=O)ccc1[N+](=O)[O-] 25199,N1(C(CC(C)n2ccnc2)=O)CCSCC1C 25200,Cn1ncc(Cl)c1C(c1nnnn1-c1ccon1)NC(=O)NC1CCC1CO 25201,c1(NC(N2CC(NC(C(C)Cc3ccco3)=O)C2)=O)cccc(Cl)c1Cl 25202,C(=O)(CCCCNC(c1cnnn1C)=O)N(CCN=[N+]=[N-])C 25203,Cc1cc(O)cc(C)c1C(=O)NC(C)CCNC(=O)C(N1CCC(O)CC1)C 25204,C1(C(=O)NCC(CNC(C(C=C)OC)=O)(C)OC)CN(C)CC(C)O1 25205,C(=O)(C(CCCC#N)N(C)CCNC(=O)CCC(C)OC)NCC(C(=O)NC)(C)C 25206,Cn1ncc(Cl)c1C(=O)NCCC1CCCN1C(C1CN(C2CCOCC2)C1)=O 25207,C1(C)(COC)CCN(C(C2CCCCCN2C(=O)CC(C)OC)=O)CC1 25208,N1(C(C(C(C)C)O)=O)CC2(COC(CNC(C3C4CCC(C4)C3(C)C)=O)C2)C1 25209,C(CC(C(=O)NCC1C(N(C)C)CC1O)OC)NC(C1CC(=C)C1)=O 25210,CC1CC(CNC(c2cscn2)=O)CN1C(c1cccc(-n2ccnc2O)c1)=O 25211,C(CCOC)(C(=O)NOCC(O)C(C)(C)C)NC(c1n(CC)nc(C)c1)=O 25212,C1(OC)(CNC(C23CCN(CC2)C3)=O)CCN(C(=O)CN2CCC(C)C2)C1 25213,C(C)(C(=O)N1CC(C(C)NC(c2coc(C(F)F)n2)=O)C1)(C(C)C)OC 25214,C(=O)(C(C(C)(C)C)N(C)C)NC(C(C)C)(C)CNC(=O)Cn1ccnc1C(C)C 25215,C(C(CC(=O)NC1CCC(=O)NC1)NC(c1cc(OC)n[nH]1)=O)OC 25216,CC(=O)CCC(=O)NC(Cn1ccnn1)C(N1CCC(F)(CO)C1)=O 25217,c1(C(=O)NCC)ccc(=NCCCNC(c2nccc3ccccc23)=O)[nH]c1 25218,c1(C(N(CCN(C(C(C=CCCC)O)=O)C)C(C)C)=O)cc(OC)nn1C 25219,CCC1=C(C(=O)NC2CCN(C(C3C=C(C)CS3)=O)C2C)CCCO1 25220,CON(CCO)C(=O)CC(C(F)F)NC(=O)C(C1CCOCC1)F 25221,C1(C(=O)NCC(CNC(C(N2CCC(O)CC2)C)=O)O)CCCCC1(F)F 25222,c1(C(=O)NCC#CCNC(c2c(C(C)C)n(C)nc2)=O)cc(Cl)c(Cl)cc1O 25223,C(c1ccccc1)=CCOCC(=O)NCC(CN(C(C(C=C)O)=O)C)C 25224,CS(=O)(=O)c1ncc(C(=O)NCC2CN(C(=O)Cn3ccnn3)C3CC23)s1 25225,C1(CC(=O)NCC2(CO)CCC2)CC2CCC1N2C(c1cnc2n1CCC2)=O 25226,C1(NCc2cn(C)nc2Cl)CC(O)C12CC(F)(F)C2 25227,Cc1ncccc1C(=O)N(CC(C)(C)C(=O)NCC1(n2nccn2)CC1)C 25228,Cc1c(F)ccc(C(=O)N(C2CCCC(NC(c3c(C)n[nH]c3C)=O)C2)C)c1Cl 25229,c1(CC(N2CC(NC(CC(CCC)O)=O)C3(C2)CC3)=O)c[nH]c2cccc(Cl)c12 25230,N1(C(C(C)(C)F)=O)CCC2C(CCN2C(=O)C(C)(O)C(F)(F)F)C1 25231,c1(CC)ccc(C(N2CCC(CCNC(c3cn(CC)nn3)=O)C2)=O)c(O)c1 25232,CCC(CC)CCC(=O)NC1C2CC1N(C(=O)C(C)CC(N)=O)C2 25233,C(=O)(CN=S(C)(C)=O)NC1CC(OCC(=O)N(c2cnn(C)c2)NCC)C1 25234,c1(CN2CC3N(C(c4c(OC)cncc4)=O)C3C2)c(C)cc(C)cc1C 25235,c1(COC)cc(C(=O)NC(C)(CNC(=O)Cc2nccn2C)C2CC2)no1 25236,O=C1COc2cccc(S(=O)(=O)NCCc3csc4ccccc34)c2N1 25237,c1(C(=O)NCC2N(C(C(n3ccc(C)n3)C)=O)CCC2)ccc(C)cc1[N+](=O)[O-] 25238,c1(C(N(CC(CC)NC(=O)CCCCN(C)C)C)=O)cc(O)n(CC)n1 25239,C1(CC(=O)N(CC(C)CNC(c2ccco2)=O)C)(CNC(C)=O)CCCCO1 25240,N1(C(Cc2cc(C)sc2C)=O)CC2(CCN(C(c3cc(F)ccc3Cl)=O)C2)C1 25241,C1(C(C)NC(=O)CSC2CC2)CCCN1C(=O)CCCc1ncco1 25242,N1(C(C(C)(C)n2cccn2)=O)CCC2(CCC2)CC1 25243,C#Cc1cccc(CNC(=O)CC(C)CNC(=O)CC=CC=C)c1 25244,C1(NC(CN2C(=O)CN(C)C2=O)=O)CCC2(CC1)CC2Nc1ncncc1Cl 25245,C(=O)(C(CC(C)C)C(N)=O)NCCCN(C(c1ccc(CC)cc1F)=O)C 25246,c1(CCC)cc(NC(=O)Nc2ccc(-c3cc(OC)ccn3)s2)n(C)n1 25247,C1(CCC)CCCCN1C(c1cnc(-c2ccc(Br)cc2)s1)=O 25248,N1(C(C2CC(CNC(=O)C=CCn3cncn3)OC2)=O)CCC(O)CC1C1CC1 25249,C1(N(C)C(=O)NCC(c2cnn(C)c2)O)CC2(C1)CC2NC(=O)OC(C)(C)C 25250,CC1(C)CCCC(O)(C(=O)NC2CN(C(c3nscc3Br)=O)CC2O)C1 25251,C(C)(CCCNC(c1csc(C(F)(F)F)n1)=O)NC(C1CC(SC)C1)=O 25252,N1(CC(=O)N(CCC(C(C)C)NC(=O)C=C2CCOCC2)C)CCCCS1(=O)=O 25253,CC1CCN2C1c1cn(nn1)-c1cccc(c1)C2=O.C1(CNC)CCCC1(C)O 25254,C1(O)(CNC(c2c(C)snn2)=O)CCN(C(c2cccc(Cl)c2)=O)CC1 25255,C(N=c1nc2sccc2c(NCc2ccccc2)[nH]1)C1(Cl)CC12CCC2 25256,CCC(CC)C(C)C(=O)N1CC(CNC(=O)CCc2ccc(N)c(F)c2)C(C)C1 25257,C1(C(=O)NCCOC2CCN(C(=O)C(F)n3ccnc3)C2)CC2(C1)CC21CC1 25258,Nc1cc(C(N2CCC(CF)(NC(=O)Cc3ccc(F)c(Cl)c3)C2)=O)cc(N)c1 25259,N1(C(=O)OC(C)(C)C)CC2(CCCC2)CCC1Cc1cnccc1Cl 25260,C1(C(=O)NCC(CN(C)C(c2ccnn2CC#N)=O)O)CCC(C)CC1 25261,C#Cc1cnn(CC(=O)NC(CCOC)C(=O)NCC(N2CCCC2)C)c1 25262,n1(C(C(=O)NC2CCC(F)(CNC(C(C)=CC)=O)C2)C)cnc2ccccc12 25263,C(C)(CN=c1nn[nH]n1Cc1ccccc1)NC(C(F)(F)C1(OC)CCC1)=O 25264,C12(CCNC(=O)CC3CC(NC(C4CCCO4)=O)C3)CC(CO1)C2 25265,C1(COCCN(C(=O)NCC(=O)NOCCF)CCO)CC12CCCC2 25266,c1(CNc2ccc(-c3ccc(OC(C)C)nc3)cc2)scnc1C1=CCNCC1 25267,N1(C(c2cnc(CC)s2)=O)C2CCC1CC(N(C)C(c1cc(C)ncc1C)=O)C2 25268,CCC(CNC(C1CC2(CC2)CO1)=O)(CC)NC(C1CC2CCC2C1)=O 25269,N1(C(CCNC(=O)OC)=O)CC2(CCC(NC(=O)C(C)C(O)CC(C)C)CC2)C1 25270,Cc1nn(C)c(N)c1C(N1CCC(OCC(=O)NC(C)C(O)C(C)C)C1)=O 25271,C(=O)(CC(C)(C)C(C)(F)F)N(CC(C)NC(c1ccc(NC(N)=O)cc1)=O)CC 25272,c1(C(=O)NC(C(C)(C)NC(C=CC)=O)C)ccc(C2(CC)CC2(F)F)cc1 25273,CCCC(CC(C)C)C(=O)N1C(C(=O)NCCC(=O)OC(C)C)C2CC(O)C1C2 25274,C1(N(C)C)CN(C(=O)COc2cncnc2)CC1O 25275,N1(CC)CC(NC(C2(F)CCN(C(c3nc(Cl)cs3)=O)C2)=O)CCC1=O 25276,CCCCC(O)C(=O)NC1(CCNC(c2[nH]ccc2C2CC2)=O)CCCC1 25277,Cn1cc(C(=O)NCC(C2CCC2)NC(=O)CCC(N)=O)c(-c2ccccn2)n1 25278,S(=O)(=O)(c1c[nH]ccc1=NC1COCC(C)(C)C1)N(CC(CC)C)CC 25279,C1(NC(c2n(CC=C)nnn2)c2cc(C)on2)CCn2nnnc2C1 25280,C1(C(=O)NC2(CN(C)C(C34CCC(C3)C4)=O)CC2)CCCC2(CCCCC2)C1 25281,c1(C(N2CCC(NC(COCC#C)=O)C(O)C2)=O)cc(C)c2[nH]nnc2c1 25282,CC1CC(C(=O)NCCC2CC(NC(=O)C3=CCCCO3)C2)CC(C)C1 25283,C12=CCOCCCC(=O)N(CC1)CC2.C1(CCC(=O)NC(C)(C)C)CCOCC1 25284,c1(C(C)(C)C)[nH]cnc1C(=O)NCC(C1CC1)NC(c1cn(CC(F)F)cn1)=O 25285,CC(C)C(C)(CNC(C1SCCS1)=O)NC(=O)Cc1csc(-c2ccoc2)n1 25286,c1(C(N2CC3CC(C(=O)NC45CC6CC4C5C6)CC2C3)=O)cc2n(c1)CCCC2 25287,C1(NC(C2CC23CCC3)=O)CCC(O)CN(Cc2ccc(-c3csnn3)cc2)C1 25288,N1(C(c2c(C)c[nH]c2)=O)CC2CCCC(C1)N2Cc1cc(Cl)ccc1F 25289,C1(N(C(c2cc(C)oc2)C(=O)N(C)C)C(C)C)CCCN(CC2CCCO2)C1C 25290,CC(C)CC(O)CC(=O)N1CC(NC(C2CCC(=O)N(C)C2)=O)C(O)C1 25291,c1(C(=O)NCCCCNC(C2(Sc3cscn3)CC2)=O)cccc(C(F)(F)F)c1 25292,c1(C(N(CCNC(c2ccc(Br)o2)=O)CC)=O)ccncc1Br 25293,C1(C(=O)NC(CNC(=O)CCCn2ccnc2)C(C)C)(CSC)CCN(C)CC1 25294,c1(CCC)cc(C(=O)NC2CN(C(=O)CCC(=O)OCC)CC2C)ccn1 25295,C1(CC(=O)NCC2C(NC(CN(C)CCO)=O)CCC2)CCC(F)(F)CC1 25296,N1(CCN(C(CC)=O)CCN(C)C)CCC(NC(=O)C(F)(F)F)CC1 25297,C1(C2CC2)(C(=O)NCC(C(C)C)OC)CN(C(=O)C=Cc2cn(C)nn2)C1 25298,Cn1ncnc1CCC(=O)NS(Cc1c(Cn2ccnc2)ocn1)(=O)=O 25299,c1(SC)c(C(N(c2ccc(C(C)C)cc2)CC2CNC2)=O)cnn1C 25300,c1(C(=O)NC2CC(N(C(C34CC(C(C)C)(C3)C4)=O)C)C2)cn(C)[nH]c1=N 25301,C1(NC(c2ccn(C)c2)=O)CC(NC(c2nnc(S)n2C)=O)C12CCC2 25302,N1(CC)CC2CC1CN2C(C1(CCNC(c2cscc2Cl)=O)CCCC1)=O 25303,C1(NC(CC(C)c2ccco2)=O)COC2(C1)CN(C(=O)CC1CC(F)C1)C2 25304,C(C)(CSC)(C(=O)NOCC(=O)N(C)C)NC(c1cccc(CC)n1)=O 25305,Cn1ccc2cccc(C(=O)NC3(C)CCN(C(c4sc(F)cc4Cl)=O)C3)c12 25306,C(CCN(C)C(c1c(C)noc1C)=O)(C(C)(C)C)NC(c1cncc(C)n1)=O 25307,C1(=O)CCCCCCNC(=O)c2coc(n2)CO1.Cc1ncncc1C(=O)O 25308,CCCCC(C)CCC(=O)NC(COC(C)C)C(=O)N(C(CO)C1CC1)C 25309,N1(C(C2N(CC)CCC2)=O)CC(C)(C)C(NC(C2CCOCC2)=O)C(C)(C)C1 25310,N1(C(=O)NC2CC(SC)(CO)C2)CCC2(CC1)CC2NC(=O)OC(C)(C)C 25311,c1(NC(CC2CCCN(C(C(CC=C)C)=O)C2)=O)ccc(Cl)nc1C(N)=O 25312,c1(C(N(CCNC(C=C(CC)C)=O)CCOC)=O)cccc(F)c1Br 25313,CCC(O)C(F)(F)C(=O)NCC(C1CCN(C(c2ccncc2F)=O)CC1)C 25314,C1(CC)C(C(=O)NC2CCN(C(=O)CCCn3nc(C)nc3C)C2C)CCN1C 25315,C12(CC(N3CCC4CN(C(CC=C)=O)CC4C3)=O)CC3CC(C)(C1)CC(C)(C3)C2 25316,C(=O)(C(C)C(O)C(C)C)N(CC(COC)C)C.C(=O)(C(C)(C)C1CCCC1)O 25317,N1(C(CC)=O)CCC(c2nc(-c3ccccc3C)nn2Cc2cccs2)CC1 25318,c1(C(=O)NCC(C)NC(C2(F)CCOCC2)=O)nc(Br)c2c(F)cccn12 25319,N1(C(CCc2ccc(C)o2)=O)CCCC2CN(C(=O)C(C)(C)C(C)(C)O)CCC12 25320,S(=O)(=O)(c1cccc(Cl)c1F)NC1CCC(C(=O)NCc2ccc(O)cc2)OC1 25321,c1(NC(=O)Nc2cn(C)nc2-c2cccc(F)c2)ccc(F)c(NC(N)=O)c1 25322,N1(CC(=C)C)CCC(NC(=NCC2CC2)NCC2CCC2)CC1 25323,C(CC(=O)NCC(C)CN(C(=O)CCc1ncco1)C)OCCC 25324,C1(F)(CNC(=O)Cc2c[nH]nc2O)CCCN(C(C2(CC3CC3)CCCO2)=O)C1 25325,c1(C(N2C3CN(C(C4(C=C)CC4)=O)C(C3)C2)=O)cc2ccc(OC)cc2s1 25326,C(CCCCC(=O)NCC1CCCC(C)(C)C1)N(C(=O)C1=CCCCC1)C 25327,CC1(C)CN(C(=O)CCc2cn[nH]c2)CCN(C(c2c(O)cc(F)cc2F)=O)C1 25328,C(=O)(C1=C(C#N)CCC1)NC(C1CCCN(C(c2c(C)nc(N(C)C)s2)=O)C1)C 25329,c1(C(N2C3C(NC(=O)CCC4CCCO4)C(C3)C2)=O)n[nH]c2c1CCC2 25330,C1(NC(C(C)OCC(C)C)=O)CC2CC(C1)CN(C(C1(O)CC(C)(C)C1)=O)C2 25331,O=C1CC2CN(C(C3CCCN(C(=O)Cn4ccnn4)C3)=O)CC2CN1 25332,C=C(F)C1(CC(=O)NC2CCCCC2N(C(=O)C(C)OCCC(C)C)C)CCC1 25333,n1(CC)cc(Br)cc1C(=O)OCc1nnc(C2CC2)o1 25334,Cn1cc(Cl)c(C(N2CC(O)(CCNC(C34COCC3C4)=O)C2)=O)n1 25335,C1(CC)CCN(C(c2[nH]ccc2CNC(=O)CCCCSC)=O)C1C 25336,c1(CN2CCN(c3nc(SC)c(Br)cn3)C(CCO)C2)cc([N+](=O)[O-])ccc1O 25337,C1(C(C)O)CCC(NC(C2CCC(C(C)C)N2C(c2ccc(Cl)cn2)=O)=O)CC1 25338,N1(C(c2c(C)nsc2)=O)CCC(C)C(NC(C2(F)CCCCC2)=O)C1C 25339,N(C(=NCCc1cnccc1OC)NC1CC1C1CCC1)CCC(=O)NC 25340,c1(C(N2CC(C)C(NC(=O)COCC(F)F)C2)=O)cccc2ccnn12 25341,C#Cc1c[nH]nc1C(=O)NC(C)CC(C)NC(=O)Cc1ccc(F)cc1 25342,C1(NC(C(COC)COC)=O)CC2(C1)CC(NC(c1ccccc1OC)=O)C2 25343,C1(CC)(NC(c2cc(Cl)no2)=O)CCCN(C(=O)CCc2cncnc2)C1 25344,Cc1nc(N(C)C)sc1C(=O)NC1CCC(CCNC(C2(O)CCSC2)=O)C1 25345,C=Cc1cnn(C)c1C(=O)NCc1cccc(NC(C2(C)CCC(C)C2)=O)c1 25346,C1(NC(C(C)N(C(C)=O)C)=O)CC(C(=O)N(CC(c2nn[nH]n2)C)C)C1(C)C 25347,C1(C(N2C(C3(NC(COCCC)=O)CC3)CCC2)=O)CC(=O)N(CC(F)(F)F)C1 25348,CCCCCC(O)CC(=O)N1CCOC(CNC(=O)CC2CC=CCC2)C1 25349,c1(CN2CCC(N(CCOC)C=O)C2)cccc(OCC2CCOC2)c1.C1CC1 25350,C(=O)(C(CNC(C1CC1(F)Cl)=O)N(C)C)N(CCCCO)CC 25351,C1(NC(c2ccc(OC)o2)=O)CC2CC1CN(C(=O)Cc1ccc(F)cn1)C2 25352,c1(NC(C2CC2Cc2ccccc2)=O)cnn(Cc2ccccc2)c1 25353,c1(CC)nc(C(N2CCC(CCNC(C3(C4CCCCO4)CC3)=O)C2)=O)co1 25354,N1(C(Cc2c(C)cccn2)=O)CCCC(N(C)C(c2cc(N)cc(F)c2)=O)CC1 25355,Cc1ccc(C(=O)NCC(C2CCCC2)NC(C2CN(C)C(=O)N2)=O)cc1C 25356,c1(N2CC(C(=O)Nc3cc(C(=O)OC)ncc3)SCC2)ncnc2cnccc12 25357,c1(C(=O)NC(CCNC(C(C)SC(C)C)=O)C)ccc2c(c1)NC(=O)CN2C 25358,N1(C(C(CNC(c2cnn(C)c2Cl)=O)CC2CCCC2)=O)CCC(O)(CO)CC1 25359,c1(Sc2c(C)cc(C3CC3)cc2)nc(S(C)(=O)=O)nc2c1ncn2C 25360,N1(C(CC(C)C2CC2)=O)CC(C(N2CC(N3CCCCC3)C2)=O)CC12CCC2 25361,c1(C(N(C(C(N2C(C)(CC)CC2)=O)C)C2CC2)=O)nc(C)ccc1C 25362,C1(CNC(CC(CCOC)(C)C)=O)CCC2CN(C(=O)C3=CCCO3)CCC2C1 25363,C(=O)(C(CNC(=O)Cc1cncn1C)N(C)C)NCC(N(C)C)C1CC1 25364,S(=O)(=O)(c1ccc(Nc2cccc(OCF)c2)c(Cl)c1)N(C(CC)(C)C)CC(F)CO 25365,c1(C(=O)NC(CNC(c2c(SC)cc(F)cc2)=O)(C)C)cc2ccc(F)cc2o1 25366,C(=O)(C1OCCc2cc(Br)ccc21)NCCNC(c1c(OC)scc1)=O 25367,c1(OC)c(NC(c2cnn(CCN(C)C)c2)=O)cccc1C(=O)O 25368,C1(NC(C2(CC#C)CC=CCC2)=O)COC2(C1)CN(C(=O)Cc1cccnc1)C2 25369,C(=O)(C1CCCc2nncn21)N1C(CNC(C2CC2(Cl)Cl)=O)CC2(CC2)C1 25370,C1(CNC(C(C)OC2CCCC2)=O)C(C2CC2)CCN1C(=O)CC(C)(F)F 25371,Cc1ccc2c(c1)C(C(=O)NC(C)CNC(c1ccc(CO)cc1F)=O)C2 25372,CC1(C(N2CCC(C)(NC(c3cc(F)cnc3O)=O)C2)=O)CCCCC1(F)F 25373,Cc1cccc2[nH]cc(C(=O)NCC3CC3NC(c3nnc(O)nc3O)=O)c12 25374,C1(NC(c2[nH]cc(CC)n2)=O)CCC2(CCN(C(=O)CC(C)CC(C)(C)C)C2)C1 25375,c1(C(C)N)ccc(N(CC(=O)NCCCC#N)C(=O)CC)cc1 25376,Cc1cc(C(N2CCC(N(CCO)C(c3cn[nH]c3)=O)C2)=O)n2ncnc2n1 25377,c1(-c2ccc(C(N3C(CCCNC(C=C(C)C)=O)CCC3)=O)s2)cccc(F)c1 25378,Cc1cccc(OCC(=O)NC(CNC(=O)C2=CCCSC2)CO)c1C 25379,C1(O)(CCNC(c2n[nH]cc2F)=O)CCCN(C(c2sccc2C(F)F)=O)C1 25380,C1(NC(C(CC=C)OC)=O)CC(NC(C23COCC(C2)C3)=O)C12CCC2 25381,C1(Cn2cnc(C(N)=O)n2)CCN(C(=O)Cn2cccn2)CC1.c12cn(nn1)C2 25382,c1(CC(=O)OCC)cc2n(n1)CCN(C(=O)CN1CCCNS1(=O)=O)C2 25383,C1(F)(CNC(=O)C(F)=CC2CC2)COCCN(C(c2ncsc2C2CC2)=O)C1 25384,n1(CCNC(=O)NCC2(C)C(C)(C)C2)ccn2nccc2c1=O 25385,O(NC(=O)C(CC(N)=O)NC(c1csc(C#N)c1)=O)CC(=C)Cl 25386,C1(C)(CCCC(=O)NC(C2(O)CN(C(CC=CCC)=O)C2)C)NC(=O)NC1=O 25387,c1(C(=O)NC(CNC(C(CC)F)=O)(C)CO)cccc(NCC)c1 25388,c1(-n2cc(CNC(c3ccc(C(CC)C)cc3)=O)nn2)cc(C)c(F)cc1Cl 25389,N1(C(c2ccc(C(C)C)s2)=O)CCC12CN(C(=O)CC13CCCC1C3)C2 25390,CC1(CNC(=O)CCC2(NC(=O)C=CC(=O)N(C)C)CCCC2)CCCCC1O 25391,c1(C(C)=O)ccn(C(c2cn(CCN(C)C)nn2)C(C2CC2(C)C)CC)n1 25392,N1(C(C2CC(C(=O)OC)C2)=O)CCC(C)C1c1ccc(C(F)(F)F)cc1 25393,C1(SCCOCCNC(CCOCCCNC(COC)=O)=O)(CO)CCCCO1 25394,C1(CN(C(CC=CCCCCC)=O)C)C2CN(C(c3cc(Cl)cn3CC)=O)CC12 25395,C(CCC(C(=O)NCCc1cccc(C)n1)NC(=O)CC1CCOC1(C)C)OC 25396,C#CC1CN(C(=O)CC2CCC(C)(C)O2)CCN1C(c1nnsc1SC)=O 25397,N1(CC)CCC(CNC(=O)CC2C=CC(NC(=O)C=C3CCOCC3)C2)CC1 25398,N1(C(CCSCC)=O)CCOC2(CCN(C(=O)CN3C(=O)CNC3=O)C2)C1 25399,c1(SC)nc(N2CCN(CCN(C(=O)CC(C)C)C)CC2)ncc1C 25400,C(C(CC(=O)N1CCC1c1cccnc1)C1CCC1)NC(=O)C(C1(O)CCCC1)F 25401,C1(CNC(c2c(C)nn[nH]2)=O)CC(F)CN1C(c1sccc1CO)=O 25402,C1(O)(CCNC(C2CC2c2ccncc2)=O)CCCN(C(C2(F)CCC2)=O)C1 25403,N1(C(Cc2c(C)scc2)=O)CCC(C2CCCN(C(=O)C(C)(F)F)CCC2)CC1 25404,c1(C(=O)NC2CC(CCNC(CC(COC)C)=O)C2)cnn2ccccc12 25405,C(=O)(CC1=CCOCC1)N1CC(C)C(CC(N2CCN(C)CC2CO)=O)C1 25406,c1(C(=O)NC2CN(C(C(CCC)N(C)C)=O)C2)ccc(C(C)C)cc1F 25407,CC1(CNC(=O)Cc2ccccc2Cl)CCN(C(C2(C)CCCC2O)=O)C1 25408,c1(C(=O)NCCCC(C)NC(CCCCCC)=O)sc2cc(CC)ccc2c1Cl 25409,Cc1cc(C(=O)NCCCN(CC2CCCC2)C)sn1.C(=O)(CCCC1(C)N=N1)N 25410,C(=O)(CCCCC(C)(C)C)NC(C(C(C)C)NC(=O)C=Cc1ccc(F)cc1)C 25411,N1(C(c2ccc(CC)[nH]2)=O)CC(C)N(C(=O)COCCc2ccccc2)CC1C 25412,CC(C)(CS(C)(=O)=O)C(=O)NCCC1CCN(C(=O)Cn2ncnn2)CC1 25413,C1(C(NOCc2cn(CC3CCC(=O)O3)nn2)=O)CC2CCCC2C1 25414,CC(CC(C)NC(=O)CCCF)NC(=O)C(CC1CC1)NC(=O)OC(C)(C)C 25415,C1(COC)CCCCN1C(=O)CCN(C(=O)CCc1ccc[nH]1)C(C)C 25416,CC(C)(F)CCC(=O)NCC1(C)CCCN1C(C1COC(=O)O1)=O 25417,CCCCS(=O)(=O)CC(=O)NC1(CNc2ccncc2[N+](=O)[O-])CCCC1 25418,C1(C(N(CC(C)NC(c2cnc(CSC)s2)=O)CC)=O)CNC(=O)N1C 25419,C=CCC(C)(C(F)F)NC(=O)CCn1cc(-c2ccc(C)cc2C)nn1 25420,C1(NC(c2ccn(CCOC)n2)=O)CN(C(=O)CNS(=O)(=O)C2CC2)CC1C 25421,S(=O)(=O)(c1ccc(OCCBr)cc1O)CC1(NCc2ccc(OC)nc2)CCC1 25422,Cc1cc2[nH]c(C(=O)NCC(C(C)C)NC(=O)CCCCCN(C)C)cc2o1 25423,c1(C(=O)NC(=O)C=CC(=O)NC(C2CCCC2)CC2CC2)cn(CC(F)F)cn1 25424,N1(S(CCOC)(=O)=O)CCC(C(=O)Nc2cnn(C(C)(C)C)c2)C(O)C1 25425,N1(C(c2n(CC#C)cnn2)=O)CC(CNC(C2(C)CCCCC2)=O)CC12CCC2 25426,N12CCN(CC1)CC(C)NC2=O.C1(NC(CC=CCC)=O)CCC(C)CC1 25427,n1(CC(=O)NCCCN(C(=O)C(O)CC[S+](C)C)C)c(O)nc2ccccc12 25428,c1(C(=O)NCCC2OCCCN(C(CC(CC)(F)F)=O)C2)cc(S(N)(=O)=O)c[nH]1 25429,c1(CN(C(=O)NC(c2cccc(F)n2)C)C)cccc(Cl)c1Cl 25430,Cc1cc(C)c(C(=O)NCCC2CCN(C(=O)C(c3ccccc3)O)C2)s1 25431,C1(C(=O)NCC(CNC(C2CCC(OC)C2)=O)(C)C)C2CCC3(COC(=O)C13)O2 25432,Cc1cnc(C(N2CCC(C)C(NC(c3cccnc3O)=O)C2)=O)c(F)c1 25433,C(=O)(C(C(C)O)NC(C)=O)NC(CC)CNC(=O)C(C)c1ccon1 25434,C1(Nc2ccc(Oc3c(OC)cccc3)cc2)CCC(=O)N(C(C)C)C1 25435,C1(C(N2CCC(N(C(=O)CCCCc3ccccc3)C)C2)=O)CCC(C)(F)CC1 25436,Cc1nsc(C(N2CCCCC2CC(=O)NC(C2CC(F)(F)C2)C)=O)c1N 25437,N1(C(C2C(CNC(c3c(COC)cc[nH]3)=O)CC2)=O)CCCC(C(C)C)C1 25438,Cc1nc(NCC(C)(C)C)cc(=NCc2ccc3ncsc3c2)[nH]1 25439,c1(C(=O)NCC(C)NC(C(CC)OC2CCCC2)=O)c(C)oc(C)c1S(N)(=O)=O 25440,C(CNC(c1cnc(SC)s1)=O)(C(C)(C)C)NC(c1cn(CC(CC)O)nn1)=O 25441,Cc1cc(F)cnc1C(=O)NC(C1(C(=O)NCC2CC(C)(C)C2)CC1)C 25442,C1(CC(=O)NC(C(C)(C)C)CNC(=O)C=Cc2cc[nH]n2)CCCC2(CC2)C1 25443,N1(C(C(=C)F)=O)CCc2[nH]nc(-c3conc3C)c2C1.c1cc(O)ncn1 25444,C1(O)(CNC(C2CCN(C(C)=O)CC2)=O)CCN(C(C2CNC(=O)N2C)=O)CC1 25445,c1(C(=O)NC2C(C)(CNC(C3(O)CCOCC3)=O)CCC2)nnc(O)cc1O 25446,C1(C(N(CC(CN(C(COCC(C)C)=O)C)O)C)=O)Cc2ccccc2S1(=O)=O 25447,c1(C(CNC(C(=O)N(CCNC(C)=O)C(C)C)=O)(C)C)ccc2c(c1)OCCO2 25448,N1(C(c2c(OC)nsc2)=O)CCCC(CC(=O)NCc2noc(C(N)=O)n2)CC1 25449,C(=O)(CCCC(C)(c1nnnn1C(C)(C)C)NC1(C)CC=CCC1)OC 25450,C1(N(C(CCCOC)=O)C)CC2CCC(C1)N2C(C12CCCC1C2(F)F)=O 25451,C(CC1CCCO1)(CC)N(C(C1(F)CC1CC)=O)OC(C=CCCC)=O 25452,N1(C(c2cc(CNC(c3ccco3)=O)no2)=O)CC2CC1CO2 25453,N1(C(C(CC(=C)C)C)=O)CCC2CCN(C(c3c[nH]c4nccc-4c3)=O)C2C1 25454,C1(C(N(CCCNC(c2c(C)oc(Cl)n2)=O)C(C)C)=O)CCOC(=O)CC1 25455,C(=O)(C1=C(CC)OCCS1)NCC(C1CC1)NC(c1oc(CC)c(C)c1)=O 25456,C(=O)(CC1COc2ccccc21)NCC(C)CNC(=O)Cn1cc(C2CC2)cn1 25457,C(C(C)CC(=O)N1CCCCC1C(C)(C)CNC(c1cc(C#N)on1)=O)OC 25458,N1(C(C2(CNC(c3ccc(C)o3)=O)CCCO2)=O)CCCC(C)CC1 25459,c1(CNC(c2c(C)cns2)=O)cncc(C(=O)N(C2CCCCC2C)C2CC2)c1 25460,C1(OC)CCC2(C(N3CCCC(CNC(c4cnn(C5CCC5)c4)=O)C3)=O)CC12 25461,c1(CCC)cc(C(=O)NCC(O)CCNC(=O)Cc2cccn2C)ccn1 25462,CC1c2cc(O)ccc2CCN1C(=O)C(=O)Nc1snc(-c2ccccc2)c1Cl 25463,c1(C(=O)NCC2C3CN(C(C4(CCCC)CC4)=O)CC32)cc(CC)nnc1C 25464,c1(CCC(=O)NC2CN(C(CCC(=C)Cl)=O)CC(C)C2)cccc(S(N)(=O)=O)c1 25465,C1(CNC(C2(CC#C)CCC2)=O)CN(C(C2(OC)CCC2)=O)CC(C)(C)O1 25466,C1(C(C(C)C)NC(C=CC)=O)CCN(C(=O)CN2CC(=O)NC2=O)CC1 25467,C(=O)(NNC(=O)C1CCCN1C(C)=O)NC(COCC(CCC)=O)C1CC1 25468,Cc1cc(C(=O)NC2CC(C(N3CCC(CCF)CC3)=O)C2)ncn1 25469,N1(C(C2CCC2)=O)CCC2(CCCCN(C(C3CCCN3C3CC3)=O)C2)C1 25470,N1(C(CSCC#C)=O)CCC2CN(C(c3cccc4c3OCC4)=O)CCC2C1 25471,CS(=O)(=O)C(CNC(=O)CCSCC(N)=O)CNC(C1CC2CCC2C1)=O 25472,C12(CC(=O)N(C3CCN(C(c4ccc(SC(F)F)cc4)=O)C3)C)COCC(C1)C2 25473,N1(C(c2nc(CC)oc2)=O)CCC(C(=O)NCC2CCC(=O)NC2C)CC1C 25474,N#Cc1c(NC(=O)CCC(=O)C(O)CC2CCNCC2)sc2c1CCCC2 25475,c1(OC)ccc(CCNC(C23CC(C(=O)NC(C)(C)C)(C2)C(C)O3)=O)cc1OC 25476,C(=O)(C1SCCc2sccc21)OC(C(C)(CN(C)C)NCCC#N)C 25477,C12(NC(c3cnc(=N)[nH]c3)=O)CCN(C(c3cnn(C4CCCC4)c3)=O)CC1C2 25478,CN1CCCC1CCC(=O)N(CC(C)O)CCNC(C1CCN(S(C)(=O)=O)C1)=O 25479,C(=O)(C1CCCc2nn[nH]c21)N1CC2CC(NC(=O)Cn3ncccc3=O)C2C1 25480,Cc1cc(C(N2CCC(NC(=O)C(=O)N(C)C)C(CO)CC2)=O)cc(C)c1C#N 25481,c1(C(N2C(CNC(c3c(C)ccc(OC)c3)=O)CC2)=O)cn(C)c2ncccc12 25482,CCCCCC(O)C(=O)NC(C)CN(C(=O)C(c1ccc(=O)n(C)c1)(F)F)C 25483,N1(C(c2cc(C)sc2)=O)CC(C)CN(C(c2ccn(C)c2C)=O)C(C)C1 25484,C1(CC(=O)NC(C)CC(=O)OC)(OC)CN(C(c2cnn(C(C)C)c2)=O)C1 25485,c1(CC)c(C(=O)NC2COCCC2C(=O)NC(c2cccnc2)CO)ccn1C 25486,c1(C(=O)NCCC=C=C)nc(CNC(c2snnc2CC)=O)oc1C 25487,Cn1c(NCC2(CNC(=O)CC=C(Cl)Cl)CCC2)cc(=O)n(C)c1=O 25488,c1(CNC(CN(C(C2(O)CCSC2)=O)CC)=O)cc(CO)[nH]n1 25489,N1(C(C2(S(C)(=O)=O)CCC2)=O)CC2CCC1CN2C(=O)CN1CC2C=CC1C2 25490,CC1CCCC1NC(=O)CCCN(C(=O)CC1CCCC1)C 25491,c1(CNC(c2cc(C)[nH]n2)C)ccc(CN2CCC(C)CC2)cc1 25492,N1(C(Cc2n(C)nc(Br)c2)=O)CCC(NC(=O)CCc2ccoc2)C12CC2 25493,C1(SC)CC(CC(=O)NC(C)CCN(C(=O)C(C)C)C)C1 25494,N12CC(C(OC)C1)OCC2=O.c1(-c2cn(CCOC)nn2)ccc(C)cc1 25495,c1(C(=O)NCC(CO)NC(CC(CC)C2CC2)=O)cc(C)ncc1C 25496,N1(C(CC=C)=O)CCC2CCCC12C(=O)NC(c1ccnn1C)C 25497,S(=O)(=O)(c1ccc(C(=O)NCC2(F)CC(NC(C3(CSC)CC3)=O)C2)cc1)NC 25498,CS(=O)C1CN(C(=O)CC2CCN2C(c2csc(Cl)n2)=O)C1 25499,c1(C(=O)NCCCC2(CNC(C(C)N(C)C)=O)CCCC2)cnc2ccoc2c1 25500,CC1CNC(C)(C)CN1C(=O)Cc1ncc(Br)s1 25501,C=CC1(C(=O)NC2CCC(NC(=O)C(C)=CCC)CC2)CCCCC1 25502,C(=O)(CCCN=[N+]=[N-])N1CCC(N(C)Cc2c(C(=O)OC(C)(C)C)occ2)CC1 25503,CN1CCN(C(=O)CC2CCCC(C)(C)C2)CC1CNC(c1ccnnc1O)=O 25504,C1(CNC(CCc2n(C)ccc2)=O)C(O)C(O)CN1C(C1CCNC(=O)C1)=O 25505,c1(C(=O)NCC2C(NC(=O)CNC(N3CCCC3)=O)C2)cnc2ncccc2c1 25506,N1(C(CSCCCC)=O)CCC(C)(CNC(=O)C2=NOC(C(C)(C)C)C2)CC1 25507,C(=O)(CC(CC(C)C)NC(C12CCC(C)(C1)OC2)=O)N1CC(C)(CC=C)C1 25508,N1(C(C)C)C(=O)CCC1C(=O)NCCCNC(=O)CC1CC2(COC2)C1 25509,C1(C)(C(=O)NC2CC(C)(OC)C2(C)C)Cc2ccc(Br)cc2C(=O)O1 25510,Cc1ncncc1NC(C1CC1NCc1cccc(CO)c1)=O 25511,N1(C(C(CC2CC2)NC(Cc2n(C)ccn2)=O)=O)CCC12CC(C(N)=O)C2 25512,C1(C(=O)NCC2(NC(C3CC34CCCC4)=O)CC2)(CC)CNC(=O)C1 25513,Cc1cc(CCC(=O)N(CCNC(=O)CC2(C)CC2(F)F)C(C)C)on1 25514,C1(NC(C(C(C)C)(C)C)=O)CC2CCC1CN(C(=O)CC1CCCCC1O)C2 25515,c1(C(N(CCNC(Cc2ccc(C)c(C)c2)=O)C2CC2)=O)cc2ccncc2s1 25516,N1(C(c2c(C)cn(C)c2)=O)CCC(F)C(NC(c2cc(C)n(C(C)(C)C)n2)=O)C1 25517,c1(SCC)cc(C(=O)N(CCNC(=O)CN(C2CCSC2)C)CC)sc1C 25518,Cc1nn(C)c(C)c1C(C)C(=O)NC1CC(CCNC(=O)CC2CCCOC2)C1 25519,c1(OC)cc(CNC(=O)NC2CNCCC2Cn2cccc2)ccc1OCCO 25520,N1(C(C(Cn2ccc(C)n2)C)=O)C2CCCC1CN(C(=O)CC(C)F)C2 25521,C1(C(=O)NCCC2CC(C)C2)CN(C(C2(C)CCCC2O)=O)CC1(F)F 25522,N1(C(C(c2ccc(C)cc2)C)=O)CC2(C1)CN(C(=O)C(C)(C)CF)CCO2 25523,C1(C(N2C3C(NC(CN(CCC)C)=O)C(C3)C2)=O)CCCC2CCCN12 25524,c1(C(=O)NCCN(C(C(CC#C)O)=O)C2CC2)ccc(OC)c(C)c1 25525,c1(OCC=C)ccc([N+](=O)[O-])c(C(N2CCC2CNC(=O)CC2CC(C)C2)=O)c1 25526,N1(CC)CCN(C2CCCN(C(=O)C(C(C)C)NC)C2)C(=O)C1.OC 25527,c1(C(N(C)CC2N(C(CS(=O)(=O)NC)=O)CCC2)=O)cc(N)cnc1Cl 25528,C1(C(N2CC(S(C)(=N)=O)C2)=O)(NC(c2scc(OC)c2)=O)CCC(C)(C)C1 25529,c1(N2CC(N(C(c3ccn(CCOC)n3)=O)C)C2)ncnc2[nH]c(C)nc12 25530,c1(C(=O)NCC2CC(NC(C(C=CC)O)=O)C2)cc2n(n1)CCCC2O 25531,Cc1ncc(Cl)cc1NC(=O)COC(C1CC1c1ccc(C2CCCCC2)o1)=O 25532,c1(CNC(C2C3CN(C(c4nc(C)nc(O)c4)=O)CC32)=O)ccc(Cl)c(C)c1F 25533,C(=O)(CC(C)C(C)C)NCC(CN(C(C1CCC(CCO)CC1)=O)CC)(C)C 25534,C(=O)(CC(C)(C)N(C)C(C1(Cl)CC1)=O)N1C(CC)CCC1 25535,C1(C#N)(C(=O)NCC(C)(C)NC(c2c(C)n[nH]c2)=O)C(C#N)C1(C)C 25536,C1(C(=O)NC2CCCC(NC(c3ccc(C(F)F)nc3)=O)C2)CCCC12CCC2 25537,N1(CC)CCCC(C)(C(=O)NC2CC(CC#N)C2)C1.c12ccc(cc1)CNC2=O 25538,C=CCC(CNC(=O)C(C#N)CCC)C(=O)N1CCC(OC(C)=O)C1 25539,c1(NC(C2CCCN2c2cc(Cl)sc2Cl)=O)cc(Oc2ccccc2)ncn1 25540,c1(COC(C)=O)ccc2nc(NC(CC(=O)N(C)C)c3cccs3)sc2c1 25541,C1(CNC(c2ccc(Cl)[nH]2)=O)CC(F)CN1C(C1CCS(=O)(=O)C1)=O 25542,CN1CCC(=CC(=O)NC2CC(CCNC(c3n[nH]cc3Br)=O)C2)CC1 25543,Cc1nc(C(C)NCC2CN(C)CCO2)ccc1OC(C)C 25544,CC1(CNC(c2cc(Cl)ccc2F)=O)CN(C(C2CCOC2=O)=O)CCO1 25545,C=CCCC(C(=O)N1CCOC(C)(C)C1)NC(=O)CCn1cnnn1 25546,C1(C(=O)NCC(CCNC(c2cnco2)=O)OC)(SC)CCOCC1 25547,C12(CNC(C)=O)CC1CN(C(=O)NC(CC(C)C)c1nc(CNC(C)=O)no1)C2 25548,N1(C(C2C(C)N(C)CC2)=O)CCC2(CCC2NC(c2cc(C(F)F)no2)=O)CC1 25549,Cc1cc(N(CC(=O)NCCn2nnnc2CC2CC=CCC2)C)cc(C)c1 25550,CC(C)(C)CCCC(=O)NCC(C)(C1CC1)NC(C1CC2(C)CC1CO2)=O 25551,C1(C(=O)NC(CCSC)C)CCN(C(=O)CCCC2CCCO2)O1 25552,C1(C(N(C2CC(OCC)C2)C)=O)CCN(C(=O)CC2(CSC)CC2)C1 25553,c1(C(=O)NCC(=O)NCC(=O)N(C(CCC)C)C)c(C)nn(C)c1N 25554,c1(N2CCC(C(N)=O)(NCC)CC2)cc(C)[nH]c(=NCCc2cccnc2)n1 25555,C(=O)(C1Cc2c(Cl)cccc21)NC1C(F)CCN(C(C2(SC)CC2)=O)C1 25556,c1(CN2CCC(C(F)(F)F)(OC)CC2)nc(O)c2cnn(-c3ccccc3)c2n1 25557,C(=O)(C1CCc2c[nH]nc21)N1CCC(CC(=O)Nc2cc(C)nc(O)c2)C1 25558,c1(CC(=O)NC2CN(C(C(CSC)O)=O)C(C)CC2)cccc([N+](=O)[O-])c1 25559,C(=O)(C(C)(CCC(F)(F)F)c1ccccc1)NCc1nc(C)c(C)[nH]1 25560,c1(C(N(CC(C)CNC(c2cnsc2)=O)C)=O)cc2c(nc1O)CCCC2=O 25561,C1(n2ncc(C)c2)CCN(C(=O)Nc2cnn(CC3CCCOC3)c2)CC1 25562,c1(OC)cc(CN2CCN(c3nc(N(C)C)cc(C)n3)CC2)ccc1Cl 25563,C1(NC(c2nc[nH]c3nccc2-3)=O)CN(C(C2CSC2)=O)C2CCCCC12 25564,C=CCC(CNC(C1(C(=O)OC)CCCCO1)=O)C(=O)NC1(C)CN(CC)C1 25565,C1(N(C(=O)CCc2cnoc2)CC)CCCN(C(=O)CC=C(C)C)C1 25566,c1(COC)nc(NCCc2c[nH]nc2O)cc(=NC2CCCC(C)C2)[nH]1 25567,c1(SCC(=O)N(C(C)CC(C)C)C2(C(C)C)CC2)ccccc1 25568,C1(NC(c2cc(CCNC(CCSCCC)=O)on2)=O)CC(CO)C2CC12 25569,c1(OCC)nc(C(=O)NCC2CN(C(C3(C)CC3)=O)CC2OC)cc(O)n1 25570,N1(CC(=O)N(C(C)C(=O)NCC(F)(F)F)CCC)CCc2sccc2C1 25571,C(CCCCC(=O)NCC(CNC(C1CC(C)(C)O1)=O)OC)OCC 25572,N1(C(C(C)(CO)OC)=O)CC2(CNC(=O)Cc3nc(C4CC4)cs3)CC1CO2 25573,N1(C(c2cccc(C(F)(F)F)n2)C(=O)NC)CC(N=[N+]=[N-])CCC1(C)C 25574,C=CCCCCCC(=O)N1CCC2(NC(=O)Cn3cc(CN(C)C)nn3)CC2C1 25575,n1(CC2N(C(=O)NCC(CCO)OC)CCC2)c(C)nc2ccccc12 25576,CC1CCN(CC(C)(C)COC(C2(c3ccc(SC(F)F)cc3)CC2)=O)CC1 25577,c1(NC(CC2CCC(NC(C=COCC)=O)CC2)=O)ccc(I)cc1I 25578,C1(CNC(COC2(C)CN(C(=O)CC3COCCO3)C2)=O)CCCC(CO)C1 25579,CC1(C)COc2c(C(=O)NCC3CCN(C(c4csc(C#N)c4)=O)C3)cccc21 25580,N1(C(c2ccc(C#C)cc2Cl)=O)CC2CCCCC2(C(N2CC(F)(F)C2)=O)C1 25581,c1(CN2CCC(CC(=O)N(CC)Cc3ccco3)C2)ccc(Cl)c(Cl)c1 25582,C1(CN(C(C2CC2CC(C)C)=O)CC)CCCCN1C(=O)CC1(OC)CCC1 25583,Cc1ccc(OC(C)C)cc1NC(c1cnn(C2CCOCC2)c1C)=O 25584,N1(C(c2c(CCC)cccc2)=O)CC2CCC2(CCNC(=O)C2=CCCCC2)C1 25585,C(=O)(CCCCCC(=O)NC(C)CNC(=O)CC1CCC2(CC1)CC2)OC 25586,C1(OCC)CCN(C(=O)C=CC(C)(C)NC(=O)CCOC(C)=O)CC1C 25587,C12(CCNC(CCc3c(C)noc3)=O)CCC1CN(C(c1cncs1)=O)C2 25588,Cc1cc(CC(N2CCCC2CCNC(=O)Cc2cccnc2C)=O)ccc1O 25589,CCCC(O)CC(=O)NC1CN(C(=O)Cc2ccnn2C)CC1O 25590,c1(C(=O)NCCc2cn(-c3n(C)nnc3)nn2)cc2cc(Br)cn2cn1 25591,n1(CC=O)cc(C(=O)NC2C(CC)CCC2)c(=O)cc1C.C(=O)(CCS(N)(=O)=O)N 25592,c1(C(=O)NCCC2CC(NC(c3nn(C)c(O)c3)=O)C2)cnc2ncccn12 25593,C12(NC(C=CC(C)NC(C(CC)=CC)=O)=O)CCN(CC1)CC2 25594,c1(NCC(CCCC)NC(=O)Cn2ccnn2)ccc([N+](=O)[O-])cn1 25595,N1(C(C(C(=O)OCC)OC)=O)CCC2(CCN(C(c3coc(Cl)c3)=O)CC2)C1 25596,C12(CCCSC1)CN2.N1(C(=O)NCC)CCCCC1CC 25597,C1(NC(c2n[nH]cc2Br)=O)CC2CC(NC(C3CC34CC4)=O)C2C1 25598,C1(C#N)(C(N(C2CC(c3cn(C4(O)CCOCC4)nn3)C2)C)=O)CC2CCC1C2 25599,CS(=O)(=NC(=O)c1cccc2ccccc12)c1cnn(C2CCCCO2)c1 25600,C(CC(C)(C)NC(C1CC(C)=NO1)=O)N(C(C(C)SCC)=O)C 25601,c1(N2CCN(C(c3cc(C#N)[nH]c3)=O)CC2)ccc(-n2cnnn2)cc1Cl 25602,C=CC1(C(N2CCC(OC(C)C)CC2)=O)CCN(C(=O)C(CC)N(C)C)C1 25603,Cc1cc(C(N2CCCC2CNC(C2(C3CCC3)CCC2)=O)=O)nc(C)n1 25604,c1(C(N2CCN(C(CCSCc3ccc(C)cc3)=O)CC2)=O)cnc(F)cc1C 25605,c1(OCCC(=O)N(CCNC(C2C(C)(CCCC)C2)=O)CC)ccc(Cl)c(Cl)c1 25606,c1(NC(N2C(CC(=O)NC3CCC(O)CC3)COCC2)=O)cnnc(Cl)c1Cl 25607,c1(CC#N)ccccc1C(=O)NCC1CC1NC(C1CC(Cc2cccs2)C1)=O 25608,CCC(C)C(C(=O)N1CCCC1(C)CNC(C1CCOC1)=O)OC 25609,c1(-c2c(CC)noc2)nc(Cc2cccnc2)nn1C(C)COc1ccccc1 25610,c1(CC(N2CC(CC(C)NC(c3c(CCC)n[nH]c3)=O)C2)=O)cnccc1OC 25611,c1(OC)cc(C(=O)NCCCCNC(=O)C(F)Cc2ccccc2)c(O)c(Cl)c1 25612,c1(OCCCC)c(OCC)cc(C(=O)NC2CCNCC2F)cc1Cl 25613,C1(NC(C2CCN(C(C(C)C)=O)CC2)=O)CN(C(C2(CO)COC2)=O)C(C)(C)C1 25614,N1(C(c2c(C)scn2)=O)CC(C)CN(C(c2ncncc2Cl)=O)C(C)C1 25615,N#Cc1cc(C(N2CC(NC(C3CC(F)(CO)C3)=O)C(C3CC3)C2)=O)ccc1F 25616,N1(C(CC(=O)NCC)=O)CCC(NC(=O)CCSc2ccccc2)C1C 25617,c1(C(N2C(CNC(c3ccc(CC)nc3)=O)CC(F)C2)=O)cccc2occc12 25618,Cc1cc(NC(C23CCN(C(c4c(I)cnn4C)=O)CC2C3)=O)cnc1C 25619,C1(N(C(CC(C)C2CCCO2)=O)C)CCC(CNC(=O)CCc2cccs2)CC1 25620,N1(C(C(CCC=C)(F)F)=O)CCC2(CC1)COC(CNC(=O)C(CC)SCC)C2 25621,c1(C(=O)NCc2cccc(C(F)(F)F)n2)cc2ncccc2o1.C12CC1NC2=O 25622,C1(CC(=O)NCc2c(C(=O)N(C3(C)CCCC3)C3CC3)nco2)CC(O)C1(C)C 25623,CCS(=O)c1ccccc1C(N1CCCN(CCNC(C2CC2C)=O)CC1)=O 25624,N1(C(C(CC#C)C)=O)CCC2(CC1)CC(NC(=O)C(C)(C)CCC)CO2 25625,C1(NC(c2cc(C)sc2)=O)CCCN(C(=O)CN2CCC(=O)NC2=O)CC1F 25626,Cc1nc(N)c(CC(=O)NCC2CC(C)N(C(=O)C(F)(F)C(C)(C)O)C2)c(O)n1 25627,Cc1nc2cc(C(=O)NCC(CNC(=O)CCSC3CCCC3)CO)cnc2[nH]1 25628,c1(C(=O)NC2C=CC(CNC(C(=O)NCC)=O)C2)cccc(C#N)c1F 25629,C(C)(CNC(C1(C2(C)OCCO2)CC1)=O)(CC)NC(C1C(=C)CC1)=O 25630,N1(Cc2c(CC(=O)OC)cccc2)CCCN(C(=O)CCC2CCOC2)CC1 25631,Cc1cc(F)cc2[nH]c(C(=O)N(CC(C)O)CCNC(c3cnnn3C)=O)cc12 25632,c1(NC(=O)NC(CO)C2CC2)cccc2ccccc12.N12CC(C1)CNC2=O 25633,n1(C(C)C)cnc2c(NCc3ccnn3C)[nH]c(=NC3CCOC(C)C3)nc12 25634,Cc1ccn2c(C(=O)NCCCNC(c3cccc(O)c3Cl)=O)cnc2c1C 25635,N1(C(C(C)N(C(CC(C)OCC)=O)C)=O)CCN(C(=O)CO)CC1 25636,C1(NC(C2C(C3C(C)C3)C2)=O)CCN(C(=O)Cc2ccccc2F)C1(C)C 25637,n1(CC(=O)NCC2(NC(C=CC)=O)CC3CCC2C3)cc([N+](=O)[O-])ccc1=O 25638,Cc1ccccc1OCC(=O)NC1CN(C(=O)CCC2NC(=O)NC2=O)CC1O 25639,c1(CC(=O)N(C2CC(NC(C3CC34CCCC4)=O)C2)C)c[nH]c2ccc(Cl)cc12 25640,c1(C(=O)NCCC(C)N(C)C(C2COC(=O)N2C)=O)ccc(SC(F)(F)F)cc1 25641,C1(C(=O)NCCCN(C(C(C)SC)=O)C(C)C)CC(=O)N(c2ccccc2)C1 25642,N1(C(C)=O)CC2CC1CN2C(C1CC(N(C)C(C2C3CCC(=O)C23)=O)C1)=O 25643,C(=O)(CC(C)C(C)(C)NC(=O)CSC1CC1)NCCCCCCC=C 25644,C(=O)(C1=C(Cl)CCC1)N(CCC)CCNC(=O)CNC(c1cnccn1)=O 25645,N1(C(C=C2CCC(C)C2)=O)CCC(C2(NC(c3cc(F)c(F)c(F)c3)=O)CC2)C1 25646,c1(CC(=O)NC)ccccc1NC(=O)NCC1CC(C)OC1C 25647,N1(Cc2cn(CCCCCN)nn2)CCOc2ncccc21 25648,C1(CNC(COCC=C)=O)CC(C)N(C(=O)Cc2cnccc2C)C1 25649,CC(CC(=O)N1CCN(CC(N2CC(F)(F)CCC2C)=O)CC1)C(C)(C)C 25650,c1(C(=O)OC)cc(C)cnc1N(CC(O)CN(C(=O)C=Cc1cccnc1)C)C 25651,c1(C(N2CCC(C3CCCO3)C2)=O)cnc(N2CCNCC2)nc1 25652,C(CN=C(NCc1c(Br)cnn1C)NC1CCN(C2CC2)C1)OCC 25653,C1(CNC(C2(CCCC)CC2)=O)CCCCCN1C(c1ccccc1OC)=O 25654,CN1CC(C)(C)CC1C(N1CC(C2CCN(C(=O)CSCC(F)(F)F)CC2)C1)=O 25655,Cc1cc(O)c(C(=O)NCCCN(C(=O)COCCCF)C)cc1Br 25656,C(CC(F)F)(C(=O)NCCCC1CCOC1)NC(C=CC=CCC)=O 25657,C=CCN=C(NCc1ccc(F)cc1)NC1CCCN(CC(F)F)C1 25658,N1(C(C2C(C(C)C)C2)=O)CC2CN(C(=O)C3=CCCC(C)(C)C3)CC2C(F)(F)C1 25659,N1(C(=O)CCc2ccoc2)CC2CN(C(c3ncc(Cl)s3)=O)CC2C1 25660,Cc1ncnc(C(N2CCC(CN(C)C(c3n[nH]cc3C(F)(F)F)=O)C2)=O)c1C 25661,N1(C(COCCC)=O)CCC(NC(C2CCCN2C(N)=O)=O)C12CCC2 25662,N1(C(C(C)NC(C)=O)=O)CCC(C2OCCC2NC(c2ccns2)=O)CC1 25663,C(C(F)(F)F)(C1CCCCC1)NC(=O)NC(c1cscn1)C 25664,N1(C(C(C)(C)C2CCOC2)=O)CC2C(CNC(=O)C(N)=O)C2C1 25665,Cc1ccc(C=CC(=O)NCC(O)CN(C(=O)CN2CCCCC2)C)c(C)c1 25666,c1(C(=O)NC2(CNC(C(CCOC)OC)=O)CCOC2)cnc(C2CC2)cc1C 25667,C1(F)(CNC(CCOCC#C)=O)CCN(C(C2CC2C2CC2)=O)C1 25668,C(=O)(C(C)C1=CCCC1)N(C)CC1CN(C(CSC(C)C)=O)CC12CC2 25669,CC(C)CC(CCO)NC(=O)CC1CN(C(C2(O)CCCCCC2)=O)CC1C 25670,C1(O)(CN(C)C(c2scnc2C2CC2)=O)CCN(C(=O)CCc2cnc[nH]2)C1 25671,CC1CN(C(=O)C(C2(O)CCC2)NC(c2cncc(CO)c2)=O)CCS1=O 25672,C(CNC(c1ccc(N2CCC(C)(C)C2)cc1)=O)(CCS(C)(=O)=O)OC 25673,C1(C(N2CC3C(CNC(CNC(C(C)(C)C)=O)=O)C3C2)=O)CC2(CCOCC2)C1 25674,C1(C(=O)NC(CNC(C2CC(CF)C2)=O)C2CCC2)(COC)CCC1 25675,C(=O)(C1=NOC(CN)C1)N1C(CN(C(=O)CSCc2ccncc2)C)CCC1 25676,C1(NC(C(C(C)C)OCC)=O)CN(C(c2csc3nccn23)=O)CCC1C 25677,C(C1CCCCC1)=CC(=O)N(CCCNC(=O)CNC(N1CCCC1)=O)CCO 25678,N1(Cc2ccc(C(=O)OC)[nH]2)CC2CCN(C(c3ccc(C#N)s3)=O)CC2C1 25679,c1(OCC)ccccc1CCS(=O)(=O)N(CC(C)C)C1CC1 25680,c1(C(=O)NCC2N(C(CCC)=O)CCCC2C)cc2ccccn2c1 25681,Cc1cc(C(N2CC3CC2CC3NC(=O)C2=COCCC2)=O)c(S(N)(=O)=O)s1 25682,C(C)(CNC(=O)CC1CCOC1)(CO)NC(C(F)=CC)=O 25683,c1(C(C)C)cccc(CNC(c2cnccc2Cl)c2nnnn2CC2(C)CC2)c1 25684,N1(C(c2cnn(C)c2Cl)=O)CC2COCCC2(NC(C2CC3(C2)CC3(F)F)=O)C1 25685,c1(C(C)C(=O)NC2CCC(NC(C3CC(Cl)(Cl)C3)=O)CC2)ccc(C#N)cc1 25686,Cc1ccc(F)c(C(=O)NCc2occc2C(=O)NC(C)C(F)F)n1 25687,C1(N(C(=O)CN2CCS(=O)CC2)C)CN(C(C2CCCCCC2)=O)CC12CC2 25688,C=CCC(C(=O)NC(C)CC(C)(C)OC)NC(C1(CO)CCCCC1)=O 25689,c1(C(N2CC(O)(C(C)NC(CCC(C)SC)=O)C2)=O)ccc(=O)n(CC(C)O)c1 25690,S(=O)(=O)(c1cccc(=NCC2CCC3CC23)[nH]1)NCCC(CC)(C)C 25691,c1(C(N2C(CNC(c3c(C)cco3)=O)CN(C)CC2)=O)ccc2nccn2n1 25692,C1(C(=O)NC(CCOC)CNC(=O)CC2(OC)CCC2)Cc2nccn2C1 25693,Cc1nn(C)c(C)c1C(C)C(=O)NC(CNC(c1cc[nH]c(=N)c1)=O)C(C)(C)C 25694,Cc1oc(S(N)(=O)=O)cc1C(N1CCC(NC(C2CCCC(CF)C2)=O)CC1)=O 25695,CC(CCCO)N=c1cc[nH]cc1S(=O)(=O)NCCCc1cccc([N+](=O)[O-])c1 25696,Cc1cc(C(=O)NC2CC3(C2)CC3NC(=O)CC2CN(C)CC2O)cc(C)c1Cl 25697,c1(CC(=O)N(C)CC2CCN(C(c3c(CC)ncs3)=O)C2)cccc(F)c1O 25698,C1(CC(=O)N(CCN(C(Cc2c(C)con2)=O)C)C)CCOC(C(C)C)C1 25699,C1(OC(=O)CC2SC3=NCCN3C2=O)C=C(c2ccc(Cl)cc2)CCC1 25700,CCCC(CCCNC(C1CCCCC1O)=O)NC(c1cc(C(C)C)no1)=O 25701,C1(NC(c2n(CC)ccc2)=O)(CF)CCN(C(=O)C=C(C)C(C)C)C1 25702,N1(C(=O)NC2(C(=O)OCC)CCC2)CC(NC2CCC=CCC2)C(C)C1 25703,c1(C(=O)NCCNC(CCc2c(C)nn(C)c2C)=O)nc(=N)[nH]c2ccccc12 25704,C(C(=O)Nn1cnnc1C)C1CN(C(Cc2c(C)con2)=O)C(C)(C)C1 25705,C(C(CC(C)C)C(=O)N(C1CCCC1O)C)NC(c1cc(C)oc1)=O 25706,C(=O)(C1=NN(C)C(=O)CC1)N1CC(NC(CC2C(C)CCO2)=O)CC2(C1)CC2 25707,C1(CNC(=O)C=Cc2cccs2)CCN(C(c2cn(C(F)F)cn2)=O)CC1 25708,c1(CCC(=O)NC(C)CNC(=O)COc2ccccc2C(N)=O)ccc(C#N)cc1 25709,C(=O)(CCC(C)(C)N(C)C)NC1CC(CNC(c2ncc(OC)nc2)=O)C1(C)C 25710,N1(C(CNC(=N)N)=O)CC2(CCCC2NC(=O)Cc2c(Cl)cccc2Cl)C1 25711,C1(CNC(c2c(C)nn[nH]2)=O)CC(O)CN1C(=O)CCCCN(C)C 25712,c1(OC)ccc(C(=O)NCc2csnc2OC)cc1.C12CCC1C1CC1NC2=O 25713,C1(CNC(CC(C)SC)=O)CN(C(C2CC=CCC2)=O)CCC1C 25714,CCCCC(CC(=O)NC1CC2OCCCC12)NC(c1cccc(CC)n1)=O 25715,CC1CCN(C(=O)CCF)C(C)C1NC(=O)C(C)C1CC1c1ccccc1 25716,C(c1cc2ccccc2o1)=CC(N1CCC(CN(C(CN(CCC)C)=O)C)C1)=O 25717,c1(C(=O)NCC(CC=C)NC(C2CC(O)CN2C)=O)c(F)ccc(C)c1Cl 25718,N1(C(C(C2CCOCC2)OC)=O)CCC(C(F)CNC(=O)CSC)CC1 25719,c1(OC)cnc(C(F)(F)F)cc1C(=O)NC1(C)CN(C(C2(F)CC=CC2)=O)C1 25720,N1(CCCC(=O)NCCN(C(C2(COC)CC2)=O)CC)C(=O)c2ccccc2C1=O 25721,C=C(Cl)CC(C(=O)NC(c1cn(C)nc1C)C)NC(=O)Cc1ccc(F)cc1 25722,c1(C(=O)NCC2(NC(C3C(C(C)C)(CC)C3)=O)CC2)cc(O)cs1 25723,Cc1ccc(C)c(C(N2CC3C(CNC(C4(n5cc(Cl)cn5)CC4)=O)C3C2)=O)n1 25724,C1(C(=O)NCc2ccc(C(C)C)cc2)CN(C(C2(F)CCC2)=O)CC1(F)F 25725,CC1CN(C(C2CNC(=O)N2)=O)CCN1C(=O)CCCC(=O)c1ccc(F)cc1 25726,CCCC(CCC)=Cc1nc(C2(C(=O)N(C)C)CC2)no1 25727,N1(C(CN(C(=O)C(Cl)(Cl)Cl)C)=O)CCC12CN(C(=O)C(CC(C)C)NC(C)=O)C2 25728,CN1C(=O)OC2CN(C(C3(F)CN(C(c4ccncc4Cl)=O)C3)=O)CC12 25729,N1(C(CCC#C)=O)CC(N(C(=O)C(C)N(C)C)C)C2(CC2)C1 25730,N1(C(CSCC#C)=O)CC(C(N2CCc3nc[nH]c3C2)=O)CC(C)(C)C1 25731,C1(C(N(CCNC(CCOCCOC)=O)C(C)C)=O)CCC(N=[N+]=[N-])CC1 25732,N1(C(C2CCC(=C)CC2)=O)CCC2(CC(NC(=O)CCOCC(C)C)C2)C1 25733,C=CC1COCC1NC(=O)C(O)CCNC(=O)CCOCC(F)F 25734,CC(C)CC(C(=O)NCC1C2CCOCC12)N(S(C)(=O)=O)C1CC1 25735,c1(NCC2(CCC)CC2)nc2ccccc2nc1NCc1cc(Br)ccc1N 25736,C12(c3onc(C)n3)COC(CN1C(=O)N(Cc1ccccc1)Cn1cncn1)C2 25737,c1(C(=O)OC)ccc(CCC=CCC(=O)N(CCCCCC)C)[nH]1 25738,c1(CN(C(CC2(OC)CC2)=O)C)cccc(C)c1.C(c1ccsc1)=CC(=O)NC 25739,C(CC(N)=O)(C(=O)N1CCCC1CC(N)=O)NC(C(C)n1ccnn1)=O 25740,C1(NC(c2occ(C)c2C)=O)CCCCCCC1NC(c1cnn(C2CC2)c1)=O 25741,c1(C(C)O)ncc(C(N2CCC2CNC(=O)C(C)OC2CCCCC2)=O)s1 25742,O(NC(=O)C(c1ccnn1C)NC(=O)CCCNC(C)=O)C(COC)C 25743,C(C(CC)(CC)C(=O)NC1CCN(C(C)=O)CC1C)NC(Cc1cn(CC)nn1)=O 25744,C1(C(=O)Nc2cncc3nc(C)[nH]c32)CC(N=c2nc(C#N)[nH]cc2Cl)C1 25745,N1(C(C=NOC)=O)CC2CCC1C1CN(C(=O)CCn3cc[nH]c(=O)c3=O)CC21 25746,CN1C(=O)NCC1C(=O)NC(C1CCCC1)CNC(=O)C=CC1CCOC1 25747,C#CCCC(O)C(=O)N(C1CN(C(=O)C2=CSCCO2)C1)C 25748,O(P(=O)(CCCC1CC(n2cc(C3(OC)CNOC3)nn2)C1)OCC)CC 25749,Nc1nccnc1C(=O)NC1CC1NC(C1COCC1C(c1ccccc1)=O)=O 25750,CC1C(NC(C2CN(C)C(=O)N2)=O)CC2CCC1N2C(c1ccsc1C(F)F)=O 25751,c1(OCC(N2CCC(NC(C3(CC)CC3(F)F)=O)CC2)=O)ccc(F)c(F)c1 25752,c1(C(N(C2CCN(C(c3scc(C)c3)=O)CC2)CCO)=O)ccn2ncccc12 25753,C1(OC)CC2CCC1(N(C(=O)C1CC1)Cc1cc(C(F)(F)C(F)(F)F)on1)C2 25754,N1(CCC(=O)NCC2(C(=O)NOCC3CCOC3)CCCO2)CCCCC1 25755,C(COC)(C(=O)NOCC(=O)NC1CC1)NC(c1c(CC)cns1)=O 25756,N1(C(CN(C(C(C)OCC2CC2)=O)CC2CC2)=O)CCC(O)C(C)(C)C1 25757,c1(C(N2CCCC(F)(CNC(c3ccncc3F)=O)C2)=O)cccc2nn[nH]c12 25758,Cc1nc(C(=O)NCC(c2ccccc2F)NC(=O)C=CC2(C)COC2)c(C)s1 25759,N1(C(c2cc(C)sc2)=O)CCOC(C(=O)NOCCF)C1 25760,N1(C(c2cccc(I)c2)C(=O)NCCOC)CCCC(O)(c2ccccc2)CC1 25761,n1(CC)ncc2cc(C(=O)NC(CNC(c3nocc3Cl)=O)CC(C)C)cnc12 25762,c1(-c2nc(C(CC)CC)nn2Cc2cccs2)cnc2n1CCCCC2 25763,C(CCC(C)(C)C(=O)NCC1CCC2(CCC2)C1)NC(COCCOCC#C)=O 25764,C#CCCCCC(=O)N1CCC(CO)C(NC(c2cccnc2C)=O)C1 25765,C1(N(CC(C)C)C)CCN(Cc2ccccc2)C2(CC2)C1 25766,CCCC(C(=O)NCc1cc(C)ns1)NC(=O)CC1CCOC1(C)C 25767,C1(CNC(C(C)=C2CCC2)=O)CC(C(=O)NCC(C)(C)CC(C)C)=NO1 25768,CCCC(CCC)CC(=O)NC(C(=O)NCC(F)Br)C1(O)CCC1 25769,c1(C(=O)NC2CN(C(C(CCC)N(C)C)=O)C2)nc2ccccc2[nH]1 25770,c1(C(=O)Nc2cc(C(=O)OC)c(C)nc2)cc2c(=O)n(C)c(=O)n(C)c2s1 25771,N1(C(C(CCO)N(C)C)=O)CC(NC(c2ccc(O)nn2)=O)C(C2CC2)C1 25772,c1(C(=O)NCC2C(C)(C)C(NC(=O)Cc3cc(Cl)cs3)C2)ccc2c(c1)CC2 25773,C1(CNC(C(C(C)O)C)=O)(CO)CCN(C(=O)CCCc2cnn[nH]2)CC1 25774,N1(C(CCC2C(C)(C)C2)=O)CCC(OCCNC(c2sccc2F)=O)C1 25775,C1(NC(C2CC(C)CC(C)C2)=O)CCOC12CCN(C(=O)OC(C)(C)C)CC2 25776,C1(C(=O)NOCCSC2CC2)CN(C(c2cnco2)=O)C2(CCC2)C1 25777,c1(C(=O)NCCC2(CNC(C3(O)C(C)(C)C3)=O)CC2)cccc(OC(F)F)n1 25778,C(CCN=c1[nH]c(=NCC2COC(C)(C)CO2)[nH]c2c1CSC2)NC(C)=O 25779,c1(C(N(CC)CC2CCCN2C(c2occc2F)=O)=O)[nH]c(O)nc1C 25780,c1(N(C)CC2COC(=O)N2)nc(=NCC2SCCS2)nc(N2CCOCC2)[nH]1 25781,c1(C(N(CC(CC)NC(=O)CSC(F)F)C)=O)ccc(-c2ccncc2)s1 25782,c1(C(N2CCC(CN(C(C=C(C)C3CC3)=O)C)C2)=O)cn2cnnc2cn1 25783,C(=O)(C(CCC=C)NC(c1cc(C)cc(O)c1)=O)N(CC#C)CC1CCCO1 25784,N1(CCNC(C(C)(C2(C)CC2)OC)=O)CCC(NC(C2CN(C(N)=O)C2)=O)CC1 25785,Cc1nc2c(C(=O)NCC3CCCN3C(=O)C=Cc3sccc3C)cccc2o1 25786,c1(OC)ncc(Br)cc1CN1CCC(CC(=O)NCCCC(F)(F)F)CC1 25787,c1(CC2N(CCC(=O)OC)CCC2C)ncc(C)cc1Cl 25788,Cc1cccc(C(C(C)C)NC(c2cccc(C(N)=O)c2)=O)c1 25789,C1(CNC(C(C)NC(=O)C2CC2)=O)CN(C(c2ccccn2)=O)CC1(F)F 25790,N1(C(CC(=O)OC)=O)CC=C(CC(=O)N2CC=CC(OC)C2)CC1 25791,CCCCC(C(=O)Nn1cnnc1C)NC(c1ccc(C#N)c(C)n1)=O 25792,CC1=C(C(=O)NC(CCC2CC2)C(=O)N2CCC(c3ccco3)C2)CCO1 25793,CC1CCN(C(c2cc(Cl)nnc2O)=O)CCN1C(C1CC1C1CC1)=O 25794,N1(C(CC(C=C)C)=O)CCCC(O)(CNC(=O)COCc2nccs2)C1 25795,N1(C(C(=Cc2cccnc2)C)=O)CC(NC(=O)CCCNC(N)=O)CCC1C 25796,C(=O)(C(O)CC(C)(C)C)N1CC(CNC(C(C(=O)OC(C)(C)C)OC)=O)(OC)C1 25797,Cn1cc2c(C(=O)NC3CCCN(C(=O)CCc4nc(=N)[nH][nH]4)C3)cccc2n1 25798,CC1CC(CCNC(c2cccs2)CO)C1 25799,C(N=c1[nH]c2c(c(=NC3CCC4CCC34)[nH]1)CCCCC2)C1(COC)CCCC1 25800,c12ccc(s1)C=CC(=O)NC1(CC1)CCN2.C(=O)(COCC1CCC1)N.CC=C 25801,S(=O)(=O)(c1ccc(Nc2cn(C)nc2OC(C)C)nc1)N1C(CCCC)CCC1 25802,n1(CC(=O)OC(CNC(C(C)OCC)=O)C)cc(Cn2ccnc2)nn1 25803,N1(C(C)C)C(=O)CCC1C(=O)NCC1C2CC1N(C(=O)COC1(C)CCCC1)C2 25804,Cc1nc2ccsc2c(=NCCN(C(=O)Cc2ccc(F)cc2)C)[nH]1 25805,C1(C(=O)NCCNC(C)=O)(NC(C2CC(OCC)C2)=O)CCCCC1 25806,N1(Cc2cccc(C#N)c2)Cc2ccc(NC(c3cc(Cl)c(Cl)cn3)=O)cc2C1 25807,C1(N(C(C(C(=C)C)(C)C)=O)C)CC2CCC(C1)N2C(=O)C1=CC2CCCC12 25808,CCC(CC)CCC(=O)N1CCOC(C(C)NC(=O)C#CC2CCC2)C1 25809,N1(C(C(N2CCC(c3nc(=N)[nH][nH]3)C2)=O)=O)CCC2(CC1)CC2C(=O)O 25810,N1(C(C(CCOCC)NC(c2ccns2)=O)=O)CC2C3CCC(O3)C2C1 25811,C1(NC(C23OCC(CC)(C2)C3)=O)CCN(C(c2cc(Cl)c(Cl)s2)=O)CC1F 25812,C1(C2CCC2)(NC(C2CCCC(C(=O)O)C2)C)CC1 25813,C1(C(=O)NCCCC(C)NC(c2cccc(F)c2)=O)COCC2(CCC2)O1 25814,N1(C(c2c(C)sc(Cl)n2)=O)CCN(C(c2ncc[nH]2)=O)CC(O)C1 25815,N1(C(CN2C(C)CC2)=O)CCC(F)C(NC(C2CCCC2)=O)C1 25816,c1(C(=O)Nc2cc(F)ccc2F)n[nH]c2c1CN(C(C1(F)CC1)=O)CC2 25817,C1(C(=O)NCc2cc(=N)[nH]cn2)(COC)Cc2ccccc2C1 25818,CCCCCC(=O)NCCC1CC(NC(c2cc(-c3cccc(O)c3)on2)=O)C1 25819,c1(C(N(C(CN(C(c2c(C)cccn2)=O)C)C)C)=O)ccc(F)c2occc12 25820,c1(C(C)=O)cc(C(N2CCC(F)(CNC(c3cnnn3C)=O)C2)=O)oc1C 25821,c1(OC)cncnc1C(N1CC2C(CNC(=O)CCC3CCCCO3)C2C1)=O 25822,C(CO)(C(=O)NCC1CC1C1CC1)NC(C(F)=CCC)=O 25823,N1(C(c2n(C)[nH]c(=N)c2)=O)CCCC1C1CCCCN1C(c1cc(=O)cc[nH]1)=O 25824,CCS(=O)CC(=O)NCCCC(C)(C)NC(=O)C(C)NC(c1ccoc1)=O 25825,CC1CN(C(=O)CCc2ncc[nH]2)CCCN1C(c1cncc(CO)c1)=O 25826,CN1CCN(c2nccc(Cc3ccccc3)n2)CC1(C)C 25827,c1(C(N2CC(C(C)NC(c3c(C)ccnc3O)=O)C2)=O)cccc2[nH]ccc12 25828,C(C)(c1ccc(OC)cc1)=CC(=O)N(C1CCCN(C(CC(CCC)O)=O)C1)C 25829,C1(CNC(C(=O)NCC(F)F)=O)CCN(C(C23CC(CO)(C2)C3)=O)C12CCC2 25830,Cc1cc(C2CCCO2)cc(C(=O)NC(CNC2(C3CCN3)CC2)CC(C)C)n1 25831,c1(CC)cc(C(=O)NC2CC(NC(c3nn(C)cc3N)=O)CC2O)n(C)n1 25832,c1(C(=O)OCCOCC2CC2)[nH]n(-c2ccccc2)c(=O)c1Br 25833,N1(C(C2CC(=O)N(c3ccccc3Cl)C2)=O)C2CCC1CC1(C2)CC1(F)F 25834,c1(CC(=O)NC2C(NC(Cc3nnc(C)s3)=O)CCCC2)cccc(O)c1F 25835,CCCS(=O)(=O)CC(=O)N(C1CC1)CC1CCN(C(C2CCCS2(=O)=O)=O)CC1 25836,CC(CS(C)=O)C(=O)NCCOCCN(C)C(c1cc(N)cc(O)c1)=O 25837,c1(C(=O)NC23C(CN(C(CSC)=O)C2)C3)c(Cl)oc2ccccc12 25838,C(=O)(CCCCCC#N)NC(C)CC(C)NC(c1cccc(OC(F)F)c1)=O 25839,C(=O)(C1=C(Cl)CCOC1)N1CCC(C(=O)NCC(CC)C(C)(F)F)C1 25840,C(=O)(CC(C)(C)O)NCC(C)NC(C1(n2cncn2)CC1)=O 25841,CC1(C)CC(NC(=O)CCC2CCOCC2)CN1C(=O)CN1CCCCCC1 25842,N1(C(C2(CCCC)CC2)=O)CCN(C(c2cc(Br)sc2C)=O)C(C)C1 25843,C1(C(C)NC(=O)C(=Cc2cn(C)cn2)F)CN(C(=O)CCc2csnn2)CCO1 25844,n1(CCC(=O)NCC(C2CC2)NC(=O)CC2CCCCC2)cnc([N+](=O)[O-])c1 25845,C1(C(C)NC(C(C)(C)OC)=O)CCCN(C(=O)CC(C)(F)F)C1 25846,C=CCCC(C(=O)NC(C(N)=O)C1CCCC1)NC(c1cc(Cl)n[nH]1)=O 25847,Cc1cc(-c2cn(CC3C(C)CCN3C(C3CC=CCC3)=O)nn2)c(Cl)cc1F 25848,c1(C(N2CC(CCNC(C(CCCC)C)=O)C(C)C2)=O)nccn2cc(C)nc12 25849,N1(C(c2cc(OC)cc(CC)c2)C(=O)OCC2CC2)CC2C3C=CC(O3)C2C1 25850,C1(C2CN(c3nnc(C)s3)C2)CN(C(c2coc(-c3ccccc3)c2)=O)CCO1 25851,N1(C(C(CC#C)O)=O)CC2(C1)CN(C(c1cccc(C(F)(F)F)c1Br)=O)C2 25852,C1(C)(NC(C(C2CN(C(c3cccc(CC)n3)=O)C2)OC)=O)CCCCC1C 25853,C1(NC(C(=Cc2ccncc2)C)=O)CS(=O)(=O)CC1NC(c1cnc[nH]1)=O 25854,Nc1cc(F)ccc1C(=O)NCC(O)CNC(C1CCC(CCO)CC1)=O 25855,C1(NC(c2c(C)nc(CCC)s2)=O)C(C)CCN(C(=O)CC(C)(C)O)C1C 25856,CS(=O)(=O)CC(=O)NC1CCOC(C(=O)NOCC(=O)OC(C)(C)C)C1 25857,N1(C(CC(CC)(F)F)=O)Cc2nccn2CC(NC(=O)C(F)C(C)C)C1 25858,c1(C(=O)NC2CCCCCN(C(CC=C)=O)C2)n[nH]c2cc(Br)ccc12 25859,Cn1cnc(I)c1CNC(N1CCC(c2nc[nH]n2)CC1)=O 25860,Cc1cncc(C=CC(=O)N(C)CCC2CCN(C(=O)CCS(C)(=O)=O)CC2)c1 25861,Cc1[nH]nc(C(=O)N(C)CC2CN(C(c3ocnc3C(F)(F)F)=O)CCO2)c1F 25862,C(=O)(CCCC(C)O)N(CC(C)(C)Nc1nccc(C(=O)OC)n1)C 25863,N1(C(c2cc(COC)no2)=O)CC2CN(C(=O)C(C)CS(C)(=O)=O)CC2C1 25864,c1(C(=O)NCC2CC(C)(C)CN2C(=O)Cn2cnc(=N)[nH]2)cc2c[nH]cnc-2n1 25865,Cc1c(C(N2CCC2CNC(=O)C(F)CC(C)C)=O)sc2[nH]cnc(=S)c12 25866,c1(C(=O)NC(CN(C(c2c[nH]cc(Cl)c2=O)=O)CC)C)n[nH]c2cc(Cl)ccc12 25867,N1(C(CCOC)=O)CCC(NC(c2cc(C(C)C)n(C)n2)=O)C1c1ccccc1 25868,N1(C(COC2(C)CCC2)=O)CC2CC1C2NC(=O)C(C)(C)C1CCCO1 25869,CC1CCn2cc(C(=O)NCC(CO)NC(c3c[nH]c(Br)c3)=O)nc2C1 25870,N1(C(c2ccc(CO)nc2)=O)CC=CC(C(N2C(CO)CCC2CO)=O)C1 25871,CCCCS(=O)(=O)CC(=O)NCCCN1CCN(C(=O)C2=CS(=O)CCC2)CC1 25872,C#Cc1ccc(C(=O)NC2CCN(C(c3c(C)ncn3C)=O)CC2O)c(OC)c1 25873,C1(CNC(C2CN(C(N)=O)C2)=O)CN(C(c2cc(F)ccc2Cl)=O)CC12CC2 25874,C1(C(N(CC(C)(C)N(C)C)C)=O)C2CC2CN1C(=O)C(C)OC1CCCC1 25875,Cc1ncsc1C(=O)NCCOCCC(=O)N(C)CCc1cnc[nH]1 25876,N(C1COc2ccccc21)CCOC(C)C(=O)NC(CCSC)C(=O)NC.CO 25877,c1(C(C)(C)C)cccc(C(c2nnnn2C2CCCC2)NCCc2cccs2)c1 25878,N1(C(C)C(=O)NC(=O)NC(C)(C)C)CCCC(C(=O)Nc2cc(O)n(C)n2)C1 25879,N12CCCC(C1)C2=O.Cc1ncsc1CCNC(=O)NC(C)C 25880,C(C)(C)(C#Cc1cn(-c2ccncc2OCC)nn1)NC(C(CC)CC(C)C)=O 25881,C(C)(CCCCNC(C12CC(C)(C1)C2)=O)NC(c1c(C)ocn1)=O 25882,C1(C(N(C)CCNC(c2sncc2Br)=O)=O)CN2CCC1CC2 25883,c1(NC(C2C(NC(c3ccc(C)s3)=O)CC2)=O)cc(F)c(O)cc1C 25884,Cc1cccc(C2(C(=O)NC(C)(C)CCNC(C3CN(C)C(=O)N3)=O)CCC2)c1 25885,C1(NC(CC2(N(C)C)CCCC2)=O)CCOC(CNC(=O)COCCCF)C1 25886,N1(C(CCCS(C)(=O)=O)=O)CCC2(CC1)CCN(c1ncns1)C2 25887,c1(C(=O)NC(C2CN(C(=O)CCCCC(N)=O)CCO2)C)cc(Cl)c(F)cc1F 25888,c1(NC(C(C)(C)CCl)=O)ccn2c(C(F)(F)F)nnc2c1 25889,c1(C(=O)NC2CCCCN(C(CC(=C=C)C)=O)C2)c(F)cc(O)cc1F 25890,c1(C(N2CCC(N(C(=O)C3=CC(C)(C)C3)CC)C2)=O)ccc2c(c1)C(=O)NC2=O 25891,c1(OCCC(=O)NC2(CC=C)CCN(C(C3C=CCC3)=O)C2)cc(Cl)ccc1Cl 25892,N1(C(=O)CN2CC3CC2CS3=O)CC(=O)Nc2ccccc21 25893,c1(CC)nn(C)cc1C(=O)NCC=C1CCN(C(C2(OC)CCCC2)=O)CC1 25894,c1(OC)ccc(F)c(C(=O)NC2CC3(C2)CC3NC(c2ncccn2)=O)c1 25895,C1(NC(CCc2c(C)noc2)=O)CC(C)N(c2nc(-c3ccccc3)ns2)C1 25896,N1(C(CCC2N(C(C3C=CCCC3)=O)CCC2)=O)CC(O)C(O)C1CO 25897,S(=O)(=O)(c1ccccc1F)NCC(=O)NCCCNC(CCCCNC(C)=O)=O 25898,c1(C(=O)NC(CNC(C(C)C2CC2)=O)(C)C2CCC2)cc(-c2cnn(C)c2)on1 25899,c1(C(=O)NCC2N(C(c3cc(C)n(C)c3C)=O)CC=C2)ccc(S(N)(=O)=O)cc1 25900,C12CN(CC1(C)C)C2=O.c1(C(N(C(CC)C)C)=O)ccc(O)nc1Cl 25901,C1(NC(CCCC2(C)N=N2)=O)CCN(CC2CCC(C(=O)N)CC2)CC1CO 25902,C(C(C)(C)C(C)(C)O)NC(C1N(C(C(C)=CCC)=O)CCC=C1)=O 25903,N1(C(c2nnn(C)c2C(F)F)=O)C2CCC1CC(NC(=O)CCC1CC1)C2 25904,C(=O)(C1CCc2nccn21)NCCCCCCC(=O)N1CC(C)(C(=O)OC)C1 25905,C12(C(=O)NCCN(C3CC3)Cc3cc(C)[nH]n3)COC(C1)C(N)C2 25906,C1(C(=O)NC2CCCN(C(C)=O)C2)CC(C)CN(C(=O)COCC(C)C)C1 25907,c1(OC)c(O)ccnc1Oc1ccccc1-c1co[nH]c1=O 25908,c1(C(=O)NC(C)C(C)NC(=O)C(C)n2cccn2)cc2occc2s1 25909,C(=O)(C(CO)C(C)(C)C)N(C(CNC(CCCC=C)=O)C1CC1)C 25910,c1(OC)ccc(C(N2CC(F)CC2C(=O)Nc2ccnc(Br)c2)=O)c(Br)n1 25911,C=CC(CCC)CC(=O)NC1C2CCN(C(=O)Cn3cnc(Br)c3)C12 25912,C(C(O)CC(=O)N(C)CC1(O)CCC1)NC(CNC(CC(C)C)=O)=O 25913,N#Cc1cnccc1N1CCCC1CN1CCCC1.C1(=O)CNC(=O)N1 25914,c1(C(N2C(C(C)NC(=O)CC3OCCC3(C)C)CCC2)=O)cc2ccccn2c1 25915,c1(C(N(C)CCNC(C2(C)CCCC2O)=O)=O)c[nH]c(=NCC(F)(F)F)cn1 25916,Cc1oc(S(C)(=O)=O)cc1C(=O)NC(C(C)NC(c1ccc(F)s1)=O)C(C)C 25917,N1(C(=O)CCc2cc(F)ccn2)CCC2C1CCN2C(=O)CCC12CC(F)(C1)C2 25918,c1(NC(c2c(CC)cc(Br)cc2)=O)ccc(S(=O)(=O)N2CCOCC2)cc1 25919,CC(C)CC(CNC(=O)C1=C(Cl)CCC1)C(=O)NC1CCCC(O)C1 25920,Cc1ccc2[nH]c(=NC(C)C3CCN(C(C4CCC=CCCC4)=O)CC3)sc2n1 25921,c1(CNC(CC(CC)C2CCC2)=O)cccc2c1CN(C(C1(CO)CC1)=O)C2 25922,N1(C(Cc2cc(C)cc(Cl)c2)=O)CCCc2c(O)cccc21 25923,C(=O)(CS(=O)(=O)CC1CCCO1)N1CCC(N(C(=O)CCCc2cccs2)C)C1 25924,c1(SC)ccc(C)c(C(N2CCCCC2CCN(C)C(c2nnc(C)s2)=O)=O)c1 25925,N1(C(COCCC=C)=O)CCN(C2CCCN(C(=O)CSC(F)(F)F)C2)C(=O)C1 25926,Cc1ncc2n1CCC(C(N1CC3(CCN3C(=O)C(c3ccccc3)C)C1)=O)C2 25927,c1(C(=O)Nc2cc(-c3cnn(CCO)c3)ccn2)c(F)cccc1Br 25928,N1(Cc2ccc(CNc3ncc(C)o3)cc2)C(=O)c2ccccc2C1=O 25929,c1(NC(C2CCCC(NC(c3n(C)cnc3)=O)C2)=O)cc(Cl)ncc1[N+](=O)[O-] 25930,c1(C(N2C(C)(C)C(CNC(=O)CSc3nc[nH]n3)CC2)=O)ncnc2c1CCC2 25931,CCCC(C)(C)CC(=O)NC(C1(O)CN(C(c2ccsc2SC)=O)C1)C 25932,Cc1ccc2cc(C(=O)NC(C3(O)CN(C(C4(C#N)CC=CC4)=O)C3)C)[nH]c2c1 25933,C1(OC)CN(C(=O)CC2(O)CCOCC2)CC1NC(c1coc(C2CCC2)n1)=O 25934,N1(C(C2(CCCC)CC2)=O)CC2CC1CN2C(=O)COCC(=O)NC 25935,CN1CC2C(NCC(=O)N=S(C)(C)=O)CCCN2C1=O 25936,c1(C(=O)NC2C(OC)CN(C(C3(C(=O)OC)C=CCC3)=O)C2)snc2ccccc12 25937,c1(C(N(CC(CN(C)C)O)C)=O)sccc1CNC(c1cnn(C2CC2)c1)=O 25938,C1(NC(CN(C(=O)CC(C)n2cccc2)CCC)=O)CC12CCOCC2 25939,c1(NCC2CCC(=O)NC2)ccc(S(=O)(=O)NC(Cc2nccs2)CO)cn1 25940,c1(C(=O)NC(CCN(C(C(C)CC(N)=O)=O)C)C(C)(C)C)ccc2occc2c1 25941,CN1CC2CCC(NC(c3ccc(CN(c4ccccc4)C)cc3)=O)C2C1 25942,c1(C(N(C(C(=O)NCC(C)Cc2cn[nH]c2)C)C2CC2)=O)cnn(C)c1 25943,c1(C(=O)NC2CCCC(CNC(C(C)(F)F)=O)C2)ncc(C(N)=O)cc1Cl 25944,c1(SCC(=O)NCC(CCOC)NC(C2CCC(CO)CC2)=O)cccc(C)c1 25945,N1(C(c2ncc(OCC)nc2)=O)CC2CN(C(=O)CCc3cccc(C)n3)C2C1 25946,c1(C(=O)NC2CC(C)SC2)c(CNC(c2cc(=N)[nH][nH]2)=O)cnn1C 25947,CCCC(C(=O)NC(C(=O)N1CCC(CC2CCC2)C1)C(C)OC)OCC 25948,C1(CN(C(C2(COC)CCOC2)=O)C)CCN(C(=O)CC(C)c2ccco2)CC1 25949,Brc1cc(I)c(CN2CCC(N3CCC3)CC2)s1 25950,n1(CC(=O)NC(C)CC2CN(C(=O)CC3CC3)C2)ccc2ccccc12 25951,N1(C(Cc2cc(C)ncc2)=O)CC(CNC(=O)C(F)=CC2CC2)C(C)(C)C1 25952,c1(CCCN2CC2=O)ccc(C(=O)O)cc1.C(CC(F)(F)Cl)SCC.CC(=O)O 25953,Cc1nc(O)[nH]c1C(N1CC(C(N)=O)(CNC(=O)C(C)OC2CCCC2)C1)=O 25954,c1(OC)ccc(N2CCCCC2)cc1NC(N1CCOC(C(F)F)C1)=O 25955,Cc1nnc(CC(N2CC(NC(c3cnc(C)s3)=O)C2)=O)o1 25956,CC(Cc1nncn1C)N=c1[nH]c(N(C)Cc2cccnc2O)nc2ccsc12 25957,Cc1cccc(CC(=O)NC2CC(O)CN(C(=O)CN3CCC(C)CC3)C2)c1C 25958,N1(C(c2n(C)ccn2)=O)CC2(CC(NC(C3(C(F)(F)F)CC=CC3)=O)CO2)C1 25959,CC1CCc2sc(C(N3CCC(C(C)(C)NC(c4csc(Cl)c4)=O)C3)=O)cc2C1 25960,c1(C(N2CCC3C(CCN3C(C3C=CCN3)=O)C2)=O)c(Cl)ccc2c1OCO2 25961,c1(CNC2CCC(C(=O)NCc3cn[nH]c3)C2)ccccc1C(F)(F)F 25962,C(CC(C)(C)C)(C(=O)NC(C)C(=O)Nc1cc(C)c(F)c(C)c1)OC 25963,c1(NC(C2CCN(C(C3CCCO3)=O)C2)=O)ccccc1NCC1CC1 25964,C(C(C)(F)C(C)(C)F)NC(CCCN(C(c1n(CC)c(O)nc1)=O)C)=O 25965,C1(CC=C)(N(C(=O)Cc2cocn2)CC)CC2CCC(C1)N2C(=O)CCC 25966,N1(Cc2ccc(C#C)s2)CCCN(C(c2noc(C)c2CC)=O)CC1 25967,N(C1CN(C(c2cncn2C2CC2)=O)Cc2ccccc21)C(CSCC#C)=O 25968,C(=O)(C(C(C)(C)C)NC(C1CN2CCN1CC2)=O)N(C)Cc1cocn1 25969,C(C(C)(C)C(=O)N1CC(C(N)=O)(CNC(c2nnn(C)c2C(F)F)=O)C1)SC 25970,c1(OC)cncc(C=CC(=O)NC2(CN(C(=O)CN3CCCC3C)C)CC2)c1 25971,Cc1cc(C(=O)NC2CCCC2NC(c2ccnc(O)c2)=O)nc(O)n1 25972,c1(C(N2CCC(C3CC3)C2)C(=O)NCC(C)C)ccc(Oc2ccccc2)nc1 25973,c1(CC)cc(C(=O)NCC(CC)NC(C2CCCCC2(C)C)=O)ccc1OC 25974,c1(C(N2CC(C(=O)Nc3cc(Br)cc(Br)c3)C(O)CC2)=O)cccc2c1CCC2 25975,CCC(CCC(=O)NCC(CC(=O)NCC(C)(CC)CO)C1CCC1)OC 25976,C1(CCN(c2cnn(C(F)(F)F)c2)C(=O)C=CC2CCCC2)CCCN(CCO)C1 25977,C(C1=CCN(C(C2CCC(F)CC2)=O)CC1)NC(C(C)C1CCCO1)=O 25978,C(=O)(CCCCCCCCC1CC1)NCC(CC)(C)NC(c1ccccc1C)=O 25979,c1(OC)cc(OC)c2c(c1)CCN(C(=O)CC1CCCC(C)C1)C2 25980,c1(C(=O)NC2CN(C(CNC(CNC(C)=O)=O)=O)C2)ncc(N)cc1Cl 25981,CCCCCCCCCCCCN(C(=O)CC1CCN1C(=O)OC(C)(C)C)C 25982,c1(C(N2C(C)(CNC(C3(C)C(C)CCC3)=O)CCC2)=O)cn2c(n1)CCCC2 25983,CC(C)CC(C)C(=O)N1CC(NC(C2(Cc3cccc(F)c3)CCC2)=O)C(O)C1 25984,CC1(C)CC(C)(C)CC(O)(CNC(N2CCC(O)C2c2ccccc2)=O)C1 25985,C1(CNC(CC(=O)NC)=O)CN(C(=O)C=CS(C)(=O)=O)CC(C)(C)O1 25986,c1(-c2ccnc(NC(N(CC(=O)NC)C)=O)n2)cccc(S(C)(=O)=O)c1 25987,C1(C(=O)NCC(CCOC)NC(C2COCCC2(F)F)=O)CC2(C1)OCCO2 25988,c1(C(N2CCC(N(C(=O)CCc3cccnc3C)CC)C2)=O)cc(C)ccc1N 25989,C12(CNC(Cc3c(Cl)cn(C)n3)=O)CCC(NC(=O)COCCN(C)C)(CO1)C2 25990,C1(NC(Cc2c(C)ncs2)=O)C2CC3C(C2)C13C(=O)NCCC1CC=CCC1 25991,c1(C(N2C(C)C(NC(=O)C(N)=O)CCC2)=O)cc2c(nc1O)CCC(C(C)C)C2 25992,CCC(C)(C(=O)N1CCC(C)N(C(=O)CCc2cc(C)no2)CC1)C(F)F 25993,C(=O)(CS(=O)(=O)CC(=O)NCC1CCN1C(=O)Cn1nc(C)nc1C)OC 25994,C(C(C)(C)C#CC(=O)N1CC(O)(C(F)(F)F)C1)NC(C(CC#C)C1CC1)=O 25995,CC1(C)CN(C(=O)C=Cc2cn[nH]c2)CC(CNC(=O)C(F)(F)CC2CC2)O1 25996,N1(C(CC2(C)CCOCC2)=O)CC2CC(NC(=O)CCN3CCOCC3)C(C2)C1 25997,Cn1cnc2c(N3CCCCC(CNC(=O)C(C)(C)C(F)F)C3)nc(Cl)nc12 25998,Cc1nc[nH]c1CC(=O)NCC1CCC1NC(=O)Cc1csc(NS(C)(=O)=O)n1 25999,C(=O)(C(=O)N=c1cc(C)o[nH]1)NCC1C(F)(F)CCN(C(CSCC)=O)C1 26000,c1(C(=O)NCCC(CCC)C)cc(C(N)=O)cc([N+](=O)[O-])c1 26001,Cc1nn2ccccc2c1C(=O)NC(CNC(=O)CSCC(F)F)C(C)C 26002,N1(C(CC(CC)OC)=O)CC(NC(c2cc3c([nH]2)CCCC3)=O)C2CCCC2C1 26003,C(=O)(C(CNC(=O)Cc1coc(C)n1)CC1CCCC1)NCCCCOCC 26004,N1(C(c2[nH]cc(C(C)=O)c2)=O)CC(NC(c2csc(CO)n2)=O)CC1(C)C 26005,c1(OC)ccccc1C(CNC(=O)Cc1ccc(F)cc1)NC(=O)CO 26006,C12(CNC(=O)C(C3CC3)C3CC3)CCCC1N(C(=O)Cn1cnnc1)CCC2 26007,Cc1nc(N2CCC(C(=O)NC3CCC4CC4CC3)CC2)c(C)c(Cl)n1 26008,C1(C(C)(C)O)(CNC(c2ccnn2CC(F)F)=O)CN(C(c2ccccc2)=O)C1 26009,c1(C(N(C)CC2CC(F)CN2C(=O)C(F)=C2CCCC2)=O)cc(N)ccc1O 26010,c1(CCC(=O)NC2(C)CC(NC(CC3C(C)OCC3)=O)C2)ccc(C#N)cc1 26011,c1(C(CC(=O)NC2CC(F)(CNC(c3c(SC)ccs3)=O)C2)O)ccc(Cl)cc1 26012,C1(C(N2CC(N(C(=O)CC3CCC3)C)C2)=O)CCCCC1C1CC1 26013,c1(CC(=O)NC(CNC(COCCOCC)=O)(C)C2CCC2)coc(C(F)F)n1 26014,C1(C(N(CC(=C)C)CC)=O)CCN(C(c2cnn(C)c2Cl)=O)C1(C)C 26015,CC(C)S(=O)(=O)C1CCN(C(CCCCC#N)c2nnnn2CCN(C)C)CC1 26016,C1(CCNC(=O)COC2CCOCC2)CSCCN1C(C1CCC(F)(F)C1)=O 26017,C1(NC(C2(C#C)CCN(C(c3cc(CC)nn3C)=O)C2)=O)CC2C(O)C(O)CC12 26018,c1(C(N2C(CNC(C3COC4(CCC4)C3)=O)COCC2)=O)coc2c1COC2 26019,c1(C(C(=O)NCC(C)(C)OCCNC(Cc2ccc(C)s2)=O)C)cccc(F)c1 26020,N1(C(=O)CC2CC3CC3C2)CCC2(CCN(C(c3ccc4nc[nH]c4c3)=O)C2)C1 26021,N1(C(c2scc(CNC(C3CN(C)C3)=O)c2)=O)CCCC2CC12.O 26022,N1(C(c2c(OC)cccn2)=O)CCC2CN(C(c3ccnc(C)c3N)=O)C(C)C12 26023,C(C)(C(=O)NOC(C)C(=O)OC)NC(c1c(CCC)[nH]cc1)=O 26024,C=CCCCCCCCC(=O)NC1CC1NC(=O)CCSc1nccn1C 26025,c1(C(N2CCC3CN(C(C(F)=CCC)=O)CC3C2)=O)n[nH]c2c1CC(C)OC2C 26026,C1(NC(C(C(C)C)N(C)C)=O)CN(C(=O)C=CBr)CC1C1CC1 26027,C(=O)(C(C)(C)C(F)F)NC(C(C)C)CNC(=O)CCN(C)CCO 26028,c1(NCC2CCN(CCC)C2)cc(=NCc2ccc(-n3ccnc3)cc2)[nH]cn1 26029,C1(C#N)(C(N2CCC(CC(=O)NC3(C)CCCC3)C2)=O)CC(F)(F)C1 26030,C(COC(C(C)C=C1CCN(Cc2cc(CC(C)C)on2)C1)=O)(C(C)(C)C)OC 26031,C12(C(=O)NCCC(=O)OCC)CC(C)(C1)OC2NC(=O)CCCCNC(=O)OC 26032,N1(c2c(CC)nccn2)CC2(C1)SCCC2N=c1[nH]c(Cl)nc(CC)c1Cl 26033,c1(C(=O)NCC(CNC(C2C(C=C)OCCC2)=O)C)cc(F)cc2nn[nH]c12 26034,C(C1=NOC2CN(C(=O)CC3CC3)CC12)NC(c1cc(CC)c(C)cc1)=O 26035,C=CC(CC(=O)NCCCCNC(C1CC1OCC)=O)c1ccccc1 26036,N1(C(C(CN(C)C)(C)C)=O)CCC(C2CC2)(CNC(=O)CCCC2CCCO2)C1 26037,c1(C(C(C)(C)C)N(C)C)nc(-c2cncnc2)nn1-c1ccccc1 26038,C1(NC(c2cnc(C(C)C)o2)=O)CCCN(C(c2coc(C3CC3)n2)=O)CC1F 26039,Cc1nc(NC(C2CCCN2Cc2ccncc2O)=O)cnc1Cl 26040,C1(C(CNC(c2c(C)onc2)=O)(C)O)CCN(C(=O)C(C)OCC(F)(F)F)CC1 26041,N1(C(C(CCNC(C(CC)NC(C)=O)=O)O)=O)CC(O)CC12CCOC2 26042,N1(C(CC2(C)CCOC2)=O)CC2CC1CC2CNC(=O)CCC1CCCOC1 26043,C1(NC(CN(C(COC)=O)C)=O)CN(C(=O)CN(C)C2CC2)CC2(CC2)C1 26044,O=C(C#Cc1ccccc1)NCC1(O)CN(c2ncncc2F)C1 26045,N1(C(c2ccc(CCC)[nH]2)=O)CC(NC(=O)CCS(N)(=O)=O)CC12CCOCC2 26046,c1(C(=O)NCCCC(C)(C)NC(=O)CC2CCOCC2)ccc2nonc2c1 26047,c1(N2CC(C)C=C(C)C2)nc(NCCc2c[nH]nc2C2CC2)c2ccsc2n1 26048,C(=O)(CC(CC1CC1)NC(=O)C(C)OCC1CC1)N1C(C=C)CC1 26049,N1(C(CC2(OCC)CC2)=O)CC(C(=O)N(C2CCOC(C)C2)C)C2(CC2)C1 26050,C(CN=c1[nH]c(=NC2CC2C(C)(C)C)c2ccccc2[nH]1)c1c(C)nc(C)s1 26051,N1(C(c2c[nH]c(C(F)(F)F)c2)=O)CC=C(CCNC(C2(O)CCOC2)=O)CC1 26052,C12(C(=O)Nc3ccc(C)c(C)c3)COCC1CN(C(c1cc[nH]c1C)=O)C2 26053,c1(NCC(CCC)(F)F)ccc(Cl)cc1N1CCN(C)CC1 26054,CN1CCCCC(C(N2CC=CC(NC(c3csc(C(F)(F)F)c3)=O)C2)=O)C1=O 26055,CCCC(CC)C(=O)NCCCN1CCC(NC(=O)C(C)C(=O)OC)C1 26056,CCC(C)C(=O)NNC(=O)C1CC1c1ccc(OC)c(C)n1 26057,N1(C(C2C(CC)OCC2)=O)CC(OC)C(NC(=O)CC23CCCC2C3)C1 26058,c1(CC(C(=O)NCCC(C)N(C)C(c2ocnc2C2CC2)=O)O)ccccc1Cl 26059,N1(C(C2CC3(CCC3)CO2)=O)CC2CC1CCC2NC(=O)C(F)(F)C(F)F 26060,C=CC1CCCN1C(C1(CC)CCN(C(=O)CCOCCCC)C1)=O 26061,c1(C(N2CC3C(CNC(=O)CC4CC5CC5C4)C3C2)=O)ccc2c(c1)COC2 26062,N1(C(c2ccccc2)C)CC2C(CNC(=O)NC(=O)CC3(O)CCCCC3)C2C1 26063,c1(OCC(C(=O)OC(C)C)(C)O)cc(C(N)=O)ncc1Br 26064,c1(CC(N2C(CNC(c3c(C)ocn3)=O)CCCC2)=O)cc2ccccc2s1 26065,Cc1ccc(C(N2CCOCC2CC(=O)NCC2COCCO2)=O)nc1O 26066,c1(SCCNC(C2CC(C)N(C(C(C)(C)C)=O)CC2)=O)ccccc1[N+](=O)[O-] 26067,C(=O)(C(CC(C)C)ONC(C1CC2(CC(=O)C2)C1)=O)NC(CC)C1CCC1 26068,C1(C(=O)NCCN(C(=O)C=C=C(C)C)CC)CCCCN1C(C)C 26069,[N-]=[N+]=NC1CCCCC1C(=O)NCC1CC(F)(F)CN1C(=O)CC1C=CCC1 26070,CCCCCC(O)CC(=O)NCC1(O)CCCN(C(=O)C2=CCCC2(C)C)C1 26071,C1(C(=O)NCC(CC)N(C)C)(SC)CN(C(=O)COCCCN=[N+]=[N-])C1 26072,c1(C(C(=O)NC2C(NC(C(c3ccc(Cl)cc3)C)=O)C2)(C)C)ccc(O)cc1 26073,c1(N(CC(C)C(C)(C)C)C)nc(N2CCCC(C)(F)C2)nc2ccc(Cl)cc12 26074,C1(C(N2CC(CCCCC)C2)=O)CCCC(NC(C2(F)CC=CCC2)=O)CC1 26075,c1(CC)ccc(F)cc1C(=O)NCC12CC1CN(C(C1(CC)CC1)=O)C2 26076,CN1CC2CCC(C1)N2C(C1CCC(O)CN1C(=O)C1=C(Cl)CCOC1)=O 26077,CC1=C(C(=O)N2CCC(N(C)C(C3CCC(N(C)C)C3)=O)C2)CCCO1 26078,N1(C(Cn2c(C)cc(C)n2)=O)CCOC2CN(C(=O)CN3CCCC3)CC12 26079,c1(CC(=O)NCC(CC)(C)NC(c2ncoc2C)=O)cc(Br)ccc1F 26080,c1(C(N(C(CNC(C(CC)c2cccnc2)=O)C)CC)=O)[nH]c(C2CC2)nc1C 26081,C(=O)(CC(C)(C)CC)N1CCC(N(C(C2(NC(C)=O)CCCCC2)=O)CCO)C1 26082,c1(C(N2CCC(F)(CNC(c3c(CC)cccc3)=O)C2)=O)ncc(N)cc1Cl 26083,N1(C(Cc2ccc(C)cc2)=O)CCCC(NC(=O)Cn2cnnc2)CC1 26084,C1(CNC(C(C)NC(N)=O)=O)(CO)CCN(C(=O)C=CCF)CC1 26085,Cc1cc(C2CCN(CC(O)CN(c3ccccc3C)CC(O)CO)C2)cc(C)c1 26086,N1(Cc2occ(C)c2)CCOCC12CN(C(=O)OC(C)(C)C)C2 26087,c1(NC(C2(F)CN(C(c3ccc(C)c(O)c3)=O)C2)=O)c(Br)cccc1[N+](=O)[O-] 26088,N1(Cc2cc(C)c(Cl)nc2)CCN(C(=O)CSc2nc[nH]n2)C(C#N)C1 26089,c1(OC)cc(C(=O)OC2CCCN(C(N3CCCCC3=O)=O)C2)cc(Br)c1 26090,N1(C(c2cncc(C)c2Cl)=O)CCCC(C2CC2NC(C2(N(C)C)CCC2)=O)C1 26091,N1(C(c2cc(COC)on2)=O)C2CCC1CC(N(C)C(c1cnc(SC)s1)=O)C2 26092,N1(C(C2(CCNC(C3(C)CCNC3=O)=O)CC2)=O)CC(O)C(C2CC2)C1 26093,N1(C(CCC#C)=O)CC2(CCCCN(C(=O)C(C)C3CCCO3)C2)C1 26094,N1(C(c2c(CC)occ2C)=O)CCCCC(NC(=O)C(C(C)(C)C)N(C)C)C1 26095,Cc1cnc(C=CC(=O)NC2COCC2NC(=O)CC2COCC2O)[nH]1 26096,c1(OC)cc(C)ccc1C(=O)NC(C1CCN(C(=O)CC=CC(C)(C)C)C1)C 26097,N1(C(CC2C(OC)CC2)=O)CCN(C(c2cocn2)=O)C(c2ncc[nH]2)C1 26098,C1(CNC(c2n(CC)ccn2)=O)CCC2(CN(C(c3csnc3Br)=O)C2)O1 26099,C(=O)(C1CCc2c[nH]nc21)NC1(C(=O)NC(C2CCCCC2)C)CSC1 26100,N1(C(CCC#CC)=O)CCCC(C(=O)N(C)CC2CCOC2)CC1 26101,c1(C(=O)NCCC2N(C(c3c(C)nns3)=O)CCCC2)cc(S(N)(=O)=O)cn1C 26102,Cc1[nH]nc(C(=O)NCC2CCCN(C(C3CC3C)=O)C2)c1C 26103,C1(CCC)CN(C(=O)C(C)Cn2cccn2)CCN1C(=O)C(F)F 26104,c1(C(=O)NCCCCN(C)C(C2CCCO2)=O)c[nH]nc1C1CCCO1 26105,N1(C(CC(C)SC)=O)CCCC2(NC(c3ccn4nnnc4c3)=O)CC2C1 26106,c1(C(N2CCN(C(c3cnn(C(C)C)c3N)=O)C(C)C2)=O)nc[nH]c2ncnc1-2 26107,N1(C(Cn2c(N)cc(C)n2)=O)CCCC(N(C)C(c2ccccc2O)=O)CC1 26108,c1(C(C)C(=O)NCC2(CNC(=O)CC3CC(F)C3)CC2)ccc(F)c(Cl)c1 26109,c1(-c2ccc(SC)c(C)c2)ccc2oc(C(N3CCC(F)CC3)=O)cc2c1 26110,c1(C(=O)OC)noc(C(C)NC(c2cscc2C)c2nnnn2C(C)C)n1 26111,c1(NC(c2c(OC)cncc2)C)ccc(S(=O)(=O)NCC2C3COCC23)cn1 26112,c1(CCC)[nH]nc(C(=O)NC(CNC(=O)C(C)CC)CC(C)C)c1[N+](=O)[O-] 26113,N1(C(c2c(C)onc2)=O)CCN(C(=O)CN2CCSCC2)CC1CS(C)(=O)=O 26114,C1(CNC(C2N(C=O)CCC2)=O)CCCN(C(c2cnc(C(F)F)nc2)=O)CC1 26115,c1(C(=O)NC(C(C(C)C)C)CNC(=O)C2=CCOCC2)c(F)ccc2occc12 26116,O=S(=O)(c1ccc(N2CC34CCC3(COC4)C2)c(F)c1)NCc1cn2ccccc2n1 26117,Cc1ncc(S(N)(=O)=O)cc1C(=O)NC1CCCCN(C(=O)CC2CCC2)C1 26118,C1(CCC)CN(C(=O)CN2CC(C)(OC)C2)CCN1C(=O)C(O)CSC 26119,c1(C(N2CC(C(=O)NCc3cc(C)on3)OCC2)=O)cc(Cl)cnc1Cl 26120,C#CCC(C)(C(=O)N1CCC(CN(C)C)C1(C)C)NC(c1ccc(F)c(C)c1)=O 26121,C(=O)(C1=COCCO1)NC1C(CNC(c2cc(C(C)=O)cn2C)=O)C1 26122,N1(C(CN(C(=O)CC2CC3CCC2C3)CC#C)=O)CCC(C(=O)OC)CC1 26123,C1(NC(C(c2cccc(Br)c2)C)=O)(CNC(=O)CC2(O)CC2)CCOCC1 26124,c1(N2CC3(CN(C(CC(CC)Cn4cncn4)=O)C3)C2)c(F)cccc1[N+](=O)[O-] 26125,C1(C(=O)OC)OC2(C)CC1(C(=O)NCC1C(C(=O)NCc3ccccc3)C1)C2 26126,c1(N2CCCC(NC(c3c(C)nn[nH]3)=O)C2)ccc(Cl)cc1[N+](=O)[O-] 26127,C1(OC)COCCC1Nc1cccc(Cn2ccnn2)c1 26128,c1(C(=O)NC2C(NC(CSC(C)(C)C)=O)CS(=O)(=O)C2)ccc2nncn2c1 26129,N1(C(C2(N(C(C(C)NC(C)=O)=O)C)CC2)=O)CCC(CO)C1(C)C 26130,C1(CN(C)C(c2ccc(F)s2)=O)CCN(C(C2(O)CCC2)=O)C1 26131,S(=O)(=O)(c1ccc2ccccc2c1)Nc1ccn(C)n1.C1(=O)CCN1 26132,C(=O)(CP(C)(C)=O)NCC(CN(C(=O)C(C)O)CC)(C)C 26133,CCCCCCC(CC)C(=O)NCC1COCCN(c2nccn3nnnc23)C1 26134,C(N=c1[nH]c(=NC(CCO)c2ccccc2F)[nH]c2c1SCC2)C1(C)CCC1 26135,C1(CN(c2ccc(Cl)o2)C(=O)NC(c2nnnn2C2(C)CC2)C)CCC(F)(F)CC1 26136,N1(C(c2ccon2)=O)CCC2C(CCCN2C(=O)Cc2cnc(C(F)(F)F)s2)C1 26137,C(=O)(C1CCCc2ncc(C)n21)N1C(CNC(c2c(OC)ccc(OC)n2)=O)CC1 26138,CCS(=O)CC(=O)NCC(=O)NCC(=O)NC(c1nccs1)CC 26139,CCC(C)C(C)(O)CNC(C1CC(C)CN(C(=O)Cc2ccc[nH]2)C1)=O 26140,c1(-c2cn(C(F)(F)F)nc2)nc(=NCc2ccn(C3CCC3)n2)[nH]cc1Br 26141,CCCCCCCCC(=O)NC(C)CN(C(=O)Cn1cc(F)ccc1=O)CC 26142,C1(NC(C(=O)NC(C)C)=O)CCC(F)(CNC(c2csc(Cl)c2)=O)C1 26143,C1(C(N2C(C)(CNC(c3nsnc3O)=O)CCC2)=O)CCCC1S(C)(=O)=O 26144,C1(CNC(CCCC)=O)N(C(c2cc(Cl)ccc2CC)=O)CCC1(C)C 26145,c1(OC)ccc(Cl)c(C(=O)N(C2CN(C(=O)Cc3ccc(O)cn3)C2)C)c1 26146,C1(C(=O)NCC2N(C(CC3CN(C)C3)=O)CC(F)C2)CC1C1CCCC1 26147,N1(C(C2(C=C)CCC2)=O)CC2CC(NC(=O)C(C)S(N)(=O)=O)C2C1 26148,N1(C(CC(C)c2cccnc2)=O)CCCCC1CCCNC(c1cncn1C)=O 26149,C(=O)(CC1=NN(C)C(=O)C1)NC(CC(C)NC(c1cc(OC)n(C)n1)=O)C 26150,N1(CC)CCC(n2nc(-c3cncc(F)c3)nc2COC)CC1 26151,C1(N(C(COC(C)=O)=O)C)CCCC(NC(=O)Cc2cnn(C)c2C)C1 26152,C12CC(=NO1)C(=O)NC2.N1(C(c2c(COC)cc[nH]2)=O)CCC(C(=O)OC)C1C 26153,C1(CC(=O)NC2CC2NC(c2cncc(C(F)(F)F)c2)=O)CN2CCN1CC2 26154,C1(NC(=O)OC(C)(C)C)CC2CC(NC(C3(O)CN4CCC3C4)=O)C1C2 26155,[N-]=[N+]=NC1(C(=O)NCC(O)CF)CCN(C(=O)CC2CCOC2=O)C1 26156,S(=O)(=O)(CCC(F)(F)F)NC1CN(C(C2CC2(F)F)=O)CC1F 26157,c1(NC(N2CCC(C)(c3ccccc3)C2)=O)c(I)cc(F)c(Br)c1F 26158,C1(OCC)(OC)CCC(C(c2nnnn2CCC2CC2)NC(C)CC(C)C)C1 26159,N1(C(CC2(C)CCN2C(=O)CC2CC(F)(F)C2)=O)CCOC(C)(CO)C1 26160,C1(C(=O)NCCc2cn(CC)nn2)C2CCC(C2)C1NC(C1(SC)CCC1)=O 26161,N1(C(c2cnc(C(C)C)nc2)=O)CC2CC(NC(c3cc4sccc4[nH]3)=O)C1C2 26162,N1(C(C2CC(C)N2C(c2ccc(=N)[nH]n2)=O)=O)CCCc2occc2C1 26163,C1(NC(COC2C(C)CCCC2)=O)CCN(C(=O)CS(C)(=O)=O)CC1O 26164,C1(NC(C(CC)C)=O)CCC2(CC1)CN(C(c1cscc1Cl)=O)CCO2 26165,C(CC(C)NC(=O)CCC1CC1(C)C)N(C(COC)=O)C 26166,C(CC(C(=O)NCC1CC1)NC(=O)C=CCOC)=CC 26167,c1(C(N(CCCNC(=O)CN2CCOCC2=O)C(C)C)=O)cc2ccsc2n1C 26168,c1(C(C)N(C2CS(=O)(=O)C2)C(=O)C2CC2)cccc(F)c1 26169,CC(N=c1cc(C(=O)O)n2[nH]cnc2n1)C(=O)N1CCc2ccccc21 26170,C1(NC(c2c(C)nc(CCC)s2)=O)CC2(CCN(C(=O)CCOC(C)C)C2)C1 26171,Cc1cccc(C(=O)NCC2(CNC(=O)C=CC3CCC3)CCCC2)c1[N+](=O)[O-] 26172,N1(C(C2N(C(C)=O)CC(O)C2)=O)CCN(C(=O)C(F)(F)C(C)O)CC1CO 26173,c1(C(=O)NC23C(CN(C(CNC(C(C)CO)=O)=O)C2)C3)ccc2c(c1)CCCC2 26174,C1(NC(C2CC(=C)C2)=O)CCCCC1CNC(=O)CCC1(C)CC1 26175,Cc1ccc(CC(=O)NC(CNC(C2CC(n3ccnc3)C2)=O)C2CC2)cc1C 26176,c1(CN(C(c2cscc2C)C(=O)NCC(=C)C)C)cccc(OCC(F)F)c1 26177,C1(C(=O)OC)CC2CN(C1)C(=O)C(C)O2.c1(C(=O)OC(C)(C)C)ccccc1 26178,CCC(C)CCC(=O)NCCOC1CN(C(=O)CCCc2ccc(C)s2)C1 26179,c1(C(N2C(CCNC(C3CCO3)=O)CCC2)=O)csc2ccc(F)cc12 26180,N1(C(c2c[nH]c(=NC)s2)=O)CC(NC(=O)C(Br)=C(C)C)CC(C)(C)C1 26181,c1(C(=O)NCC2C3N(C(C4CC(OC)C4)=O)C(CC3)C2)c(Cl)c([N+](=O)[O-])nn1C 26182,CCC(CCC(=O)N(CC(C1CCC1)OC)C)NC(c1ccc(F)c(O)c1)=O 26183,C1(C)(CNC(C2C(CNC(c3cc(COC)no3)=O)C2)=O)CNC(=O)O1 26184,c1(CC(=O)N(C)CCNC(C2(P(C)(C)=O)CC2)=O)ccc2c[nH]nc2c1 26185,c1(SC)c(C(=O)NC(C2CCOC2)CNC(=O)CN2CCCC2=O)cccc1F 26186,c1(C(=O)NC2C(C)(C)C(=O)NC2)cccc2oc(O)nc12 26187,CCCCCC(=O)NCC(C1(O)CN(C(c2ncn(C)n2)=O)C1)(C)C 26188,c1(N2CC(O)(CNC(C(CC)Oc3cccc(C)c3)=O)C2)nc(Cl)c(C#N)s1 26189,C1(C(=O)NCCCc2n(C)nnn2)CCN(C(c2ccc(=O)n(C)c2)=O)C1(C)C 26190,n1(CC(=O)N(C(CNC(=O)OC(C)(C)C)C2CC2)C)cc(Cl)c(C(F)(F)F)n1 26191,C1(C(=O)NCC2(CC)CC2)CCN(C(=O)COCC2CCCO2)C1 26192,c1(CNC(=NCC)NCC23COCC2C3(F)F)ccc(OC(C)(C)C)nc1OC 26193,C12(CNC(=O)C=Cc3cscn3)CCC(CC1)N2C(c1ncc[nH]c1=O)=O 26194,C1(C)(CNC(c2ccc(C(C)C)cc2)=O)CCC(NC(C2CCC3CC23)=O)CC1 26195,c1(CCCC(=O)NCCC(C)NC(C2COCCO2)=O)ccc(F)c(F)c1 26196,CC1CCN(C(C2(F)CCN(C(=O)CCN3CCC3)CC2)=O)CC1O 26197,C(C1CN(C(c2coc(C(F)F)c2)=O)CC1C(=O)NC1(CO)CCCC1)=CC 26198,CCCCC(CC)C(=O)NC1CN(C(c2cccc(C(N)=O)n2)=O)CC12CC2 26199,C(=O)(C(C(C)(C)C)n1cc(C2CN(C(c3cnn(C(C)C)n3)=O)C2)nn1)OCC 26200,C(=O)(CS(=O)(=O)C1CC1)NCC1N(C(C(C2CCOCC2)OCC)=O)CC=C1 26201,c1(OC)ccc(C(=O)N(CCC(C)NC(C2(C)CC2(C)C)=O)C)cc1S(N)(=O)=O 26202,N1(C(c2c(Cl)ccc(C#C)c2)=O)CC2(C1)C(NC(=O)C(O)C=C)CCS2(=O)=O 26203,Cc1nc2c(NC(C3C=CC(NC(c4cc(F)cnc4Cl)=O)C3)=O)cccn2n1 26204,N1(C(=O)CN2CCOCC2)CC(C2CCCCN(C(=O)C(F)(F)CO)C2)C1 26205,CON1CCC(C(N2CCCC2CC(=O)NC(C)CN(C)C(C)C)=O)CC1 26206,C1(CC(=O)NCCCN2CCCC2=O)C=CC(NC(=O)CC(C2CC2)C2CC2)C1 26207,c1(OC)cc(OC)cc(CN2CCCCC2C(=O)Nc2nc(Cl)nc(Cl)n2)c1 26208,CC1CCC(CNC(=O)COCC2CCCO2)CN1C(=O)C=Cc1nccs1 26209,Cc1sc(Cl)c(C(N2CCCC(C)(NC(=O)CCNC(C3CCC3)=O)C2)=O)c1C 26210,N1(C(CCC=CCC=C)=O)CCN(C(C2COCCN2CC)=O)C(C)C1 26211,C1(COCCCOC)CN(C(=O)C=Cc2ccccc2)CC12CC2.C1CC(=O)N1 26212,C(=O)(CC1=NNC(=O)C1)NCC1C(OCC)CN(C(=O)COCC2CC2)C1 26213,c1(C(N2CC(NC(C)=O)CC(C)(C)C2)=O)nnn2cc(C)nc(O)c12 26214,N=c1ncc(C(=O)NCC2(C(F)F)CCN(C(=O)Cc3ccc(F)cc3)C2)c[nH]1 26215,C(CNC(C)=O)(C(C)C(C)C)NC(C1(OCC)CCOCC1)=O 26216,N1(C(C(CC)C(F)(F)F)=O)CC2(C=C(C(=O)NCC3CCSC3)CO2)C1 26217,Cc1cc(C)n(CCCCNC(=O)CC2CCN(C(c3ccco3)=O)C2)n1 26218,C(C#N)(C(=O)C(C)(C)CNC(c1ccc(C)cc1)=O)c1ccc(OC)cc1 26219,c1(OC)cc(C(=O)NC23CCC(CN(C(C4CC4(F)F)=O)C2)C3)sc1S(N)(=O)=O 26220,N1(C(C=CC=CC)=O)CC(O)(C2(CNC(c3ccc(=NC)[nH]c3)=O)CC2)C1 26221,Cc1nscc1C(=O)NC(Cc1ccoc1)C(=O)NCC(C)C#N 26222,N1(C(C2C(C=C)C2)=O)CC(CNC(=O)C(=O)N(C)C)(COC)C1 26223,c1(N2CCC(OCC)C2)ccnc(NC(Cc2ccco2)CO)n1 26224,S(=O)(=O)(c1cn(C)nn1)NC(=O)NC(c1cccc(C)c1OC)c1ccccc1 26225,c1(C(=O)NCC(C)N(C(=O)COc2ccc(F)cn2)C)cnc(Cl)cn1 26226,C(Cn1cccn1)(C(=O)NC(c1nc(=O)o[nH]1)C)NC(C(C)=C(C)C)=O 26227,c1(C(=O)NC2C(CNC(C(CCC)(C)CC)=O)CC2)ccc2nccc(C)c2c1 26228,c1(CC(=O)NC(CO)C2CC2)cc(Cl)ccc1Br.c12ncccc1NC2=O 26229,C1(C(=O)NCCCC(C)CO)CC2CN(C(=O)C=Cc3cc[nH]n3)CC2C1 26230,C(CC(C(=O)N1CCC(C)(C(N)=O)C1)NC(c1cccc[n+]1[O-])=O)N(C)C 26231,c1(C(N2C(CC)C(C(=O)N(C3CC3C3CC3)C)CC2)=O)cccc(C)c1N 26232,C1(CCC)CN(C(=O)Cc2csc(Cl)n2)CCN1C(=O)C(C)OCC 26233,N=c1[nH]c(CCC(=O)NCCOC2CN(C(C3CC3Cl)=O)C2)cs1 26234,Cc1cc(C(c2nnnn2C2COC2)NCCn2ncc(Br)n2)ccn1 26235,C1(C(=O)NCC2N(C(C)(C)C)CC2)C=CCN(C(=O)CN2CC(=O)NC2=O)C1 26236,CCCC(C(=O)NC(C)C(=O)NCC(C)(CC)CC)NC(N)=O 26237,N1(c2nc(C)c(F)cn2)CCc2ccc(NC(=O)CC3COCCO3)cc2C1 26238,n1(CC(=O)NC2C(NC(c3c(C)ncn3O)=O)CCCC2)ccc2ccccc12 26239,c1(C(=O)NCC(=O)N(CCNC(C2CCCC(=O)O2)=O)CC)cc(F)cc(F)c1 26240,N1(C(C(c2ccc(Cl)s2)C)=O)CC(NC(C2CCCC(CF)C2)=O)C(C)(C)C1 26241,C1(CCNC(C(C)(C)SC)=O)CN(C(=O)CCc2nnc(C(C)C)o2)CC(C)O1 26242,c1(CC(=O)NC(C2CC=CCC2)C(=O)NCCN(C(=O)OC)C)ccccn1 26243,CC(CC(N)=O)C(=O)NC1CC(CNC(c2cc(C3CCOCC3)nn2C)=O)C1 26244,N1(C(c2n(CC#C)ccc2)=O)CC2CCC2(CC(=O)N(CC)CC)C1 26245,c1(CC(=O)NCC2(NC(c3cccc(F)c3O)=O)COC2)nc2ncccn2n1 26246,N1(C(C(C)NC(=O)OC)=O)CC(CCNC(=O)C(C)N2CCCC2)OC(C)C1 26247,Cc1cc2c(cc1C)C(C(=O)N1CCCC1CNC(c1cnc(N)s1)=O)CO2 26248,N1(C(C(C)=CC2CC2)=O)CCN(C(=O)CNC(C2CCC2)=O)CC1CC(F)F 26249,Cc1cccc(C)c1CC(=O)NC1CC12CC(NC(C13CCCC1C3)=O)C2 26250,CCC(C)C(O)C(=O)NC1CCN(CCNC(=O)C(F)(F)C2CCCC2)CC1 26251,CC1(C)CC2(CC(C(N3CCN(C(c4ccccc4Cl)=O)CC(CO)C3)=O)C2)C1 26252,CC(C)C(CN(C)C)C(=O)N1CCOCC(NC(=O)CCCN=[N+]=[N-])C1 26253,c1(C(N2CC3C(CNC(C(C)=CC)=O)(C3)C2)=O)cccc2cccc(O)c12 26254,c1(C(N2CCC(c3cccc(C#N)c3)C2)=O)c(F)ccc2c1OCO2 26255,c1(NC(c2ccc(CC3CC3)cc2)c2n(C)nnn2)ccccc1OC(F)F 26256,C=Cc1ccc(C(N2CCC(C(=O)NC(C)CN3CCCC3)(OC)C2)=O)cc1 26257,C(=O)(CC(O)CC(C)(C)C)N(C(CC(=O)NC(CCC)C1CC1)C)C 26258,c1(C(=O)NC(CCCNC(CSCC#C)=O)C)ccc(Cl)c(Cl)c1C 26259,C1(NC(C2(C)CC(=C)C2)=O)CCC(F)(CNC(=O)COCC2CCCCO2)C1 26260,CC(C)C(F)(F)CC(=O)N1CCCC(N(C(=O)C(c2ccc(Cl)cc2)C)C)C1 26261,c1(OC)cc(C=CC(N2CC(F)CC2CNC(c2cnc(Cl)s2)=O)=O)ccc1N 26262,Cc1cc(C(=O)NC2CCN(C(=O)CN3CSCC3=O)CC2F)c2[nH]cnc2c1 26263,n1(CC)cnc2c(NCC(C)(C)OC)[nH]c(=NCC(C(C)(C)C)OCCO)nc12 26264,C1(C(=O)NCCCCNC(c2ccc(CN(C)C)o2)=O)CCCCCCC1 26265,c1(-n2c(CN3CCC(O)(CC)C3)ccc2)cn(C)c2ccccc12 26266,N1(C(C2(CC)CCN(C(=O)C=Cc3cncn3C)C2)=O)CC2CCCC(C1)N2C 26267,c1(NC(C2N(C(COCC#C)=O)CC2C)=O)cncc([N+](=O)[O-])c1 26268,C1(NC(CCOCC(C)C)=O)CCC2(CCN(C(=O)CCn3ccnc3C)C2)C1 26269,c1(CN2CC(CC)S(=O)C(C)C2)cnn2cc(Br)cc(C(=O)OC)c12 26270,N1(C(c2n(CCC)ncc2)=O)CC2C(CNC(c3cnoc3)=O)C2C1 26271,c1(OC)cc(C)c(C(=O)NCC2(F)CCN(C(C3COC(=O)N3)=O)C2)cn1 26272,C1(NC(c2c(CC=C)cccc2)=O)CN(C(=O)C(O)C=CC)CC12CCC2 26273,C1(C(F)(F)C(=O)Nc2ccc(OC3CNC3)cc2)(OC)CCCCC1 26274,C=CCC(CC=C)C(=O)N1CCC(C(=O)NC2(C)CCC(C)(C)CC2)CC1C 26275,Cn1nnc2c1CC(C(N1CCC(NC(=O)COCc3nc[nH]n3)C1)=O)CC2 26276,C1(C(=O)NC2CC(N(C(=O)CC3(C(F)(F)F)CCC3)C)C2)CCCOC1 26277,c1(OC)ccc(C(=O)N(C(C)C(=O)Nc2cccc(Cl)c2)C2CC2)nn1 26278,c1(C(=O)NC2C(NC(=O)CNC(=O)CC(F)(F)F)CCOC2)ncc(F)cc1F 26279,c1(C(N)=O)nn(CC(C2CCC23CCNCC3)=O)c(=O)c2ccccc12 26280,C(=O)(C1=COCCO1)NCC(C1CCC1)NC(C1(C(=O)OC)CCCO1)=O 26281,N1(C(c2cnn(CC)c2)C(=O)NC(CC)C)CC(CC(=O)OC)C(O)C1 26282,C1(CCN(C(c2n(CC#C)ccc2)=O)C)CCCCN1C(=O)COCCOC 26283,c1(C(N(C2CCN(C(=O)C(C)(Cl)Cl)C2)C)=O)cnn2cccnc12 26284,CC1(C)CN(C(=O)CC2(CO)CCC2)CC1NC(c1ccccc1F)=O 26285,N1(C(c2ccc(Cl)cc2Br)=O)CCC2(CCN(S(=O)(=O)c3cccc(Br)n3)C2)C1 26286,c1(NCC2C(c3c(C)nn(C)c3C)OCC2)cc(F)cc(F)c1CO 26287,c1(C(=O)NCCOCCN(C(=O)Cc2cc(C3CC3)on2)C)cnnn1C 26288,C(=O)(CCC(F)F)NC(C1(O)CN(C(c2cc(N3CCCC3)ncn2)=O)C1)C 26289,C(C1CCOC1)=CC(=O)NCC1CCN1C(c1cn(C2C=CCCC2)nn1)C1CC1 26290,Cc1nc(=N)[nH]cc1C(N1CCC(N(C(=O)C(C)O)C)C1)=O 26291,c1(CC(=O)NC2CCC(NC(C3C(C)(C(F)F)C3)=O)C2)cccc(Cl)c1 26292,C1(CNC(C(c2scc(C)n2)C)=O)CCN(C(c2cnn(C(C)C)c2)=O)C(C)C1 26293,N1(C(C(CC(C)C)C)=O)CCc2cc(CNC(C3CC3F)=O)ccc2C1 26294,Cc1cc(N(C)C)cc(C)c1CC(N1CCC(=CCNC(=O)CC(C)F)CC1)=O 26295,N1(N(c2ccccc2)C)CC2(CC(NC(C3CC(C)(C)C3)=O)C2)C1.C1(C=O)(N)CC1 26296,N1(C(C(C=C)(C)O)=O)CC(C2CCCN(C(=O)C(c3ccccc3)F)C2)C1 26297,C1(C(=O)NC(CCOC)COC)CN(C(C2CC(C)=NO2)=O)CC1(C)C 26298,Cc1ncnc(C)c1C(=O)NCc1cc(C(=O)NCCC2CCCC2)cs1 26299,O=C1Cc2c(C(N3CC4(CC4)CC3CNC(=O)C(F)C3CCC3)=O)cccc2N1 26300,C1(NC(CC(OCC)OCC)=O)CCN(C(=O)CC2CC(C(F)F)C2)CC1CC 26301,c1(C(N(CCCNC(CC(CCC)C)=O)CC)=O)csc(=NC2CC2)[nH]1 26302,c1(C(C(=O)NCC(CN(C(c2csnn2)=O)CC)(C)C)O)ccc(Cl)cc1F 26303,C(=O)(N1CC(O)CCO1)C1CCCN(C(c2c(NC)nccc2)=O)CC1 26304,C(C1(C)CCOCC1)=CC(=O)NC(C(C)C)(C)CNC(=O)C(C)NS(C)(=O)=O 26305,c1(CC)ccc(C(=O)C(=O)NCC(C2CC2)N(C)C(C2(C(F)F)CCCO2)=O)s1 26306,CCC(CC(F)(F)F)C(=O)N1CC2CC3CC2C1C3NC(=O)CCCF 26307,n1(CCC)cc(C(=O)N(CCCNC(=O)CNC(=O)NCC)C)cn1 26308,Cc1sc(C(=O)NC2CCC(CCNC(=O)Cc3ccn(C)n3)C2)cc1Br 26309,N1(C(=O)Cc2ccc(Cl)s2)CC2CC(C1)CN(C(C1CCCC1)=O)C2 26310,c1(OC(c2ccc(CC)o2)=O)cc(C)ccc1F.C12(CC1)CC(=O)NC2 26311,C1(C(=O)NC23CC(C(=O)Nc4cn(CC)nc4C)(C2)C3)CCCCCCC1 26312,N1(C(C2COCC2C(F)(F)F)=O)CCN(C(c2ccc[nH]2)=O)C(CC2CC2)C1 26313,N1(C(c2n(C)ncc2I)=O)CC2(C1)SCCC2NC(C1CC12CCSCC2)=O 26314,c1(C(CNC(COCC=C)=O)NC(=O)CCCc2ccsc2)ccc(OC)cc1 26315,c1(C(N2CCC3CCN(C(=O)C(F)(F)CC4CC4)CC23)=O)cc2cc(F)ccc2[nH]1 26316,c1(C(=O)NC2C3(NC(c4nnn(C)c4N)=O)CCC(C2)C3)cccc2[nH]ncc12 26317,CCCCCC(O)CC(=O)N1CC2CC2(CNC(=O)CNS(=O)(=O)N(C)C)C1 26318,Cc1cnc(C(N2CCOC(CNC(=O)C=CC(C)C)C2)=O)nc1 26319,c1(CN=C(NCc2cc(C)on2)NC(c2ccn(C)c2)C)cn(C)c(=O)nc1O 26320,CCC(CC)(CCNC(=O)C=NOC)NC(C1CCC1n1cccn1)=O 26321,c1(NC(c2cc(I)ccc2-n2cnnn2)=O)ccc2nnn(O)c2c1 26322,c1(C(N2C(CNC(c3c(C)cco3)=O)CCC2)=O)[nH]c2cc(F)cc(F)c2c1C 26323,C(C1=CCN(C(=O)COCC(F)F)CC1)NC(C1C(C)(C(C)C)C1)=O 26324,C(=O)(CCC(C)N(C)C)N(CC(CNC(CSCCC(C)C)=O)(C)C)C 26325,C1(C(=O)NC2(C)CCN(C(=O)CNS(N)(=O)=O)CC2)CC2CC1CC2(F)F 26326,CCCCC(CC)CC(=O)NC1CN(C)CCN1C(=O)COC1(C)CCCC1 26327,N1(C(C2(CNC(CCn3cnc(=N)[nH]3)=O)CC23CCC3)=O)CCC(C2CCC2)C1 26328,C(=O)(CCC(=O)NCC)NCC1(NC(CC=CCC)=O)CCC1 26329,N1(C(C(CN(C)C)NC(=O)COCCCF)=O)CCCN(CCO)CC1 26330,C1(n2cc(C3CCN(C)C3)nn2)C=CCC(C(=O)NCCC2CC(O)C2)C1 26331,C(C(C)(CNC(c1cnc(CC)[nH]1)=O)OC)NC(C(C)OCC=C)=O 26332,CC(C)C(CCNC(c1ccc(N(C)C)cn1)=O)NC(=O)CCN1CCCCC1 26333,c1(C(N2C(CNC(=O)CCC3CCCCC3)C=CC2)=O)ccn2ccnc2n1 26334,N1(C(c2c(C)nc[nH]2)=O)CC(CNC(=O)Cc2cnc(C(F)(F)F)s2)C(C)C1 26335,N1(C(C(C(C)C)C(C)C)=O)CCC2CCN(C(C3CC(n4cnnc4)C3)=O)CC12 26336,CCCCC(C)C(=O)NCCCC(O)C(=O)NCCCC(=O)NO 26337,N1(C(C2CC(C#N)(O)C2)=O)CCC2CC(NC(=O)CS(N)(=O)=O)CCC2C1 26338,c1(C(=O)NC2CC(C)(NC(=O)COc3ccccc3Cl)C2)c(O)cccc1Cl 26339,n1(CC)ccc(C(=O)NCc2cc(C(=O)NCC(=O)OC(C)C)on2)n1 26340,CN=c1[nH]c(=NCN2CCC(CF)CC2)[nH]c(=NCc2ccnc(C(N)=O)c2)[nH]1 26341,C(CC(CC)C(=O)NC1CN(C(c2cnn(C)c2OC)=O)C(C)(COC)C1)=CC 26342,C1(NC(c2n(CC)ccc2)=O)CN(C(=O)C(C)C2CC2)CCC12CCOCC2 26343,C1(F)(C(=O)NCC(CN(C)C(C2CC23CCOC3)=O)(C)C)CCCCCC1 26344,CC1(C)CCN(C(=O)CN2C(=O)CCCC2=O)CC1C(N1CCC=C(Cl)C1)=O 26345,C12CC3CCC1CC3C(=O)N2.C(C(=O)OC(C)(C)C)N(C(C1CC1F)=O)CC 26346,c1(C(N(CCN(C(=O)CCc2ccnc(Br)c2)C)C)=O)ccccc1C#N 26347,C1(C)(C(=O)OCC)CN(C(c2cc(C#N)n(C)c2)C(=O)NCC2(C)CC2)CCO1 26348,c1(C(=O)NCC2(OC)CCN(C(=O)CCS(C)(=O)=O)CC2)ccc2c(c1)NCC2 26349,CCC(C)(C)CC(=O)N1CCCC(C(C)(O)CNC(c2cc(CO)oc2C)=O)C1 26350,C1(NC(C23CC(C)(C2)C3)=O)CCC2(CC1)CCN(C(C1CCOC1)=O)C2 26351,Cc1c(OC(F)(F)F)cccc1Br.C12CN(CCO1)C(=O)C2 26352,c1(OC)c(Cl)ccc(Cl)c1C(=O)NCC(C)NC(c1ccc(C(F)F)o1)=O 26353,C1(C(N2CCC(C)C2CNC(c2ccoc2Br)=O)=O)CCCNS1(=O)=O 26354,Cc1ccc(C)c(C(=O)NC2CC2CNC(=O)C(C)Sc2nncn2C)c1 26355,c1(CS(N2CC(NC(Cc3cn(CCOC)nn3)=O)C2)(=O)=O)ccc(Br)cc1 26356,N=c1[nH]cc(C(=O)NCC2CC(O)(CNC(C3(C(F)F)CCC3)=O)C2)o1 26357,Cc1oc(-n2cccc2)c(C#N)c1C(=O)NCC(O)CNC(C1(O)CCSC1)=O 26358,Cc1ccc(N)cc1C(=O)NCCC1CN(C(c2ccc(=O)n(C)c2)=O)CCO1 26359,C12CCCC(N=C3NC(=NCC4(CC4)C1)NC1=C3CSC1)C2.N(C)(C)CC.C1CC1 26360,c1(C(N(c2nc(OC)nc(OC)n2)C2CC3(CNC3)C2)=O)ccc2ccsc2c1 26361,N1(C(C(CCC)O)=O)CC2(CCN(C(C3CCCCO3)=O)CC2)CC1C 26362,Cc1cc(C(N2CCC(C)C2CNC(=O)Cn2ccnn2)=O)cc(F)c1 26363,C1(C(N(C2CCCC2)CCNC(c2ccc(CC)o2)=O)=O)CC(C)CC(C)(C)C1 26364,c1(CC(=O)NCC(C2CC2)NC(C(C)OCCC=C)=O)ccc([N+](=O)[O-])c(N)c1 26365,C=CC(C)CC(=O)N(C1CCN(C(c2cc(C)sn2)=O)C1)CC 26366,N1(C(=O)NC(CC)C(c2nnnn2C)SC(C)(C)C)CC2(C(=O)O)CC2(CO)C1 26367,CCCCC(O)C(=O)N1CC(NC(=O)CCc2ncccn2)C(n2ccnn2)C1 26368,N1(C(Cc2c(F)ccc(C)c2)=O)CC2CCC(C1)N2C(C1C(C)CC1C)=O 26369,Cc1ccc(F)cc1C(=O)NCC(CNC(C1CC2(CSC2)C1)=O)CO 26370,N1(C(c2n(C)nnc2)=O)CCC(C(=O)NCCNS(N)(=O)=O)C1(C)C 26371,C1(CNC(C=CCCC)=O)CC2CC(C1)N(C(=O)CCc1cccnc1)C2 26372,CC(C)(CCCNC(c1sc(OC(F)F)nc1Cl)=O)NC(C1CCC(=O)O1)=O 26373,c1(C(=O)NC2C3CN(C(CC(C=C)CCC)=O)CC32)c(O)nnc2c1CCC2 26374,N1(C(C2CC(NC(C(C)(C3(C)CC3)OC)=O)C2)=O)CC(C)CC(C)C1 26375,Nc1c(C(=O)NC2CC(NC(C3C4C5CCC(C5)C34)=O)C2)ccc(Cl)c1O 26376,c1(OC)cnc2ncnc(N3CCCCCC3CCO)c2c1 26377,C1(OC)CCC(C(=O)NCCN(C(=O)CCc2cccs2)C)C1 26378,C1(N(C)C(c2csnn2)=O)CCC(NC(=O)C(O)Cn2cncn2)CC1 26379,C(=O)(CC1COCc2ccccc21)N1CCC(CNC(CSC)=O)C1(C)C 26380,CCCCCCCC(=O)N1CCC(NC(=O)COc2cc(F)cc(F)c2)C12CC2 26381,c1(C(=O)NC2C(NC(c3c(C)onc3C3CC3)=O)COC2)cccc(S(C)=O)c1 26382,c1(C(=O)NCC(CC)(CC)NC(=O)Cn2cncn2)cc(F)cc(Br)c1 26383,N1(C(C2C(CC)CCC2)=O)CC2(NC(=O)CC3CC4C=CC3CC4)CCC1CC2 26384,N1(C(c2ncc(C)nc2)=O)CCC2(CC1)CN(C(=O)Cc1nccs1)CCO2 26385,C1(N(C(COCCNC(C(C2CCCC2)OCC)=O)=O)C)COCCO1 26386,c1(CNC(C(c2cc(-c3cnn(C)c3)[nH]n2)N(C)C)=O)nnn(C)n1 26387,CC#CCC(C(=O)NCC(C)(O)CCO)NC(=O)C(C1CC1)SC 26388,C1(c2n(CCC)nnn2)(Nc2cnn(CC(=O)OC)c2)CCN(C(C)C)C1 26389,C1(NC(CCN(CCC)C)=O)CCCN(C(=O)CCCSC)C1 26390,c1(C(C)C)ccc(C(N2CCC(N(C)C(C3C(C(F)F)C3(C)C)=O)C2)=O)c(O)c1 26391,c1(C(=O)NCCCCN(C(=O)CC2CCC2)C)cc(=NS(C)(=O)=O)cc[nH]1 26392,c1(CN2CCC(O)(NC(CNC(CC(C)C)=O)=O)C2)ccc2ncccc2c1 26393,C1(NC(CCC2(CCC#C)N=N2)=O)CCC12CN(C(=O)COC1CC=CC1)C2 26394,c1(CC(=O)NCC2CN(C(c3cc(Cl)no3)=O)CCO2)cc(F)c(F)cc1F 26395,C12(CNC(C(=Cc3ccc(F)cc3)C)=O)CN(C(=O)CC3CCC3)CC1CCO2 26396,C1(NC(c2c(C)noc2)=O)CCN(C(=O)C(C)(C)c2cnn(C)c2)CCC1CO 26397,S(=O)(=O)(c1ccccc1)NCC(=O)N(C(C)CCNC(C1CCC(C)CC1)=O)C 26398,C(=O)(C1CCCn2ccnc21)NC1CC2(C(NC(CC(C(C)C)(F)F)=O)C2)C1 26399,c1(OC)cc(C(=O)N(C)CC2CCCN2C(c2ccn(C3CC3)n2)=O)sc1Cl 26400,C(=O)(C(CC)CCc1ccccc1)NC1C(CC)CN(C(c2coc(Cl)n2)=O)C1 26401,c1(C(N2C(C3(NC(C=CC=CC)=O)CC3)CCCC2)=O)cccc2ncc(C)n12 26402,Cc1onc(C(F)(F)F)c1C(N1CCC(CNC(=O)CN2CCCC2=O)C1)=O 26403,c1(C(N(C)CCOCCNC(C2CC3(CC3)CO2)=O)=O)nc(N(C)C)nc(=N)[nH]1 26404,c1(OC)cc(F)c(C(=O)NCC2COCC2NC(C2CC(F)(F)C2)=O)c(F)c1 26405,c1(CN(C(CCC#C)=O)C)cccnc1N1CCN(c2ncc(Cl)cn2)CC1 26406,CC(C)C(F)(CNC(=O)C(F)C(F)(F)F)C(=O)N1CCC2(CCC2)C1 26407,c1(CC)nc(C(=O)NC2CCC(NC(=O)COCc3cc(C)on3)C2)co1 26408,C#Cc1ccc(CC(N2CCN(C(c3ccc[nH]3)=O)C(CO)C2)=O)cc1 26409,N1(CCCNC(N2C(CC(c3onc(C)n3)(C)C)CCC2)=O)CCCC(C)C1 26410,C1(NC(CSC)=O)C2CC1N(C(=O)CCC(=O)N(C)C(C)C)C2C 26411,Cc1csc2ncc(C(=O)NC(C)(CNC(C3(Cl)CC3(C)C)=O)C3CC3)c(=O)n12 26412,c1(NC2CC(NCc3ccc(SC)s3)C2)ncnc2[nH]cc(C)c12 26413,N1(C(CN(C2CC2)CC)=O)CCCC1C(C)NC(=O)C=Cc1ccsc1 26414,C1(C(=O)OC)CC(C)N1C(C1(NC(c2cnc(C(C)C)o2)=O)CC1)=O 26415,c1(C(=O)NC2CCN(C(C(CC=C)C)=O)CC2F)ccc2c(c1)C(=O)NCC2 26416,c1(CC)cc(C(N2CCOCC2CCNC(=O)CC2C=CCCC2)=O)cc(O)n1 26417,c1(SC)ccccc1CC(=O)NCC(O)CNC(=O)C(C)O 26418,C1(NC(C(C)(C)SC)=O)CN(C(c2cncc(C(C)(F)F)c2)=O)CC1C(F)F 26419,C1(CC)CCN(C(C2CCC2C(N)=O)=O)C1C(=O)NCCCC1(C)CC1 26420,c1(C(C(=O)NCC(CNC(C2C(CC)CCC2)=O)C)C)ccc2ccccc2c1 26421,C(C(O)CC(=O)Nc1c(C)coc1C(=O)NC)NC(COC(CC)C)=O 26422,C1(C(N2C(CNC(C(CC)N(C)C)=O)CCCC2)=O)OC2CCC1CC2 26423,C1(OCCNC(c2coc(O)n2)=O)CCN(C(C2(C(F)(F)F)CCC2)=O)CC1 26424,c1(C(=O)NCCC2CCC(NC(c3cc(OC)n(C)n3)=O)C2)cn2ccsc2n1 26425,C(=O)(C(C)(C)CC(=O)NCc1nc(CNC(=O)CCc2csnn2)cs1)OCC 26426,C(=O)(C(CCS(C)=O)N(C)C)NC1CCN(C(CCCOC)=O)C1(C)C 26427,C12(C(=O)NC(C)CNC(C3COC(=O)N3C)=O)CC3CC(C)(C1)CC(C)(C3)C2 26428,C1(NC(C(CC=C)C)=O)CCN(c2ncc(Br)cn2)CC1C 26429,c1(OCCC)ccc(C(=O)NC2(CNC(C3SCCCS3)=O)CC2)cc1N 26430,c1(CC(N2CCN(C(c3scc(C#N)c3)=O)C3C2C3)=O)c[nH]c2cnccc12 26431,c1(C(c2n(C)nnn2)NCc2cnoc2C(C)(C)C)nn(C)cc1I 26432,c1(OC)c(C)cc(NC(C2(O)CCN(C(=O)C(O)C(C)(C)C)C2)=O)cc1C 26433,Cc1ccc(C2CC2)c(NC(=O)NCc2c(C)noc2-c2ccc(C)cc2)c1 26434,C1(C(=O)NCC(C)(O)CNC(=O)C=Cc2ccsc2)CCOCC12CCC2 26435,C(CCS(=O)(=O)OCC(=O)NCCOCCOCCNC1CCC1)OC.OC 26436,c1(CC)ccccc1NC(=O)C(Cc1ccoc1)NC(=O)OC(C)(C)C 26437,C1(OC)CCCC1CNC(c1cn(CCNC(C2CNC(=O)N2)=O)nn1)=O 26438,c1(OC)c(C(=O)NC2CCC2NC(C23CC(F)(C2)C3)=O)cc([N+](=O)[O-])cc1Cl 26439,C(CCCCCC(=O)N(CC(=O)N(C)C)C)NC(C(C=C)CC)=O 26440,C1(COC)CCCCN(C(=O)C(N2CCSCC2C)=O)C1 26441,CC1CC(NC(=O)C=Cc2ccc(Br)s2)CN(C(=O)C(C)NC(N)=O)C1 26442,c1(NC(c2ccc(Br)c(Cl)c2)c2n(CCSC)nnn2)ccc(Br)c(C)c1 26443,C1(C(=O)NC(c2ccncc2)C)CN(C(=O)CN2CCC(F)CC2)C2(CCC2)C1 26444,c1(NC(C)=O)ncc(S(=O)(=O)N2CCCC2c2cc(F)cc(Br)c2)s1 26445,CCC(F)(F)C(=O)NCC(O)CCNC(c1nc(Cl)sc1C)=O 26446,N(C(=NCC1CCOC1)NC(c1ccccc1F)=O)CC1(C2CCCO2)CCCC1 26447,C=CCCCC(C(=O)NCc1cn(C2CC2)cn1)NC(=O)CC1(COC)CC1 26448,CCCC(C(O)C(=O)NC1(C)CC(F)C1)NC(C1(CCC)CC1)=O 26449,c1(C(N(CC(C)CNC(=O)CC(C)P(C)(C)=O)C)=O)ccc(F)c2ncccc12 26450,C(=O)(CS(=O)(=O)CC(=O)N(C)CC1CCCN1C(=O)C(C)CC(C)C)OC 26451,c1(OC)cccc(CC(O)C(=O)N(C)CC2CN(C(C3CCC(=O)N3)=O)C2)c1 26452,c1(CC)cc(C(N2CCCC2c2ccc(F)cc2)C(=O)NC(C)(C)C)ccc1Br 26453,N1(C(c2cnn(C)c2C(C)(F)F)=O)CCC(NC(C2CC2CF)=O)CC(O)C1 26454,C1(C)(CN(C)C(C2OCCC2C(F)(F)F)=O)CN(c2nnnn2C)CCO1 26455,C1(CNC(C#CC(C)C)=O)C(C2CC2)CCN1C(=O)C=Cc1ccc(Cl)s1 26456,N1(C(C2CC(OC)C2)=O)CC(NC(C2(C(C)C)CCCO2)=O)CC1(C)C 26457,N1(C(CC(=O)OC)=O)CCC2C1CCCN2C(c1ccc([N+](=O)[O-])c(C)c1)=O 26458,C1(NC(c2ncc(SCC)nc2)=O)CCSC12CN(C(C1CC1CC(=O)OC)=O)C2 26459,CCCCCC(O)C(=O)NCC1CN(C(=O)C(=O)NCCOCCOC)CCO1 26460,N1(C(c2c(C)cno2)=O)CC2CC(NC(=O)CCOC3CCOC3)C1C2 26461,c1(C(=O)NCC2(Cn3cc(C=CC)nn3)CC2)cc(F)ccc1Cl 26462,C1(C)(C(=O)NCC(C(=O)OCC)C)CCN(C(=O)CC=CCOC)C1 26463,C12(NC(c3ccc(CC)o3)=O)CN(C(c3cc4c(s3)CCC4)=O)C(COC)(C1)C2 26464,C(C#N)(C(=O)C(C)(C)CO)C1CCN(C(=O)Nc2c(C)ncc(F)c2)CC1 26465,N1(C(C(CC)F)=O)CCc2nc(NC(=O)COCCS)sc2C1.c1nc[nH]n1 26466,c1(C(=O)NCC2(C(=O)OCC)CC(F)(F)C2)cccc(Cl)c1F 26467,CC(C)C(F)(F)CC(=O)NC1CC(CNC(c2ccc(O)nc2)=O)C12CCC2 26468,c1(CNC(C(CC)C)=O)ccc2c(c1)CCN(C(C1(C)CCN(C(C)=O)C1)=O)C2 26469,N1(C(CC(C)CF)=O)CC2COCCC2(NC(c2cccc([N+](=O)[O-])c2N)=O)C1 26470,C1(C(=O)NC(CNC(C(CC)C2CCC(=O)N2)=O)C)CCC(OC)CC1 26471,c1(-c2occc2)cncc(N2CCN(Cc3csc(-c4cn[nH]c4)n3)CC2)c1 26472,c1(N2CCN(C(=O)OC)CC2)nc(=NC2CCCSCC2)[nH]c2c1COC2 26473,N1(C(C2(C)COC2)=O)CCC2(NC(c3ccc(-c4cccs4)[nH]3)=O)CC2C1 26474,c1(CN(Cc2c(C)cncc2)Cc2ncccc2C(=O)O)cc(F)cc(Cl)c1 26475,C1(C(N(C2CN(C(c3cnc(C(F)F)nc3)=O)CC2F)C)=O)CCC(C)(C)CC1 26476,n1(CC(=O)NCCCOCCOCCNC(=O)C(Cl)=CCl)cc2ccccc2n1 26477,c1(C(N2CCC(NC(C3(CC)CCNC3=O)=O)C2C)=O)cnc2sccc2c1 26478,C#CC1CC2CCC1N(C(=O)CC1(OC)CN(C(c3cnn(C)c3CC)=O)C1)C2 26479,CC1(C)OC2(C(N3CC(OCCNC(=O)CCn4cccn4)C3)=O)CCC1CC2 26480,C1(C(=O)NCC2CC(C(=O)OC)C2)C(C)CCN1C(=O)CC1C(=O)NN=C1C 26481,C1(C)(CNC(C(CC)SC)=O)COCCN(C(c2ccn(CCOC)n2)=O)C1 26482,C1(c2nc(C3(CO)CC3)on2)(CC2CCCO2)CCCCCC1 26483,C1(C(=O)NCC2CC(O)CN2C(c2cn(C)c(O)n2)=O)(COC)CCOCC1 26484,N1(C(c2cnc(OCC)nc2)C(=O)NC(C)C)CC(N(C)C)C2(CC2)C1 26485,C12(CSCC)CC(C(N3CCC(C)(CNC(=O)CC=C(C)C)C3)=O)(CO1)C2 26486,c1(C(N2C(C)CC(NC(c3cnn(C)c3C3CC3)=O)C2)=O)cc(Cl)ncc1O 26487,C12C(C)CCCN1C(=O)CC1CN(C1)C1CC21.N1(C(C)=O)CC(F)C1 26488,C1(NC(CN(CCC)C)=O)(CNC(C2(CC#N)CCOC2)=O)CCCC1 26489,CC1CC(C(=O)NCC2(NC(=O)CS(N)(=O)=O)CCCCC2)CCS1(=O)=O 26490,C(=O)(CCCC(F)F)NCC(CCCC)NC(=O)CN1CCCC1C 26491,C1(F)(CNC(c2cnsc2)=O)CC(NC(C2CC2F)=O)C1 26492,C1(C(=O)NCCC(CNC(=O)C(C)O)OC)CCCOCC1 26493,C=C(C)CCCC(=O)NCC=CCNC(=O)C(C)c1cncs1 26494,c1(C(=O)OC)ccncc1C(=O)NC1CCCCC1NC(C1CC12CCC2)=O 26495,CC1CCN(CC(=O)N(CCCN(C)C)CCNC(C2CCSCC2)=O)C1 26496,C(CCCCCF)NC(c1nccs1)=O.C(CC(=O)CCO)n1cc(C2CC2)nn1 26497,c1(OC(C)C)cc(NC(C2C=CC(Nc3csc(Cl)n3)C2)=O)ncn1 26498,c1(C(N2CCC(C(C)NC(=O)C(c3ccccc3)O)C2)=O)cncc(N=[N+]=[N-])c1 26499,CCC(C)(CC)C(=O)OCCCC1=NOC(C(N2CCC(C)CC2)=O)C1 26500,N1(CC)CCCCC1C(=O)NCC1CCCCN1C(C1(O)CCCCC1)=O 26501,CC(O)CCCCCC(=O)N1CCN(C(=O)C(F)C(F)(F)F)C2(CCC2)C1 26502,c1(C(C)(C)C(=O)NCC2(O)CC(NC(C3CCCO3)=O)C2)cccc(Cl)c1F 26503,c1(C(=O)NCCC2N(C(C3=CCCC3C)=O)CCSC2)n[nH]c2ccc(F)cc12 26504,N1(Cc2cccc(OC)c2)CCC(O)(C(=O)NC2CCOCC2F)CC1 26505,C1(C(=O)NC)CN(C(=O)CN(C)C(=O)C2CC2)CC1(C)C 26506,C1(CNC(Cn2c(C)ccn2)=O)CN(C(=O)CC2C=CCC2)CC1(C)C 26507,c1(SC(CC(=O)NC23CC(COC)(C2)C3)C)ccc(N)cc1.C12(CC1)C(=O)NC2 26508,c1(C(=O)NC(C2(O)CCN(C(=O)CCc3ccccc3O)C2)C)cnccc1Cl 26509,C(=O)(C1SCc2cccnc21)NC1(CN(C(C2CCN(CC(C)C)C2)=O)C)CC1 26510,c1(C(N2CCCN(c3ccccn3)CC2)=O)ccc2c(c1)CCC2 26511,c1(OC(C)C)cccc(F)c1C(=O)NC(C)C(O)Cc1ccccc1 26512,c1(OCC(=O)Nc2nc(C(C)C)nc(C(C)(C)C)c2)c(Cl)cc(Cl)cc1Cl 26513,CCC(CC)(C(=O)NC1CC(N(C)C(C2CC(C)(C)CO2)=O)C1)C(C)C 26514,C1(NC(C(=O)NCCOC)=O)CCC(CCNC(=O)CC2CCOC2)C1 26515,c1(OC)cc(CNCC(C(=O)O)OC)cc(I)c1OC 26516,C1(NC(CCC)=O)CCS(=O)(=O)C12CN(C(=O)C(F)(F)C(C)(C)O)C2 26517,c1(OC)cc(C=CC(=O)Nc2ccn(C)c(=O)c2C)ccc1OCC(N)=O 26518,c1(CC)cc(C(N2CC(CC(F)C(=O)NCCCc3cc(C)[nH]n3)C2)=O)ccn1 26519,C1(NC(C2CC(C)(CC)C2)=O)CCCC2CN(C(=O)C=Cc3ccccc3)CC12 26520,c1(CCC(=O)NC2(CNC(C3CC(Cl)(Cl)C3)=O)CC2)cnc2ncccn12 26521,c1(NC(C2N(C(C3(C)CC3)=O)C3C(C2)C3)=O)c(F)cc(C#N)cc1F 26522,c1(C(N(CC(C)NC(C2CCCSC2)=O)CC)=O)cc(SC)ccc1Cl 26523,C1(C(=O)NC(CSC)C)(NC(=O)CCN(C)CCO)CCCCC1 26524,CCCCC(CNC(=O)Cc1ccn(-c2ccc(F)cc2)n1)NC(=O)CC(C)O 26525,Cc1cccc(OCCCC(=O)N2CCC(CNC(c3c(C)nsc3N)=O)C2)c1 26526,N1(C(CC(=C)C)=O)CCC(NC(c2ccnc(CC)c2)=O)C(CC)C1 26527,c1(N2CCC3(C)C(C)(C2)C3(F)F)nc(=NCc2cscc2Cl)[nH]c2cccnc12 26528,c1(N(C)C)ncccc1C(=O)NC1CC(NC(c2ccn(C3CC3)n2)=O)C1 26529,c1(C(=O)NC(CN(C(=O)Cc2ccon2)C)(C)C)ncc(Cc2ccccc2)s1 26530,C(=O)(C(C(=O)N1CCC(CN(C)C(c2cncn2C(C)C)=O)C1)OC)OC 26531,C1(CC=C)(NC(c2snnc2CCC)=O)CCCN(C(c2ccnc(F)c2)=O)C1 26532,c1(C(=O)Nc2c(C)cc(NC(C3CCC(=O)N3)=O)cc2)c(Br)ccc2c1CCC2 26533,C1(NC(C(c2ccccn2)C)=O)CN(C(c2cccc(Cl)c2)=O)C2CCCCC12 26534,C(CCNC(=O)CCC=CC(C)C)(C(C)C)NC(CCSCC)=O 26535,c1(C(c2n(CCCC)nnn2)NC2CCC3(CC3)C2)sc(Br)c(C)c1C 26536,Cn1nc(C(=O)NCCC2(CNC(=O)CCc3ccc(=N)[nH]c3)CC2)ccc1=O 26537,C(CN=c1cc(C)nc(N2CCOC3(CCSC3)C2)[nH]1)(c1ccccc1)OC 26538,C1(C(=O)NC23C(CN(C(CC4(C)CCC4)=O)C2)C3)CC2CCCC(C1)C2 26539,c1(C(=O)NCC(CNC(c2ncc(C)c(C)c2)=O)O)ccn2ccccc12 26540,C1(C(=O)NCc2ccc(C(C)NC(C(C)OCC=C)=O)cc2)CC2C(C1)C2(C)C 26541,S(=O)(=O)(c1ccc(NCCCCCCSC)c(C#N)c1)NC(CC=C)C 26542,c1(OC)nccc(C(=O)NC2CCCN(C(=O)C(C)CC(F)F)CC2)c1F 26543,C(=O)(CCCC(=O)OC)N(C1CCN(C(C(C(C)C)OCC)=O)CC1)CCO 26544,c1(CC)nc(N2CC3CC(NC(=O)CC(C)CC(C)C)CC2C3)c(C)c(Cl)n1 26545,C#CC1CCCN(C(C2(CNC(=O)C=Cc3ccoc3)CCC2)=O)C1 26546,c1(OC)cc(F)ccc1C(N1CC(C)(C)CC1CNC(=O)CCCC1CC1C)=O 26547,c1(C(N2CCC(NC(CN3C(C)CC3)=O)CC2C)=O)cccc2[nH]ccc12 26548,Cc1ccnc2nc(C(=O)NC3CN(C(C4CC4(C)Br)=O)CC4(CC4)C3)nn12 26549,Cc1ccc(C(=O)NC(C)CCCNC(c2coc(CO)c2)=O)cc1S(N)(=O)=O 26550,C(=O)(CC(C)C(C)(C)C)N1C(CCC)CN(C(=O)CCCc2cnccn2)CC1 26551,N1(C(CC(CC)C)=O)CCC(CNC(=O)C=Cc2ccc(Cl)s2)C12CC2 26552,N1(C(C(COC)OC)=O)CC(C(=O)N(CCCC(C)(F)F)C)CCC1C 26553,C(=O)(C#CC1(C)COC1)NC1CC(F)(CNC(Cc2cc(CC)nn2C)=O)C1 26554,c1(C(N(C2CC(CNC(=O)CSc3nncs3)C2)C)=O)cccc(=O)n1C 26555,c1(C(N2CC(C(C)NC(C(COC)(C)O)=O)OCC2)=O)cncc2[nH]ccc12 26556,CC(C)CC(C)CC(=O)N(C1CCC(NC(=O)COCc2nccn2C)CC1)C 26557,C(=O)(C1=CCCOCC1)NC(CC)(CC)CCNC(=O)Cc1c(C)nn(C)c1C 26558,CCC(C)C(C(=O)N1CCC(n2cc(Cn3cncn3)nn2)C(O)C1)N(C)C 26559,N1(C(c2c(C)nn(C)c2Br)=O)CCN(C(C2CCC(O)C2)=O)CC(O)C1 26560,C1(N(C)C)CCCN(C(C2C=CCN(C(=O)C=Cc3ccnn3C)C2)=O)C1 26561,C1(C(=O)NCC2CCC(C)CN2C(C23CC(F)(C2)C3)=O)CC2(COC(=O)N2)C1 26562,N1(CC(=O)NCc2scc(CC)n2)CCN(C(c2cnc(Br)s2)=O)CC1 26563,c1(C(N2C(CC(=O)NC3CC=C(C)CC3)CCC2)=O)ncn2ccccc12 26564,CP(C)(=O)CC(=O)N1CC2(NC(C3CN(C(C4CCCCC4)=O)C3)=O)CC1C2 26565,C1(C(N(CC#C)Cc2cccnc2)=O)CCCC(C(F)(F)F)C1 26566,c1(Cc2c(-c3ccc(OCC)c(CO)c3)nccc2)cc(OC)c(C)cc1C 26567,C1(CNC(C(C(C)C)C)=O)CCN(C(=O)CCC2(C)CC2)CC1(F)F 26568,CCC(C(=O)NC(C)(CNC(c1cc(C2CC(F)(F)C2)[nH]n1)=O)CO)C(C)C 26569,N1(C(C(=O)NCCC)CC2CC(F)(F)C2)CCC(C2CCCCC2)CC1 26570,c1(CC(=O)NC2(C)CC(NC(C(CC)(C)O)=O)C2)cccc(F)c1Cl 26571,C1(NC(=O)COC(=O)CO)CCN(CCNC(c2cocn2)=O)CC1 26572,c1(CCN2CCC(CNC(C(COCC)C)=O)C2)cccc(S(C)(=O)=O)c1 26573,CC1CC(C)N(C(c2ccns2)=O)CCN1C(c1ccc(CC2CC2)cc1)=O 26574,N1(C(c2cn(C)cn2)C(=O)NCCC2(C)CC2)CCC(CO)C1c1ccccc1 26575,CC1CC(NC(C2CCC2)=O)CCN1C(c1cnn(C2CC2(F)F)c1)=O 26576,c1(C(=O)NCC2(NC(=O)CC(F)(F)F)CCC2)cc2c(nn1)CCC2 26577,n1(CC)cnc2[nH]c(=NC3CC3CC)nc(N3CCCC(OC)C3)c12 26578,C1(CNC(C(C)(C)O)=O)CC(C)(C)CCC1NC(=O)COc1ccsn1 26579,c1(C(=O)NC(CC)CNC(=O)C=CC2CC2)cccc(NC(N)=O)c1 26580,C1(CNC(=O)CCN2CCCCC2)CC(NC(C2(C3CC3)CCC2)=O)C(O)C1 26581,c1(OC)ncc(Cl)c(C(N2CC(N(C)C(c3ccccn3)=O)C(O)C2)=O)c1Cl 26582,c1(C(=O)NCc2ccc(OCCCN(C)C)cc2)ccc2c(c1)C(CN)CCC2 26583,C1(CNC(c2ncccc2Cl)=O)CN(C(=O)C2=CC(O)CCC2)CC12CCC2 26584,C#CC1(CNC(C2(NC(c3ncc(F)cc3F)=O)CCSC2)=O)CCOCC1 26585,c1(OC)ccc(F)cc1CCC(N1CCCC1CNC(c1cc(O)nn1C)=O)=O 26586,C1(C(=O)NCC(C)(C)C#N)CCCC(NC(=O)CC(C)(C)C)CC1 26587,c1(SCC(=O)NC(CC(C)NC(CCOC)=O)C)nc(C)nc2sc(C)c(C)c12 26588,c1(C(N)=O)cccc(C(N2CC3(CO)CCC2C3)=O)c1N.C1(=O)CCOCCN1 26589,C1(C(=O)NC(CCOC)CO)C=CCCN1C(=O)Cc1cc(C)cs1 26590,C=CCC(CNC(C1(C2CC2)CC1)=O)NC(c1c[nH]nc1-c1ccc(Cl)s1)=O 26591,N1(CC(C)C)CCC(C(=O)NCC(C(C)(C)C)NC(=O)C=CC2CCCO2)CC1 26592,C1(C(=O)NCC2CC2CNC(C2(O)CCOCC2)=O)C2CCCCCC12 26593,CCCC(C#N)C(=O)NCC1(O)CCCN(C(c2c(C)cnn2C)=O)C1 26594,C(=O)(CCC(C)(C)C(=O)N(CCNC(C1CCCCC1F)=O)C1CC1)OC 26595,N1(C(C2CC(=C)C2)=O)CCN(C2CCC(NC(=O)Cc3ncccc3C)C2)CC1 26596,c1(NC(C(C(C)NC(=O)C(F)C(C)(F)F)(C)C)=O)cc2ccccn2n1 26597,N1(C(c2c(C)nc(NC(c3c(C)nc(C)o3)=O)s2)=O)CCc2ccc(Br)cc2C1 26598,c1(C(=O)NC2CN(C(C3C(CC)CCCC3)=O)C2)cc2c(C)ccc(F)c2[nH]1 26599,C(c1ccccc1OC)=CC(=O)NCC1CCC(NC(C(CC=C)C)=O)C1 26600,N1(C(C(CSC)O)=O)CC(C(=O)NCC2(C(C)C)CC2)CC1(C)C 26601,N#Cc1c(Cl)cc(-c2cn(CCNC(C3(O)CCC3)=O)nn2)cc1Cl 26602,CC1(CNC(C2C3COCC23)=O)CCN(C(C2(C(N)=O)CCC2)=O)C1 26603,N1(CC(c2cccc(C)c2)=O)CCC(C)C(NC(c2cc(C3CC3)nn2C)=O)C1 26604,C1(NC(COCC=C)=O)CCCC(NC(c2cccc(CCN(C)C)c2)=O)C1 26605,CCC(C)(C#N)C(=O)NCCOCCNC(c1ccccc1-c1nncn1C)=O 26606,c1(OC)ncc(C(N2CC(NS(=O)(=O)C(F)(F)F)CC(F)C2)=O)cc1Br 26607,c1(N(C(N2CC(=C(C)C)C2)=O)CC2CC2)cccc([N+](=O)[O-])c1 26608,N=c1nc[nH]n1CC(N1CC(CC(F)C(=O)NCC2CCCCC2)C1)=O 26609,N1(C(C(CCC2CCC2)NC(C(C)OCCC(C)C)=O)=O)CC(C)N(C)C(C)C1 26610,N1(C(c2c(C)nn(C(C)C)c2)=O)CCN(C(=O)CN2CSCCSC2)CCC1C 26611,N1(CCC)CC(C(=O)NC(C2CCN(C(c3sccc3SC)=O)CC2)C)CC1=O 26612,N1(C(c2c(NCCCC)cccc2)=O)CC2CCC1C(CNC(C1CC1F)=O)C2 26613,c1(C(=O)NCC2N(C(C(CCOC)(C)C)=O)CCC2)cccc2ccc(O)nc12 26614,C1(OC)(CNC(=O)C(C2CCOCC2)C)CCN(C(=O)CCc2ccco2)CC1 26615,S(=O)(=O)(CC(=O)NCC1(F)CC(NC(c2cccn2CC)=O)C1)NCC 26616,CCC(CCCC(=O)N1CC2(C1)CC2(F)F)NC(C1(O)CCSC1)=O 26617,c1(C(=O)Nc2n(C)ncc2)csc(=NCc2c(Br)cnn2C)[nH]1 26618,c1(NC(C(C2CCC(C)CC2)N(C(CC)C(=O)OC)CC)=O)cn(C)nc1Cl 26619,C1(CN(C(C=C(C)C)=O)C)CCCCN1C(=O)CCc1cn(C)nn1 26620,C(=O)(C#CC(C)(C)C)NC1(CC(=O)NCc2nnn(CC)n2)CCCCC1 26621,CCS(=O)c1ccccc1C(N1CCN(C(=O)CP(C)(C)=O)C(C2CCC2)C1)=O 26622,C1(c2cn(C(C)C)nn2)C(C)CCN1C(c1ccc(CSC(F)(F)F)o1)=O 26623,C(c1ccccc1)=CC(=O)O.N=c1nc[nH]n1CC(=O)N=CCN1CCC(N2CCC2)C1 26624,c1(OC)ccc(S(=O)(=O)N2CCOCC2C2CCCCC2=O)cc1-c1cc[nH]n1 26625,CCCCCC(F)C(=O)N(CC(N1CCc2nc[nH]c2C1)=O)CCOC 26626,C1(NC(=O)C=CC2CCCC2)CCCN(C(C2(F)C3CCCC23)=O)CC1 26627,c1(NCCCSC(C)(C)C)ccc(C(F)(F)Cl)cc1 26628,N1(C(CCCOC(C)(C)C)=O)CC2(C=C(C(=O)N3CC(F)CC3CO)CO2)C1 26629,C1(CN(C(=O)CC2CC(F)C2)C2CC2)CCN(C(=O)CC2(O)CCC2)CC1 26630,C1(O)(CCNC(C=CCNC(C2C(C)(C)C2)=O)=O)CCOC1 26631,c1(OCC)ccc(N)c(C(=O)NCC2CCN2C(=O)CCCn2cc(C)cn2)c1 26632,C1(C)(n2cc(C(N3CC(F)(SC(c4ccncc4F)C)C3)=O)nn2)CC(C#N)C1 26633,N1(c2nnc(CC)o2)CC(C)CN(C(c2ccc([N+](=O)[O-])s2)=O)CC1C 26634,c1(C(N2CCCC(N(C(c3cc(COC)cs3)=O)CC)C2)=O)cc(C)c(C)cn1 26635,c1(C(N(CC(C)NC(C2(SC)CCCCC2)=O)CC)=O)cc2cc(C)ccc2[nH]1 26636,C(=O)(CC1=CCOCC1)NCCC(C)NC(C(C)(c1ccccc1)OC)=O 26637,C(=O)(C(C)S(=O)(=O)C(C)C)N1CCC(OC)(CNC(C2(CC(C)C)CC2)=O)CC1 26638,c1(C(=O)Nc2nc(C(F)(F)F)c3ncnc-3[nH]2)cc(F)cc2nccnc12 26639,C1(CNC(CCC)=O)CCC12CCN(C(=O)COc1ccc(Cl)cc1C)CC2 26640,C1(=O)C(c2ccccc2)CN1.S(C)(=O)(=O)N(CCN(CC)CC)C(C)C 26641,c1(NC(C2CC2C(=O)Nc2cc(Br)cnc2Br)=O)c(Cl)cnnc1Cl 26642,c1(C(=O)NCC2N(Cc3c(C#C)cccc3)CCCC2)cc(Br)c(F)cc1C 26643,N1(C(CCC(C)C)=O)CCN(C(c2cc3n(n2)CCNC3=O)=O)C2COCC12 26644,c1(C(N2CCC(CNC(c3c(CC)scc3)=O)C2)=O)n[nH]c2c1COC2 26645,N1(C(C(C=CC)O)=O)CCC2CCCC12C(=O)NC1CCC2CCC12 26646,N1(C(C(CC)C)=O)CCC2CN(C(=O)C3=C(C)OCC3)CC2CC1 26647,C(=O)(C1=CC2(CCOC2)C1)N1CCC(C(C(=O)NCC2(CCC)CCC2)C)CC1 26648,C(=O)(C(F)(F)C(C)(C)O)N(C(C)CCC=Cc1ccccc1)C 26649,C1(F)(CNC(C(=O)N(C)C)=O)COCCN(C(C2COCC2(C)C)=O)C1 26650,C#CCC(C)(CC)C(=O)NCCN(C(c1cnc(C2CCC2)o1)=O)C(C)C 26651,C#Cc1ccc(C(=O)NC(Cn2cncn2)C(=O)NCC2C=CCC2)cc1 26652,Cc1c(O)ccc(C(N2CC(F)CC2CNC(C2(C)CCN(C)C2=O)=O)=O)c1C 26653,c1(C(=O)NCC23N(C(C4C(C)(C)CCC4)=O)C(CC2)CC3)ccsc1S(C)(=O)=O 26654,c1(C(=O)NCC(CC=C)NC(=O)CN2CC=CC2)ccn(C)c1CC 26655,c1(NC(C2CN(Cc3cccc(F)c3)CCC2O)=O)cccc2nc(O)ccc12 26656,CC1(C)CCN(C(c2cncnc2)=O)CC1NC(c1cc(-c2ccns2)on1)=O 26657,c1(C(N2CCC(N(C(=O)CCCCC#N)C)CC2)=O)cc2ccncc2cc1F 26658,c1(-c2cc(Cc3ccccc3)[nH]n2)nc(CC2CCCC2)nn1-c1ccccc1 26659,c1(C(=O)NC2C(CNC(C(n3ncc(C)c3)C)=O)C2)cncnc1C(C)C 26660,C1(CCN(C(CN2CC(CC)C2)=O)C)CCCCN1C(=O)CCNC(=O)NC 26661,N1(C(c2c(C)con2)C(=O)NC(c2ccccc2)C)CC(C)(C)C1C(C)C 26662,C1(C(=O)NC(c2ccsc2)C)CN(C(=O)C(=O)NC2CC2)CCC1(C)C 26663,c1(OC)cc(C(=O)N(C)CCNC(=O)CC2(O)CCCC2)cc(Br)c1OC 26664,C12(C(=O)NC3C(NC(CC=CC=C)=O)CCCC3)CCC(CC)(C1)OC2 26665,C(C(=O)Nn1cnnc1)(C(C)CC)NC(c1cc(=NC)[nH]cc1)=O 26666,C(=O)(CCC(C(C)C)NC(c1ocnc1C(C)C)=O)NCC(C1CC1)OC 26667,C1(NC(C)=O)CCN(C(C2CCOC2CN(C(C)=O)CCO)=O)C1 26668,N1(C(c2n(CC)ncc2)=O)C2CCC1C(NC(=O)Cc1nn(C)cc1Br)C2 26669,N1(C(c2c(C)n(C)nc2)=O)CCC2(CCCN2C(=O)CCCc2cccs2)C1 26670,CC(C)CC(C(=O)NC(CNC(C1(n2ccnn2)CC1)=O)C(C)C)N(C)C 26671,C1(C)(CC)CC(C(=O)N(CCNC(c2coc(C3CC3)n2)=O)C2CC2)CCO1 26672,c1(C(=O)NC(CC)CN(C(=O)C(C(C)C)SCC)C)ccc2nc(C)oc2c1 26673,S(=O)(=O)(c1ccc(Br)cc1N(C)Cc1cccc(Cl)c1)NCC1OCC(C)C1 26674,N1(C(CCC(=O)NCC)=O)CC(NC(C2CC=CC2)=O)CC(F)C1 26675,c1(C(=O)NC(C)CCNC(C2(CO)CC2)=O)cn(C)cc1C(F)(F)F 26676,C12(C(=O)NCC3N(C(c4c(C)n[nH]c4C)=O)CCC3)CCC(CC1)C(C)O2 26677,N1(C(C2N(C(Cn3ccc(C)n3)=O)CSC2)=O)CC(C(N)=O)C2(CC2)C1 26678,c1(C(=O)NCC(CC)NC(=O)C(O)CC2CC2)cc(F)n(C)n1 26679,N1(C(CCC=C)=O)CC2CC(C(=O)NCc3cccnc3OC)C(C2)C1 26680,C(C1=CCN(C(=O)C2=CCCOC2)CC1)NC(C(c1ccc(CC)cc1)C)=O 26681,N1(C(C2(F)CN(C(C(C(C)C)SC)=O)C2)=O)CC2CN(C)CC2C1 26682,c1(C(N(CC(O)CNC(=O)CN2CCNC(=O)C2)C)=O)cc2nc[nH]c2cc1F 26683,N1(C(C(CC)F)=O)C2CCC1CC(N(C(=O)COc1ccccc1O)C)C2 26684,C(CC(C)CC)(C(=O)N(CC(C)(C)CN(C)C)C)NC(c1c(C)nc(CC)o1)=O 26685,c1(C(=O)OCC)cnn(CCNCCC2OCCC2C)c1 26686,CCC(CC(C)C)C(=O)N1CC(C(=O)NCc2ccccn2)C2(CC2)C1 26687,Cc1ccc(Br)c(C(=O)NC23CC2CN(C(=O)COCC(C)(C)C)C3)c1 26688,C1(CNC(c2c(C)nco2)=O)CN(C(C2CC2c2sccc2C)=O)CC12CCC2 26689,c1(NC(C(=O)NCCCCSC)=O)ccc(Br)cc1-n1cncn1 26690,C1(C2(O)CN(C(=O)CC3CNC(=O)O3)C2)(CNC(=O)CCc2cnco2)CC1 26691,CN1CCCC(C)(C(N2CC(NC(C3CCCN3N=O)=O)C(C)(C)C2)=O)C1 26692,C1(OC)CC(C(=O)OC)N(C(=O)NC(C)C(C)SC)C1.C(C)(C)O 26693,c1(CC)[nH]c(C(=O)NCC(C)(CO)NC(c2cc(C)nn2C)=O)nc1Cl 26694,c1(C(C)C)cccc(-c2cn(C3CCC(C(=O)NCCCO)CC3)nn2)c1 26695,C1(CNC(C(=O)NCc2n(C)nnc2)=O)CCC(C)(C)CO1 26696,c1(C(=O)N(C2CC2)CC2(C(F)F)CCC2)cccnc1-c1nc(C2CCC2)no1 26697,c1(CC)noc2ncc(C(=O)NC3CC4CC(C3)N(CC(C)OC)C4)cc12 26698,Cc1cnc2n1CC(C(N1CC(N(C)C(C3SCCCS3)=O)C3(CC3)C1)=O)CC2 26699,N1(C(=O)CC2CCN(C(c3cccs3)=O)C2)Cc2n[nH]cc2C1CO 26700,c1(C(N2CCC(C)C2c2cn(Cc3cnco3)nn2)=O)ncn2c1CCC2 26701,c1(OC)ccc(C=CC(=O)NC2CC(C)N(C(c3ccc[n+]([O-])c3)=O)C2)c(C)c1 26702,c1(OC)cc(C)c(C(N2CC3CC3(CNC(C3(C)CC4CC4C3)=O)C2)=O)cn1 26703,N1(CC(=O)N(CCC(=O)N(CCC=C)CC)C(C)C)CCCCC1=O 26704,c1(CN(C(C(=O)NCCOC)C2CC(OC)C2)C)ccc(F)cc1.C(C)C 26705,C1(NC(c2cncc(C)c2Cl)=O)CCN(C(=O)CCOCC2CC2)CC1(C)C 26706,Cc1nn(C)cc1CC(=O)NC(CNC(=O)C(C)Sc1ccc(Cl)cc1)C1CC1 26707,CC(C(O)C(=O)NC1(CCNC(c2cccnc2S)=O)CC1)c1ccccc1F 26708,c1(NC(CC2CCCN(C(C(CCCC)O)=O)C2)=O)c(I)cc([N+](=O)[O-])cc1I 26709,N1(C(CCC2CCN(C(c3cnn(C)c(=O)c3)=O)CC2)=O)CC2(CNC(=O)C2)C1 26710,C1(C(N(C)CC2N(C(CCc3cc(OC)no3)=O)CCC2)=O)CC(C)OC(C)C1 26711,N1(C(c2c(F)ccc(C)c2O)=O)C2CCC1CC(F)(CNC(C1CC13CC3)=O)C2 26712,C1(C(=O)NC(CNC(c2c(C)scn2)=O)(C)C)CCCC(F)C1 26713,N1(C(CN(C)CC)=O)CCC(c2n[nH]c(CNC(=O)C=CC3CC3)n2)CC1 26714,C(=O)(C(O)CC(C)(C)C)NC1(C)CCN(c2snc(C(C)(C)OC)n2)C1 26715,C1(NC(CNC(CSC)=O)=O)CCN(C(=O)CCNC(C)=O)CC1C(N)=O 26716,N1(C(C(CNC(c2cc(C)sn2)=O)C)=O)CC2(C1)CN(C)CCO2 26717,c1(C(=O)NC23CCCC(NC(CC=C)=O)(C2)C3)ccc(Cl)c(F)c1N 26718,c1(N2CCCC(CN(C(C3(OC)CCCOC3)=O)C)C2)cccc(F)c1[N+](=O)[O-] 26719,C1(C(=O)NCC2(COC)CCCC2)(CNC(=O)COCCCF)CC12CCC2 26720,c1(C(=O)OC)cc(C(=O)NCC2(CN(C)C(c3ccn(C)n3)=O)CC2)nn1C 26721,N1(C(c2nccc(C)c2)=O)C2CCC(C2)C1CNC(=O)COCc1ccccc1 26722,c1(C(=O)NCCN(C(=O)Cc2cc(Cl)ccc2F)C)cncc([N+](=O)[O-])c1 26723,N1(C(C)C(=O)NCCC2CCCN2C(=O)COC(C)(C)C)C(=O)CCC1=O 26724,C(=O)(C1OCCc2ccccc21)N(CCNC(CC(C)OC)=O)C(C)C 26725,C=Cc1ccc(C(=O)NCC(F)CNC(=O)C(C)(C)C#N)cc1 26726,C1(C(=O)NCC2C(C)OCC2)CN(C(C2CC(N=[N+]=[N-])C2)=O)CC12CCC2 26727,Cc1cc(C(N2CC(NC(=O)C(=O)NCC(F)F)C2)=O)c(C)cn1 26728,C1(CN(C(C(C)NS(CC)(=O)=O)=O)C)CN(C(c2cc(Br)n[nH]2)=O)CCO1 26729,C#CCC(CC(=O)N1CCCC1C(C)CC)NC(c1cc(O)ccc1F)=O 26730,N1(C(CCCC(C)C)=O)CC2(CCN(C(c3cc(C(F)(F)F)n(C)n3)=O)C2)C1 26731,c1(C2N3CCC(C3)NC2=O)ccc(F)cc1Cl.C(=O)(N(C)C)NC 26732,C12(NC(c3c(C)nsc3)=O)CCN(C(c3cnc(N)cn3)=O)CCC1C2 26733,C1(CCN(C(COCc2onc(C)n2)=O)C)CCCCN1C(C1CC1F)=O 26734,CCC(C(=O)N1CCOC(CNC(=O)Cn2ncc(O)nc2=O)C1)C(C)(F)F 26735,CC1CC2(CC2)CN1C(C1OCCC1CNC(=O)Cc1cccnc1O)=O 26736,S(=O)(=O)(c1ccc(I)cc1)N1CCN(C(C(C)=O)=O)C2C1C2 26737,N1(C(C(CCC)OC)=O)CCC2(CC1)CC(NC(=O)CC(C)CC)C2 26738,C1(NC(C2(CC)CCCO2)=O)CCC(O)CN(C(c2cc(C)no2)=O)C1 26739,C=CCCCC(C(=O)NCC1CN(C(=O)OC)C1)NC(=O)C(C)CC(=C)C 26740,CC(C)(C)CC(O)C(=O)NC(c1cccc(O)c1)CO 26741,c1(CCC(=O)OCC2C(C)CCO2)nc2ccccc2oc1=O 26742,N1(C(c2c(CC)ccs2)=O)CCOCC1CNC(=O)C(C)Oc1ccc(F)cc1 26743,c1(C(N2CC3N(C(CCCCSC)=O)C(CC3)C2)=O)n[nH]c2c1CC(F)(F)CC2 26744,C(CN=c1cc[nH]cc1S(=O)(=O)N1CCC(C)(CO)C1)N(C)N(C)C 26745,C(CC(=O)NC1(CCC(=O)NC2CC(F)C2)CCC1)=C(C)C 26746,c1(C(N(C)CCNC(C2COCC3(CCC3)O2)=O)=O)cccc2nc(O)[nH]c12 26747,c1(C(=O)NC2(C)CCN(C(C(C(C)(C)O)F)=O)C2)cc(O)c2ccoc2c1 26748,c1(C(C(=O)NCc2n(CC)cnc2)NC)ccc(OC)cc1 26749,C1(NC(COCCCC)=O)CN(C(=O)CCc2cnoc2)CC1CC1CC1 26750,N1(C(C=C(CC)C)=O)CC2CC3CC2C1C3NC(=O)CCc1ccccc1OC 26751,C1(NC(C2C(C)=CCS2)=O)CCN(C(=O)CCc2ncnn2C)CC1O 26752,c1(CCOC(C)=O)nc(-c2cccc(Cl)n2)nn1CC(C)O 26753,C(=O)(CC(F)(F)C(F)F)N1C(C(=O)NCC(CCOC)(C)O)CCCC1 26754,C1(C(=O)NC2CCC(C(=O)NC3(CO)CCOC3)C2)CCCCC1(F)F 26755,C(CCCCC(=O)NCC(CC)NC(=O)CC1CN(C)C1)OCC 26756,C1(NC(=O)CCC2CCCCO2)CCN(c2nnc(C(F)F)o2)CC1O 26757,Cc1cccc(C(N2CC(CNC(=O)Cc3ccc(F)cc3)C3CC23)=O)n1 26758,C=Cc1cc(C(=O)NCC(CNC(c2cc(C#N)on2)=O)C(F)(F)F)cc(F)c1 26759,Cc1cn2c(C(=O)NCC3(CNC(c4cn(C)nc4C)=O)CC3)cnc2s1 26760,c1(CCNC(=O)NC(c2ccccc2Cl)C)c[nH]c2ccc(O)cc12 26761,Cn1cnc2c(C(=O)Nc3cccc(Cc4ccc(C#N)cc4)c3)ccnc12 26762,CCC(CCOC)C(=O)N1CC(OC)C(C(=O)NCCCCN(C)C(C)C)C1 26763,C1(COC)(CNC(=O)Cc2ccccc2C)CCCN1C(=O)C(C(C)C)NC=O 26764,N12CCN(C(C)C1)C(=O)c1cnc2nc1.C1(C(=O)NCC)CSCN1C(C)=O 26765,CC1(C)CN(C(C2CCCCS2(=O)=O)=O)CCC1NC(c1cc(F)cnc1Cl)=O 26766,c1(C(C(=O)NC2CCOC2)N(C2C(C)C2)C)ccc(S(=O)(=O)C(C)C)cc1 26767,N1(C(=O)C2=CCCO2)CCC(C2CCN(C(c3cc(O)nc(O)n3)=O)CC2)C1 26768,Cn1cc(CNC(=O)C(C2CC2)NC(c2cnns2)=O)nn1 26769,C(=O)(C1=CCC(C)CC1)N(CC(CNC(CCC#C)=O)(C)C)CC 26770,c1(COC)ccc(C(=O)N(CC(O)CNC(c2cc(C)ccc2O)=O)C)cc1F 26771,C1(NC(C(CC=C)C)=O)CN(C(c2cccc(F)c2NC)=O)Cc2ccnn2C1 26772,N1(C(c2c(CC)c[nH]n2)=O)CCCCC1C1(NC(c2ccc(C)n2C)=O)CC1 26773,N1(C(CC(=O)N(C)C)=O)C2CCC1CC(CNC(C13CCC(C)(C1)OC3)=O)C2 26774,C1(NC(CC(CN(C)C)O)=O)CCN(C(c2cc(F)ccc2Cl)=O)C12CC2 26775,C(=O)(C1Cc2ccc(F)cc21)NCC(C(C)(C)C)NC(=O)CCc1cc[nH]n1 26776,C=CCC(C)C(=O)N1CCOC(CCCNC(=O)CCc2nncs2)C1 26777,c1(C(C(=O)NCCCNC(CC(C)CN(C)C)=O)O)ccc(Cl)c(Br)c1 26778,c1(C(=O)NCC(CNC(c2ccn(CC(C)C)n2)=O)F)cccc2c1CCOC2 26779,c1(C(N2CC(C(C)NC(=O)CCc3nncs3)OCC2)=O)cc(Cl)ncc1N 26780,C(C(C)(C)CC(=O)N1CC(NC(=O)CCc2nnc(S)n2C)C1)OC(C)=O 26781,C1(C(=O)NCC=CC(=O)N(CCCCC=C)C)CC2(CC2)CO1 26782,N1(CC)C(=O)CCC1CC(=O)NC1CN(C(C2(c3n[nH]cc3C)CC2)=O)CC1O 26783,C(=O)(CCCC(=O)NC12CC(CC(C)C)(C1)C2)NN1CCCC1C(=O)NC(C)C 26784,N1(C(C2C(=C)CC2)=O)CCN(C(c2ccc(C(C)(C)C)cc2)=O)CC1CO 26785,c1(C(N(C2CCN(C(=O)COc3cccnc3)C2)CC)=O)ccc2cccnn12 26786,c1(C(N2CC(NC(C3C(C)(C)CC3)=O)CC3(C2)CC3)=O)[nH]c2ccccc2c1Cl 26787,CC(C(=O)NO)NC(c1nc(C(C)(C)C)cs1)c1nnnn1C1CCC1 26788,c1(CC(C(N2CCC(CNC(C3CC(CF)C3)=O)C2)=O)O)cc(Cl)cc(Cl)c1 26789,C(=O)(CS(=O)c1ccc(Cl)cc1)NCC12CCCC(NC(=O)OC(C)(C)C)(C1)C2 26790,c1(C(=O)NCC(C)N(C(=O)Cc2sc(O)nc2O)CC)c[nH]c(C)c(Br)c1=O 26791,C1(C(=O)NC(CCC)C)CCCCCC1NC(c1ncoc1C)=O 26792,Cc1snnc1C(=O)N(CCNC(C1CC(C(F)(F)F)CO1)=O)C1CC1 26793,N1(Cc2cc(C)sc2C)CC2(CCC(CNC(C3(C(F)F)CCOCC3)=O)O2)C1 26794,c1(C(=O)NC(C(=O)N(C(C=C)C2CC2)C)CC2CCC2)cc(C)oc1C 26795,c1(CNC(CC)=O)ccc(CN(C(=O)CC=CC(C)(C)C)C)cc1 26796,c1(C(=O)NC2CN(C(Cn3nnc(C)n3)=O)C(C)CC2)cnn2ccc(O)nc12 26797,N1(C(C(COC)N(C)C)=O)CC(CNC(=O)Cc2c(C)n[nH]c2C)C(C)C1 26798,c1(C(=O)NCCNC(C(N2CCCC(O)C2)C)=O)c(Cl)cc(Br)cc1Cl 26799,c1(C(=O)NC(CCOC)CNC(=O)CN(C)C(C)=O)nccc2ccccc12 26800,C1(NC(C2CCCN2C(c2ncccn2)=O)=O)CCOC12CCCC2 26801,c1(CC(CNC(CCOC(C)=O)=O)NC(=O)COc2ccsn2)ccccc1 26802,C(CC(C)(C)C#N)(c1n(CCOC)nnn1)NCCC(=O)NCC(C)C 26803,COn1cnc(C)c1C(=O)NC1CC(=O)N(C2CN(C(C3CC3C#N)=O)C2)C1 26804,n1(CC)ncc(Cl)c1C(=O)NCC(O)CN(C)C(C1CC1C(C)(C)C)=O 26805,N1(C(CSCCC(C)C)=O)CCCCCCC1C(=O)N(C)CC1CC1C 26806,c1(OC)cc(Br)c(NC(C2CC2NCc2ccc(O)c(O)c2O)=O)cc1C 26807,C(=O)(C(C(C)(C)C)N1CCNC1=O)N1C(C)C(NC(c2cc(N)ccn2)=O)CC1 26808,n1(CC)nnc2c1C(C(=O)NCCc1cccc(F)c1)CN(C(=O)C(O)CC)C2 26809,c1(C(N2CCC(C)(N3CCCC3)C2)C(=O)NCC=C)cc(Cl)cc(Cl)c1Br 26810,O=S(=O)(c1ccc(NCc2ncnn2C2CC2)cc1Br)NC1CC2CCC1C2 26811,Cn1nc(O)cc1NC(C1CC1NCc1cscn1)=O 26812,CC1CN(C(=O)CCc2cccc(C#N)c2)C(C)CN1C(=O)CCc1nc[nH]n1 26813,c1(CC(N2C(CNC(C(C)CC(C)(F)F)=O)CC2)=O)cc(F)cc2c1OCOC2 26814,C(=O)(CC(C)CF)NC(C)CCN(C)C(c1c[nH]nc1-c1cnn(C)c1)=O 26815,N1(C(C2(COC)CN(C(c3c[nH]c4cccnc34)=O)C2)=O)CC2(C1)OC(=O)NC2C 26816,C=CCC(C)(C)CNC(c1cnccc1OC)c1nnnn1CCC(=O)OCC 26817,CN=C(NCC1(C(O)C(C)C)CC1)N1CC2(CCC2)c2ccccc21 26818,CC(CC(=O)N1CCN(C(=O)C(C)(C)N=[N+]=[N-])CC12CC2)CC(C)(C)C 26819,C1(C(=O)NCC(COC)OC)CC12CC(NC(c1ccc(=N)[nH]c1)=O)C2 26820,N1(C(c2c(C)sc(O)n2)=O)CC2COCC2(C(=O)NCC(C)CO)C1 26821,Cc1cc(C(=O)N(CCC(=O)N(C)Cc2ncc[nH]2)CCO)nc(O)c1 26822,c12ccc(F)c(c1)CN(C)C(=O)c1ccncc1-2.c1(C(C)C2CC2)ccccc1 26823,Cc1nc(O)nc(C)c1C(=O)NC1CC(C)N(C(c2ccc(N)c(Cl)n2)=O)C1 26824,CC1CN(C(=O)C(O)Cn2cncn2)CCC1CNC(=O)CCC(C)(F)F 26825,C(=O)(CCCC(=O)NCc1cnc(Cl)cc1F)NC 26826,CC1CN(C(=O)Cc2c(F)cccc2Cl)CCC1NC(c1cc(C(F)F)no1)=O 26827,C1(F)(C(=O)NCC(C(C)C)NC(=O)Cn2cnc(C(N)=O)n2)C2CCCC12 26828,N1(CC)CCCC(N(C)C(C2CN(C(=O)OC(C)(C)C)CC2C)=O)C1 26829,c1(C(N2CC(C(C)=O)C2)=O)cc(C(F)(F)F)cc(N=c2[nH]c(Cl)ncc2F)c1 26830,N1(C(C2CC(F)(F)C2)=O)CCCC(NC(C2(CC3CC3)CC2)=O)C1 26831,C=C(Cl)CCC(=O)NC1CCN(C(c2cncc(N(C)C)n2)=O)C1 26832,N1(C(C(C)C=Cc2ccccc2)=O)CC2CCC1C(NC(=O)C(C)(F)F)C2 26833,N1(C(C2C(CC)C2)=O)CCC2(CC1)CC(NC(c1cc(Br)nn1C)=O)C2 26834,c1(C(=O)NCC(CNC(=O)C(O)Cc2ccccc2)OC)ccnc2c1CCO2 26835,C(=O)(C(CC(C)C)C(C)C)NC(C1CCN(c2nc(COC)nc(C)c2)CC1)C 26836,c1(C(=O)NCC2(O)CN(C(=O)CCc3cn[nH]c3)C2)csc2cccc(F)c12 26837,c1(C(=O)NCC2(C(C)(C)C)CN(C(C3CCCC3(F)F)=O)C2)cccc(=O)n1C 26838,c1(C(N2C(CNC(CC(C(=C)C)O)=O)CCCC2)=O)cn2nc(OC)ccc2n1 26839,CC1CC(C(=O)NC2CCC(CNC(=O)COc3cnn(C)c3)CC2)=NO1 26840,N1(C(c2c(C)nc(C(F)(F)F)o2)=O)CCC2C(C1)CN2C(=O)Cn1nnc(=O)[nH]1 26841,C1(CC)CC(C(=O)NCC(CNC(c2ccc(CF)cc2)=O)OC)CC(=O)N1 26842,C(=O)(C(C)(F)F)NC1C(NC(C2(C(=O)NC)CCC2)=O)CC1 26843,c1(C(N2CCCC(NC(C(CC)NC(C)=O)=O)C2)=O)cc2cccnc2[nH]1 26844,CCC1=NOC(CC(=O)NCC2C=CCN2C(c2csc(C)c2)=O)C1 26845,Cc1ncc(CCNC(=O)C(F)CC2CN(C(c3cn(CCO)nn3)=O)C2)[nH]1 26846,N1(C(c2c(CC#N)ccs2)=O)Cc2nccn2CC(NC(C2CN(C(N)=O)C2)=O)C1 26847,c1(C(C(C)NC(=O)NCCOC(CC)(C)C)C)cccc(F)c1 26848,c1(C(=O)NCCCC(C)NC(C2OCC2(C)C)=O)c(Cl)cccc1Br 26849,O=C(CN=c1cc[nH]cc1)NCC1OCCC1C(=O)Nc1ccc(F)c(CO)c1 26850,N1(C(COCC)=O)CCN(C(C23CCC(CO2)C3)=O)CC1C1CC1 26851,S(=O)(=O)(c1ccc(=NCc2ccnc(CO)c2)[nH]c1)NC(c1nnc(CO)s1)C 26852,c1(NC(C(C2CCN(C(c3cccc(C)c3)=O)CC2)C)=O)cc(Br)c(Cl)cc1F 26853,C1(CCNC(C2(CNC(C=CC(=O)OC)=O)CCC2)=O)CCOC1(C)C 26854,C(=O)(C(C#N)C(C)(C)C)NCC(C(C)C)C(=O)N1CCOCC1C(F)F 26855,c1(CC(N2CC3CCN(C(COCCC#C)=O)C3C2)=O)oc2ccccc2c1C 26856,CCC(C)(CC1CCCCC1)C(=O)N1CCN(C(=O)C(F)F)CC1 26857,c1(-c2c(C(=O)NCC(C)NC(c3cccnc3N)=O)c[nH]n2)ccccc1F 26858,N1(C(C(C)(F)F)=O)CCC2(NC(c3coc(C(F)F)c3)=O)CCCC12 26859,C=CC(C)(O)CCCC(C)C(=O)N1CCCN(C(c2cc(Br)co2)=O)CC1 26860,C(=O)(C1=C(C#N)CCC1)N1CC2(C1)C(=O)N2.C(C(=O)OC)(C1CC1)OC 26861,c1(C(CC(=O)NCCC2CCCC2)NC(c2cncc(Cl)c2)=O)ccc(F)c(F)c1 26862,c1(C(=O)NCC(C2CC2)OCC(=O)NCC(F)(F)F)cccc2c1COC2 26863,C1(C(=O)NCCn2cc(C(N(CC=C)CC)=O)nc2)CCSC(C)C1 26864,C(c1cccnc1)=C(C)C(=O)NC(C)CCCNC(=O)CC1C=CS(=O)(=O)C1 26865,C(CCC(C)(F)F)N(C(=O)CN(C(=O)CC1CC2CC2C1)C1CCC1)C 26866,C12(CNC(=O)C=Cc3ccco3)CC1CN(C(c1nccnc1C(F)(F)F)=O)C2 26867,C(CN=c1[nH]c2c(c(=NCc3noc4c3CC(C)CC4)[nH]1)SCC2)OC 26868,O=C(Nn1ccnn1)C1(c2ccccc2)CC1Br 26869,C(=O)(C(CC(C)C)CC(C)C)N1CC2(NC(C(CC=C)(C)C)=O)CC1(COC)C2 26870,C=CCC(Cc1ccccc1)C(=O)NC(CNC(=O)CCC=C(C)C)CO 26871,C(CC1=CCN(C)CC1)NC(C1(CC#C)CCN(C(C2CCN(C)C2C)=O)C1)=O 26872,Cc1ccc(C(=O)CCC(=O)N(C)CC2CN(C(c3cnccn3)=O)C2)cc1 26873,Cc1onc(C(=O)NC2CCN(C(c3cnn(CC(F)F)c3C)=O)C2)c1[N+](=O)[O-] 26874,Cc1cc(C(=O)NCC2CN(C(c3ccc(F)cc3)=O)CCC2C)cc(C)c1O 26875,C#CCCCC(=O)N1CCN(C2CN(Cc3cnc(Cl)nc3)C2)CC1 26876,C(=O)(C(C)C(O)C(C)CC)N1C2C(C(=O)NCCCCC)CC(C=C2)C1 26877,c1(C(N2C3(CNC(CCCC)=O)CCC(CC3)C2)=O)ccc(Cl)c2occc12 26878,N1(C(c2ccc(NCC=C)cc2)=O)CC(CO)OCC1C 26879,N1(C(c2c(C)ccnc2)=O)CCC(NC(=O)C(F)(F)c2csc(Cl)c2)C(O)C1 26880,c1(NC(C(c2cc(C)ccc2I)N(CCC(N)=O)CC)=O)c(C)cccc1C 26881,C1(C)(C(=O)NC2CCC(N(C(C=C(C)Cl)=O)C)C2)COC(=O)OC1 26882,CCC(C)C(C)C(=O)NCC1CC1NC(=O)CS(=O)(=O)NCC(=O)NC(C)(C)C 26883,C(C1=NOC2CN(C(c3cc(O)nc(O)c3)=O)CC12)NC(=O)C1=CCS(=O)(=O)C1 26884,N1(C(C(C2CCC2)OCC)=O)CC(C(=O)N(C)CCN(CC)CC)C2(CC2)C1 26885,C(N=c1ccn(C(=O)OC)[nH]1)(C1(C=C)CCCC1)c1nnnn1CC(=C)C 26886,CCC(C)C(C(=O)NCCN(C(=O)C(c1ccc(C(C)(C)C)cc1)(C)C)CC)N(C)C 26887,N1(C(CCCCOCC)=O)CC2(C1)C(NC(=O)C(F)F)CCS2(=O)=O 26888,Cc1cccc(C(C)C)c1C(N1CCC(CO)C(NC(c2cscc2C)=O)C1)=O 26889,CCC(C(=O)NC(CNC(=O)CSCC(=O)OC(C)(C)C)(CC)CC)C(C)C 26890,CCC(C)(C#N)C(=O)NCCCOCCCNC(C1CCCC(C(N)=O)C1)=O 26891,C1(C(=O)NCC(c2ccccc2)NC(=O)Cc2ccoc2)CCCCO1 26892,N1(C(C2CC2F)=O)CCN(C(c2[nH]nnc2C2CC2)=O)C(c2cccc(Cl)c2)C1 26893,Cc1cc2cc(C(=O)NC34CC3CN(C(C3(O)CC3)=O)C4)c(Cl)cc2[nH]1 26894,C1(C(=O)NCC2N(C(CC3(C=C)CC3)=O)CC(C)CC2)(CO)CC2CCC1CC2 26895,N1(CC)CC(C(=O)NCC(C2CC2)N(C(=O)CN2C(=O)CNC2=O)C)CC1=O 26896,O(P(C)(=O)CNC(C1(OC)CCN(C(=O)C(C2CC2)OC)C1)=O)CC 26897,C1(C(=O)NCCCN(C(c2coc(CO)c2)=O)CC)CC(C(F)(F)F)CO1 26898,C1(NC(c2cccc3[nH]ccc23)=O)CN(C(C2CCC3CC23)=O)CCC12CCC2 26899,N1(C(c2cc(OCC)no2)=O)CCCCC(N(c2cc(OC)cc(C)n2)CC)C1 26900,C(C(CC(F)(F)F)NC(C1(C)CC1)=O)NC(COc1c(OCC)cccc1)=O 26901,C1(C(N2CCN(CC)CC2)=O)CNC(=O)CN1C(c1ccc[n+]([O-])c1)=O 26902,C1(CNC(CN(CCOC)C)=O)CC2CCC1N(C(C1CCC1C)=O)C2 26903,c1(C(C)=O)ccc(Cl)c(NC(C2COCCN2Cc2ccnn2C(C)C)=O)c1 26904,N1(C(C(C)CC2CCC2)=O)CC2(CCCN(C(=O)C=CC3(C)CCOCC3)C2)C1 26905,c1(OCC(=O)NCC2(F)CCN(C(C3CC=CCC3)=O)C2)ccc(F)nc1 26906,c1(OC)ccc(CC(=O)NC2(C)CN(C(=O)C(C)C3CCCC3)C2)cc1F 26907,c1(NC(c2cc(-c3cc(C)cc(F)c3F)[nH]n2)=O)ccc2ncnc(O)c2c1 26908,C#Cc1ccc(C(=O)NC(CNC(c2cccn2C)=O)CC)o1 26909,c1(C(N2CC(N(C(c3nc(CC)oc3C)=O)C)C2)=O)cc(C)nc(O)n1 26910,C1(C(=O)Nc2c(C)ncnc2)CC2CCC1N2C(C1CCC1C#N)=O 26911,N1(C(C(C=C)O)=O)CCC(CCCCNC(=O)C(n2ccc(C)n2)C)CC1 26912,S(=O)(=O)(c1cc(-c2cc(F)cc(F)c2)ccc1OC)N(Cc1onc(CC)n1)CC 26913,Cc1cc(C(N2CCC(C)(NC(=O)CC3CCC(C)(C)O3)C2)=O)ccc1Cl 26914,c1(C(=O)NC2CC2CNC(c2cc3ncccc3s2)=O)cc2ccc(Cl)cn2c1 26915,CCC(C)(COC)C(=O)N1CCCC(CNC(=O)Cc2cc(C(F)(F)F)co2)CC1 26916,C(C(=O)NOCC(N1CCC(C(C)(C)C)C1)=O)=CC 26917,C1(C)(CC)CC(NC(c2ccc(N)cc2Cl)=O)CN1C(c1cn(C(F)F)cn1)=O 26918,c1(N2CCC(c3c(C)cccc3)C2)nc(N2CC3CC3C2)c2ccsc2n1 26919,N1(C(c2cc(C)nc(Cl)c2)C(=O)NC(C(=O)OC)C)CCc2n[nH]cc2C1 26920,N1(c2c3ncn(CC(CO)OC)c3ncn2)CC=C(c2ccc(Br)cc2)CC1 26921,CC1CN(CC2CCCN2Cc2ccc(N(C)C)cc2)CC(C)O1 26922,C1(NC(c2cc(CC)oc2C)=O)(CO)CCCN(C(=O)C(F)=C(C)C)C1 26923,c1(CNC(CCC=CC)=O)ncccc1C(N1CCC(Cc2ccccc2)C1)=O 26924,c1(C(N2CCCCC2CC(O)C(F)(F)F)=O)cc2c(Br)cccc2[nH]1 26925,c1(C(C)NC(CC2CCOC2)CO)cccc(COc2ccccc2)c1 26926,Cc1cc(F)ccc1COC(C1(C(F)F)CCCC1)=O 26927,CC1CCN(C(=O)C2CC2)CC1.C1(=O)CS(=O)(=O)NC(C)C2CCN1C2 26928,N1(C(CCC(C)C)=O)CCCCC2C1CCCN2C(C1CCNC(=O)C1)=O 26929,C1(NC(C2CC2c2ccsc2)=O)CN(C(c2nocc2Cl)=O)CC1C1CC1 26930,Cc1cc(C(=O)N(CCCNC(c2cnn(C3CC3)c2)=O)C)cn1C(C)C 26931,CC1CN(C(c2csc(S)n2)=O)CC1NC(c1ccncc1-n1cccn1)=O 26932,CCCCCC(O)C(=O)N1CC(N(C)C(c2cc(C(C)(F)F)ccn2)=O)C1 26933,N1(C(C(c2c(C)nns2)N)=O)CC(=O)NC(C)C1 26934,c1(C(N2CC3C(C(=O)NCc4ncc(C)nc4)(C3)C2)=O)c(Cl)ccc(Br)c1F 26935,c1(C(N2CC(CNC(C3(CCC=C)CC3)=O)C(C)C2)=O)ccc(N)c(Cl)n1 26936,C(=O)(C1=Cc2ccccc2C1C)NC(CCOC)CNC(c1nc(Cl)cs1)=O 26937,Cc1ccc(C=CC(N2CCCC(C(C)NC(=O)CC(F)(F)F)C2)=O)cc1Cl 26938,Cc1c(C(N2CC=CCC2C(=O)NOC2CCCC2)=O)nnn1C 26939,c1(C(C)C)nccnc1N1CCCC(C(C)NC(=O)CSCC(N)=O)C1 26940,C1(CC)CN(C(c2ccnn2C2CCC2)=O)CCC1NC(=O)CC(C)(F)F 26941,N1(C(CN(C(c2ncc(C)cc2F)=O)C2CC2)=O)CC2(C)COCC2(C)C1 26942,c1(C(=O)NCC(CNC(C(C)C(F)(F)F)=O)F)ccc2c(c1)NCCC2 26943,C#Cc1cc(F)c(C(=O)N(C2CCC(NC(c3csc(C#N)c3)=O)C2)C)cc1F 26944,CCC(CC)(CC)C(=O)N1CCC(OCCCNC(C2CCC2(F)F)=O)CC1 26945,c1(CNC(C2ON=C(CC)C2)=O)nn(C)c2c1CN(C(=O)C=C(C)C(F)F)CC2 26946,C1(C(=O)NCC(n2cc(C3CCOC3)nn2)C)CCC2(CC1)CC(O)C2 26947,CCC(C(=O)NCCCN(C(=O)C(C)N(C)C(C)=O)CC)OC 26948,C(CCC(C(=O)N(C)Cc1nncn1C)NC(c1csnc1Cl)=O)OC 26949,c1(C(C)=O)ccccc1C(=O)NC1CCCC1(C)NC(c1cc(CO)n(C)n1)=O 26950,Cc1ccc(C(=O)NCCC(O)CNC(C2CC(O)C2)=O)c(N)n1 26951,c1(CCC(=O)NCC2CC(C(N(CC(=O)OC)CC3CC3)=O)C2)nc(O)n[nH]1 26952,N1(C(C(c2ccc(C)cc2)C)=O)CC2CCN(C(=O)C(CO)N(C)C)C2C1C 26953,C(CCCC(=O)NC(CCF)C(=O)N(C)C)N(C)CCNC1CC1.C(=O)O 26954,N1(c2ccnc(C(=O)OCC)n2)CCC(C)C(NC(=O)C(F)C(C)C)C1C 26955,C1(CC(N2CCC(C(=O)NC)C2)=O)CCN(C(=O)Cc2cnnn2C)CC1 26956,c1(COC2CCCN(C(CNC=O)=O)C2)cccc2cncn12 26957,N1(C(C2C(=C)C2)=O)CC=C(C(=O)NCC2Cc3nccn3C2)CC1 26958,c1(C(=O)NC(C(=O)NC(C2CCOCC2)C)Cn2cccn2)cccc(CO)n1 26959,c1(CC)cc(C(=O)NCC(O)C(=O)N(CCCCO)C)n[nH]1 26960,Cc1nc(C=CC(=O)NC2(CCNC(C3(CC(C)C)CCC3)=O)CC2)cs1 26961,C1(C)(C(=O)NCC(CN(C)C(c2csc(-c3ccco3)n2)=O)O)C(C)(C)C1(C)C 26962,C1(C(N(C2CCCNC2=O)C)=O)CCN(C(=O)C(c2cccn2C)=O)C12CC2 26963,C1(C)(C(=O)OC)CCN1C(=O)CCOC1CN(C(=O)C(=O)C2CC2)C1 26964,C1(CC)(CC)CCN(C(C2CCC(C)(C)C2)C(=O)Nc2cccc(Cl)c2C)CC1 26965,N1(C(c2cnc(SC)s2)=O)CC2CN(C(c3ccc(C)nc3)=O)C2C1 26966,C1(NC(C(C)(C)OC(C)=O)=O)CCCC1(C)NC(=O)C=C(C)Cl 26967,C1(c2nnnn2C2COC2)(Nc2ccc(NS(C)(=O)=O)cc2)CCCC2(CC2)C1 26968,C1(C(N2C3CC(NC(C4(C#C)CCC4)=O)CC2CC3)=O)CCc2c(n[nH]c2C)C1 26969,N1(C(C2(C(=O)OCC)CCC2)=O)CCC(N(C(=O)CC2(C)CC2)CCO)C(O)C1 26970,CCCCCCCC(=O)NC(CC)CCC(=O)N(C)CC1CCOCC1 26971,C1(C(N2CCC(CCC(=O)NC(c3nccs3)CC)C2)=O)CCCC1C1CC1 26972,CCCCC(CC)C(=O)N1CCN(C(=O)Cc2ccnn2C)CCC1C 26973,N1(C(C(C)NC(CC)=O)=O)CCC12CN(C(=O)C(C)(C)c1cc[nH]n1)C2 26974,O=C1Cc2c(C(N3CC4(CCN(C(C5C6CCC(=O)C56)=O)C4)C3)=O)cccc2N1 26975,C1(NC(CCCC)=O)CCN(C(c2ccc(C#N)s2)=O)CC1C 26976,c1(C(=O)NC2(C)CC(NC(C3CCN(CC(C)C)C3)=O)C2)n[nH]c2c1CCC2 26977,C1(C(=O)NCC(C(CC)C)C)CCN(C(c2cc[nH]c(=NC)c2)=O)C1(C)C 26978,c1(C(=O)NC2CC(C)(C)CN(C(C3CC3(C)C)=O)C2)cccc2nc(CO)[nH]c12 26979,N1(C(CC2C(C)CCC2)=O)CCCC(C)(CNC(c2scnc2C(C)(C)C)=O)C1 26980,c1(C(N2CCC(NC(C3CCCCS3)=O)CC2)=O)ccc([N+](=O)[O-])cc1O 26981,N1(C(C2C(NC(c3c(C)snn3)=O)CC=CC2)=O)CC(F)(F)CC1CO 26982,c1(CSC)cc(C(=O)NCC2CC(OC)CN2C(=O)C2=COCCO2)ccc1F 26983,N1(C(CC(C)(C)C#N)=O)CC2CCC1CN2C(c1cccc2nccn12)=O 26984,C1(NC(=O)CCN2CCCC2)CN(C(c2cnc(O)o2)=O)C2(CCOC2)C1 26985,N1(C(C(C)NC(N)=O)=O)CC2(C1)C(NC(C1CCCC13CCC3)=O)CCS2(=O)=O 26986,C1(NC(c2cc(CC)nn2C)=O)CC2CCC1(CNC(c1cnc(CC)s1)=O)C2 26987,n1(CCc2onc(-c3ccc4ccn(C)c4c3)n2)cnc2ccccc2c1=O 26988,c1(NC2CCCC(NC(=O)CCCc3cccnc3)C2)ncnc2c1CCO2 26989,C1(C(=O)OC)(C(=O)NCC(O)CN(C)C(c2cc(O)ncn2)=O)CCCCO1 26990,C(=O)(C(C)(C)CS(C)(=O)=O)NC1CC(C)CN(C(=O)Cn2nc(O)ccc2=O)C1 26991,C(N(C)N1CCC(OCC(N2CCC(OC)C(C)(OC)C2)=O)CC1)OC 26992,N1(C(CCC2CCC(=O)N2)=O)CCCC(F)(C(=O)NC2CN(CC(F)F)C2)C1 26993,N(C1CCOc2ccc(F)cc21)C(c1ccc(SC(F)(F)F)cc1)C(=O)OC 26994,NS(=O)(=O)c1ccc(C(N2CCC(CCNC(C3CC3c3ccsc3)=O)C2)=O)o1 26995,c1(C(=O)NCC(CCNC(CCCC(C)=O)=O)(C)C)cc2c([nH]1)CCCC2 26996,c1(C(C(=O)NC2CC(F)(F)C2)N(CC(=O)NC)CC)nc(Cl)cc(Cl)c1C 26997,c1(OCCOC)ncccc1C(=O)NC1CCC(NC(=O)C(F)(F)CO)CC1 26998,N1(C(c2c(NC)nsn2)=O)CCC2(C(N3CC4CC3CO4)=O)CC2C1 26999,N1(C(COC(CC)C)=O)CCC(CNC(=O)Cc2cnsc2)C(CC)C1 27000,c1(OC)cc(Br)c2c(c1)CCN(C(=O)NCC1(OCCO)CCOCC1)C2 27001,N1(C(c2cccc(SCC#C)c2)=O)CCC2(CCCN2C(=O)C(C2CC2)OC)C1 27002,N1(C(C2(CCCC)CC2)=O)CC(NC(=O)CC2CC(N(C)C)C2)C(SC)C1 27003,CCCC(C)(CC)C(=O)NC1CN(C(c2cc(C3(C)CC3)n[nH]2)=O)CC1F 27004,Cc1cc(N)c(C(=O)NCC#CCNC(=O)C(C)(O)c2ccccc2)cc1C 27005,C(CN(C(=O)Cn1cnnn1)C)(CO)(CO)NC(C(N1C(=O)CCC1=O)CC)=O 27006,N1(C(c2[nH]cc(C#N)c2)=O)CCC(CCNC(=O)CC2OCCCO2)C(F)(F)C1 27007,S(=O)(=O)(c1ccc(Br)cc1NC(Cc1cnc[nH]1)CO)NC(c1ccoc1)C 27008,C1(CC(C)NC(C2C(OCC)C2C)=O)CCN(C(=O)C(C)OCC)CC1 27009,CC1(C(=O)N2CC(NC(c3sccc3Cl)=O)C3(CCC3)C2)COc2ccccc21 27010,c1(C(=O)OCC)ccccc1C(N1CCCC1CC(=O)NCC1CCCCO1)=O 27011,CCCCCCC(CC)NC(C1CCCCCN1C(c1n[nH]c(C)c1O)=O)=O 27012,N1(C(C2(C)CCN(C)C2)=O)CC=C(CC(=O)NC2(C)CC(F)C2)CC1 27013,N1(C(CC(CC)C2CC2)=O)CCC2C(C1)CN2C(c1csc(Br)n1)=O 27014,C(C1=NOC2OCCC12)SCC(C(=O)OCC)C 27015,CC1CCC(=CC(=O)N(C(C)(C(=O)NCc2cscn2)C2CC2)C)CC1 27016,CCC(CC(=O)NC(C)CN(C)C(C1CCN(C)C(=O)C1)=O)C(C)C 27017,C1(NC(CC2C(C)=NNC2=O)=O)C2CCCN(C(=O)CCC3CCC3)C2C1(C)C 27018,c1(C2C(=O)N2)ccc(N2CCCCC2)cc1.CC1CC(CS(=O)(=O)C(C)C)CN1 27019,N1(Cc2nnc(OC)c(OC)c2)CCC2CN(C(C)=O)C2C1 27020,N1(C(CN2CCN(CCCC=C)CC2=O)=O)CCn2c(C)nnc2C1 27021,C1(C)(NC(C2(C)N(C(CCSCC)=O)CC=C2)=O)CCC(C)=C(C)C1 27022,n1(CC)c(C(=O)NCC(O)CN(C)C(c2cc(-c3ccoc3)[nH]n2)=O)cnc1O 27023,C(=O)(C1CSc2ccccc21)N1C(C)CN(c2ccc(C(F)(F)F)cc2)CC1 27024,C(=O)(C(CC1CC1)NC(=O)CCC1(C)N=N1)N(CCN=[N+]=[N-])CC 27025,C(C)(C(N)CC(=O)N1CCCC1CC(c1cccs1)O)OCC 27026,N1(C(=O)NCCc2ccsc2)CC2(CCC(F)(F)CC2)C1 27027,N1(C(C(=O)N(CC(C)NC(CSCC)=O)C)CC)C(=O)c2ccccc2C1=O 27028,c1(C(N)=O)ccc(CC(=O)NCC(C)(C)NC(=O)CC2CCC3CC23)cn1 27029,C(=O)(C1=NOC2(CCC2)C1)N(CC(CC)NC(c1cc(C#N)no1)=O)C 27030,CC(C)(O)CC(=O)N1CCC(N(C)C(C2C(c3ccccc3)C2(F)F)=O)CC1 27031,CC1(C)CC(CNC(=O)CC23COCC(C2)C3)N(C(c2cnc(C(F)F)s2)=O)C1 27032,CS(=O)(=O)c1ccc(C(=O)NC2CCN(C(=O)C(F)C3CNC3)CC2)cc1 27033,C1(CNC(c2scc(C)c2)=O)CN(C(=O)CC2CCCC23CC3)CCO1 27034,c1(C(=O)NC(C(=O)NC)C(C)(C)C)coc2c1CN(C(=O)CSCCC#N)C2 27035,c1(C(N(CC(C)(C)CNC(=O)CCc2nncs2)CC)=O)cc(OC)ccc1C 27036,CC1(C)CC(CO)(Nc2ccc(Br)c(F)c2)CO1 27037,C(=O)(C1=C(Cl)CCOC1)NC(COCC)C(=O)NC1CC1(C)C(F)F 27038,c1(OCC)ncc(C(=O)NC(C)(C)CCCNC(=O)Cc2ccno2)cc1Cl 27039,N1(C(N2CCN(C)CC2)=O)CCc2cc(C(=O)NC3CC3)ccc2C1 27040,c1(C(N2CC(N(C(CC(C=C)(C)C)=O)C)C(O)C2)=O)ccc(C)c(Br)c1N 27041,c1(C(=O)NCCOC(CNC(C(C(C)O)C)=O)(C)C)cc2n(c1)CCCC2 27042,c1(C(=O)NC(C)Cn2cc(C(C)(C)C)nn2)cc2c(cnn2C)nc1C(F)(F)F 27043,c1(NC(=O)NCC2CC(SC3CCCO3)C2)cccc(OCCN(C)C)c1 27044,N1(C(C(C)NC(N)=O)=O)CCCC(C)(NC(C2CCC(=O)NC2)=O)C1 27045,N1(C(c2nc(CC)oc2)=O)CC2CCC2(C(=O)NC(CO)CC(C)C)C1 27046,n1(CC(=O)NCC(C)CNC(=O)Nc2cc(C3CC3)on2)cc(Br)cn1 27047,c1(CC(=O)NC2CCCC(NC(C(C=C)O)=O)C2)cc(F)ccc1Cl 27048,N1(C(c2c(C)cco2)=O)CC2CCC1C1CN(C(c3occc3F)=O)CC21 27049,c1(CC(=O)NCC(O)CNC(C23CCC(C2)C3)=O)cccc(Cl)c1 27050,C1(C(=O)NC(C#C)CC2CCCC2)C(CC)CCN1C(c1csc(CC)n1)=O 27051,N1(C(c2cccc(F)n2)=O)CCCC(C2CCN(c3ncnc(Cl)c3F)C2)C1 27052,N1(C(CCCOc2ccc(C(C)=O)cc2)=O)CCC(C2(C(=O)O)CC2)CC1 27053,C1(COC)CCC(C(N(C2(C(=O)Nc3ccsn3)CC2)C)=O)C1 27054,Cn1ccc(=O)cc1C(N1CCOC(C(=O)Nc2nccc(Cl)c2Cl)C1)=O 27055,C1(OCC#C)CCCN(C(C23CC(NC(=O)C(Cl)Cl)(C2)C3)=O)C1 27056,N1(C(c2nc(C(C)OC)sc2)=O)CCCC(N(C(=O)CC2CCC(=O)N2)C)C1 27057,C1(C(N2CC(Cl)CC(OC)C2)=O)CC12CCC1(CC1)CC2 27058,c1(C(=O)NCC(CC)NC(=O)COCC2CCOC2)ccnc2c(Br)cccc12 27059,C1(NC(c2cncc(C)n2)=O)COC2(CCN(Cc3cnn(C4CC4)c3)CC2)C1 27060,C1(C2CC2)(C(N2CCC(NC(CCC(=O)OCC)=O)C2)=O)CCOCC1 27061,C(=O)(C1CCc2nccn21)N1CC2C(NC(C3CCN(C(C)=O)C3)=O)(C2)C1 27062,c1(OCC)cncc(N2CCCC2Cc2ccc(C)cc2)n1 27063,c1(C(N2CC(CC(=O)Nc3ncncc3Cl)C2)=O)ccc2scnc2c1 27064,c1(C(=O)NCC(c2cccc(C)c2)NC(C2ON=C(C)C2)=O)cc(C)nc(C)c1 27065,C(=O)(C(C)C(=O)OCCC(C)C)NC(CN(C(COC)=O)C)C 27066,c1(C(N(CCNC(c2c(C)nc(CC)s2)=O)C)=O)c(F)c(F)cc(F)c1F 27067,c1(C(=O)NCCC2CCN(C(c3cnc(C(=O)OC)s3)=O)C2)nnn(C)c1C 27068,N(C(=NCCF)NCC1(O)CCS(=O)(=O)C1)CC1CC(OC)CN1C 27069,N1(C(Cn2ncc(C)c2)=O)CC(C)(CNC(C2(F)CC=CC2)=O)CC1(C)C 27070,C1(C(N(CCCNC(COCC(C)(C)C)=O)C2CC2)=O)OC(C)(C)OC1(C)C 27071,c1(C(=O)NCCCCC(C)NC(CSCC=C)=O)ccc2n[nH]cc2n1 27072,C(=O)(C1=CSCCO1)NC1C(CNC(CC2C(C)=NNC2=O)=O)CCC1 27073,C(=O)C(=O)CC(C)CC.c1(C(=O)NCCC=CCCC)ncoc1C 27074,Cc1c(C(N2CC3C(CN(C(=O)CCCC4CCC4)C)C3C2)=O)cnn1C(C)C 27075,N1(S(CC)(=O)=O)CCCC1C(=O)NCC(c1ccccc1)NC(=O)C1=CCC1 27076,N1(C(CCP(C)(C)=O)=O)C2CCC1CC(NC(C1CCOC3(CCC3)C1)=O)C2 27077,CC1CCC(CO)N(C(C2C3CC4C(C3NC(c3cc(O)ncn3)=O)C24)=O)C1 27078,N(C(=NCCc1ccc(Br)cc1Cl)NC1CCC1)CCC1CCCN(C)C1 27079,CC1C2CCC(C2)C1C(=O)N(C)CC1CCC(CNC(=O)Cc2nc[nH]n2)CC1 27080,N=c1nc(O)c(CC(=O)NCC2CC2CNC(=O)C(O)CN(C)C)c[nH]1 27081,CCCS(=O)(=O)C(C)C(=O)NCCCOCCNC(=O)CSc1nccn1C 27082,C1(NC(c2c(C)cns2)=O)CC2CC1CN(C(=O)C(C1CCCCCC1)O)C2 27083,CCC(F)C(=O)NCCN(C(=O)CC1CC=CC1)C 27084,c1(C(=O)NCC(CC(=O)NCC(C(=O)OC)C)C2CCC2)cccn2ccnc12 27085,N1(C(C(c2cccc(F)c2)C)=O)CC(CNC(c2cc(Cl)on2)=O)C(C)C1 27086,N1(C(C2C(C=C)C2)=O)CCCN(C(c2ccnn2CCOC)=O)CC1CO 27087,C(=O)(C1=CC2(CCN(C(C34C=CC(CC3)C4)=O)C2)C1)N(CC(F)Cl)C 27088,C1(CNC(c2scc(C)c2)=O)N(C(=O)CC2CC(C)(C)C(=O)N2)CCC1(C)C 27089,N1(CC(N2CC(C)(NC(=O)Cc3ccc(C#N)cc3)C2)=O)CCn2ccnc2C1 27090,C=CCCC(C(=O)NCC(CC)C(C)(F)F)NC(C1CCC1COC)=O 27091,c1(C(=O)NCC(C)NC(=O)CN(C)CCO)cc(Cl)c2n[nH]cc2c1 27092,Cc1cc(C(=O)NCCC2CCC(NC(=O)CC(C)C)C2)c(N)c(Cl)n1 27093,c1(NC(=O)C=CC2CC2)cccc(CNC(c2nc(C(F)(F)F)cs2)=O)c1 27094,C1(CNC(C(C)n2ccnc2)=O)CCC(N(C(=O)CC2CCCC(=O)N2)C)CC1 27095,c1(C(=O)NCC2(C(N(CCCCN(C)C)C)=O)CCCO2)ccc(C2CC2)cc1 27096,C1(CCOC)CN(C(c2ccc(C(O)CF)cc2)=O)CCN1C(C1CC1F)=O 27097,c1(C(=O)NC(CC)CN(C(=O)CC2CCOC2)C)ccnn1C(F)F 27098,C(C)(CCCC(=O)NCc1c[nH]nc1C1CC1)NC(COCCC=C)=O 27099,C1(C(=O)NC2CON(CC)C2=O)CN(C(c2ccc(C)nc2O)=O)CC1(F)F 27100,N1(C(c2cccc(COC)n2)=O)CC2CCC2(CCNC(C2(CF)CC2)=O)C1 27101,c1(CCC)onc(C)c1C(=O)NCCC1(C)CCN(C(C2(C#N)CCCO2)=O)C1 27102,C=CC1CN(C(=O)C2=CCN(C)C2)CC1NC(c1c[nH]nc1-c1ccoc1)=O 27103,C1(CC)CN(C(c2cccc(C)c2)C(=O)NC)CC(=O)N1 27104,CC1CC(C)CC2(C1)NC(=O)N(CC(=O)NC1CC3CC1C(O)C3O)C2=O 27105,Cn1cc(C(F)(F)C(=O)NCC2CCCC2NC(c2cocn2)=O)ccc1=O 27106,c1(-c2cccc(C3C(C(N4CCC5(CCCC5)C4)=O)C3)c2)cccc2c[nH]nc12 27107,CN=c1ccc(C(=O)NC(C(=O)NCC2CCOC(C)(C)C2)C(C)C)c[nH]1 27108,c1(C(=O)NCC2C(NC(c3cc(CC)oc3C)=O)CCC2)ccc(C)cc1OC 27109,N1(Cc2c(=N)cc[nH]c2)CCCC(C(N2CC3CCCC23)=O)CC1 27110,Cc1cccn2ncc(C(N3CC(O)(CN(C)C(C4CNC(=O)N4C)=O)C3)=O)c12 27111,C1(C(=O)NCC2CC(NC(C(C)OC)=O)C2)CC2CCC1O2 27112,N1(C(CCC#CC)=O)CC(NC(c2ncccc2O)=O)CC2(CC2)C1 27113,C1(CC(=O)NCC(=O)NCCOC)CCCN(C(=O)CC(=O)OC)CC1 27114,CN1CC(F)CC1C(=O)NCC1CCC(NC(C2CC2CC(C)(C)C)=O)C1 27115,C1(CNC(CC(C)C#N)=O)CC2(C1)CN(C(=O)Cc1ccoc1)C2 27116,C1(CCNC(C2C(OCC)C2)=O)CCCN1C(=O)CSC(F)F 27117,c1(C(=O)NCC2(F)CC(NC(c3c(CC)ocn3)=O)C2)ccc2c(c1)CCC=C2 27118,C1(C(=O)NCCCCN(C(C2(COC)CC=CC2)=O)C)CCC(C)(C)CO1 27119,C1(NC(c2ncnc3ccsc23)=O)COC2(CCN(C(c3ccc[nH]3)=O)C2)C1 27120,c1(C(=O)NC2CC3C2CCN3C(C2(F)CC2)=O)nnn2c1C(=O)NCC2 27121,C(=O)(C1=NOCC1)N1CCC(CN(C(C(CC)OC)=O)Cc2ccccc2C)C1 27122,C(C(CC(C)C)C(=O)NCC(CC(C)C)OC)NC(CC(C=C)(C)O)=O 27123,c1(C(=O)NC(C(C)NC(c2c(CC)c[nH]c2)=O)CO)ccccc1[N+](=O)[O-] 27124,C1(C(=O)NC(C)CC2CN(C(=O)CCc3cnoc3)C2)CCc2nncn2C1 27125,C1(C(=O)Cl)(NC(c2cccnc2C2CC2)=O)CCOCC1.N12CCCC(C1)C2 27126,c1(OC)cc(C(=O)Oc2ccccc2OCC2CCOC2=O)cc([N+](=O)[O-])c1 27127,C(=O)(C(F)CC(C)(C)C)NCCN(CCC)C(c1ncccc1N)=O 27128,C1(N(C(C(C2(O)CN(C(c3c(C)ocn3)=O)C2)F)=O)C)CS(=O)(=O)C1(C)C 27129,Cn1nc(Br)c2ccc(C(=O)NC3CCCC3C(N3CCS(=O)CC3)=O)cc12 27130,N1(C(C(CC(CC)C)C)=O)CC(C)CN(C(c2cccc(OC)c2N)=O)CC1C 27131,C12(CNC(C(CC3CC3)NC(=O)CC34CCCC3C4)=O)CCC(CC1)O2 27132,C(=O)(CCC(=O)c1ccc(Br)s1)NC(C)CNC(C1COCCO1)=O 27133,N1(C(C(C=C)(F)F)=O)CC2(C=C(C(=O)NC(c3cnn[nH]3)C)CO2)C1 27134,N1(C(C(C(=O)NC)(C)C)=O)CC(C(=O)N(C)CCc2nccs2)CCC1(C)C 27135,C(=O)(CC(CC)C(C)(C)C)N(C1CCN(C(=O)CCCNC(C)=O)CC1)CCC 27136,C(CC(C)(C)C(=O)NC(CNC(=O)COCCF)C1CCC1)OC 27137,S(=O)(=O)(c1cc(F)cc(F)c1)N1C2CC(N(CCC#N)C)C(C2)C1 27138,C(=O)(CC1OCCc2ccsc21)N1CC(NC(C(CC#C)CC#C)=O)C(C)(C)C1 27139,C(C1c2ccccc2CC1C)NC(N1CCC(c2ccc(C)cc2)C1)=O 27140,c1(OC)cc(C(=O)N=c2ccn(C3CN(Cc4ccsc4)C3)[nH]2)c(F)c(F)c1F 27141,C1(C(N2C(C3(C)CC3)CCC2)=O)CC(O)CN1C(C1CCC1C(=O)C1CC1)=O 27142,n1(CC(=O)NCC2COCCN(C(=O)CSC3CC3)C2)nc2c(n1)CCCC2 27143,C1(CCNC(c2ccc(N(C)C)cc2)=O)CN(C(C2(F)CCC2)=O)CCCO1 27144,c1(N2CC(NC(c3ccnc(N4CCCC4)c3)=O)C2)nc(Cl)ncc1C(=O)O 27145,c1(C(N2CC(NC(=O)CCCn3c(O)nnc3O)C(O)C2)=O)n[nH]cc1[N+](=O)[O-] 27146,CN1CC2CCC(C1)N2C(C1CC12CN(C(C1CC1c1ccc(O)cc1)=O)C2)=O 27147,CC1(NC(=O)CNc2ncccn2)CC(NS(C)(=O)=O)C1 27148,N1(C(C(C)O)=O)CCN(C(c2sc(Br)nc2Br)=O)CC1CO 27149,C1(C(=O)NCC(CNC(c2ccc(CC)c(CC)c2)=O)O)CN2CCN1CC2C 27150,N1(C(c2n[nH]c(C)c2O)=O)CCC2CN(C(C3CCCC(O)C3)=O)C2C1 27151,Cn1c(=O)n(C)c2cc(CS(=O)CC3CC4(CCC(C(=O)O)CC4)C3)ccc12 27152,C(CN=c1cc[nH]cc1S(=O)(=O)NC1CCCSCC1)c1c(C)c(Cl)c(Cl)cc1 27153,c1(OCc2scc(CCC)n2)ccc([N+](=O)[O-])cc1.C(=O)(CCCCOC)NCCS 27154,c1(C(=O)NCC=CCNC(CN2CCC(C)C2)=O)cc(Br)cnc1NC1CC1 27155,N1(C(C2C(C)=CCS2)=O)CCOCCC1C(=O)Nc1cnc(C(C)C)nc1 27156,CCC(F)(F)CC(=O)N1CCC(C)C(NC(c2cc(N)cc(N)c2)=O)C1 27157,C(CNC(=O)Cn1cc(N)cn1)(C(C)(C)C)NC(C1(CC=C)CCC1)=O 27158,c1(C(N(C2CCCCN(C(C3CC3C(N)=O)=O)C2)C)=O)cc2cn[nH]c2cn1 27159,C1(NC(C2CCC(CC)O2)=O)CCN(C(c2cc(C)cc(Cl)n2)=O)CCC1CO 27160,C1(CNC(C2(CCCC)CCCC2)=O)CCN(C(=O)CCc2nncs2)CC1O 27161,C(CNC(C1CC1c1cccc(Cl)c1)=O)(C(C)(C)C)NC(C12CC(C)C1C2)=O 27162,C1(CC(C)NC(C2CC2)=O)CN(C(=O)C=CC(=O)NC2CCC2)C1 27163,N1(C(C(=O)NCC)=O)CCCC(CC)(NC(c2cnccc2N(C)C)=O)C1 27164,C1(C(N2CCC=C(C)C2)=O)CCN(C(=O)CCCC(C)(C)C)C(C)(C)C1 27165,N1(C(CNC(=O)OC)=O)CCCC(C2CCN(C(=O)C=Cc3csc(C)n3)C2)C1 27166,N1(C(C(C(C)C)OCC)=O)CC2CC(NC(c3c(C)csc3Cl)=O)C1C2 27167,N1(C(c2c(CN(C)C)cco2)=O)CCOC(CNC(c2cccc(=O)o2)=O)C1 27168,Cc1ccc(CC(C)C(=O)N2CCC2CNC(=O)Cc2ccc(Cl)cn2)cc1 27169,N1(C(CSCCC#N)=O)CC2CC(NC(=O)Cc3csnn3)CC2C1 27170,C(CC(C)(C)C)(C(=O)NC1CCC1NC(c1ccc(F)c(CC=C(C)C)c1)=O)OC 27171,O=C1CCN(CC(=O)NCCNC(=O)CC2CC=CCC2)CC1 27172,C(=O)(C(C)C(O)CC)NC(CC=C)C(=O)Nc1ccc(CO)cc1O 27173,C(C(C)C(=O)NOCC1CCOCC1)NC(C(COC)(C)OC)=O 27174,CC(=O)CCCC(=O)NCCN(C1CCCCC1)C(C1CCCC1P(C)(C)=O)=O 27175,N1(C(c2ccn3c2CCCC3)=O)CC2CCCC(O)C2C1 27176,N1(C(C(C2CC2)SC)=O)CCC(O)(C(C)NC(C2CCCN2C(=O)C2CC2)=O)C1 27177,c1(C(=O)NC2C3(CC(NC(C4=NOC(C)C4)=O)C3)C2)cc2cc(Cl)ccc2o1 27178,c1(C(N(C)CC2CCCN(C(C(C(C)O)(F)F)=O)C2)=O)c(F)cc(F)c(F)c1F 27179,c1(SC)cc(C(=O)NCCC(C)N(C(=O)C=CC(C)(C)C)C)ccc1N 27180,C(=O)(C1=CCCOC1)NCC1(NC(c2[nH]ccc2CC)=O)CCOCC1 27181,c1(C(N2C(CCCNC(c3ccno3)=O)CCC2)=O)cnc(C(F)(F)F)cn1 27182,Cc1c(C(=O)NCC(C)N(C)C(C2CCC(=O)N(C)C2)=O)nn2ccccc12 27183,N1(C(C2C(C)C2)=O)CC(NC(=O)C2=CCCCO2)CC12CCC2 27184,n1(CC(=O)NCC2CC2CNC(C2CCC(CCO)CC2)=O)ccc(O)nc1=O 27185,N1(C(c2c(C)cc(C)s2)=O)CCC(CO)C(NC(=O)Cc2cccnc2C)C1 27186,C1(CC(=O)NCCN(C)C(c2ccnc3ncnn23)=O)CCCCCC1(F)F 27187,c1(C(N(C2CCCN(Cc3ccccc3CO)CC2)C)=O)cccn(C)c1=O 27188,c1(OC)cccc(C(=O)NCC2CC(NC(=O)CCCC(N)=O)C2)c1O 27189,N1(C(C2C(CC)CCCC2)=O)CCC(COC)(NC(=O)CCC2(C)CC2)CC1 27190,N#Cc1ccsc1C(N1CCC(NC(=O)C=Cc2ccco2)C1)=O 27191,CCC(C(=O)NCC12CC(NC(=O)C(F)OC)(C1)C2)n1ccnc1 27192,c1(NC2CCC(NC(C3N(CC)CC3)=O)CC2)cc(OC)nc(C(F)(F)F)n1 27193,Cc1cc(C)c(CNCC2COCCN2c2ncc3ccsc3n2)c(C)c1 27194,Cc1ccc(C(=O)N(CCCNC(C2C3CCCCCC23)=O)C)c(O)c1C 27195,c1(C(c2nnnn2CC)NC(c2scc(CC)n2)C)nccc(C(F)(F)F)n1 27196,C1(CC(=O)NC2CCC2CNC(c2cccc[n+]2[O-])=O)CCCC2(CC2)C1 27197,C1(NC(CCSCCC)=O)CC2CCC1CC2NC(c1csc2nccn12)=O 27198,c1(C(C)=O)oc2cccnc2c1C(=O)NC1CCN(Cc2cccc(OC)c2)C1 27199,N1(c2ccnc(OC)n2)CC2(CCCN2C(c2ccsc2C)=O)C1 27200,C1(CNC(C2CCCC2)=O)CCCN1Cc1ccc(Cl)o1 27201,c1(C(N2CC(NC(C3CCOC(=O)N3)=O)CC(C)C2)=O)ccc2ccn(C)c2c1 27202,C1(F)(C(=O)NCCc2onc(C)n2)CCCN(C(=O)C=C2CCC2)C1 27203,Cc1c(O)ccc(C(N2CCCC(C(C)NC(C3(CF)CCC3)=O)C2)=O)c1C 27204,C1(NC(CCc2cc(C)on2)=O)CC2CCC(C1)N2C(C1COC(=O)O1)=O 27205,C(=O)(C1=CCCCO1)N1CC(n2cc(CNC(C3(COC)CCCO3)=O)nn2)C1 27206,C(=O)(CC1OCc2ccccc21)NCC(C1CCCCC1)NC(=O)C#CC1CC1 27207,C1(C(N2CC3(CN(C(c4cc(=N)[nH]cc4)=O)C3)C2)=O)C2Cc3c(Cl)cccc3C12 27208,C1(C)(COC)CN(C(=O)C(c2ccc(F)c(Cl)c2F)O)Cc2ccccc2O1 27209,CC1CN(C(=O)C(C)Cc2cccc(F)c2)CCC1CNC(=O)C1=C(Cl)CC1 27210,CC1CC(NC(C2(C)CSC2)=O)CCN1C(C1CN(C(N)=O)C1)=O 27211,N1(C(C(COC)NC(c2[nH]nnc2C)=O)=O)CCN2CC(F)CC2C1 27212,c1(C(N(C2CN(C(C3CC(CF)C3)=O)CC2F)C)=O)cnc2c(C#N)cnn2c1 27213,CC1(C)CC(c2nn[nH]n2)CN(S(=O)(=O)CC2(C)CCCC2)C1 27214,Cc1cccc(CNC(C2CC2c2ccccc2-c2cncn2C)=O)n1 27215,c1(CN2CC3(C(C(N(CC(O)CO)C(C)C)=O)C3)C2)cc(Br)c(F)cc1Cl 27216,C1(C(=O)NCC2CCCN(C(C3OCCN(C)C3)=O)C2)CCC(=O)N(C)C1 27217,c1(C(N2CCC(NC(CC(CC)C3CC3)=O)C2)=O)cc2ccccc2n1CC 27218,C(C(O)C(=O)NCC1(C(C)NC(=O)CC(C)NC=O)CC1)OC.C(C)(C)(C)S 27219,c1(C2(N(C)CC3CCCCO3)CCC2)nnc(N2CCCC2)n1CC1CCOC1 27220,C1(NC(CCC(=C)Cl)=O)CCCC12CN(C(C1C3CC4C(C3=O)C14)=O)C2 27221,C=CC1CCN(c2nnc(-c3[nH]c(=N)[nH]c3Br)n2C)CC1 27222,N1(C(c2cc(SC)c(C)o2)=O)CCC2CN(C(C3CC(N(C)C)C3)=O)CCC2C1 27223,N1(C(C(CCOC)(C)C)=O)CCCC(C2CN(C(C3(S(C)(=O)=O)CCC3)=O)C2)C1 27224,c1(C(=O)NC(C(=O)N(C)CCn2ccnc2)Cc2cc[nH]n2)cn2ccccc2n1 27225,C12(CNC(C(COC)C)=O)CCC1CN(C(c1csc(Br)c1C)=O)C2 27226,c1(C(N(CCOCCNC(CC(CCCC)O)=O)C)=O)cccc2c1OCC2C 27227,C1(C(=O)NCCC(C)(C)NC(c2c(C(C)(C)C)noc2)=O)C2CCCC(F)(F)C12 27228,CCCCCC(O)C(=O)NCC1CN(C(C2COCCN2C)=O)C1 27229,N1(C(C(CCNC(CCN(CCC)C)=O)O)=O)CCCCC(C)(F)C1 27230,c1(C(=O)NCCCN2CCC(NC(c3cc[nH]n3)=O)C2)cc(F)cc([N+](=O)[O-])c1 27231,C12(CNC(c3c(OC)c[nH]n3)=O)CCC1CCN2C(c1cnco1)=O 27232,C1(NC(CCCOC(C)(C)C)=O)CN(C(=O)CN2CCN(C)C(=O)C2)CCC1C 27233,CC1COc2c(C(=O)NC3CN(C(=O)CC4(C5CC5)CC4)CCC3O)cnn2C1 27234,CCC(CNC(C1CC(OC)CN1C(=O)CSc1ccccn1)=O)CC(C)C 27235,N1(C(C2N(C(CC3CC(=C)C3)=O)CCC2CC)=O)CC(C2CCCC2)C1 27236,C(C)(C)(CC(C)NC(=O)C(F)C1CC(NC(=O)CCN2CCCC2=O)C1)OC 27237,c1(C(=O)NCCN(C(C2(CC)CCOC2)=O)C)ccc(C(C)C)nc1O 27238,c1(CNC(C2(C)C(C)(C)C2)=O)nnc2n1CCN(C(c1ccc(Cl)c(N)c1)=O)C2 27239,Cc1sc(C(=O)NCCCN(C(=O)CC23CCC(CC2)C3)C2CC2)nc1O 27240,c1(C(=O)NCCN(C)C(C2CCCOCC2)=O)ccc2c(c1)CCCC(=O)N2 27241,C1(CNC(=O)NC(c2ncccc2Br)C)CCCOC1c1cn[nH]c1 27242,N1(C(CC=C=C)=O)CCCC(NC(c2coc(Cl)n2)=O)CCC1 27243,Cc1cc(O)cc2c1CN(C1CC3CC1N(C(c1ccoc1I)=O)C3)CC2 27244,c1(CCC(=O)N(CC(C)NC(c2ncccn2)=O)C)nc2cc(Cl)ccc2s1 27245,n1(CCC)cc(C(=O)NC2CC(N(C(=O)Cc3cccn3C)C)C2)c(C)n1 27246,C1(C#N)(COC)CCN(C(c2cc(C3CCCN3S(C)(=O)=O)[nH]n2)=O)CC1 27247,c1(OC)cccc2c1CN(N1CCC(CCN(C)C)CC1)C2 27248,CC(C(CO)NC(c1cnc(C2CC2)[nH]1)=O)NC(=O)C(c1cccn1C)=O 27249,c1(C(=O)NCC2(NC(c3ccn(CCC)n3)=O)CC2)sc(C)c(Br)c1C 27250,Cc1ccc(C(N2CC=CC(NC(c3cccn3C)=O)C2)=O)c(F)c1F 27251,c1(C(N2CCCC(NC(CCOC)=O)C2C)=O)c(C)c2cc(O)ccc2oc1=O 27252,c1(CC(=O)NC(CC=C)CNC(=O)Cc2cccc(Cl)c2)ccc(C)cc1Cl 27253,c1(C(=O)NC2CCN(C(c3c(SC)ccs3)=O)C2)cc2c(cn1)OCCC2 27254,C1(NC(c2cn(CCC)nn2)=O)(CO)CCCN(C(C2(F)CC=CC2)=O)C1 27255,CCC(CC)C(C)C(=O)NCCCC(C)(C)NC(C1CCC(C)O1)=O 27256,N12CCC(F)(F)C(C1)C2.Cc1c(CNC(c2ccccc2)C2CC2)c[nH]c1C#N 27257,c1(C(=O)NC2(C)CC(NC(C3(C)N(C)CC(O)C3)=O)C2)cc(F)c(Cl)cc1F 27258,N1(C(C(COC)C)=O)CCCCCC(NC(c2cc(C)cnc2C)=O)C1 27259,c1(C(=O)NCCNC(Cc2c(C)n[nH]c2C)=O)ccc2c(c1)N(C)C(=O)C(C)O2 27260,Cn1cc(S(N)(=O)=O)cc1C(N1CC(NC(=O)CCCN=[N+]=[N-])CC(C)(C)C1)=O 27261,N(C(=NCCc1ccccc1F)NCC1=CCOCC1)Cc1cc(C)on1 27262,C1(C)(CNC(c2c(C)nco2)=O)CCN(C(=O)CSCc2cccnc2)CC1 27263,C(C(C(C)(C)C)NC(C1(O)CC1)=O)NC(c1cc(C(=O)OC)sn1)=O 27264,C1(C(N2CC(OCCOC)C2)=O)(OC)CCN(C(=O)COCC(C)C)CC1 27265,C(=O)(CC(=O)N(CC(=O)N(C1CC1(C)C)C)CC1CC1)NCC 27266,c1(CC=CCC(=O)NCCCCN(C)C(C2CCC3CC23)=O)ccccc1 27267,C(C(CC(C)C)C(=O)NC(c1ccccc1)CO)NC(c1cnn(C=C)c1N)=O 27268,CCC(CC(=O)NCC1COCCN(C(=O)C(F)C2CCC2)C1)CC(C)C 27269,CCC(C)(C)CCCC(=O)NCC1CCN(C(=O)C#CC(=O)N(C)C)CC1C 27270,O=C1NC2CCC1CN(C(=O)C(F)C1CC(NC(C3CC4OC3C3CC43)=O)C1)C2 27271,Cc1cc(C)c(C(=O)NCC(C)C(=O)NCCc2nccs2)s1 27272,C1(OC)(CNC(=O)C(C)c2ccsc2)CN(C(=O)CC2CC(=O)C2)C1 27273,C1(CCNC(CSCC=C)=O)CCCN(C(=O)C(C)Cn2ccc(C)n2)C1 27274,C(=O)(C#CC(C)(C)C)N(C1CCN(C(c2ccccc2-n2cnnn2)=O)C1)C 27275,c1(C(N(C(CSC)C)C)=O)cn(C2CCCNC2)nn1 27276,C1(NC(c2cc(C)c(F)cc2Cl)=O)CN(C(C2CNC(=O)N2)=O)CC12CCCC2 27277,Cc1ncc(C(=O)NCC2CC(O)CN2C(=O)CC2CCN(C)C2)n1C(F)F 27278,c1(N2CCC(OCC)CC2)nc(=NCc2cc[nH]n2)[nH]c2c(C)nn(C)c12 27279,CCCCC(CC)C(C(=O)NC1CCC1)N1CCc2sccc2C1C 27280,C(CC(C)C(=O)NCc1ocnc1C(=O)NCCCC1CCC1)OC 27281,c1(NC(C(C)(C)c2cnsc2)=O)nc(O)ccc1-c1ccccc1 27282,C1(c2onc(Cc3n(C)ccn3)n2)CC12CCSCC2 27283,c1(CC)cc(CC)nc(N2CCC(CNC(=O)CC(C)(O)C3CC3)(OC)CC2)n1 27284,N1(C(COCCCC)=O)CC2CCC(CNC(C3CC3(C)CC)=O)(C2)C1 27285,C(C(CO)C(C)CC)NC(C1C(CCC)CN(C(=O)C(C)(C)N(C)C)C1)=O 27286,C1(CC(=O)NCC2CCCCS2)CCN(C(c2cc(Cl)ns2)=O)CC1 27287,C12(Cn3cc(CCC(=O)NCCC(COC)(C)O)nn3)CCCC1C2(F)F 27288,C1(C(N)=O)CCN(c2nnnn2-c2nc3c(s2)CCC3)CC1O 27289,c1(C(=O)NC(CCCC)CNC(c2ccc[nH]2)=O)cnc(O)c2ccsc12 27290,CCCCC(CNC(=O)CCCc1ccccc1)NC(=O)CC1CCC12CCC2 27291,N1(C(c2nc(C)[nH]n2)=O)CCN(C(c2sc(C(C)C)nc2C)=O)CC1C(F)F 27292,N1(C(C(C)Cn2cccn2)=O)CCCC(CC(N2CCC(CCO)CC2)=O)CC1 27293,Cc1nn(-c2ccncc2)cc1C(=O)N(CCCNC(=O)C(C)(C)CF)C 27294,C(=O)(CCC(=O)NC1CC1CNC(=O)CCCCN1C(=O)CCC1=O)OC 27295,CCCCCC(C)CC(=O)NCc1cc(C(=O)N(c2cccc(C)c2C)C)cs1 27296,C(=O)(CC(CC)CC(C)C)NC(CCC(=O)NCCC(=O)NCC(C)C)C(C)C 27297,N1(C(=O)Nc2cn(CCN(C)C)nc2)CCc2nc(Cl)cc(Cl)c2C1 27298,c1(C(N(CC(C)NC(CCCn2c(C)nc(C)n2)=O)C)=O)cc2ccsc2n1C 27299,c1(NC)ccc(C(N2CCN(C(c3ccncc3F)=O)C(C)C2)=O)cc1F 27300,CCC(CCC(=O)NCC(O)Cn1cccn1)NC(c1nc(CC)oc1C)=O 27301,C1(NC(C(C)c2ccco2)=O)CN(C(=O)C=CC2(C)COC2)CC1C1CC1 27302,N1(C(C(C)(C)CF)=O)CCOCC(C)(CNC(c2ccccc2)=O)C1 27303,Cc1cnc(CNC(C2CCN(C(=O)C(c3ccccc3)C3CC3)C2)=O)o1 27304,C12(NC(CC(CC)SC)=O)CCCCC1CN(C(=O)CCCS(N)(=O)=O)C2 27305,N1(C(C(C)n2cncn2)=O)CC2CC2(C(=O)NOCCF)C1 27306,CC(c1ccccc1)=CC(=O)NCC1(NC(C2CC3CC2C2CC32)=O)CCCC1 27307,c1(C(N2C(COC)(CNC(=O)C=C(C)C(C)C)CCC2)=O)cccc(F)c1C#N 27308,C1(C(N2C(C(C)NC(c3c(C)csn3)=O)CCC2)=O)CCCN(C)C1 27309,c1(C(C(=O)NCC2CCN(C(=O)C=Cc3nccs3)C2)O)cc(Cl)cc(Cl)c1 27310,C1(NC(c2c(C)ncnc2)=O)(CO)CCCN(C(c2ccccc2Br)=O)C1 27311,C=CCCCCCC(=O)N1CCCC(CCC(=O)N(C(C)C(C)CC)C2CC2)C1 27312,c1(C(=O)OC)cc2c(s1)CCOC2CNCC1C(C)(C)C1(F)F 27313,C1(SC)CN(C(C2(OC(C)C)CCCCC2)=O)CC1NC(=O)C=C(C)C 27314,C(=O)(C1=NOC(C)C1C)N1CC2C(CC(N3CCC(SCC)CC3)=O)(CC2)C1 27315,N1(C(CC(C)F)=O)CCc2sc(CNC(=O)CN3CCCC3C)nc2C1 27316,C1(C(=O)NC23C(CN(C(C4N(C(N)=O)CCC4)=O)C2)C3)CS(=O)(=O)CC12CC2 27317,c1(C(N2CCN(C(C(C(C)C)C)=O)CC2C)=O)cccc2ccnn12 27318,N1(C(C(CC(F)F)NC(=O)C(C2CC2)C2CC2)=O)CCN2C(=O)OCC2C1 27319,C#Cc1cncc(CN2CCN(C(=O)CN3C(C)CCCC3C)C(CCO)C2)c1 27320,N1(C(CCOCC#C)=O)CCC(C)C(NC(c2ccc(NC(C)=O)cc2C)=O)C1 27321,c1(CCC)ccc(C(=O)NCC(C(C)C)NC(=O)C(C)CSC)cc1[N+](=O)[O-] 27322,C(=O)(CC1=CCOCC1)NC(C1CC(NC(C2CCCC2(F)F)=O)C1)C 27323,CC(C)CCCC(C)CNC(C1CC(C)CN(C(c2cncc(F)c2)=O)C1)=O 27324,CCCCC(C)(F)C(=O)N(CCC)CCNC(c1nccnc1N)=O 27325,c1(-c2c(C)n[nH]c2)ccc(CN(C)C(C2CCC(=O)O2)=O)c(F)c1 27326,c1(C(=O)NCC2C(C)(C)C(NC(=O)C=CC3CCC3)C2)cncc2[nH]ccc12 27327,C(=O)(C(F)(F)C1CC1)NCCNC(C1(n2cncn2)CC1)=O 27328,N1(C(C(COC)C)=O)CCCC(O)(CNC(c2ccc(C(F)(F)F)cc2Cl)=O)C1 27329,C(=O)(C(C)C(C)(C)O)NC1CCCN(C(CCSc2c(OC)cccc2)=O)C1 27330,c1(C(=O)NCCCC2N(C(CC(C)SC)=O)CCCC2)cccc2nncn12 27331,c1(C(C)C)n[nH]cc1C(=O)NCC(O)CN(C(=O)CCc1ccsc1Cl)C 27332,C1(NC(c2csc(C)c2C2CC2)=O)CCCC12CN(C(=O)Cn1ccnc1C)C2 27333,C(=O)(CC(C)(C)C#N)NC12CC(CNC(c3c(C(=O)OC)cco3)=O)(C1)C2 27334,c1(CN(C(CCNC2CC(=O)C2)=O)Cc2cnccn2)ccccc1 27335,C1(CNC(C(C(C)C)(C)C)=O)CN(C(c2ncccc2Cl)=O)CC2(CCC2)O1 27336,N1(C(C(CSC)O)=O)CCCC12CCC(NC(=O)CN(C)C1CC1)CC2 27337,C(CC(F)F)(C(=O)N(C)Cc1ccccc1F)NC(C1C(C)SCCC1)=O 27338,N1(C(CNCc2c(C(=O)OC)cco2)=O)C(C)CCC1C 27339,CC(C(CO)NC(=O)CCc1cncn1C)NC(c1cn(C2CCC2)nn1)=O 27340,c1(C(=O)NC2C3CN(C(C=CC(C)C)=O)CC2CC3)ccc2c(c1)CNC2=O 27341,C1(NC(C(CSC)C)=O)CCSC12CN(C(=O)CCc1ccc(O)c(F)c1)C2 27342,CCCCCC(CC)C(=O)NC1CC(NC(c2ccc(Br)cc2C)=O)C1 27343,c1(C(N2C(C)(C(=O)Nc3cccc(OC)c3)CCC2)=O)cc(Cl)cnc1Cl 27344,C(=O)(C(CN=[N+]=[N-])NC(=O)C(C)NC(=O)Nc1cccs1)OCC 27345,C1(C(=O)NC2CC3CN(C(c4c(CC)sc(=N)[nH]4)=O)C2C3)CCC2(CCC2)CC1 27346,c1(OC)ccc(C(=O)NC2CC2NC(c2cc(C)cc(F)c2)=O)cc1C(C)C 27347,CC1(CNC(=O)CN2CC=CC2)CC(NC(c2ncsc2Br)=O)C1 27348,Cc1noc(C(C)C)c1C(=O)N(C)CC1(O)CCN(C(=O)CC(C)NC(N)=O)C1 27349,c1(C(=O)NC(C(C)NC(c2cc(N)cnc2Cl)=O)C)ccc(Cl)c2ccccc12 27350,C12(C(=O)OC)CCCC1CCN2CCn1cnnc1 27351,C1(CC(=O)Nc2c(C(C)C)c[nH]n2)CCN(C(=O)COC(C)(C)C)CC1 27352,CC1CN(C(=O)C2=CCCCC2)CC(CCNC(=O)CCc2ccn(C)c2)O1 27353,c1(C(=O)NC2CC2NC(c2noc3c2CCCC3)=O)ccc2cccnc2c1 27354,Cc1nn(Cc2ccccc2Cl)c(Cl)c1C(=O)OCC1C(C)(C)C1(F)F 27355,c1(NC)ccc(C(N2CCC(CC)C2C(N2CC(OC)C2(C)C)=O)=O)cc1 27356,C(=O)(CCCCC(=O)N1CC(O)(C(F)C(=O)N(C)C(C)C2CC2)C1)OC 27357,CC1(F)CCC(C(N2CCC(CNC(=O)C(F)(F)c3cncs3)C2)=O)CC1 27358,CC(C)C(CC(=O)NCC(C)CNC(c1cnc(C2CCC2)s1)=O)C(C)C 27359,CC#CCCCC(=O)NC1(CCO)CN(C(=O)C(C)SCCC(C)C)C1 27360,c1(CNC(C(C)O)=O)ccc2c(c1)CCN(C(c1coc(CO)c1)=O)C2 27361,C1(C)(CNC(C2(C)C(C)CCC2)=O)CCCN(C(c2ccc(F)s2)=O)C1 27362,C1(C(=O)NCC2N(C(c3cc(C)oc3)=O)CCC2C)CCc2nncn2C1 27363,N1(C(C=CCC(C)NC(C2(O)CCCCC2)=O)=O)CC(CO)CC12CCC2 27364,c1(OC)cccnc1C(=O)NC1(C)CC(NC(=O)CCC2CCCO2)C1 27365,c1(CC)c(C(=O)N(CC(C)NC(=O)CC2(O)CCCC2)CC)cnn1CC(C)C 27366,Cc1ccc(C(=O)NC2CC(CNC(=O)CS(C)(=O)=O)C(O)C2)c2c1CCCN2 27367,C(C)(C)(CC(=O)N1CCCC(C(=O)NC2(CO)CCC(C)C2)C1)OC 27368,C(=O)(C1=COCCO1)NCCC(C)(C)NC(CCC(=O)NCCCC(C)O)=O 27369,C(=O)(C(CO)NC(C1CCCN1CCC)=O)NCC=C 27370,c1(C(=O)NC2CCCC2c2nc(S)n[nH]2)cc(O)nc(C2CC2)n1 27371,C1(CC)CN(C(c2cc(C)oc2C)=O)CCC1NC(c1cnn(CC(F)F)c1)=O 27372,Cc1ncnc(C)c1C(=O)NCC12CC1CN(C(=O)C(=Cc1cccnc1)F)C2 27373,c1(NCC2(CNC(c3c(F)cccc3Cl)=O)CCCC2)ncnc2ccccc12 27374,c1(NC(C)=O)cccc(C(N2CC(O)(C(C)NC(C3CC34CCCC4)=O)C2)=O)n1 27375,Cc1cc(C)c(C(=O)NC(C)(C)CCCNC(=O)CCC2CCCC(O)C2)[nH]1 27376,CCCC(C)(C)C(=O)N1CCC(C)(NC(N2CCC(C)C2c2cccs2)=O)C1 27377,C1(C(=O)NCc2ccc(F)nc2F)CC12CCN(C(c1cc[nH]n1)=O)C2 27378,C#Cc1cccc(CNC(=O)C=C(C)CNC(=O)C(C)(C)C(N)=O)c1 27379,C#Cc1cn(C)nc1C(N1CC(NC(C2CC3CC(=O)C2O3)=O)CC(O)C1)=O 27380,C(=O)(CCC(C)(C)N(C)C)NC1(CCNC(C=C2CCC(C)C2)=O)CC1 27381,C1(C(=O)NCCNC(c2c(OCC)oc(C)n2)=O)CC1C1CC(F)(F)C1 27382,c1(SCCC(=O)NC2CC(C)(NC(C(CCN(C)C)O)=O)C2)cc(F)ccc1F 27383,C1(CC#C)CC(=O)N1.C1(n2cc(-c3ccc(F)cc3)nn2)(CC#C)CCOCC1 27384,C(=O)(CC(O)CCSC)N1CCC(N(C(=O)C(C)C(F)F)CCOC)CC1 27385,Cc1ccccc1C(C)C(=O)NC(C)CN=[N+]=[N-] 27386,Cc1cc(C)c(C(=O)NC2(CNC(C3(CF)CC3(F)F)=O)CCC2)s1 27387,c1(OC)ncccc1-c1cn(C(C)CNC(c2nc[nH]c2C(C)(C)C)=O)nn1 27388,c1(C(=O)NCC#CCC(=O)NCCC(COC)O)ccc2c(c1)CCC2 27389,C1(C(N2CC(COC)(NC(=O)C=C(C)C3CC3)C2)=O)CCCC(O)C1 27390,c1(C(N(C2C(N(C(C=C(COC)C)=O)C)CCCC2)C)=O)cnc2sccn12 27391,N1(CC#CC)CCN(C(=O)C(c2ccoc2)NC(=O)C(N2CCOC2=O)C)CC1 27392,CC(C)C(C(=O)N(C1CCOC(C)C1)C)C(C)NC(c1cc([N+](=O)[O-])n[nH]1)=O 27393,C1(C(=O)NC2CC3CC(NC(C4=CC(C)(C)C4)=O)CC32)COc2ccccc2O1 27394,C(=O)(C(C)CC(N)=O)NCc1cn(CC2N(C(CSCCOC)=O)CC=C2)nn1 27395,C(=O)(C(C)CN(C(=O)CC1CNC(=O)O1)C)NC1CC(CSC)C1 27396,N1(C(Cc2ncn(C)c2)=O)CCOC(C(=O)NC2CC3CC4C(C3)C24)CC1 27397,C1(CC(N2CCC(CC=C)C2)=O)CN(C(c2cc(O)n(C)n2)=O)CC1C 27398,Cc1c(C(=O)NCC(C(C)C)NC(=O)COC(F)F)cnn1CCC(C)C 27399,CC(C)CCC(F)C(=O)NC1CC2CC1N(C(c1cnc3n1CCCC3)=O)C2 27400,c1(C(N(CC(C)(C)CNC(C2(CC)CCCC2)=O)CC)=O)cc(C)cc(O)c1 27401,c1(CC(=O)NCCCC(C)NC(=O)CC2CCN(C)C2)ccc(N)cn1 27402,N1(C(c2cn(CC=C)nc2)=O)CC(NC(c2onc(CC)c2C)=O)CC1CO 27403,C=CC(C)C(C)C(=O)NCCCN(C)C(c1cncc(C#N)c1)=O 27404,C1(C)(CNC(C(C=CCCC)O)=O)COCCN(C(c2ccccc2O)=O)C1 27405,CC1(C(=O)NCCn2cnnn2)CC(O)CN1C(=O)Cc1ccon1 27406,Cc1cccc2nc(NC(C3CCN(c4cccc(Br)n4)C3)=O)[nH]c12 27407,c1(CC(=O)NCCC2CCCCN2C(=O)C=C2CCC2)n[nH]c2ccccc12 27408,c1(OC)ccc2ccccc2c1CNC12CC(NC(c3c[nH]nc3C)=O)(C1)C2 27409,C1(C)(CNC(c2ccc(C#C)cn2)=O)CC(F)(F)CN1C(C1COC(=O)O1)=O 27410,c1(OC(C)C)ncccc1CN1CC2CC2(C(=O)N(C)Cc2ccccc2Br)C1 27411,C1(N(C)C(C2(C3CC3)CCCO2)=O)CCN(C(c2ccc(CO)nc2)=O)CC1 27412,C1(N(C(=O)CC2CCCC2)CC)CCCN(C(c2oncc2CC)=O)C1 27413,N1(C(C(C)O)=O)CCC(C(=O)NC2CCC(C3CC3)C2)C(C)(C)C1 27414,C(C)(C)(CCC(=O)Nc1ccccc1O)NC(CCC1N(C)CCC1)=O 27415,N#Cc1ccc(S(N)(=O)=O)c(N2CC3CC2CC3O)c1 27416,C1(O)(CNC(C2(C(=O)OCC)CC2)=O)CCN(C(=O)C(N2CCC(O)CC2)C)C1 27417,n1(CC)cnc(C(=O)NCC(C)(CO)NC(=O)CNC(C2CCC2)=O)n1 27418,C(C1CCCCCC1)=CC(N1C(CNC(c2c(C)noc2C(F)F)=O)CCC1)=O 27419,C1(O)(CNC(CCCN(C)C)=O)CCCN(C(=O)CC2CCC(C)(C)CO2)C1 27420,N1(C(C(C)N(CCC)C(c2ccc(OC)o2)=O)=O)CCSCC1CO 27421,CC1CN(C(c2cncc(-c3ccc(Cl)cc3)c2)=O)C2(COC2)CO1 27422,c1(CC)cccc(OCC(=O)N(CCNC(=O)CCC2CCC(C)O2)C(C)C)c1 27423,CC1(C)COC(C(=O)NC2CCC(CC(N3CCOCC3CO)=O)C2)C1 27424,C1(NC(C(C)CC2CCCCC2)=O)CCN(C(=O)CCc2nncn2C)CC1C 27425,c1(C(=O)NC(CNC(c2[nH]cc3c2CCC3)=O)CO)ccc2c(c1O)CCC2 27426,C=CCC(CC=C)C(=O)N1CCC(NC(C23CC(C#N)(C2)C3)=O)CC1C 27427,CC(C)C(CCN(C(=O)CCC1(NC(=O)CNC(N)=O)CCCC1)C)N(C)C 27428,N1(C(C2CC(SC)C2)=O)CCN(C(c2ccnn2C2CCOCC2)=O)CC1 27429,N1(C(C2CCC(=O)OCC2)=O)CC2(CCCN(C(C3CN4CCC3CC4)=O)C2)C1 27430,N1(C(COC2(C)CCC2)=O)CCOC(C(C)NC(c2ccc(C(N)=O)[nH]2)=O)C1 27431,C1(C)(C(=O)NCc2cn(C(CC)C)nn2)CCC2CC2C1 27432,C1(NC(c2cc(COC)no2)=O)CCN(C(=O)C(F)(F)C(F)(F)F)CC12CCC2 27433,c1(CC(=O)NC2CC(F)(CNC(c3cn[nH]c3)=O)C2)cccc2ccccc12 27434,Cn1nc(CNCc2cc(Br)cnc2Br)c2c1CNCC2 27435,C(=O)(C1CCCn2cnnc21)NCC1C2(CC(NC(CSCC(C)C)=O)C2)C1 27436,C(=O)(C(O)C(C)(C)CC)NCCCOCCC(NOCCC(=C)C)=O 27437,C(CCCC(=O)OCCOc1ccccc1)NC(c1ccc(CC)s1)=O 27438,CC(C(=O)NC1COCCN(C(C2CN3CCCC2C3)=O)C1)S(C)(=O)=O 27439,C(CC(=O)NC(c1ccccc1C)C)(C(F)(F)F)NC(CC(C=C)C)=O 27440,CC1(C(=O)NCC2(NC(=O)CCNC(=O)CC3CCCCC3)CC2)CNC(=O)C1 27441,C1(CC=C)(C(=O)NCC(C)N(C)C(C2CCCN2CC(C)C)=O)CCCCC1 27442,c1(C(N2C(CNC(CC(CC)C3CC3)=O)CCC2)=O)ccc(OC)c2ccsc12 27443,c1(C(N2CC(COCC)(NC(C3CCCC(C)C3)=O)C2)=O)ccc(C)cc1F 27444,C1(CC(=O)NCc2c(C)non2)CCCN(C(C2SCCS2)=O)CC1 27445,N1(C(Cc2n[nH]c(=N)s2)=O)CC2CC1CCC2NC(c1cncc(C2CC2)c1)=O 27446,c1(OC)ccc(O)cc1C(=O)NCC(C)CNC(=O)CC(C)=C(C)C 27447,c1(NCC(C2CCCC2)NC(c2ccn(C)n2)=O)ncc2c(ncn2C)n1 27448,c1(N2CCN(C)C(CNC(c3cccc(C(F)F)n3)=O)C2)ncc(C#N)cc1F 27449,c1(CC)ccsc1C(=O)NCC=CC(=O)N(C1CCSC1)CC 27450,c1(CN(CCCO)C(=O)Nc2cc(-n3cccc3)ccn2)ccc(Cl)cc1 27451,c1(C(N2CC(CC(=O)Nc3cnc(Cl)nc3)OCC2)=O)cnn2ccccc12 27452,C1(CC(=O)OCC)COCCN1C(=O)COCC.N12CCN(CC1)C(=O)C2 27453,C(=O)(C#CC1CCCC1)N1CCN(C)C(C(N2CCC(F)(CF)C2)=O)C1 27454,C1(c2ccc3c(c2)OCCO3)CCCN(N2CCC23CCCCC3)C1 27455,N1(C(c2[nH]cc(CC(C)C)c2)=O)CC2CCCC2(CNC(=O)CCCC#N)C1 27456,Cc1[nH]c(C)c(C(=O)NCC(C)(C)CNC(=O)CCOCC(C)C)c1C 27457,c1(OC)ccc(CCC(=O)NC2CC(C)(NC(C3CCCC3(C)C)=O)C2)cc1F 27458,C1(NC(C(CC)SC)=O)CC1C1CCCN(C(=O)C(=O)C(F)(F)F)C1 27459,C(=O)(C(C)CCCC(C)=O)NCCn1cc(C(=O)NCC(C(F)(F)F)OC)nn1 27460,N1(C(CNC(CNC(c2ccc(C)cc2)=O)=O)=O)CCC2C(C(N)=O)C2C1 27461,Cc1cc(C(N2CCC(C)(NC(c3cc(F)c(Cl)cc3Cl)=O)C2)=O)cc(F)c1C 27462,c1(C(=O)NCCCN(C(c2nc(Cl)cs2)=O)CC)ccnc(C(C)(F)F)c1 27463,CC1(CF)CN(C(C2(C3CCCN3C(c3cnccn3)=O)CC2)=O)C1 27464,C(CCC(O)C(=O)NC(C)C(=O)NCC(C)C)NC(C(C=C)CC)=O 27465,N1(C(CC(COC)C)=O)CC2CCN(C(c3cnn4c3OCC4)=O)CCC2C1 27466,CC1OC2(CNC(C3C(C)OC(C)C3C)=O)CC1(NC(C1CCCOCC1)=O)C2 27467,CCCCCCC(C)NC(=O)C1=CCN(C(=O)CCC2CC2)C1 27468,S(=O)(=O)(c1ccc(N2CCn3ncc(Cl)c3C2)nc1)N1CC(C)C(C)C1 27469,Cc1ccc(C(N2CCSCC2C(N2CCC(OCC(C)C)C2)=O)=O)nc1O 27470,C(=O)(CCCS(C)(=O)=O)N(C)CC1(CNC(=O)CCCC2CCCC(=O)N2)CC1 27471,C1(C(=O)NCC2C(C)C2C)CCN(C(c2ncccc2Cl)=O)C1(C)C 27472,c1(C(N2CCOCC(C(N(CCC(=O)NC)CC)=O)C2)=O)cccc2ccoc12 27473,C1(CC(=O)N(CC(O)CNC(=O)C=Cc2cccs2)C)CCC(F)(F)CC1 27474,c1(NC(C(=O)NC(c2c(C)cccc2C)C)=O)ccc2c(c1)CCC2 27475,c1(C(N2CCC(N(C(=O)CC3C=CCC3)CCC)C2)=O)ncc(OC)nc1OC 27476,C1(NC(CNC(N)=O)=O)(CNC(c2ccn(C3CCCCC3)n2)=O)CCOC1 27477,CCCCC(CC)C(=O)NC1(CC(=O)NC2CCOC2C2CC2)CCC1 27478,c1(CN(c2nccc(N(C)CC3C(C)C3)n2)C)ccc(Br)cc1[N+](=O)[O-] 27479,CC1(C)OCCC1C(=O)NCCn1ccc(C(N2CCC3CC23)=O)c1 27480,C1(NC(C=CC)=O)CC=C(C(=O)NCc2cnc(CC)[nH]2)C1 27481,C(=O)(CC(C)(C)C(=O)N(CCCNC(=O)C(C)CSC)C(C)C)OC 27482,c1(C(=O)OC)cc(Br)cc(I)c1NC(=O)CCc1cccc(Cl)c1 27483,C(CCCC)(CN=c1[nH]c(Cl)ncc1C1CC1)NC(C=CC(=O)NCCCC)=O 27484,c1(CCC(c2n(CCOCC)nnn2)NC2CC(C)(C)C2)cccc(Br)c1 27485,C1(NC(CN(C)CC)=O)CC(NC(c2cc(C(C)C)ccc2C)=O)C12CCC2 27486,c1(C(=O)NC(CCNC(CN(C(C)C)C)=O)C)ccc2c(=O)ccoc2c1 27487,C(=O)(C(C)CC(C)C)N1CCC(C)(CC(=O)NCCNC(=O)OCC)C1 27488,Cc1c(NC(c2oc(CNC(=O)CC3CCC(C)C3)nc2C)=O)cnn1C(C)C 27489,c1(C(C(F)F)NC(=O)Nc2cn(C(C)(C)C)nc2)ccc(F)cc1F 27490,C(=O)(CN=c1cc[nH]cc1)NC1C(CNC(=O)CCC(=O)c2cccc(Cl)c2)C1 27491,C1(C(N(CCC(=O)NC)C)=O)(CC)CCCN1C(c1ncn(C(C)C)n1)=O 27492,N1(C(c2cc(=O)n(-c3ccc(Cl)cc3)[nH]2)=O)CCn2cncc2C1 27493,c1(N2CC(O)(C(C)NC(c3ccncn3)=O)C2)nc2c(F)cccc2o1 27494,C1(NC(CCc2cnn(C)n2)=O)CN(C(=O)C=C(Cl)Cl)CC1N=[N+]=[N-] 27495,Cc1cc(Cl)c(CN2CCCC2CC(N2CCC(C)(O)CC2)=O)c(Cl)c1 27496,C1(CC(=O)NCC(C(C)C)OC)CCN(C(=O)CC2CCCC2)CC1 27497,c1(OCCC(=O)N(CCN=[N+]=[N-])CCOC)ccc(C)cc1Br 27498,C1(CNC(C(c2cn(C)nc2)=O)=O)CCCCCN1C(c1ccsc1Cl)=O 27499,c1(CNC(C=CCC2(NC(c3n(C)ncn3)=O)CCC2)=O)cc(=O)cc[nH]1 27500,CC1(C)CN(C(C2(CNC(c3ccc(=N)[nH]n3)=O)CC=CC2)=O)CCC1O 27501,c1(C(N2CC3C(NC(C4C(CCC)C4)=O)(CC3)C2)=O)cc(S(C)(=O)=O)co1 27502,N1(S(CCCC)(=O)=O)CCC(O)C(C(=O)NCC2CC(=O)N(CCC)C2)C1 27503,CCC(C)(CC)C(=O)NCCNC(C1CN(C(C23CCC(C2)OC3C)=O)C1)=O 27504,c1(C(N(C2CCN(C(C34C(=O)C5CC3C4C5)=O)C2)CC)=O)cc(=O)n(C)cn1 27505,CC(C)C(CNC(=O)COCc1ccccc1)NC(=O)CCc1cc(Cl)no1 27506,c1(OC)cc(C(N2CCC(CNC(c3ccc(CF)cc3)=O)C2)=O)cc(F)n1 27507,C(=O)(C1=C(Cl)CCCC1)NC(C(=O)NCCC(C)N1CCC1)CO 27508,CCCC(CC)CCC(=O)NC1C=CC(C(N2CCC(O)C2C)=O)C1 27509,C1(C(=O)NCC2(O)CC(CO)C2)(COC)C=CCN1C(=O)CC1COCCOC1 27510,CCC(CC(=O)NC1CCC(NC(c2cc(F)cc(Cl)c2)=O)CC1)C(F)F 27511,N(C1COc2ccccc21)C(CC1CCN(C(c2cnc(C)n2C)=O)C1)=O 27512,CCCC(C(=O)NC(C(=O)NOCCN1CCCC1=O)C1(O)CCC1)C(C)C 27513,Nc1c(C(=O)NC2CC(NC(C3(F)CCC3)=O)C2)cc(Cl)cc1F 27514,c1(CC(C)(CO)N(CC(O)C2CNC2)C)cccc(Br)c1 27515,C#Cc1cc(C(=O)NCCC(C)NC(c2csc(C#N)c2)=O)cc(C(F)(F)F)c1 27516,C12(C(=O)O)CCC(C(=O)NCC3=CCSC3)(C1)OC2 27517,N1(C(c2cc(COC)cn2C)=O)CCN(C(=O)CN2CCSCC2)CC1CF 27518,c1(OC)[nH]c(=NC(=O)C2CC(F)CN2C(=O)C(Cl)(Cl)Cl)cc2cccnc12 27519,C1(N(C(c2c(OC)csc2)=O)C)CCCC2CN(C(C3CCN(C)C3=O)=O)CC12 27520,C1(CC=C)(NC(COCC=C)=O)CN(C(=O)Cc2cc(-c3ccccc3)on2)C1 27521,c1(C(=O)NCC(CNC(=O)CC2(O)CCOC2)O)ccc2ccccc2n1 27522,C1(CNC(CC(C)OC)=O)CC2(CCC2)CN1C(C1CN(CC(F)(F)F)C1)=O 27523,C1(C(N(CCCNC(C2C(C)C2C)=O)CC2CCCC2)=O)C(F)(F)C12CCC2 27524,c1(C(=O)NCCC2N(C(C(C)CCO)=O)CCCC2)c([N+](=O)[O-])cnn1C 27525,CC1CCC(C)(C(=O)NCCCOCCNC(=O)CCc2cc(Cl)no2)C1 27526,C1(C(=O)NC2COCCN(C(=O)Cc3ccoc3)C2)CC2(C1)CC(F)(F)C2 27527,CC1(C)CN(C(C2CCCOC2)=O)CC(C)(C)C1NC(C1CC(C(F)F)C1)=O 27528,c1(CC)ccc(CC(N2CC(N(C(=O)CC34CCCN3CCC4)C)C2)=O)cc1F 27529,C1(C(N2CCC(OCC)C2)=O)CC2(CC2)CN1C(=O)CC1CCC=CCC1 27530,C1(NC(C=CSC)=O)CCCCC12CCCN(c1cccc(SC)c1[N+](=O)[O-])C2 27531,CCC(CO)C(=O)N1CCC(N2CC(C)(CNC(=O)C3=NOCC3)C2=O)CC1 27532,C#CC(C)(C)C(=O)NCCCC1CN(C(c2ccc(CC(N)=O)cc2)=O)CCO1 27533,c1(C(N2CCOCC(NC(=O)CCOCC(F)F)C2)=O)cccc2[nH]ccc12 27534,c1(OCC)cc(C(=O)NCC2(C)CN(C(=O)C=CCN(C)C)CCO2)cc(F)c1 27535,c1(C(=O)NC(CNC(C(C2CC2)SC)=O)CO)cc(C(F)(F)F)cc(Cl)c1 27536,c1(C(=O)NCC(CNC(C(C=C=C)C)=O)(C)C)cnc2c(cnn2C(C)C)c1 27537,c1(C2(C(=O)NC3CCOC3)CC(NCCCCCC)C2)c[nH]c2cc(F)ccc12 27538,Cc1cc(C(=O)NC2CCC(C(=O)NCC34CCC(C3)C4)C2)c(C)o1 27539,Cc1nc2c(o1)CCCC2CC(=O)N1CC2CCC1CN2C(=O)Cn1cncn1 27540,C1(C(N2CCCC(C)(CC)C2)=O)CCCCCCN1C(c1cncc(OC)n1)=O 27541,C(=O)(CCCC(F)(F)F)N(CC(CC)NC(C1(C)CCC(O)CC1)=O)C 27542,CC(CC(=O)NCCN(CCCN(C)C)C(=O)CC1CCC2CC12)C(F)(F)F 27543,C1(CNC(C2(C#C)CC2)=O)CCCC2(CN(C(=O)C(C)(C)C(C)(F)F)C2)O1 27544,C1(CCC)CN(C(C2CC=CCO2)=O)CCN1C(=O)CC1CCCCCCC1 27545,c1(NCc2cccc(C)n2)cnc(Cl)cc1C(=O)N(CCC#N)CC1CC1 27546,CC1CC(C)N(C(c2c[nH]nc2F)=O)CCN1C(c1cncc([N+](=O)[O-])c1)=O 27547,C1(C(=O)NC(C)C(=O)NCC#CCNC(=O)CC23CCCC2C3)CCCCC1 27548,c1(C(=O)NCC(C)N(C(=O)COc2ccsn2)C)scc2c1CCCC2 27549,C1(NC(Cn2c(C)ccc2C)=O)CC(C(N2CC(CC(C)C)C2)=O)C12CCC2 27550,N1(C(C(CSC)OC)=O)CCN(C(=O)C(C(C)(C)C)c2cccc(C)c2)CC1C 27551,N1(C(C2C(CCC)CN(C(=O)C(C)C(O)C(C)C)C2)=O)CCc2oc(C)nc2C1 27552,N1(CCNC(=O)N(C2CCC2)CC2(c3ccco3)CC2)CCn2cnnc2C1 27553,C12(CNC(CCCC(=C)C)=O)CCC(CC1)N(C(c1ncc([N+](=O)[O-])n1C)=O)C2 27554,N1(C(C(C2CCN(C(c3c(CC)c[nH]c3)=O)C2)F)=O)CC=CC1(C)C(=O)OC 27555,C(=O)(CCCCN=[N+]=[N-])N1CCCC(N(C(c2c(CC)nn[nH]2)=O)CC2CC2)C1 27556,C(=O)(C(O)CC(=O)OC(C)(C)C)NC1(C)CN(C(C(CCC)C)=O)C1 27557,N1(C(C2C(C)CCCC2)=O)CCCCC(CNC(c2cccc(F)c2N)=O)C1 27558,Cc1cccc(F)c1CC(=O)NC1CC2(C1)CC(NC(=O)C(C)C1CCC1)C2 27559,Cc1nc(C(=O)NCC(C)(O)CNC(=O)Cc2nc(=N)[nH][nH]2)c(C)n1C1CC1 27560,CC(CC(=O)NC1CC(F)(CNC(=O)Cc2c[nH]nc2O)C1)P(C)(C)=O 27561,C(=O)(C(C)(C)CCCF)N1CCCC(N(C(C(c2ccc(C)cc2)C)=O)C)C1 27562,C(C(C(=O)OC)NC(=O)CC(C)NC(=O)CCN1CCOC1=O)OC 27563,C(CCCCC(=O)NCC(c1ccc(F)cc1)NC(c1cccn1CC)=O)=CC 27564,CC(C)CC(C(=O)NC1(C(O)CO)CC1)NC(c1nnc(O)nc1O)=O 27565,Cc1nn2cccnc2c1C(=O)NCC12CC1CN(C(C1CCS(=O)CC1)=O)C2 27566,c1(C(C)C)c(NC(=O)NCC2CC2C(=O)OC(C)(C)C)cccc1Br 27567,C(=O)(CCCCC(C)CC)NC(CC(=O)NCC1(OCC)CC1)CC 27568,C1(NC(c2cc(C)oc2)=O)CCC(C)(C)CC1CNC(=O)CSc1ccncc1 27569,Cc1cc(O)cc(=O)n1CC(=O)NCC1(F)CC(NC(=O)C(CN(C)C)N(C)C)C1 27570,c1(C(N2CCC(NC(C(C(CC)O)(F)F)=O)C(O)C2)=O)cc(S(N)(=O)=O)oc1C 27571,C1(C(=O)NC2C=CC(C(=O)NCC(=O)OCCCC)C2)COCCN1CC 27572,Cc1cnc(Cl)cc1NC(C1CCCN(C(c2cccnc2C)=O)C1)=O 27573,c1(OC)ccc(F)c(C(=O)NC2CCC(C)N(Cc3cc(Cl)ccc3F)C2)c1F 27574,N1(C(COCCN(C)C)=O)CCN(C(c2cccc(N)c2O)=O)CC(C)(C)C1 27575,c1(OC(C)(C)C(=O)NC2CC(CNC(=O)C3=NOCC3)C2)cccc(N)c1 27576,c1(C(N2CCCCC(NC(c3c(C)c[nH]n3)=O)C2)=O)cccc2nc[nH]c12 27577,c1(C(N(C)CC2CCCN(C(C(C3CCC3)OCC)=O)C2)=O)ncnc(O)c1F 27578,N1(C(C2N(C(C)=O)CSC2)=O)CCCCC(CNC(c2nc(C)nn2C)=O)CC1 27579,c1(NCC2(CO)CCCCC2)nc(N2CCCC(F)C2)nc2ccsc12 27580,c1(-n2c(C3CCCCN3C(=O)C(C)C)nc(COC)n2)cccc2ncccc12 27581,C(=O)(C(N)CCC(=O)Nc1cnc2n[nH]c(Br)c2c1)OC 27582,c1(OC)ccc(C(=O)N(CC(C)N(C(=O)Cc2ccoc2C)C)C)nc1 27583,C1(C(=O)NCC(C)S(N)(=O)=O)C(C)OCCN1C(=O)CC1CCOC1(C)C 27584,Cc1nc(NCC2CN(C(C3C=CCC3)=O)CCC2C)ncc1Br 27585,N1(C(COCCCOC)=O)CCCC(NC(c2cc(CO)on2)=O)C1C 27586,C(=O)(C(F)C(C)CNC(C1C=C(C)CS1)=O)NC(C(=O)OC)C 27587,CC1CN(C(c2ccc(-c3ccncc3)s2)=O)CC(C)C1NC(c1cc[nH]c1)=O 27588,C1(CC)NC(=O)N(CC(=O)Nc2cc(C3CCCCC3)no2)C1=O 27589,Cn1c(C(=O)NC2(CNC(=O)CS(N)(=O)=O)CC(F)(F)C2)cc2sccc12 27590,c1(C(=O)NCC2(F)CN(C(=O)C(F)F)C2)c(C(F)(F)F)cncc1F 27591,C(CC(C)N=c1[nH]c2cc(Cl)ccc2s1)NC(CCOc1ccc(C)cc1C)=O 27592,C1(C(=O)NC2(CC=C)CN(C(C3CCS3(=O)=O)=O)C2)CCCCC1O 27593,N1(C(CCN(CCCCC)C)=O)CCC2CCN(C(C3(C#N)CC3)=O)CC2C1 27594,c1(C(C)C)nc2ccc(NS(=O)(=O)c3cc(Cl)sc3Cl)cc2[nH]1 27595,C1(C(=O)Nc2c(C)n(C)nc2)CC(F)CN(C(C2CCCCN2C)=O)C1 27596,c1(C(N(C)CC2(O)CN(C(c3c(C)nc[nH]3)=O)C2)=O)[nH]c(C)c(S(N)(=O)=O)c1C 27597,C1(N(C(C(C)CO)=O)C)CC2CCC(C1)N2C(=O)CC1=NNC(=O)C1 27598,C12(NC(=O)CCC3CCC3)CCN(C(c3cc(CC4CCC4)c[nH]3)=O)CCC1C2 27599,Cc1c(Br)ccc(F)c1C(c1ccccc1)NC(=O)C(=O)NCC1=CCCC1 27600,c1(C(N2CCC(C)(O)C2)=O)cc(-c2ccco2)cc2[nH]ncc12 27601,C1(C(=O)NCC(CN(C)C(C2(F)CCCCC2)=O)(C)C)CC2C=CC1C2 27602,N1(C(C2(C)C(C)(C)C2)=O)CC2CCCC(NC(=O)CSCc3cccs3)C2C1 27603,c1(NCCSCC)nc(N2CCN(CCN(C)C)CC2)nc2c1cnn2C 27604,C(=O)(C(C(C)CC1CCCC1)N1CCC(F)(C(=O)OC)C1)NCC 27605,n1(CC)ccc(C(=O)NCC2CN(C(c3ncc(F)cc3N)=O)CC2C)cc1=O 27606,c1(C(N2C(CNC(c3cc(O)cc(F)c3)=O)CC2)=O)ccc(=O)n2c1CCC2 27607,CC(C)C(CC(=O)NC1CCCC(NC(c2scnc2C(F)F)=O)CC1)C(C)C 27608,c1(OC(C)CN(C)C(C2(C)CC=CC2)=O)cccc(N)c1 27609,CC(F)(CNC(=O)NC1CCC1C(F)F)C(F)(F)F 27610,C1(NC2CC(Cc3ccc(OC(F)(F)F)cc3)C2)CCC2CC=CC12 27611,N1(C(CN2CCC(C)CC2)=O)CCCC(O)(CNC(=O)C(c2cncnc2)C)C1 27612,S(=O)(=O)(c1ccc([N+](=O)[O-])cc1OC)N1CC(C(=O)NC(CC)C)C(O)CC1 27613,N1(C(C(C)NC(=O)N(C)CCS(C)(=O)=O)=O)CCc2ccsc2C1 27614,N1(C(C=CC(=O)OCC)=O)CCC2(COC(CNC(c3ncccc3F)=O)C2)C1 27615,c1(C(=O)NC(CC=CC)C(=O)NC(CCOC)C(C)C)c[nH]c2nccc-2c1 27616,N1(C(c2c(C(C)C)cco2)=O)C(CNC(C2CC(C(C)C)C2)=O)CC2CCCC12 27617,c1(C)ccc(NC(=S)NN(CC(c2cccs2)O)C)cc1.N1CCCC1 27618,C12(C(=O)OC)CC(NCc3ccccc3)C1C2.C1CO1 27619,N1(C(c2c(SC(C)C)cccc2)=O)CCN(C(C2(C(F)(F)F)CC2)=O)CC12CC2 27620,c1(C(=O)NCc2cccnc2Br)n[nH]c2cc(C3=CCCCC3)ccc12 27621,C(C(=O)N(C)CC1CCCN1C(c1occ(C)c1C)=O)(C(C)C)N(CC)CC 27622,Cc1cccc(C(=O)NC2CCC(NC(C3CSCN3CC3CCC3)=O)C2)c1F 27623,Cc1nocc1C(=O)NCC(C1CCCC1)NC(=O)C(C)c1cccs1 27624,N1(C(CCSc2n(C)cnn2)=O)CCCC(CNC(=O)COC2CCOC2)C1 27625,N1(C(Cc2cc(CC)nn2C)=O)C2CCC1C(NC(=O)C(C)OCC(C)C)C2 27626,S(=O)(=O)(c1ccc(CCC(=O)O)cc1)N1CCC(C)CC1C(N)=O 27627,CCCCC(F)C(=O)N1CCCCC(C(=O)NCCc2ccc(C)c(C)c2)C1 27628,N1(C(C(=O)NCCC2CCCCC2(F)F)=O)CCc2ccc(Cl)c(F)c2C1 27629,N1(C(C=CC)=O)CC2CCCC2C1C(=O)N(CCC(C)C)C 27630,C1(NC(C(n2ncc(C)c2)C)=O)CCC(C)(NC(c2ccc(Cl)nc2N)=O)CC1 27631,C=CCCC(F)(F)C(=O)NC(CC)CCCC(=O)NCc1nccn1C 27632,c1(C(N2CC3C(NC(C4CCC(C)(CC)O4)=O)C3C2)=O)c(C)nn(C)c1F 27633,CC1CCC(CC(=O)Nc2nn(C)cc2Br)CC1C 27634,N1(C(CNC(=O)OC)=O)CC(CNC(=O)CC(C)C(F)F)C(F)(CO)C1 27635,C(=O)(C(O)CC(C)C)NC1(CCNC(C(c2ccc(CCCC)cc2)C)=O)CC1 27636,C1(CNC(c2ccc(SCC)nc2)=O)CC12CCN(C(C1CCOCC1)=O)CC2 27637,CCC(C)C(O)C(C)C(=O)NCC(C)(F)CNC(C1CCC(C2CC2)C1)=O 27638,C(C)(C(C(=O)N(C)CC1CCCC1)C(C)C)NC(c1snc(C)c1N)=O 27639,Cn1ncc(C#N)c1C(=O)NCc1ccnc(C(N2CCC(CO)C(O)C2)=O)c1 27640,C1(CC)CC(C(=O)NCC(C)N(C(=O)C(F)OC)C)CC(=O)N1 27641,NS(=O)(=O)c1csc(C(=O)NC2CCCN(C(C3CCSC3)=O)C2)c1 27642,c1(CC)cc(C)c(C(=O)NC(C)(CNC(=O)CC2CCCOCC2)C2CCC2)o1 27643,c1(C(=O)N)cc(CO)on1.C(CNCCSCC(=O)O)(C1CC1)OCC 27644,N1(C(C(CCC)OC)=O)CCN(C(c2cnc(O)o2)=O)CC(CO)C1 27645,c1(C(=O)NCCN(C(=O)NC2CCN(CC(C)C)C2)CC)cc(C(F)(F)F)c[nH]1 27646,c1(CC(N2CCC(NC(COC(CC)C)=O)C2)=O)ccc(F)cc1 27647,c1(OC)ccc(NC(C2(C)CCCN(Cc3cc(Br)co3)C2)=O)c(F)c1 27648,C1(CC)CCN(C(C)=O)C1C(=O)N(CCNC(c1scnc1C)=O)CC 27649,N1(C(c2c(SCC)cccn2)=O)CCN(C(=O)Cc2ncccc2C)CC12CC2 27650,c1(C(N2CC(CCC)C(C(=O)NC3CCSC3)C2)=O)ccc(=O)n(C)n1 27651,c1(SCC(=O)N(C(CCNC(C(C)OCC=C)=O)C)C)cccc(F)c1 27652,c1(C(=O)NCCC2N(C(C3CC=C(C)CC3)=O)CCOC2)cc(C)c(C)cc1C 27653,CCCC(C(=O)NC(C)(CNC(=O)C(N1CCOC1=O)C)C1CC1)OCC 27654,CC1CC(C(=O)NCC2(F)CCN(C(=O)CCC(=O)c3cccc(Cl)c3)C2)=NO1 27655,N1(C(C=COCC)=O)CC(C)CN(C(=O)COc2cccc([N+](=O)[O-])c2)C(C)C1 27656,c1(C(=O)NC2CN(C(Cc3cccc(C)c3)=O)CC2C(F)F)[nH]c(C)c(C)c1C 27657,C(=O)(C1=CCCCO1)C(=O)Cn1ccc(C(F)(F)F)n1.C(CN)(N(C)C=O)C1CC1 27658,Cc1cccc(CNC(=O)CC2CCN2C(=O)CSC(C)(C)C)c1F 27659,CC1CCN(C(c2cncc(O)c2)=O)CC1CNC(C1CCCC1)=O 27660,C(C(C(=O)N(C(C)C(C)(C)C)C)C(C)(C)C)NC(c1n(C=C)ncc1)=O 27661,C(=O)(C1=COCCC1)NCC1(NC(=O)Cc2ccccc2F)CC(O)C1 27662,CC1CN(C(c2nnn(C)c2N)=O)CCN1C(c1cccc(OC(F)F)n1)=O 27663,C(=O)(C1CCc2c(Cl)cccc21)NCC(CCCC)NC(=O)CS(=O)(=O)C1CC1 27664,C#Cc1cc(C(=O)NCC2(O)CC(NC(=O)CC3CCC3(C)C)C2)ccc1C 27665,N1(C(CCc2cnc(C)o2)=O)CC2CC1(c1cn(Cc3cnn[nH]3)nn1)C2 27666,N1(C(c2nc(CCC)oc2)=O)CC2(CCN2C(C2C(C#N)C2(C)C)=O)C1 27667,c1(CC(=O)NCC(CN(C)C(C2CC(C)(C)CO2)=O)O)ccc2[nH]ccc2c1 27668,C(=O)(C(F)CCC(C)C)N1CCC(NC(C2(CCC=C)CC2)=O)CC1CC 27669,c1(C(N2CCC2CC(=O)NCC2(C(=O)OC)COC2)=O)nc(C)c(C)s1 27670,N1(C(C(CCC)C#N)=O)CCCC(C)(C)C1C(=O)NCC1CC(SC)C1 27671,C1(C(=O)NCCOC2CCNCC2)CC(=O)N(C2CCCCCC2)C1 27672,N#CCCCC(=O)NCC1CCN(C(c2ccc(CN3CCCCC3)o2)=O)CC1 27673,Cc1cc(C)n(CCN(C(C2CN(C(=O)OC(C)(C)C)CCO2)=O)C(C)C)n1 27674,c1(C(N(CCNC(C2(CCCC)CCC2)=O)CCOC)=O)ccc2oncc2c1 27675,C12(CNC(c3cc(C)oc3)=O)CCC(CNC(=O)C=Cc3cnc[nH]3)(CC1)CO2 27676,N1(C(CC(COC)C)=O)CC2C3CCC(C2C1)N(C(c1cc(Br)co1)=O)C3 27677,c1(CNC(CCC=CC)=O)nc(CNC(=O)C(C)=C2CCCC2)cc(O)n1 27678,c1(S)cncc(OCCNC(=O)NCC(N2CCCC2)C2CC2)c1.C(C(F)(F)F)O 27679,N1(C(C23C(C)OC(CN)(C2)C3)=O)CCC2(C1)Oc1ccccc1O2 27680,c1(CC)c(C(=O)NCC2(OC(C)C)CC2)nnn1CC.C12(CCCCC1)C(=O)N2 27681,C1(C(=O)NC2C(NC(c3ccon3)=O)COC2)CC2(C1)CC(F)(F)C2 27682,c1(C(=O)NC2CCCCN(C(C3(COC)C=CCC3)=O)C2)cc(N)c(C)cc1C 27683,c1(SC(C)C)ccc(C(=O)NCCOC2CN(C(=O)C(C)SC(C)C)C2)cc1 27684,C12(C(=O)OC)CCC(CC1NC(c1cccc3[nH]nc(O)c13)=O)C2(C)C 27685,N(C1CCCn2ccnc21)C(C1CCN(C(c2cc(CC)ncc2)=O)C1C)=O 27686,C1(NC(c2cc(C#N)[nH]c2)=O)CC2CCC1(NC(=O)Cn1cc(Cl)cn1)C2 27687,CC(C)CC(CNC(=NCc1ccsc1C(F)(F)F)NCc1cncnc1)OC 27688,CCCC(O)C(=O)N1CC(CNC(=O)C(C)OCCC(C)C)C1 27689,C1(C)(COC)CC(NC(=O)CCC(C)(C)F)CN1C(=O)C=C(Cl)Cl 27690,c1(C(N2CCC(NC(c3c(CC)non3)=O)C2CC)=O)cc(S(N)(=O)=O)co1 27691,c1(NCC(C)(C)C2CCC2)[nH]c(=NCC2CCCSCC2)nc2scnc12 27692,N1(C(=O)NC(c2c(C)cccc2)C)CCCCC1(CO)CO 27693,C(=O)(CC(C(F)F)NC(=O)C(C)(C)CCSC)NCC1(CCC)CCC1 27694,C1(C(=O)OC)CCC1S(=O)(=O)N1CCCSCC1C1CC1 27695,Cc1ccc(Cl)cc1C(=O)NC1COCCC1NC(c1cnn(C)c1F)=O 27696,C12(NC(CCCCCN(C)C)=O)CCCC1N(C(C1CCC(=O)C1)=O)CC2 27697,Cc1cnc(C(=O)NC2CCCN(C(=O)C(C)OCCC(C)C)CC2)c(C)c1 27698,N1(CN(C(=O)CC(C)C)CC(=O)NOCC)CC(=O)NC(c2cn[nH]c2)C1.CC 27699,N1(C(C(C(C)C)SC)=O)Cc2ccnn2CC(NC(c2cc(C)cs2)=O)C1 27700,Cc1cc(C(N2CC(NC(c3cnn(C)c3N)=O)CC2C)=O)nc(O)n1 27701,C1(COC2CCC2)CC(N(C)C)C1.C12(CC1)CC(=O)N(SC)C2 27702,C1(NC(CCSC)=O)CS(=O)(=O)N(C)C12CCN(C(=O)C1=CCCC1C)CC2 27703,CC1CN(C(C2CCCCC(=O)N2)=O)CCN1C(C1(O)CC(C)(C)C1)=O 27704,C1(N(C(=O)CSSC(F)F)CC)CCN(C(C2CC2c2ccccc2)=O)C1 27705,C1(C(=O)NC(C2CCN(C(C(C)=CC3CC3)=O)C2)C)C2CCC1(C)C2(C)C 27706,N1(C(C=NOC)=O)CCOC(C(C)NC(c2csc(C(F)F)n2)=O)C1 27707,c1(C(=O)NCCCN(C(C2CC(C#N)C2)=O)C2CC2)ccc(-c2nc[nH]n2)cc1 27708,c1(C(=O)NC2C(NC(c3cc(C4CCOC4)[nH]n3)=O)COC2)cc(O)nc(O)n1 27709,c1(CC)ccc(C(=O)NC(Cn2ccnn2)C(=O)NC(C)(C)CN(C)C)cc1 27710,c1(C(N2CC(F)(c3cn(C4CCOCC4O)nn3)C2)=O)c(O)cccc1Br 27711,C1(NC(=O)CCCCc2cnc[nH]2)CC2CCC1N(C(c1ccc(=O)oc1)=O)C2 27712,C1(C(C(=O)OC)N(c2ccc(NC(=O)C3CC3)cc2)C2CC2)CC2C=CC1CC2 27713,N1(C(c2c(C)c3c([nH]2)c(F)ccc3)=O)CCC12CCOC(C)(C)C2 27714,Cc1nn(CC(N2CC(N(C)C(C3CC4(CCC4)CO3)=O)C2)=O)c2ncccc12 27715,N1(C(C(=O)NCCOC)=O)CC(NC(C2CC23CC(F)(F)C3)=O)CC(C)(C)C1 27716,C(C(C(=O)NCCc1cc(C)[nH]n1)C(C)(C)C)NC(C(CCOC)C)=O 27717,N1(C(=O)CCN2CCC(F)C2)CCC2C(CCN2C(c2cnc(O)s2)=O)C1 27718,C1(CNC(C(n2ccc(C)n2)C)=O)CC(NC(c2cnc(C(F)F)s2)=O)CC1O 27719,C12(NC(c3cc(C)c(F)cc3)=O)CCCC1N(C(c1cc(O)nn1C)=O)CCC2 27720,N1(C(CCNC(CC(C)C)=O)=O)CC(C(=O)NC2COCC2N(C)C)CC1(C)C 27721,CC(C)CC(CCO)CN=C(NCc1cccn1Cc1cccs1)NCC(F)F 27722,N1(C(c2cc(C)n(C)n2)C(=O)NCC)CC(OC)CC(OC(C)(C)C)C1 27723,N1(C(C(C)CF)=O)CC(C2CCN(C(=O)C(C3CC3)C3CC3)CC2)C1 27724,C(=O)(CC(C)CCC(=O)N1CCOCC1CCNC(c1ncc(C)cn1)=O)OC 27725,c1(C(N(CC(C)NC(C(CC=CC)C)=O)CC)=O)ccc2nc(C)nn2c1 27726,c1(CC)cc(C(N2CCC(C(C)NC(c3c[nH]ccc3=O)=O)C2)=O)nn1C 27727,c1(C(N2CCC3(NC(=O)C(F)=CC4CC4)C(C2)C3)=O)ccc2nnc(S)n2c1 27728,C(=O)(C#CC1CCOCC1)N1CCC(NC(C(C=CC)O)=O)C1 27729,c1(C(N2C3CN(Cc4cccc(N(C)C)c4)CC32)=O)cc(O)ccc1I 27730,C1(COC(c2ccc(Cl)nc2)=O)CC(=O)N(C(C2CCCCC2)=O)C1 27731,c1(NC(C(CC)(C)C)C)ccc(CCO)c([N+](=O)[O-])c1.C(C(O)COC)S 27732,n1(CC(=O)NC(CCNC(CC(C=C)CC)=O)C)ccc(=O)n(C)c1=O 27733,N1(C(c2cc(OC)n[nH]2)=O)CC(C(=O)NC23CC(F)(C2)C3)C2(CCC2)C1 27734,N1(C(COC)C)CCC(C)C(NC(C2CCCCC2c2ccccc2)=O)C1 27735,Cc1ccc(C(=O)NC(CC(N)=O)C2CCOCC2)nn1 27736,c1(C(=O)Nc2nc(SCC)nc(Cl)c2)cnc2[nH]cnc2c1 27737,N1(C(CC)=O)CCOCC(CNC(=O)CC2CCCN2C(C)=O)C1 27738,c1(OC)cc(OC)c(-c2c(C)n[nH]c2C)cc1CN1CC2COC(=O)C2C1 27739,C1(C(F)(F)F)CCNC(=O)C(C)N1.c1(C(=O)NC(C)(C)C)cccc(F)c1 27740,C1(C(=O)Nc2cnn(-c3ccc(OC(F)F)cc3)c2)CCCN(CC(F)F)C1 27741,C(=O)(C1COc2ccc(F)cc21)N1CC2(CCN(C(C(CC=C)CC)=O)C2)C1 27742,N1(CC(=O)N(C(CNC(C(c2cccnc2)C)=O)C)C)CCC(N(C)C)CC1 27743,C1(C(=O)NC2C3CCCOC23)COCCN(C(c2ccc(C3CC3)o2)=O)C1 27744,Cc1cc(C(=O)NCCCN(C(=O)C=C2CCCCC2)C(C)C)nnc1C 27745,C(=O)(C(F)(F)C1=CCOCC1)NCC(CO)NC(C1SCCCS1)=O 27746,C1(NC(CCOC(CC(C)C)C)=O)CCN(C(C2CCCC(C#N)C2)=O)C1(C)C 27747,c1(OC)ccc(C(=O)NC2(C)CCCN(C(C3(CCN(C)C)CC3)=O)C2)cc1Cl 27748,N1(C(CCSC)=O)CCN(C(=O)C2=CCCC2)C(C)C1 27749,N1(C(C2CC3C=CC2C3)=O)CCC2(CCC2)C(NC(C2(C3CCC3)CC2)=O)C1 27750,N1(C(C2N(C(C(CC)N(C)C)=O)CCC2CC)=O)CCC2C(O)CC12 27751,c1(C(=O)NCC2CCC(C(N3CC4(CCOC4)C3)=O)CC2)nccc2cc[nH]c12 27752,c1(C(=O)NCCC2CCCN(C(=O)Cc3cnoc3)C2)c[nH]c2cccc(Cl)c12 27753,C12(NC(c3ccc(CC)nc3)=O)CCCC(CN(C(C)=O)C1)C2 27754,CC(C)(C)CC(=O)N1CC(O)CC1C(=O)NC(Cc1ccco1)CO 27755,C(=O)(C(C)S(C)(=O)=O)N1C(C(C)NC(=O)C=Cc2cc(C(N)=O)co2)CCC1 27756,c1(C(N2C(CNC(=O)CSCC3CCCO3)CC2)=O)cnc2c(c1)CCOC2 27757,C(=O)(C(C)CC(C)(C)C)NCc1ccc(CN(C(c2onc(C)c2C)=O)C)cc1 27758,c1(CC(=O)NCCNC(C2(c3ccccc3)CC2)=O)cncc(F)c1 27759,C1(O)(CN(C)C(c2ccc(Cl)cn2)=O)CCN(C(C2CCC(CCO)CC2)=O)C1 27760,N1(c2ncnc3n[nH]c(C)c32)CCC2CC(NC(c3ccno3)=O)CCC2C1 27761,Cc1cncc(C(=O)NCC(O)CCNC(C2(c3ccccc3C)CC2)=O)c1 27762,c1(C(N2CC3CN(C(C(CC)(C)C)=O)CC3C2)=O)cccc2c1C(=O)OC2(C)C 27763,C1(C(=O)NC2CCCC(CC(=O)NCC3C(C)(C)COC3)C2)CCC2(CCC2)C1 27764,C(=O)(CC1=CCOCC1)N(CCCC(=O)NC1CCNC1=O)C 27765,C(CC)(C(=O)NCC(C)(C)CNC(=O)CC1(c2ccccc2)CCCO1)OCC 27766,c1(SC)cc(C(=O)NC(C)CN(C)C(C2(c3ccccc3)CCCC2)=O)c(C)o1 27767,N1(C(c2scc(C)n2)=O)CCC(F)(CNC(C2CC2(Cl)Cl)=O)CC1 27768,CC1CN(C(=O)CC2CCC(=O)NC2=O)CCN1C(C1(NC(N)=O)CC1)=O 27769,C=CCCC(C(=O)NCC)NC(=O)C=CCN(C(CCO)C(F)F)C 27770,c1(C(=O)NCCC2N(C(Cc3nnc(C)o3)=O)CCSC2)cnn2cnnc2c1 27771,c1(C(=O)NC(C(C)NC(C2CNC(=O)C2)=O)CO)cnc2nccn2c1 27772,c1(CN2CC(COC(c3ccc(F)cc3C(F)(F)F)=O)C2)cc(F)c(O)c(Cl)c1 27773,C12(NC(C3Cc4cscc4C3)=O)COCCC1CN(C(=O)CN1CCCC1=O)C2 27774,c1(C(=O)NCCN(C(=O)C(C)n2cccn2)CCC)cc2c(C)c(C)ccc2[nH]1 27775,c1(C(N2C3C(C(N4CCN(C)CC4)=O)C(C3)C2)=O)ccc2[nH][nH]c(=N)c2c1 27776,C1(NC(c2cc(C)[nH]n2)=O)CCCC(N(C(=O)C(F)=CC2CC2)C)C1 27777,C1(NC(c2noc(CC)c2C)=O)CN(C(c2c(C)noc2N)=O)CC1S(C)(=O)=O 27778,C(=O)(C1CSc2ccccc21)N1CCC(C(C)NC(c2ccnnc2Cl)=O)C1 27779,Cc1cc(NC(C2CCCN(C(=O)CCCF)CC2)=O)cc(Cl)c1 27780,c1(C(N2C(C(=O)NCCSCCC=C)CCC2)=O)cccc(=O)o1 27781,N1(C(CC)=O)Cc2n[nH]cc2C1C(=O)OC.c12cn(nn1)C1CCC(C1)C(=O)NC2 27782,N1(C(c2c(CCNC(C(CN(C)C)O)=O)n[nH]c2)=O)CC(C2CCCCC2)C1 27783,C1(CNC(C(C(C)C)n2cnnc2)=O)CC2COCC2N1C(=O)Cc1nncs1 27784,c1(CNC2CN(C(CC(C)(C)C)=O)C2)ccc(OC2CCCCO2)c(F)c1 27785,c1(CCC)c(C(=O)NC(C)CC(C)NC(c2ncn(C)n2)=O)nnn1CC 27786,C1(C(=O)NCC(C)C2CC2)(CNC(c2cc(CC)on2)=O)CCCCC1 27787,c12cc3n(n1)CC1(CCN(CC1)CC2=O)OC3.c1(CC(N)=O)nccc(O)n1 27788,C1(N(C(COC)=O)C)CCCN(C(C2CCCS2(=O)=O)=O)CC1 27789,c1(C(=O)NC2CN(C(C3(C)CC3(F)Cl)=O)C2)cccc(NC(N)=O)c1 27790,C1(CC(C)NC(c2cccnn2)=O)CCN(C(C2CNC(=O)C2)=O)CC1 27791,C(C)(C)(C=CC(=O)NC(C1CC1C(=O)NCCCn1cnnn1)C)SC 27792,C1(C(=O)NC2CC3CN(C(C=CC(=O)NC4CC4)=O)C2C3)CCn2nncc2C1 27793,C=C(CNC(C1(C2CC2)CN(C(C2CC2=C)=O)C1)=O)C1CCOCC1 27794,C1(C(=O)OCC)(NC(=O)NC2CC2(c2ccc(Br)cc2)C)CCOCC1 27795,N1(CC(=O)NC2CN(C(C(C)OCCC(C)C)=O)C(C)C2)CCc2ccccc21 27796,c1(C(C2C(Cl)(Cl)C2)NCCOCC2CCCC2)nnnn1CC1CCOCC1 27797,C1(C(N(CC#C)CCOC)=O)(NC(=O)Cc2ccccn2)CC1(C)C 27798,N1(C(c2n(C(C)C)ccn2)=O)CCN(C(C2CC3CCCCC23)=O)C(CO)C1 27799,C1(C(N(CC(N2CC=CC2)C)C)=O)CSCCN1C(=O)C(=O)NCC(F)F 27800,c1(C(=O)NCCN(CCC)C(c2scnc2Cl)=O)cn(CC)nn1 27801,N1(C(C(CCC)(C)CCC)=O)CCC2(CC1)CC(NC(C1CCSC1)=O)CCO2 27802,C(=O)(C(CC=C)CC(C)C)NC(CC#C)CC(=O)NCC1(OC)CCCC1 27803,CC1(C)CC(CNC(=O)C=Cc2nccs2)N(C(=O)CCc2cnn[nH]2)C1 27804,C1(NC(C2=NOC(C)C2)=O)CC1C1CCCN(C(C23CC(C2)C3)=O)C1 27805,N1(C(C2(OC)CCSC2)=O)CC(C)CN(C(c2cccc(=O)n2O)=O)C(C)C1 27806,N1(C(=O)CCC2CCOC2)CC2CC1CN2C(C1C2(CC2)C12CC2)=O 27807,c1(C(N2CCC(C)(NC(C(CC=C)C)=O)C2)=O)c(C)ccc2ncccc12 27808,C1(CNC(C2CC(NC(=O)Cc3cc(Cl)cs3)C2)=O)CCS(=O)(=O)CC1 27809,c1(C(N2CC3CC(NC(c4c(O)cc(C)nn4)=O)C3C2)=O)ccc(C#N)nc1C 27810,C1(CSC)CCCN1C(C1CCOC1CNC(=O)CCCC1CCC1)=O 27811,N1(C(c2c(OC)c(F)ccc2)=O)CCC2CN(C(=O)CCC(C)N(C)C)CC12 27812,c1(C(=O)NCc2ncoc2C2CC2)ccc(C(F)(F)F)c([N+](=O)[O-])c1 27813,C1(C2CCN(C(=O)C=CCO)CC2)(NC(c2c(N)cccc2[N+](=O)[O-])=O)CC1 27814,C(=O)(C1=C(Cl)CCC1)NC(C(=O)N(C)CCc1cccs1)CCF 27815,c1(OC)cc(F)c(F)cc1C(N1CC(c2ocnc2CNC(C2CC2F)=O)C1)=O 27816,N1(C(C(C(=O)OC)OC)=O)CC(F)(F)CC1CCNC(C1CCCN1C(C)C)=O 27817,C#CC1CN(C(=O)CC2C(CC)C2(F)F)CCN1C(c1cc(Cl)cs1)=O 27818,C1(C(=O)NC2(C(=O)NCC=C=C)CC2)CCNC1=O 27819,C(=O)(C(C)(C)C(C)O)NC.c12cccc(c1)-n1cc(nn1)C1CC21 27820,C(=O)(C(C(C)NC(c1cccn1C)=O)C(C)C)Nc1c(C)noc1 27821,c1(CNC(C2CNCCN2Cc2ccc(Br)c(Cl)n2)=O)ccc(O)c(O)c1O 27822,CN1C(=O)NC2(CCC(C(=O)Nc3ccsc3-c3ccncc3)CC2)C1=O 27823,C(=O)(C(CC)CC(F)(F)F)NCC(C1CC1)NC(c1c(C=C)cnn1C)=O 27824,c1(OC)ccc(C)nc1C(=O)NCC(c1ccccc1)NC(=O)C(C)C(C)(C)O 27825,c1(C(=O)NC2(CNC(=O)Cc3ccccn3)CC2)nc(O)[nH]c(=O)n1 27826,CC1CC(F)(F)CCN1C(=O)CC1CCC(NC(=O)C(C2CC2)C2CC2)C1 27827,c1(NCc2c(C)cccn2)ncc(S(=O)(=O)NCC2CC2C)cc1Cl 27828,CC1(C)CC(=O)OC1CNS(=O)(=O)Cc1cc(Cl)cc(Cl)c1 27829,Cc1ncnc(NC2CC(CNC(c3cnc(Cl)s3)=O)C2)c1Br 27830,C1(C(=O)NCC2(O)CC2)(CNC(=O)CC2CC3CC3C2)CC12CCC2 27831,Cc1[nH]c2ccccc2c1CC(=O)NCC1(O)CCN(C(=O)COC(F)F)CC1 27832,c1(C(=O)OC)c(F)cc(CNCCCc2cncnc2)cc1F 27833,c1(CCN(C(C)=O)C)nc(-c2cc(C3CCC3)on2)n(-c2cnc(C)s2)n1 27834,C1(CSCC(=O)NC(C)CC2CN(C(C3CC(F)C3)=O)C2)CCCCO1 27835,c1(C(N(CCOCCNC(C(C=CC)O)=O)C)=O)cc(OC)c(Br)s1 27836,C1(C(=O)NC2C(NC(C(=O)NCCNC(C)=O)=O)C2)CCC12CCC2 27837,Cc1[nH]nc(C(N2CCC(C(C)C(=O)NCC)C2)=O)c1C(=O)NC1CC(C#N)C1 27838,c1(CC)nn(C)c(CC(=O)NCCCC(C)NC(=O)C(C)C(F)(F)F)c1Cl 27839,Cc1cc(NC(=O)NCC2CCSC2(C)C)cc(C(F)(F)F)c1 27840,n1(CC(C)C)c(N2CCCC2C(C)C)nnc1CS(=O)(=O)Cc1ccccc1 27841,Cc1c(C(=O)NC2CCCC(NC(c3csc(Cl)n3)=O)C2)cc(O)cc1N 27842,CON1CCC(C(=O)NC2CCC(C)N(C(=O)CCc3ccc(Cl)s3)C2)CC1 27843,CCCC(C)C(=O)NC1CC(C)(NC(=O)CCc2ccccn2)C1 27844,C1(O)(C(=O)NCC2(O)CN(C(CCc3cnc(C)o3)=O)C2)CCCC(C)CC1 27845,c1(C(CNC(C2CCCC2)=O)NC(CCOC(C)C)=O)ccc(N(C)C)cc1 27846,C1(C(=O)NCCCCNC(C(C(=O)OC)C)=O)CCc2nc(C)ncc2C1 27847,C(=O)(C(F)(CNC(C1CCCOC1)=O)C(C)C)N1CCCN(C(C)C)CC1 27848,C1(O)(CN(C)C(c2cnns2)=O)CN(C(=O)CCN2CCC2)C1 27849,C1(C(=O)NC2CCC(NC(C(OC)OC)=O)CC2)CC(F)(F)CCC1(C)C 27850,N1(C(C(COCC)C)=O)CC(CC(=O)NCCn2cc(C)cn2)CC1(C)C 27851,c1(C(N(C2CCN(C(C(COC)(C)OC)=O)C2)CCO)=O)cncc(F)c1Cl 27852,c1(OC(CC)C)cc(C(=O)NC(C)CN(C(c2nocc2C)=O)CC)ccn1 27853,c1(C(N2CCCC(Cn3cc(C(COC)(C)O)nn3)C2)=O)cncc(F)c1Cl 27854,c1(CCCC(=O)NC23C(CN(C(CC(=C)C)=O)C2)C3)csc2ccccc12 27855,c1(N(C(C)(C)C(=O)NC(=O)CN2CCCC2=O)C(=O)OC(C)(C)C)ccc(Cl)nc1 27856,Cc1nc(CCNC(c2ccc(-n3cncn3)nc2)=O)cc(O)n1 27857,Cc1ccc(-c2cc(C(N3CCC(C(=O)OC4C=CCC4)CC3)=O)on2)cc1 27858,C(=O)(C#CC1CC1)NC(CC)CN(C(C1CCCN(CC)C1)=O)CC 27859,c1(OC)cnc(C(=O)NC(C)CNC(c2sccc2-n2ccnn2)=O)c(OC)n1 27860,c1(-c2cn(CC(CNC(c3ccc(CCC)[nH]3)=O)OC)nn2)c(F)cccc1F 27861,C#CCCC(C(=O)NC1(C)CN(C(=O)OCC)C1)NC(=O)CC1OCCCO1 27862,C(CC)(CC)(CCNC(=O)C(C)S(N)(=O)=O)NC(CCN(C(CC)CC)C)=O 27863,c1(C(=O)NCC(CN(C(C(C)C(F)(F)F)=O)C)O)cccc2c1N(C)C(=O)CO2 27864,O=C1NC(C(=O)NCC23CC2CN(C(=O)CN2CCCNC2=O)C3)CCO1 27865,CC(C)C#CC(=O)N(CC(C)NC(c1cnn(C(C)C)c1Cl)=O)C 27866,CC1(C)CN(C(=O)CCCNC(C2(C)CCC(=O)NC2)=O)CC1O 27867,C(CN=c1ccnc(C2CCCC2)[nH]1)(C(C)(C)C)NC(C1N(CC#C)CCC1)=O 27868,OC1CCCCC(NCc2ccccc2F)CCNC1 27869,N1(C(c2cn(CC)nc2)=O)CCCCC1CNC(C1CS(=O)(=O)C1)=O 27870,C1(C2CCN(c3ncnc4c3COC4)CC2)(NC(c2cccc(F)c2Cl)=O)CC1 27871,N1(C(COCC#C)=O)CCCC1CN(C(C1(C#C)CC1)=O)C1CC1 27872,CC1CCC(C)(C(N2CC3CC2(C(=O)NCC(O)CN(C)C)C3)=O)CC1 27873,c1(C(C(=O)NCCCOC)N(C2CCOC2)CC)cncc(OC)c1 27874,CC1(C)C(C(=O)NCC(C)(F)CNC(C2COCCO2)=O)CC1(F)F 27875,CC1=NC(C)(CNC(c2coc(C(C)NC(c3cnc(C)o3)=O)n2)=O)CS1 27876,C(=O)(CC(C(F)(F)F)n1cccn1)N(C1CCN(C(=O)C(C)(F)F)C1)C 27877,C(=O)(C(CC(=O)OC)N(C)C)NC(C(C)NC(C=CC=CCC)=O)(C)C.C1CC1 27878,c1(OC)cc(F)cnc1NC(C1CCN(Cc2ccc(C)s2)CC1)=O 27879,C1(NC(c2nnc(C(F)(F)F)s2)=O)CN(C(c2c[nH]cc2Br)=O)CCC12CCC2 27880,C1(C(=O)NC(CNC(C(CC=C)(F)F)=O)CCCC)CCC(S(N)(=O)=O)CC1 27881,n1(CC=C)cc(CNC(=O)C(F)CC2CN(C(=O)CSC(C)C)C2)nn1 27882,CCC(C)C(C(=O)NCc1cc(C)ncn1)NC(C1C2CCC(F)C12)=O 27883,c1(SC)ncc(C#N)c(N2CCN(c3ccnc(Br)n3)C3CC23)n1 27884,c1(C(N2CCCN(C(Cc3c(C)nsc3)=O)CC2C)=O)cccc2c1OCC2C 27885,N1(C(c2n(CC)ncn2)=O)CCCN(C(c2cc(C#N)oc2C)=O)CC1CO 27886,c1(C(N2CCC(N(C)C(C3CCCC3)=O)CC2)=O)cc(O)nc2ccccc12 27887,C(F)(C(=O)NN1CCCC1C(=O)NC(C1CCCOC1)(C)C)=C(C)C 27888,CCC(C)CCCCC(=O)NC(c1cn(-c2cc(OC)ccc2C)nn1)(C)C 27889,S(=O)(=O)(c1ccc(C(N2CCCCC2)C)cc1)NC1CCC(OC)C1 27890,N1(CC)CCC1C(=O)NC1(CC(=O)NC2(c3cc[nH]n3)CC2)CC1 27891,c1(C(=O)NC(C2N(C(C(C)=C3CCCC3)=O)CCC2)C)cn2c(n1)C(C)CCC2 27892,C1(NC(C2CC2c2ccncc2Cl)=O)CCCN(C(C2(F)CC=CC2)=O)CC1 27893,C=CCC(CNC(=O)COC(C)(C)CC)C(=O)NC(C)CN1CCCC1 27894,C1(CC(=O)NCCCN(C(=O)CSc2ccccc2)C)CCOC1(C)C.C1CS1 27895,c1(OC)ccc2c(c1)CCN2C(C1CCCC(c2nn[nH]n2)C1)=O 27896,C(CNC(=O)C(=O)NC(c1ccc(OC)c(F)c1)C)(CC(C)(C)C)OC 27897,Cc1nc2c([nH]1)CC(C(N1CCC3CN(C(=O)C(=O)NC4CC4)C3C1)=O)CC2 27898,Nc1cc(C(=O)NC2(CNC(C3CC34CCCOC4)=O)CC2)cc(F)c1 27899,CCS(=O)(=O)CC(=O)N1CC(CNC(c2cccc(-n3cccn3)n2)=O)C2CC12 27900,c1(C(=O)NCCOCCN(C(=O)Cc2ccoc2)C)c(Cl)ccc(F)c1N 27901,C1(C(N2CCC(O)(CNC(Cc3cnc(C)o3)=O)C2)=O)CC(C)(C)CN1C 27902,Cc1ccc(N(C(c2ccc(C(c3cc(Br)ccn3)=O)cc2)=O)CC2CC2)cc1 27903,C1(CNC(c2cn(CC)nc2)=O)C2CN(CC(=O)Nc3cncc(Cl)n3)CC12 27904,CCC(CC(=O)N1C2CCC1CC(CNC(=O)CCCS(N)(=O)=O)C2)C(C)C 27905,N1(C(C2(C)CCCC2)=O)CC2(CC(CC(N3CCOC(C#N)C3)=O)C2)C1 27906,N1(C(C(CC)n2ccnc2)=O)CCC2(CC1)CC2NC(c1cnc(COC)s1)=O 27907,CC(CS(C)=O)C(=O)NCCCCN1CCCN(C(=O)CCN(C)CCO)CC1 27908,c1(C(=O)NC2CC(CC(=O)N(CCCCCC)CC#C)C2)cccc(C)c1N 27909,C1(C)(C(=O)NC(C2(CN3CCCC3)CC2)C)CCCN1C(=O)CN1CCCCC1C 27910,N1(C(c2ccc(CNC(C(CCC=C)(C)C)=O)cn2)=O)CCc2c(O)noc2C1 27911,Cc1ccc(O)cc1C(=O)NC(C)C(c1ccccc1)NC(=O)CSC1CC1 27912,C(CC(C)(C)C(=O)NC(C1CN(C(C2CCC(C)CC2)=O)C1)C)SC 27913,C(C(=O)NCCc1c[nH]nc1O)(C(C)(C)O)NC(c1c(CC)n(C)cc1)=O 27914,C1(C(N(c2c(C)csc2)C)=O)CC12CC2(F)F 27915,C1(OC)CC(CNC(c2ncc(F)cn2)=O)N(C(c2cnc(C(C)(C)C)o2)=O)C1 27916,c1(C(N2CCCC(NC(CC(=C)C)=O)CC2)=O)c(F)ccc(O)c1F 27917,C1(C(=O)NC(C)C2CC2)CC12CCN(Cc1noc(C(F)(F)F)n1)CC2 27918,N1(C(C(CC)(C)OC)=O)Cc2cccc(CNC(c3ccn(C4CC4)n3)=O)c2C1 27919,C(CC(C)C(=O)NCCN(C(=O)C(c1cnn(C)c1)=O)CC)=CCC 27920,Cc1nc(O)nc(C)c1C(=O)NCCCCCCNC(c1cc[nH]c1)=O 27921,S1(=O)(=O)c2ccc(OC)c(c2OC)C(=O)N1.c1(N(CC)CC)ccccc1 27922,N1(C(c2ccn(COC)n2)=O)CCC(C)C(NC(=O)C(C)(O)C2CC2)C1 27923,C1(N(C(CCOCCC)=O)C)CN(C(=O)Cn2c(C)c(C)sc2=O)CC1(C)C 27924,C1(C(=O)NCc2cc(C(N)=O)no2)CCCN(C(C2CC3CC2CC3O)=O)CC1 27925,c1(CC)ccc(S(C)(=O)=O)cc1C(=O)NC1C2CC3CN(C(=O)C4CC4)C1C3C2 27926,c1(OCC(=O)NC(C2CCCN2C(=O)COc2ccon2)C)cc(F)cc(F)c1 27927,C1(OC)(NC2CCC(n3cc(CCC(C)(C)CO)nn3)CC2)CC(C)(C)C1 27928,c1(CNC(c2cccc(CN3CCCC3=O)c2)=O)ccc2c(c1F)OCCO2 27929,c1(N2CC(CNC(=O)CN3CCCNC3=O)OCC2)ncnc2scc(Br)c12 27930,N1(CC)CCC2(CCCCC2)CC1.C1(n2c3ccc(s3)c2=O)CCCCCCCC1 27931,C(=O)(CCCCc1ccccc1)N(C1CCN(C(C)Cc2cnccn2)C1)CCO 27932,c1(C(N(C2CN(C(c3cccn3C)=O)CC2F)C)=O)ccc2cc(F)ccc2n1 27933,N1(C(C2C(CC)OCC2)=O)CC2(CC(C(=O)NC(COC(C)=O)CO)C2)C1 27934,C1(OC(C)=O)(OCc2cc(F)ccc2Cl)CCC(C(F)F)CC1 27935,c1(NCC2CCC(NC(c3c(CC)nco3)=O)C2)ncccc1C#N 27936,C1(CC(=O)NCC(CNC(C2(CCO)CC2)=O)OC)CC2(C1)CC1(CCC1)C2 27937,Cc1nnc2n1CC(c1nc(C3CC=CCC3)nn1-c1nccn1C)CC2 27938,c1(C(=O)NCCC2(OC)CN(C(C3CCCC3C)=O)C2)c(C)nn(C(C)C)c1C 27939,C1(NC(C2CC3(C2)CC(O)C3)=O)CCN(C(=O)C(F)(F)C(O)C2CC2)CC(O)C1 27940,C1(NC(CCc2cnc(C)s2)=O)CCN(CCC2CCOC2)CC1(C)C 27941,c1(C(=O)NC2(C)CCN(C(C(c3cnn(C)c3)C)=O)C2)ccc(N)c(Cl)n1 27942,C1(F)(CNC(c2c(CCC)nco2)=O)CCC(NC(=O)C=Cc2cscn2)C1 27943,C1(O)(CNC(C2(OC)CC(C)C2)=O)CCCN(C(c2cnc(C3CC3)s2)=O)C1 27944,c1(C(=O)NC(CC2CN(C(C(CSC)C)=O)C2)C)coc2c1CCCC2 27945,c1(SCC)nccnc1C(N1CC(OC)CC1CCNC(c1ncoc1C)=O)=O 27946,O=C1CCc2ccc(C(=O)NC3CCCC(NC(c4n[nH]cc4Cl)=O)C3)cc2N1 27947,c1(OC)ccnc(CNC2CC(C(=O)O)CCC2C)c1C 27948,C(C(=O)N1CC(O)(C(F)(F)F)C1)(C(C)(C)C)NC(c1cc(C)sc1)=O 27949,C1(NC(C2CN(C(C)C)C2)=O)C2CC(CN(C(=O)CCCCN(C)C)C2)C1CO 27950,N1(Cc2c(C#N)c(F)ccc2)CCC2(CC1)CCN2C(c1cc[n+]([O-])cc1)=O 27951,c1(CCC)[nH]nc(C(=O)NCC2CCN(C(C3CC3C)=O)C2(C)C)c1[N+](=O)[O-] 27952,N1(C(C2(OC)CCC2)=O)CC2CCC(NC(=O)C=Cc3ccc(C)s3)CC2C1 27953,C=CCCCC(=O)NCCCC1CN(C(=O)CCN(C)CCO)CCO1 27954,N#Cc1cc(CNC(C2CC2NC(c2ccncc2Cl)=O)=O)cc(F)c1 27955,N1(C(C2(C#C)CCCC2)=O)CCOC(C(=O)NC(COCC)CO)CC1 27956,O=C(CC(C(F)(F)F)N1CCOCC1)OCC1C2CCC(C2)C1C(F)(F)F 27957,N1(CCN(C)Cc2ccc(-c3cnc(C)s3)s2)CCC(F)(F)CC1 27958,C1(N(C(=O)CSc2nc[nH]n2)C)CCCC(NC(=O)Cc2ccc(Cl)cn2)C1 27959,C1(C(=O)NC(CC(C)NC(C(C)S(N)(=O)=O)=O)C)CN(C)CCN(C)C1 27960,N1(C(C2CCC(CCCCC)O2)=O)CCN(C(c2ccc(C)cc2)=O)C(C)C1 27961,C1(OC)CC(CNC(C2(N3CCCC3)CCC2)=O)N(C(c2cnc(C)s2)=O)C1 27962,C1(CNC(C2(CCOC)CCCC2)=O)CCN(C(c2nnc(C)s2)=O)C12CC2 27963,Cc1ccc(F)c(C(=O)NC2CCN(C(C3CC3C3CC3)=O)CC2)c1F 27964,C1(C(=O)NC2C(CNC(c3cnn(CC)c3C)=O)CCC2)CC12CCCCCC2 27965,N1(C(C2CCCC2O)C(=O)NCCOCC)CC(NC(C)=O)Cc2ccccc21 27966,N#Cc1ccc(C(=O)NC2CCN(C(=O)CSc3nncs3)CC2F)cc1 27967,c1(C(=O)NC(CC=C)CNC(=O)C#CC2(C)COC2)nc2ccccc2[nH]c1=O 27968,CC1(C)CCN(CC(=O)NCC(C)(O)CNC(c2cc(C#N)c[nH]2)=O)C1 27969,Cc1ccc(C(F)CC(CC(=O)NC(C)C(C)C)c2ccccc2)cc1C 27970,C1(CCC(=O)NC2(CNC(c3cc(C(C)=O)sc3)=O)CC2)CCCCN1C 27971,C1(NC(Cc2c(C)ncs2)=O)C2CC(NC(C3(C)CCCC3C)=O)CC12 27972,Oc1nc(CN2CCCCC2C2CCCC2)nc2c1COCC2 27973,N1(C(c2sccc2OC)=O)CCN(C(=O)NCCC2CCN(CCCC)C2)CC1 27974,C#CCCCCC(=O)NCCC12CC1CN(C(c1ccc(C)cc1)=O)C2 27975,c1(CNC(C2CCCN(c3ccncn3)C2)=O)ccc(C(=O)O)c(F)c1 27976,CC(C)(C)C(=O)C(=O)N1CCCCC1CCC(=O)NCC(C)(C)C1CCCC1 27977,C1(C)(COC)CC(NC(c2n[nH]c3c2CCC3)=O)CN1C(c1ccnc(S)c1)=O 27978,C(=O)(C(C(C)(C)O)NC(c1nonc1N)=O)NC(c1nnc(C)s1)C 27979,C1(CCNC(c2n(C=C)ncc2)=O)CC2CCC(C1)N2C(C1CCN(C)C1C)=O 27980,c1(C(N2CCC(C(C)(C)NC(C3OCCCO3)=O)C2)=O)cn2c(n1)CCC2 27981,c1(CC)cc(C(=O)NCC2(COC)CCCN2C(c2cocc2C)=O)cc(Cl)n1 27982,c1(CC(N2C(C)CC(NC(c3cc(C)nc(C)n3)=O)C2)=O)cnc2ncccn12 27983,C(=O)(C1CCc2snnc21)N1C2CN(C(C(C)c3cc[nH]n3)=O)C(C2)C1 27984,O=C1CCCC(C(=O)NCC(N2CCN(C(=O)CCn3cncn3)CC2)=O)O1 27985,Cc1ccc(CC(=O)NC(C)CCCNC(C2C=CCC2)=O)c(C)c1 27986,CCCCCCNC(=O)C(Cc1cnc[nH]1)NC(=O)CSc1cn[nH]c1 27987,c1(C(N2CCC(CNC(=O)C(F)(F)C3CC3)C(O)C2)=O)ccc2ncnn2n1 27988,N1(C(c2c(OCC)nccc2)=O)C2CCC1CN(C(c1noc(C)c1C)=O)C2 27989,Cc1cnc(Cl)c(C(N2CCC(CC(C)NC(c3ccc(F)nc3)=O)CC2)=O)c1 27990,c1(C(=O)NCC2OCCN(C(CS(CC)(=O)=O)=O)C2)ccc(OC)c([N+](=O)[O-])c1 27991,C(N=c1[nH]c(C)c(C(=O)NC(CCO)C(C)C)s1)c1c(F)ccc(OC)c1 27992,Cc1cc(NC(=O)C(=O)N(C)Cc2ccnc(Cl)c2)cnc1C 27993,c1(C(=O)NCC(Cc2ccccc2)CO)csc(=NCc2ccc(O)c(Cl)c2)[nH]1 27994,Cc1cc(C(F)F)oc1C(=O)NC(C)CC(C)NC(c1ccncn1)=O 27995,Cc1ccc(C(=O)NC23CC(NC(=O)C(Cl)(Cl)Cl)(C2)C3)c2ccccc12 27996,c1(C(C)=O)ccc(OCC(N2CCC(C)C2CNC(c2ccon2)=O)=O)cc1 27997,N1(C(CCn2ncn(C)c2=O)=O)CC2CC(NC(c3cnccc3Cl)=O)C2C1 27998,C1(NC(CCC=CC)=O)CC2CC(NC(c3cc(OC)cnc3F)=O)CC2C1 27999,N1(C(C(C2CCCC2)NC(=O)Nc2ccncc2)=O)CC(F)(C(F)(F)F)C1.CCO 28000,c1(C(N2CC(COC)(CNC(=O)C(C)(Cl)Cl)C2)=O)ccnc(S(N)(=O)=O)c1 28001,C12(CNC(c3c(CC=C)cccc3)=O)CN(C(=O)CN=S(C)(C)=O)CC1CCO2 28002,CC1CN(c2ncnc(Cl)c2F)CCC1CNC(C1CCC(C)O1)=O 28003,N12CCC3(C=C(C(=O)NC(C(C)C)C1=O)C3)C2.C12(CNC(N)=O)CCC(CO1)C2 28004,C1(CN(CCC(CC)C)CCOC)COc2ccccc2O1 28005,c1(OC(C(=O)OC)C)cccc(Nc2nc(C3CC3(F)F)cs2)c1 28006,Cc1ccc(-c2cn(CCCNC(c3nccn3-c3ccccc3)=O)nn2)cn1 28007,C1(NC(c2ccc(C#C)o2)=O)CCN(C(c2ccc(SC(F)(F)F)s2)=O)CC1C 28008,N1(C(C(CSC)(C)C)=O)CCOC2(C1)CN(C(=O)CCc1cccnc1)C2 28009,C1(C(=O)NCCc2cn(CC(=O)O)nn2)COc2ccc(F)cc2C1 28010,Cc1nnc2n1CC(C(N1CC3CC1CN(C(=O)Cc1ccsc1)C3)=O)CC2 28011,N1(C(C)=O)CCC2C1CCN2C(=O)OCc1ccc(F)c(C(=O)O)c1 28012,C1(C=O)CN(C(c2c(C)nc(-c3ccccc3)s2)=O)CC(F)(F)C1.C(C)C1CC1 28013,N1(C(C(=O)NCc2cc(OC)c(C)cc2)=O)CC2CCC(C1)C(=O)N2 28014,c1(CC(=O)NCC(C2CC(F)(F)C2)NC(CCC)=O)c(C(F)(F)F)coc1C 28015,c1(C(N2CC(C)C(F)(F)C2)C(=O)NCCCSCC)ccc(C#N)c(C)c1 28016,C1(C(=O)NC2(c3ccccc3)CCCN(C(CC)=O)C2)CCOC(C)(C)C1 28017,c1(CC(=O)NC(CNC(C(CCC)(C)O)=O)(C)C)ccc(S(C)=O)cc1 28018,C1(NC(CN(C(=O)Cc2c[nH]nc2C)CC#C)=O)CCCCC1N(C)C 28019,N1(C(C=C(CC)C)=O)CC2C(CNC(=O)CNC(N3CCOCC3)=O)C2C1 28020,N1(C(C(C)N(C)C)=O)CCC(C(=O)NCCc2cc(C3CCCN3)no2)C1 28021,C1(Cc2cn(CCN(C(CCOC)=O)C)nn2)(CO)CCOCC1 28022,N1(C(c2ccc(CC)cc2C)=O)CC(C)N(C(c2cnc(S)[nH]2)=O)CC1C 28023,C1(CNC(C(CC)CC)=O)CN(C(=O)C(C)(C)n2cccn2)CCCO1 28024,Cc1oc([N+](=O)[O-])cc1C(N1CC2CC1CC2CNC(=O)CC1=CCCC1)=O 28025,c1(C(=O)N(CC(CO)NC(CC2C(CC)C2)=O)CC)ccc2ccccc2n1 28026,Cc1oc(C(=O)N(CC(C)O)CCNC(C2(C)CCCN2C)=O)cc1Br 28027,N1(C(C(CCC)O)=O)CC(NC(c2cncc(C)n2)=O)CC12CCCCC2 28028,CC(C)(CCC(=O)NC1CCCC(F)(F)C1)NC(=O)Cc1ccsc1 28029,CC1CCN(C(=O)CCSC2CCCC2)C(C(=O)NC2CC3CC4C(C3)C24)C1 28030,C1(C(=O)NC2CCC(CNC(c3[nH]ccc3CN(C)C)=O)C2)CCS(=O)(=O)CC1 28031,c1(C(N(CCC(C)NC(C2CCCC2(C)C)=O)C)=O)cnc(N)c(Br)c1 28032,O=C(C(O)C(F)(F)F)N1CCN(C2CN(C(C3(Cl)CC3(F)F)=O)C2)CC1 28033,N1(C(C(CN(C(CSCCC)=O)C(C)C)N(C)C)=O)CCCC(F)CC1 28034,c1(C(N(C(CCNC(CN(CC)CC)=O)C)C)=O)cc(C(=O)OC)ncc1F 28035,C1(CC#C)(C(=O)NCc2ccc(Cl)cn2)CCN(C(=O)CCSC)C1 28036,c1(C(C)=O)cccc(C(=O)NCC(F)CNC(C2(c3ccc(F)cc3)CC2)=O)c1 28037,c1(SC)nc2ncnc(NCC3(F)CCN(C(=O)CCC4CCCO4)CC3)c2s1 28038,C1(CNC(C2C(OCC)C2)=O)CC(C(C)C)CCN1C(=O)CCS(=O)(=O)CC.OCC 28039,c1(OC)ccc(OC)c(C=CC(=O)N(C(C)CNC(c2cc(OC)no2)=O)C)c1 28040,Cc1ccc(C(=O)NC2CCOCC2NC(=O)CCc2ccoc2)cc1N 28041,C1(C(=O)NC(CCOC)C(C)C)CCCCC1(C)NC(c1c[nH]c(=N)c(C)c1)=O 28042,c1(C(N2CCC(NC(CC)=O)C2)=O)ccc2c(c1)CN(C1CCC(=O)NC1=O)C2=O 28043,N1(C(c2n(C(CC)C)ncc2)=O)CCN(C(C2CC(OC)CN2C(C)=O)=O)CC1 28044,C1(C(=O)NC(C)(C)CCNC(=O)CC2CCCS2(=O)=O)CC2COCC2C1 28045,CCCS(=O)(=O)C(C)C(=O)N(C(C)CCNC(c1cc2sccc2n1C)=O)C 28046,N(C1CCc2c(Br)cccc21)c1cc(NCCCSc2ccccc2)ncn1 28047,c1(NC(=O)NC(CC)C)ccc(NCC(F)(F)C(C)C)c(C)c1 28048,c1(C(=O)NC(CN(C(CC(=C)C)=O)CC)CC)cc(OC)c(OC(C)C)c(Cl)c1 28049,c1(C(c2nnnn2CC(F)F)NCCC(C)CO)ccc(Cl)c(F)c1 28050,N1(C(c2c(CC)sc(=N)[nH]2)=O)CCCOC(CNC(=O)C2=C(Cl)CC2)C1 28051,CN1C(CN=C(NCC2CCCSC2)NC2CC2)CCS1(=O)=O 28052,c1(C(N2C(CNC(=O)CCCCc3cnn[nH]3)CC2)=O)ccc(F)cc1Cl 28053,N12CC(C(O)C1)CN(C)CC2=O.c1(CNC(c2cc[nH]n2)=O)ccccc1 28054,CN1c2ccc(C(=O)NCCCNC(c3coc(Cl)c3)=O)cc2C(C)(C)S1(=O)=O 28055,C1(NC(c2c(CC)non2)=O)CCN(C(C2COCC(C)O2)=O)C1C1CC1 28056,N1(C(C(N)=O)=O)CC2(CCC2CNC(C2CCCS2)=O)C1 28057,c1(CC(C(=O)OC)NC(c2ncc(C)cn2)C)ccc(OC)cc1Cl 28058,c1(C(=O)NC(CN(C(C2(c3ccoc3)CC2)=O)CC)C)cc(C)cc(C#N)c1.C 28059,CN=c1[nH]cc(C(=O)N(C2CCN(C(c3ccncn3)=O)C2)C)s1 28060,c1(C(=O)NCC(CN(C(C2(CCOC)CC2)=O)C)(C)C)[nH]c(C)c([N+](=O)[O-])c1C 28061,N1(C(CC2(C=C)CCCCC2)=O)CC2(C1)CN(C(=O)C(O)COC)CC2CO 28062,c1(CCNC(C2(CCCC)CC2)=O)ccc(CNC(=O)CCCCN(C)C)cc1 28063,c1(C(C)NC(C2C(C#N)C2(C)C)=O)ccc2nc(O)[nH]c2c1 28064,C(=O)(CC1=CCN(C)CC1)NCC(C#C)OC.O1NC(=O)C2CC2C1C 28065,c1(C(N2CCN(C(CSCCCC)=O)CC2C(C)C)=O)cccc2cncn12 28066,CC1CCCCC1C(=O)N(C1CCCCC1)CCNC(=O)COc1ccccc1 28067,N1(C(c2nc(N(C)C)oc2)=O)CCC2(CCN(C(=O)Cn3cc(CO)nn3)C2)C1 28068,C1(CNC(c2c(CCC)n(C3CCCC3)nc2)=O)CC2(CC2)CN1C(=O)COC 28069,N1(C(c2c(O)ccc(C#N)c2)=O)CCC2(CCCC2NC(=O)CC(F)(F)F)CC1 28070,c1(CC)cc(NC(=O)C(C)(C)C2CCN(C(=O)C(C)C(F)(F)F)C2)ccc1C 28071,c1(OC)ccc(C)nc1C(N1CC(OC)C(NC(=O)COc2cc(C)on2)C1)=O 28072,C(=O)(C(C(C)(C)C)n1ccnn1)N(CC(CC)NC(c1csc(=NC)[nH]1)=O)C 28073,Cc1[nH]nc2c1CCC(C(=O)NC1CCCN(S(=O)(=O)c3ccc(Br)cc3)C1)C2 28074,C1(O)(C(C)NC(COC)=O)CCN(C(=O)Cc2ccccc2CC#N)C1 28075,c1(NC(=O)C(N2CCN(c3ccnnc3)CC2)=O)ccccc1-n1ccnn1 28076,C1(NC(=O)CC2CC3(CC3)C2)CC(CNC(c2csc(Br)c2)=O)C12CCC2 28077,c1(C(N2CCN(C(C=CCOCCOC)=O)CC2C)=O)cc(S(N)(=O)=O)sc1C 28078,N1(S(CC(=O)OC)(=O)=O)CCCC2C1CCN2Cc1ccc2occc2c1 28079,C1(OC)CN(C(=O)Cc2nccn2C)CC1NC(C1CCOCC1)=O 28080,CCCCS(=O)(=O)NC(=O)C(=Cc1cccnc1)F.C1(CC)CNCC(=O)N1 28081,C(=O)(N1CC=CCO1)C1(C(F)F)CC1.C12CCN(CC1)NC2C 28082,c1(OC)ccc(C(=O)NCC2CC(O)CN2C(=O)C(F)=CCCF)nc1OC 28083,S(=O)(=O)(c1[nH]c(=NCCCCC(C)(C)NC)ccc1Br)N1CCC(N(C)C)CC1 28084,Cc1cn2ccc(C(=O)NC(C3CN(C(c4cnns4)=O)C3)C)cc2n1 28085,N1(C(C(C)(C)NS(C)(=O)=O)=O)CCOCC(NC(c2coc(Br)c2)=O)C1 28086,Cc1ccc(CC(=O)NCC2(NC(=O)CSCCN(C)C)CCOCC2)cc1C.C(C)C 28087,C=CC1CN(C(=O)CCN(C(=O)CCCCCC)CC)CCO1 28088,CCC(C)(C)CCCC(=O)N1CC(NC(C2(C)CCCCO2)=O)CCC1C 28089,Cc1cc(Br)oc1C(=O)NCC1COC(CNC(=O)C=Cc2cocn2)C1 28090,C1(CC)CCCCCN1C(=O)Cn1cc(CN)nn1.c1(C=O)cc(N(C)C)ccn1 28091,c1(C(=O)NCC(CNC(c2c(N)nc(Cl)cc2)=O)CO)ccc2nonc2c1 28092,CCC(C)C(O)C(C)C(=O)N(C)CC1CCCN1C(C12CCCN(CC1)C2)=O 28093,C1(C(N(C)CC2CN(C(c3cn(C4CC4)nn3)=O)CCO2)=O)CCC=CCCC1 28094,C1(CCC(=O)NCC(C2CCCC2)NC(c2cc(Cl)ccn2)=O)NC(=O)NC1=O 28095,CC1CN(C(=O)C2=CCSC2)CC2(CCN(c3nnc(C(N)=O)s3)C2)O1 28096,C(CN=c1nn[nH]n1-c1ccccc1)NC(C1CC2CC2C1)=O 28097,C1(CC(=O)NC2(CF)CCN(C(CCC(C)C)=O)C2)COC(C)(C)CO1 28098,N1(C(CCC(CC)CC)=O)CC(C2CCCN(C(C3CC(=O)NC(=O)C3)=O)C2)C1 28099,c1(C(N(CCNC(c2cscc2Br)=O)C2CC2)=O)cc2ncccc2[nH]1 28100,C12(NC(CCOC(C)C)=O)CC(CNC(c3csc4nnsc34)=O)(C1)OC2(C)C 28101,C12(C(=O)NC3CCC(N(C(c4ccc(COC)s4)=O)C)C3)CCOC(C)(C1)C2 28102,C1(CC(=O)NC(C(=O)OC)CN2CCOCC2)CCNC2(CC2)C1 28103,C12(C(N(C(CN(C(CNC(CCC)=O)=O)C)C)C)=O)CC1COC2(C)C 28104,C1(C(=O)OCC2(F)CCN(C(=O)OC(C)(C)C)C2)CCCS(=O)(=O)C1 28105,C1(CN(C)C(c2ccnc(F)c2)=O)CCCN(C(C2CCCCN2C(N)=O)=O)C1 28106,C(C(C)(C(=O)Nc1conc1C)NC(c1ccc(C#N)o1)=O)SC 28107,C(C[Si](C)(C)C)NC(CN(CC#C)C(c1cc(Cl)cs1)=O)=O 28108,C(CC(N)=O)(C(=O)NC(C)C(=O)NC1CC1)NC(c1nccc(CC)c1)=O 28109,c1(C(=O)NCC2CN(C(CCSCC)=O)CC2O)cc(CC)cnc1O 28110,N1(C(c2cnc(COC)s2)=O)CCC2(NC(=O)CSS(C)(=O)=O)CCCC12 28111,N1(C(CCC(=O)N(C)C)=O)CCC(C2CCN(C(c3ccc(F)cc3Cl)=O)C2)C1 28112,c1(CCC(=O)NC2C(NC(Cc3c(C)scc3)=O)COC2)cccc(N(C)C)c1 28113,c1(C(N(c2n(CC)nc(C)c2)C2CC3CNC2C3)=O)cc(F)ncc1NC(C)=O 28114,N1(C(CC)=O)CCC(C(=O)NCC(CC)NC(=O)CC(O)c2ccccc2)C1 28115,c1(C(=O)NC2CN(C(CC(C)C3CC3)=O)CC(F)C2)ccc2n[nH]cc2c1Cl 28116,N1(C(C(C2CC(F)(F)C2)OC)=O)CCC(NC(c2ccns2)=O)CC1C 28117,N1(C(Cc2n(C)cnn2)=O)CCC(CNC(C2CC(n3cnnc3)C2)=O)C12CC2 28118,C1(C(N2CCC(C3(C)N=N3)CC2)=O)CN(C(c2ccccc2Cl)=O)CC1(F)F 28119,CCCCCCC(C)(c1nnnn1CCCF)NCC=C1CCSCC1 28120,C=CC(C)(O)CC(=O)NC1CCN(C(=O)CCc2nc(CSC)no2)C1 28121,c1(NCC2CCCCN(C(CCCCOC)=O)C2)nnc(C)c(C)c1C#N 28122,C=C(C)C(C)(C)C(=O)NCCNC(c1ccnc(C(C)(C)O)c1)=O 28123,N1(Cc2cccc(C)c2F)CCC2(C1)CN(c1ncc(C3CC3)cn1)CCO2 28124,c1(CNC(NCc2ccc(C#N)nc2)=NCCCF)ccc2c(c1)OCCCO2 28125,N1(C(CC2(C)CCN(C(CSC)=O)C2)=O)Cc2cccc(F)c2C1 28126,N1(C(CSCC2CCCO2)=O)CC2CCCC(C(=O)NCc3[nH]c(=N)sc3)(C2)C1 28127,C(=O)(C1=CCS(=O)(=O)C1)NCC1CC(C)(C)CN1C(C1CC1C(F)F)=O 28128,C#CCCCC(C(=O)Nc1ccc2c(c1)CCC2)N(C1CCCS(=O)(=O)C1)C 28129,c1(-c2nc(CCC)nn2C2CCS(=O)(=O)CC2)ccnc2c(I)cnn12 28130,Cc1c(C(=O)NCC2CCN(C(=O)C(F)=C3CCC3)C2)cnn1CCO 28131,c1(OC)c(CC(=O)NC(C)CCNC(C2CCC(C)CC2)=O)cccc1C#N 28132,CC1CN(C(c2cnn3c2SCC3)=O)CC(C)N(C(c2cncs2)=O)C1 28133,C(=O)(C(F)C(C)CNC(c1ccc(C)o1)=O)N(C(CC)C(=O)OC)C 28134,N1(C(c2c(F)cccc2Cl)=O)CCC2(CC1)CN(C(C1CC1F)=O)CCC2O 28135,c1(C(=O)NC(C(C(C)C)NC(Cc2c(C)ocn2)=O)C)ccsc1S(C)(=O)=O 28136,N1(c2c(C#N)cnc(C)n2)Cc2ccc(NC(=O)C(c3ccccc3)O)cc2C1 28137,Cc1ccc(N)c(C)c1C(=O)N(CC(O)CN(C(=O)CC(C)C1CC1)C)C 28138,CCC(CC(=O)N(CC(C)C(=O)NC(C)CC1CC1)C)CC(C)C 28139,C1(NC(C=C2CCN(C(C3(COC)COC3)=O)CC2)=O)CC(=O)N(C)C1=O 28140,C1(CNC(C(CCCC)C)(C)c2nnnn2CC(F)F)Cc2ccccc2CO1 28141,c1(C(=O)NC(c2cc(F)cc(Cl)c2)CNC(C2CC(O)C2)=O)n[nH]cc1[N+](=O)[O-] 28142,N1(C(CCCn2c(C)ncc2)=O)CC(NC(=O)CC2COCCO2)CC(C)(C)C1 28143,CON(Cc1ccccc1)C(=O)C(CNC(c1csc(C#N)c1)=O)N(C)C 28144,C(=O)(C1=CC2C=CC1C2)N1CCCC(C(=O)Nc2c(C(C)C)nccc2)CC1 28145,C12(CCNC(=O)Cc3ccsc3)CCC1CN(C(c1ccc(CO)c(Cl)c1)=O)C2 28146,C(CCN(C)C)(C(=O)NCC1(O)CCOC1)NC(Cn1ncc(CC)c1)=O 28147,C#Cc1cccc(CNC(C2(CCNC(=O)C(c3cnccn3)C)CCC2)=O)c1 28148,N1(C(C2(C)CCCOC2)=O)CC2CCN(C(c3ccc(Cl)cc3O)=O)C(C2)C1 28149,CC1(C)CC1(C#N)C(N1CC2C(NC(c3cn[nH]c3)=O)C2C1)=O 28150,c1(C(=O)NCC2C(C)CN(C(c3nnc(C(C)(C)C)s3)=O)C2)cc(C#N)cn1C 28151,c1(C(=O)NC2C(C)(C)CCN(C(C3CC(C)(C)O3)=O)C2)cc2nn[nH]c2cc1F 28152,C(=O)(C1=CCCC(C)(C)C1)N(C1CCN(C(C2(S(C)(=O)=O)CCCC2)=O)C1)C 28153,CC(C)(C)C(CNC(C12CC(F)C1C2)=O)NC(C1CCC(=C2CCC2)CC1)=O 28154,N1(C(c2cnn(C)n2)=O)CCCC(C2CCCCN2C(=O)C(=O)NCC2CC2)C1 28155,c1(C(=O)OC)ccc(NC(=O)CC2CC(NCc3ccc(O)cn3)C2)cn1 28156,CN(S(=O)(=O)N1CC(O)C1)CC1CCCCC1 28157,Cc1csc2nc(CC(=O)N(C3CN(C(=O)CC4CC(C)C4)CC3O)C)cn12 28158,C12(C(=O)NCCNC(c3c(OC)cc(C)cc3)=O)CCC(F)(CNC1=O)C2 28159,C(=O)(C(O)CCn1cncn1)NC(C(C)NC(c1cnn(CC2CC2)c1)=O)(C)C 28160,C1(OC)(CNC(=O)C(=Cc2cccs2)C)CCN(C(C2C3CCCCC23)=O)C1 28161,N1(C(c2c(-c3ccn(C)n3)n[nH]c2)=O)CCC2(NC(c3ccsc3)=O)CC2C1 28162,C(=O)(CS(=O)(=O)CC(F)(F)F)NCC1(C(F)F)CCN(C(C(CC)(C)O)=O)C1 28163,c1(C(N(CC(C)NC(C2CCCO2)=O)C)=O)ccc(N)c(C(F)(F)F)c1 28164,C1(C(=O)NC(C(C)C)(C)CNC(=O)C(C)(C)N(C)C)CCCC(=O)N1C 28165,n1(CCCC)ccc(C(=O)NC2(CNC(=O)Cc3c[nH]nc3C)CCCC2)n1 28166,c1(CC)ccc(C(=O)NCC(C)CN(C)C(c2cccn2C(C)C)=O)cc1F 28167,c1(C(N2C3CC(CNC(C(C(=O)OCC)F)=O)C2CC3)=O)ccc2c(n1)CCC2 28168,Cn1ncc2ccnc(C(=O)NCC=CCNC(=O)C(O)P(C)(C)=O)c12 28169,c1(NC(C2N(Cc3c(C)c(O)ccc3)CC3(CC3)C2)=O)cnn2ccc(Cl)nc12 28170,Cc1nc(O)sc1C(=O)NC(C)(CSC)C(=O)NC1CCN(C(N)=O)CC1 28171,N1(C(c2sccc2Br)C(=O)NCCCSCC)CCCC2(CO)CCCC12 28172,CC(C)C(C(=O)NCC1CN(C(=O)Cc2ccccc2F)CC(C)(C)O1)C(C)C 28173,C(=O)(C(CCSC)NC(=O)C(C)NC(=O)CC)NC(CC=C)C1CC1 28174,C1(NC(c2cscc2Br)=O)CN(C(=O)CCc2cncnc2)CC1(F)F 28175,c1(CC)ccccc1CNCC1(C(=O)Nc2cc(CC3CC3)ncn2)CCC1 28176,c1(NC(C(C)NC(c2c(COC)cco2)=O)C(C)C)ncc(Cl)c(C)c1C#N 28177,c1(C(N2C3(CN(C(C4CN(CCC)C(=O)C4)=O)C3)CC2)=O)cc(F)cc(F)c1F 28178,N1(C(CCc2cnn(C)n2)=O)CCC2(CC1)CCN(C(C1CC(O)C1)=O)CC2 28179,c1(C(N2CC(C)C(NC(c3cscc3S(C)(=O)=O)=O)C2)=O)ccn2ccnc2c1 28180,C(c1csc2ccccc12)=CC(=O)NC1CCCCN(CC)C1=O 28181,c1(CC(=O)NCC2COCCN(c3ncc(C)cn3)C2)cccc2c1OCCO2 28182,CC(C)CCCCCC(=O)NC(C1(CNC(=O)Cn2cc(C(F)F)cn2)CC1)C 28183,c1(CC(=O)NCC(C)NC(c2c[nH]nc2-c2ccccc2)=O)cc(F)cc(F)c1 28184,c1(CNC(N2CC(c3ccn(C)n3)OCC2)=O)ccc(I)c(Br)c1 28185,C1(OC)CC(NC(=O)CN(CC(C)C)C(=O)Cc2cccnc2)C1(C)C 28186,C1(CC(=O)NC)CN(C(=O)C(O)CC(F)F)CCN1C(c1nc(C)sc1C)=O 28187,N1(C(C(CC2CCCC2)NC(c2c(C)nc(O)s2)=O)=O)Cc2n[nH]cc2C1CO 28188,C1(CNC(C(CC=CC)NC(=O)OC(C)(C)C)=O)CC(c2ccc(C)cc2)=NO1 28189,N1(C(c2cccc(CCC)c2)=O)CCC2CN(C(=O)Cc3cn[nH]c3)C2C1 28190,Cc1c(C(N2CCC(CCNC(C3CC(=O)N(CC4CC4)C3)=O)C2)=O)ncn1C 28191,N1(C(CS(N)(=O)=O)=O)CCOCC(NC(=O)C(O)Cc2ccccc2)C1 28192,Cc1nc(Cl)ccc1CC(=O)N(CC(O)CN(C)C(c1ccn(C)c1)=O)C 28193,Cc1ccc(C(=O)NC(C)C(N2CCC(N(C)C(C34CC(CO3)C4)=O)C2)=O)cc1 28194,c1(OC)ccc(C(N2CC(O)CC2C(=O)NCc2ccc(Br)c(Br)c2)=O)cc1I 28195,C1(C(=O)NC(CNC(CC2(C)CCCCC2)=O)C2CC2)CCOC(=O)CC1 28196,c1(C(N(CCN(C(Cc2cnc(C)[nH]2)=O)C(C)C)C)=O)ccc(OC(F)F)nc1 28197,C12(CC(N3CCC(n4cnnn4)C3)=O)CCC1CN(C(=O)C=C1CCCCC1)C2 28198,C1(N(C(=O)Cn2cnnn2)C)CCCN(C(C2(C#N)CCCO2)=O)CC1 28199,C1(CCC(N2CC(N(CC(=O)N(C(C)C)C(C)C)C)C2)=O)CCCCO1 28200,c1(CNC(NCc2cn(C)nc2)=NCCC2CCOC2)ccc2oc(O)nc2c1 28201,N1(C(c2c(C)cncc2C)=O)CCC2C(CCCN2C(=O)C(F)CC(C)C)C1 28202,c1(C(=O)NC(c2ncc(N(C)C)cn2)C)ccc(Cl)c(O)c1 28203,C1(NC(C2CC(=O)NCC2)=O)C2CC(O)C1N(C(=O)CC1(C(F)(F)F)CC1)C2 28204,CC1CCCCC1(CNC(=O)Cc1sc(O)nc1O)NC(=O)CC1CCCCC1C 28205,N1(C(c2nc(OCC)sn2)=O)CCC(C2(NC(c3cc(CO)[nH]n3)=O)CC2)CC1 28206,CCCCCS(=O)(=O)CC(=O)N1CCN(Cc2cc(OC)c(O)c(OC)c2)CC1 28207,C1(NC(c2n(CCOC)ncc2)=O)CC(C)N(C(c2nn(C)cc2SC)=O)C1 28208,N1(C(=O)NC(Cc2cccc(OC)c2)C)CCC(C2CCN(C)CC2)C1 28209,c1(C(N(CC(C)O)CCNC(c2cncc(C=C)c2)=O)=O)cnc2scc(C)n12 28210,S(=O)(=O)(c1c[nH]ccc1=NCC1CCC2(CCCC2)O1)N1C(C)CSC1 28211,N1(C(Cc2cccc(OCC)c2)=O)CCC(NC(=O)COc2cccnc2)C1(C)C 28212,c1(C(N2CC3C(NCc4c(Cl)ccc(Cl)c4Cl)C3C2)=O)cnc2cc(Cl)ccn12 28213,c1(C(N2CC(OC)C(NC(=O)C(C)S(C)(=O)=O)C2)=O)ccc2c(c1)NC(=O)C2 28214,N1(C(C(CC)SC)=O)CCC2(CC1)CCN(C(=O)C=C(C)c1cccs1)CC2C 28215,CC1=C(C(=O)NC23CCN(C(=O)CC(C)(C)C)CC2C3)CCC1 28216,N1(C(C=CCCC)=O)CCC(CNC(=O)Cn2ccnc2)C(C)C1 28217,C(=O)(CC1OCCc2ccsc21)N1CC(NC(C(CC(C)C)(F)F)=O)CC1(C)C 28218,c1(C(=O)NC(CNC(CN2CC(C)C2)=O)C2CCC2)cc2cc[nH]c2cn1 28219,C(=O)(CCCCCN(C(C1CCC1C)=O)C(C)C)N(CC(F)F)CC 28220,C(C)(C)(CC(F)C(=O)NCCc1cccnc1)NC(c1scc(C)c1)=O 28221,c1(C(N2CCCC(NC(C(C)n3cccc3)=O)C2)=O)ccc2c(c1)COC2 28222,C(CC(=O)N1CC(CC(C)(C)C)C1)N(C(=O)C=CC(F)(F)F)CC 28223,C(C(C)(C(C)C)NC(=O)Cc1csc(C(C)=O)c1)NC(CCOCCCOC)=O 28224,C1(NC(C(C#C)(C)C)=O)CCC(C)(CNC(c2coc(C(F)F)n2)=O)CC1 28225,c1(C(=O)NC2C=CC(CNC(C(C)CN(C)C)=O)C2)ccc(=O)n(CCF)n1 28226,CC1CCC(C)(NC(c2conc2CNC(C2C3CCC(=O)C23)=O)=O)C1 28227,c1(CN2CC(NC(c3c(Cl)ccnc3Cl)=O)C(F)(F)C2)ccc2c(c1)CCO2 28228,C1(C(=O)NCC2(C(N)=O)CN(C(C3CCCC34CC4)=O)C2)(OC)CCS(=O)(=O)C1 28229,C1(NC(C(C)NC=O)=O)CCN(C(c2ccnn2CC#N)=O)CC1(C)C 28230,CC1CCCCC1C(=O)NC(C)(C)C=CC(=O)NCC(F)Cl 28231,C1(CNC(C(C(CC)C)O)=O)CCCC2(CN(C(=O)Cc3cccc(Cl)c3)C2)O1 28232,Cc1c(C(=O)NC2CN(C(=O)CC3C=CCCC3)C2)c(C(F)(F)F)nn1C 28233,Cc1cccc2c(C(N3CCCC(N(CCF)C(C4CC4(F)F)=O)C3)=O)coc12 28234,N1(C(C2CCOC2C(=O)NC2(c3nc[nH]n3)CCC2)=O)CCCC1(C)C=O.CO 28235,N1(C(C(C(C)C)SC)=O)CCN(C(=O)Cn2nnnc2-c2ccsc2)CC12CC2 28236,Cc1cccc(C(=O)NCC(F)CNC(c2cnc(CC(C)C)[nH]2)=O)c1C 28237,c1(C(=O)NCC2CCOC2)cc2c(s1)CCN(C(c1cc(Cl)c(Br)cc1Cl)=O)C2 28238,C(=O)(C(F)(F)C(F)(F)F)NC1C(CNC(c2cc(C)n(CCO)n2)=O)COC1 28239,c1(C(=O)NCC)ccc(NC(=O)Cn2cc(CCCNC(N)=O)nn2)cc1C 28240,CC1(C)CC(CNC(=O)CCCNC(N)=O)CN(C(C2(F)CC2)=O)C1 28241,N1(C(C(C)=C2CCCC2)=O)CC2CCCCC2(CNC(=O)CCC2CCCO2)C1 28242,C#Cc1ccc(C(=O)NC2CCN(C(=O)CC(C)C(F)(F)F)C23CC3)cc1C 28243,CP(C)(=O)C(O)C(=O)NCCCOCCOCCNC(c1ccc(Cl)nc1)=O 28244,C#CC1CN(C(C2CCC2C#N)=O)CCN1C(c1cnc2[nH]nnc2c1)=O 28245,C(=O)(CCCCCCNC(=O)C(C)(CO)NC(C)=O)NC(C(C)NC(C)=O)CO 28246,N1(C(C(F)=CCC)=O)CC(CNC(=O)CSC2CCC2C(C)(C)C)CCC1=O 28247,c1(OC)ccc(C(=O)NC(C)C(C)NC(c2[nH]ncc2C#N)=O)c(C)c1 28248,C#CCC(C)(C(=O)NCC(C)S(N)(=O)=O)NC(c1cccnc1NC)=O 28249,Cc1c(F)ccc(CN2CCC(F)(C(=O)NC(c3cccnc3)C)C2)c1Cl 28250,CCCC(CCC)C(=O)NCCN(C1CCCCC1)C(C1CC1COC)=O 28251,c1(C(=O)NCC(CO)NC(c2cc(SC)oc2)=O)ccc([N+](=O)[O-])s1 28252,n1(CCC(N2CCC(C(C)NC(c3ccc(CC)[nH]3)=O)C2)=O)ccc(O)nc1=O 28253,CCCC(C(=O)OC)C(=O)N1CCC(C)(C)C1C(=O)NCc1cnc(O)nc1O 28254,C1(Cl)(CNC(c2nnnn2C2CC2)(COCC)C)CC12CCC2 28255,C(=O)(CCN=c1[nH]ccs1)NCC1CC(OC)CN1C(c1c[nH]c(Br)c1)=O 28256,c1(N2CC(C)(CNC(C(C)N(C)C)=O)OCC2)ncnc2sc(C(F)(F)F)nc12 28257,C(=O)(C1=NOC(C)(C)C1)N1CC(C(=O)NCC(COC)C(C)C)C(F)C1 28258,N1(C(c2cnn(C3CCOC3)n2)=O)CCN(C(c2csnc2Br)=O)CC1 28259,c1(OC)cc(CNC(=O)C(F)C2CC(NC(C3(n4nccn4)CC3)=O)C2)on1 28260,C(=O)(C(C)(C)C(F)F)N1CCCC(CCNC(C2C(C)(C)C2(F)F)=O)C1 28261,N1(C(c2ccc(C)cc2)=O)CCC(C2CC2)C1CNC(c1nsnc1O)=O 28262,N1(C(c2c(CC)ncs2)=O)CCCC(C(C)NC(c2c(C)nnn2C)=O)C1 28263,C(CCCCCNC(=O)C(Br)=C(C)C)N(C(c1c(CC)cco1)=O)C 28264,c1(C(=O)NCC#CCNC(=O)C=CC2CCCO2)cc2ccccn2n1 28265,c1(C(=O)NC(CC(C)NC(=O)Cn2cc(Cl)cn2)C)ccc2c(c1)CCC2(F)F 28266,S(=O)(=O)(c1ccc2c(c1)COCC2)N1CC2C(C)(C)C2C1 28267,C1(C(=O)NC2CCCC(NC(=O)CSCC(F)(F)F)C2)(CC)CCC(O)CC1 28268,c1(C(=O)NCC2(NC(=O)CO)CCC2)cnn2c(-c3cccs3)ccnc12 28269,C[Si](C)(C)CCCNC(=O)CONC(C1CC(F)CN1)=O 28270,Cc1ccccc1CC(C)C(=O)NCCC1(NC(=O)CCSCC(N)=O)CC1 28271,CS(=O)(=NC(=O)CC1CCCCS1(=O)=O)c1ccccc1 28272,c1(C(N(C)CC2CCCN(C(CCC3CCC(C)O3)=O)C2)=O)c[nH]cc(F)c1=O 28273,C12(NC(CC(CC)C(C)C)=O)CCCC(CN(C(c3cccn3C)=O)C1)C2 28274,N1(C(C(C)(C)F)=O)CC2CCC(C1)N2C(C1CC1c1ccc(Br)s1)=O 28275,c1(NCC(=O)NCCCN(C)C(=O)NC)cccc(C(N)=O)c1 28276,Cc1nnc2n1CCN(C(c1ccc(CNC(=O)Cc3cccc(F)c3)nc1)=O)C2 28277,N1(C(C2CC(CCC)OCC2)=O)C2CCCC1CN(C(c1cccc[n+]1[O-])=O)C2 28278,C1(NC(c2c(OC)scc2)=O)CC2CC(NC(=O)C(C)(O)C3CCC3)C1C2 28279,C(=O)(C(CCCOC)NC(=O)CSCCOC)N1C(CC)CC1 28280,CCC(CCCC(=O)NC1(CC)CCC1)NC(C1(NC(N)=O)CC1)=O 28281,N1(Cc2cccc(CC)c2)CC2CC(NC(=O)CS(=O)(=O)C(C)C)CC1C2 28282,CCC(CC(=O)N1CCC(C(C)O)CC1)NC(=O)C(=CC1CCCC1)C 28283,NS(=O)(=O)CCC(=O)N1CC(Cn2cc(C3(O)CCOC3)nn2)C1 28284,Cc1nc(C(F)(F)F)ccc1CNC(=O)C=CC(C)NC(C1CC1(C)C)=O 28285,N1(C(C2(NC(C)C)CC2)=O)CCC2C(C1)CN2C(=O)CC1(C(F)(F)F)CC1 28286,C#CC1CN(C(=O)CCOCCN(C(=O)C(C)CC(C)C)C)CCN1C 28287,N1(C(c2c(CC)occ2)=O)CCCC(C)(OC)CC1.C12(C)C=C(C(=O)NC1)C2 28288,Cc1ccc(CN2C(C(=O)NCC3CCC(O)CC3)CC3CC23)c(Cl)c1Cl 28289,C1(C(=O)NCC(CNC(CSCCN(C)C)=O)(C)C)CCc2nccn2C1 28290,N(C1CC(C)n2ccnc21)C(CCC(Cn1cc(CNC(C)=O)nn1)(F)F)=O 28291,C1(C(=O)NCC(C=C)O)CCN(C(C2CN(C)CCO2)=O)CC1(C)C 28292,C(=O)(C1Cc2ccc(Cl)cc21)NC1C2CN(C(C3(C)COC3)=O)CC1COC2 28293,C1(C(=O)NCC(N2CCN(C(c3ncccc3F)=O)CC2)C)CC2(CCC2)C1 28294,C1(C(C(=O)NCc2ccco2)N(CCC)CCc2ccccc2)CCOC(C)C1 28295,N1(C(CNC(CNC(c2cc(C)sc2N)=O)=O)=O)CC2CCCCC2C1C 28296,C(=O)(C(C)(C)C(F)(F)F)NCCC1CCC(NC(CCC(=O)NCC)=O)C1 28297,CCCCCCCC(=O)N1CC(C(=O)NCc2ccc(Cl)cc2Cl)C1 28298,C1(N(C)C)CCCCC1C(=O)NC1CC(C)(NC(=O)CCC2CC2(C)C)C1 28299,C1(NC(CCCCOCCC=C)=O)CC2C1CCN2C(=O)CC(CC)C1CCC1 28300,N1(C(CCCOCC=C)=O)CCC2(CCCN(Cc3ccc(Cl)c(F)c3)C2)C1 28301,N1(C(C(CC)C#N)=O)CCCC(C(=O)NC2COCC2CO)CC1 28302,N1(c2nnc(CCC)n2CC(C)C)CC2C3CCC(CC3)C2C1 28303,Cc1ccccc1C1CC1C(N1CCCC(C(=O)Nc2cncn2C(C)C)C1)=O 28304,c1(OCC#C)cncc(CN2CCC(SC)CC2)n1 28305,C(CC(C)(C)CC(=O)NCC1(C)CC(F)(F)CN1C(c1cnsc1)=O)OC 28306,c1(C(=O)NC2(CC=C)CCN(C(=O)CSCCC(C)C)C2)cnc(C)c(C)c1 28307,CC1C2CCC(C2)C1C(N1CCC(C)(CC(N2CCC2C2CCCC2)=O)C1)=O 28308,N1(C(C=C(CC)C)=O)CCC2CCC12C1C(NC(=O)Cn2cc(Br)ccc2=O)C1 28309,c1(-n2c(C3CCC(C(C)OC)CC3)nc(CCCCCC)n2)cc(C)ccc1C 28310,c1(C(=O)NC(CC=C)CNC(=O)CCCC2CCCCC2)ccc(C(C)C)cn1 28311,c1(C(=O)OC)cncc(C(=O)NC23CC(NC(C4CCCNC4=O)=O)(C2)C3)c1 28312,C(C(C(=O)NCc1nc(C2CC2)n[nH]1)C(C)C)NC(C(C)SCC)=O 28313,C(C(CC1CCCC1)C(=O)NC1CCC(C)CC1)NC(COC(C)=O)=O 28314,CC(C)(C)COCC(=O)NC(C(=O)NCCCC(C)(C)n1ccnc1)C1(O)CCC1 28315,N1(C(C2C(COC)CC2)=O)CCN(C(c2ccccc2Cl)=O)CC(O)C1 28316,CCC(C(=O)OC)C(=O)NC1(CNC(c2cccc(SC(F)(F)F)c2)=O)CCC1 28317,c1(C(=O)NC2(CCC(=O)NC(c3cn(CC)nc3)C)CCC2)cnnc(C)c1 28318,c1(CC)cc(F)c(C(N2CCN(C(c3cccc(O)c3C)=O)CC2)=O)c(F)c1 28319,N1(c2cc(CC)nc(C)n2)CCOC2(CCCN(C(=O)CC3CCC(C)C3)C2)C1 28320,C1(NC(C(C)C2CCC2)=O)CN(C(c2cncn(C)c2=O)=O)CC12CC2 28321,C1(NC(CCC(C)c2ccc(Br)cc2)=O)CC=C(C(=O)N2CCOCC2)C1 28322,C(C(C)C(=O)NC(C)(CNC(=O)COCCCC(C)C)CC)OCC 28323,N1(C(C2CCOCC2)=O)CCN(C(=O)CNC2CN(S(CC)(=O)=O)C2)C2CCC12 28324,C(=O)(CS(=O)(=O)N(C)C)NC(C1CN(C(c2cn(C(C)(C)C)cn2)=O)CCO1)C 28325,N1(C(C2C3CN(C(c4cc(OCC)c(Br)cc4)=O)C2C3)=O)CCC(C)C(F)(F)C1 28326,N1(C(CC2C(CNC(C3(CF)CC(=O)C3)=O)C2)=O)CC2(CSC2)C1 28327,N1(C(C(C)CS(C)(=O)=O)=O)CCN(C(C2(C)CCN(C)C2=O)=O)CC(C)(C)C1 28328,N12CC(C)(C)C1Sc1cc(cs1)C2C(=O)NCCC.C(C)(C)(C)OC(=O)NCCl 28329,C1(C(=O)NCCC2(CNC(C=C3CCC(C)C3)=O)CC2)(CO)CC(C)(C)C1 28330,C=CCC(CC(F)F)NC(=O)C(CCC1CC1)NC(c1ccncc1CC)=O 28331,C1(C(=O)NCC2CC23CCN(C(=O)C(F)OC(F)(F)F)C3)CC2(CCO1)CC2 28332,C1(NC(C(c2ccc(Cl)cc2)(C)C)=O)CN(C(C2CC(C)(C)C2)=O)CC(F)(F)C1 28333,CCS(=O)CC(=O)NCCN(CCOCCO)C(c1cccnc1OC)=O 28334,n1(CC(=O)NCC2C(CNC(C3CC(CC)C3)=O)C2)ccc2ccccc2c1=O 28335,CC1=C(C(=O)N2CCC(CO)(NC(c3ccc(CC(C)C)nc3)=O)C2)CCO1 28336,c1(C(N2C(CN(C)C(C3CC3(C)C)=O)CCC2)=O)ccc(F)c(O)c1F 28337,c1(C(=O)NCCCC(C)NC(C2(CO)CCCO2)=O)cc2cccnc2nc1O 28338,c1(C(=O)NC2CCCC23CN(C(=O)Cc2cccs2)C3)ccc2nccnc2n1 28339,C1(C)(C(N2CC=CC(NC(C(CCC)=CCC)=O)C2)=O)CCS(=O)(=O)CC1 28340,C(=O)(C(C)(C)CCC(=O)OCO)NCC1CCCN(C(COCC(=O)NC)=O)C1 28341,C1(C(N(C2CC(CO)C2)C)=O)CCOC1C(=O)NC1CCCC1F 28342,C1(COCC)CCCN(C(=O)C(Cn2cccn2)NC(c2ccc(C#N)o2)=O)C1 28343,C(=O)(Nn1nnc2c1CCCC2)C1C2(CC(NC(C(C)(C)OCC)=O)C2)C1 28344,C(=O)(C1=CC2(CCN(C(=O)CN3CCNC3=O)C2)C1)Nc1cn(CC)c(=O)cc1 28345,c1(N(C(c2cccc(Br)c2)C(=O)NCC(F)F)C)cccc(Br)c1 28346,c1(C(=O)NC2C3CN(C(CC(CC)SC)=O)CC32)cccc2c(C)coc12 28347,c1(C(=O)NCC(CCNC(=O)CC2COCC2(C)C)OC)cc2nccnc2[nH]1 28348,C(=O)(CS(=O)C(F)(F)F)NCC(C1CCC1)NC(CNC(CC(C)(C)C)=O)=O 28349,C(CCC(C)(C)C(=O)Nn1nnc(C)c1C)NC(C(CC#C)O)=O 28350,N1(C(C2C(C(C)C)OCCC2)=O)CCN(C(=O)C(C)(C)c2ccsc2)CC(O)C1 28351,CCC(C)C(O)C(C)C(=O)N1CCCC(CCNC(c2cscn2)=O)CC1 28352,N1(C(C2C(OCC)C2)=O)CCCC(C)(C)C1CNC(c1cnn(CC)n1)=O 28353,C1(NC(c2ccnnc2O)=O)C2CC(O)C1N(C(=O)Cn1cnnc1O)C2 28354,N1(C(CC2(C)CC2)=O)CCC(O)(CCNC(=O)Cc2cncc(F)c2)C1 28355,c1(CNCC(=C)Cl)csc(C2OCCO2)c1 28356,C1(C(=O)Nc2c(C)nsc2C)CCN(C(c2cncc(C#N)c2)=O)C(C)(C)C1 28357,c1(C(N2C(CC)C(NC(c3cccnc3)=O)CC2)=O)ccc(OC)c(Cl)c1F 28358,CC1(CNC(C2(CF)CCOCC2)=O)COCCN(C(C2CN(C(N)=O)C2)=O)C1 28359,C1(C(=O)NCCC(C)N(C)C(c2ccc(C3CC3)o2)=O)C2CC(F)(F)CC12 28360,Cn1nnc(N2CCCC2C2CCN(C(=O)CN3CCC3)C2)n1 28361,Cc1nc(N2CCCC(NC(c3cc(C)c(F)cc3C)=O)C2)c2c(n1)CCC2 28362,CCC(C(=O)NC1(C)CCN(C(C2CCN2CC)=O)C1)C(C)O 28363,c1(C(=O)OC)ccc(F)c(C(=O)NCC(C)N(C(=O)COC2CC2)C)c1 28364,N1(C(C(=O)NC2CN(C(=O)OC)CC23COC3)=O)CCCCCC(F)(F)C1 28365,C(=O)(CCC(C)(C)C#N)N(CC(=O)NCC1(C#C)CCC1)C 28366,C=CCC(C)(C)C(=O)NCC1(O)CC(NC(c2nnn(C)n2)=O)C1 28367,C1(CNC(C2(CC)CC2(F)F)=O)CCCN(C(C2(C(C)(C)C)CCC2)=O)C1 28368,C1(C(N2CCC(C(C)NC(=O)CCn3cc(Cl)cn3)CC2)=O)CCCCC(=O)C1 28369,N1(C(C(CCC)(C)O)=O)CC(C)(C)OC2(C1)CN(C(=O)C(C)C(C)COC)C2 28370,N1(C(C=C(CCN(C)C)Cl)=O)CCC2(CCN(C(c3ncccc3N)=O)C2)C1 28371,C1(C(N2CCN(C(c3ccc(C(C)=O)nn3)=O)CC2)=O)CCc2ncncc2C1 28372,c1(N(C)C)ccc(C(N2CC3C(NC(c4nc(Br)c[nH]4)=O)C3C2)=O)nn1 28373,c1(C(=O)NCC2N(C(c3cc(C(C)=O)oc3)=O)CC2)c(Br)ncn1C 28374,C(=O)(C1=NOC(CNC(=O)CC2C=CCC2)C1)N(C(CCO)C(F)F)C 28375,c1(C(=O)NC23CCN(C(c4ccc(C)c(O)c4)=O)CC2C3)nccn2cnnc12 28376,C1(C(N2CCN(C(c3cnc(Cl)s3)=O)C3C2C3)=O)CCc2ccccc2CC1 28377,c1(NC(c2c(SCC)cn(C)n2)=O)ccc(N(C)C)cc1OC 28378,N1(C(C)=O)CCN(C(C2(NC(=O)CC3CCOC3)CCOCC2)=O)CC1 28379,N1(C(C=CCCC)=O)C2CCC1C1CC1(NC(C1CCCC(F)(F)CC1)=O)C2 28380,c1(OC)cc(CNC(=O)C(=O)NCC2CC3CCC2CC3)c(F)cc1F 28381,C(CCC(=O)N(C)CC1CN(C(c2occc2Br)=O)C1)N(C(C)=O)C 28382,Cc1nc(C)c(C(=O)NCCN2CCC(NC(=O)CS(N)(=O)=O)CC2)[nH]1 28383,Cc1ccc2c(C(N3CC=CC(NC(c4cnc(N(C)C)o4)=O)C3)=O)csc2c1 28384,C1(C(=O)NN2CC(NC(c3nccc(CC)c3)=O)C(F)C2)CN2CCN1CC2C 28385,Cc1ncn(C)c(=O)c1C(=O)NCC#CCNC(=O)CSCC(=O)OC(C)(C)C 28386,N1(C(C(C)=C(C)C)=O)CCN(C(c2cc(C#N)ccc2C)=O)C2CCC12 28387,N1(C(c2c(SC)n(C)nc2)=O)CCN(C(=O)COCCOCCO)C(C)C1 28388,C1(OC)CC2(C1)CC(NC(c1cnn(CCNC(=O)CC3CCC3)c1)=O)C2 28389,C1(N(C)C)(C(=O)NCC2C=CC(NC(c3cccnc3S)=O)C2)CCCCC1 28390,N1(C(c2cn(CCC(C)C)nn2)=O)CCC(NC(=O)CCC(C)(C)O)C(C)C1 28391,N1(C(CNC(C)=O)=O)CCCC(N(C)C(C2COCC(=O)N2C(C)C)=O)CC1 28392,C1(C(=O)NCC2CC(F)CN2C(c2cc(Br)c[nH]2)=O)CCCC12CCC2 28393,c1(COc2ccc(NCCCCN3CCC(OCC)C3)cc2)ccc(F)cc1 28394,c1(C(N2CC3C(NC(c4c(CC)nco4)=O)(CC3)C2)=O)cc(N)c(C)cc1Cl 28395,c1(C(N2CC(NC(CN(C)CC)=O)C3(C2)CC3)=O)cc(C)c(C)cc1C 28396,c1(NC(CC)COC)ccc(S(=O)(=O)NCC(N2CCOCC2)C)cc1Br 28397,c1(OC)ncnc(N(C2CNCCOC2)C(c2cc(SC)oc2C)=O)c1C 28398,C(=O)(CS(=O)(=O)CC1CCCO1)NC1(CNC(C(C)n2cncn2)=O)CCC1 28399,c1(C(=O)NC(C2CCOC2)C#C)oc(CNC(=O)CNC(=O)CC)cc1C 28400,N1(C(c2ncc(-c3c(C)cnc(F)c3)nc2)=O)CC2CC(C1)c1ccccc12 28401,c1(C(=O)N(C(C2CCC(F)(F)C2)C(=O)OCC)CC)cc2ccsc2n1C 28402,C1(C(=O)NCCC2CN(C(C3(C)CC4CC4C3)=O)C2)CCC2(CCCO2)CC1 28403,n1(CC(=O)NC(C2CCCN2C(=O)CC2CCNC2=O)C2CC2)ccsc1=N 28404,CC1CC2(CC(C(=O)NCC(O)C(=O)NC3(CO)CC=CC3)C2)C1 28405,C1(CNC(CCC2(NC(CSC)=O)CCCC2)=O)CCCCC1(C)C 28406,C1(N(C(C(CSC)C)=O)C)CN(C(c2c(O)cccc2F)=O)CC12CC2 28407,CCC(c1ccc(C)cc1)=CC(N1CCN(C)CC1CNC(=O)CSC(F)F)=O 28408,c1(CCC(N2C(C(=O)NC3(CC)CCOC3)CCCC2)=O)ccc(OC)c(F)c1 28409,N1(C(C(C2CC(NC(C3CS(=O)C3)=O)C2)F)=O)CC(O)(CC2CC2)C1 28410,C1(NC(c2cn(CCC)nc2)=O)CCCCCC1NC(=O)C(F)(F)c1cncs1 28411,C(=O)(CC(F)(F)C(F)F)NC1CCCC(CC(=O)NCc2c(C)nc(C)s2)C1 28412,c1(CC(=O)NCCC2CC(NC(c3c(CC)c[nH]n3)=O)C2)cccnc1OC 28413,C(=O)(C(CC(C)C)N(C)C(c1ccc(O)nn1)=O)NC(CC#C)C(N)=O 28414,c1(OC)cc(C(N2CCC(C)C(CNC(=O)CC3=CCCC3)C2)=O)oc(=O)c1 28415,N1(C(C(C)=C(CC)C)=O)CCC2(CCC(CNC(=O)CN3CC(C)(C)C3)O2)CC1 28416,C1(CNC(C(CCC)OCC)=O)CN(C)CCN1c1cnc(C#N)cn1 28417,C1(C(C)NC(c2cc(Cl)c[nH]2)=O)CCCCN1C(=O)CCc1cccs1 28418,N1(Cc2cc(C)on2)CCC(NC(C2CCC3CCCCN23)=O)C(C)(C)C1 28419,CC1COCCC1NC(C1CC12CC(NC(C1(c3cc[nH]n3)CC1)=O)C2)=O 28420,N1(CC(=O)NC(C)(C)C(F)F)CCN(C(C2SCCS2)=O)CC1 28421,c1(C(=O)NCCCN(C(C=CC(C)C)=O)CCO)cscc1OC(F)F 28422,c1(OC)ccccc1OCC(=O)NCC(O)CN(C(=O)C1=CCSC1)C 28423,C1(NC(=O)CNC(C2CCCCC2)=O)COCCC1C(N1CCCC1)=O 28424,N1(C(C2C(C)CC2)=O)CCOC(CC(=O)N(C2CCCCC2)CCO)C1 28425,N1(C(C=C2CCN(C)C2)=O)CCC2CN(C(C3CC(N4CCOCC4)C3)=O)CC12 28426,Cc1cc(C(=O)NCC2C3CCC(C3)N2C(c2cnc(Cl)cn2)=O)cc(F)c1 28427,N1(CCCC2C(C)C2)CC2(CO)CC2(CO)C1 28428,c1(C(c2nnnn2CCCF)NC(COC)(C)CCO)cnc2cc(Br)ccn12 28429,c1(NC(C2C3(CC(NC(c4ccn(CC)c4C)=O)C3)C2)=O)cccc2occc12 28430,C1(CC(=O)NCCC(=O)OCC)C2CC(C2)N1C(c1cc(C)oc1C)=O 28431,Cc1cc(C(N2CCCC(C(N3CC(C(C)(C)C)C3)=O)CC2)=O)cc(O)c1 28432,c1(NC(C2(C)CN(Cc3cccc(C=O)c3Br)C2)=O)csc2nccnc12 28433,N1(C(C(C=C)(C)C)=O)CCN(C(=O)CCN2CCC(F)C2)C(CC(=O)NC)C1 28434,c1(CSCCNC(C2C(c3ccccc3)CCC(=O)C2)=O)nnc2ccccn12 28435,C1(NC(C2N(C(c3c(C)cc(CC)o3)=O)CCC2)=O)C(=O)NCCC1C 28436,C#CCC(C(=O)NOCC=CC)NC(=O)Cc1cn(C)cn1 28437,c1(OCCC)ccc(C(=O)NCc2ccc(CO)c(F)c2)cc1C 28438,c1(CC(=O)NC(C)CN(C(=O)CNC(c2cn[nH]c2)=O)C)csc(NC(C)C)n1 28439,C1(NC(C2CN(CC)C(=O)CC2)=O)CN(C(=O)CSC(C)C)CC2(CC2)C1 28440,c1(C(=O)NCCC(C)N(C)C(c2cccnn2)=O)csc2ccc(F)cc12 28441,c1(CNC(C(N2C(C#N)CCC2)c2ccc(CO)cn2)=O)ccc2c(c1)CCC2 28442,C(C1=NOC2CN(C(=O)C#CC3CCOCC3)CC12)NC(c1c(C)scc1)=O 28443,c1(C(=O)NCC2(O)CCN(C(C3(C#N)CC3)=O)C2)ccc2ncnn2c1 28444,C1(C)(NC(CNC(CNC(c2cnc(C(C)C)o2)=O)=O)=O)CCCC1(C)C 28445,CCCCC(C)CCC(=O)NC1COCC1(C)NC(=O)OC(C)(C)C 28446,N1(C(c2cc(C)sc2C)=O)CC(C)OC2(CCN(C(C3CC3C(C)C)=O)CC2)C1 28447,c1(N2CC(C(=C)C)OCC2)nc(=NCCc2ccoc2)[nH]c2c1cnn2C 28448,C(=O)(C1CCCc2c1ncn2C)NCC(C)(CO)NC(c1cc(C)on1)=O 28449,N1(C(c2ccc(CSC)o2)=O)CCC(NC(C2CCN2C(C)(C)C)=O)C1C 28450,c1(Cn2cc(C3CC(NC(C4(CC)CCCC4)=O)C3)nn2)cc2n(n1)CCCO2 28451,c1(OC)cc(C(N2CC(NC(c3ncc(C)nc3OC)=O)C(C)C2)=O)c(F)cn1 28452,C1(CC(=O)NCCNC(C)=O)CC2(C1)CN(C(c1cc(C)cs1)=O)C2 28453,C1(NC(C2CC(OC)C2)=O)CC2(C(=O)NCC(C)CN(C)C)COC1C2 28454,C1(C(N(CCN(C(C)C)C(c2ncc(Cl)n2C)=O)C)=O)CCC2CC2CC1 28455,N1(C(c2scc(NC(=O)OC(C)(C)C)n2)=O)CCC(C2CCC(=O)N2)CC1 28456,N1(C(C2CC(CC)N(C(=O)Cc3cn(C)cn3)CC2)=O)CCC(F)(F)C(O)C1 28457,CCCCC(C)(F)C(=O)N(C)CC1(O)CCN(C(=O)C=Cc2cccc(F)c2)C1 28458,c1(C(=O)O)ccc(CCNC(=O)C(C2CCNCC2)F)cc1 28459,C1(CNC(CCCn2cc(-c3ccc(C(=O)O)s3)nn2)=O)CCCOCC1 28460,N1(C(c2c(OC)cnnc2)=O)CCC2(CCN(C(=O)C(N=[N+]=[N-])C(C)C)C2)C1 28461,C12(CCS(=O)(=O)CC1)C(=O)N2.c1(CC(C(=O)NCC2CCC2)N)ccc(Cl)cc1Cl 28462,n1(CC)cnc2c(NCCc3cc(F)c(F)c(F)c3)[nH]c(=NC(C)CF)nc12 28463,c1(CC)cc(CNC(=O)C(c2ccc(-c3nn[nH]n3)cc2)O)cc(F)c1 28464,c1(C(=O)NCC(CN(C(c2ccc(C(F)(F)F)o2)=O)CC)(C)C)cnnc(C)c1 28465,C#CCCCCC(C(=O)Nc1ccccc1C)N(C)Cc1cc(C)n(C)n1 28466,C1(NC(c2scc(C)c2)=O)CN(C(c2ncncc2Cl)=O)C2(CCOCC2)C1 28467,C(COC)(CCCC)NC1(C)CN(C(C=CCOC)=O)C1.C1C(=O)N1 28468,C1(CCNC(CN(CC)CC)=O)COCCN1C(c1ccn(CCF)n1)=O 28469,C(=O)(C1=C(Cl)CCC(C)C1)N(CCN(C(CC(C)P(C)(C)=O)=O)C)C 28470,C(=O)(CS(=O)(=O)CC(C)C)N1CCN(C(c2ccc(C)nc2)=O)C(C(C)C)C1 28471,Cc1ccccc1-n1cc(C(N2CC(NC(C3(C(F)F)CCC3)=O)C2)=O)nn1 28472,CCN=C(NCc1ccc2c(c1)OCO2)N1CCC(O)CC(C)(C)C1 28473,N1(C(C23C(CN(Cc4cccc(N(C)C)c4)C2)C3)=O)CC2CCCC2C1 28474,c1(CC(=O)NCCC(C)NC(=O)CCCCN(C)C(C)C)ccc2c(c1)CCO2 28475,c1(C(=O)NCC2CCC(NC(CCCOC(C)C)=O)C2)ccc(C(F)(F)F)cc1 28476,N1(C(c2c(C)n(C)nc2)=O)CCCC2(CCN(C(c3cc(N)cc(O)c3)=O)C2)C1 28477,C1(NC(c2n(CC)ncc2)=O)CC2CN(C(c3cccc4c[nH]nc34)=O)CC2C1 28478,C1(CNC(COC2CN(C(C3C(C(C)C)C3)=O)C2)=O)CCCCC1C 28479,C1(NC(C2C(=C)C2C(=O)OC)=O)CC(CO)N(C(=O)C(C)CC2CC2)C1 28480,c1(CCC2(C(=O)N(CCOCCNC(=O)CO)C3CC3)CC2)ccccc1 28481,N1(C(C(C)CC2CCC2)=O)CC2CCC1C(NC(=O)CN1CCS(=O)(=O)CC1)C2 28482,C1(NC(CCCOC)=O)CS(=O)(=O)C2CN(C(C3CC4CC3CO4)=O)CC12 28483,C(=O)(C(CO)C(C)(C)C)NCCCN(C(c1cnn(CC)c1C)=O)CC 28484,c1(COC)nc(N2CC(CNC(=O)CN3OC(C)(C)CC3=O)CC2C)cc(O)n1 28485,C1(CC)CCCN(CC(=O)NC2CCC(NC(c3cc(C4CC4)[nH]n3)=O)C2)C1 28486,CCCC(C)CCCC(=O)N1CC2(CCCN(C(c3cn4ccnc4s3)=O)C2)C1 28487,CC1=CCCN(C(C2CC(=O)CN2C(C2CC(O)C(F)C2)=O)=O)C1 28488,N1(C(C(COC(C)C)NC(C)=O)=O)CCC(C(=O)NC2(C(C)C)CCC2)C(O)C1 28489,c1(CCC(N2CCC(O)(CNC(C3(C)CSC3)=O)C2)=O)cc(F)cc(F)c1 28490,N1(CCC(=O)NCCOCCNC(CCCOCCOC)=O)CCCCCC1 28491,c1(C(=O)NCC(C2CCCC2)NC(c2cnn(C)c2Cl)=O)c(F)cc(Cl)cc1F 28492,N1(C(CCC=C)=O)CCN(C(=O)CNC(=O)C=Cc2ccco2)CC1CC(F)F 28493,O=C1NCC2(CO1)CN(C(c1ccc(CNC(C3(CO)CCCO3)=O)cn1)=O)C2 28494,C1(CC)CCCCCCN1C(C1CCCC1NC(c1ccncc1)=O)=O 28495,CCCC(CC)C(=O)NCC1(F)CCCN(C(c2cc(O)ccc2Br)=O)C1 28496,N1(C(c2c(CC)nc[nH]2)=O)CCC(CO)(CNC(c2ccccc2C(F)F)=O)C1 28497,N1(CCC(=O)NC2(C)CN(C(C3CCCC34CCC4)=O)C2)C(=O)NC(C)(C)C1=O 28498,N1(CCNC(C(C)CC2CC2)=O)CCC(NC(C2CCOC2(C)C)=O)CC1 28499,Cc1nn(C)cc1C1OCCC1NC(C1CCCCN1C(c1ccnn1C)=O)=O 28500,c1(C(C(=O)NCc2ccoc2)N(C2CCOC2)C2CC2)ccc(Br)cc1 28501,C(C(C)(C)CN=C(NCC1(c2ccccc2C)CC1)NC1CCS(=O)(=O)C1)OC 28502,C(C)(C(C)C(=O)N(C)CCc1noc(C)n1)NC(CSCCOC)=O 28503,C1(COC)CC(CNC(=O)C(C)Cc2ccnn2C)N(C(c2cccn2C)=O)C1 28504,Cc1ccc(CN2CCC(CNC(c3ccn(C4CCC4)n3)=O)C2)o1 28505,c1(C(=O)NCC(C)CNC(=O)CNC(C2CCCC2)=O)coc(Br)c1 28506,CC(C)CC(C(=O)NC(CC1CC1)C(=O)NCCCc1cnn[nH]1)C(N)=O 28507,C12(C(N(C)CC)=O)CC(CN(C(c3cnn4c3CCC4)=O)C1)C2 28508,CCCC(C)(CC)C(=O)NC(C)CCNC(=O)C1=CSCS1 28509,c1(C(N(CCCNC(C=Cc2n(CC)ccn2)=O)C)=O)cc2c(s1)CCCC2 28510,C12(CC(N3C(COC)(CNC(c4ccn(C)c4)=O)CCC3)=O)CCC(CC1)OC2 28511,C(CC(=O)N1CCN(C(c2ccc(C)nn2)=O)C(C(F)F)C1)(C(F)(F)F)OC 28512,C1(CC)(CC)CC(C(=O)NC(C)CC(C)NC(=O)CN(C)C(C)=O)C1 28513,C1(NC(C2C(C)C2)=O)CN(C(C2(C)CCN(CC(F)F)CC2)=O)CCC12CCC2 28514,CCCC(C)(CC)C(=O)N1CC(CC(N2CCCC2CC(C)O)=O)(OC)C1 28515,C(C)(C)(CN=c1[nH]c2ccccc2o1)NC(C(C(CC)C)O)=O 28516,c1(CSCC(=O)NCCN(C(C2CCC(CO)CC2)=O)CC)ccc(C#N)cc1 28517,c1(C(=O)NCC23CC(NC(CC)=O)(C2)C3)ccnc2[nH]c(CC)nc12 28518,Cc1cncnc1C(N1CCCCC1CNC(=O)CC1CC(=O)NC1=O)=O 28519,N1(C(CN(C)CC)=O)CCC2(C=C(C(=O)NC3CC(CSC4CC4)C3)C2)C1 28520,CCCC(CNC(C1CCCCCN1C)=O)C(=O)NCCc1ccnn1C 28521,N1(C(c2csc(C)n2)C(=O)NC(CC)C)CCC(CSc2cnn(C)c2)CC1 28522,CC1CC(CCNC(=O)CCOC2CC2)CCN1C(=O)CC(Cl)Cl 28523,Cc1cc(C(=O)NCC2(C(=O)NCCN3CCCC3)CC=CC2)ncc1F 28524,CC(C)CC(F)(F)C(=O)NC1CCCCC1NC(C1(NC(N)=O)CCCCC1)=O 28525,C1(NC(C(CCCCC)O)=O)CCN(C(c2ncc(C)cc2C)=O)CC12CCC2 28526,C1(CNC(c2coc(CO)c2)=O)OCCC1C(=O)NCCCC1CCOC1=O 28527,CC1CCC(CNC(=O)CC(C2CC2)NC(=O)CCc2ccnn2C)C1 28528,c1(OC)ccnc2c(Nc3ncn(C4CCC(N)CC4)n3)cccc12 28529,C(=O)(C(C)(O)C(C)(O)C(=O)OC)OC.c12csc(n1)COC2=O 28530,N1(C(c2c(CC)scc2)=O)CCN(C(=O)COC2CC2(F)F)CC1C1CC1 28531,CC(C)C(CNC(c1cc(Cl)on1)=O)NC(C1(CO)CCCO1)=O 28532,Cc1ccc(N)c(C(=O)N(CC(C)(C)CNC(=O)CC2CCC(C)(C)C2)C)c1 28533,C(CNC(=O)Cn1cc(C)cn1)(CC(=O)NCCn1nncc1C)OC 28534,c1(C(=O)NC2(C)CC(NC(=O)Cn3cnc(C(N)=O)n3)C2)ccc2oncc2c1 28535,c1(OCC(=O)NC)cc(CN2CCC(CO)CC2)ccn1 28536,N1(C(C2(OCCNC(C=CC=C(C)C)=O)CCC2)=O)CCC12CCCC2 28537,N1(C(CCOC(C)=O)=O)CCCC(C(N2CCC(N3CCCC3)C2)=O)CC1 28538,c1(C(=O)NCC(CCOC)NC(=O)Cn2cccc2)ccn(C(C)C)c1C 28539,Cc1cccc(C(O)C(=O)NC2CC2NC(=O)CCC2(C)CC2)c1 28540,C1(C(=O)NCC2C(C)C2C)CN(C(C2C(C)(C)C2(F)F)=O)CC1(F)F 28541,C(=O)(C(C)(C)C(C)O)N(CCNC(C1CC1c1ccnn1CC(C)C)=O)CC 28542,CCC(CCC(=O)NC1C=CCN(C(=O)CCc2ccc(C)s2)C1)OC 28543,Cc1csc(=O)n1CC(=O)NCC1CC(C)N(C(=O)C=CC(C)(C)C)C1 28544,CCC(C)CC(=O)C(=O)N1CCC2(CC(C(N3CCOC(C)C3C)=O)C2)C1 28545,c1(C(=O)NC(CN(C2CCCN(C(C(C)C)=O)C2)C)=O)ccc([N+](=O)[O-])cc1 28546,C1(C)(N)COC(C)(C)CO1.CCN=C(NCCCN(C(=O)OC)C(C)C)NC1CC1 28547,Cc1n[nH]cc1CNC(C1OCCC1CNC(C1(C)CCC1)=O)=O 28548,n1(CC)nnc2cc(C(=O)NCC(O)CNC(C3COC3)=O)ccc12 28549,C1(CC)CN(C(c2ccc([N+](=O)[O-])s2)=O)CCN1C(C1CCN(C)CC1)=O 28550,C(=O)(C1=CCCOC1)NCC(C1CCCC1)NC(C1(CCC=C)CC1)=O 28551,C=CCCC(F)(F)C(=O)NCC1CN(C(c2cnn(CCC)c2CC)=O)CCO1 28552,c1(C(=O)NCC2C(NC(c3c(OCC)cccn3)=O)C2)cc2cc(O)ccc2[nH]1 28553,c1(C(N(C2CCN(C(=O)CSC3CC3)C2)CC#C)=O)cc(Cl)n(C)n1 28554,N1(c2nc(CC)nc(Cl)c2CC)CC(NC(=O)C(O)C(C)C)C2(CCOCC2)C1 28555,C1(C(N2CCC(c3cccc(Br)c3)CC2)=O)CC2CC2N1C(C1CC1F)=O 28556,Cc1nn(C)c2ncc(NC(=O)NCCCOc3c(F)cccc3Cl)cc12 28557,c1(SC)ccc(CC(=O)NC2CCCC(NC(=O)Cc3ccc(Cl)cn3)C2)cc1 28558,C1(O)(CCNC(C(COC)OC)=O)CCCN(C(=O)CCC(C)(C)OC)C1 28559,c1(C(N(C(CN(C(C(CC=C)CC)=O)C)C)C)=O)cccn2nccc12 28560,C1(C(C(=O)NCCC(C)N(C(=O)CC2(C)CC2)C)OCC)CC(F)(F)C1 28561,C(CC(=O)NC1CCCN(C(N)=O)C1)(C(N)=O)N(C(=O)CN1CC2CC2C1)C 28562,c1(OC)cnc(Cl)c(NC(C2CCN2Cc2ccc(C(C)(C)C)cc2)=O)n1 28563,c1(CN(C)C)cc(O)c(Br)cc1O.C12CN(CCC1O)CC1CN(CCO1)C2=O 28564,c1(C(=O)NC2(c3c(C)cccc3)CCC2)cccc2nscc12.n12cc(nn1)C2 28565,C(=O)(CC(F)(F)F)NC(C)C(=O)NC1(CNC(=O)CC2(C)CCCC2)CCOC1 28566,c1(C(=O)NC(C2CCN(C(c3ccnc(C(F)(F)F)n3)=O)C2)C)cncc(N)c1 28567,c1(OC)cc(C(=O)NC(CNC(C2CC(=C3CC3)C2)=O)C2CC2)c2occc2c1 28568,C(=O)(CC(O)c1ccccc1)NCCC(C)N(C)C(C1(C)CCCC1)=O 28569,CCC(C(=O)N1CC(CN(C)CC)C1)N(C)C(C1CC(CC(=O)OC)C1)=O 28570,c1(C(N2C3C(NC(CSCC#C)=O)CC(C3)C2)=O)cccc2nccnc12 28571,c1(C(=O)NCc2ccsc2C(N2CCC2C2CCC2)=O)n[nH]cc1[N+](=O)[O-] 28572,C(=O)(C(F)(F)F)NN(C(C)C(=O)NCCCN(C1COC1)C1CC1)C(C)=O 28573,CCC(C(=O)NCC1CN(C(c2ccc(C)c(CO)c2)=O)CC1(F)F)C(C)C 28574,c1(NC(C)=O)c(C(N2CCC(NC(=O)Cn3cccc3)C2C)=O)cccc1C 28575,C#CC1CN(C(=O)CCc2cn[nH]c2)CCN1C(c1cnc(O)o1)=O 28576,CN1CCC(C(=O)N2CC(NC(=O)C3=CCCC3(C)C)C2)c2ccccc21 28577,c1(C(N(C)CC2C3CN(C(CN(C(C)=O)C)=O)CC32)=O)ccc(F)c(C(F)F)c1 28578,C1(N2CCOCC2)(CNC(=O)Nc2nc(N(C(C)=O)CC)sc2)CCN(C)CC1 28579,N1(C(C2(C(C)C)COC2)=O)CCOCC(NC(=O)C(C)Oc2ccccc2)C1 28580,C1(CNC(CC2CC(C(=O)OC)C2)=O)CCCCN1C(=O)COCP(C)(C)=O 28581,N1(C(CCC=C(C)C)=O)CCOC2(C1)CN(C(=O)C(C)Oc1ccccc1)C2 28582,CC1CCC(C)(C(N2CC3(CC(NC(c4[nH]cc5c4CCC5)=O)C3)C2)=O)CC1 28583,Cc1ccnc(O)c1C(=O)NCCC1CC(N)C1 28584,n1(CC(=O)NCC2(CO)CCN(C)C2)c(=O)c(F)cn(-c2ccccc2)c1=O 28585,S(=O)(=O)(c1ccc(C)c(C)c1)N1C2(CNC(C(CCCC)O)=O)CCC1CC2 28586,C1(NC(c2c(CC)oc(C)c2)=O)C2CC3C1C3C2C(N1CCC1C(C)(C)O)=O 28587,CC1CN(C(=O)CCC2CCCOC2)CC1(C)C(=O)NC1CC2CCC1O2 28588,Cc1ccc(O)c(CC(N2CCN(C(c3nc(O)sc3C)=O)C(C)C2)=O)c1 28589,CC1CCCCCN1C(=O)CSCCNC(c1cncc(F)c1)=O 28590,N1(C(c2cccc(N3C(=O)NCC3)c2)=O)CC2(CO)CCC2(CO)C1 28591,c1(C(=O)NCC2(CNC(C(c3cncnc3)C)=O)CCC2)ncc(Cl)cc1F 28592,C1(C(N(C)CCNC(C2CCC(C(F)(F)F)CC2)=O)=O)CCc2nnc(O)n2C1 28593,C1(NC(CSC(C)C)=O)CC2CN(C(=O)CN3CC(=O)NC3=O)CC2C1 28594,C1(C)(NC(CC2OCCN(C(C3CCN(C)CC3)=O)C2)=O)CCC(C)(C)C1 28595,CCC(CCCO)NC(=O)C(CO)NC(=O)CC(C)=C(C)C 28596,c1(CC(=O)NC(CC2CN(C(c3cc(C)oc3)=O)C2)C)cnc(Cl)cc1C 28597,C1(O)(CC(=O)N(C(C)CNC(=O)C(c2ccc(Cl)s2)C)C)CCCCCC1 28598,CC1=C(C(=O)N2CCC(N(C)C(c3ccncc3F)=O)CC2)CCC1 28599,c1(C(N2C(C)(C)CC(NC(C34CCCC3C4)=O)C2)=O)cc(F)cc2nn[nH]c12 28600,C1(NC(c2nnc(C)s2)=O)C2CC1CN(C(C1CC1C1CCCC1)=O)C2 28601,C(=O)(C(C)(C)CS(N)(=O)=O)N1C(CNC(c2ccc(COC(C)=O)cc2)=O)CC1 28602,C1(O)(CCNC(c2csc(O)n2)=O)CN(C(c2ncoc2Br)=O)C1 28603,c1(C(=O)NC(CC)(C)CNC(c2nn(C)cc2Cl)=O)cc(C)n(CCOC)c1C 28604,CC1(C(=O)N2CCC(C(C)(C)NC(c3cn[nH]c3)=O)C2)COc2ccccc21 28605,C(=O)(CCS(=O)(=O)CC(C)C)N1CC(NC(Cc2cc(C)on2)=O)C(CO)CC1 28606,c1(C(=O)NC(CC=C)CNC(c2cnc(C(F)F)nc2)=O)cc2n(n1)CCC2 28607,CC(Cc1cccn1C)N=c1ccnc(NC2CCC(=O)NC2)[nH]1 28608,N1(C(C(C)OC)=O)CCC(O)C2(CCN(C(c3ccn4ccnc4c3)=O)CC2)C1 28609,c1(C(=O)NC2C(CNC(c3ccn(CC)n3)=O)CC2)ccc(=O)n(CCOC)c1 28610,CC(=NO)C1CC(C(N2CC(NC(=O)CSCc3cccs3)C2)=O)C1(C)C 28611,Cc1cccnc1C(=O)NC1(CCO)CN(C(c2cncc(C(C)(F)F)c2)=O)C1 28612,N1(C(c2c(CNC(CC=CC=C)=O)n[nH]c2)=O)CCc2ccncc21 28613,Cn1nc(C(=O)NC2CC2NC(C2CC3(CC3)CO2)=O)cc1C1CC1 28614,c1(-c2ccc(CN3CCN(CCC(=O)OC)CC3)cc2)ccc(Cl)c(CO)c1 28615,c1(C(N(C(CN(C)C)(C)C)C2CC2)=O)ccccn1.C1CC(=O)N1 28616,C1(C(N(CC(C)O)CCNC(=O)C(C)(C)C)=O)CCn2nccc2C1 28617,c1(C(N2CCC(CC)C2)=O)ccncc1N(C)C.C1(O)COCC1CN(C)NC(CC)=O 28618,c1(C(=O)NCC23C(CN(C(CC=CCC)=O)C2)C3)ccc(F)c(C(F)(F)F)c1 28619,C1(CNC(C(C)c2cccs2)=O)CC(C(F)(F)F)CN1C(N)=O.n12cc(nn1)C2 28620,c1(C(=O)NCC2N(C(CC(C)C)=O)CC(C)CC2)cccc2cc[nH]c12 28621,C(CC(=O)N1CC(N(C)C(C23CCC(C)(CO2)C3)=O)C1)(C(C)C)OCC 28622,c1(-n2ccc(C)n2)ccccc1C(=O)NCC(F)CNC(C1CCOCC1)=O 28623,C1(C(N2CC(NC(c3cc4c(s3)CCC4)=O)C(F)C2)=O)CC2(CCCC2)C1 28624,N1(C(Cc2cncc(C)c2)=O)CC(F)(F)CC1CNC(c1nc(C)ccc1C)=O 28625,c1(C(N(CCN(C)CC2CCC(C)(C)CC2)C)=O)occ2c1CCC2 28626,N1(C(C2C(CCC)C2)=O)CC(NC(=O)C=C2CCCCC2(C)C)C2CCCC12 28627,c1(C(=O)NC2CC(NC(C3C(C)(C)COCC3)=O)C2)ccc2cc[nH]c2n1 28628,O=C1CC(NC(=O)CN2CCCCC2c2ocnc2C(=O)O)C(=O)N1 28629,C(C(=O)N1CCC(C=C)CC1)(C(C)(C)O)NC(CC(=O)NCC#C)=O 28630,CC1(NC(=O)Cc2ccn(C3CC3)n2)CCN(C(=O)CCCn2cccn2)C1 28631,c1(OC)snc(C)c1NC(=O)NCC1CCN(C(C2CCCN2C)=O)C1 28632,C1(CC)CCC(C(=O)N(C2(C(N3CC(C(F)(F)F)C3)=O)CC2)C)CC1 28633,C1(CNC(COCC(=O)NC)=O)CN(C(=O)CCc2ccc(NC)cc2)CCO1 28634,c1(C(N(CCN(C(C(C(=O)OC)OC)=O)C)C)=O)ccc(C(C)C)c(C)c1 28635,C1(C(N2CC(c3cn(CC(COC)O)nn3)(O)C2)=O)CCC(C(=O)OC(C)C)CC1 28636,n1(C2CC(C)OC2)ncc2cc(-c3ccc(C(=O)OCC(F)(F)F)cn3)cnc12 28637,CCC(C(C)(F)F)C1CCN(C(=O)CCCOCCN)CC1 28638,C#CCCCCC(=O)N(C)CC1(NC(=O)CC2CCCS(=O)(=O)C2)CC1 28639,N1(C(C2(OCC)CCC2)=O)CCCCC1CNC(=O)C(c1cccc(F)c1)O 28640,Cc1cn2cc(C(=O)N(C3CCN(C(=O)C4=COCCC4)C3)C)sc2n1 28641,C1(C(=O)NC(C=C)CO)CCCCN1C(c1cncn1C(C)C)=O 28642,c1(C(=O)NCC(CN(C(C(C)N(C(C)=O)C)=O)C)(C)C)cccc(CS(C)=O)c1 28643,C1(CC(=O)OC)CN(C(CC2CCC3CC23)C(=O)NC2CC2)CC(C)O1 28644,CC1(C)CC1(S(C)(=O)=O)C(=O)OCc1cc(Br)cc(I)c1 28645,Cc1cnc2cc(C(N3C4CCC3CC(CNC(=O)COC(C)C)C4)=O)ccn12 28646,c1(C(=O)NCC(c2ccc(OC)cc2)O)c[nH]c2cc(-c3nn[nH]n3)cnc12 28647,C(=O)(CC(C(F)F)C(C)(C)C)NCCCN(C(c1cccc(OC)c1)C)CC 28648,c1(C(=O)NC(C2CCCN(C(COCC(=O)NC)=O)C2)C)c[nH]c(=N)nc1C 28649,C1(C(=O)NC(C)(C)CNC(c2[nH]ccc2-c2ccccc2)=O)CCC2(CCC2)O1 28650,C(C)(C(=O)N(C(C)CO)C)N(C(=O)C=CCC1CCC1)CC 28651,c1(C(=O)NC(C2CCCN(C(C(C=CCCC)O)=O)C2)C)ccc(N)c(Cl)c1O 28652,c1(C(=O)NC(C)CC(F)(F)F)cc(NCC=CCO)ccc1Cl 28653,C(=O)(CC(CC)CC(F)(F)F)NCC1CCCCN(C(CC(=C)C)=O)C1 28654,N1(C(C=COCC)=O)CCCC2(CCC(NC(c3cc(C)c(C)nc3O)=O)C2)C1 28655,n1(CC)nccc1C(C(=O)NC1CCOCC1)N(C)C(C1CCCC1)C 28656,c1(C(=O)NC2CC3(C(NC(CCCC4C(C)C4)=O)C3)C2)cccc2c1C(=O)NC2 28657,Cc1cc2[nH]c(C(=O)NCC(C3CC3)NC(C34CC(C3)C4)=O)cc2s1 28658,C1(NC(c2c(C(C)C)ccs2)=O)CC2CC(NC(c3cnco3)=O)CC2C1 28659,c1(OC)nc(C(C(=O)NC(C)(C)C)N(C)Cc2cccc(C(C)(C)C)c2)sc1C 28660,C12(C(=O)NC3CC(N(C(CCCCCOCC)=O)C)C3)CCC(CC1)C2(C)C 28661,N1(C(C)=O)CCc2cc(C(=O)NCC(C)NC(C3(c4nc[nH]n4)CCC3)=O)ccc21 28662,N1(C(c2c(C)ccc(C)c2)=O)CC2CCC(C1)C2NC(=O)CC1CCC(C)CO1 28663,c1(C(=O)NCC2(C)C(C)CN(C(=O)C=Cc3cocn3)C2)nnn2c1CCCC2 28664,CC1CN(C(c2nc(C3CC3)cs2)=O)CC(CCNC(=O)COCC(F)F)O1 28665,C1(C(N2CCOC(CCCNC(C3CC3F)=O)C2)=O)(OC)CCC(C)CC1 28666,C(=O)(C(C)(F)C(=O)OC)N(C1CCN(C(C(CC#C)C)=O)CC1)CC 28667,Cc1ccc2c(c1)CC(C(=O)NCC(C)N(C(=O)CCSc1nccn1C)C)O2 28668,N1(C(C2C(NC(CC(CC(C)C)C)=O)CCO2)=O)CC2C(=O)NC(=O)C2C1 28669,Cc1sc(C(=O)NC2CCN(CC(=O)NC3CCCCC3)C2)c(C)c1Br 28670,N1(C(CCC=CC)=O)CCOC(C)C1C(=O)NC(C)C(=O)N(C)CC 28671,C(=O)(CCCCCOC1CCCC(C(N)=O)C1)NC(C)(C)C 28672,C=C(C)C(C)(O)C(=O)N1CC(N(C(=O)C=Cc2ccc(Cl)cc2)C)C2(CC2)C1 28673,N1(C(Cn2c(C)c(Cl)cn2)=O)CCC2(CC1)CC2NC(=O)C(C)CC(C)C 28674,N1(C(c2cc(Br)co2)=O)CCC2(CO)CN(C(c3ccnc(O)c3)=O)CC2C1 28675,CCC(CC(=O)NC(C)(C)C(C)CC(=O)N1CC(CC)(CC)C1)C(F)F 28676,c1(C(=O)NC(CCCC)CNC(=O)CNS(=O)(=O)NC)coc2c1C(=O)NCC2 28677,N1(C(C(C)=C(C)C)=O)CCN(C(=O)C(C)S(N)(=O)=O)CC1CCO 28678,C1(NC(COCCCOC)=O)CCN(C(C2CC2C2CC2)=O)CC1F 28679,C(C)(CNC(c1nnsc1C)=O)(CC(C)C)NC(CCCC)=O 28680,Cc1c(C(=O)NC(C)(CNC(=O)CCC2CC2(C)C)CO)nnn1C(C)C 28681,c1(C(=O)OC)ccc(CNCC2CCCC2N)cc1Cl 28682,c1(C(=O)NC(C)(Cc2ccncc2)C(=O)O)ccc([N+](=O)[O-])cn1 28683,C1(C(=O)NC2C(COC)(CO)C2)CN(CO)CC12CCC2.C1(C(=O)N)CC(CO)C1 28684,N1(C(=O)NC2CC(c3ccc(Br)cc3)C2)CCC12CC1CCC2C1 28685,C1(C)(C(N2CCC(NC(CCC(CC)OC)=O)CC2)=O)CC2CCC(C1)S2(=O)=O 28686,c1(C(=O)NCC2(NC(CC(=O)NCC#C)=O)CC2)ccc2c(c1)C(=O)CCC2 28687,C(=O)(CCCC(=O)OC(C)(C)C)NC1CCCC(N(C(c2c(C)coc2)=O)C)C1 28688,N1(C(C(OCC)OCCCO)=O)CCCC(c2nn[nH]n2)(OCC)C1 28689,C1(NC(c2cc(C)c(C)[nH]2)=O)CS(=O)(=O)C12CCN(C(=O)C(C)(Cl)Cl)CC2 28690,c1(C(=O)NC2CC(OC)CN(C(c3c(Cl)n[nH]c3C)=O)C2)c(C)cc(C)nc1O 28691,c1(-c2ccc(OCCN(C)C)cc2)ccc2c(C(=O)NCC3CCO3)cnn2c1 28692,c1(C(C(=O)NCCCC)NC(C2CCN2C(C)(C)C)=O)cccnc1 28693,C(=O)(CC(F)(F)C(F)F)NC(C1N(C(CCN(CC)CC)=O)CCCC1)C 28694,C1(NC(C(CCC)O)=O)CCN(C(c2cc(NC(C)=O)ccc2C)=O)C12CC2 28695,c1(C(C(=O)NC2CC(CCNC(C=C(C)C)=O)C2)=O)ccc(O)cc1 28696,CCCCC(CC)C(=O)N(CC(N1CCC2(CSC2)C1)=O)CC(C)C 28697,C1(C)(CNC(c2c(C)sc(Br)c2)=O)CCCN(C(=O)CC2CCC2)C1 28698,N1(CCC)C(=O)CCC1C(=O)NCC(C)(C)CN(C(=O)Cn1nc(C)nc1C)C 28699,c1(CC(COC)C)cn(CC(CNC(=O)C(=O)Nc2cc(C)cs2)OC)nn1 28700,Cc1c(CS(N2CCCC(OC3CCC3)C2)(=O)=O)cccc1Br 28701,CC1CN(C(c2ccn(C)c(=O)c2)=O)C(C)CN1C(C1CCNC1=O)=O 28702,C1(C(C)C)CCCN(C(c2ncoc2CNC(C2(C(F)(F)F)CC2)=O)=O)C1 28703,C1(CC)(NC(=O)C(F)F)CCN(C(=O)C(C)(C)C)CC1 28704,c1(C(N2C(C(C)C)CN(C(=O)C(C)n3ccnc3)CC2)=O)ccc([N+](=O)[O-])cn1 28705,CCC(CC)CC(F)C(=O)N1CC2CC1CC2CNC(C1CC(F)(F)C1(C)C)=O 28706,c1(C(N(C2CC(NC(C(C)c3cncs3)=O)C2)C)=O)cccc2c1CCO2 28707,c1(C(=O)NC2C(F)CCN(C(C3(C)CC(=C)C3)=O)C2)sc2cncn2c1C 28708,c1(CC(=O)NC2CCN(C(C=NOC)=O)C23CC3)cccc2[nH]ncc12 28709,c1(COC(c2cccc(C(F)C(F)(F)F)n2)=O)cc(Cl)ccc1F 28710,CC1(C)C2CCC(NC(=O)NC(C3CCCCC3)Cc3ccccc3)C1C2 28711,C(=O)(C1=CCC2CCC1N2C(=O)COC1CC1)N(C(CC)COC)C 28712,n1(CCC)nc(C)c(C(N2CCC(NC(=O)CCC3CC3CC3CC3)C2)=O)c1C 28713,C1(NC(c2c(OCC=C)cccn2)=O)CN(C(c2cc[nH]c2C)=O)CC2(CC2)C1 28714,N1(C(Cc2c(C)scc2)=O)CCC(C)(O)C1C(=O)NCCc1nnc(O)o1 28715,c1(C(=O)NCC(C)CN(C(=O)COc2ccc(Cl)nc2)C)cccc(CO)n1 28716,CC(C)CC(F)C(=O)NC1CCC(NC(c2ncccc2OC(F)F)=O)CC1 28717,N1(C(c2cccc(C)c2F)=O)CCCC(C2CCN(C(C3CCOCC3)=O)C2)C1 28718,C1(NC(C2CC(=C)C2)=O)CC(NC(=O)COCc2cccc(Cl)c2)CC1O 28719,C1(C(=O)OC)CC(F)(F)CN1C(c1cc(C)c(C)s1)C(=O)NC(C)C 28720,C1(CNC(C(CC)(C)C)=O)C2CCCC1N(C(c1cc(C#N)no1)=O)C2 28721,C1(NC(CC(CC=C)(C)C)=O)CC2(CCC(CNC(C3C4COCC34)=O)CC2)C1 28722,n1(CC(C)(C)C)cc(C#N)cc1NC(C1COC(=O)N1)=O 28723,CCCC(C)(C)CC(=O)C1C(CNC(CSc2cn(CC(=O)O)nn2)=O)CC1O 28724,N1(C(C(C)OCC2CC2)=O)CC(CNC(C2(C)CCN(C)C2=O)=O)CC(C)C1 28725,C(=O)(C(O)CC(C)(C)C)NC(CC#CC)C(=O)NCc1cccc(F)c1 28726,c1(C(N(C2CCN(C(c3cnsn3)=O)C2)CCC)=O)cc(Cl)cc(Cl)c1F 28727,c1(OC)nccc2c(C(N3CC4C(NC(c5cc(C)oc5C)=O)C4C3)=O)c[nH]c12 28728,N1(C(CCc2ncc(C)[nH]2)=O)CCCCC(NC(c2n[nH]c(C)c2F)=O)C1 28729,C12(C(CO)NC(=O)NC(C(C)C)C3CC3)CC3CC(CC(C3)C1)C2 28730,c1(C(C(=O)NC(CNC(Cc2cc(CC)no2)=O)C)O)ccccc1F 28731,CC1(CC(N2CC(CO)(NC(c3coc(Br)c3)=O)C2)=O)CCS(=O)(=O)N1 28732,C(C1CCCN1C)=CC(=O)NC(CC=CC(=O)NCC(C)Sc1ccccn1)(C)C 28733,CC(C)(C(=O)N1CCC(NC(c2cc(Br)sn2)=O)C1)c1cc[nH]n1 28734,C12(NC(CSCCOC)=O)CCC(CNC(=O)C=Cc3ccnn3C)(C1)OC2 28735,c1(CNC(c2n(C)cc(Cl)c2)=O)ccc2c(c1)CN(C(=O)Cc1cc[nH]n1)C2 28736,c1(C(=O)NCC2N(C(CSCCOC)=O)CCCC2)cccn2nncc12 28737,N1(C(C=CCCC)=O)CCCC(C(=O)NCc2conc2C)CC1 28738,c1(C(N(C2CN(C(c3cc(Cl)cnc3O)=O)CC2F)C)=O)ccc2nonc2c1 28739,C1(NC(c2cc(Cl)ns2)=O)CN(C(c2nc(C3CC3)cs2)=O)CC12CCC2 28740,C(=O)(CCCCNC(C1CCC2CC12)C)OCC 28741,c1(C(N2C(CNC(CC(CC)OC)=O)CN(C)CC2)=O)cc(C)c(F)cc1O 28742,Cc1ccc(C(=O)NC(C)(CNC(=O)C(F)F)CC(C)C)c(=O)n1C 28743,c1(SCC(=O)NCCC2CCN(C(c3c(CC)csc3)=O)C2)ccccc1F 28744,c1(C(=O)NC2CC(NC(C(c3scc(C)n3)C)=O)C2)cc2nccnc2cc1C 28745,c1(OC)ccccc1CCC(=O)NC(C)CC(C)NC(c1nocc1C)=O 28746,c1(C(N2CCC(NC(=O)N(CC=CCl)C(C)C)C2=O)C)ccc(F)cc1 28747,c1(C(C)NCCCOCc2ccc(Cl)cc2)nnc2n1CCC2 28748,c1(C2C(=O)N2)cc(F)c(F)c(Cl)c1F.c1(N(CCOC)C)ccc(OC)cc1 28749,c1(OC)ccc(CC2(C(=O)N(C)C)CC2)c(COc2ccccc2)c1 28750,C1(C(N(C2CCN(C(c3c(C)nc(C4CC4)o3)=O)C2)C)=O)CC2CCCCCC12 28751,C1(CNC(c2cc(Br)cs2)=O)COCCN1C(C1C2CCCOC12)=O 28752,N1(C(Cn2ncc(CC)c2)=O)CC(NC(C2(CC)CCCC2O)=O)C(CO)C1 28753,c1(OC)ccc(C(c2cccnc2)NC(C2CCC2(C)C)=O)cc1 28754,c1(C(N2CCC(NC(COCCCC)=O)C2C)=O)cc2cccnc2cc1F 28755,c1(C(N(CC(C)NC(=O)C=CCOCCO)CC)=O)c(F)cc(OC)cc1F 28756,c1(C(NOCC2(C)CC2)=O)cccnc1C(=O)NCC1CC(O)C1(C)C 28757,CC1CCC(C(=O)N(CCNC(c2cncc(CO)c2)=O)C2CC2)CC1 28758,C1(C(F)F)(NC(C2CS(=O)(=O)C2)=O)CC(NC(=O)C(O)C2CCC2)C1 28759,Cc1csc(=O)n1COC(c1ccc(CC2CCC3CC23)cc1)=O 28760,C12(CNC(Cc3cncc(C)c3)=O)CCCC(CN1C(c1nc(O)c(C)s1)=O)C2 28761,N1(C(c2c(CC)cccn2)=O)CCN(C(C2CCC(=O)N2)=O)C(COC)C1 28762,CC(C)CCC(=O)NC(c1ccccc1F)CNC(c1ccco1)=O 28763,N1(C(CCCC2C(C)C2)=O)CCC2CC1CN(C(c1cc3ncccc3s1)=O)C2 28764,Cc1cc(O)c(C(=O)NC(C2(O)CCN(C(=O)CN3CCC(C)C3)CC2)C)nn1 28765,CCC(CC(=O)NC1CCN(C(=O)CCOc2cc(F)cc(F)c2)C1C)C(C)C 28766,C1(C(=O)NC(C2CC(NC(=O)CC3CC(C)(C)CO3)C2)C)CCC(O)CN1C 28767,C1(N(C)C)CC2(CCC(CNC(C3CCC4CCCCN4C3)=O)CC2)C1 28768,N1(C(C2(CC=C)CC2)=O)CCC(C)C(N(C(c2ncc(F)cc2N)=O)C)C1 28769,c1(CN2C(CNC(C(C)NC(C)=O)=O)CC2)csc2ccc(F)cc12 28770,N1(C(C2=CC(C)(CC)C2)=O)CCN(C(=O)CCCC(C)=O)CC2(CC2)C1 28771,n1(CC)nc(C(C)C)cc1C(=O)N(CC(C)NC(c1cc(C)c(Cl)s1)=O)C 28772,c1(C(=O)NCC(CNC(C(c2ccccc2Cl)OC)=O)O)nccc2nn[nH]c12 28773,CCCC(F)C(=O)NC(COC)CC(=O)NCC1(CN(C)C)CCC1 28774,Cc1nnc(O)c(C(N2CC(NC(=O)CCCN=[N+]=[N-])C(C)C2)=O)c1C 28775,N1(C(C(C=CC)O)=O)CCC(CO)(CNC(C2(OC)CCC(C)(C)C2)=O)CC1 28776,C=CCCCC(=O)NCCOCCN(C)C(c1cnc(SC)n1C)=O 28777,c1(C(N(C2CCN(C(=O)CC3CCCO3)C2)C)=O)cnc2n1CCCC2 28778,C1(CNC(CC2C(C)C2)=O)COCCN(C(c2ccc(CC3CC3)s2)=O)C1 28779,c1(C(=O)NCC(CNC(C2CCN(C)C2=O)=O)S(C)(=O)=O)ccn2ncnc2c1 28780,C(=O)(C(O)C(C)(C)C)NC(C)CC1CCN(C(c2cc(C(C)(C)C)no2)=O)CC1 28781,C#CCS(=O)(=O)CCNC(=O)NC1(C)CCCC1(F)F 28782,C(=O)(C(=O)C(C)(C)C)NCC1(OC)CCN(C(=O)CCn2ccccc2=O)C1 28783,C1(CNC(CCC2CCC(C)O2)=O)CN(C(c2coc(C(F)F)n2)=O)CC1(C)C 28784,c1(NC(C2CC(NC(CNC(CCC)=O)=O)C2(C)C)=O)n[nH]c2ccccc12 28785,c1(OC)nn(C)cc1C(=O)NCC12CC(CN1C(c1csc(O)n1)=O)C2 28786,C(=O)(C(O)(C(C)C)C(F)(F)F)NC1CN(C(CC(=C=C)C)=O)C(C)(C)C1 28787,CCC(C(=O)N1CCN(C(=O)C=CC2CCOCC2)CC(C)C1)C(F)(F)F 28788,N1(C(c2cc(CCC)[nH]n2)=O)CC(C)(CNC(=O)CS(=O)CC)CC1(C)C 28789,c1(C(N2C(CNC(C3CC4(CC4)CO3)=O)CCCC2)=O)ccc2[nH]nc(Cl)c2c1 28790,N1(C(=O)OC(C)(C)C)CC2CC(O)C1C2CNN1CCCCC(NC(N)=O)C1=O 28791,N1(C(C2N(C)CCC2)=O)CCCC2(CCN(C(c3cnn(C)n3)=O)C2)C1 28792,C(=O)(C1=CCCOCC1)NC1C(CNC(C2=CC(C)(C)C2)=O)COC1 28793,c1(C(N(C2(C(=O)NC3(C(=O)NCC)CC3)CC2)C)=O)occc1C 28794,N1(C(C2C3COCC23)=O)CCCC(Cn2cc(Cc3ccccc3F)nn2)(CO)C1 28795,C(=O)(CCC(C)S(C)(=O)=O)N(C1C2CN(C(c3cc(C)cc(F)c3)=O)CC21)C 28796,C1(CNC(COCCCC)=O)(CO)CCN(C(c2nc(CC)ns2)=O)CC1 28797,c1(NC(CN(C(=O)C(CC)=CC)CC#C)=O)ccc(N(C)C)cc1 28798,C(=O)(C(CC(C)CC)NC(c1cc(=N)[nH][nH]1)=O)Nc1cnc(COC)nc1 28799,N1(C(C2C3CN(S(=O)(=O)C4CCOCC4)CC23)=O)CCc2ccc(F)cc2C1 28800,C(=O)(C(C(C)(C)C)c1ccccc1)NC1CC(NC(c2cn(COC)nc2)=O)C1 28801,C(=O)(CC(C)C(C)(C)C)N1CC=C(C(=O)OC)C1.C1(C)(C2CC2)C(=O)N1C 28802,Cc1nc2ncc(C(N3CC4C(NC(C5CC=CC5)=O)C4C3)=O)cc2o1 28803,C1(C(NOCCOCCOC)=O)CC(O)C1NC(=O)C=CC(C)CC 28804,c1(C(=O)NC2C=CCN(C(=O)CN3CCC3)C2)csc2ccccc12 28805,N1(C(C(=O)N(C)C)=O)CCC(C)(NC(c2cccc(N3CCOC3=O)c2)=O)C1 28806,CC(C)CS(=O)(=O)CC(=O)N1CC(O)CC1CNC(c1ccccc1)=O 28807,C(=O)(CCC(c1ccccc1)N(C)C)NC(C1CCN(C(=O)C(C)(C)F)CC1)C 28808,CC1(C)CC(CC(N2CC(NC(c3ccc(Cl)o3)=O)C(C)(C)C2)=O)CCO1 28809,N1(C(=O)NCCCC#C)Cc2nnc(C)n2CC1C(=O)OC 28810,c1(C(=O)NCCN(CCC)C(c2cccc(CF)c2)=O)nn(C)c2c1CCC2 28811,N1(C(CSSC)=O)CCN(c2cc(CNC(=O)CCC(F)F)ccn2)CC1 28812,n1(CCNC(=O)C(O)Cc2cnc[nH]2)cc2ccccc2n1 28813,CCC(C(=O)NC(c1cccnc1)C(=O)NCCn1nncc1C)n1ccnc1 28814,C12(CNC(C=CC(C)(C)C)=O)CN(C(=O)C=CSc3nc[nH]n3)CC(F)(C1)C2 28815,CC(C)CC(C(=O)NC(CO)CC(C)C)NC(C1C2CCC(F)C12)=O 28816,C1(C(N(CCCNC(C2CCN(C)C2)=O)CC)=O)CC12CC(C)(C)C2 28817,C1(NC(C(CSC)OC)=O)CCN(C(=O)CC2(O)CCCC2)C1(C)C 28818,N1(C(CC(C(F)F)NC(c2c(C)ccc(O)c2)=O)=O)CC(C)C12CCOCC2 28819,c1(NC(CC2CCN(Cc3c(C)n[nH]c3)C2)=O)ccc(C(F)(F)F)cc1 28820,N1(C(c2c(OC)nsc2)C(=O)NC2CC2)CCCC(C)(O)CC1 28821,CC(Cl)(Cl)C(=O)NCC(C1CCOC1)NC(=O)C=Cc1cc[nH]n1 28822,C1(CNC(C(COCC)C)=O)CN(C(=O)Cc2cccnc2Cl)CC1O 28823,c1(CC)nc(C)c(C(N2CC(NC(C3CC3CN(C)C)=O)C(SC)C2)=O)s1 28824,CCCC(C(=O)NCc1cc(C(N2CCC23CC(C)(CO)C3)=O)ccn1)C(C)C 28825,c1(C(=O)NC(CN(C(c2cc(C)[nH]c2)=O)C)C)cc(C#N)ccc1C 28826,c1(CN(CC=C)C)cc(C)c(-c2ccccc2OC)s1 28827,c1(NC(C)C)ccc(C(=O)NCCCC(C)NC(=O)C(C2CCCCC2)F)cn1 28828,C1(NC(CSCC#C)=O)C(CNC(c2cc3ccncc3s2)=O)CCC12CCC2 28829,c1(C(C(=O)NCC(C)N(C(Cc2cnc(C)[nH]2)=O)C)O)ccc(Cl)c(F)c1 28830,N1(C(CC=CC(C)(C)C)=O)CC(NC(c2cc(C3CC3)no2)=O)CC(O)C1 28831,C1(C2CCC2)(C(=O)NCC2N(C(=O)Cc3ccccc3F)CC2)CC1(F)F 28832,c1(C(=O)CNC(C2CCC3NCCC3C2)=O)ccc2c(c1)CCOC2 28833,N1(C(c2cc(SC)oc2)=O)CC(CC(=O)N(C)CC2C(C)(C)C2(C)C)C2(CC2)C1 28834,C1(c2nnnn2C(C)(C)C)(NCC2(SC)CCCC2)CCCC2CC12 28835,C(=O)(C(F)C(C)CNC(c1cc(C)cc(O)c1)=O)NC(COC)(C)C 28836,CCC(C(=O)NCC1(F)CC(NC(C2(C)COC2)=O)C1)Nc1ccccc1 28837,Cc1cc(F)cc(C)c1C(=O)NC1CC1NC(C1CN2CCCC2CO1)=O 28838,C=CCCCCCN(C(=O)CC1CCCN1C(=O)C(O)C1CCC1)C 28839,C(CCCCC(=O)N(CCCCN(C)C(C1CCCN(C(C)C)C1)=O)C)OC 28840,C1(NC(C(CCSC)O)=O)CCC2(CCN(C(C3(CCN(C)C)CC3)=O)C2)C1 28841,Cc1cccc(C(O)C(N2CC(O)(CNC(C3CCC(C)(O)CC3)=O)C2)=O)c1F 28842,C1(O)(CC(=O)NC2(CF)CCN(C(c3c(C(C)C)ocn3)=O)C2)COC(C)(C)C1 28843,O=C(C1=CCCO1)NCCCN(C(=O)C(F)(F)C1CC1)CC1CCCC1 28844,N1(C(C(C2CCC2)OCC)=O)CC(C)(C)CC1C(=O)NCC1(C)CNC(=O)O1 28845,N1(C(CCc2n(C)ccn2)=O)C(C(=O)NC2CCOC2)CC2CCCC12 28846,c1(C(C(=O)N(C2CN(C(C3C(OCC)C3C)=O)C2)C)C)cccc(Cl)c1 28847,C1(NC(C(C)=C(C)C)=O)CCC(N(C)C(c2cc(-c3ccccc3)[nH]n2)=O)CC1 28848,c1(OC)cc(C(=O)NC2CCCC2NC(C2(F)CC2)=O)cnc1O 28849,C(=O)(CCCCCNC(N)=O)NCC(CNC(C1(COC)CCCO1)=O)(C)C 28850,c1(-c2c(OC)ccc(CO)c2)cncc2sc(C(=O)Nc3conc3C)cc12 28851,c1(OC)c(C(=O)N(C(C)CC2CN(C(C3CCC3OC)=O)C2)CC)cccc1Br 28852,C1(NC(c2sccc2C#N)=O)CCC(O)CN1C1(CCCC)CC1 28853,C(=O)(N=c1[nH]oc2c1CC(C(C)(C)C)CC2)c1nn(C)c(NC(C2CC2)=O)c1Br 28854,C(CCC(C)(C)NC(C1CSCN1C(=O)C(C)OCCN(C)C)=O)OC 28855,C12(NC(C(C)Sc3ncccn3)=O)CCCCCC1N(C(=O)CC(C)(F)F)CC2 28856,N1(C(C2CN(C(C)=O)C2)=O)CC(CNC(=O)CC2CCC(O)C2)C2(CC2)C1 28857,Cc1cc(C(N2CC3CC(CNC(c4cnco4)=O)C3C2)=O)n2nccc2n1 28858,c1(CNCc2c(OCCCC)nccc2)nc(Cl)c(C)cc1F 28859,N1(C(C(C)N(C(C2CCCCCN2C)=O)CC)=O)CC2CCCCC12C 28860,C1(C(=O)NCCCOCCCNC(COCCOC)=O)(CO)CC=CCC1 28861,C(C(=O)NCC1CCC(F)(F)C1)(C(C)(C)C)NC(c1c(CC)cno1)=O 28862,C1(c2nc(C3(CN)CCCCO3)on2)CC12CCOc1ccccc12 28863,N1(C(c2ccc(O)cc2)=O)CCC2CCCC12CNC(C1(CCF)CC1)=O 28864,C1(C(N2CCC(N(C(C3(c4cc[nH]n4)CCC3)=O)CC)C2)=O)CC(C)(C)CN1C 28865,C1(O)(CN(C(c2c(CC)occ2C)=O)C)CCCN(C(=O)C(F)(F)C(F)F)C1 28866,N1(C(C2CC(SC)C2)=O)CCC2CN(C(c3cnc4ccccn34)=O)C2C1 28867,c1(C(=O)NCCC2CC(NC(C3CCC3)=O)C2)cnoc1-c1ccccc1 28868,c1(C(=O)NCC2CC(NC(C=C(C)Cl)=O)C2)ccnc2c1ccn2C 28869,c1(CNC(CC(=O)Nc2c(C)nc[nH]2)Cc2cccs2)cccc(F)c1I 28870,C1(CC=C)(NC(=O)CS(=O)(=O)CCO)CC2CCC(C1)N2C(=O)C(C)CF 28871,C1(OCC)CC(NC(C2CC23CCC(F)(F)CC3)=O)C12CCCCC2 28872,C(=O)(C1=CC2(CCOCC2)C1)NCC(C(C(C)C)C)NC(c1c[nH]ccc1=O)=O 28873,N1(C(c2cc(C)oc2)=O)CCN(C(c2ccnnc2S)=O)C2CCCCC2C1 28874,N1(C(CC(=O)OC(C)(C)C)=O)CC(C(=O)NCC(F)CO)CC12CCC2 28875,C1(O)(CCNC(c2c(CC)c[nH]n2)=O)CCCN(C(=O)CCc2cccs2)C1 28876,CCCCC(C(=O)N1CC2CCC2(CNC(=O)Cc2cccc(Cl)c2)C1)N(C)C 28877,c1(C(N(C2CCC(NC(CCC(=O)N(C)C)=O)C2)C)=O)oc2ccccc2c1Cl 28878,c1(OC)nn(C)cc1C(N1CC(CNC(=O)Cn2nc(C)oc2=O)CC1C)=O 28879,C#CCC(C(=O)N1CCCC(CCNC(c2cnn(C3COC3)c2)=O)C1)C1CC1 28880,C12(C(=O)NC3C(C)(NC(C4N(C)CC4)=O)CCC3)CC=CCN1CCC2 28881,N#Cc1cccc(-c2cn(CCCCNC(=O)Cc3nc[nH]n3)nn2)c1 28882,C1(CC(=O)NC(CCCNC(c2c(CC)nco2)=O)C)CCC(F)(F)CC1 28883,C(=O)(CCCC(F)(F)F)NCC(C)NC(C(c1ccc(OC)cc1)C)=O 28884,C(=O)(C1CCCc2nn(C)cc21)NCCC(C)NC(=O)CC1CCS(=O)(=O)CC1 28885,C1(F)(C(N2CCN(CCCCCNC(C=CCC)=O)CC2)=O)C2CCCCC12 28886,Cc1cc(C(=O)NC2CN(C(=O)Nc3cccc(CO)c3)C2)cc(NC2CC2)n1 28887,c1(C(C(=O)NCCN(C(=O)COC2CCC2)CC)C)cn(C)c2ccccc12 28888,N1(C(C(C)OC2CCCC2)=O)CCC(C(N2CC3CCC(C2)N3C)=O)C12CCC2 28889,Cc1ccnnc1C(=O)NCC(C)N(C(=O)C#CC(=O)N(C)C)C 28890,N1(C(C2(C#C)CC2)=O)CC2(CC(NC(=O)C(CC)N(C)C)C2)C1 28891,C(CNC(c1ncsc1C(F)(F)F)=O)(C(C)C)NC(C1CC(N(C)CC)C1)=O 28892,C1(C(=O)Nc2cc(CCC)n[nH]2)COCC1(C)C 28893,CC1CCN(C(c2ccc(Cl)cc2N)=O)CC1NC(=O)CSc1ccccc1 28894,C=CC1(CNC(=O)NCCN(C)CCO)CCC1 28895,C12(CNC(C(C)CC(N)=O)=O)CCC(CN(C(c3cc4cccnc4[nH]3)=O)C1)C2 28896,N1(C2CCN(CCC)CC2)CCN(C(c2cccnc2)=O)C(=O)C1 28897,C=CCC(CC)C(=O)NCC1CC1CC(=O)NC1CNC(=O)C1 28898,N1(C(C2CCCC(OCC)C2)=O)CC2OCCN(C(=O)C=CCO)C2C1 28899,C(CCS(C)=O)(C(=O)N1CCOC(CNC(=O)C2=CCCOC2)C1)N(C)C 28900,N1(C(C(c2cn(C)nc2)=O)=O)CC2CC(NC(C3CC4(CCCO4)C3)=O)C1C2 28901,Cc1nccc(C(=O)NC2C3CN(C(c4c(Cl)nsc4Cl)=O)CC23)c1O 28902,C#Cc1ccc(C(N2CCN(C(=O)Cc3ccoc3C)C3CC23)=O)cc1F 28903,CC1=NOC(=O)C1CC(=O)NCC1(CNC(C2(O)CC(F)(F)C2)=O)CC1 28904,N1(C(C=CCC(C)(C)NC(c2cc(CC)n(C)n2)=O)=O)CC2CC1CN2C(C)C 28905,C(=O)(C#CC1CCOCC1)NC(C1CCCCC1)C(=O)NC1C(C)C1C 28906,c1(C2(C(=O)O)CN(Cc3cccc(-n4cncn4)n3)C2)ccc(Br)cc1 28907,N1(C(C(N2CCCCCC2)C)=O)C2CCCC1CN(C(=O)CC1(C)OCCO1)C2 28908,C1(C(N2CCC(CC3CC3)CC2)=O)CS(=O)(=O)CC1O 28909,C#Cc1cccc(C(=O)N(C(C)CCNC(C2CC(C)(C)CN2C)=O)C)c1Cl 28910,N1(C(C=CC(=O)OCC)=O)CCC2(C(=O)Nc3ncc(Br)cn3)CCCC12 28911,c1(NC(c2n(C(CC)C)nnn2)c2cccnn2)ccc(SC)cc1OC(C)C 28912,Cc1cccc(C(N2CC(NC(=O)C(C(C)(C)C)NC(N)=O)C(C)C2)=O)c1N 28913,c1(C(=O)NC(C#C)C2CC2)cccc(CNC(C2CC3(CC3)CO2)=O)n1 28914,N1(C(c2cc(COC)sc2)=O)CCC(N(C(=O)Cc2cc(C)no2)C)C(C)C1 28915,C1(CC(=O)NCC2C(NC(C(c3ccccc3)C)=O)COC2)CCC=CCC1 28916,C=C(C)CC(C(=O)N1CC(OCCF)C1)NC(=O)Cc1nocc1C 28917,C(=O)(CC(CC)c1cn[nH]c1)N(CCN(C(C(=O)NCC)=O)C)C(C)C 28918,C1(NC(C(C)c2cncs2)=O)CC2CCCCC2C1 28919,CN1CCC(O)(CNC(c2cc(CNC(C3(C)CC3(C)C)=O)cs2)=O)C1 28920,N1(C(C2CC(C)C2)=O)CCC(C(=O)NC2CC=CCC2)C(O)C1 28921,C1(Cn2c(C)ccc2C)CN(C(=O)OCC2CC[Si](C)(C)C2)CCCO1 28922,C(N=c1[nH]c(=NCC2=CCCC2)c2cccc(F)c2[nH]1)C1(OC)CCS(=O)(=O)C1 28923,c1(C(N(CC2N(CC)CCC2)CC2(COC)CCC2)=O)sc(Br)c(C)c1C 28924,Cc1cnc(NCC2(C)CCN(C(=O)CCC(C)(C)C)C2)c([N+](=O)[O-])c1 28925,c1(C(C)NC(C2COCCN2C(c2cc(Cl)ncn2)=O)=O)ccc(Cl)cc1Cl 28926,C1(N(C)C(c2cc(C3CCC3)[nH]n2)=O)CCCN(C(c2cnn(C)n2)=O)C1 28927,N1(CCOC)CC(NC(=O)NCC(Cl)Cl)C(C)C1 28928,c1(OC(C)=O)ccc(CNC(=O)CCCc2ncc(-c3ccccc3)o2)nc1 28929,C1(CNC(c2c(C)nns2)=O)CC(C)N(C(C2CCC(NC(N)=O)CC2)=O)C1 28930,C1(C(N2CCC(NC(CCC(N)=O)=O)CC2)=O)C2C3CC4C1C1C2CC3C41 28931,c1(SCC)ccccc1CC(=O)NCC1CCN(C(=O)CC2CC3(CC3)C2)CC1 28932,CC1(C)CCC(C(N2CCOCC2CCNC(C2COCCN2C=O)=O)=O)CC1 28933,C(=O)(CCCC(C)(C)C)NCC(C)=CC(=O)NCCC(O)C(C)C 28934,N1(C(c2nc(CC(C)C)sc2)=O)CC2CC(NC(=O)CCN3CCCC3=O)C2C1 28935,N1(C(C2(C)CCC(=O)N2)=O)CCCC2(C1)CN(C(c1ccc3cnnn3c1)=O)C2 28936,n1(CC)ncnc1C(N1CC(CN(C(=O)Cc2cnn(C(C)C)c2)C)C1)=O 28937,CCC(C(=O)NCC1(OC)CN(C(=O)CC(C)F)C1)N(C)C 28938,Cc1sc(NC(=O)C2CC2)c(C(=O)N(C2CC2)CC2CCCN2C(=O)CC#N)c1C 28939,c1(-c2cn(CC(CNC(=O)C(c3cncnc3)C)OC)nn2)cc(C)ccn1 28940,C=Cc1ccc(C(=O)NC2CCC(CNC(c3cc(CC)[nH]n3)=O)C2)cc1 28941,CS(=O)(=O)CC(=O)NCC1C=CCN1C(=O)Cc1cccnc1O 28942,c1(-c2cc(CC)no2)nc(CCOC)nn1Cc1ccccn1 28943,Cc1cc(C(=O)NCCCN(CCCCNC(C2CC=CCO2)=O)C)sc1C 28944,C1(N(C(CS(=O)(=O)NC)=O)C)CN(C(C2CC(F)(F)C2)=O)CCC1O 28945,C1(NC(COCCC=C)=O)CC(C2CCN(C(=O)C=Cc3cccc(C)c3)C2)C1 28946,c1(C(C)C)nccn1CC(=O)NCCN(C(=O)C(F)CC1CCOCC1)C1CC1 28947,c1(NCC2(C(N(C(C#C)C)C(C)C)=O)CC2)ccc(F)s1 28948,c1(C(N(CCCN(C)C(C2CSCCS2)=O)C)=O)ccc(-n2cccn2)nc1 28949,N1(C(CCc2cncc(OC)c2)=O)CCC(NC(=O)CCc2cnco2)C(O)C1 28950,C1(n2ncc(C(N(C3CCCN(C(=O)C(C)(F)F)C3)CC)=O)c2)CCC(C)CC1 28951,c1(C(=O)OC(C)(C)C)ccc(C=C(F)Cl)cc1.C1(C(=O)NC2CC2)CCCSS1 28952,C(=O)(C1=CCCN(C(C23CC(C(F)(F)F)(C2)C3)=O)C1)Nc1ccc(N(C)C)cc1 28953,CCC(CC(C)CO)NCc1cn(Cc2occc2C(=O)O)nn1 28954,C=C(Cl)C(C)(C)C(=O)N1CCC(NC(C2CC23CCCCC3)=O)C1 28955,O=C(C1=CCS(=O)(=O)C1)N1CCC2(C1)CN(C(c1cc(F)cc(F)c1)=O)C2 28956,C1(NC(C(C)Oc2ccccn2)=O)CCCN(CCn2cc(Cl)cn2)CC1 28957,Cc1ccc(F)c(C(=O)NCC(O)CCNC(c2cc(Cl)ncc2N)=O)c1 28958,C(CCS(C)=O)(C(=O)N1CCC(CCNC(c2ccc(Cl)c(F)c2)=O)C1)N(C)C 28959,C(=O)(C1=CCC(C)CC1)N1CCC(O)(CN(C(C2(CCOCC)CCC2)=O)C)C1 28960,C(=O)(CCCCC(=O)OC)NCC1N(C(C23C(CN(C(C)=O)C2)C3)=O)CCCC1 28961,C1(COC)(NC(c2ccccn2)=O)CCN(C(c2ccc(C(N)=O)[nH]2)=O)CC1 28962,c1(SCCC(=O)NC2CC(NC(CCN(CCC)C)=O)C2)ncnc2[nH]cnc12 28963,C1(NC(C2CC(OCC)C2)=O)CCC2(CCN(C(C3(C)CC(C)(C)C3)=O)C2)C1 28964,C1(C(=O)NCCc2c(C)noc2C)CC(O)CCN1C(c1cnc(O)o1)=O 28965,N1(C(c2c(C)nn(CC(F)F)c2)=O)CCN(C(C2C3CCC(=O)C23)=O)CC1C 28966,CC(CCCO)(N=c1ccn(Cc2ccc(F)cc2)[nH]1)c1ccccc1 28967,C1(CC(=O)NC(c2c(C)nccc2)C)C2CCCC2N1C(=O)C(C#N)C(C)C 28968,c1(N(C(=O)C(C)N(C(=O)C(C)C=C)C)CC#C)ncc(CC)s1 28969,C(c1cccc(F)c1Cl)=CC(=O)NCCC1(CNC(CCN(C)CCO)=O)CC1 28970,c1(N(C(COC(CNC(C(C2CCOC2)OC)=O)(C)C)=O)C)ccccc1 28971,c1(C(N2CC(c3c(C(N(CC)CC)=O)nco3)C2)=O)cccc(C(N)=O)n1 28972,C1(C(=O)NCC2(COC)CN(C(=O)CCCC(F)(F)F)C2)CC2C=CC1CCC2 28973,c1(CC)cc2c(cc1Br)CCC2.C12=NC(=NCc3ccccc3C1=O)NC(C)=C2 28974,CC1CN(C(=O)CCC(=O)c2cccc(F)c2)CC1NC(C1CCC1)=O 28975,c1(NC(=O)CCNC(c2ccc(Cl)o2)CO)ccc(Cl)cc1F 28976,CC(C)CC(CCO)NC(C1OCCC1CNC(c1ccn(C2CC2)n1)=O)=O 28977,c1(C(=O)OC)cc(C)cnc1N1CC(NC(C2CC(=O)N(C)C2)=O)C1 28978,Nc1cc(C(=O)NC2CCC(NC(=O)CC34CCCC3C4)CC2)c(F)c(O)c1F 28979,c1(COC)cccc(C(=O)NC(C)CN(C(=O)CCSCC(C)C)C)n1 28980,N1(CCOC)C(=O)NC(c2csc(C#N)c2)C2=C1CN(C(C)(C)C)C2=O 28981,S(=O)(=O)(c1ccc(N2CCCC(OCC(F)F)C2)cc1Br)NCC1(C)CSC1 28982,C#Cc1ccc(Cl)c(C(=O)NC2CCCC(NC(c3cnsc3C)=O)C2)c1 28983,c1(C(N2C(CCc3cn(CC4CNC(=O)O4)nn3)CC2)=O)ccccc1C1CC1 28984,C1(CNC(C2CCC(C)C2)=O)CCCN(Cc2sncc2Br)C1 28985,c1(NCc2c(-c3c(F)cccc3)nccc2)cccc2c(Br)cccc12 28986,C1(NC(=O)CONC(=O)CC2C=CCCC2)(CO)CCOCC1 28987,C(N=c1[nH]c(=NCC2CN(C3CCC3)C2)[nH]c2ccsc12)c1c(C)cccc1Cl 28988,c1(C(=O)NC2C(CNC(C(C)(C)c3cnc[nH]3)=O)C2)cccc(-n2ccnc2)c1 28989,N1(C(Cc2c(OC)nccc2)=O)CC2CC(NC(C3CCC3C(F)F)=O)CC1C2 28990,C(=O)(C1CCCc2nncn21)N1CC2CN(C(CN(C)C3CC3)=O)C2CC1 28991,N1(C(C2N(C)CCC2)=O)CCN(C(=O)C(O)C2CC2)C(CO)C1 28992,c1(C(C)C)ccc(-n2nc(COc3ccccc3)nc2C2CC2F)cc1 28993,c1(C(=O)NCCC(=C)CNC(=O)CCn2ccnc2)c(Br)cnn1C 28994,C(N=c1nc2scnc2c(N2CCOCC(F)(F)C2)[nH]1)c1n(C)nnn1 28995,C1(C(=O)NC(CO)C2(C)CC2)(NC(C(CO)N(C)C)=O)CCCCC1 28996,c1(C(=O)NC(C(C)NC(C=CC)=O)C)c(C)nn(C)c1Sc1ccccc1 28997,c1(C(N2C(C)CC(CNC(=O)CC3CCOCC3)C2)=O)cncc(C#N)c1 28998,c1(C(N2CCC(NC(C(CCC)OCC)=O)C2(C)C)=O)cc(F)cc(Cl)c1N 28999,c1(C(=O)NCC2(F)CN(C(=O)C=C3CCC3)C2)cc2cccc(Br)n2c1 29000,c1(C(=O)NCC(CC)NC(=O)CCc2scnc2C)cccc(C#CC2CC2)c1 29001,C(c1nc2cc(Br)cnc2s1)=C(C)C(C)(C)C 29002,CC1(CNC(c2ccc(CNC(c3cccc(F)c3F)=O)o2)=O)CCCCC1O 29003,c1(CC(=O)NCCC2CCC(NC(C(C(=C)Cl)(C)C)=O)C2)ccccc1[N+](=O)[O-] 29004,C(=O)(C1=C(Cl)CCOC1)N1CCC(C(N2CC(CC)NC(=O)C2)=O)C1 29005,C(CN=c1nc(N2CC=C(Br)CC2)c2c([nH]1)CCS2)N1CC(C)OC(C)C1 29006,N1(C(CNC(CNC(CC(C)SC)=O)=O)=O)CCCC2OCCC12 29007,c1(CC)cn2c(n1)CC(C(=O)NCC(C)N(C)C(c1cc(C)cc(O)c1)=O)CC2 29008,N1(C(C(C)Oc2ccccc2)=O)CC2CC2(NC(C2(c3ccn(C)n3)CC2)=O)C1 29009,c1(CC)ccc(F)c(C(N2CC3CCOC3(CNC(=O)C(CC)SC)C2)=O)c1F 29010,n1(CC(N2C(C(=O)NCC(C)OC)CCC2)=O)ccc2ccccc12 29011,C1(C(N2CCCC2CCNC(C2(CF)CC2)=O)=O)CC12CCC(F)(F)CC2 29012,CCCCC(C)CCC(=O)N1CCC1CNC(c1sccc1CC#N)=O 29013,C(=O)(C1=C(C)OCCS1)N1CC(OCC)C(CNC(C2CCC(C)(C)OC2)=O)C1 29014,N1(C(C2(C)C(C)C2)=O)CC2CN(C(c3ccc(C(N)=O)cc3)=O)CC2C1 29015,N1(C(C2=CC(C)(CC)C2)=O)CC2CC(C1)CN(C(c1cc(Br)c[nH]1)=O)C2 29016,c1(OC)ccc(C(=O)NCCNC(=O)NC2CC2)c(Cl)c1 29017,N#CC1CCN(C(C2CN(C(c3ccc(O)c(I)c3)=O)CCC2O)=O)CC1 29018,c1(C(N2CCCC(O)(CNC(c3ccco3)=O)C2)=O)cc(F)c2c(c1)CCC2 29019,c12ccnc(c1F)NC2=O.C(=O)(C(C)(C)OC)N(CC(C)NC(COC)=O)C 29020,C(=O)(C1=CCOCC1)NC(COC)C(=O)NCCC1CCN(C)C1=O 29021,CN1N=C(C(=O)Nc2cccnc2C(N2CCCC(NC(C)C)C2)=O)CCC1=O 29022,c1(C(=O)NCCC2CSCCN2C(c2ccncc2)=O)csc2c(F)cccc12 29023,c1(CCCC)ccc(C(N2CCN(C(C)C(=O)NC3(C(N)=O)CC3)CC2)=O)cc1 29024,c1(OC)nc(C)ccc1C(=O)NCC1(C)CN(C(c2c[nH]nc2C)=O)CCO1 29025,c1(C(N2CC(CC)N(C(=O)CCC(=O)OC)CC2)=O)cc2c(C)nn(C)c2s1 29026,c1(C(N(c2nc(C#N)cs2)C(=O)NCc2ccn(C)n2)C2CC2)ccc(F)cc1Br 29027,CC1CC2CN(C(=O)C(CO)C(F)(F)F)CC2N1C(=O)CCC(=O)C1CC1 29028,c1(CCC)cc(C(N2CCCC2CNC(=O)CCCOC)=O)no1 29029,Cc1noc(C)c1C(C)C(=O)NCC1(CNC(C2(C)CNC(=O)C2)=O)CC1 29030,n1(CC)nc(C(=O)NC2C(OC)C2C(=O)OC)c2cccc(O)c12 29031,c1(C(=O)NCC2CN(C(C3CCCC3)=O)C3CC23)cc2c(cn1)OCCC2 29032,Cc1cc(C)n(CCNC(=O)CC(C2CC2)NC(=O)CC2CC(C)(C)CO2)n1 29033,c1(OC)cc(C(=O)N(C2CC(NC(=O)C(C)(C)CO)C2)C)cnc1OCC 29034,c1(NCC)scnc1C(=O)NC(C)CNC(=O)COCCc1cccs1 29035,CCCC(C)(C)CC(=O)NC1C(C)(C)C(NC(C2CSCCS2)=O)C1(C)C 29036,Cn1cccc(C(=O)NCC2C3CN(C(C4(CCF)CC4)=O)CC23)c1=O 29037,C1(NC(CSS(C)(=O)=O)=O)CCN(C(=O)CCN2CCCC2=O)CC1CO 29038,c1(COC)nc(Cl)cc(=NC(C)CCNC(c2nc3cccnc3s2)=O)[nH]1 29039,C1(NC(C)=O)CN(C(=O)C(Cc2cccc(Cl)c2)NC=O)CC2(CCOCC2)C1 29040,C1(C2CCN(C(=O)CC3OC(C)(C)OC3=O)CC2)(NC(C2CC(SC)C2)=O)CC1 29041,C12(NC(Cn3c(C(C)C)ncc3)=O)CCN(C(=O)COCCN(C)C)CCC1C2 29042,c1(C(=O)NC2C3CCN(C(CC(C=C)CC)=O)C32)cc2c(=O)[nH]c(C)cn2n1 29043,N1(C(C(c2ccccc2)OC)=O)CCCOC(CNC(=O)CCCCSC)C1 29044,C1(CC(N2CC(O)(C(C)NC(c3n(C(C)C)ccn3)=O)C2)=O)COCC(C)(C)O1 29045,c1(CNC(C(COC)C)=O)ccccc1CNC(C)=O 29046,C(C(C(=O)N(C)Cc1nc(C)cs1)NC(=O)CCSC)SCC 29047,C1(CC)CCN(C(=O)C=CC2CCOCC2)C1C(=O)N(C)Cc1ccsc1 29048,N1(C(C)=O)CCCC1(C)CNC1C=CCN1C(=O)CC=CC(C)(C)C.c1c(=O)n1 29049,C1(NC(COCC=C)=O)CCN(C(c2ccc(OC)cc2N)=O)CC1F 29050,c1(C(=O)NCC(=C2CN(C(c3nc(OCC)oc3)=O)C2)F)cccc(C(C)C)c1 29051,C(=O)(CCCn1cccc1)NC1C(C(=O)NC(CC)CC)CC1 29052,Cc1[nH]c(C)c(C(=O)NCCCNC(c2cccc(N(C)C)c2)=O)c1C 29053,c12cccc(c1)-c1cc(n[nH]1)-c1nccn1CC2.C1(C)(CC#N)CCCCC1 29054,c1(C(=O)NCC2(O)CCN(C(C3(CC4CC4)CC3)=O)C2)csc2ccc(F)cc12 29055,C1(NC(C(C)SCC)=O)CC(C(=O)N2CC=CC2(C)CO)=CC1O 29056,c1(C(N2CC(OC)C(NC(=O)C=Cc3cnc[nH]3)C2)=O)sc([N+](=O)[O-])cc1Cl 29057,CC1CCN(C(=O)C=Cc2ccccc2)CC1NC(=O)CC1CC(=O)NC1=O 29058,C1(NC(c2c(CC)ocn2)=O)C(C)CN(C(=O)C2=C(C)CCCC2)CC1C 29059,C1(CC(C)NC(c2cc(OC)ns2)=O)CCN(C(=O)CC2CCS(=O)(=O)C2)CC1 29060,N1(C(c2ccc(NC(C)=O)s2)=O)CCN(C(=O)Cc2cnccc2C)CC1C#N 29061,c1(NC(c2cnn(C(CC)C)c2C)=O)ccc(C)c(OCC(=O)O)c1 29062,C1(CCC)CCC(C(=O)NCC(C)N(C)C(c2cnc(OC)s2)=O)CC1 29063,c1(CC)ncc(C(=O)NC(C)C(C)(C)NC(C2CC(n3ccnn3)C2)=O)s1 29064,CCCCC(O)C(=O)NCC(CC1CC1)C(=O)NC12CCC(CC1)C2 29065,C1(NC(C(F)=C(C)C)=O)CCCCCN(C(C2CN3CCCN2CC3)=O)C1 29066,c1(C(=O)NCCCCC(C)NC(C(CC)OCC)=O)ccc([N+](=O)[O-])cc1C 29067,c1(C(=O)NCCNC(c2occ(C)c2)=O)ccccc1Oc1ccccc1F 29068,C(CC(C(=O)NC(C(C)(C)O)C1CC1)NC(=O)CCc1ccc(C)o1)=CC 29069,N1(C(C=C(C)C)=O)CCC(C(=O)NCc2ccnc(O)c2)(C(C)C)C1 29070,Cc1sc(-c2ccccc2)nc1C(=O)NC1CN(C(C2CCCO2)=O)C1 29071,C1(C(=O)NCC(CN(C(c2c(C)occ2)=O)C)C)C2CCC1(c1nccs1)C2 29072,C1(CC)CN(C)C(=O)CN1C(=O)NC1CCCC=C1Br 29073,N1(C(c2cncc(NC(c3ccncc3Cl)=O)c2)=O)C2COCC1CC(F)C2 29074,C(=O)(C1COc2ccccc21)NCC1CC(C)N(C(c2cc(F)ccc2N)=O)C1 29075,C1(C=O)CCCC(=O)C1.C1(N(N(C2(CC(=O)OC)CC2)C)C)(COC)CCOC1 29076,C1(NC(c2cc(C)oc2)=O)CCCCN(C(c2c[nH]c(=N)s2)=O)CC1 29077,CCCCC(=O)C(=O)N(CCCNC(c1nnc(S)n1C)=O)Cc1cccnc1 29078,C=CC(F)(F)C(=O)N(CCCNC(=O)CC1COC(C)(C)C1)C 29079,c1(N2C(C3CCCN(C(C4CC(=C)C4)=O)C3)CCCC2)nc2c(C)cccc2o1 29080,C12(C(N3CCC(C(C)(O)CNC(=O)Cc4cncs4)CC3)=O)CCC(F)(CC1)C2 29081,C1(C(N2CC(CCO)(NC(COCCC)=O)C2)=O)OCCOC1c1ccccc1 29082,c1(NC(CNC(C2N(C(C)C)CCC2)=O)(C)C)nc2cc(Cl)cc(Cl)c2o1 29083,c1(C(=O)NCc2occ(C(N(C)OCC(F)(F)F)=O)c2)nc(=N)cc[nH]1 29084,c1(CC)nc(Cl)nc(N2CCCCC(CNC(C3(CO)CCCO3)=O)C2)c1C#N 29085,C12(C(N(C)CC3CCN(C(C(=O)NC(C)C)=O)C3)=O)C=CC(CC1)C2 29086,C1(NC(C2CC(C#C)(O)C2)=O)CCCC(C(=O)N(C)Cc2occc2C)CC1 29087,CC(C)(F)CC(=O)NC1(CF)CCN(C(=O)CCNC(=O)OC(C)(C)C)C1 29088,CC1(C)CCCC1(O)CNC(=O)CC1(NC(C2OC3CCC2C3)=O)CC1 29089,CCCCC(O)CCC(=O)NC1CCSC12CN(C(=O)Cc1ccc(F)cc1)C2 29090,Cc1noc(Cl)c1CC(=O)NC1(C)CCN(C(=O)CCCn2cnc(C#N)n2)C1 29091,c1(C(=O)NC2CC(C)N(C(c3nccn3C)=O)C2)ccccc1S(=O)(=O)C(F)F 29092,C1(NC(C2N(C(C)C)C(=O)CC2)=O)CCCCN(C(=O)C(F)C2CCC2)C1 29093,Cc1cccc(C(N2CCCC2C(=O)N(CCC#N)C2CC2)=O)c1Cl 29094,CCCC(CCCNC(=O)Cc1ccc(Br)cn1)NC(c1c[nH]ccc1=O)=O 29095,CC1(C(=O)NCc2nocc2C(=O)N(C2CC2)CC2CC2)COCCO1 29096,C(=O)(C1=C(Cl)CCC1)NC(CCCCNC(C(CC)(C)C)=O)C 29097,n1(C(C(=O)NCC(C)(C)NC(C(C)NC(=O)NC)=O)C)nccc1C 29098,CC(CC(=O)N1CCC(c2cnco2)C1)C(C)(C)NC(=O)CN(C1CCC1)C 29099,C1(CNC(C2(OC)CCSC2)=O)CN(C(c2c[nH]c(=O)cn2)=O)CCC1(F)F 29100,CC1CC=C(C(=O)NCc2cncc(C(=O)NC(c3nnc(O)n3C)C)c2)CC1 29101,C(=O)(CC(C)(C)C(=O)N(CCCN(C(=O)C(=Cc1cccnc1)C)C)C)OCC 29102,C(CCCCC(=O)NC1CC(NC(=O)CC2CC(F)C2)C12CCC2)OCC 29103,c1(C(C)=O)ccc(CC(=O)NC2CC(C)(NC(C3(C4CCCO4)CC3)=O)C2)cc1 29104,N1(C(=O)OC(C)(C)C)CCC2(C1)CN(N1CCc3nc(Cl)ccc3C1)C2 29105,c1(N(C)C)cc(F)c(NC(=O)NC2CCNCC(C)(C)C2)cc1[N+](=O)[O-] 29106,c12cccc(Cl)c1OC2.c1(CNC(=O)NCCCOCC)ccc(F)cn1 29107,C1(CCC(=O)NCC2CC(NC(C(C#N)C3CC3)=O)C2)NC(=O)NC1=O 29108,C1(NC(C(CC)(C)C#N)=O)CC2(C1)CC1(CC(NC(=O)C3=COCCO3)C1)C2 29109,N1(C(C2C(C(=O)OC)CC2)=O)CC(NC(c2n[nH]cc2Br)=O)C2(CC2)C1 29110,c1(C(=O)NCCN(C(c2cnn(C(F)F)c2)=O)CC)cc(N)c(Cl)c(O)n1 29111,C1CN=C(N2CCS(=O)(=O)CC2)NC(C)C(=O)N1CC.N1(CC)CCCCC1C 29112,c1(C(=O)NCC2CCN(C(C(OC)OC)=O)CC2C)cc2c(C)ccc(F)c2o1 29113,C(c1ccco1)=C(C)C(N1CCC(CNC(=O)C(F)=CC2CC2)C1)=O 29114,CCC(C)(O)C(=O)N1CC(C(C)NC(C2(O)CCC2)=O)C1 29115,N1(C(C2=NOC(C)C2)=O)CC(C)(C)OCC1CNC(C12CCC(C)(CC1)OC2)=O 29116,C1(C)(C(=O)Nc2cc(C)sc2)CCCN1C(c1ccc(C(N)=O)[nH]1)=O 29117,C(=O)(C#CC1CCOCC1)N1C(C)CC(CC(=O)NCCN2CCOCC2=O)C1 29118,C1(NC(CCCOCCOC)=O)CC2CCC1N2C(c1cc(OC)ccn1)=O 29119,CC1CN(C(=O)C=Cc2cncc(F)c2)CC1(C)CNC(c1ncncc1F)=O 29120,N1(C(C)=O)CCCC2(C1)CN(C(c1cc3ccc(C)cn3n1)=O)CCO2 29121,Cc1cc(C(=O)N(CCNC(c2ccn(CC#N)n2)=O)CCOCCO)sc1C 29122,CC1(C)CC2(CC(C(N3CCC(CNC(=O)CCS(N)(=O)=O)C3(C)C)=O)C2)C1 29123,CCCCC(O)CC(=O)N1CC2C(C(=O)NCC(=O)NCC)C2C1 29124,N1(C(c2ccc(COC)o2)=O)CCCCC(CNC(=O)C(CBr)=CC2CC2)C1 29125,c1(C(=O)NC2CCC(NC(C(CC(C)C)(C)C)=O)C2)cn2cc(Cl)cnc2n1 29126,C(=O)(C(C)C(F)(F)F)NC(C(C)NC(Cn1c(CCC)nnc1S)=O)C 29127,C1(CNC(c2n(C(CC)C)ncc2)=O)CC2CCC1N2C(=O)C(F)(F)C(F)F 29128,C(c1cccc([N+](=O)[O-])c1)=CC(=O)NCCC(C)NC(c1ccc(Cl)c(Cl)c1)=O 29129,c1(OC)ccc(NC(C2CCCN2C(C2CCC2)=O)=O)cn1 29130,Cc1c(CC(N2CCCCC2c2cn(-c3cccc(N)c3)nn2)=O)nc(Br)n1C 29131,C#CC1(O)CC(C(=O)NC(c2cnn(C)c2)C(=O)NC2CC(C)(CO)C2)C1 29132,C1(CC(=O)N(CCOCCCNC(CC(C)O)=O)C)CCC(=O)NC1 29133,Cn1nc(C(=O)NCC2C3CN(C(C4(C)CCC(=O)C4)=O)CC23)cc1Br 29134,C1(CNC(C2(Cc3ccccc3)CCOC2)=O)NCC12CCC2 29135,N1(C(C2C(C=C)C2)=O)CCC(NC(=O)Cc2sc(O)nc2O)CC1c1ccccc1 29136,c1(SC)ccc(C(N2CC(C)(NC(C3CC4CC4C3)=O)C2)=O)cc1Br 29137,c1(C(=O)NCCOC2CN(C(C(CCCC)O)=O)C2)ccc(Cl)c(S(N)(=O)=O)c1 29138,n1(CC(=O)NC2C(CNC(c3c(CC)cco3)=O)C2)c(C)nc2ccccc12 29139,c1(CC)ccccc1CC(N1CC(CNC(=O)C=C(C)c2ccco2)(OC)C1)=O 29140,Cc1nccc(CCC(N2CC(NC(C3CCN(C(C)C)CC3)=O)CC2C)=O)n1 29141,C1(O)(C(C)C)CCN(C(c2ncccc2NS(C)(=O)=O)=O)C1 29142,c1(C(N2CC3CCN(C(CC(C)C(F)(F)F)=O)C3C2)=O)cnn(C)c1S(N)(=O)=O 29143,C1(C(N2CSCC2C(N)=O)=O)(CC)CNC(=O)C1 29144,C1(C)(CC)CC(NC(c2cc(N)c(Cl)cn2)=O)CN1C(C1COCC1C(N)=O)=O 29145,N1(C(Cc2c(Br)cn(C)n2)=O)CCOCC12CCS(=O)(=O)C2 29146,N1(C(C(N2CC(C(C)NC(C(CCC)C)=O)C2)=O)C)C(=O)NC2(CCCC2)C1=O 29147,C1(NC(CC(=C)Br)=O)CC2CC1CN(C(=O)C(C)Cc1ccncc1)C2 29148,N1(C(c2c(C)nccn2)=O)CCN(C(C2CCCS2(=O)=O)=O)C2(CC2)C1 29149,O=S(=O)(c1cc2sc(=NCCCCO)[nH]c2cc1Cl)NC1C2CCC(F)(F)C12 29150,N1(CC)CCC(CNc2cn(C3CCCC3)nn2)CC1 29151,Cc1cc(NNC(=O)C2CCCN2C(c2cccc(C(C)C)c2)=O)cc(C)c1Br 29152,c1(C(C)OC(=O)C(C)Sc2ccccc2)cccc(OC(F)(F)F)c1 29153,C1(C(=O)NC(c2cccc(F)c2)C)CCN(C(=O)C2=CC(C)(C)C2)CC1C 29154,C(=O)(C(CC(C)C)NC(=O)OC)NC1CCN(C(CNS(CC)(=O)=O)=O)C1 29155,CC1=C(C(=O)N2CC(NC(c3cc(Cl)cn3C)=O)CC2CO)CCCC1 29156,c1(N2CCC(NC(=O)NCc3cc(Cl)ncc3Cl)CC2)ncc2c(n1)CCC2 29157,c1(C(N(CCC)CCNC(=O)CN(C)C(N)=O)=O)cc(F)ccc1OC 29158,O=C(CCCCN1CCCC1)NCC12CC1CN(C(C1(O)CCSC1)=O)C2 29159,Cc1c(C(=O)NC(C2CCN(C(=O)CSC3CCOC3=O)CC2)C)c(Cl)nn1C 29160,c1(CCC(=O)NC(C(C)C)CNC(C2(C(C)(F)F)CC2)=O)ccc(F)cc1F 29161,Cc1ccn(C)c1C(=O)NCCC1CN(C(C2CC2C(C)(F)F)=O)CCO1 29162,C1(C)(CNC(C(CCC)C)=O)COCCN(C(c2ccc(CO)cc2F)=O)C1 29163,c1(OCC)sc2ncn(-n3cc(-c4ccccc4F)nn3)c(=O)c2c1C 29164,c1(OC)ncnc(C(=O)NCC2(F)CN(C(=O)Cc3ccc(C#N)cc3)C2)c1F 29165,N1(C(CCC=C=C)=O)CCN(C(=O)C(C)(C)COC)CC1C(C)C 29166,c1(C(=O)NC2CC(CNC(Cc3nc(C)sc3)=O)C2(C)C)ccc(CO)c(Cl)c1 29167,Clc1ccc2c(c1Br)CN(c1ccn3nccc3n1)CC2 29168,O=C1CCCC2C(C(N3CCCC3Cc3cn(C4CCCC4)nn3)=O)C12 29169,CN1CCC(NC2CNC(=O)C2)CC1.N12CCCC(C1)NC(=O)C1CN(C1)CC2=O 29170,c1(CN2C(C(=O)NC(C(C)C)C)CCC2)ccc(C23CCC(C2)OC3)cc1 29171,Cc1nc(S)sc1CC(N1CCC(F)(CNC(c2cncc(F)c2)=O)C1)=O 29172,C1(N(C)CC)CN(C(c2ccc(C3CCC3)cn2)C(=O)NC)CC12CCC2 29173,C1(NC(c2cc(CN(C)C)on2)=O)CCCCC1CNC(=O)C(C)(C)C1CCC1 29174,Cn1ccc2cc(-c3nc(-c4ccncc4)nn3CCc3ccccn3)ccc12 29175,c1(C(N(CCC)C(c2occc2C)=O)=O)scc2c1CCCC2 29176,c1(C(N2C(C)CC(NC(C(CCC)(C)O)=O)C2)=O)c(F)cc(F)cc1F 29177,c1(CC(=O)N(CC(C)O)CCNC(CCc2cnc(C)s2)=O)ccccc1C 29178,C1(C(C)NC(c2c(CC)noc2)=O)CCCCN1C(c1cccc(C(N)=O)n1)=O 29179,N1(C(c2c(CC)c[nH]c2)=O)CCOC(CNC(=O)C(C)(CO)OC)C1 29180,CCCCC(C)(F)C(=O)N(CC(C)NC(c1cc(N(C)C)ccn1)=O)C 29181,N1(C(CC(C)(C)NC(=O)CC2CC3C=CC2C3)=O)CCC2C(C1)C2(F)F 29182,C1(C(N2CCC(C(=O)OCC)C2)=O)CCCCN1C(=O)CNc1sccc1OC 29183,N1(C2CCN(C(=O)CCF)CC2)C2CCC1CN(C(C1C=CCC1)=O)C2 29184,C(C(F)(F)C(=O)NC1CCC1CNC(c1cc(-c2ccccc2F)no1)=O)OC 29185,c1(C(N2CCC(CNC(C3(C)CC3(F)F)=O)C2)=O)cc2nc(F)ccc2o1 29186,C=CCCC(c1nnnn1CCCNc1cnc(CSC)s1)NC(C)COC 29187,O(C1CCCc2ccccc21)CC(=O)NCCS(=O)(=O)c1cnn2cccnc12 29188,C=C(Cl)CCC(=O)NC(c1ccccc1)CNC(c1cnccc1Br)=O 29189,C(=O)(C1=C(Cl)CCC1)N1C(CCNC(CSCC)=O)CCC1 29190,N1(C(c2ccc(C(C)=O)c(O)c2)=O)CC2CCC1CN2C(c1c(C)csc1C)=O 29191,c1(CC(=O)NC2(CO)C(C)C2)csc(-c2cccnc2)n1 29192,C1(CC(=O)NC(C2CCN(C(=O)C(F)CC3CCOC3)CC2)(C)C)SC(=N)NC1=O 29193,C1(NC(c2c(SC)cn(C)n2)=O)C2COCC1CN(C(C1CCCO1)=O)C2 29194,c1(C(=O)NC(CCNC(C2N(CC)C(=O)CC2)=O)(C)C)ccc2c(c1O)CCC2 29195,C1(CNC(c2cnsc2)=O)CCCCN1C(=O)CCC1CC1CC1CC1 29196,CC(C)C(C(C)NC(c1nocc1Cl)=O)NC(=O)CCNC(N)=O 29197,n1(CC)nc(C)cc1C(=O)N(C)CC1CCCC1NC(C1(C)CC1C)=O 29198,c1(CCC(=O)N(CC(C)NC(CCOC)=O)C)ccc(Br)cc1 29199,c1(C(N2CC(COC)N(C(C)=O)CC2)=O)cc2c(cc1Br)OCCO2 29200,c1(-c2cn(C(C(=O)NCc3ncc(C)o3)C)nn2)cc(Cl)c(Cl)c(Cl)c1 29201,C1(C(=O)NC(C2N(C(c3n(CC)ncc3)=O)CCC2)C)CCCC(C)(C)CC1 29202,c1(C(=O)NCC(F)CNC(C2CCC2)=O)cc2sc(Br)cc2[nH]1 29203,Cn1c(C(=O)N(CCNC(C2CC2F)=O)CC2CC2)cc2occc12 29204,Cc1nc(O)[nH]c1C(=O)NC1CCN(C(c2cscc2C#N)=O)C1 29205,N1(C(COCc2onc(CC)n2)=O)CCN(C(c2ccns2)=O)C(CCO)C1 29206,C1(C(N2CCN(C(=O)Cc3cccnc3)CC2)=O)CC12CCCOC2 29207,c1(OC)cccc2c1CC(C(=O)NC1CN(C)CC1C)N2C(=O)OC(C)(C)C 29208,C(c1ccc(Cl)cc1F)=CC(=O)NC1CCC(CNC(c2n(CC)ncn2)=O)C1 29209,C(C)(CCC(=O)NCC(c1ccc(OC)cc1)NC(=O)CCOC)OC 29210,c1(C(N(CC(CC)NC(C2CC23CCOCC3)=O)C)=O)ccc(C)c(C(=O)OC)c1 29211,c1(NC(C)=O)ccc(Cc2nc(-c3ccc(C(=O)C(C)C)cc3)no2)cc1 29212,c1(C(=O)NCCN(C)C(c2nocc2Cl)=O)cncc2c1CCC2 29213,c1(NCc2nc3ccc(C)cn3c2)cc(=NCCS(=O)(=O)N(C)C)[nH]c(C)n1 29214,c1(C(N2CC(C(C)NC(CC(COC)C)=O)C2)=O)ccc2c(c1)CCO2 29215,N1(CCC(=O)NC(C2CCCN(C(=O)CCF)C2)C)CCCCC1=O 29216,c1(OC)ccc(C(=O)NCCCCCCNC(C2CCCCN2C)=O)nc1N 29217,Cc1cccc2c1ccn2CC(=O)NCCCCNC(C1CC(=O)NC(C)C1)=O 29218,C1(OC)COc2c(C(=O)NC34CC5CCC(C3C4)N5C(=O)CSC)cnn2C1 29219,Cc1nccn1CC(=O)NC1(C(=O)NCCN2CCC(C)C2)CCC1 29220,N1(C(CC2(O)CC(C)(C)OC2)=O)CC(N=c2cc(C(C)(C)C)nc(Cl)[nH]2)C1 29221,C1(NC(C2(NC(CSCCCC)=O)CCC(C)(C)C2)=O)CC(C2CCCC2)C1 29222,CC1(NC(c2cc(C3CC3)n[nH]2)=O)CCCN(C(=O)C(F)F)C1 29223,N(C1CN(C(c2cc[nH]n2)=O)Cc2ccccc21)c1nc(C)nc(O)c1C 29224,CC1(C)CCC2CC(NC3CCCOC3)c3cccc1c32 29225,c1(NC(C(Cc2cn[nH]c2)NC(CCC2CCC(=O)C2)=O)=O)cnc(F)nc1 29226,N1(C(c2n(C)ccn2)=O)CCCC2CN(C(c3cncc(C#N)c3)=O)CCC12 29227,c1(CN(C(c2ncc(Cl)n2C)C(=O)NCCCC)C)noc2ccccc12 29228,C(C(=O)NCCn1cc(COCCO)nn1)(C(C)(C)O)NC(=O)OC(C)(C)C 29229,c1(N(CC(C)(C)CO)C(=O)NC(COC(C)C)C)cccnc1 29230,c1(CN2C(C(=O)NCc3nc(C(F)(F)F)cs3)CC2)csc2ccccc12 29231,Cc1cc2c(C(=O)NC(C)CC(C)NC(c3cnc(O)nc3O)=O)cccc2o1 29232,c1(C(N2C(C(=O)NCCc3c(C)nn(C)c3)CC2)=O)cc(C#N)cn1C 29233,Cc1ccc2c(c1)CC(C(N1CCN(C(C3(C(C)(C)O)CC3)=O)CC(O)C1)=O)S2 29234,C12(C(=O)NC(c3cnc[nH]3)C)CCCC1CCN2C(C1OCCO1)=O 29235,C=CCCCC(=O)NCCC1(NC(=O)C(C)NC(C2CCCC2)=O)CCCC1 29236,C1(NC(CC2CCCC(CC)C2)=O)CC12CCN(C(c1ccc[nH]1)=O)CC2 29237,C=Cc1ccc(C(N2CC(O)CC2CNC(=O)Cc2ccc(Cl)c(F)c2)=O)cc1 29238,CCCCN=C(NCc1ccncc1OCC)NC1CC1(c1cccc(F)c1)C 29239,c1(C(=O)NCCCCC2CCCN(C(=O)CO)C2)cc(Cl)c2c(c1)OCCCO2 29240,CC(C)CC(CNC(=O)CSCC(C)C)NC(=O)CSc1cccs1 29241,c1(-c2cccc(NC(N3CCc4ncncc4C3)=O)c2)cncc2ccccc12 29242,C#CCC(C(=O)NCC1CCN(C(=O)C(C)O)C1)C1CC1 29243,c1(CC(=O)N(C2CC3CNC2C3)C(CC)=O)ccc(CC)cc1 29244,N1(C(C=Cc2cn(C)nn2)=O)C2CCC(C2)C1C(=O)NCc1ncn(C)n1 29245,c1(C(N2CCC(C(C)NC(=O)C(F)(F)C(F)(F)F)C2)=O)ccc2nsnc2c1 29246,N1(C(CC2CCC(C(C)C)CC2)=O)CC2CCC1CN2C(c1cc(CO)n(C)n1)=O 29247,N1(C(C(=O)OC)C)CCC(C(N2CCCCC2CO)=O)(OC)CC1 29248,C1(C(=O)NCCOC2CCN(C(CC3CN(C)CC3O)=O)C2)CCCCCCC1 29249,C=C=CC(C)C(=O)N1CC(O)(C(C)NC(=O)CCOCC2CCC2)C1 29250,c1(C(=O)NCC(=C)CCNc2cc(=O)n(C)cn2)ccc2c(c1)COCC2 29251,N1(C(C(C)NC(=O)NC)=O)CCC(C(N2CCCC(CC(N)=O)C2)=O)C12CCC2 29252,CCS(=O)(=O)c1ccc(F)c(C(=O)NC(C)C(C)NC(=O)Cc2cccs2)c1 29253,C12(NC(CC(C)O)=O)CCC(CC1)N(C(=O)Cn1cnc([N+](=O)[O-])n1)C2 29254,C#CCC(C)(C(=O)NC1CC(COC)C1)NC(C1CC(=O)CS1)=O 29255,C1(NC(CC(COC)NC(C2CC3(C2)CC32CC2)=O)=O)CCCCCC1(C)C 29256,C(C(C)(O)CCC)NC(C=C(CNC(C(C)OCC=C)=O)C)=O 29257,N1(C(C2C(OC)CC2)=O)CC2C(C(=O)NOCCCN3CCCC3)C2C1 29258,c1(C(=O)OC)cc(C(=O)NC(C)CNC(C2(C)CCN(C)C2)=O)cc(C)c1 29259,N1(C(CCCC)=O)CCCCC1CNC(C1(c2ccn(C)n2)CC1)=O 29260,c1(C(N2C(C)(CNC(=O)CS(C)(=O)=O)CCC2)=O)cc(=O)n2ccccc2n1 29261,N1(C(c2cnc(C(C)OC)s2)=O)CCCC(N(C)C(c2c(C)nsc2C)=O)CC1 29262,N1(C(c2ccc(CC)cc2O)=O)CC2CC(NC(c3snc(Cl)c3Cl)=O)CC2C1 29263,N1(C(CC2CC(C)(C)OCC2)=O)CCC2(CCCN2C(=O)C(O)C2CCC2)C1 29264,c1(C(N2C3(CNC(C4CNC(=O)N4)=O)CC(C2)C3)=O)cn2cc[nH]c(=O)c2n1 29265,S(=O)(=O)(c1c[nH]ccc1=NC1CC1C1CCCC1)NCc1scc(C(C)C)n1 29266,C=C(C)CC(C(=O)NCCCCNC(N)=O)NC(c1ccsc1)=O 29267,C1(C)(C(N2CCC(NC(c3ccn(C)c3)=O)C(CO)C2)=O)CC(C2CC2)=NO1 29268,Cc1ccc2[nH]nc(C(N3CC(F)(F)CC3CNC(C3CCC(C)O3)=O)=O)c2c1 29269,Cn1cc(-c2cc(C(=O)NC3(C)CN(C(C4(c5nccs5)CC4)=O)C3)no2)cn1 29270,C1(C#CC(=O)N2CCC(OCCNC(C3CC3F)=O)C2)(CC)COC1 29271,C1(C)(NC(C=CC)=O)CCN(C(c2oc(-c3ccccc3)nc2C)=O)C1 29272,C1(CNC(CC(CC)SC)=O)CCCCCN1C(=O)COc1cc(C)ccc1C 29273,n1(CC)nnc2c(N3CC4CC(NC(=O)Cc5ccc(Cl)cn5)C4C3)ncnc12 29274,N1(C(CNS(CCCC)(=O)=O)=O)CC2CCCN(C(=O)C(C)C(F)F)C2C1 29275,S(=O)(=O)(c1ccc(=NCC23CCC(CO2)C3)[nH]c1)N1C(CC)CCCC1 29276,N#CCCCN=c1[nH]c(N2CCC3(CC(C(F)F)=NO3)C2)nc2ccccc12 29277,Cc1oc(C(=O)NCCNC(C2CCCCN2C2CCCC2)=O)cc1S(N)(=O)=O 29278,C(=O)(C(C(=O)NCC(C)(C(C)C)NC(=O)C1=CCC1)c1ccccc1)OCC 29279,C(=O)(CCC(C)(C)NC(c1cc[nH]c(=N)n1)=O)N(C)Cc1onc(CC)n1 29280,c1(CCNC(C2CCN(c3ncc(I)cn3)CC2O)=O)c[nH]c2ccc(Br)cc12 29281,c1(C(=O)NCC2CCCC(NC(CCCSC)=O)C2)coc2c(F)cc(Cl)cc12 29282,c1(C(N2CC(CC)(NC(=O)C(C)OCCC(C)C)C2)=O)cc(N)c(Cl)cn1 29283,N1(C(C(c2cccc(O)c2)C)=O)CC(CNC(C2(C)COC2)=O)C(C)C1 29284,c1(OCC)ncccc1CC(N1CC(CNC(=O)C=C=C(C)C)(OC)C1)=O 29285,N1(C(C(n2ncc(C)c2)C)=O)CCCCC1CC(N1CC(F)(CF)C1)=O 29286,C(c1cnc2ccccc2n1)=CC(=O)NC1CC2CC1N(C(c1cocn1)=O)C2 29287,C1(C(N(CCCCC(=O)NCC2CC(F)(F)CO2)C)=O)CC2COCC2C1 29288,N1(C(C2CCCN(C(=O)OC)C2)=O)CC2(CCC2NC(=O)C(F)=C(C)C2CC2)C1 29289,C1(NC(CS(=O)(=O)NCC)=O)CN(C(C2(C)CCC(=O)N2)=O)CCC1C 29290,C(=O)(C(CC)CCc1ccccc1)NCCC(C)NC(CC=CCC)=O 29291,c1(C(N2CC(C#C)N(C)CC2)=O)sc2ccccc2c1C(=O)OC 29292,C1(C(N2C(CCNC(C(=Cc3cn[nH]c3)C)=O)CCC2)=O)CCCC2CCCN12 29293,CCN=c1ccc(C(=O)NCC23CC2CN(C(c2cnc(C(C)C)o2)=O)C3)c[nH]1 29294,c1(NC(C2CC3CCN(C(CCC(C)C)=O)CC32)=O)cccc2ccccc12 29295,C1(NC(C(=O)N(C)Cc2cccc(C(=O)OCC)c2)=O)CCC(P(C)(C)=O)C1 29296,C1(O)(CC(=O)NC(C2CCCCC2)CC)CN(C(=O)Cc2nocc2C)C1 29297,c1(C(=O)NC(CC)C(C)(C)O)cc(S(=O)(=O)N2CCOCC2)ccc1F 29298,CC1CC(C)N(C(c2cccc(NC(N)=O)c2)=O)CCN1C(=O)C=C1CCCC1 29299,C1(O)(CCNC(c2c(OCC)ccs2)=O)CCN(C(=O)C(C)P(C)(C)=O)CC1 29300,N1(C(C(C=C=C)C)=O)CC2CCC2(CNC(c2cnoc2CC(C)C)=O)C1 29301,N1(C(C#CC(=O)N(C)C)=O)CC2CC(NC(=O)CSC3CC3)C2C1 29302,N1(C(C(COC)C)=O)CCC(CNC(c2c(N)cnn2C)=O)C1(C)C 29303,C1(C)(OC)CC(NC(C2(C)CN(C(C3(OC)CCOC3)=O)C2)=O)C1(C)C 29304,Cc1ncc(Br)c(NC2CCCC2C(=O)Nc2ncc(Br)cc2I)n1 29305,CC1CC(=O)NC(C(=O)N(C(C)CNC(c2ccc(CO)cn2)=O)C)C1 29306,C1(NC(CCC#CC)=O)CC(O)CN(C(=O)CCC2CC2)C1 29307,c1(C(=O)NCCC(C)NC(C2N(C(C)=O)CC(O)C2)=O)ccc(=O)n(C)c1 29308,C(=O)(C1=CCCOC1)NCC1CCC(NC(c2ccc(OC)s2)=O)CC1 29309,c12cccc(n1)NCC2.c1(C(CCCOC)(C)OC)nnnn1C(C)C 29310,c1(CNC(=O)NCC2(C)N=C(C)SC2)cc(C)c(F)cc1Br 29311,n1(CC)nnnc1C(c1ccn(-c2ccccc2)n1)NCc1csc(COC)n1 29312,N1(C(C)=O)CCN(C(c2cccc([N+](=O)[O-])c2C)=O)CC12CCCCC2 29313,N1(C(CC(C)C)=O)CCCCC1C(N1CCC(C)C1C)=O 29314,C#Cc1ccc(C(N2CCN(C(C3C4CCCC34)=O)CC2CC(=O)NC)=O)nc1 29315,C(=O)(C(C)CCC(C)(C)C)NC1C2CCN(C(c3cc(C)c(O)c(C)c3)=O)C2C1 29316,C1(NC(c2n(C=C)nnc2)=O)CCC(C)N(C(C23CC4CC2C3C4)=O)C1 29317,C12(CNC(c3ncc(C)c(C)c3)=O)CCC(CNC(=O)COC(F)F)(CC1)OC2 29318,c1(C(=O)NCC(CC)NC(=O)C(F)(CC)C(=O)OC)ccnc2nc(C)nn12 29319,c1(NC(C(N2CCOCC2)C)=O)cc(CNC(c2csnc2C2CC2)=O)[nH]n1 29320,CCCC(C(=O)NC1CCC(CNC(c2ccc(F)cc2)=O)C1)N(C)C 29321,N1(C(c2nn(C)c(I)c2)C(=O)NCC(F)F)CC(N=[N+]=[N-])CCC1(C)C 29322,c1(C(=O)NCCN(C(C(C)C)=O)C2CCCC2)cc(CN(C)C)ccc1O 29323,c1(C(C)NC(=O)Cn2cc(C(C)O)nn2)cc(Cl)ccc1Oc1ccccc1 29324,C1(CNC(c2cnc(SC)s2)=O)CN(C(c2cnn(CC3CC3)c2C)=O)CCN1C 29325,C(=O)(C(CN=[N+]=[N-])NC(=O)C#CC(C)(C)O)Nc1cnc(C)nc1 29326,C(=O)(CCCCC(=O)NC)NCCOCCCNC(C(CCC)NC(N)=O)=O 29327,C12(NC(C(C)OCCC(C)C)=O)COC(C1)C(NC(c1cccc(CO)c1)=O)C2 29328,C1(C(=O)NC(c2nc(C(C)(C)C)no2)CC)CCC(=O)NC1 29329,C1(C(=O)NC(C)CN(C)C(C2(C#N)CCCC2)=O)(COC)CC=CCC1 29330,C1(NC(=O)CN2CCCCC2)CN(C(=O)C=CC2CCCO2)Cc2nccn2C1 29331,N1(CC(N2CCCC(CNC(=O)Cc3ccsn3)CC2)=O)CCCCC(O)C1=O 29332,c1(OC)ncccc1CC(=O)NCC1C2CC1N(C(=O)CN1CCCC1C)C2 29333,N1(C(c2nncc(OC)c2)=O)CCC(O)CC1C(=O)NC1CC1c1ccco1 29334,CC1CC(NS(=O)(=O)Cc2cccc(O)n2)CN(C(=O)OC(C)(C)C)C1 29335,N1(C(Cc2ccc(NC(C)=O)cc2)=O)CC2CCC(N(C)C)CC2C1 29336,C(=O)(C(C)N=c1cc[nH]cc1)NCCN(C(COCCCC#C)=O)CC(C)O 29337,c1(C(=O)NCC2N(C(C(C)CC3CCCC3)=O)CC(O)C2)nc(O)nc(O)c1N 29338,c1(N2CC(NC)C2)nc(NCC2COCC(C)O2)c2ncn(C(=O)OC)c2n1 29339,C1(C(=O)NC(CC)(C)O)CC(O)CN1c1nncs1 29340,C1(C(=O)NC(c2ncc(C)[nH]2)CC)C2CC3C(C2NC(C2C4COCC24)=O)C13 29341,C(=O)(CCCC(=O)NCC(=O)Nc1cccs1)OC(CC(C)C)c1nn[nH]n1 29342,Cc1cccc(C2(C(=O)NC3CCCC(CNC(c4cocc4C)=O)C3)CC2)c1 29343,C(=O)(C1=C(CSCC(=O)NCC(CNC(=O)C(C)(F)F)CO)NC(=O)NC1C)OCC 29344,c1(C(=O)NC2C(NC(c3[nH]c(=N)sc3)=O)C2)cnc2cccnn12 29345,C1(C(=O)NCCN(C(C(C)OC)=O)Cc2ccccc2)CC2CCC1CC2 29346,c1(C(=O)NC2CCC(NC(CC=C(C)C)=O)CC2)[nH]nc([N+](=O)[O-])c1Cl 29347,N1(C(c2c(C)nns2)=O)C2CCC1CN(C(c1cccc(C(F)F)n1)=O)C2 29348,C1(CCOC)CN(C(c2[nH]c(C)nc2C)=O)CCN1C(c1cc(C)ncc1C)=O 29349,c1(C(N2CCCC2C2CCOC2)C(=O)NC(CC)(C)C)ccc(C)c(C)n1.CCOC 29350,C(=O)(CCCC(=O)N1CC(CNC(C2(F)CCOC2C)=O)CC1C)OCC 29351,C(C#Cc1cc(Cl)cnc1F)NC(N1CCC(O)(C(C)O)CC1)=O 29352,C1(NC(C(C)OC2COC2)=O)CCC2CN(C(c3ccnn3C)=O)CCC2C1.CC 29353,N1(C(C2CCC(C)O2)=O)CC2CCCC1(CNC(c1ccc3c(c1)CCO3)=O)C2 29354,c1(C(N2CCC(C)(NC(CCN(C)CC)=O)C2)=O)cc2n(c1)CCSC2 29355,C12(C(N3CC(C)C(NC(=O)Cn4ccc(=N)[nH]4)C3)=O)CCCCN1CCC2 29356,N1(C(CCC2(C#N)CCC2)=O)CCOCC(NC(C2CC3CCCCC23)=O)C1 29357,CC1(C)C2CN(C(c3ccnc(Br)c3)=O)C(C(=O)N3CC(O)CO3)C12 29358,C#Cc1ccc(C(=O)NCC2(NC(c3cncc(OC)c3)=O)CCCCC2)o1 29359,CCCC(C)CC(C(=O)NC(C)(C)C)N1CCCC1(CC)CO 29360,C1(NC(CC(COC)C)=O)(CO)CCCN(C(=O)Cc2conc2C)C1 29361,c1(C(N(CCN2CCOCC2)CC)=O)cn(CCNC(=O)Cc2ccsn2)nn1 29362,N(C1CC(F)(F)c2ccccc21)C(=O)C(N1CCC(O)(c2cccc(F)c2)C1)=O 29363,c1(C(C(=O)NCCC(C)NC(=O)CCCCCSC)N(C)C)c(F)cccc1F 29364,CCCC(CCNC(=O)CN(C(=O)CC1CCCN1C)C(C)C)C1CC1 29365,C1(CC)CCN(C(=O)CCOC)C1C(=O)Nc1ccnc(C(=O)OC)c1 29366,S1(=O)(=O)c2ccc(cc2)OC(=O)N2CCCC(C2)N1.C=CCOCC 29367,C1(C(N2C(C(C)NC(c3c(C)occ3)=O)CCC2)=O)CSC(c2ccccc2)=N1 29368,c1(C(=O)NCC(COC)NC(=O)CCc2cnc(C)s2)ccnn1C 29369,c1(C(N2CCC(CCNC(C(C)=CC)=O)CC2C)=O)cccc2c1ccn2C 29370,C1(NC(C)=O)CCCN(C(c2cnc(CNC(C3CCCC(C)C3)=O)nc2)=O)C1 29371,n1(CC)ncc(C(=O)N(CCCNC(=O)COCP(C)(C)=O)C2CC2)c1Cl 29372,C1(CNC(C2C(C(=O)OC)C2)=O)CCCC(CNC(c2ccc(C)cc2)=O)C1 29373,C1(C(N2CCC(c3cn(-c4ccncc4)nn3)C2)=O)(SC)CC(=O)C1 29374,CC1CN(c2cc(NC3CC4OC(=O)CC34)ncn2)CCC1N(C)C 29375,c1(CC)ccc(C(=O)NCC2(C)CCCN(C(c3csnn3)=O)C2)c(O)c1 29376,C1(C(=O)NCC)(CC2CCOC2)CC12CCC2.c1(C(N2CCC2)=O)ccc(C)cc1 29377,N1(C(c2c(CCNC(CCN(CCC)C)=O)n[nH]c2)=O)CCOCC(O)C1 29378,C1(NC(CC(=C2CCCC2)NC(C(C)=CCO)=O)=O)CC2CC1CC2CO 29379,O=S(=O)(c1cnc(NC2CC(CO)C2)c(Cl)c1)NC1CCC2(CC1)CC(O)C2 29380,Cc1ccc2c(N3CCSCC3C(=O)NCc3ncco3)ncnc2c1 29381,c1(CN(C(c2snc(C)n2)C(=O)NC2CCC2)C)ccnc(Cl)c1 29382,c1(CNC(C23CC(COC)(C2)C3)=O)ccc(CO)cc1.C1(C)CC(=O)N1 29383,N1(C(C(c2ccccc2F)C)=O)CCCC(CO)(NC(c2cccn2C)=O)C1 29384,CC(C)(O)C(F)C(=O)NCCC1CC(F)CN1C(=O)C1CC1 29385,C(C(C(C)(C)C)NC(=O)CCc1nc(C(C)OC)no1)NC(C1C(CC)C1)=O 29386,c1(C(N(C(C)CC(=O)N2CC(CN=[N+]=[N-])C2)C)=O)ccc(Cl)nc1 29387,c1(N2CCN(C(C(=O)NC)C)CC2)nccc(=NC(C)c2ccn(C)n2)[nH]1 29388,N1(C(C(C)=C(C)C)=O)CCOC2CN(C(C3COCCC3(F)F)=O)CC12 29389,c1(NC(C2CN(S(CC)(=O)=O)C2)=O)cc(-c2ccco2)nn1C 29390,CC1CCN(C(=O)Cn2[nH]cnc2=N)C(C(N2CCCC(CO)(CO)C2)=O)C1 29391,C1(CNC(COC(C)C)=O)CCN(C(=O)C(C)(C)CC2CCOCC2)CC1C 29392,N1(C(CCC)=O)CCc2nc(CNC(C3CC(C)CC(C)C3)=O)sc2C1 29393,c1(CC)nn(C)cc1C(N1CCCC(NC(c2cc(C(=O)OC)c[nH]2)=O)C1)=O 29394,CCCCCC(C(=O)NC1CCCCC1)N1CCC2(CSC2)C1 29395,C(CN=c1ccc(N2CCc3nncn3CC2)n[nH]1)OCCN(CC)CC 29396,N1(C(C(CC)=CCCC)=O)CCN(C(=O)CCc2nncnc2O)C(CO)C1 29397,N1(C(=O)COC2CCCC2O)CC2CCCC(C1)N2C(C1CC(F)(F)C1)=O 29398,C(C(CC1CCCC1)C(=O)Nc1ccc(SC)cc1)NC(CC(=O)NCC#C)=O 29399,c1(C(=O)NC(CCCNC(C(Cn2ccc(C)n2)C)=O)(C)C)cnc(N)c(N)c1 29400,c1(C(N2CCN(C(CNC(C(C#C)(C)C)=O)=O)CC2)=O)ccnc2c1nnn2C 29401,CC(C)C(C(C)NC(c1ncccc1C(F)F)=O)NC(c1ccc(CO)nc1)=O 29402,C(N=c1cc(NCC(Cc2ccccc2)N(C)C)nc(C)[nH]1)C1(OCC)CC1 29403,N1(C(c2c(C)c(Cl)cnc2)=O)CCCC(C2CN(C(=O)COC3COC3)C2)C1 29404,c1(N2C3CN(C(C4CC(C)(C)OC4)=O)C(C3)C2)ccc([N+](=O)[O-])c(C#N)c1 29405,c1(CN2CCC3(C(C(=O)NCCc4ccc(F)nc4)C3)C2)cc(Cl)cc(Cl)c1O 29406,c1(CNC(C2(CNC(c3n(C)nnc3)=O)CCCO2)=O)cccnc1F 29407,C1(CN(C(=O)Cc2cn(C)cn2)C)CCN(C(c2csc(C#N)c2)=O)CC1 29408,C(=O)(CCCCCNC(N)=O)NC(C)CCCCNC(C12CCC1C2)=O 29409,C1(CC)CC(C(=O)NCC(c2ccsc2)O)CCN1C(c1csc(C)n1)=O 29410,C12(CC(N3CC(C4N(C(=O)COCCF)CCC4)(O)C3)=O)CCC(CC1)C2 29411,N1(C(C(C)=C(C)C)=O)CCN(C(c2nn[nH]c2C(F)(F)F)=O)C2(CCC2)C1 29412,N1(C(C(CC=C)CC)=O)CCC2(CC1)CN(C(=O)C=Cc1ccn(C)c1)C2 29413,C1(C(N2CC3CC(C2)C(=O)N3)=O)CCCCC(C)(C)C1.C1(COCC)(CC)CC1 29414,Cc1nn(C)c(Cl)c1C(N1CCC(F)(CNC(=O)CN(C)C2CC2)CC1)=O 29415,C1(NC(c2ccnc(C)n2)=O)CCCCCN(C(c2ccc(C3CC3)cc2)=O)C1 29416,c1(NCCNC(c2nc(C(F)(F)C(=O)O)cs2)=O)ccc(F)cc1 29417,c1(C(=O)NC(C2N(C(C(CC=C)C)=O)CCC2)C)ccc(C)c(OC)c1 29418,C1(C(=O)NCC2N(C(C(CC)N3CCCC3=O)=O)CC=C2)CC2(C1)CC(C)(C)C2 29419,C(=O)(C1=CCCN(C(C2CC2C(C)(C)C)=O)C1)NC1CN(C)CC1(F)F 29420,C1(NC(N(CC(O)COCc2ccccc2)C)=O)CC12CCCC2 29421,N1(c2nnc(-c3c(C)ocn3)n2CC2CCOC2)CC2CC1c1ccccc12 29422,C(C(CCC(F)(F)F)NC(c1ncc(Br)cc1F)=O)OC 29423,C(=O)(C1=NOC(C)(C)C1)NCC1C(N(C)C)CN(C(CC2CCCN(C)C2)=O)C1 29424,C(CC(CC)C(=O)NCC1CN(C(=O)CN2CCN(C)C(=O)C2)CC1(C)C)=CC 29425,C1(NCC(C)Cn2cccn2)CCCC1C.C1(OC)CN(C(=O)OC(C)(C)C)C1 29426,C1(NC(C2(OC)CCN(C(CCC#C)=O)C2)=O)CCn2nccc2C1 29427,c1(N2CC(N(C)Cc3cnn4c3CCCC4)C2)ncnc2cc(I)sc12 29428,C(=O)(C1CCCc2nc[nH]c21)NC(C)(CNC(c1snc(O)c1Cl)=O)C1CC1 29429,CC(C)C(C(F)F)NC(C1CCN(c2cccc(C(=O)O)c2)CC1)=O 29430,c1(C(N2CCC(CC(C)NC(C3C(C=C)CC3)=O)CC2)=O)c(C)nn(CC)c1C 29431,N1(C(CC=CCC)=O)CCOC(CNC(c2sc(-c3cnn(C)c3)nc2C)=O)C1 29432,C(=O)(C1=C(C#N)CCC1)N(C1CCCC(NC(=O)C=CC2CC2)C1)C 29433,CCC(CC)(C(=O)NCCC1CN(C(C2(COC)CC2)=O)CC(C)O1)OC 29434,C12(NC(=O)C=C3CCC3)CCCN(C(=O)CCOC3COC3)CC1C2 29435,CC1CN2CC(C)N1C2.C1(C)(n2cc(-c3cnccc3Cl)nn2)CCC(=O)N1C 29436,C(=O)(CN=c1cc[nH]cc1)NC1CC(NC(c2cc(CC)no2)=O)C12CCC2 29437,C(=O)(CCC(C)(C)C)N1CC(NC(C(CC)C)=O)C(C)C1 29438,C1(C(N2CC(O)(CCNC(C(C=CC)O)=O)C2)=O)COc2ccccc2O1 29439,c1(OC)cc(C(=O)NC2CCCCC2NC(c2ncccc2N)=O)cc(F)c1F 29440,Cc1nc(C)c(C(=O)NC(C2CCN(C(C3CCCC3C(C)C)=O)CC2)(C)C)[nH]1 29441,c1(C(N2CC(C)(CC(=O)NCc3cc(F)ccc3Cl)C2)=O)cc(F)ccc1C#N 29442,c1(CC(=O)NC2(CCNC(CCCSC)=O)CC2)ccc(O)c(F)c1 29443,C1(NC(C2(CC#C)CCCC2)=O)CC2CC1CN(C(c1ncc(C(N)=O)s1)=O)C2 29444,C1(C(N2CCC(O)(CC)C2)=O)Cc2nnsc2S1 29445,C12(CNC(c3cc(SC)nn3C)=O)CN(C(=O)C=CC3CC3)CC1CCO2 29446,C1(NC(C2CCOCC2)=O)CS(=O)(=O)C2CN(C(c3ncccc3Cl)=O)CC12 29447,C1(CC)CCN(C(=O)OC(C)(C)C)C1CNC(c1ccc(OCCO)nc1)=O 29448,c1(NC(C(c2cccc(Br)c2)NCc2nc(C)sc2)=O)cc(F)ccc1O 29449,C1(F)(CNC(=O)Cn2c(O)nnc2O)CCCN(C(C2C3CC4C(C3)C24)=O)C1 29450,N1(C(c2nn[nH]c2Cl)=O)CCN(C(=O)C=CBr)C2CCCCC2C1 29451,C1(CNC(COCCCCC)=O)CC(CO)CO1.C12CC(C1)CNC2=O 29452,O=CN1CCCN(C(=O)CC2CC=CCC2)CC1 29453,C#CC1(O)CCN(C(=O)C(CC(=C)C)NC(c2ccccc2C#N)=O)C1 29454,N1(c2nnc(-c3ccc(C(F)F)s3)n2CC2CCC2)CCc2nc(Cl)ccc2C1 29455,c1(C(N2CCC(NC(C(CCC)OC)=O)C2)=O)coc2cc(OC)ccc12 29456,Cc1oc(C(=O)NCCCN(C(C2(C#N)CC2C)=O)C2CC2)cc1S(N)(=O)=O 29457,CN1C(=O)CCN(C(C2CCC3C2C3(F)F)=O)c2ccc(F)cc21 29458,c1(NC(CC2CCN(Cc3ccc(OCC)c(Cl)c3)C2)=O)cc(Br)c(Cl)cc1F 29459,O=C(C1=NN2CCCN=C2N1)NCC1CC1NC(C1(Oc2ccc(F)cc2)CC1)=O 29460,C1(C)(C(=O)NC23CC(C(=O)OC)(C2)C3)CCN(C(=O)CCCCc2ccccc2)C1 29461,c1(C(N(C)CC2CCCN(C(C(C)S(C)(=O)=O)=O)C2)=O)ccc(S(C)(=O)=O)s1 29462,C1(n2c(-c3ccc(F)cc3Cl)nc(C3CCN(C)CC3)n2)CCN2CCOCC12 29463,C(=O)(C(CO)C(C)(C)C)NC(CNC(c1ccc(C#C)o1)=O)CC(C)C 29464,C1(CNC(c2c(CC)onc2)=O)CN(C)CCN1C(=O)CCc1ccn(C)c1 29465,N=c1[nH]c2cc(C(=O)NCC3C4CN(C(=O)CSc5nncs5)CC34)ccc2o1 29466,c1(C(=O)NC(CC)C(=O)O)cc(Br)c(C(F)(F)F)cc1OC.c1(S)cccc(F)c1 29467,N1(C(CC(c2scc(C)c2)O)=O)CCC(C)C(Cn2cc(CNC=O)nn2)C1 29468,C1(NC(C23CC(C)(OCC2)C3)=O)CCC2CN(C(=O)C(C)(C)C3CCC3)CC12 29469,c1(C(N2C(C(=O)Nc3ccc(C#N)cc3)CC(F)C2)=O)c(Br)cc(F)c(Cl)c1F 29470,c1(C(=O)NC2C(CNC(C(C)(C)c3ccc(Cl)s3)=O)CCC2)cc2n(n1)CCO2 29471,N1(CCNC(=O)CC(F)(F)F)C(=O)CCN(CC2CCCc3nc[nH]c32)C1=O 29472,O=S(=O)(c1cc(Br)c(F)cc1F)NCC1CCN(Cc2cc[nH]n2)C1 29473,C(=O)(C(C)CCCC(C)C)N1CC(CCNC(=O)C(C)C2CCOC2)(OC)C1 29474,CONC(=O)C(=O)NC1CN(C(=O)COCP(C)(C)=O)CC1C 29475,C(=O)(C(C)(C)CCC#N)NC1CN(C(C(c2ccc(F)cc2F)C)=O)C1 29476,n1(CC)c(S(=O)(=O)NCC2COC(C)(C)C2)cnc1C 29477,Cc1coc2ccc(C(=O)NC3CCC3NC(C3CC3C)=O)cc12 29478,CCC(CC(=O)N1CCOCC1CCNC(=O)C=Cc1nccs1)C(F)F 29479,CC(C)(C)C(CO)NC(C1CCN1C(=O)CCC1CCCCC1)=O 29480,C1(CCC)(NC(=O)CC2(OC)CN(C(C3(CSC)CC3)=O)C2)CCNC1=O 29481,C(CC(=O)NC1(CO)CC2CCCC12)(CC(C)C)NC(C(C)NC(=O)OC)=O 29482,N1(C(CCCC#C)=O)CC2CCCC2C1C(=O)NC(C)CC(=O)NC 29483,Cc1cc(C(=O)N(C)C)c[nH]c1=NCc1ccc2c[nH]nc2c1 29484,C1(CC=C)(NC(c2sc(COC)nc2C)=O)CCN(C(c2ncoc2C)=O)C1 29485,c1(NC)ccc(C(=O)NCCCCC(C)NC(c2cccc(F)n2)=O)cc1 29486,C(C(F)(C(=O)NCC1CC2CCC(C1)C2)C(C)C)NC(CCC(CC)=O)=O 29487,C(CCC1CC1)(C(=O)NC1CC2C=CC1C2)NC(C(C1CCC1)OCC)=O 29488,c1(CC)cc(C(N2CCC(N(C(=O)CC3CCCC(O)C3)C)C2)=O)c(C)o1 29489,C(=O)(C1(C)CCn2c(C)nnc21)N1CC(O)(CNC(C(CC)O)=O)C1 29490,C(=O)(C1CCCn2ncnc21)N1C2CN(C(c3nccc(OC)c3C)=O)C(C2)C1 29491,c1(OC)cc(C)c(C(=O)NC2CN(Cc3ccncc3Cl)CC2O)c(C)c1 29492,N1(C(C(CC(C)C)ONC(C2CC(=C)C2)=O)=O)CC2CCC1C(O)C2O 29493,C1(C(=O)NC2C(OC)CN(C(c3cnc(C)cc3Cl)=O)C2)CCc2ccnn2C1 29494,C1(C(=O)NC(CCNC(c2nn(CC)c(O)c2)=O)C(C)C)CCc2nccn2C1 29495,Cc1nc(C2CC2)nc(C)c1C(=O)NC1CCN(C(C2CC(C)OC2C)=O)C1 29496,C(=O)(C(O)Cc1cnn(C)c1)NCCN(C(C(c1ccc(Cl)s1)C)=O)C1CC1 29497,C1(COC)CCCCN(C(c2ccc(SCCCC3C=CCC3)cc2)=O)C1 29498,c1(C(N2C(C)CC(NC(C3CC(C#C)(O)C3)=O)C2)=O)cccc2c(C)[nH]nc12 29499,N12CC(C3(CC3)C1)CSCCC2=O.n1(CC)c(ON(C2CC2)CC)nnc1CO 29500,c1(COC)ccc([N+](=O)[O-])cc1.CON1CC23OCC(CC1=O)(C2)C3 29501,N1(C(c2cc(OC)ncc2)=O)CCC2CN(C(c3cnn(C)c3Br)=O)CC12 29502,c1(C(COC)N(C)C(c2nnsc2C)=O)ccc(Cl)cc1 29503,c1(OC)c(F)ccc(C(N2CC(NC(c3ccc(Cl)o3)=O)CC2C)=O)c1F 29504,CC(CCC(=O)N1CCC1Cn1cc(-c2ccccc2Cl)nn1)N(C)C 29505,c1(C(=O)OCC)nc(C(=O)NC(C)CNC(=O)C(C)(C)c2csc(C)c2)c(C)s1 29506,O(NC(=O)C(CNC(c1cnsc1)=O)C(C)(C)C)CC(C)(C)C 29507,C1(CC(C)C)CC1N=c1[nH]c(N2CCCC(c3cccnc3)C2)nc2c1CCC2 29508,NS(=O)(=O)C1CC(C(=O)NCc2cccc(CNC(C3CC3CF)=O)c2)C1 29509,c1(C(=O)NC2C(NC(CCOCCC)=O)CC2)csnc1C 29510,C#CCC(C(=O)NC)NC(C1CC(NC(=O)C(C)OCC2CC2)C(O)C1)=O 29511,C1(F)(CNC(CNC(=O)OC)=O)CCN(C(c2coc(C(C)(C)C)n2)=O)C1 29512,c1(C(N(C)CCNC(=O)CCOC2CCC2)=O)c[nH]c2cccc(F)c12 29513,c1(C(N2C(c3ncc(-c4ccc(OC)cc4)[nH]3)CCC2)=O)c(Cl)cc(Br)cc1Cl 29514,c1(C(C)C(N2CCCC3CC23)=O)cc2ccccc2o1 29515,C(=O)(CC1=NN(C)C(=O)C1)N1CCC(C)CC1CNC(C1COC(C)(C)CO1)=O 29516,C(CC(C(C)(C)C)NC(c1cc(C2CC2)cs1)=O)N(C(=O)CCCN1CCCC1)C 29517,C1(N(C)C(C2CCNC2=O)=O)CN(C(c2cc(C(C)(C)C)ccn2)=O)CC1(C)C 29518,N1(C(c2c(OC)n[nH]c2)=O)CC(C)(C(=O)NCc2ncc[nH]2)CC1(C)C 29519,C1(NC(Cc2cc(COC)on2)=O)CN(C(=O)CP(C)(C)=O)CCC1C 29520,C(C(N=c1cc(C)nc(NC2CC3(C2)CC(O)C3)[nH]1)C1CC1)OC 29521,c1(NC(=O)CCC2(N3CCCC3)CCC2)ccc(NCCc2ccc(Br)cc2)cc1 29522,Cc1nc(Br)sc1C(=O)NC1CCC(NC(=O)CCc2cccn2C)CC1 29523,N1(C(CC2C(OCC)C2)=O)CCC2CCN(C(=O)CO)C2C1 29524,C1(C(N2CC(CC=C)(NC(CC=CC=C)=O)C2)=O)CCCC2(CCC2)O1 29525,C(=O)(CC(C)(C)CC(=O)NCC1CCCN1C(C1CC2(CCC2)C1)=O)OCC 29526,C(CC(C)C)(C(=O)NCC(CNC(=O)CCc1cnoc1)CO)OC 29527,CN=c1nc(C(=O)NCC2(CNC(=O)CC(C)P(C)(C)=O)CCC2)cc(C)[nH]1 29528,C1(CNC(C(CC(C)C)C)=O)CC2CCC(C1)N2C(c1nn(C)cc1N)=O 29529,C=CCCC(C(=O)N(C)Cc1cn(C)nc1C)NC(=O)CC1CCCCN1C 29530,c1(-n2cc(CN(C(COc3ccn(C)n3)=O)C3CC3)nn2)cccnc1Br 29531,C1(COC)CC(Cn2cc(C3CC3)nn2)N(C(=O)C(C)(C)F)C1 29532,C(N=c1[nH]c(=NCC2CCOC2)c2[nH]ccc2[nH]1)C1CC(N(C)C)C1 29533,c1(C(N2CCC(C3(C(F)(F)F)N=N3)C2)=O)cc2ccsc2s1 29534,c1(CC)ccc(C(=O)NC2CCC2NC(=O)CCc2nnc(O)nc2O)cc1N 29535,N1(C(=O)Cc2ccc(Br)cn2)CC2CCC(C1)C2NCc1c(F)cccc1Cl 29536,N1(C(CC(C)C2CCCCC2)=O)CCC2(CC1)CN(C(=O)C=CI)CCO2 29537,c1(C(c2cn(C(CCCNC(N)=O)c3ccccc3)nn2)CC)cccnc1 29538,c1(C(N2CCC(N(C(CS(CC)=O)=O)C)C2)=O)ccc(Br)cc1OC 29539,N1(C(C2(CC)CC(F)(F)C2)=O)CCOc2cccc(C(=O)O)c2C1 29540,C1(O)(CC(N2CC(O)(CN(C)C(c3ccc(NC=O)cc3)=O)C2)=O)CCCCC1 29541,N1(C(C2OCCN(C)C2)=O)CC(NC(c2cccnc2Cl)=O)CC2(CC2)C1 29542,C1(CNC(C2(N(C)C)CC2)=O)COCCN1C(c1ccc(Br)s1)=O 29543,C(C(COC)C(=O)NC(Cc1ccco1)C(=O)NCCC1CC1C)OC 29544,C(C)(CO)(C(=O)N1CC(C)(C)C1C(C)C)NC(c1c(OC)nsc1)=O 29545,N1(C(c2c(C)sc(O)n2)=O)CC(C)C(NC(c2cc[n+]([O-])cc2)=O)C(C)C1 29546,c1(C(=O)OC)cc(C)c(F)c(S(=O)(=O)NC(c2c(C)ccnc2OC)=O)c1 29547,C1(N(C)C)CCCCC1CNC(=O)C1=C(Cl)CC1.C12CCCC1C(=O)N2 29548,c1(CC(=O)NCCOCCNC(COC(CC)C)=O)csc(Cl)n1 29549,c1(CNS(C)(=O)=O)cccc(C(=O)NCC2CC(NC(C3(C)CCC3)=O)C2)c1 29550,C(=O)(CCCCCC)N(C1CC(NC(COCC#C)=O)C1)C 29551,Cc1ncc(F)c(=NCC2(C)CCN(C(=O)CC3CCC(C)C(C)C3)C2)[nH]1 29552,N(C(=NCC(C)Oc1ccccc1F)NC1CCOCC1)Cc1cnc(C)o1 29553,C1(C(N2CCC(CNC(C(CCC)c3ccccc3)=O)C2)=O)CCC(F)(F)CC1 29554,c1(CC(=O)NC(C)CCNC(=O)CC2(C)OCCO2)ccc(C#N)nc1 29555,C=CCN=C(NCc1nnn(C)c1C(F)F)NCC(CC1CC1)CO 29556,Cc1ccccc1CC(C)C(=O)NCC(C(C)C)NC(=O)CN(C(=O)C(C)C)C 29557,C1(CNC(C2(N(C)C)CCCC2)=O)C2CC1N(C(C1CCS(=O)CC1)=O)C2 29558,C(c1ccc(C)c(Cl)c1)=CC(=O)NCC1C=CC(NC(Cc2ccc(C)s2)=O)C1 29559,c1(COC(C(c2ccoc2)NC(=O)OC(C)(C)C)=O)c(C)nc(O)nc1O 29560,C1(C(=O)OC)COCCC1NC(=O)CC1CSCCS1 29561,N1(C(CC2(COC)CC2)=O)CC2CC(NC(C3CCS(=O)(=O)CC3)=O)C(C2)C1 29562,c1(CC(=O)NC(C2CCN(C(c3ns[nH]c3=O)=O)C2)(C)C)c[nH]c2cnccc12 29563,S(=O)(=O)(c1ccc(NC2CC(C3CC3)C2)c(Br)c1)NC1(CC(C)C)CC1 29564,N1(CC)CCC(NC(=O)Nc2ccc(CO)cc2)C1c1ccc(C(F)(F)F)cc1 29565,C1(C(C)CNC(=O)C=CCO)CCN(C(C2CCC23CCC3)=O)CC1 29566,n1(C2CN(C(c3cccc(C)c3C)=O)C2)ccc(=Nc2ncnc3[nH]ncc23)[nH]1 29567,Cc1cnc(N2CCSCC2C)c(S(=O)(=O)N2CCOC(C3CCCC3)C2)c1 29568,C1(C)(CNC(CC(C)(O)c2ccccc2)=O)CCCN(C(C2(CF)CCC2)=O)C1 29569,C(=O)(C1=CCC(NC(c2ccc(C#N)n2C)=O)C1)NC1C(C=C)COC1 29570,C1(C(C)C)(CO)CCN(C(c2cnc(Cl)s2)=O)C1.C1(=O)C(=O)NCCN1 29571,C1(C(=O)NCCCN(CCCNC(=O)Cc2cccn2C)C)COC(C)(C)CO1 29572,Cc1coc(C(=O)C(=O)O)c1C.C(C)(CN(C(C1CC1NC(C)(C)C)=O)C(C)C)N 29573,C(=O)(CCS(N)(=O)=O)N1CCCC(CCCC(=O)N(C)Cc2onc(CC)n2)C1 29574,N1(C(C(CC=C)CC)=O)CCC2(CCCN2C(=O)CCCOC(C)C)C1 29575,CCCCC(CNC(c1ccc(OC(C)CC)cc1)=O)NC(C1CCCCO1)=O 29576,c1(CC(=O)NC2CCN(C(=O)C3=COCCO3)CC2O)ccc2c(c1)NC(=O)C2 29577,CC1(C)CN(C(=O)C(F)(F)F)CCS1.C1CCCCCn2cc(nn2)OCCO1 29578,C1(CNC(C(C(C)C)N(C)C)=O)CN(C(=O)C=CC(F)(F)F)CCC12CCC2 29579,C1(C(N2CC(CCNC(c3c(OC)n[nH]c3)=O)C2)=O)CC(c2cnn(C)c2)=NO1 29580,C1(C)(CNC(C2(CC=C)CCOC2)=O)CCN(C(C2(OC)CCSCC2)=O)C1 29581,C12CC(O)CN1C2=O.c1(C2(CNC(=O)CO)CC2)ccc(C(F)(F)F)cc1 29582,C(=O)(C1=CS(=O)CCC1)N1CCC(NC(C(C)NC(=O)CC(C)(C)C)=O)C1C 29583,N1(C(=O)CO)CCSC2CCCCC12.C1(OCC(=O)NC2(C)CCC2)CC=CC1 29584,C=C1CC2(C1)CC(C(=O)NC1CCOC(CNC(=O)CN3CCCS3(=O)=O)C1)C2 29585,C(=O)(CCCN(C)C(c1cc(Cl)c[nH]1)=O)NC1(C(=O)NC)CC1C 29586,N1(C(C(C)(C)NS(C)(=O)=O)=O)CCN(C(=O)Cn2[nH]cnc2=N)CC(O)C1 29587,N1(C(CN2C(C)CC2)=O)CCC2(CCC2)C(NC(=O)Cc2csc(S)n2)C1 29588,N1(C(c2c(CC)nc[nH]2)=O)CC2CC1CN(C(c1ccsc1-n1cnnn1)=O)C2 29589,CC(CC(=O)N1CCCC1CN(C(=O)C(C)(C)c1ccns1)C)P(C)(C)=O 29590,N1(C(C2C(=C)CC2)=O)CCC2(CCC2)C(CNC(c2ccc(N)cn2)=O)C1 29591,O=S(=O)(c1ccc2c(c1)CCC2)NCC1CCCCC1F 29592,CCC(C)C(C(=O)NCCN(CCOC)C(c1cnc(C)o1)=O)OC 29593,N1(C(C(=O)NC(CN(C(c2cnc(C3CCC3)s2)=O)CC)C)C)CCC(O)CC1 29594,c1(C(=O)NC2CC(C(N(CC(F)(F)CO)C)=O)C2(C)C)cnn(C)c1C#N 29595,N1(C(CC2CC(OC)C2)=O)CCCC(O)(CNC(=O)C=Cc2ccc(C)o2)CC1 29596,Cc1noc(CCC(=O)NC(C2CCN(Cc3nc(CC4CC4)no3)C2)C)n1 29597,N1(S(c2c(C)nc(C)s2)(=O)=O)CCCC2(CCS(=N)(=O)C2)C1 29598,C1(C(=O)NC2CC(O)(CNC(C3(CC(C)C)CC3)=O)C2)CCS(=O)(=O)N1 29599,CC1(NC(C2CCC(NC(C3CCCC3F)=O)CC2)=O)CC(F)(F)C1 29600,c1(C(=O)NCC2CCN(C(c3cc(C(C)=O)oc3)=O)C2)cnn(C)c1C 29601,c1(C(=O)NCC(C)NC(c2c(CC)nco2)=O)ccc(OCC(C)C)cc1 29602,c1(C(=O)NCC2C(NC(C=C(C)Cl)=O)COC2)cnn2c1C(C)CCC2 29603,c1(C(=O)NCC2(F)CCC(CNC(C(CC#C)O)=O)C2)cccc(C2CC2)c1Cl 29604,c1(OC)ccc(C(C)=CC(N2CC(OC)CC(NC(C3(O)CCC3)=O)C2)=O)cc1 29605,C12=C(C)NNC1=NC(=O)c1scnc1OC2.c1(C(=O)OC)cc(OC)ccc1Br 29606,Cc1ccncc1C=CC(=O)NCC(CC(C)C)NC(c1ccnc(C)c1C)=O 29607,C12(NC(CCC#CC)=O)CCOCC1CN(C(c1cc3sccc3s1)=O)C2 29608,c1(N2CC(CCOC)OCC2)nc(NC(c2cccc(F)c2)C)c2ncsc2n1 29609,S(=O)(=O)(CCCCCS(N)(=O)=O)N(CC(C)(C)C(F)F)CCCC 29610,N1(C(CCCC(N)=O)=O)CCCC12CCN(C(c1cnc3nccn3c1)=O)C2 29611,C1(C)(CNC(Cc2n(C)nnc2)=O)COCCN(C(C2CCC3CCC2O3)=O)C1 29612,N1(C(C(CNC(C(C)(C)OC(C)=O)=O)CC2CC2)=O)CCC(O)C(C)(C)C1 29613,Cc1cccc(C)c1OCC(=O)NCC1CC(NC(C2(C)CC3CCC2C3)=O)C1 29614,C12(NC(C3C4CN(C(C5OCC(C)(C)C5)=O)C3C4)=O)CCC(CC1)OC2 29615,CC1(OCC(=O)NCCCN(CCC(O)CO)C)CN(CCC2(C)CC(F)C2)C1 29616,C1(NC(=O)CC2CC=CCC2)CN(C(C2(CC(F)F)CC2)=O)CC12CCC2 29617,C1(CNC(C2(C(N(C)C)=O)CC2)=O)CC2CCC1N2C(=O)Cn1cc(CO)nn1 29618,CC1CCCCC1(C)C(N1CCC(CF)(NC(c2ccc(C(N)=O)[nH]2)=O)C1)=O 29619,N1(C(c2n(CC)ccn2)=O)CC2CCC1CN(C(=O)C(c1ccc(O)cc1)=O)C2 29620,c1(C(=O)NC(CC)CN(C(c2nccnc2C)=O)CC)ccc(S(=O)(=O)NC)o1 29621,C(CCS(N)(=O)=O)NC(C=C(C)CNC(C1CC1(Cl)Cl)=O)=O 29622,C1(C(N(CCC=C)CC)=O)(NC(C2(C(N)=O)CC2C)=O)CC(CO)C1 29623,N1(C(c2c(C)cncn2)=O)CCC2(CCC(NC(C3CCCOCC3)=O)C2)C1 29624,Cc1c[nH]c(CC(N)=O)c1C(=O)NCC1CCC(O)CC1 29625,N1(C(C2(CC)CC2)=O)CCC2(CC1)CCN(c1ncnc3c(C)cccc13)CC2 29626,c1(C(N2C(C)CC(CNC(CCc3cc(C)no3)=O)C2)=O)ccc(N)c(O)c1 29627,C1(C(N2C(C(=O)NCCC3CCCCC3)C=CCC2)=O)CC2CCC(C1)C2 29628,c1(OC)cccc(CC(=O)NC2CC(CO)N(C(c3cnc(C4CC4)s3)=O)C2)n1 29629,C#CC1CN(c2ncnc(N3CCCN(CCC)CC3)c2C)CCO1 29630,C1(C(=O)NCC(C)CC2CCCC2)CCCN(C(c2ccc(C(F)F)o2)=O)C1 29631,N1(C(CCC(N)=O)=O)CC2CC1CC2NC(=O)C#CC1CCC1 29632,C1(c2scc(C)n2)CCCN(C(=O)CNC(=O)CCC2CCCC2)C1 29633,C1(C(=O)NC(C)(CNC(=O)COC(F)F)C2CCC2)CCC1(F)F 29634,C#CCCC(=O)NC(C)C(CO)NC(=O)C(Cc1ccc[nH]1)NC(=O)OCC=C 29635,Cc1ccc(C(O)C(=O)NC2CC(NC(c3cnc(O)n3C)=O)C2)cc1 29636,Cc1nn(CC(N2CC3CCC3(NC(=O)CCCNC(N)=O)C2)=O)c(C)c1Br 29637,CC(C)CC(CNC=O)CC(=O)NC1CC1NC(c1ccc(CCO)cc1)=O 29638,C(=O)(CCCCN1CCCCC1)NC1CC(CNC(C=CCN(CC)CC)=O)C1 29639,CCCCCC(O)CC(=O)NCC12CC(NC(=O)CC3OCCC3(C)C)(C1)C2 29640,C1(CNC(CSCC=C)=O)CC2(CN1C(c1cc(C)no1)=O)CC2(F)F 29641,CCS(=O)(=O)CC(=O)NC1CCC(C)(CNC(=O)CS(=O)(=O)N(C)C)C1 29642,C(=O)(C1=CCC(C(F)(F)F)OC1)C(C(C)OC1CCCCC1)=O.C1(N)CC(C)C1 29643,CC1CC(CCNC(c2ccc(C(N)=O)[nH]2)=O)CCN1C(c1ccoc1)=O 29644,N1(C(C(C)OC)=O)CCCN(C(=O)C(C)(C)C2CCC2)CC1C 29645,C1(NC(CC=C)=O)(CC)CCN(C(c2cccc(C(C)(F)F)n2)=O)CC1 29646,c1(C(=O)NCC=CCNC(C2C(CC)CCC2)=O)ccc2c(c1F)CCC2 29647,C1(N(C(COC(C2C(c3n(CC)ccn3)OCC2)=O)=O)C)CC2CCC1O2 29648,c1(NC(c2ccn(C)n2)C)ccc(C(=O)N(C)C)cc1F 29649,C1(C(=O)NC2(CN(C)C(c3nccn3C)=O)CC2)C2CCC1(c1ccccc1)C2 29650,Cc1ccc2c(c1)C(NCCCC(N)=O)C(C)C2 29651,C1(NC(COCCCCCCCC)=O)CCN(C(=O)C(C2CC2)OC)CC1(C)C 29652,N1(C(C2C(CCC)CN(C(=O)C(C)CC(N)=O)C2)=O)CC2(C1)CC(C)(C)C2 29653,N1(C(C(C)CN(C)C(C2CCCOCC2)=O)=O)CCc2sccc2C1 29654,N1(C(c2c(C)n(C)nc2)=O)CC2C3CCC(C2C1)N(C(=O)CS(=O)(=O)C(C)C)C3 29655,N1(C(C(C(C)(C)C)SC)=O)CCC2(CC1)CCN(C(C13CC(C1)C(C)O3)=O)C2 29656,c1(C(=O)OC)cccc(C(N)=O)c1.n12nnnc1C(C(OC)OC)NCC2 29657,C(C(CC(F)(F)F)NC(C1(CO)CCOCC1)=O)NC(C1(COC)CC1(F)F)=O 29658,c1(N(C2CCCCC2S(C)(=O)=O)C)ccc2c(n1)CCCC2=O 29659,Cc1sc(O)nc1C(=O)NC(C)C(C)NC(=O)C(C)(C)CN1CCOCC1 29660,N1(C(c2c(C)cc[nH]2)=O)CCC(NC(c2ccc(C(=O)N(C)C)cc2)=O)C1(C)C 29661,CC(CC(C)(C)C)C(=O)NC1CC(O)CN(C(c2cscc2C2CC2)=O)C1 29662,N1(C(c2c(C(C)=O)ccs2)=O)CCC(C(C)NC(C2(C)CCCCC2)=O)CC1 29663,C(C)(C)(CC(=O)N1CCCCC1CNC(=O)C(c1ccc(C)s1)C)SC 29664,O(NC(=O)C(C)SC)CC.c12coc(c1)CN(C(C)C)C2=O 29665,CC1CC1N=c1nc2c(ncn2C)c(NC(c2ccc(F)cc2)CN2CCCC2)[nH]1 29666,c1(C(N2C(CNC(CC(C)(F)F)=O)CCC2)=O)ncnc2sccc12 29667,Cc1ccc(O)cc1C(=O)NCC1CC1NC(c1cn(C(F)F)cn1)=O 29668,C1(C(=O)NC2CCCC(CNC(C3CCCN(CC)C3)=O)C2)CN2CCN1CC2 29669,Cc1cccc(OCCCC(=O)NCCCCCNC(c2cc(C)[nH]n2)=O)c1 29670,C(CC(N)=O)(C(=O)N1C(CO)CC1CO)NC(CC1(CSC)CC1)=O 29671,c1(C(=O)NCC(C)N(C(=O)COCc2cccc(O)c2)C)cccnc1C1CC1 29672,n1(CC)nnc(C(=O)NCCCCC(=O)NCC2(F)CCN(C)C2)c1C 29673,C12(C(=O)NCC3N(C(C=CC(CC)=CC)=O)CC3)CCOC1CCOC2 29674,c1(CC)cc(C(=O)NCC2CCCN(C(=O)C(=O)N(C)C)C2)oc1CC 29675,c1(C(=O)NC(C(C)NC(C2CCCN(C3CC3)C2)=O)CO)cnc2[nH]ncc2c1 29676,c1(CCC(=O)NCC2(NC(=O)CC3CCCCO3)CCC2)cccc(F)c1 29677,C1(CNC(=O)CCC2CC2(Cl)Cl)CC2(CCC2)CN1c1nc2ccccc2o1 29678,Cc1cncc(CCC(c2ccn(C(F)F)n2)=O)n1.c12oc(cc1C)CNC2=O 29679,CC1CCc2nnc(C(N3CCN(C(C)C(=O)N(C)C)CC3)=O)n2C1 29680,C1(NC(c2n(C)ncc2)=O)CC2CCC1(NC(c1cc(C(N)=O)co1)=O)C2 29681,N1(C(c2ccc(CC)o2)=O)CC2CCC(CC(=O)NCC3CC[Si](C)(C)C3)(C2)C1 29682,C1(NC(c2cn(CC)nc2C)=O)CC12CCN(C(=O)Cc1nc(=N)[nH][nH]1)C2 29683,S(=O)(=O)(c1cc(Cl)ccc1Cl)NCC1(F)CCCN(C(C(CC)O)=O)C1 29684,c1(OC)ccc(CC(C)C(=O)NC(C)CCNC(=O)Cc2sccc2C)cc1F 29685,C1(NC(C2CN(CC)C(=O)C2)=O)CC2CCC(C1C)N2C(c1cc(C)c(C)o1)=O 29686,C1(C(N(C2CCC(NC(C3CCC(CC)O3)=O)C2)C)=O)C2CCC3C(C2)CC13 29687,C(C)(C)(CC(F)C(=O)N(CCCF)C)NC(CCC(N(C)C)N(C)C)=O 29688,C(CC1=CCN(C(C2(C)CCCO2)=O)CC1)NC(C(C(C)C)n1cc(C)nc1)=O 29689,c1(C(=O)NCC2CC(O)CN2C(=O)CCOCC(F)(F)F)cncc(Cl)c1Cl 29690,N1(C(c2ccc(S(C)(=N)=O)cc2)=O)CC2C3CCC(C2C1)N(Cc1cccs1)C3 29691,c1(OCCC)cccc(CC(=O)NC(C)C(C(C)C)NC(c2cncnc2)=O)c1 29692,N1(C(=O)NC2C(C(=O)OC)CCCN2)CCCC(C(=O)O)C1C 29693,C(=O)(C1CCCn2nccc21)N1CCC(CCc2cn(C(C)CO)nn2)CC1 29694,Cc1cc2c(COC(c3ccnc(SCC(F)(F)F)c3)=O)csc2s1 29695,N1(C(c2ccc(OC)o2)=O)CCC(O)(CN(C)C(c2cnc(S)nc2)=O)C1 29696,n1(CC(=O)NC2CC(C(N(C(CF)CF)C)=O)C2)cnc(C#N)n1 29697,c1(CC(=O)NCCN(C(c2cc(C)c(CO)cn2)=O)C)ccc2c(n1)OCCO2 29698,C(CC(Cc1ccccc1)NC(C1(Br)CC1)=O)NC(c1cnns1)=O 29699,c1(C(=O)NCC(C2CCCC2)NC(C2CC=C(C)CC2)=O)cccc2nc[nH]c12 29700,C1(NC(CNS(CCCOC)(=O)=O)=O)CN(C(c2ccc(C)s2)=O)CC2(CC2)C1 29701,C1(C(=O)NCC(C)(C)CO)CC2CC1CN(C(=O)CC1CCC(C)(C)O1)C2 29702,C(=O)(C(CCC(C)C)NC(c1cnn(C)c1Cl)=O)N(CC#C)Cc1ccco1 29703,c1(C(=O)NCCC(C)N(C(CC)=O)C)cccc2c(I)n[nH]c12 29704,C(c1ccc2c(c1)OCCO2)=CC(N1CCCC(N(C(C(CC)CC)=O)C)C1)=O 29705,C#CCCCCCC(=O)N1CC2(CC(C(=O)NC3CC(=O)N(C)C3=O)CO2)C1 29706,c1(C(=O)OC)cc(C(=O)NCC2CCCC2NC(=O)CN2CCOCC2)ccn1 29707,Cc1nnc2cnc(C(=O)N(C3CC(NC(c4ccc(Cl)[nH]4)=O)C3)C)cn12 29708,c1(NC(C2C(NC(c3cccc(-c4ccccc4)c3)=O)C2)=O)ccc(I)c(Br)c1 29709,C1(C(N(C(CN(C(Cn2nnc(C)n2)=O)C)C)C)=O)CCC(C)CC1 29710,c1(C(C)C)conc1C(=O)NC(C)CC(=O)NC1COCC1CN(C)C 29711,C(=O)(C(CC1CCC1)NC(c1cc(F)c[nH]1)=O)N(C)CCOCC1CC1 29712,n1(CC(=O)NCCN(C(c2ncncc2C#N)=O)CC)cc(C)ccc1=O 29713,C1(NC(=O)OC(C)(C)C)CN(C(=O)OC2CC3CCCC3C2)C2CCCC12 29714,C(=O)(CCCCC(N)=O)N1C(C)CC(CCNC(=O)COCP(C)(C)=O)CC1 29715,c1(CNC(C(C)C#N)=O)cccc(CNC(=O)CC(C2CC2)C2CC2)c1 29716,C1(C2CC2)(NC(CN2CC(CCN(C)C)OCC2)=O)CCCCCC1 29717,CC1(C)CN(Cc2ccc(C(=O)NO)cc2)CC1c1cc[nH]n1 29718,Clc1ccccc1Cn1nnnc1N1CCN(CCSc2ccccc2)CC1 29719,C(=O)(CCN=c1[nH]c(=NCC2(C)CC2)[nH]c2ccsc12)NC(c1ccco1)C 29720,C1(NC(c2nc(C)oc2C)=O)CCN(C(=O)C(F)C(C)C)CC1CO 29721,C1(CNC(c2cc(O)ccc2I)=O)CCN(Cc2c(F)cncc2F)CC1(F)F 29722,c1(C(N(CC(C)C)CC(=O)NCC2CC(=C3CCC3)C2)=O)ncccc1N 29723,N1(C(C(COC)NC(CCOC)=O)=O)CC2CC=CCC2C1 29724,CC(CC(=O)NCC1CC12CC2(F)F)C(C)(C)NC(=O)C=C1CCOCC1 29725,C(=O)(C(C)(C)C(F)(F)F)NCC(CNC(c1cc(-c2c(C)n(C)nc2)no1)=O)C 29726,CCC(CNC(=O)CC(CC1CC1)NC(=O)CC1C(=O)NN=C1C)(CC)OC 29727,Cc1nn(C)c(C(=O)NCC2CN(C(=O)COC(F)F)CCCO2)c1Cl 29728,S(=O)(=O)(c1ccc(Br)cc1NCc1cn2ccsc2n1)NCC1ON=C(CC)C1 29729,C=CC1OCCC1C(N1CCN(CC2(NC(=O)Cn3ccnc3C)CC2)CC1)=O 29730,c1(C(=O)OCC)ccc(C(c2nnnn2CCc2nncs2)NCCSC)o1 29731,C1(CCN2C(CNC(c3ccc(C)n3C)=O)CCC2)COc2ccccc2O1 29732,c1(C(=O)NCC2N(C(C3=C(C)OCC3)=O)CCOC2)ccc([N+](=O)[O-])c(F)c1 29733,C1(NC)CCN(C(=O)C=O)C(C)C1.n1(CC)nc(NCC2CC2)cc1C1CC1 29734,C=CCC(C(=O)NC1CCCN(C(c2snnc2CC)=O)C1)OC 29735,C(=O)(C(C)(C)C(F)F)N(C)CC1CN(C(C(C)SC)=O)C1 29736,CCC(C)(CNC(=O)C(C1CCCCC1)C)NC(c1occc1C1CC1)=O 29737,c1(CNC(C2CC(NC(COCCOC)=O)C2(C)C)=O)ccc(O)c(C)c1 29738,c1(C(C)=O)ccc(C(N2CCCC(C)C2)=O)cc1F.C1(=O)C(=O)N(CC)CCN1 29739,c1(C(=O)NC2(CC=C)CN(C(C3CC3COC)=O)C2)ccc(S(=O)(=O)CC)cc1 29740,C1(COC)CN(C(c2cc(F)c[nH]2)=O)CCN1C(=O)CCCc1ccc(O)cc1 29741,N1(C(C2CC(SC)C2)=O)CC2CC(NC(=O)CC3(O)CCCC3)CC(C2)C1 29742,c1(C2CCN(CC3CCN(Cc4c(Cl)c[nH]n4)CC3)C2)cccc2c1OCO2 29743,c1(OC)ccc(C(=O)O)cc1CN1CC(C)(C(N2CCCC(C)C2)=O)C1 29744,c12sc(C)cc1NC2=O.N1(CCN(C(CNC(=O)OCC)=O)C)CCC(C)C1 29745,Cc1cc2ccc(C(N3CCC(NC(c4[nH]c(O)nc4C)=O)CC3C)=O)cn2c1 29746,N1(C(C2N=C(C)SC2)=O)CCOCC(CNC(=O)Cc2cccc(N)c2)C1 29747,C1(C(N2CC=CC(C(=O)NCCC3CC(F)(F)C3)C2)=O)C2CCC(F)(F)C12 29748,C(=O)(C(C)CC(F)(F)F)NCCN(CC(C)O)C(c1ccn(C(C)C)n1)=O 29749,c1(C(=O)NC(C(C)NC(c2c(C)cc(F)cn2)=O)CO)cnc2c(c1)COCC2 29750,C1(C(=O)NCCOCCCNC(=O)Cn2cccc2)CC(=O)N(c2cn[nH]c2)C1 29751,c1(C(=O)NCC2(C(N)=O)CN(C(C3(OC)CCC(C)C3)=O)C2)ncc(C)cc1C 29752,c1(NC(=O)Nc2cc(C)c(Br)cn2)cc(C(F)(F)F)cc(S(C)(=O)=O)c1 29753,C1(C)(C(=O)NCC(C)(CO)NC(CC2CC(=C)C2)=O)CC(=O)N(C)C1 29754,c1(C(N(CCCNC(C(CC)C)=O)Cc2ccccc2)=O)nc(C)ccc1F 29755,c1(C(N(C)CCn2cc(CN3CCSCC3)nn2)=O)snc(Cl)c1Cl 29756,CCCCC(O)C(C)C(=O)NCCCC(=O)N(CC(C)OC)C 29757,N1(C(c2c[nH]nc2Br)=O)CC2C(CNC(C34COCC3C4)=O)C2C1 29758,C1(C)(CC)NC(=O)N(CC(=O)NC(C)C(C)NC(c2c(Cl)n[nH]c2CC)=O)C1=O 29759,C(=O)(C(C(C)C1CCC1)N1CCC2CC12C)NC(C(=O)OC)Cc1ccccc1 29760,CC(C)C(F)(CNC(C1CCCCCN1C)=O)C(=O)NCC1CCC1(F)F 29761,C#Cc1ccccc1CC(=O)NCC(C1CC1)N(C(=O)C(O)C(C)C)C 29762,Cc1cc(C)n2nc(C(N3CCC3CNC(=O)C3=CCCCO3)=O)cc2n1 29763,C1(CNC(c2scc(C)c2C)=O)CN(C(c2ccc(C(F)F)o2)=O)CCC1C 29764,N1(C(=O)NC(c2cnn(C)c2)C(C)C)CCOC(C)(C(F)F)C1 29765,c1(-n2c(CC(C=C)C)nc(C3CCCCC3)n2)ccnc2ccccc12 29766,C1(NC(CCC(=O)NCCC)=O)CC2CC1CN2C(c1cnc(CC)s1)=O 29767,CC(O)C(C(=O)NCC1(CO)CC1)NC(C1CC(F)(F)C1)=O 29768,c1(-c2nc(COC)nn2-c2cccc(OC(F)(F)F)c2)cnn2ccc(O)nc12 29769,N1(C(CC)=O)CCCC2(CCN(C(C3CCn4nccc4C3)=O)C2)C1 29770,C=CC1(CC(N2CCC(NC(c3cscc3C)=O)C(CC)C2)=O)CCOCC1 29771,C1(NC(C2C(OC)CCC2)=O)CN(C(c2cnsc2C)=O)CCC1C(F)(F)F 29772,CCCC(C(=O)OC)C(=O)N(C)CCNC(c1csc(-c2ccccc2C)n1)=O 29773,CC1CCN(C(c2n[nH]cc2Br)=O)CC1NC(C1(F)CC2(CCC2)C1)=O 29774,c1(C(=O)NCCCC2N(C(C(CCCC)O)=O)CCC2)c(C)nc2sc(C)cn12 29775,C(CCC(C)C(=O)NCCOCCCNC(C12CCCC1OCC2)=O)OC 29776,c1(C(=O)NC2C(CC)N(C(=O)CCc3cncs3)CC2)cc(C2CC2)ccc1F 29777,C1(CNC(CC(C)n2ccnc2)=O)C(C)CCCN1C(=O)CC1(O)CCCOC1 29778,c1(NC(C2CSCCN2C(c2ccc(Br)s2)=O)=O)cccc(O)c1F 29779,c1(-c2cn(CC3N(C(CCN(C)CC)=O)CCC3)nn2)ccc(C#N)nc1 29780,N1(C(C2(CC)CC2)=O)CCCC2CN(C(=O)C(=O)Nc3ccc(C)cc3)CC12 29781,C(C(CC1CC1)C(=O)NCCCCOC(=N)O)NC(C(C1CCCC1)OC)=O 29782,n1(CC(C)CO)nc(-c2ccc(Cl)nc2)nc1C1CCC(=O)N1C(C)(C)C 29783,N1(C(C(CC(C)C)OC)C(=O)NC2CC2)CC2OCCCC2(CO)C1 29784,c1(C(=O)NC2CN(C(c3c(C#C)cn(C)n3)=O)C2)ccc2c(O)nc(C)nc2c1 29785,CCC(C#N)(CC)C(=O)NCC(O)CN(C)C(C1(OC)CCC1)=O 29786,C(=O)(CCCCCCNC(C1CCOC1(C)C)=O)NCC(C(C)O)C 29787,c1(C(=O)NCC(CC)NC(C2(O)CCCCC2)=O)cn(C)nc1C(C)(F)F 29788,N1(C(C2CCN(C(C3(C)CC4CC4C3)=O)C2)=O)CCC2C(C(N)=O)C2C1 29789,C1(COC)(CNC(c2csc(C)c2N)=O)CCN(C(=O)C(C)c2ccsc2)CC1 29790,N1(C(C(C2(C)CC2)NC(C(COC)C)=O)=O)CC2(CC(C)CO2)C1 29791,C1(OC)CC2CCC1CC2C(N1CCC(N(C)C(c2ccc(C)c(C)c2)=O)C1)=O 29792,c1(C(=O)NC2C(NC(C3(C=C)CC3)=O)CCCC2)cc(C)nc(O)c1 29793,N1(C(C2COCCO2)=O)CC2C(NC(C3(C(F)(F)F)CC(F)(F)C3)=O)C2C1 29794,C(N=c1cc(CO)nc[nH]1)C1(NC(C(C(C)C)N2CCCCC2)=O)CCOCC1 29795,c1(CNC(C(=O)N(C)CCc2ccc(C#N)cc2)=O)sccc1S(C)(=O)=O 29796,c1(OC)ccnc(C(=O)NCC2CCCCN(C(c3csnc3C)=O)C2)c1F 29797,c1(C(=O)NCC(C)CN(C)C(c2cc3nc[nH]c3cn2)=O)cncc2sccc12 29798,c1(OC)ccc2c(c1)CCC(CNC(=O)C(=O)Nc1c(C)nc3sc(C)cn13)C2 29799,C1(C(N(CCCC=C)C)=O)(NC(=O)COC)CCCC1C 29800,CN1CCN(C(=O)CCC2NC(=O)NC2=O)C(CNC(=O)C(C2CC2)C2CC2)C1 29801,c1(N2CC(=C(CNC(C3C=CCCC3)=O)F)C2)ncc2cccnc2n1 29802,N(C(=NCCN1CCCC1)N1CCCC2(CC2)C1)Cc1oc(CC)c(C2CC2)n1 29803,C1(NC(C(n2ncc(C)c2)C)=O)CC(CNC(=O)C=Cc2cnc[nH]2)CC1O 29804,C(=O)(CC(C(=C)C)OCC)NCc1cc(C(=O)NC2(CC#C)CCCCC2)sc1 29805,c1(C(=O)O)ccc(CN(c2cnsc2)Cc2cccc(-c3cnco3)c2)cn1 29806,C1(C)(C(N2C(CNC(C(c3cccc(C)c3)C)=O)CCC2)=O)C(C)(C)C1(C)C 29807,C1(NC(C=C(C)C(C)C)=O)C2CC1N(C(=O)CC(c1ccccc1)NC(N)=O)C2 29808,C(N=c1[nH]c(N(C)CC2CCCO2)nc(=N)[nH]1)c1c(C)ccnc1 29809,CCCC(C#N)C(=O)NCC1(F)CC(NC(=O)Cc2cncn2C)C1 29810,C(=O)(CC(C(F)(F)F)NC(=O)C(F)C(C)(F)F)NC(C)C(=O)NCCF 29811,N1(C(c2ccc(C)s2)=O)C(C(N2CC(OCC(C)C)C2)=O)CCC1C(C)C 29812,c1(NC2CCN(C(CC)=O)C2)ncnc(N2CCCC(F)(CO)C2)c1C 29813,N1(C(CC2N(C)CCC2)=O)CCC(C2CCCN(C(c3ccc(Cl)o3)=O)C2)CC1 29814,N1(C(c2cc(C(C)C)ncc2)=O)CC2CCC(C1)N2C(=O)Cc1cnn(C)c1 29815,C1(C(N2CCC(NC(c3cnn(C)c3Cl)=O)C2)=O)Cc2ccccc2CO1 29816,c1(CN2CCC(C(=O)OC)C2C)cc2ccccc2[nH]1.c12ccc(o1)NC2 29817,CCC(C)C(C(=O)NCCc1cc(C)on1)NC(=O)CC(C)n1cccc1 29818,CC(C)CCCC(C)C(=O)NC1C2CC3C(C2)C13C(=O)N(C(CO)C1CC1)C 29819,c1(C(N(C2CCN(C(C(=CC3CCCC3)C)=O)C2)C)=O)nc(Cl)c(Cl)s1 29820,C1(C(=O)NC(C)Cc2nccn2C)COc2ccc(Cl)cc2C1 29821,CCCCC(=O)C(=O)NC(CO)C(N1CC(CO)CC1CO)=O 29822,C1(NC(=O)C=CCn2cncn2)CCC(NC(C23CCOCC2C3)=O)CC1 29823,N1(C(CCSCC)=O)CC(NC(c2cc(C)n(CC(F)F)c2C)=O)CC1(C)CC 29824,C(=O)(CS(=O)(=O)C(C)(C)C)N1C2(CNC(CC(CC)C)=O)CC(C1)C2 29825,CCCC(CC)C(=O)N1CCC(CNC(c2csc(CC)n2)=O)C12CC2 29826,C(=O)(CCC(F)(F)C(=O)N1CCCCC1CNC(C1(C)CNC(=O)C1)=O)OCC 29827,N1(CCNC(C=CC2(C)COC2)=O)CCC(NC(C2CC=CCC2)=O)CC1 29828,Cc1nc(C(C)(C)C)sc1C(=O)NCC1(NC(C2CCCC2)=O)CCCC1 29829,C(=O)(CC(O)CC(C)(C)C)N1CCC(N(C(c2cncc(C)c2)=O)CC2CC2)C1 29830,c1(C(N2C(C)CC(NC(=O)C3=COCCO3)C2)=O)cccc2c3c([nH]c12)CCC3 29831,C(CO)(CCF)NC(C(C)N(C(=O)C=C1CCC1)C1CC1)=O 29832,Cc1cccc2c1c(CNc1cc(F)cc3cc[nH]c13)cn2C 29833,c1(C2CC(CC(=O)NCC(C)CN(C)C(C3(C)CCCO3)=O)C2)ccccc1 29834,Cc1oc(C#N)cc1C(=O)NCC1(C)CCN(C(C2CCCC(C)CC2)=O)CC1 29835,CCC(CC(=O)N1CCCC1(C)C(=O)NCC1(C)CCOCC1)C(C)(C)C 29836,CC1(C)OCCC1CC(=O)NC1CCCC1NC(c1ncccc1O)=O 29837,N1(C(c2c(C)n(C)cc2)=O)CCCCC(NC(c2ccc(CO)s2)=O)C1 29838,Cc1ccc(O)nc1CNC(C1CCCN(CC2CCCCC2)C1)=O 29839,N12CCC3(CC1)COC(C3)C2.C(CC(F)(F)F)C1(C(=O)OC(C)(C)C)CCC1 29840,N1(C(CC(=O)OCC)=O)CCC(NC(=O)Cn2nnc(C)n2)CC(C)(C)C1 29841,N1(C(c2c(C)nn(C(C)(C)C)c2)=O)CC2CCC1C2NC(=O)COC(C)C 29842,C1(C(=O)NC2CN(C(c3c(C)onc3)=O)CC2(C)C)Cc2ccccc2S1 29843,C(C1=NOC2CCCC12)NC(C(=O)N(C(COc1ccc(C)cc1)C)C)=O 29844,C=C(C)C1CCC(C)=CC1CC(N1CCCCC1C=Cc1cccs1)=O 29845,c12cc(ncn1)N2.N12CCC(C1)CN2C.c1(CNCCO)ncccn1.CC 29846,CCCC(CC)C(=O)NCC1CCC1NC(=O)COCC1CCCC1 29847,C12(C(=O)NCC(CC)(C)OC)CC(CN1C(=O)CCOCC(C)(C)C)C2 29848,C(=O)(CC(C)P(C)(C)=O)NCCCN(C(CSCC(=O)OC)=O)C(C)C 29849,C(=O)(C1=CCCN(C(C2CCC=CCC2)=O)C1)NCc1n(C)nnn1 29850,CCC(C)(CCNC(=O)C=Cc1c[nH]cn1)NC(=O)CCCc1ncco1 29851,N1(C(C(c2ccc(C)cc2)C)=O)CC2=C(C1)CN(C(c1c[nH]cc1C)=O)C2 29852,C12(C(=O)NC3(C(=O)OCC)CC3)CCC(CN(C(=O)C3=NOCC3)C1)C2 29853,CCCC(C)(CCC)C(=O)NCC1COCCN1C(=O)CCCCN(C)C 29854,C(N=c1nc(O)c(Br)c[nH]1)C1CCC(NC(c2ccc3nncn3c2)=O)C1 29855,c1(C(N2C(CNC(C3CC(=O)N3)=O)CC(C)(C)C2)=O)cnc(O)c2ncccc12 29856,Cc1nc2ccnn2c(C)c1C(N1CCN(C(c2cnc(O)n2C)=O)C(C)C1)=O 29857,Cn1cnc(C(O)CNC(=O)CC2(NC(C3CC(F)(F)C3)=O)CC2)c1 29858,Cc1ccc(C(=O)NC2(CNC(=O)Cn3nnc(=N)[nH]3)CC2)cc1C(C)(C)C 29859,N1(C(CCC2N(C)CCC2)=O)CCN(CCN(C(=O)CCCCC2CC2)C)CC1 29860,C1(CNC(CNC(c2c(C)occ2)=O)=O)CN(C(=O)CCCCF)CCC1C 29861,c1(C(=O)NC23CC2CN(C(C2CC4(C2)CC(O)C4)=O)C3)cn2cc[nH]c(=O)c2n1 29862,C1(c2cccc(NC(c3n(C)cc(Br)n3)c3nnnn3C)c2)CCC(F)(F)CC1 29863,C1(NC(CCCc2n(C)cnn2)=O)(CNC(=O)CSCCC#N)CCOCC1 29864,c1(C(=O)NCC=CCNC(C2CC3CCC2CC3)=O)ccc2cc[nH]c2c1 29865,CC1OC2(C(=O)NCCC(C)(C)NC(c3cnn(C)c3Br)=O)CCC1C2 29866,N1(C(C#CC2COC2)=O)CCN(C(C2Cc3ccccc3O2)=O)CCC1C.CCS 29867,C1(C(=O)NCC2C(NC(C(C3CCCC3)OC)=O)C2)C2CCC3C(C2)CC13 29868,Cc1c(Br)c(C(N2CCC(C)(CNC(C3CC(C)CCO3)=O)C2)=O)nn1C 29869,C1(CNC(C2CC(O)(CC#C)C2)=O)CCN(C(=O)C(C)=CC)CC1 29870,C(=O)(C1=CCOCC1)N1CC(C2CN(C(CCC3(C)CC3)=O)C2)OCC1 29871,C1(CC(=O)NC(C(C)C)CNC(=O)CCN2CCCC2=O)CCCS(=O)(=O)C1 29872,c1(C(=O)NCCCCNC(CSCCOC)=O)cc(C)ccc1C1CC1 29873,c1(CC)cccnc1C(=O)NC(C)CN(C(=O)C(=Cc1ccccc1)C)CC 29874,Cc1ccc(C(N2CCCCC2CC(=O)Nc2ccnc(F)c2F)=O)c(I)c1 29875,N1(C(Cc2cccc(CC)c2)=O)CCC(NC(C2CC(=O)N(C)C2)=O)C(O)C1 29876,C(=O)(CC(C)(C)C#N)N1CCCC(C(C)NC(CCC(=C)C)=O)C1 29877,C1(CNC(C=Cc2c(C)nn(C)c2Cl)=O)CCC2(CC1)OCCO2 29878,n1(CC)nccc1C(=O)NC(C1CCCN1C(c1cc(CCO)on1)=O)C 29879,C12(C(=O)NCc3c(C)nccc3)COCC1CN(C(=O)C1CC1)C2 29880,C12(C(=O)NCCc3cncc(C)n3)CC(CN(C(C3(C(N)=O)CCC3)=O)C1)C2 29881,CCCCCC(C)(C)C(=O)NCCC1(C)CCN(C(=O)CC2CCCO2)CC1 29882,C(=O)(C1OCCn2ccnc21)N1CCC(CNC(c2n(C(C)C)ccn2)=O)CC1 29883,c1(OC)ccc(C2CCN(C(=O)NC(C)C(C)(C3CC3)OC)CC2)cc1 29884,N1(C(c2nn(CC)nc2C)=O)CCC(NC(c2cc(Cl)sc2Cl)=O)C(CO)C1 29885,N(C(=NCCCC(=O)NC(C)C)N1CCCc2ccccc2CC1)CCOC 29886,CC1(C)CCN(C(c2nnsc2C(F)F)=O)CC1NC(c1ccc(C(N)=O)o1)=O 29887,C1(CNC(C2CCN2Cc2ccccc2)=O)CC(O)CN1C(C1CCC(O)C1)=O 29888,c1(OC)c(C(=O)NC(C2CCCN2C(=O)CC2(OC)CCCC2)C)ccnc1F 29889,C1(C)(C(=O)NCC(CNC(CCOc2c(C)cccc2)=O)C)CCS(=O)(=O)CC1 29890,c1(C(=O)NC(CC(C)C)CNC(=O)C(F)=CCCF)cc(Cl)ccc1C(C)C 29891,C(CCC)(C(=O)NC1CCN(C2CCN(C(=O)Cc3ccsn3)C2)CC1)=CCC 29892,Cc1cc(C(N2CCC(CF)(NC(=O)CC(C)CF)C2)=O)cc([N+](=O)[O-])c1 29893,C1(C2CC2)(CNC(c2ccn(C)n2)=O)CCN(C(C2(C(N)=O)CCC2)=O)C1 29894,C1(C2CCC2)(C(=O)NCC(c2ccccc2F)NC(=O)CC2CCCO2)CC1 29895,C1(NC(=O)Cn2cc(C3CCC3)nn2)CN(C(C2CCC2)=O)C2(CCCC2)C1 29896,N1(C(c2cnc(C(N)=O)s2)=O)CC2(CC(NC(C3COCCC3(F)F)=O)C2)C1 29897,C#CC1CCCN(C(=O)C(C)(C)NC(C2CC3(CCC3)C2)=O)CC1 29898,C1(CCC(N2CC(CC=C)(NC(C3CNC(=O)N3)=O)C2)=O)CC(C)(C)CO1 29899,c1(C(=O)NCCC(C)NC(=O)C=Cc2ccc(F)cc2)cc2c(Cl)cccc2[nH]1 29900,N1(C(COC(CC)C)=O)Cc2[nH]nc(C(=O)NCc3cc(C)sc3C)c2C1 29901,c1(CC(=O)N(C2CCN(C(=O)C3=COCC3)C2)CC)cc(C)ccc1F 29902,Cc1cc(CC(=O)N(CC(=O)N(CCC(C)C)CCO)CC(C)C)c[nH]1 29903,CC1CC(C(N2CC(F)(CNC(=O)C(C)Cc3ccccc3)C2)=O)(CO)C1 29904,C(=O)(C(CC=C)CC(C)C)NC(C(=O)NCC(=O)OCC#C)CCF 29905,c1(CCC)[nH]nc(C(=O)NCC2CN(C(C3CCN(C(C)=O)C3)=O)C2)c1[N+](=O)[O-] 29906,CC1CCCN(C(=O)CC2CCCC2C)C1CNC(c1cnc(C#N)s1)=O 29907,N1(C(c2c(CC)con2)=O)CCCC(N(C(c2cscc2F)=O)CC)C1 29908,C1(N(C)C(C2C3COCC23)=O)CCCN(C(=O)CSc2ncccn2)CC1 29909,c1(C(C2CC2)C2CC2)ccc(C)o1.C1(C(COC)NC(=O)N)CCCOC1 29910,C1(C(=O)NC2C(NC(C3(CCCC)CCC3)=O)CC2)CCSCC1 29911,N1(C(C(c2cccnc2)C)=O)CCC(N(C(=O)C=CCF)C)CC1 29912,c1(C(N2C(C(C)NC(=O)CCc3cncnc3)CCC2)=O)c[nH]c2ncccc12 29913,Cc1cc(=NC2CCC(=O)N(C)C2)[nH]c(N2CCC(F)(CO)C2)n1 29914,C1(C(=O)NC(CCNC(CC(CC)OC)=O)(C)C)CC12CCS(=O)(=O)CC2 29915,C1(C(=O)OCC)C=CC(NC(c2nnnn2C2CC2)c2ccon2)C1 29916,CC1CSCC1NC(=O)CC1(NC(C2CCN2C2CCCC2)=O)CC1 29917,N1(C(C2C(C)N(C(=O)Cc3ccc(O)cn3)CC2)=O)CCOC(C#N)C1 29918,C(CCCC(=O)N1CCCC1(C)CNC(C1C(C(F)F)C1(C)C)=O)OCC 29919,C1(NC(c2ccc(CO)cc2)=O)CCC(NC(=O)C(F)Cc2ccccc2)CC1 29920,C1(c2n(CCOCC)nnn2)(NCCC2CCC2)CC2CCCCCC2C1 29921,c1(C(N2CC3C(CNC(CC)=O)C3C2)=O)oc2ccccc2c1CS(C)(=O)=O 29922,C1(CC(=O)NCCC2CN(C(Cc3nc(CC)sc3)=O)C2)CCCCN1C 29923,c1(C(C)=O)cc(C(=O)NCCCN(C(=O)C(c2ccccc2C)C)C)c(C)o1 29924,C12(C(N(CCNC(C(CN(C)C)O)=O)C3CC3)=O)C3CCC(CC13)C2(F)F 29925,CC1CCC(CNC(c2cnc(N(C)C)cn2)=O)CN1C(=O)C=CC1CC1 29926,C1(NC(CC2CN(C)C(=O)C2)=O)CCCCN(C(=O)C=CC=C(Cl)Cl)C1 29927,C(CC(C)(C)C)(C(=O)N1CC(CNC(=O)C=Cc2cccs2)C2(CC2)C1)OC 29928,C12(CCOCC1)C(=O)NC(C)C(=O)NCCO2.C(CCOC1CCC1)SC 29929,Cc1ocnc1CC(=O)N(C)CC1(CNC(C2CC(=O)C2C)=O)CC1 29930,c1(C(N(CC(C)NC(=O)C=C(C)C)CC)=O)ccc(OC)cn1 29931,C#Cc1cccc(C(N2CCC(CN(C)C(C3CC(=O)NC3(C)C)=O)C2)=O)c1F 29932,Cc1noc2nc(C(N3CC(n4cc(C5CCCO5)nn4)C3)=O)ccc12 29933,N1(C(c2nc(Br)nn2C)C(=O)NCC=C)CCCC(O)(C(F)F)C1 29934,c1(CN2CCC(CC(N3CCC(N4CCCC4)C3)=O)CC2)cccc2nonc12 29935,CCCC(CC(C)C)C(=O)NC1CC(NC(=O)CCCC(F)(F)F)CC1O 29936,C(=O)(CCCC(=O)NC(c1cc(C(=O)OC)on1)=O)N1CCC(CNC)C1 29937,N1(C(C(CC=C)C)=O)CCC2C(C1)CN2C(C12CC(c3ccccc3)(C1)C2)=O 29938,CCCCCC(C)CC(=O)N1CC(C(C)NC(=O)C2=NNC(=O)C2)C1 29939,Cc1noc(N)c1C(=O)NCc1cn(CC(N2CC3CC3(CN(C)C)C2)=O)nn1 29940,C(CNC(=O)C(O)CN(C)C)(CC(=O)Nc1ccccc1Cl)OC 29941,C(=O)(C(CC)C(=O)NC(C)Cn1cccn1)OCC 29942,CC1CN(C(=O)CC2COC(=O)N2)CC1CNC(=O)C(=O)Nc1ncc[nH]1 29943,Cc1cc2ccc(C(=O)NCC3(O)CCN(C(=O)Cc4ccoc4)CC3)cc2o1 29944,N1(C(c2c(C)snn2)=O)CCC(C(C)CNC(C2(P(C)(C)=O)CC2)=O)CC1 29945,N1(C(c2c(C)cns2)=O)CCC2CCN(C(c3cc4n(n3)CC(F)C4)=O)CC12 29946,c1(C(N(C)CCOCCNC(c2cccc(Cl)c2Cl)=O)=O)cccc2ncnn12 29947,c1(NC(=O)NCC2(OC)CCS(=O)(=O)C2)nccn2cccc12 29948,C1(NC(CCC(C)(C)C#N)=O)CC(NC(c2occc2F)=O)C12CCOCC2 29949,C1(NC(CC2CCC(NC(CCC(=O)N(C)C)=O)CC2)=O)CCN2CCC1C2 29950,C1(C2CC2)(CNC(COCCCC)=O)CCN(C(c2cnn3c2OCCC3)=O)C1 29951,C=C(C(=O)Nc1ccc(CCC(=O)NCC=C(C)C)cc1)C(C)(C)C 29952,CC1(C)CNC(=O)CN1c1ccn(-c2cccc(CN)c2)n1 29953,Cc1ccc(-n2nc(C3CCCO3)nc2CN2CCOC2=O)cc1Cl 29954,O(S(=O)(=O)CCC(C(C)C)NC(=O)OC(C)(C)C)c1cc(OCC)cc(F)c1F 29955,c1(C(=O)NC(C)CN=[N+]=[N-])nccc2ccn(C)c12 29956,C(=O)(C(C(C)C)c1ccncc1)N(CCCNC(C(c1ccncc1)OC)=O)C 29957,C(CCNC(c1ccc(CC(C)C)s1)=O)(C(C)C)NC(C1(CC#C)CCCO1)=O 29958,c1(OC)cc(CC(N2CC(O)(C(C)NC(c3cnc(CC(C)C)s3)=O)C2)=O)on1 29959,N1(C(c2c(C)snc2)=O)CCC(F)(CNC(c2nnn(C3CC3)c2C(F)F)=O)C1 29960,c1(C(C(=O)NCCCN(C(CCC(=C)Br)=O)CCO)O)ccc(C#N)cc1 29961,C1(C(N(CCCNC(CS(=O)(=O)NCC)=O)CCO)=O)CCCC2(CCOC2)O1 29962,c1(C(=O)NC)ccc(OCC(N2CC(CO)(NC(C3CCCN3C)=O)C2)=O)cc1 29963,C(=O)(CC1=CCN(C(c2cccnc2O)=O)CC1)N(CC(C1CC1)OC)C 29964,C(=O)(C1c2c[nH]nc2CN1C(=O)C(Cl)Cl)N1C(C)COCCC1 29965,C1(C#N)(C(=O)OCC)CCN(C(=O)CC2CCOC2=O)C1 29966,CCC(CC(C)C)C(=O)NC1CCC(NC(=O)Cc2ccc(C#N)cc2F)CC1 29967,C(=O)(CC(O)CNC(C1CC1C(F)(F)F)=O)N(CC(CC)CC)C1CC1 29968,c1(OC)ccc(F)cc1C(=O)C(=O)NCC1CC(OC(C)(C)C)C1 29969,c1(C(=O)NC(C)C(C)C(=O)O)ccc2nc(O)nc(O)c2c1 29970,C(=O)(C(F)CC1CC1)N(C(C)CN(C(=O)CCOC1CC1)C)C 29971,Cc1cnc(C(=O)NC2CCCCC2CNc2nccc(CC#N)n2)cn1 29972,C1(C)(CNC(C2C(C(=O)OCC)C2)=O)CN(C(c2ccc(F)c(F)c2)=O)CC1C 29973,C(CC1=CCN(C(=O)CO)CC1)NC(C1CCCN1Cc1cn[nH]c1)=O 29974,N1(C(Cc2c(C)non2)=O)CCCC(CC(=O)NCC2CCN(C(C)C)C2)C1 29975,Cc1c(C(=O)NC(C(=O)N(CCO)CC2CCCC2)C(C)O)[nH]ccc1=O 29976,CC1CCCN(C(c2cnc(C(F)F)s2)=O)C1CCNC(=O)CCNC(N)=O 29977,c1(CC)ccc(F)c(C(=O)NCC(O)CNC(c2c[nH]c(=N)o2)=O)c1 29978,C1(C(C)NC(c2[nH]nnc2C2CC2)=O)C=CC(NC(=O)CC2CCCC2)C1 29979,c1(NCCC2CCN(C(C3(COC)COC3)=O)C2)ncnc2scc(C)c12 29980,C(C(CNC(C1SCCS1)=O)S(C)(=O)=O)NC(CCNC(=O)NC)=O 29981,CC1CCCCC1OCC(=O)NCC(=O)NCCCNC(=O)Cc1csc(Cl)c1 29982,N1(C(C(C)=C(CC)C)=O)CCCN(C(C2CC3CCC(C2)C3O)=O)C(C)C1 29983,CCCC(C)(CC)C(=O)N(CCCCC(=O)NC1(C(=O)OC)CC1C)C 29984,c1(C(=O)Nc2ccc(OC(C)C)cc2Cl)cccc2oc(O)nc12 29985,c1(CN(C2CNC(=O)C23CC3)C=O)c(F)c(F)c(Cl)c(F)c1F 29986,c1(C(COC(=O)CCc2ccc(I)cc2)=O)ccc(F)c(Br)c1 29987,c1(C(=O)NCC2CN(C(CCNC(=O)NC)=O)C(C)C2)cccc2c1CC(=O)N2 29988,C12(NC(c3[nH]cc(CC(C)C)c3)=O)CCCC1N(c1nnc(C)s1)CCC2 29989,C1(NC(CN(C2CCC2)C)=O)(CO)CCN(C(=O)C(CCSC)NC(C)(C)C)C1 29990,N1(C(Cc2c(F)ccc(OC)c2)=O)CC2CCCC2(NC(=O)CC(O)C(C)C)C1 29991,n1(-c2cccc(NCCOc3cc(C)c(Cl)cc3)c2)c(=O)oc2ccccc12 29992,c1(C(N2CC(n3ncc(NC(c4cccnc4O)=O)c3)C2)=O)ccc(Br)c(F)c1 29993,c1(C(=O)NC2(CCCNC(C3(CO)CCCC3)=O)CC2)ccc(F)cc1N 29994,OCCC(N=c1[nH]c(=NCCc2cccc(Br)c2)c2ccccc2[nH]1)C1CCC1 29995,C#Cc1ccc(C(=O)NCC2(COC)CCCN2C(C2CC2CC)=O)c(C)c1 29996,C(=O)(C(O)CC(C)C)N(CCOC)CCNC(=O)CCCc1cnn[nH]1 29997,Cc1nc(C(c2nnnn2C2CC2)NCC(C2CC2)OC)sc1C 29998,c1(OC)ccc(Cl)c(C(N2CC(NC(c3cc(O)ncn3)=O)CC(O)C2)=O)n1 29999,N1(C(C(CNC(C(C)SCC)=O)CC(C)C)=O)CCc2c(C#N)cccc21 30000,C(=O)(CCCCC(=O)NCc1ccc(C(=O)NCC(C2CC2)OC)s1)OC 30001,N1(C(c2c(OC)nn(C)c2)=O)CCC2(NC(=O)CCc3cnn[nH]3)CC2C1 30002,n1(C(C)C)cc(CC(=O)NCC(O)CN(C)C(C2(C)CCCO2)=O)cn1 30003,c1(C(=O)NCC(C)NC(N)=O)cn(-c2nc(C3CC3)ns2)cn1.C1(=O)C(C)N1 30004,C1(O)(CCNC(C(=O)NCC)=O)CCN(C(=O)CCOCCN(C)C)C1 30005,C(=O)(CCCCC(N)=O)N1CCCC(CCC(=O)N(CC(C)(C)OC)C)C1 30006,c1(CC(=O)NC2(CNC(c3ccc(O)c(Cl)n3)=O)CC2)cnc2cccnn12 30007,c1(NCCOCC)[nH]c(=NCc2ccc3c(c2)nc(CO)n3C)nc2scnc12 30008,Cn1cnc2c(N3CC(CNC(c4cn(CC5CCOC5)nn4)=O)C3)ncnc12 30009,C(CCCC(C)(C)C(=O)NNC(=O)CCCCC(C)C)OCCC(C(=C)C)OC 30010,N1(C(C2CCN(C(CC3CCCC(C)O3)=O)C2)=O)CC(C)CCC12CC2 30011,N1(C=O)CC(OCc2cccnc2)CC1C(=O)NN1CCCC1=O.CC(C)(C)O 30012,c1(C(=O)NCC(C(C)C)NC(=O)C(C)(C)c2ccccc2)nn(C)cc1Cl 30013,c1(C(N(C2CN(C(C(CC)OC)=O)CC2O)C)=O)cc(F)cnc1O 30014,c1(C(C)(C)C)cncc(C(=O)NCC(=O)NCCCOCC(F)F)c1 30015,N1(C(C2(C)CCN(Cc3c[nH]ccc3=N)C2)=O)CCc2ccc(C#N)cc2C1 30016,C(C(C(=O)NCC1CCCO1)N(C)Cc1cocn1)(C1CCCC1)OC 30017,C(c1ccc2[nH]ccc2c1)=CC(=O)NC(C(C)NC(C1CCCS1)=O)CO 30018,Cc1cc(C(N2CCCC(C)(NC(C3CC(CF)C3)=O)C2)=O)cc(N)c1Cl 30019,C1(NC(C2C(NC(c3c(CC)n[nH]c3)=O)COCC2)=O)CC(C)(C)C12CCC2 30020,c1(C(=O)NC2(C)CC(NC(c3cn(CC=C)nc3)=O)C2)ncccc1Br 30021,c1(C(=O)NCC2(F)CCC(CNC(C3C(C)C3)=O)C2)n[nH]c2c1CS(=O)(=O)CC2 30022,CCC(C(C)(C)O)NC(C1(NC(C2CC3(CC3)C2)=O)CC1C)=O 30023,N1(C(C2C(CCC)C2)=O)CCC(C(=O)NC2C=CCCC2CO)CC1(C)C 30024,c1(C(C(=O)NCC(C)N(C(=O)C(O)P(C)(C)=O)C)=O)cc(Cl)cc(Cl)c1 30025,c1(N(C)CC)cccc(S(=O)(=O)N(CC(C)(C)S(C)(=O)=O)CC)n1 30026,CC(C)CCC(O)C(=O)NC1CCC(CC(=O)NCC(O)CNC(N)=O)CC1 30027,C(=O)(CCC(C)(C)OC)NCC(CNC(C(CC)OC)=O)(C)C 30028,c1(CC)cc(C(N2CCC3(NC(c4coc(CO)c4)=O)CC3C2)=O)cn(C)c1=O 30029,C(CCCCNC(c1ncsc1C)=O)N(C(C1(CC#C)CC1)=O)C 30030,C(CCCC(=O)NC(COC)CC(=O)NC(C)Cc1nc[nH]n1)OCC 30031,c1(C(=O)NCCN(C2CCCC2)C(c2c(COC)cc[nH]2)=O)ccn(C)c(=O)c1 30032,CCCCC(O)C(=O)N1CC(NC(=O)CCc2ccc(F)cc2)C2(CC2)C1 30033,CC1C(C(=O)NCCN(C)C(=O)OC(C)(C)C)CCN1C(c1cc(CF)on1)=O 30034,C1(F)(CNC(C2C(C(=O)OC)CC2)=O)CCC(NC(=O)CN2CCCC2=O)C1 30035,C1(C(N(CCOCC=C)C)=O)CC(NC(=O)CCCNC(N)=O)CCO1 30036,N1(C(CCNc2ccc(C)cc2)=O)CC(CNC(c2cc(C)on2)=O)CCC1C 30037,C(c1cc(F)c(F)c(F)c1)=CC(N1CCN(C(CC(C)SC)=O)CC1CF)=O 30038,c1(OCCOCC)ncccc1C(=O)NC(C)CNC(=O)C(CC)n1ccnc1 30039,O=C1CN(S(=O)(=O)c2ccc(C(F)F)cn2)CC2(CO)COCCN12 30040,Cn1ccc(C(=O)NC2CCC(NC(=O)CS(=O)(=O)NCC3CC3)C2)c1C1CC1 30041,C1(C(N2CC(NC(c3nc(CCC)sc3)=O)C(OC)C2)=O)CC2(CCCCO2)C1 30042,c1(C(=O)NCC2(CCCNC(C3CCO3)=O)CCCC2)[nH]nc2ncccc12 30043,c1(-n2cc(C3CN(C(C4CCS(=O)CC4)=O)C3)nn2)cc(F)ccc1Br 30044,N1(C(C(CCC)N(C)C)=O)CCN(C(C2(C)CCC2)=O)CC1C 30045,C1(CNC2(CC(N)=O)CCC2)CC1(Br)Br 30046,CC(O)(CNC(c1cc(CCNC(=O)C(F)=CC2CC2)on1)=O)CO 30047,CCN=c1[nH]cc(CN2CCN(C(=O)CC(C(C)C)c3ccon3)CC2)s1 30048,C(=O)(C1=CCCC1)NCC(CO)NC(c1cc(CC)on1)=O 30049,c1(C(N2CCN(C(c3sccc3Cl)=O)C(C(F)F)C2)=O)cc2cnccc2o1 30050,C1(C(C(=O)NC2CCCC2)N(C)Cc2ccc(C)o2)CC=CCC1C 30051,c1(C(=O)NC2C(NC(c3nc(COC)sc3)=O)CCC2)cnc2sc(C)c(C)n12 30052,c1(C(=O)NCCOCCOCCNC(C2C(=C)CC2)=O)cc(C)c(F)c(C)c1 30053,C1(CC)CCOC1C(=O)N(CCCCN(C)C(c1sccc1CN(C)C)=O)C 30054,CC(C)(C)CCC(=O)NC12CCC(NC(C3CCC(C)(C)CC3)=O)(CC1)C2 30055,N1(C(C(CCNC(=O)CCc2nc[nH]n2)OC)=O)CCC2(CCOC2)CC1 30056,N1(C(c2ccsc2Br)C(=O)NC(C)(C)C)CC(C)CC2CCCCC12 30057,Cc1ccc(C(N2CCC(CCC(=O)NC(C3CCCC3)CO)C2)=O)cc1 30058,n1(CCCC)nc(C)c(C(N2CCC(CC(N3CCCCC3CO)=O)C2)=O)c1C 30059,N(C(=NCCS(=O)(=O)N1CCCC1)NCC1(CO)COC1)C(COC)C 30060,c1(C(=O)OC)c(C)n(COCC)c(CCNC(c2ccccc2)COCC)c1C 30061,C1(C(=O)NCCN(C(=O)CC2C=CCC2)C)(OC(C)=O)CC(C)C1 30062,C(CNC(=O)Cn1cnccc1=O)(C(C)(C)C)NC(CN(S(C)(=O)=O)C)=O 30063,c1(C(N2CCCCC(NC(c3ccc(CO)o3)=O)C2)=O)cc2cc(O)ccc2[nH]1 30064,C1(CC(=O)N(C)CCOCCCNC(=O)CC2COC(=O)C2)OCCC1(C)C 30065,N1(C(CCCc2n(C)cnn2)=O)CC2CC1CCC2NC(=O)Cc1ccnn1C 30066,Cc1ccc2nc(C)c(C)c(C(=O)NS(=O)(=O)CC3CNCCO3)c2c1 30067,N1(CC=C)CCc2nc(C(=O)NCC3(CCOCC)CCCC3)cn2CC1 30068,CC(=O)n1cc(-c2ccc(C(=O)Nc3ccc(O)c(C)c3)nn2)cn1 30069,CN1CC(C)(C)CC1C(N1CCC(C(=O)NCCCN2CCCC2)C1)=O 30070,CCC(N=c1[nH]c2c(c(=NC(C)c3ncc(C)s3)[nH]1)CSC2)C1CCCC1 30071,Cn1cc(C(=O)COc2cccc3[nH]cc(NC(=O)C4CC4)c23)c2ccccc12 30072,CCC(CC)C(F)C(=O)N1CC(F)CC1CC(=O)NCc1ccc(F)c(C)c1 30073,n1(CC(=O)NCC(CNC(Cc2c(C)nsc2)=O)CO)ccc(=O)cc1C 30074,CCC(CC)CCC(=O)NCCC1(O)CCN(C(=O)CCNC(=O)C=CCl)CC1 30075,c1(C(c2nnnn2C(C)(C)C)Nc2c(CC)nc(C)cc2)ccc2c(c1)CCC2 30076,c1(OC)ccc(S(=O)(=O)N2CCC23CN(Cc2c(Cl)cccc2I)C3)cn1 30077,CCCCC(O)C(C)C(=O)NC1(C)CCCC1NC(=O)C=CC1CCC1 30078,C(=O)(C=C1SCC(=O)N1C)N1CCC(C)(CNC(c2c(N)cc(C)c(C)c2)=O)C1 30079,c1(C(N2CC(CC=C)(NC(C(C)OCC#C)=O)C2)=O)c(C)nc(O)nc1S 30080,C123CCCC1N(CC2)C3=O.C1(CNC(c2sccc2F)=O)CCC=CCC1 30081,Cc1ccc(C(=O)NC(C(=O)NOC2CC3CCC2C3)c2cccnc2)nc1C 30082,N#Cc1ccc(C(c2nnnn2CC(F)F)NCCC(O)c2cccs2)cn1 30083,C1(OC)CC2CC1CN(C(C1CC(O)CN1C(c1sncc1C)=O)=O)C2 30084,c1(CC)ccnc(C(C(=O)NCC2CC2)N(C)CC2(C#N)CCC2)c1 30085,c1(C(C(N2CC(CN(C)C(C3CCCOC3)=O)C2)=O)O)ccc(Cl)cc1 30086,CP(C)(=O)C(O)C(=O)NC1CCC(NC(=O)CN2CCC(O)CC2)CC1 30087,c1(N(C(COCCC=C)=O)CCCNC(C2CCC2F)=O)ccccc1 30088,CC(CC(=O)N1CCN(C(c2cnn(CC3CC3)c2)=O)C(CF)C1)C(C)(C)C 30089,N1(C(COCC(=C)C)=O)C2CCC(C2)C1CC(=O)NCCCCCOC 30090,C1(CC#C)(C(=O)NCC2C=CCN2C(=O)CC2CC(=O)C2)CCCC1 30091,C1(NC(=O)CC2CCOC2)C2CC1N(C(=O)C=CCO)C2 30092,Cc1cc(C(=O)N(C(C)CNC(c2ncn(C(C)C)n2)=O)C)c(Br)s1 30093,C1(NC(C(CCC)C)=O)CN(C(=O)C2=CCC(C)(C)CC2)CC2(CCC2)C1 30094,N1(CCNC(C(Cc2ccco2)NC(CC2(SC)CC2)=O)=O)C(=O)CCC1=O 30095,C(=O)(CC(O)CN(c1nc(Cl)cs1)C)NCCCNC(=O)NC 30096,N=c1nc[nH]c(=NCCOC2CCN(C(=O)C=C3CCC3)CC2)[nH]1 30097,N1(C(c2cnc(C(C)C)nc2)=O)CC(O)C(O)C1CNC(=O)C(F)C1CCC1 30098,n1(CC(=O)NCCN(C)C(C2CCSC2)=O)cc(C2CC2)cn1.C1CC1 30099,c1(C(=O)NCC(C)(C2CCC2)NC(CSC(C)(C)C)=O)ccnc2ccncc12 30100,c1(CC)ccc(F)cc1C(N1CC2CC1CN2C(C1(C(C)(C)O)CCC1)=O)=O 30101,c1(C(=O)NCC(n2cc(-c3c(COC)nns3)nn2)C)cc2n(n1)CCCO2 30102,O=S(=O)(c1sccc1I)N1CCCC(Oc2cccc(F)c2)C1 30103,Cc1nc(=N)[nH]cc1CNC(=O)NC1CCN(CC2CC2)CC1 30104,C(CC(CNC(=O)C(CO)N(CC(C)(C)C)C)NC(=O)CO)OC 30105,N1(C(=O)NCC2(CO)COC2)CCC(c2nncs2)C1 30106,c1(C(=O)NCC(CO)NC(=O)CSc2ccncc2)cc(Br)c(Cl)s1 30107,C(=O)(CCCCCn1cc(CNC(N2CCC(C)(C#N)C2)=O)nn1)OCC 30108,CCC(C)C(=O)C(=O)N1CC(C)C(C)(C(N2CC(C)C(C)C2C)=O)C1 30109,N1(C(COCCC=C)=O)CCC2(CCN(C(C3(S(C)(=O)=O)COC(=O)C3)=O)C2)C1 30110,C12(CNC(C(c3ccc(F)cc3)C)=O)CC1CN(c1ccnc(N(C)C)n1)C2 30111,c1(C(N2C(C)CC(CNC(c3ccc(F)nc3)=O)C2)=O)ccc(F)c(N)c1 30112,c1(C(=O)NC2C(NC(c3nc(CCC)oc3)=O)CCOC2)cn2cccnc2n1 30113,N1(C(CNC(C(CC)CC)=O)=O)CCN(C(=O)C(F)=CC2CC2)C(C2CC2)C1 30114,C=CC(C)(CC)NC(c1cc(CNC(c2cocn2)=O)[nH]n1)=O 30115,N1(C(C)CNC(c2cc(C(N)=O)c[nH]2)=O)CCN(C(=O)CN2CCOC2=O)CC1 30116,CC(C(C)C(=O)NCCOCC(C)(C)O)NC(C1SCCS1)=O 30117,CC1CN(C(c2cn(C)cn2)=O)CC(C)C1Nc1ncnc(Cl)c1F 30118,Cc1nncc(C(N2CCC(C)(C)C2C(=O)N(C2CCCC2C)C)=O)c1C 30119,N(C(=NCCOC)NCC(C)Oc1ccccc1Cl)Cc1nc(CC)oc1 30120,c1(C(N2CCN(C(c3scc(C#N)c3)=O)C3C2C3)=O)ccc2ccccc2c1 30121,Cc1nc(C(C)(C)CNC(=O)NC(c2ccoc2)C)n[nH]1 30122,C(=O)(CCCS(N)(=O)=O)NCCCN(C(C(C)NC(COC)=O)=O)CCO 30123,C1(NC(C=CC(C)(C)SC)=O)CN(C(c2cn(C)c(=O)cn2)=O)CC2(CC2)C1 30124,c1(C(=O)NCC2(O)CCN(C(CCCCC)=O)C2)cc(OC)c(O)c(N)c1 30125,C(C)(CCC(=O)NCC1OCCC1C(=O)N(C)C1CC1)OCC 30126,c1(CN(C)C(c2cccc(CNC(=O)CCC3CC3(F)F)n2)=O)ccc(O)cc1 30127,C1(N(C(C(N2C(=O)CCC2=O)C)=O)C)CCCN(C(=O)Cn2cnnc2O)CC1 30128,Cc1ccncc1C=CC(=O)NC1(CO)CCCN(C(=O)CCc2cc[nH]n2)C1 30129,Cc1cnc(C(N2CC(CCNC(=O)C(c3ccc(F)c(F)c3)O)C2)=O)cc1Cl 30130,CC1CC(=O)NC(C(=O)NC2CN(C(=O)CSCC(N)=O)C(C)(C)C2)C1 30131,CCCC(O)(CCC)CC(=O)NC1CC2CC(C1)N(C(c1c[nH]c(=O)cn1)=O)C2 30132,C1(NC(C2CCCCC2(F)F)=O)CC2CC(NC(=O)CC3=CCOCC3)CC2C1 30133,N1(Cc2ncc(C(C)(C)C)o2)CCC2(CN(C(c3coc(Br)c3)=O)C2)C1 30134,N1(C(c2cc(C)ncc2)=O)CCC2CCN(C(=O)COCC(F)F)CC12 30135,n1(C(CC)C)ccc(=NC(=O)C2(NC(=O)C(C#N)C(C)C)CC(CO)C2)[nH]1 30136,Cc1cnn(CCC(=O)NCCOC2CN(C(C3CCCN3C)=O)C2)c1 30137,C(=O)(C(CC(C)C)NC(C)=O)NCC(CC)NC(C1CCN1Cc1cccs1)=O 30138,c1(CCC)onc(C)c1C(=O)NCCCN(C(=O)C=CC(CC)=CC)C 30139,c1(C(=O)NCC2C(NC(CN(C)C(N)=O)=O)COC2)cc(C(F)(F)F)nn1C 30140,C(=O)(C(C)(C)C#N)NCC(C)(C)CC1CN(C(c2ccsn2)=O)C1 30141,C(C(O)C(=O)N(CC(C)C(=O)NCC1CSCCO1)C)SC 30142,C(C(=O)NC(CO)C(C)NC(C1(CCF)CCC1)=O)(C(C)C)SCC 30143,N1(C(C(OCC)OCC)=O)CCC(CNC(C2CCC2(C)C)=O)(OC)CC1 30144,N1(C(C(N2CC(CC(=O)OCC)CC2(C)C)=O)=O)CC23CCCCC2(CNC3)C1 30145,N#CC1CCCC(C(N2CCN(Cn3cc(CCC4CCCO4)nn3)CC2)=O)C1 30146,c1(C(N(CC(CNC(Cc2cc(C)nn2C)=O)(C)C)C)=O)cc2n(c1)CCOC2 30147,C=C1CCN(C(=O)CC=CCC)C(C(N2CCC(CF)CC2)=O)C1 30148,c1(C(C)OCC)noc(SCC(=O)NC(C2CCOC2)CC)n1 30149,C1(CC(=O)NCC2(NC(C(C(C)C)C)=O)CCCC2)COC(C)(C)CO1 30150,c1(C(=O)NCCC2(O)CCN(C(=O)C3=CCSC3)CC2)cc2c(nn1)CCC2 30151,C12(CCOC1)C(=O)N2.C1(NC(C)=O)CCCC1CNC(=O)CNC(=O)C(C)(C)C 30152,C(=O)(C(C)S(=O)(=O)C(C)C)N1CCC(CCNC(C(COC)(F)F)=O)CC1 30153,CCC(C)C(=O)C(=O)N(C)CC1(O)CCCN(C(c2sccc2CO)=O)C1 30154,c1(C(=O)NC2CCCC(CNC(C3(N(C)C)CCCC3)=O)C2)cc(F)cc(F)c1 30155,N1(C(c2cnc(C(C)C)s2)=O)CCCC(CCNC(=O)CC2CCN(C)C2)CC1 30156,C1(C(N2C(CC(=O)N(CCC#C)CCOC)CCCC2)=O)CCOCC1(C)C 30157,N1(C(C=Cc2c(C)nccc2)=O)CC(C2CCCCN(C(=O)CSC(F)F)C2)C1 30158,C(C1=NOC2OCCC12)OC(C1CCC=CC1O)=O 30159,C1(C(=O)NC(CC#C)CCOC)CCN(C(=O)c2csc(C)c2)O1 30160,N1(C(C(C)OC)C)CCC(O)(C(=O)N(CCCN(C)C)C)CC1 30161,N1(C(C(C)SC)=O)CCCCC(CNC(c2cnoc2C)=O)C1 30162,C1(OCC)CCCC1NC(=O)C(c1ccnn1C)C 30163,CCCC(CC(=O)N1CCC1COC)c1ccccc1.n12nnnc1C2C1CC1 30164,C(=O)(CCC(=O)N1CCOC(CC(N2CCC23CCC3)=O)C1)NCC 30165,c1(C(=O)NCCCN2CCN(C(C3(O)CC3)=O)CC2)cc([N+](=O)[O-])ccc1Br 30166,N1(C(=O)C2=C(Cl)CC2)CCCN(C(c2cc[nH]c3nccc2-3)=O)C(CO)C1 30167,C1(C(N2C3CN(C(c4ccc(C)nc4)=O)C(C3)CC2)=O)CCc2ncccc2C1 30168,Cc1ccc2c(CC(=O)NC3CC(NC(C4(CO)CCCCC4)=O)C3)coc2c1 30169,N1(C(c2cccnc2S)=O)CCC2(CCCN2C(c2ccc[n+]([O-])c2)=O)C1 30170,c1(CN(C(c2ccc(C(=O)OC)n2C)C(=O)NC2CC2)C)c(C)nn(SC)c1C 30171,C1(C(=O)Nc2cnc[nH]2)CN(Cc2ccc(Br)cc2)CCC1O 30172,N1(C(C2C(NC(CCCN=[N+]=[N-])=O)C=CCC2)=O)CCC12CCCCC2 30173,c1(C(N2C(CO)CC(NC(C=C(C)C)=O)C2)=O)cc2c(Br)coc2cn1 30174,N1(C(c2c(CC)nn[nH]2)=O)CCC2(CCCN2C(=O)CCCC2OCCO2)C1 30175,c1(C(N2CCC(O)(CNC(C(n3c(C)ncc3)C)=O)C2)=O)nnn2c1CCCC2 30176,Cc1cccc(N2CCC(N(C)Cc3ccn(-c4ccccc4)n3)C2=O)c1 30177,C(=O)(CCCCCN(C)C)N(CC(CC)NC(=O)CSc1n[nH]c(C)n1)C 30178,C1(NC(c2c(C(=O)OC)[nH]cc2)=O)CCC(NC(=O)COCC(F)(F)F)CC1 30179,Cc1cc(C(N2CC3CCC2C(NC(C2CCC2)=O)C3)=O)c(N)c(F)c1 30180,C(CC(=O)NC1CC(CCO)C1)(C(F)F)NC(Cc1c(C)ccs1)=O 30181,CC(C)CC(C)C(=O)N(CC(O)CNC(=O)CCOc1ccc(C(C)C)cc1)C 30182,c1(C(N2CC(NC(C34CCN(CC3)CC4)=O)C2)=O)ccc([N+](=O)[O-])[nH]1 30183,c1(C(=O)NC2C(CNC(CN(CCC#C)C)=O)C2)ncccc1OC 30184,C(CC1=CCN(C(c2ccc(C)c(C(=O)OC)c2)=O)CC1)NC(CCC=CC)=O 30185,N1(CC(N2CC(NC(C3CCS(=O)CC3)=O)CC(C)C2)=O)CCc2ccccc21 30186,N1(C(c2c(C)coc2)=O)CC(NC(c2[nH]nnc2-c2ccnn2C)=O)CC1C 30187,C#CCCCC(=O)NC(Cc1ccoc1)C(N1CC2C=CC2C1)=O 30188,C1(NC(CCC=C=C)=O)CC=C(C(=O)N2CCC(OC(C)=O)C2)C1 30189,Cc1cccc(F)c1C(=O)NC1CCC(NC(C2CC23CC3)=O)CC1 30190,N1(C(C(C)(C)c2cccs2)=O)CCCC(O)(CNC(c2ccc(C(F)F)o2)=O)C1 30191,CCC(CC(=O)NOCC(=O)NC(c1nccs1)(C)C)C(C)(C)C 30192,N1(C(CCOCCOC)=O)CCC(C(=O)NC(CCO)C2CCC2)(CC)CC1 30193,n1(CC(N2C(C)CC(CNC(=O)CC3CS(=O)(=O)C3)C2)=O)nnc2c1CCCC2 30194,c1(C(=O)Nc2ccc(C#N)cc2)cnc2c(-c3ccc(CO)nc3)cccc2c1 30195,CCCCC(CC)C(=O)NCC(C)(F)CNC(c1ccn(CC)c1C)=O 30196,c1(C(N2CC(NC(c3ccccn3)=O)C3C2C3)=O)ccc2cnccc2n1 30197,C1(C)(NC(CCCN(C)C)=O)CCN(C(=O)C2=CCCC2)CC1 30198,N1(CC)CCCCC1C(=O)NCCC1(NC(c2cnn(CC(F)(F)F)c2)=O)CC1 30199,N1(C(=O)OC(C)(C)C)C2CCC1CC(CNC1CCC(O)CC1)C2 30200,C(=O)(C(Cc1ccco1)C(F)(F)F)NC1(CCNC(=O)CC2CCC2)CCC1 30201,c1(C(N2C(CC)C(NC(=O)CCC3CCOC3)CC2)=O)cnn2c(Cl)cccc12 30202,c1(-c2n(C)cnc2)ccc2oc(C(=O)Nc3cc(O)ccc3Br)cc2c1 30203,c1(C(=O)OCC)cnc(NC2CC(C)N(C(C3CC4(CCCO4)C3)=O)C2)nc1C 30204,C12(NC(CCSC)=O)CC(C1)N(C(=O)CSc1nccn1C)C2 30205,c1(C(=O)NCC(CC)NC(=O)C(CC)Nc2nc(C)cs2)cccc(=O)o1 30206,Cc1c(C(N2CCN(C(=O)CC3C=CCCC3)CC2CO)=O)nn(C)c1Br 30207,CC(F)(F)C(C)(C)CNC(C1(NC(=O)COCC2CCCO2)CSC1)=O 30208,N1(CC(=O)NCC(O)CNC(c2csnn2)=O)CCCC1CO 30209,Cc1cc(C(=O)NC2CC23CCN(C(=O)OC(C)(C)C)CC3)nc2nccn12 30210,CN1CCOC(C(=O)NCC2(F)CCC(NC(=O)CSCCC(F)(F)F)C2)C1=O 30211,c1(OC)ccc2c(C(N3CCC(N(c4c([N+](=O)[O-])cnn4C)C)C3)=O)cnn2c1 30212,C1(C(=O)OC)CCCC(C(N2CCCCC2CN(C)C(c2cocn2)=O)=O)C1 30213,N1(CC(N2CC(O)(CCNC(CCCOCC)=O)C2)=O)OC(C)(C)CC1=O 30214,C#CCCCCCC(=O)N1CCCOC(CNC(=O)CCSC2CCCC2)C1 30215,C1(NC(c2cc(O)nc(O)n2)=O)COC2(CCN(C(c3cccnc3Cl)=O)C2)C1 30216,CC1CN(C(=O)CC(C)(C)CCC2OCCO2)CCC(c2nc(C3CC3)no2)O1 30217,c1(NC2(CC(=O)NCC(N3CCCS3(=O)=O)(C)C)COC2)ncc(C#N)cc1Br 30218,c1(C(=O)NCCCNC(CC2(C)CCCO2)=O)ccc(-c2ccccc2)cc1F 30219,Cc1ccnc(CNc2c[nH]nc2C(=O)Nc2nccnc2C(F)(F)F)c1 30220,C1(C2(C(=O)NC(C3CCOCC3)C#C)CC2)CCCN1C(=O)CSC 30221,c1(CC)cc(NC2CCCN(C(C3CC3NC3CCC3)=O)C2C)c2c(c1)CCO2 30222,N1(C(CCNC(C(C=C)C)=O)=O)CC=CCC1C(=O)NC 30223,N1(C(c2cc(N3CCOCC3)ccn2)=O)Cc2cccc3c2C(CCC3)C1 30224,n1(C(CC)C)ncc(C(=O)NCC2C=CCN2C(c2cccs2)=O)c1C 30225,CCC(CN1CCCC1)NC(=O)C(=O)NCC(n1ccnn1)c1cnc[nH]1 30226,c1(C(C)C)cc(C(=O)NCCCOCCOCCNC(C2C(C)C2C)=O)on1 30227,C=CCC(C)(CO)CN=c1[nH]c(=NCC2CCCS2)[nH]c2c1COC2 30228,c1(NC(C2CN(C(c3ccnc(C(F)(F)F)c3)=O)CCO2)=O)cc(Br)ccc1I 30229,Cc1ccc(OCC(=O)NC(C)(CNC(c2cn(C)cn2)=O)C2CCC2)cc1C 30230,Cc1c(C(N2CC(NC(C34CC(C(C)C)(CO3)C4)=O)C2)=O)[nH]c2ccccc12 30231,c1(C(C(=O)NC(CSC)CC(C)C)C)c(Cl)cccc1Cl 30232,N1(C(CN2CC(C)(OC)C2)=O)CCN(C(=O)C2=CCCN(C)C2)CC2CCCCC12 30233,S(=O)(=O)(CCC(=O)NCC1CC(O)CN1C(c1cccc(=O)n1C)=O)N(C)C 30234,c1(C(=O)NC(CC)CNC(=O)CN2CCN(C)CC2)cnc2ccccn12 30235,N1(C(c2c(C)oc(C(C)C)n2)=O)C2CCC1CC(NC(=O)C(C)CC1CC1)C2 30236,C1(C(=O)OCC)CNC(=O)CC12CCN(C(c1cccc(=O)n1C)=O)CC2 30237,C=CC1OCCC1N=c1[nH]c(C(F)F)c(C(=O)OC)o1 30238,N1(C(C2CCC(CNC(CCC(C)(F)F)=O)C2)=O)CCn2ncc(O)c2C1 30239,C12(C(N(C(CNC(CC(C=C)C)=O)C)CC)=O)C3CC(CC13)C2(F)F 30240,C1(C(C)O)CCN(CCN(c2cc(Br)n(C)n2)C(=O)C2CC2)CC1 30241,N1(C(C(C)NS(CC)(=O)=O)=O)CCCC(C)(CNC(=O)Cc2ccns2)C1 30242,CCC(C)CCC(O)CC(=O)N1CCC(NC(c2csc(C)c2C2CC2)=O)CC1 30243,CC1CCN(C(=O)CCc2cnn(C)n2)CC1N(C)C(C1COC(C)(C)CO1)=O 30244,O(NC(=O)C(C)(C)C#C)CC(=O)NC(C#C)C(C)C 30245,Cc1cccnc1C(N1CCC(C)C1CNC(C12CC(C(C)C)(CO1)C2)=O)=O 30246,C1(CC(=O)NCC2(NC(=O)CSc3ccc(F)cc3)CCOC2)CCCC12CC2 30247,c1(CN2CC(CC(=O)NC3CCS(=O)(=O)C3)OCC2)cc(F)c(Cl)cc1O 30248,c1(C(=O)NCC2(CNC(CC=C=C)=O)CCC2)c(C)cc(C)nc1O 30249,c1(CC)nn(C)c(CC)c1C(=O)NCCC(C)N(c1cc(Cl)c(O)nn1)C 30250,c1(C(=O)NC(C(CC)C)C(N2CCC3(CC(CO)C3)C2)=O)ccn2nccc2c1 30251,c1(C(N(CC(CN(C(C(C)OCCCC)=O)C)O)C)=O)cc(O)cc(C#N)c1 30252,C1(CNC(C2(C)CCC(=O)C2)=O)CC(C(=O)NC2(CC(N)=O)CC2)=NO1 30253,N1(C(Cc2c(C)nc(Cl)cc2)=O)CC2CN(C(=O)Cc3ccc(F)cn3)CC2C1 30254,CCC(CC)C(C)C(=O)NCCC1(C(=O)NOCCCN(C)C)CC1 30255,C1(C(=O)NCC2CCN(C(C3(n4ccnn4)CC3)=O)C2)CCCCC(F)(F)C1 30256,CCC(C(=O)NCC1CC2(CC(NC(=O)C=CCOCCOC)C2)C1)C(C)C 30257,N1(C(C(C)CC(C)(C)C)=O)CCC(O)(C2(NC(C3CCC(F)(F)C3)=O)CC2)CC1 30258,C1(C2CC2)(C(=O)NCC2N(C(CCC3C(C)=NNC3=O)=O)CC2)CCOCC1 30259,c1(C(N)=O)ncn(CC(=O)NCC2CCC(NC(C3CC4CC4C3)=O)C2)n1 30260,N1(CCCC(=O)NCC(C)N(C(=O)CC=CC(C)(C)C)C)C(=O)NC(C)(C)C1=O 30261,c1(C(N2CCCN(C(C34CCC(OC)C3C4)=O)CC2)=O)ccc2c(c1)CCCS2 30262,C1(C)(N)CCN(C(C)=O)C1.C(CCC=O)OC.C1(C(C)C)CNC(=O)N1 30263,c1(OC)ccc2sc(CNC(C)C(=O)Nc3ccc(C)c(C)c3)c(C)c2c1 30264,Cc1cn(C)nc1C(=O)N(CCC(C)NC(C1CCCN1S(C)(=O)=O)=O)C 30265,c1(C(N(CCCN(C(C(CC)(C)O)=O)C)C)=O)nc2ccccc2nc1C1CC1 30266,CC1C(NC(=O)COC2CCOC2)CCN1C(=O)C=CC1CCC1 30267,N1(C(c2scc(C)c2)=O)CCC2(CC1)CC(C(N1CCCC(C)(F)CC1)=O)C2 30268,C=C(C)C(C)(C)C(=O)NC1CCC(N(C)C(c2ccccc2C(C)O)=O)CC1 30269,S(=O)(=O)(c1ccccc1F)NC(C1C(NC(c2cccc(F)n2)=O)C2CCC1C2)=O 30270,c1(C(N(CC(=O)NCCC(=C)C)C)=O)ccn(C)n1 30271,CC1CN(C(=O)COCCF)CCCN1C(=O)CC12CCC(CC1)OC2 30272,CC1OCCC1C(=O)NCC1CCOC1C(=O)NCCc1cnnn1C 30273,C1(NC(N(C)CC)=O)CCN(C(=O)Cn2ccnc2C(C)C)CC1 30274,C(C(C)(C)C(=O)N1CCCCC1CCO)NC(C=C(C)C(F)F)=O 30275,Cc1sc(=O)n(CC(=O)NC(C2CCCN2C(c2cc(Cl)ccn2)=O)C)c1C 30276,C(C)(CO)(C(=O)NCC(O)C(C)O)NC(CC(C)n1cccn1)=O 30277,C=C(Cl)CC(C(=O)N=c1cc(C)n(CCO)[nH]1)NC(=O)C1=CC2(CCOC2)C1 30278,C(=O)(C1=NOC2(CCOC2)C1)NCCOCCNC(C1(c2c(C)c[nH]n2)CC1)=O 30279,CC1C(=O)N(CC(=O)NCCCN(C)C(c2nc(=N)cc[nH]2)=O)C(=O)C1C 30280,C1(C(=O)NCCC2CCN(C(C(C)n3cncn3)=O)CC2)CC(F)(F)C12CCC2 30281,C(C(=O)N=c1ccn(CC(C)C)[nH]1)N(C1CN(C)CCO1)CCC 30282,N1(C(C(CC(C)C)OC)=O)CCC2(CCC(NC(c3cc(O)nc(C)n3)=O)C2)C1 30283,C1(C(=O)NC23CC(NC(C4(CN(C)C)CC4)=O)(C2)C3)CCC(N(C)C)CC1 30284,C1(CNC(C=CCC)=O)CC(CNC(=O)CCOC2CCC2)CO1 30285,C(=O)(C1CCC(=O)c2cccn21)NCCCCC(C)NC(c1cc(OC)ns1)=O 30286,C1(NC(c2cc(CC)ncn2)=O)CN(C(=O)C(=O)C(C)CC)CC(F)(F)C1 30287,C(=O)(C(CCF)NC(c1scnc1Cl)=O)NC1C(C(C)C)C1 30288,C(CCC(C)C)(C(=O)N1CCC(C)=C(C)C1)NC(C=CCCC)=O 30289,C1(CC(=O)NC2(CNC(=O)CC3CCCCC3)CCOC2)CCCS1(=O)=O 30290,C(=O)(C(F)C(C)CNC(=O)C=C1CCCCC1)N(C(C)C(=O)OC)CC 30291,c1(C(N2CCN(C3CN(C(C(=O)N(C)C)=O)C3)CC2)=O)n[nH]c2ccc(F)cc12 30292,N1(C(c2ncn(C)n2)=O)CCOC2CN(C(=O)CC3CCC(C)(C)O3)CC12 30293,c1(C(=O)NCCC2(C(=O)NC(c3ccncn3)C)CCC2)ncccc1N 30294,N1(CCC)CC(C(=O)N(CCCCCNC(=O)COCC(C)(C)C)C)CC1=O 30295,S(=O)(=O)(c1ccc(C#N)c(N2CCC3CC23)c1)N1CCCC(=C)C1 30296,c1(C(=O)NCC2(CNC(CC(C)OC)=O)CC23CCC3)ncc(C)cc1F 30297,C12COC3(CC1C3)C(=O)N2.c1(OC)ccc(C(=O)N(C2CCCC2)CCO)cc1 30298,c1(C(=O)NC(CCN(C(c2c(CC)nn[nH]2)=O)C)C)cccc(Cl)c1F 30299,c1(C(=O)NC2(C)CC(NC(Cn3c(C)nnn3)=O)C2)cccc2c1OCC2(C)C 30300,CC(C)CC(C(=O)NC1CC2CC(NC(=O)CSc3nnnn3C)C1C2)C(N)=O 30301,C(=O)(C(C(=O)C1CC1)OC(C)CC)OCC.C1(=O)CCNC(=O)NCCN1C 30302,C1(CC)CCC(C(=O)ON2CCC(O)(c3ccc(C)nc3)C2)CC1 30303,N1(C(C(CC(F)F)N(C(CNC(=O)NC)=O)C)=O)CC2(CNC(=O)N2C)C1 30304,c1(OC)ccc2nc(N3CCC(NC(=O)Cn4cc(C(C)O)nn4)C3)sc2c1 30305,N1(C(C(ON=C(C)C)C)=O)CC2(CCCN(S(=O)(=O)N3CCCCC3OC)C2)C1 30306,C1(COC)CN(C(=O)Cc2cncc(Br)c2)CCN1C(=O)CC(C)OC 30307,C(C(CC(C)C)C(=O)NC(C)(C)CNC(C1(C)CC1)=O)OC 30308,c1(N2CCC(CC)C2)ncc(C)cc1S(=O)(=O)N1CCC1(C)NC(=O)NC 30309,C(=O)(C1=CC(O)CCC1)N1C(CN(C(=O)CCCC2CCOCC2)C)COCC1 30310,Cc1ccc(C(=O)NCC(=O)N(C(C)CCNC(=O)CC(C)C)C)cc1C 30311,N1(C(c2c(C)nsc2C)=O)CC2(CO)CC1(C(=O)NCC1(C)CC1(C)C)C2 30312,N1(C(COCCCC(C)C)=O)CC2CCC2(CCNC(=O)C=C2CCCC2)C1 30313,C1(NC(C2(C#C)CC(=O)C2)=O)CS(=O)(=O)CC1NC(=O)Cc1csc(C)n1 30314,C1(C(=O)NCCC(N2CCCCC2)C)CC2CCC(N2)C1C(F)(F)F 30315,CC(C)CC(O)CC(=O)N1CCC=CC1C(=O)NCC1(C)CC1(F)F 30316,C1(CNC(c2ccc(Cl)cn2)=O)CC2COCC2N1C(=O)CCCN1CCCC1 30317,N1(C(C)C)C(=O)CCC1C(=O)NC(C)(CNC(c1c[nH]c(=N)o1)=O)C1CC1 30318,CC1c2ccc(Br)c(Cl)c2CCN1C(c1c(F)cccc1F)=O 30319,CC1=C(C(=O)NCC2C=CC(NC(=O)CC3CCC3)C2)C(C)n2nnnc2N1C 30320,C(=O)(CC(CC)C(C)(C)C)N(C1CCN(C(=O)CCc2nc(C)c(C)[nH]2)C1)CC 30321,C(=O)(C1=CCC(C)CC1)NCC(CC=C)NC(c1ncsc1S(N)(=O)=O)=O 30322,c1(C(N2C(CNC(c3c(CCC)cccc3)=O)CCC2)=O)ccc2cncn2c1 30323,C1(CNC(Cn2c(CCC)ncc2)=O)CC(F)CN1C(c1cnncc1OC)=O 30324,C(=O)(CC(F)(F)C(F)F)N1CC(NC(=O)C=Cc2ccsc2)C(F)C1 30325,c1(C(=O)NC2CC(CC(=O)N(CCO)CCO)C2)ccnc(C(F)(F)F)c1 30326,C#CCCCCCC(=O)N1CCC(NC(c2c(C)cccc2Cl)=O)CC1C1CC1 30327,c1(CC(=O)NCCC2CN(C(=O)N(C3CCC3)C3CC3)CCO2)cccc(I)c1 30328,N1CC(NCc2scc(OC)c2)CC1(C)C.C1(=O)CC(C)(C)O1.c1(CN)ccccc1 30329,c1(C(=O)NC2CC(N(C(=O)CC(C)(C)C3CCCCC3)C)C2)ccc2c(c1)CCC2 30330,N1(C(c2cc(C)c(C)s2)=O)CCCC(O)(CN(C)C(C2(C)CC(C)(C)C2)=O)C1 30331,c1(CC(=O)NCC(CC=C)NC(c2ncc(C)cc2C)=O)csc2ccccc12 30332,Cc1cccc2c1c(CN1CCC(C#N)(NC(=O)C(C)n3cccn3)C1)cn2C 30333,C1(C(=O)NCC2CN(C(=O)CC3CCCCO3)C2)(COC)CCCCO1 30334,C1(NC(=O)CC(O)c2ccccc2)CN(C(c2ccsc2Br)=O)CC12CC2 30335,N1(C(C2C(C)=NOC2=O)=O)CCCCC(CNC(=O)C(C)Cc2ccccc2)C1 30336,C1(CCCCNC(c2c(C)c[nH]n2)=O)CCN(C(c2c[nH]ccc2=O)=O)CC1 30337,C=C=CCCC(=O)NC1(CCNC(=O)CC2(OOc3ccccc3)CC2)CCC1 30338,CN1CCC2CN(C(C3CC(NC(C4(O)CCC4)=O)C3)=O)CC2C1 30339,N1(C(C2CCC(OC)CC2)=O)C2CC1CN(C(C1(C)CNC(=O)C1)=O)C2 30340,N1(C(C2C=CCN(C(C(C(=O)OCC)F)=O)C2)=O)CCC(C2=NOCC2)C1 30341,C1(NC(CCCOC)=O)CC=C(C(=O)NC2(C(C)O)CC2)C1 30342,C1(C(N(C(C)C(N2CCC(CN=[N+]=[N-])C2)=O)CC)=O)CCOC1(C)C 30343,n1(CC)cc(C(=O)N(C)CC2CN(C(C3CC3(C)C)=O)CCO2)c2ccccc12 30344,C1(NC(c2c(N)cncc2)=O)CC(NC(c2cc(C(F)F)cs2)=O)C12CCC2 30345,N1(C(CCC)C)CC(C(=O)NC(C)CNC(C2(C(F)F)CCCC2)=O)CC1=O 30346,CC1C(C=CC(N2CCCC2CCNC(=O)C(=C2CCCCC2)F)=O)C1(Cl)Cl 30347,Cc1cccc2cc(C(=O)NC3CCCC3NC(=O)C#CC3CCC3)oc12 30348,N1(C(c2ccc(OC)c(OC)n2)=O)C2CCC1CC(N(C)C(C1OCCO1)=O)C2 30349,c1(NC(c2cn(Cc3cccnc3)nn2)=O)cccc(O)c1 30350,c1(C(=O)NC(CC(C)NC(c2c(C)nncc2)=O)C)ncc(C#N)cc1Cl 30351,CC12COC(C(=O)NCCC3CSCCN3C(=O)CC3CCCCC3O)(C1)C2 30352,c1(NC(N2C(C(C)C)CC(O)C2)=O)cccc(C(F)F)c1Cl 30353,Cc1cc(C(=O)NC2CC(CNC(c3cccc(Cl)c3C)=O)C2(C)C)cc(O)n1 30354,Cc1cnc(F)cc1NC(=O)CN(C)C(=O)OC(C)(C)C.c12ccc(cc1)s2 30355,N1(C(C(C)c2cccs2)=O)CCC(C)(C(N2CCC(C(C)(C)O)C2)=O)C1 30356,C1(C(=O)NC(CC#C)C(=O)NCCc2nc(CC)no2)CC2(CCO1)CC2 30357,c1(N(C)C)ccccc1NC(C1C=CC(NCc2csc(Br)c2)C1)=O 30358,C(=O)(CCC(=O)NN(C)C)NC(C1C(C(=O)NCC(CCC)C)C1)C 30359,C1(NC(C(C)N2CCC2)=O)(CO)CCN(C(C23CC(C2)C(C(F)(F)F)O3)=O)CC1 30360,n1(C(C)C)nnnc1C(C1C=CCC1)NCCCN(S(C)(=O)=O)C 30361,C1(NC(c2c(CC)nc(C)n2C)=O)CCN(C(=O)Cc2cncn2C)CC1(C)C 30362,N1(C(C(C)C2CCCOC2)C(=O)NCC(F)F)CCc2ccc(F)c(F)c2C1 30363,N1(C(c2ccc(Oc3ccccc3)o2)C(=O)NC)CC2CCC1CN2CC 30364,Cc1ccc(F)cc1C(=O)NC1CCCN(C(=O)Cn2ccc(C(F)(F)F)n2)C1 30365,C(=O)(C(C)(C)C(C)O)NCc1cccc(CN(C(CC(C)O)=O)C)c1 30366,C(CC1CCOCC1)(C(=O)N1CCCCCO1)NC(C1CN2CCC1C2)=O 30367,CCC(COC)C(=O)N(C(C)CN(C)C(c1cc(Cl)cnn1)=O)C 30368,CCCCCC(O)CC(=O)NCCC1CCCCN1C(=O)C(CC)SC 30369,C1(NC(c2ncnc(=N)[nH]2)=O)CC2CC(NC(c3ccno3)=O)CC12 30370,C1(C(CC)C)CCN(c2cc(N3CCOC(c4nncn4C)C3)ncn2)CC1 30371,C#CC1(C)CCCN(C(=O)C(CC(=C)C)NC(c2cc(C3CC3)[nH]n2)=O)C1 30372,C1(CNC(Cc2[nH]cc(C)c2)=O)COCCN(C(c2csc(CO)n2)=O)C1 30373,C(=O)(C(C)(C)CCSC)NC(C1CC1C(=O)NCC1(F)CC(CNC(N)=O)C1)C 30374,CC(C)N=C(NCC1CC(OC(C)(C)C)C1)NC1CC12CC2 30375,c1(CC)ccc2c(c1)CN(c1nnc(-c3ncc[nH]3)n1CCC#N)CC2 30376,c1(OC)nn(C)cc1NC(c1ccc(CNC(=O)C(O)CC2CCCC2)cc1)=O 30377,Cc1ncc(C(=O)N(C)CC2CN(C(C3COCC(C)(C)O3)=O)C2)c(C2CC2)n1 30378,Cc1cccnc1C(N1CCCC1C(C)(C)CNC(=O)CC1CCC(C)(C)C1)=O 30379,c1(OCCCC)ccc(-n2cc(-c3c[nH]nc3C(F)(F)F)nn2)cc1 30380,N1(C(c2cnc(CC)s2)=O)CCCCC(NC(=O)C(O)CC2CCOCC2)C1 30381,c1(C(N2CC(NC(C(C)n3ccnc3)=O)C(C)(C)C2)=O)c(O)cc(Cl)cc1F 30382,C1(NC(C2(CCOC)CC2)=O)CCCCC1CNC(=O)Cc1ccncc1 30383,c1(C(N)=O)cc(C(N2CCC(F)C(NC(C3CCCSC3)=O)C2)=O)ccc1Cl 30384,C(=O)(CCCCC(=O)N(C)CCNC(=O)Cn1cc(Br)c(C)n1)OC 30385,c1(OC)ccc2cccnc2c1C(N1CCC(CNC(=O)C(C)C#N)C1)=O 30386,N1(C(c2c(CC)csc2)=O)C2CCC1CN(C(c1ccn(C(C)C)c(=O)c1)=O)C2 30387,c1(C(=O)OC)cc(Cl)nc(Cl)c1NC(C1(C)CCN1C(c1cscc1C)=O)=O 30388,c1(C(N2CCCC2CCNC(C23C=CC(CC2)C3)=O)=O)ccc2c(c1)COC2=O 30389,C(=O)(CCCC(=O)N(C)C)N1CC(OC)C(NC(c2cnn(C(C)C)c2Cl)=O)C1 30390,N1(c2nnc(C(CC)(C)C)o2)CCCC(C)(NC(=O)C(C)=C(C)C)C1 30391,C1(C(=O)NCC2CC3(CC3)CN2C(c2ccc[nH]2)=O)CCC(C2CC2)CC1 30392,C1(C(=O)OCCn2nccc2N)(CNC(=O)OC(C)(C)C)CCCO1 30393,N1(C(C2CCCC(C(N)=O)C2)=O)CC2(C1)CN(C(C1CCC=CCCC1)=O)C2 30394,c1(SNc2ccnn2C2CC2)cccc(C(C)=O)c1.C123CC(C1)(C2)C(=O)N3 30395,C1(C(=O)NC(CC=CC)C(=O)N2CCC(CC3CC3)C2)CCC(O)CN1C 30396,N1(C(c2c(C(C)(C)C)ocn2)=O)CCC(F)C(NC(C2(F)CC2(C)C)=O)C1 30397,C1(NC(C2C(C)(C)OC2(C)C)=O)CC2CN(C(=O)C(F)(F)C(F)F)CC2C1 30398,C1(CN(C(C(C)NC(=O)Cc2cccs2)=O)C)CN(C(=O)C(N)=O)CCO1 30399,C1(N(CCC)C(c2cscn2)=O)CCN(C(c2ccsc2CC)=O)C1 30400,N1(CCC#C)CCN(C(=O)COCCNC(=O)CC2CCCN2C)CC1 30401,N1(C(C(CC)(C)CC)=O)CCC2CC(NC(=O)COc3ccsn3)CCC2C1 30402,Cc1nc(NC2CC3CN(C(c4ccn(O)c(=O)c4)=O)CC23)c(F)c(C)n1 30403,Cc1ncc([N+](=O)[O-])n1CC(N1CCN(C2CCCC2O)CC1)C 30404,c1(C(=O)OC)ccc(F)cc1C(=O)OC(c1nccs1)C 30405,C1(C(N2CC(C=C)C2)=O)CN(C(=O)CCc2cccs2)CCO1 30406,N1(CC(C2CC2)NC(=O)OC(C)(C)C)C2CCCC1CC1(C2)NC(=O)NC1=O 30407,c1(-c2ccc(C(N3CCCC3C3CC3(F)F)C(=O)NCC=C)s2)cn(C)nc1C 30408,CC1C(C(=O)N2CCCC2CC(=O)NCC2CN3CCC2C3)=NOC1C 30409,N1(C(c2ccc(CC)o2)=O)CCN(C(c2cc(Cl)cn2C)=O)CC1CC(F)(F)F 30410,CC1CN=C2NC(C(=O)N3C4CCC3C(CNC(c3cccnn3)=O)C4)=NN2C1 30411,C(C1=CCN(C(C2CCC(CCO)CC2)=O)CC1)NC(c1cn(C)nn1)=O 30412,Cc1cc(C(=O)NCC2C(CNC(c3cc(C)oc3C)=O)C2(F)F)c(C)[nH]1 30413,CC(C)(C(=O)NC1CC(F)(CNC(c2cc(C3(C)CC3)on2)=O)C1)C(N)=O 30414,c1(CCC(=O)NCC2(CN(C(CCSC)=O)C)CC2)ccc(Cl)cc1 30415,c1(C(N2CCC(OCCNc3snc(COC)n3)C2)=O)cnc(C(F)(F)F)cn1 30416,C(=O)(C1=NOC(C)C1C)N1CCC(C(C(=O)NCCC(=O)NC)F)C1 30417,CC1C(C(N2CCN(CC3(NC(C4(C)CCCN4C)=O)CC3)CC2)=O)CCN1C 30418,c1(CC)nc(CC(=O)NCC2CCN(C(=O)CSC3CCCCO3)C2)cs1 30419,C1(C(=O)NCCC2CCC(NC(COCC)=O)C2)CC12CCC1(CC1)CC2 30420,c1(C(=O)NC(CNC(C(CC=C)CC)=O)CC)ccc2c(c1)COCO2 30421,c1(C(=O)NC(CNC(CCOCC)=O)(C)C2CC2)ccc(C2(C#N)CC2)cc1 30422,c1(C(N2CC(CNC(COC)=O)N(C)CC2)=O)cc2ccccc2n1CC(F)(F)F 30423,c1(SC2CC2)cccc(CC(=O)N(C)C(C2ON=C(C)C2)c2ccccc2)c1 30424,C1(NC(C(CCC)C)=O)CCC12CN(C(=O)CCCCN1CCCCC1)C2 30425,c1(C(=O)OC)cc2ccc(N3CCCCC3)cc2o1.N12CCCC(C1)C2=O 30426,C(=O)(C(C)Cc1cn(CC(=O)N(C)Cc2cn(CC(C)(C)O)nn2)nn1)OC 30427,CCC(C)C(C(=O)NC1CCCCC1C(N1CC=CC1(C)COC)=O)N(C)C 30428,c1(C(N(C2C3CN(C(=O)CC4(C)CC4)CC23)C)=O)ccc(Cl)cc1 30429,C=CCC(C(=O)NCC1(O)CCN(C(c2ncoc2CC)=O)C1)C(C)C 30430,CC(C)(O)C(F)(F)CNC(=O)C(CNC(=O)Cn1cccc1)CC1CCCC1 30431,c1(C(N2CCN(C(C=CSC)=O)C(C)C2)=O)cc2c(F)ccc(F)c2s1 30432,c1(C(=O)OC)ccc(C(=O)NC(C)CNC(=O)C(=O)NCC2CC2)nc1C 30433,c1(OC)ccc(SCC(=O)NCC(C2CC2)NC(=O)CCCc2ncco2)cc1 30434,c1(C(N2CCCN(C(C3CCCC(O)C3)=O)CCC2)=O)cnc2c(c1)CCCO2 30435,N1(C(CC(C)OC)=O)CCCC(C2CN(C(=O)Cc3cc(F)ccc3C)C2)C1 30436,CN1CCCCC1CC(=O)NC1CC1C(=O)Nc1ccccn1 30437,c1(C(=O)NC2CCCC(CNC(C3CC3C(F)F)=O)C2)cn2ncccc2n1 30438,C1(NC(C2CCCOC2)=O)(CO)CCCN(C(c2cnn[nH]2)=O)C1 30439,C(=O)(CC(C(F)F)C(C)(C)C)N1C(C)CC(NC(c2cc(C3CC3)on2)=O)C1 30440,C1(C(=O)NC2(CCC)CC2)CCN(C(=O)Cc2csc(Cl)n2)C1CC 30441,C(=O)(C1=CS(=O)CCC1)N1CCC(NC(C2C(F)(F)C23CCC3)=O)(CF)C1 30442,C1(NC(CCOC(C)C)=O)CC(NC(c2cc(O)cc(F)c2)=O)C12CCOCC2 30443,C1(COC)(NC(C2CCN2S(C)(=O)=O)=O)CN(C(=O)CCCN2CCCC2)C1 30444,C1(CCNC(CSCCC)=O)C(C)CCCN1C(c1cc(=O)cc[nH]1)=O 30445,c1(C(N2CCC(C)(CNC(CN(C)C)=O)CC2)=O)ccc2c(c1)C(C)(C)CO2 30446,C1(C(N2CCC(C)(NC(CCc3n(C)cnc3)=O)C2)=O)C2Cc3ccccc3C12 30447,C1(NC(c2c(C)nc(C)o2)=O)CCC2CN(C(C)C(=O)NC3CC3)CC2C1 30448,NC(Cc1ccccc1Br)CC(=O)NC(c1ccccn1)C(N)=O 30449,CC(C)C(C)(O)C(=O)N1CCC(CCC(=O)NC(CN(C)C)CCO)C1 30450,C12CCc3nc(sc3C1)-c1nc(CCSC)nn1C2.c1(CC)cccnc1 30451,c1(CN(CCC#C)CC)cc(OC)c(OC)c(Br)c1 30452,O=C(NNc1ccc(S(=O)(=O)Nc2nncs2)cc1)C1CCCC(C(F)(F)F)O1 30453,C1(CCNC(=O)NCc2ccc(I)o2)CCN(C(c2ccccc2)=O)CC1 30454,C1(C)(C(N2CCC(N(C(c3c(COC)noc3)=O)CCO)C2)=O)CCC(F)(F)C1 30455,C1(NC(c2cnc(C(F)F)s2)=O)CN(C(=O)C2=CCCC2)CCC1F 30456,C1(OC)CCOCC1NC(=O)C(c1ccc(Br)cc1)(C)N 30457,C1(CCC(C)(C)NC(C2CC2(F)F)=O)CCN(C(=O)COCCF)CC1 30458,C=Cc1ccc(CNC(C23CC2CN(C(C2Cc4ccccc4O2)=O)C3)=O)cc1 30459,C(=O)(C(F)C1CCOC1)N(C)CCOCCCNC(=O)C=C1CC1 30460,CC1CN(C)CC1C(=O)NC1(CCNC(c2ccc(C3CCOC3)s2)=O)CCC1 30461,c1(C(=O)NCC(CNC(COCc2onc(C)n2)=O)O)c2c(nn1C)CCSC2 30462,C(=O)(CCCCN=[N+]=[N-])N1C(C)CN(C(c2ccc[nH]2)=O)CC1 30463,CN1CCC(C(=O)NCCCNC(C2(C(=O)N(c3ccccc3)CC)CC2)=O)C1 30464,c1(C(=O)NC(C2CN(C(C3CC3(C)C)=O)C2)C)ccc(N(C)C)cn1 30465,C1(CNC(c2cnn(C(C)C)c2N)=O)CCN(C(=O)CC(C)(C)N(C)C)C1(C)C 30466,N1(C(CC2C=CC(NC(C3N(C)CC(O)CC3)=O)C2)=O)CC(O)CC12CCOC2 30467,C#CCCCC(C)OC(C1CC1c1ccccc1Nc1ccccc1)=O 30468,N1(C(CC(=O)NC)=O)CC2C(CNC(C3(c4ccccc4F)CC4(CC4)C3)=O)C2C1 30469,Nc1ccc(C(N2CC(CC(N3CCC3CO)=O)C3(CC3)C2)=O)nc1F 30470,C1(C(N(CC)Cc2nc[nH]n2)=O)CC(F)CN1C(=O)Cc1ccc(C(C)(C)C)cc1 30471,c1(C(=O)NCCCCCNC(C(N2CCOCC2)C)=O)cc(O)ncc1Br 30472,Cc1cc(=NCc2n[nH]c3c2CCC3)[nH]c(=NCc2ccc(C(F)(F)F)cc2)[nH]1 30473,C=CCC(C(=O)N(C(C)CNC(=O)C(c1ccc(Cl)cc1Cl)(C)C)C)C(C)(C)C 30474,N1(C(CCC2C(C)(C)C2)=O)C(CC(=O)NCC23CCCC2C3)C2CCCC12 30475,c1(C(N2CC(C)C(CNC(=O)CC3CCCCO3)C2)=O)c[nH]c2c(F)cccc12 30476,c1(OC)ncnc(C(N2CC3C(CN(C)C(C4(C)CCCCC4)=O)C3C2)=O)c1F 30477,C1(C(N2CCN(C)CC2)=O)CCC2(CC2)N1C(C1(CO)CCC1)=O 30478,C1(NC(CC=C)=O)CN(C(=O)Cc2c(Cl)cccc2Cl)CC12COC2 30479,N1(C(=O)Cc2ccn3cncc3c2)CCC2CCN(c3ccncn3)CC2C1 30480,c1(N2CCCC(CNC(c3cc(C(C)C)nn3C)=O)C2)cc(S(C)(=O)=O)ncn1 30481,C(=O)(C(C)(C)CC(F)F)NCC(C(C(C)C)C)NC(c1ccsc1Cl)=O 30482,C1(C#N)(Cc2n(-c3ccccc3)nc(Cn3cccn3)n2)CCOCC1 30483,N1(C(C2C(C)SCCC2)=O)CC(CC(=O)NC(c2ccon2)(C)C)C2(CC2)C1 30484,Cc1cncc(C(=O)NC2CCC(NC(C3CN(C4COC4)C3)=O)CC2)c1C 30485,CCC(CCO)CN=c1nc(N2CCC(CC(C)C)C2)c2c(ncn2C)[nH]1 30486,CC1(C)CCC(C(N2CC(C#N)C2)=O)CN1C(=O)CCc1ccncn1 30487,CC(C)C(C)(CN=c1cc(F)nc[nH]1)NC(C1CCN1C1CCCC1)=O 30488,c1(C(N2C(C(=O)Nc3ccc(C)nc3)C=CCC2)=O)ccc2c(c1)CCCC2 30489,C12(NC(c3cnc4n3CCS4)=O)CCCCCC1N(C(C1CCOCC1)=O)CC2 30490,c1(C(N(CCC2N(C(CSC)=O)CCCC2)C)=O)[nH]c2cc(F)cc(F)c2c1C 30491,N1(C(C2CCC(=O)C2)=O)CCc2ccccc2C(NC(=O)Cc2ccc(Cl)s2)C1 30492,N1(C(c2c(CNC(C(c3cnn(C)c3)C)=O)occ2)=O)CCCN(C)CC1C 30493,Cc1cc([N+](=O)[O-])ncc1C(=O)NCCCN(C(C1CCCS1)=O)C1CC1 30494,c1(N(C(C)=O)C(=O)C2CC2)cccc(C(N2CCCCC2c2ccccc2)C)c1 30495,c1(-c2nc(C(CC)C)nn2C23CC(C2)C3)ccc(Cl)c(S(C)(=O)=O)c1 30496,c1(OC)cc2cc(C(=O)NC(C)CCS(C)=O)[nH]c2cc1F 30497,N1(C(C=CS(C)=O)=O)CCN(C(c2ccccc2C(N)=O)=O)CC1c1cn[nH]c1 30498,c1(CCC)cccc(OC(C2CC2c2cccs2)=O)c1 30499,Cc1ccc(Br)cc1C(=O)NCC1CC(C)(C)CN1C(=O)C(F)C(F)(F)F 30500,N1(C(CC(C)SC)=O)CC(NC(c2cc(C)cc(F)c2)=O)CC(F)C1 30501,c1(C(N(C(C)CNC(=O)C(F)(F)C(F)F)CC)=O)ccc2c(c1)COC2 30502,N1(C(c2cnc(C)nc2C)=O)CC(CO)C2(C1)CN(c1nc(C)nc(C)c1F)C2 30503,C(=O)(CC(CC1CC1)NC(=O)CS(=O)CC)N(c1cccc(F)c1)CC 30504,c1(CCN(C(=O)C(C2CCN(C(=O)OC(C)(C)C)C2)F)C)cc(F)cc(F)c1 30505,c1(N2CCC(N(C)C)C2)[nH]c(=NCC23CC2CN(C)S3(=O)=O)nc2sccc12 30506,C1(C(=O)NC2(C)CC(NC(c3c(C)ocn3)=O)C2)CCOC2(CCC2)C1 30507,N1(C(C(CN(C(c2ccc(C)cc2)=O)C)C)=O)CCCC(C(N)=O)C1C 30508,c1(C(N2CC(CCNC(C(CCC)OC)=O)C(C)C2)=O)c(F)ccc2nc[nH]c12 30509,C(=O)(C(F)C(C)C)NC(CCOC)CNC(c1ccc(CN2CCCC2)o1)=O 30510,c1(C(N2CCC(CC)(NC(c3cnoc3)=O)CC2)=O)ccc2c(c1)nc(O)n2C 30511,C1(C(=O)NC(C)CN(C(=O)CCc2sccc2Br)C)CC(C)(C)CO1 30512,CCC(C)(CNC(C1(C(C)C)CCN(C(=O)CC(C)SC)C1)=O)CO 30513,C1(NC(C2SC3C=CC2C3)=O)CC2CCC1N2C(=O)C1=C(Cl)CCC1 30514,CC(C)(C(=O)NC(Cn1ccnn1)C(=O)NCCc1cnco1)C1CCOC1 30515,C(=O)(CC(C)C(F)(F)F)NCC1=CCCN(C(C2=CCCC2C)=O)C1 30516,C1(CC=C)(C(=O)N(CC(=C)C)C)CN(C(C2C=C(C)CS2)=O)C1 30517,C(C(CC(F)(F)F)NC(=O)CC(CC1CCCC1)CC)NC(COCC)=O 30518,C1(C(C)(C)CNC(C2COC(=O)N2)=O)CCN(C(C2CCC23CCC3)=O)CC1 30519,CC(C)(CS(N)(=O)=O)C(=O)N1CC(CCCCNC(C2CC3(C2)CC3F)=O)C1 30520,C(=O)(C1=CC2C=CC(C1)C2)NC(CC(=C)C)C(=O)NC1CC(CCF)C1 30521,C1(NC(CC(=O)OC)=O)CCC(N(C(=O)C=CBr)C)CC1 30522,S(=O)(=O)(c1cc(C)cnc1NCc1csc(C)c1C)N1CCCC(CSC)C1 30523,Cc1cc(=NCC2(CNC(=O)Cc3c(O)ncnc3O)CC2)[nH]c(C2CC2)n1 30524,C(=O)(CCCCCCc1ccccc1)N(CCC)C(c1ccccc1OC)C 30525,c1(OCC(=O)NC2C(CC)CN(C(=O)CC(=O)NC3CC3)C2)ccc(F)c(F)c1 30526,Cn1ncc(C(=O)N(CCC(=O)NC2COC(C)(C)C2)CC2CC2)c1C#N 30527,CC1CC(C(N2CCCC(CN=[N+]=[N-])C2)=O)CN(C(=O)CCNC(=O)CO)C1 30528,c1(N(CCN2CCC(CC=C)(NC(=O)CC(C)CC)C2)C)c(Cl)cc(Cl)cc1Cl 30529,C1(C(N2CCN(Cc3ccc(Br)cc3)CC2)=O)CC2CC2N1Cc1cnco1 30530,N1(C(c2ccnc(C)n2)=O)CC2C3CCC(C2C1)N(C(C1(N(C)C)CCC1)=O)C3 30531,CC1CCC(C)(C=CC(=O)NCc2ccccc2SC(F)(F)F)C1(C)C 30532,C1(C(=O)NCCC2(OC)CN(C(c3ccccc3C(N)=O)=O)C2)CC(O)C(F)C1 30533,c1(CCC(=O)NCC(C)NC(=O)CC2CCN(C)C2=O)ccc(Cl)cc1 30534,C(CS(=O)c1cccc(Br)c1)N1CCCC(NC(C)=O)C1 30535,N1(C(C)=O)CCC(N2CCC(NC(C3CC3NC(=O)COC3CC3)=O)CC2)CC1 30536,c1(OC)ccc(NC(C2(O)CCN(CC3C4COCC34)C2)=O)c(C)c1 30537,C1(CNC(C(C)OCC)=O)(CNC(C2CC(F)C2)=O)CC12CCC2 30538,c1(C(N2CCN(C(CCOCC)=O)C(CCO)C2)=O)oc2ccccc2c1CC 30539,C(=O)(C(C)(C)CS(N)(=O)=O)NCC1CN(C(c2c(CC)ncs2)=O)C(C)C1 30540,c1(-c2cn(C3CN(C(Cc4cc(C)[nH]n4)=O)C3)nn2)cncc(C(N)=O)c1 30541,c1(CN2CCCC(CC(=O)Nc3c(CC)nccn3)C2)ccc2c(c1)CCO2 30542,c1(CN(C(C2CCCN(S(=O)(=O)CCCCl)C2)=O)C2CC2)ccc(F)c(I)c1 30543,C1(CN(C(CCN(C(c2nccn2CC)=O)CC)=O)C)CCOC1C 30544,c1(C(N2CC(O)CC(NC(CC=CC=C)=O)C2)=O)nc2ccccc2nc1C 30545,CC(C)(C(=O)NCCCCNC(C1(C)CC1F)=O)C1CC1 30546,C(C(C(=O)NCCN1CC=CCC1)NC(c1ccn(C(F)F)n1)=O)OC 30547,N1(CC(C)(C)NC(C(CC)OC2CCCCC2)=O)CCN(C(C2CC2C)=O)CC1 30548,C1(C)(C(=O)NC2C(N(C(CCOCCC)=O)C)CCCC2)CCCCCCC1 30549,C(C1CCCCCC1)=CC(=O)NCCCC(C)NC(C1CC(C(C)C)C1)=O 30550,N1(C(c2c(CC)[nH]nc2Cl)=O)CCC(NC(=O)CCc2cccc(C)c2)C(C)C1 30551,C(C)(CCCC(=O)NCC1CCC(O)C1)NC(C(c1ccn(C)c1)C)=O 30552,c1(CC(=O)NCC(CC)NC(=O)CSCCN(C)C)scnc1C 30553,C(=O)(CC(C)CC(=O)NC1CCN(C(C2(C3CC3)CCOCC2)=O)C1)OC 30554,C(C(CCC)C(=O)N1CCN(C)CC1CCO)NC(C1(C=C)CCCC1)=O 30555,C12(NC(=O)CSc3ccccc3)CCC1CN(C(c1cccnc1)=O)C2 30556,N1(C(C=COCC)=O)CCOC2CCN(C(=O)C=CC(C)C)CC12 30557,N1(C(c2cc(C)on2)=O)CCCC(C)C1CCN(C(=O)CN1CCCS1(=O)=O)CO 30558,C(=O)(C(C)CC(F)F)NC(C(=O)NCCc1cnc(C)[nH]1)CO 30559,CC1CCN(CC2CCCC(=O)N2)CC1NC(c1ccsc1-n1cnnn1)=O 30560,C12(C(=O)NCC(CNC(c3nc(OCC)oc3)=O)(C)F)CCCCC1C2 30561,CC1CCC(C(=O)NCCCc2cncnc2)CN1C(=O)C(=O)NC1CC1 30562,c1(NC(C2(NC(CN(C)C(=O)C3CC3)=O)CC2(C)C)=O)ccc2ccoc2c1 30563,C(C(C(=O)NC1COCC1NC(=O)C(C)(C)c1cocn1)OC)OC 30564,N1(C(Cc2cn(CC)nn2)=O)CC(F)CC1C(=O)NCc1csc(C)c1 30565,N1(c2nc(OC)nc(C)c2)CCC(F)(F)C(CNC(c2sccc2F)=O)C1 30566,CC1CCN(C(=O)CC2N(C(=O)CN3CCSCC3)CCC2(C)C)CC12CCC2 30567,CC1(C)CCN1CC(=O)NC1CCCC1NC(C1(c2cccnc2)CCCC1)=O 30568,C(CC(C(C)C)NC(=O)CCNC(C)=O)NC(C1CC(C(F)F)(OC)C1)=O 30569,c1(CC(=O)NC(C(C)NC(COCCCCC)=O)CO)ccc(C2CC2)cc1 30570,c1(C(=O)NC2C3(CC(NC(C4(C)CC(=C)C4)=O)C3)C2)cn2c(n1)CCC2 30571,C1(C(=O)NCC2(C(=O)OC)CCC2)C=CC(NC(=O)CC2CC(=O)C2)C1 30572,Cc1cnn2cc(C(N3CC(O)CC3c3ccc(F)cc3)=O)cnc12 30573,CC1CN(C(=O)CCSC2CCCC2)CCCN1C(C1CSCCS1)=O 30574,C1(OC)CCCCC1C(=O)NCc1cccc(CNC(=O)COC2CCOC2)c1 30575,C1(CNC(c2c(OCC#C)nccc2)=O)CN(C(c2cnn[nH]2)=O)CC(C)(C)O1 30576,N1(C(C(C)N(CC(F)(F)F)C)=O)CC2(CCC2)CC1CNC(c1nn[nH]c1Cl)=O 30577,c1(C(N2CCC(N(C(=O)CCS(C)=O)CCC)C2)=O)ccc(Cl)c(C)c1 30578,O(C1CCCc2ccccc21)CC(=O)NC1CCN(C(c2cnc(C)o2)=O)C1C 30579,C1(C(C)NC(CNS(NC)(=O)=O)=O)CN(C(=O)CC2CCCC2)CCO1 30580,C1(C(=O)NCC2CCCN2C(C2C=CC=CC=C2)=O)CC2CCC(C1)S2 30581,N1(C(c2ccc(CNC(C(CC)CN(C)C)=O)nc2)=O)CC(O)CC1(C)C 30582,c1(C(=O)NCC(N(C(CC(CCC)C)=O)C)C2CC2)cnc2scc(C)n2c1=O 30583,N1(C(CCN(CCC)C)=O)CC(NC(c2ccc(=NC)[nH]c2)=O)CC(C)(C)C1 30584,C(C(C(=O)NC(c1cn[nH]c1)C)C(C)C)NC(C1CC(CCC)C1)=O 30585,C(N=c1cc(CC(C)C)nc[nH]1)C1CN(C(C(C=C)c2ccccc2)=O)C(C)C1 30586,c1(C(=O)NC(C2N(C(C(C)c3cncs3)=O)CCC2)C)n[nH]c2ccc(Cl)cc12 30587,Cc1cnnc(O)c1C(=O)NCCCCC(C)NC(=O)CC(C)NC(N)=O 30588,c1(C(N2C(CN(C(c3cn(C)cn3)=O)CC)CCC2)=O)cc(OC(F)F)n(C)n1 30589,C(=O)(C1=NOC2(CCC2)C1)N1CC(CCNC(=O)C2=CCC(C(F)(F)F)OC2)C1 30590,N1(C(c2c(OC)cc(Cl)cc2)=O)CCN(C(=O)OC(C)(C)C)CC12CCC2 30591,CC1(C)CCC(C(=O)NCC2(C)CCCN(C(c3ocnc3C(F)F)=O)C2)OC1 30592,c1(C(=O)NCC2CCC(NC(=O)COCC3CCC3)C2)ncccc1Cl 30593,c1(OCCCC(=O)NCC2CCN(C(C(CSC)C)=O)C2)cccc([N+](=O)[O-])c1 30594,Cc1cc(C(N2CCCC(CC(=O)NC3CN(C)CC3C)CC2)=O)cnc1O 30595,N1(C(C(CNC(c2oc(C)c(CO)c2)=O)CC2CC2)=O)CC2COCC2(CO)C1 30596,c1(NCCN2C(=O)CCCC2)nccc(=NCC2(CF)CC(F)(F)C2)[nH]1 30597,C12(C(N3CC(NC(C4(OC)CCOCC4)=O)C3)=O)CCOC1CS(=O)(=O)C2 30598,c1(C(N2CCC(N(C(c3cncc(OC)c3)=O)C)C2)=O)c(F)ccc(F)c1Cl 30599,c1(OC)ccc(CCNC(c2ccccc2-c2ccccc2F)=O)c(F)c1F 30600,C(=O)(C(F)C(C)CNC(c1ccsn1)=O)N(C(C)C)CCN(C)C 30601,c1(C(N(C2CC(C(=O)NC3CC3(F)F)C2)C)=O)ccccc1S(C)(=O)=O 30602,C=CCC(C(=O)NC(C)CCN(C)C(c1cnn(C)c1OC)=O)C(C)C 30603,c1(OC)ccc(C(N2CCC(CNC(c3csnc3OC)=O)C(C)C2)=O)c(F)n1 30604,C1(NC(COCCSC)=O)CC12CCN(C(c1csc3cncn13)=O)CC2 30605,c1(C(=O)N(CC(CCNC(CN(c2ccccc2)CC)=O)O)CC)c(C)n[nH]c1C 30606,C1(C(=O)NC(C2(O)CCCCC2)C)CCC(C)(C)N(C(=O)CN2CCCC2)C1 30607,c1(C(=O)NCC2(C)N(C(=O)C=CC(C)C)CC(OC)C2)cc2cnn(C)c2s1 30608,N1(C(C2CCN(C(CC)=O)CC2)=O)CCC(CNC(C2CC(OC)C2)=O)C(O)C1 30609,N1(C(=O)CCF)CCCC(C2CCCN(C(c3ccc4nncn4c3)=O)C2)C1 30610,CCCCCCN(C(c1sncc1C)C(=O)NCc1cccs1)C1CC1 30611,Cc1[nH]nc(C(=O)N(C)CCOCCCN(C(=O)Cc2ccnn2C)C)c1Cl 30612,N1(C(c2c(C)c(Br)cnc2)=O)CCCN(C(=O)C(C)NC=O)CC1C 30613,Cc1noc(C)c1NC(=O)CC1(NC(C2CCCC2C(C)C)=O)CCC1 30614,n1(C(C(=O)N(CCNC(c2c(C)ccnn2)=O)C(C)C)C)cnc2ccccc12 30615,CC1=C(C(=O)N2C3CCC(C3)C2CC(N2CCCCC2C(F)F)=O)CCC1 30616,c1(C(N(C2CCN(C(C3CCCOC3C)=O)C2)CC#C)=O)cc(C(N)=O)nn1C 30617,c1(CCC(=O)NCC(C2CCCC2)NC(COC(C)C)=O)cnn(C)c1 30618,n1(C(C)C)cnnc1CC(N1CC(CCCCNC(C2CC2C)=O)C1)=O 30619,C1(NC(Cc2cnc(C)s2)=O)CC2CC1CN(C(C1(O)CC1)=O)C2 30620,C1(CNC(C2(SCC)CC2)=O)CCN(C(=O)Cc2cccc(C)c2)C12CCC2 30621,C1(C(N(CCCCC)CC(N)=O)=O)CC12CCc1cc(Br)ccc12 30622,CCC(=O)CCC(=O)N(CCCCN(C)C(c1cocc1C(N)=O)=O)C 30623,N1(C(C(C)SCCCC)=O)CC(C2CC2)(C(=O)NCc2csc(C)c2C)C1 30624,C1(NC(C=NOC)=O)CCC2(CCN(C(=O)CCc3ncc(F)cn3)C2)C1 30625,c1(C(=O)OC)cncc(CNC(=O)C(=O)NCCCCN(C)C)c1 30626,N1(C(C2N(CCC)CCC2)=O)CCc2ccccc2C1CNC(c1ccns1)=O 30627,c1(-n2cc(CN)nn2)ccc(C(=O)NCCc2cccc(Br)c2)cc1 30628,C1(NC(C2CCN(C)C2)=O)CCC12CN(C(=O)C=CCF)C2 30629,N1(C(C(CCC)NC(C)=O)=O)CC2CCC(NC(=O)CSC(F)(F)F)C2C1 30630,Cc1snnc1C(=O)NCC(C)N(C(=O)CC1(Oc2ccccc2)CC1)C 30631,N1(C(C(CCC)CNC(c2nccnc2C)=O)=O)Cc2nncn2C(C)C1 30632,N1(C(CCC(=O)NC)=O)CC(NC(C2(C(F)F)CCCCC2)=O)CCC1C 30633,Cc1cccc(C)c1NC(=O)CNC1CCC(Nc2ncccn2)CC1 30634,CCC(F)(F)C(=O)N1CCC(C(C)CNC(=O)CCC2CC(F)(F)C2)CC1 30635,N1(c2n(CCS(=O)(=O)N(CC)CC)c(C(C)C)nn2)CCOC2(CCSC2)CC1 30636,N1(C(C2=CCN(C(c3cc(C)c(O)nn3)=O)C2)=O)CC2CCC1C(CO)C2 30637,S(=O)(=O)(c1ccc(C(=O)O)nc1)NC(C(c1ccccc1)OCC)=O 30638,N1(C(c2c(OC)csc2)=O)CC(CNC(C2CC(=C3CCC3)C2)=O)C(O)C1 30639,c1(C(=O)NCCN(C(c2c(CCC)nns2)=O)C(C)C)cccc2ccncc12 30640,c1(C(N2C(C(C)NC(CNC(CC)=O)=O)CCCC2)=O)cc(C)n(C(C)C)c1C 30641,C(=O)(C#CC1CCOCC1)N1CC(CCCCNC(c2n(CC)c(O)nc2)=O)C1 30642,C(=O)(CCC(=O)C(C)(C)C)N1CCC(C)C1CNC(=O)C(c1ccccn1)O 30643,N1(C(c2c(COC)noc2)=O)CC2CCN(C(c3cc(N)ccc3C)=O)C2C1 30644,CC(C)C(C)C(CNC(=O)COC(F)F)NC(c1cc(N)ccc1F)=O 30645,C(=O)(C(C)(F)C(F)(F)F)NC(C1CCN(C(C2(C(=O)NC)CC2)=O)CC1)C 30646,S(=O)(=O)(c1cccc(C(=O)NC23CC(NC(=O)Cc4conc4C)(C2)C3)c1)NC 30647,Cc1cc(C(=O)NCCCN(C(C2CC(C)C2)=O)C2CC2)nn1C 30648,c1(CC(=O)NCC(CC)NC(C(CCC)NC(N)=O)=O)cc(Cl)cc2c1OCC2 30649,C(CNC(c1ccc(C(N)=O)cc1)=O)(C(C)(C)C)NC(c1cnc(COC)s1)=O 30650,N1(C(C(C(C)(C)C)O)=O)CC2(C(=O)NCCn3ccnc3)CCC1CC2 30651,C1(NC(C2(COC)CC=CC2)=O)C2CCN(C(C3CC(C)(C(C)=O)C3)=O)CC12 30652,c1(CC(=O)NC(C2CCCO2)COC)cccc(NCc2ccccc2Cl)c1 30653,C1(NC(c2n[nH]c(C)c2C)=O)CC2CC(NC(=O)CCn3cccc3)CC2C1 30654,Cc1nc(C(C)C)ccc1C(=O)N(C)CC1(O)CN(C(=O)COc2ccon2)C1 30655,c1(C(=O)NCC(C)N(C)C(c2cnco2)=O)c(F)ccc(N)c1Br 30656,CCC(F)(F)CC(=O)NOCC(=O)NCc1sc(C)nc1C 30657,N1(CCCNC(c2cscn2)=O)CCN(C(c2cnn[nH]2)=O)CC1 30658,c1(COC)cc(C)c(C(=O)NCCC2(C(=O)NCCN3C(=O)CCC3=O)CC2)o1 30659,N1(C(CCOCC(C)C)=O)CCC(C(C)NC(=O)C(F)(F)c2ccncc2)CC1 30660,C1(F)(CNC(C=C(C)C(C)C)=O)COCCN(C(=O)CC2(CS(C)(=O)=O)CC2)C1 30661,Cc1cncc(N)c1.c1(CCC(NOC(=O)C(F)(F)F)=O)ccc(O)nn1 30662,C(=O)(CCCCN(C(=O)C(C)(C)C1(O)CCC1)C)NCC(C)CCO 30663,S(=O)(=O)(c1ccc(=NCCCC(F)(F)F)[nH]c1)N(C1CC(C)OCC1)C 30664,c1(C(N2CCCC(NC(C3(COC)CCCO3)=O)C2)=O)ccc(C)cc1C 30665,CC(C)C(C(=O)N1CCN(C(c2ccc(F)cc2)=O)CC1)NC=O 30666,C(=O)(CC(O)C1CCCC1)NC1C(NC(=O)Cc2ccsc2)C1 30667,c1(OC)ncccc1C(=O)NC1CN(C(c2cn(C(C)C)cn2)=O)CC1O 30668,N1(C(C(=O)NC2CCC2)=O)CCC2CCC12C.CC1(C#N)CC(N)C1 30669,c1(C(=O)NCC2C(NC(c3cnc(OCC)nc3)=O)C2)c(F)ccc2nc[nH]c12 30670,C(=O)(C(CCC(N)=O)n1cc(-c2cncc(Cl)c2)nn1)N(C(C)C(F)F)C 30671,N1(C(c2nc(CS(C)(=O)=O)oc2)=O)CCN(C(c2cncc(O)c2)=O)C2(CC2)C1 30672,c1(NC)ccc(C=CC(=O)NCC(C)(C2CCC2)NC(=O)C(C)CF)cc1 30673,Cc1c(C(=O)NC2C=CCCC2C(=O)NCCCNC(N)=O)nnn1C 30674,c1(C(=O)NCC2CCN(C(C(C)(CO)OC)=O)C2)cc(Cl)c(F)cc1N 30675,CCCCC(=O)C(=O)NCC1CN(C(C2CC23CCOCC3)=O)CCO1 30676,c1(CC(=O)N(C(c2ccccc2)CNC(c2nncs2)=O)C)nnc(O)s1 30677,c1(-c2ccc(CCC)cc2)ccc2[nH]cc(CC(=O)NCCc3cccs3)c2c1 30678,C1(NC(C(=O)N(CC(N)=O)C)=O)CCN(c2ncccn2)C1 30679,C=CC1(C(=O)N(CCCCO)C)CCN(C(c2ccn(C)c2)=O)C1 30680,c1(C(=O)NC(CC)CNC(=O)CC2CC(OC)C2)ccc(N)cc1Cl 30681,N1(C(C2CC(C(C)C)C2)=O)CC(NC(c2ccccc2C(N)=O)=O)C(F)C1 30682,O(NC(=O)C(CCF)NC(=O)CC12CCCC1C2)C(CC)CC 30683,c1(C(=O)NCC2(CN3CCN(C(=O)C4CC4)CC3)CC2)ccc2nncn2c1 30684,Cc1nc(C)c(C(=O)NC(C2CCN(C(c3cc(C(F)(F)F)no3)=O)CC2)C)[nH]1 30685,N1(C(=O)N(Cc2cccnc2)CC2CCCO2)CCCN(CC2CCCO2)CC1 30686,c1(C(N2CCC(C)(NC(C34CCC(OC)C3CC4)=O)C2)=O)cc(F)c(F)cc1F 30687,c1(C(=O)NCCC2CCCC2)ccc(CNC(c2cc(=O)cc[nH]2)=O)nc1 30688,C(=O)(CC(O)CC(C)(C)C)N1C2C(N(C(CCCCCCC)=O)C)CC(C2)C1 30689,C1(C(=O)NCC(C)N(C(=O)C(=O)NCC2CC2)C)CC2CSCC(C1)C2 30690,C1(NC(c2cc(O)cs2)=O)CN(C(C2CC3C=CCC(C2)C3)=O)C2(CCC2)C1 30691,C1C(C)(CO)NCCCC(=O)N1.n1(COC(C2C(C)(C)CO2)=O)cnccc1=O 30692,C1(C(N(CCC(C(C)C)NC(=O)C(C)c2ccco2)C)=O)CN2CCCN1CC2 30693,Cc1cc(C(=O)NC2CCCC(C(=O)Nc3ncc(C#N)s3)C2)n(C(F)F)n1 30694,C#Cc1ccc(C(=O)N(CC(O)COC)C)c(C)c1.c12ccc(s1)C(=O)NC2 30695,Cc1c(-c2nc(-c3cccnc3O)nn2CC2CCOC2)cnn1CCO 30696,C12(CNC(C3CC3(Cl)Cl)=O)CC3CC(CC(NC(=O)C(O)C(F)(F)F)(C3)C1)C2 30697,N1(C(C(CC)(CC)OC)=O)CCN(C(C2CCCC(C)C2)=O)C2(CC2)C1 30698,CC1CN(C(C2CCC3(CCC3)C2)=O)CCCN1C(=O)CCc1cn(C)nn1 30699,C12(C(N(CCN=[N+]=[N-])CC)=O)CC1CCN2C(=O)CC1CC2CC2C1 30700,n1(CCS(CC)(=O)=O)c(=NCCc2sc(N(C)C)nc2C)[nH]c2cc(Cl)ccc12 30701,C1(C(C)CO)CCN(C(=O)C(c2ccnn2C)NC(=O)CCN(C)C)CC1 30702,N1(CCC(N2CCC(C)(C)SCC2)=O)C(=O)C2CC=CCC2C1=O 30703,COn1cnc(C)c1C(=O)NC1CC1CNC(c1cc(C)ccc1C1CC1)=O 30704,C1(CCNC(c2ccc(Cl)s2)=O)CCN(C(=O)COc2cccc(O)c2)CC1 30705,C(C(=O)NC(CC)CO)(C1CC1(Br)Br)N(CC(=O)NC(C)(C)C)CC 30706,c1(C(=O)NCCCCNC(c2ccnc(C)n2)=O)cccc2c1COC2 30707,c1(C(=O)NCCN(C(=O)C(F)CC2CCC2)CC)ncncc1Cl 30708,CC1Cc2ccccc2N1C(C1CC2CCCC2N1)=O 30709,N1(C(C(CC)NC(N)=O)=O)CCN(C(c2n[nH]c(O)n2)=O)CC1c1ncc[nH]1 30710,n1(CC)cc(CN2CCC(CC(N3CCCC(CN(C)C)C3)=O)C2)c(C)n1 30711,c1(C(C2CCOC2)OCC)nc(-c2ccccc2)nn1-c1cnn(C)c1 30712,c1(OC)ccc2nc(C)c(C(=O)NCC3CCC3NC(c3ccsn3)=O)n2n1 30713,C1(NC(c2c(CC)nns2)=O)CN(C(=O)CSc2cccc(C)c2)CCC1C 30714,C1(C(=O)NCC2C(NC(=O)Cc3ccc(Cl)cc3)C2)CN2CCC1CC2 30715,Cc1cnc(C(=O)NC2CCN(C(=O)C(=CC3CCCCC3)F)C2(C)C)cc1C 30716,Cc1ncc(C(=O)NC2(C)CCN(C(c3c[nH]c(Br)c3)=O)C2)c(=N)[nH]1 30717,c1(C(N2C(CNC(C(C)Oc3cccnc3)=O)CCCC2)=O)cccc(N)c1O 30718,N1(C(Cc2nc(C)[nH]n2)=O)CCCC12CCN(C(=O)CCc1nncn1C)CC2 30719,C(=O)(CC(O)(C(F)(F)F)c1ccc(C)o1)NC(CNC(C=C(CC)CC)=O)C 30720,C1(C)(C2CCCN(C(C(=O)NCC)C3CC(OCOC)C3)C2)NC(=O)NC1=O 30721,C1(NC(=NCCSC)NCCc2cccc(O)c2)CCOC2(CCSC2)C1 30722,N1(C(c2ccn(COC)n2)=O)CCC=C(C(=O)N2CC3CCC2CC3)C1 30723,n1(CC)ncc(CNC(N2CC(CC(=O)OC)C2)=O)c1C 30724,c1(C(N2CCCCC(NC(C(CCC)C#N)=O)C2)=O)noc2ncccc12 30725,c1(-c2onc(C3(c4cccc(F)c4)CC3)n2)cc2c[nH]nc2s1 30726,N1(CCN(C)C(C2CN3CCCN2CC3)=O)CCc2ccccc2C1 30727,C1(C(=O)O)C=CCN(Cc2ccc(N3CCCC3)nn2)C1 30728,c1(C(=O)NC2C(NC(c3cnc(C)[nH]3)=O)CCC2)cccc(F)c1F 30729,C1(C(=O)NCc2ccc(C#N)o2)(NC(CC=CCCCCC)=O)CCCCC1 30730,c1(-c2nn(C)c([N+](=O)[O-])c2)ccc(Cl)c(S(=O)(=O)N2C3CCCC2CC(O)C3)c1 30731,C1(C(=O)NC2CCC3(CC3)C2)C2CC(O)C(C2)N1C(=O)CN1CCCC1=O 30732,C1(OC)(CNC(C2(C)CCCCCC2)=O)CCN(C(c2[nH]c(O)nc2C)=O)CC1 30733,CC1(C#CC(=O)N2CCC3C(C2)CN3C(C2CCC(C(F)(F)F)C2)=O)COC1 30734,C1(NC(C(CC)C)=O)CN(C(C2(C(F)(F)F)CCCC2)=O)CC1n1cccn1 30735,C1(N(C)C(c2ccnc(S)c2)=O)CCCCN(C(=O)Cc2c(O)ncnc2O)C1 30736,C1(C(=O)NCC2C=CC(NC(C3(OC)CC3)=O)C2)CS(=O)(=O)CC(=O)N1 30737,C(C)(CC(=O)N1CCC(CF)(NC(C2CCCCC2)=O)C1)(C(F)(F)F)N(C)C 30738,c1(COC)cccc(CNC(C2COCCN2C)=O)c1 30739,c1(C(=O)NC(CNC(c2nccc(C#C)c2)=O)C(C)C)ccc(F)c(C#N)c1 30740,c1(CC(=O)NCC2Cc3cc(Br)ccc3O2)ccc2c(n1)OCCO2 30741,C#Cc1cn(C)nc1C(=O)NCC(O)CC(=O)N1CC(OCCO)C1 30742,C1(C(F)(F)F)(OC)CCCN(C(=NCC(C)C)NC2CN(c3ncccn3)C2)C1 30743,C(=O)(CCCS(C)(=O)=O)NCC1(C(C)(C)C)CCN(C(c2c(C)c[nH]n2)=O)C1 30744,CCC(O)(C(=O)NCC1CC2CC2N1C(=O)C=CC(C)C)c1ccccc1 30745,C1(NC(c2cc(C)no2)=O)CCC2CN(C(c3cncc(C(N)=O)c3)=O)CC2C1 30746,CC1CCCCN1CC(N1CCC(CCC(=O)NCCC(O)C2CCC2)CC1)=O 30747,c1(CNc2nc(-c3cn(CC=C)nc3)sc2)sc(C)nc1C 30748,C1(SCC)CCC(NC(c2c[nH]nc2-c2ccccc2Cl)=O)CC1 30749,c1(C(C)NCC(c2ccc(OC)cc2)(C)O)nc(O)c2c(C)c(C)sc2n1 30750,N1(C(C=CCN(C)CC)=O)CCC(CCC(=O)NC(C)CC2(O)CCC2)C1 30751,c1(CC)cc(C)c2[nH]cnc2c1.N12CCC(C)N(CC1)C(=O)c1ccsc1C2=O 30752,c1(C(=O)NCC(C(C)C)(C)NC(C2CC3(C2)CC3F)=O)cnc(C2CC2)[nH]c1=N 30753,c1(C(C)=O)ccc(NC(c2ccc(NC(c3cccc(I)n3)=O)nc2)=O)cc1 30754,N1(C(c2c(C3CC3)ccc(C)c2)=O)CC2CC(NC(c3[nH]ccc3C)=O)CC1C2 30755,N1(CCNC(=O)CSC2CC2)CCN(C(C2(C(F)F)CCC2)=O)CC1 30756,C12(NC(CC(=O)N(C)C)=O)CC(CNC(c3coc(Cl)c3)=O)(C1)OC21CCC1 30757,C1(C(=O)NC2CCN(CC)C2)CCC(CNC(C2C3COCC23)=O)CC1 30758,C1(OC)(OC)CC(C)(C(=O)NC(C)COCC(C)(C)C)C1 30759,c1(C(=O)NC2(C3N(C(c4nncc(OC)c4)=O)CCC3)CC2)c(Cl)cccc1Cl 30760,c1(-n2cc(NCC3CC34CN(OC)C4)nn2)cc(C(=O)OC)ccc1C 30761,c1(CCCC(=O)N(C2CCN(C(CC=C(C)C)=O)C2)C)ccccc1Cl 30762,CCC(CC(C)C)C(=O)N1CCC(CO)C(NC(=O)CC2CCCC(C)C2)C1 30763,c1(C(N2CC3C(CNC(C(CCN(C)C)O)=O)(C3)C2)=O)c(Cl)cncc1Cl 30764,Cc1cc(NC(c2cc(CNC(c3cc(CO)ccn3)=O)on2)=O)c(=O)n(C)c1 30765,N1(C(C(CCCC)O)=O)CC(CNC(=O)C=C2CCCCC2)OC2(CCC2)C1 30766,N1(C(C2CCN(CC)C2)=O)CCC(O)(C(=O)NCC2(O)CC2)C1 30767,c1(NC2CCN(CC=C)CC2)ncc(S(=O)(=O)N2CCCC(C)C2)cc1Cl 30768,CCC(CCOC)C(=O)N(CC)CC1CCCN1C(c1nccc(OC)c1O)=O 30769,C1(C(=O)NCc2c(C)nco2)C2CC2CN1C(=O)CC1COCCO1 30770,C(CC#CC(C)(C)C)NC(CC(CC)NC(C1(CC)CC1)=O)=O 30771,Cc1cc(C(=O)NC2CCN(C(=O)COCCCF)CC2F)cc2nc[nH]c12 30772,c1(CC(N2CCC(C(C)(C)NC(=O)CC34CCCC3C4)C2)=O)cccnc1Cl 30773,Cc1cc(Cl)cc(C)c1OCCNC(=O)NCc1ncnc(C(C)C)n1 30774,c1(NCC(C)S(N)(=O)=O)ncccc1S(=O)(=O)NC(CC(N)=O)C1CC1 30775,c1(C(N2C(=O)CCC2)c2ccccn2)nnc(C(F)F)n1Cc1ccco1 30776,Cc1ccc(C(=O)N(CCC(N2CC3(CCC3)CC2C)=O)C2CC2)cc1C#N 30777,CN1CCCC(F)(C(=O)NCCOC2CCN(C(C3(C)CCC3)=O)CC2)C1 30778,C1(C)(COC)CCN(C(N2CC(OC(C)(C)C)C2)=O)CC1.N12CCCC1C2 30779,C1(C(N2CCC(N3CCN(C(=O)Cc4cnco4)CC3)C2)=O)CCCCC1(F)F 30780,C(=O)(C(C)CC(F)F)NC1CC(C(C)NC(c2ccn(CCC)n2)=O)C1 30781,CCC(C)C(=O)N(C(CNC(C1CC2CC2C1)=O)C1CC1)C 30782,c1(-c2cccc(C3C(C(=O)NC(CC(C)=O)C)C3)c2)ccc(S(=O)(=O)N(C)C)cc1 30783,C1(NC(c2n(CC)ccn2)=O)CCCN(Cc2nnc(C3CC3)s2)C1 30784,C(=O)(N=c1nc[nH]n2c(C(=O)OC3CC3)cnc12)c1ccc(SC)cc1 30785,C(=O)(C(C)=NOCC#N)NCC1C(C(=O)NCC(COCC)C)C1(C)C 30786,CCC1=C(C(=O)NCC2CCN2C(C2CCc3n[nH]c(C)c3C2)=O)CCCO1 30787,C1(NC(c2c(C)cccn2)=O)C2COCC1CC(NC(=O)C1=NOC(C)C1)C2 30788,N1(C(C(C)NC(C)(C)C)=O)CC(C2CN(C(=O)CSC3CCCCO3)C2)C1 30789,C1(COC)(NC(=O)C(F)CC2CCCC2)CN(C(=O)Cn2cc(Cl)cn2)C1 30790,CCC(CCC(=O)NCC1(C)CC(NC(=O)CSc2ccc(C)cc2C)C1)OC 30791,Cc1c(O)ccc(C(=O)NCC2CC2CNC(=O)CCCOC(C)C)c1C 30792,C1(C)(C(=O)NC2CC(CNC(C(C)OC3CCCC3)=O)C2)CCC(F)(F)CC1 30793,c1(C(=O)NC(CCCCNC(C2(C)ON=C(C)C2)=O)C)c(C)nc(O)nc1C 30794,c1(OC)cc(CN2CC3(CC(CC(=O)Nc4cccc(C)c4Cl)C3)C2)cc(F)c1 30795,C(CCCCCC(=O)OC)n1c(-c2onc(C3CN(OC)C(=O)C3)n2)ccn1 30796,C(N)(CCC(=O)NS(N)(=O)=O)c1nc(C2(C)CC2(F)F)on1 30797,CCCC(CN1CCS(=O)(=O)CC1)CCC 30798,O=C(CC1=CCOCC1)N1CCCN(C(=O)C(C2CC2)C2CC2)CC1 30799,N1(C(C(C)OC)=O)CCN(C(c2ccc(NC(=O)C(C)(C)C)cc2)=O)CC1 30800,CC1(C(=O)NCCOCCNC(C2CCCCNC2=O)=O)CCCNC1=O 30801,C1(CNC(CCCOCCOC)=O)Cc2ccccc2CN1C(c1cc[nH]c1)=O 30802,C(=O)(CCCCCCCC=C)NCC(C)N(C(COCCC#C)=O)C 30803,c1(CCN)cc(C(N2CC(F)(c3cccnc3)C2)=O)no1 30804,C(=O)(C1=NNC(C(F)(F)F)C1)N1CC(C)(NC(C(C(C)O)C)=O)C1 30805,c1(NC(=O)OCC)ccc2c(NCC(=O)OCC)ncn2c1.c1ccccc1 30806,C(=O)(C1c2ccccc2CN1C(c1cnc(O)c(Cl)c1)=O)NC1CC(=O)NC1 30807,Cc1nc(C(N2CCC(CC(N3CCC(C(C)(C)O)C3)=O)C2)=O)c(C)s1 30808,C1(NC(N(C)C2CC2)=O)CCN(C(=O)C#N)CCC1CO 30809,c1(C(=O)NCC#CC(=O)NCc2onc(COC)n2)cnnc(C)c1C 30810,c1(C(=O)NCC(CNC(CC(CC)CC)=O)OC)ccc(F)c2ccoc12 30811,CCCC(CCCNC(=O)CC(c1ccc(F)cc1)C)Nc1ccncn1 30812,C1(CC=C)(NC(c2coc(O)n2)=O)CCCN(C(=O)CC2CCC(C)(C)CC2)C1 30813,C1(C(=O)Nc2ccc(OC)c(N3CCOC3=O)c2)CCC(C2CC2)CC1 30814,N1(C(CN2CCC(C)(C)C2)=O)CCC(NC(c2cnc(C3CC3)[nH]2)=O)C(OC)C1 30815,N1(C(C(C(C)C)SCC)=O)CC(NC(c2cnnn2C(C)C)=O)CC1(C)C 30816,c1(C(N2CC(C)(C)C(NC(=O)C(F)=CCCF)C2)=O)cc(F)c(O)c(F)c1 30817,c1(C(=O)NCC(C)CNC(c2ccnc3ccnn23)=O)cc2c(s1)CCCCC2 30818,c1(NCC2OCC(CNC(CSc3cn(C)nc3)=O)C2)ccnc2ncnn12 30819,C(=O)(CCCCC(F)(F)F)NC1CC(CCNC(C2CCCN(C(N)=O)C2)=O)C1 30820,c1(C(C)C)[nH]nc2cncc(C(N3CCC(C)(NC(=O)C=CCO)C3)=O)c12 30821,c1(OC)cccc(CNC2(c3ccc(-c4cccc(CC#N)c4)cc3)CC2)c1C 30822,c1(NCCC2(O)CN(C(C(CC)SC)=O)C2)ncc(Br)cc1[N+](=O)[O-] 30823,C1(C)(C(=O)NCCCN(C(=O)CC2(C#N)CC2)C)CCC(=O)N1 30824,CC1(C2CC2C(=O)NCC=CC(=O)Nc2cncc(C(N)=O)c2)COC1 30825,NS(=O)(=O)N1CCCC(C(=O)NC2(C3CN(C(=O)CCC(F)F)C3)CC2)C1 30826,NS(=O)(=O)c1ccc(O)c(C(=O)NC2CC(NC(c3ccc(O)nn3)=O)C2)c1 30827,C1(NC(CCC(=O)NCCC)=O)CN(CCOCC)CCC1C 30828,C1(CC(=O)NCc2cn(CCNC(C=CSC)=O)nn2)CC2(CC2)CO1 30829,C1(C(N(CCCSC)C)=O)CCN(C(=O)C(C)c2cccs2)C1C(C)C 30830,C(c1ccccc1)=CCN(C)C(=O)NCc1cc(C(C)(C)C)n[nH]1 30831,S(=O)(=O)(c1cnccc1N1CC(OC)CC(C)C1)NCc1nnc(COC)s1 30832,CC1(C)CC=C(C(=O)N2CC3CC2(CNC(C2CCCN2S(C)(=O)=O)=O)C3)CC1 30833,C(CC(C)(C)C(=O)N1CCN(CCO)CC1)NC(C(c1ccc(C)o1)C)=O 30834,CCC(C(=O)N(C1(C(N2CCC3CCC23)=O)CCC1)C1CC1)C(F)(F)F 30835,N1(CCCNC(C(CC)C)=O)CCN(C(=O)C=CC(N2CCC(C)CC2)=O)CC1 30836,Cc1[nH]c2ncnc(N3CCC(C)(NC(C4C5CCCC45)=O)C3)c2c1C 30837,C1(C)(CC)CCCN(C(C2CCC(O)CN2C(=O)CC2CCOC2=O)=O)C1 30838,N(C(=NCCn1cccn1)NC(C)Cc1cnccn1)CC1(OC)CCOC1 30839,C(=O)(CS(=O)(=O)C1CCCC1)N1CC(CN(c2cc3nncn3cn2)C)OCC1 30840,c1(C(N2CCOC(CCNC(C3CC(C(F)F)C3)=O)C2)=O)ccc2nnnn2c1 30841,C1(NC(C=C(CC)CC)=O)CN(C(=O)C(c2cccc(C)c2)(F)F)CC1O 30842,C1(CNC(C(CC)OCC)=O)CC(NC(=O)Cc2cscn2)C(O)C1 30843,C=CC1(CO)CCN(C(=O)C(C)(CSC)NC(=O)COc2cccnc2)CC1 30844,Cn1cc(CC(O)C(=O)NCC2(CNC(=O)C=CC=C(Cl)Cl)CC2)cn1 30845,C1(C(=O)NCCC(CC)C)CC12CC(NC(c1cnccc1C)=O)C2 30846,c1(C(=O)NC(C2CCN(C(=O)C(F)=C3CCC3)CC2)C)ccc(N)cc1[N+](=O)[O-] 30847,c1nnn2c1CN(c1nc(N3CCN(C4CCC4)CC3)nc(C3CC3)n1)CC2 30848,C(=O)(N=c1nc2ncc(Cl)cn2[nH]1)Nc1ncc(C(C)(C)C)o1 30849,n1(CC)nc(C)c(CC(=O)NCC2CN(C(=O)CCCC(C)C)CC2C)c1C 30850,N1(CCCC=C)CCC2C(CCCN2C(=O)C(c2cnn(C)c2)C)C1 30851,Cn1c(=O)oc2c(C(=O)NCC(CNC(c3ccnc(O)c3)=O)CO)cccc12 30852,OCC1CN(CC2CC3(CCC(F)(F)CC3)C2)Cc2ccccc21 30853,N1(C(CC2(C=C)CCC2)=O)CC(NC(=O)C(C)NS(C)(=O)=O)CC(C)(C)C1 30854,N1(C(C(COCC)C)=O)CC2(CCN(C(=O)C(C)(C)c3cccs3)CC2)CC1C 30855,c1(C(N(C(CNC(c2cc(CC)c(CC)o2)=O)C)C)=O)ccn2cncc2c1 30856,N1(CC2CC2)CCC(c2n[nH]cc2CN(C(=O)C(C)C(C)C)c2c(C)cns2)CC1 30857,c1(CCC(N2C(CN(C(=O)C(=Cc3c[nH]cn3)F)C)CCC2)=O)cccc(F)c1 30858,N1(C(c2cn(CCC=C)nn2)=O)CCC(O)(C(C)NC(C2CCC(=O)N2C)=O)C1 30859,C1(NC(CCNC(C)=O)=O)COC2(CCN(C(C3(F)CC=CC3)=O)C2)C1 30860,N1(CCC)CCCN(C(C2CSCCN2Cc2ncccc2C)=O)CC1 30861,S(=O)(=O)(C(F)(F)F)N1CC2C(C(N3CCOC(C4CCC4)C3)=O)C2C1 30862,N1(C(CC(C)n2ccnc2)=O)CCC2(CC1)CC2NC(C1(C(F)(F)F)CC1)=O 30863,c1(C(N2CC(O)(CNC(C3(C)C(CC)CCC3)=O)C2)=O)ccc2oc(=N)[nH]c2c1 30864,C12(NC(Cc3cc(CC)no3)=O)CCCCCC1N(C(c1nnsc1N)=O)CC2 30865,CC#CCCC(=O)N1CCC(C(N2CCC(N3CCCC3)C2)=O)O1 30866,N1(C(=O)CCN(C(c2ccco2)=O)C2CC2)CC2(CCC2O)C1 30867,n1(CC(=C)C)nnnc1C(c1csnc1OC)NCCn1cccn1 30868,CCCCCCC(=O)N1CCC2(NC(=O)Cc3c(OC)cccc3OC)CC2C1 30869,c1(-c2ccccn2)cc(-c2noc(C3CCC(=O)O3)n2)ncn1 30870,C(=O)(CCS(N)(=O)=O)NCC(C(C)(C)C)NC(CCC(C)SC)=O 30871,c1(CC(C(=O)N(CCNC(=O)Cc2cc(C)[nH]n2)CC)O)ccccc1Cl 30872,C(C(=O)NC(C)CCOC)(C(C)C)NC(CCOCCC)=O 30873,C1(C(N2CCCC(NC(=O)CN3C(=O)CCC3=O)C2)=O)COc2ccccc2O1 30874,C1(C(C#C)NC(=O)N(CCCN(C)C)C)CC(F)(F)C1 30875,S(=O)(=O)(c1cc(F)c(OC)cc1C(C)C)NC(c1c(OCC)scc1)=O 30876,C1(CNC(c2c(CC)ccs2)=O)CCCCC1NC(c1cc(OC)n(C)n1)=O 30877,c1(N2CCC(Nc3c(C(=O)OC)c(C)sc3)C2=O)cc2ccccc2o1 30878,Cc1ccn(C)c1C(=O)NCC1CCCN(C(C2CCC(=O)N2C)=O)C1 30879,N1(C(c2ccnnc2S)=O)CCCS(=O)(=O)CC1c1cccc(C(F)(F)F)c1 30880,C(=O)(C(O)C(C(C)C)OC)NCCC(CNC(C(F)=CCC)=O)(C)C 30881,c1(CN2CCC(CNC(CSCC)=O)C2c2cccnc2)cc(Cl)c(F)c(Cl)c1 30882,c1(OC)ccc2c(c1)C(C(=O)NCC1C(NC(c3ccoc3C3CC3)=O)C1)CC2 30883,C1(C(=O)NCCC2(O)CCN(C(CS(=O)(=O)NC)=O)CC2)CCC12CCOCC2 30884,N1(C(c2cn(CCCOC)nc2)=O)CC(NC(c2ccoc2Br)=O)C(O)C1 30885,c1(C(=O)NC2C(C)CN(C(c3nn(C)cc3Cl)=O)CC2)cc2c(cc1O)OCO2 30886,N1(C(C(C#C)(C)C)=O)CC2CC(NC(c3cnccc3C(F)F)=O)C(C2)C1 30887,c1(NC(C(COCC)NC(=O)CC2CC2(C)C)=O)ccn2nccc2c1 30888,c1(C(=O)NCCCCCCNC(C2N(CC)CCC2)=O)c(C)ccc(C)c1N 30889,C1(C(=O)NC(C2(C(N3CCC3CC(N)=O)=O)CC2)C)CC=CC(O)C1 30890,C12(CNC(=O)C=C(Cl)Cl)CCC(CC1)CN2C(c1cc(C(F)(F)F)cc(O)c1)=O 30891,CC1CCN(C(C2(C(F)F)CC2)=O)CCN1c1ncc(I)cn1 30892,Cc1nn(-c2cccc(F)c2)cc1C(N1CCCC(NCC(F)F)C1)=O 30893,c1(C(=O)NC2CC(C)N(C(=O)C3=CCOCC3)C2)c[nH]c(=N)nc1O 30894,Cc1cnncc1C(N1CCC(N2CCC(NC(=O)C3=CCOC3)C2)CC1)=O 30895,N1(C(C(C)OCCCCCC)=O)CC(NC(c2ccnnc2C)=O)CC(C)(C)C1 30896,N1(C(C=CCC)=O)CC(O)(C2(CNC(c3c(C)cc(F)cc3Br)=O)CC2)C1 30897,C1(CNC(C(CN(C)C)(F)F)=O)CC2CCC1N2C(C1(C2CCCO2)CCC1)=O 30898,CCCCCC(O)C(=O)NCC1CN(C(c2cnc(NC)cn2)=O)CC12CCC2 30899,n1(CCOC)ccc(C(=O)N(CCCNC(=O)Cc2nonc2C)CCOC)n1 30900,C1(CNC(C(CC)=CCCC)=O)CN(C(=O)COC)CCN1C 30901,N1(C(C(C)CC(C)(F)F)=O)CCOC2(C1)CN(C(=O)CCCC1CCOCC1)C2 30902,C=CCCC(CO)NC(=O)C(O)C1CN(C(c2cn(C3CC3)nn2)=O)C1 30903,c1(NC(C2(C)CCN2C(c2ccc3nc[nH]c3c2)=O)=O)ccc(Cl)c(C#N)c1Cl 30904,n1(C(C)C(N2CCC(F)(CNC(=O)CCNC(N)=O)C2)=O)cc2ccccc2n1 30905,C(c1ccncc1)=C(C(=O)NC(CCN(C(C(CC)F)=O)C)C)C 30906,c1(CNC(c2ccc(-c3ccc(SC(C)C)cc3)cn2)=O)c(O)ccc(F)c1F 30907,C(=O)(C(CO)NC(c1[nH]ccc1C)=O)OC.C12CC(C1)NC2=O 30908,C1(NC(C)=O)CCN(C(=NCC2CCCN2Cc2cccs2)NC2CCC2)C1 30909,c1(C(C(C(=O)NCCC2(C)COC2)N)=O)ccc(F)cc1F 30910,c1(OC)cc(C)c(Br)cc1C(N1CCC2(CC2C(=O)Nc2cc(O)ncn2)C1)=O 30911,N1(C(CC2CC(=C)C2)=O)CCN(C)CC1C(=O)NCC(CC(C)C)N(C)C 30912,CON(CCC(=O)NC1C2CCCCCC12)C(=O)C1CC(C#N)(OC)C1 30913,C12(CC(=O)N(C(CC#C)C)C)CCC1CN(C(=O)CC1CC3(CCC3)C1)C2 30914,N1(C(C2C(CC)CCC2)=O)CCC(CCOC)(C(=O)N(C2CCC2)C)CC1 30915,c1(-c2cncc(COCC)c2)ccn2nc(C(=O)Nc3nc(C#N)cs3)cc2c1 30916,C=C1CCN(C(C2CC(C)CN2C(=O)CC(C)c2ccco2)=O)CC1 30917,Cc1nc2c(s1)CCCC2C(=O)NC1CCN(C(c2c[nH]c3cccnc23)=O)C1 30918,c1(C(=O)NCC(CC)NC(=O)CCC2CCN(C)CC2)oc(C)cc1C 30919,C1(C(=O)NCCC(CN=[N+]=[N-])F)CC12CCOc1ccc(F)cc12 30920,N1(c2cc(NCC3(CCO)CN(C)C3)ncn2)CCCC2(CCCCCC2)C1 30921,C(CCC1CCC1)(C(=O)NCc1cnn(C)c1O)NC(c1c(C)ocn1)=O 30922,c1(C(=O)NC2C(NC(=O)CC3CCCCC3(F)F)CCC2)ccc2nnnn2c1 30923,c1(C(=O)NC2CC(N(C(CCC(=O)NC)=O)C)C2)cc(N)nc(Br)c1 30924,C(C(=O)N(CC)OC)NC(C(CNC(C1(CC#C)CC1)=O)C)=O 30925,N1(C(c2c(C)nsc2N)=O)CC(C2CN(C(=O)CCC3CCCOC3)C2)C1 30926,N1(C(C2CNC(=O)N2)=O)CCCC2(CCN(C(c3cocc3C(N)=O)=O)C2)C1 30927,C(=O)(C1CCc2cccc(F)c21)NC(CC)CNC(=O)Cn1ccc(=O)cc1C 30928,C=CC1(C(=O)NCC23CCCC(CO2)C3)CCN(C(=O)Cc2ccccn2)C1 30929,CCC(C)CCCCC(=O)NCC(CC)N(C(=O)Cn1cc(C)cn1)C 30930,N1(C(c2ccn(CCC)n2)=O)CC2CCC(C1)N2C(c1cnc(C2CC2)s1)=O 30931,c1(C(=O)NC2CCC(CCNC(C(C(C)C)C)=O)C2)nn(C)c(Cl)c1Br 30932,N1(C(C(CC)OCC)=O)CC(OC)CC(NC(C2CC(C)CC2)=O)C1.OCC 30933,C(=O)(C(COC)COC)NCC1(C(=O)NCC2C(CC)C2)CCC1 30934,C(=O)(C(CC(C)C)NC(c1nc(N2CCCC(N(C)C)C2)ncc1Cl)=O)NC 30935,C1(CN(C(=O)CN(C)C(C2(C)COCCO2)=O)C)CCCCCC1 30936,c1(C(=O)NCC(C2CCCCC2)NC(C(C(C)C)F)=O)csc([N+](=O)[O-])c1 30937,C(C(=O)N(C)CCN(C)CCO)(C(C)(C)O)NC(C(CC)C#N)=O 30938,N(C(=NCCN1CC=C(C)CC1)N1CCC(C(O)C(F)(F)F)C1)CC(=C)C 30939,C1(NC(COCCN(C)C)=O)CN(C(C2CCCC23CC3)=O)CC12CCOCC2 30940,N1(C(c2cccc(OCC#N)c2)C(=O)NC)CCOc2cccc(Br)c2C1 30941,C(=O)(C(C)(CC)CC)NC(CNC(Cc1c(SCC)cccc1)=O)CCOC 30942,c1(NC2CCC(C(=O)Nc3cnc(C)nc3Cl)CC2)nccc(S(C)(=O)=O)n1 30943,c1(N2CC(C)C(NC(c3cnsn3)=O)C2)ncc([N+](=O)[O-])cc1Cl 30944,c1(CNC(=O)NCC2C(c3n(C)ccn3)OCC2)cccc2c1SCCC2 30945,N1(CC)CCCC1(C(=O)NCc1cc(CO)[nH]n1)C(C)C.C12CCC1C(=O)NC2 30946,c1(N(C(=O)CCc2nc[nH]n2)C)ccc(Br)cc1CC#N 30947,N1(C(C(CC)c2ccccc2)=O)CCN(C(c2n[nH]c(C)c2F)=O)C2(CCC2)C1 30948,N1(C(C2CC(CC)C2)=O)CCc2cc(NS(=O)(=O)c3cccc(Cl)n3)ccc2C1 30949,CC1CCC(NC(c2c[nH]ccc2=N)=O)CN1C(c1csc(-c2nc[nH]n2)n1)=O 30950,C1(C(N(CCNC(C(CC)(C)O)=O)C)=O)CCC(=O)N(C(C)C)C1 30951,CC1CN(C(=O)Cn2cc(C34COC(C3)C(O)C4)nn2)C(C)C1C 30952,c1(C(N2CCC(NC(Cc3c(C)con3)=O)(CF)C2)=O)c(C)cccc1[N+](=O)[O-] 30953,C(=O)(C1CCCc2nn[nH]c21)N1C(C)CC2CN(C(c3c(C)coc3C)=O)CC21 30954,N1(C(CCCC(C)=O)=O)CC2CCCN(C(C3OCCN(C)C3=O)=O)C2C1 30955,N1(C(c2c(OC)nsc2)=O)CC(CC(=O)NCC2CC2C(C)C)C2(CC2)C1 30956,c1(CC)cc(C(=O)NCCCCCNC(=O)C(CC)n2nccc2C)c(C)nn1 30957,C1(NC(C=C(C)C)=O)CCN(C)C12CCCN(C(C1CCCN1C1CC1)=O)C2 30958,c1(C(=O)NC2CN(C(c3cc(OC)cc(F)c3)=O)CC2F)cc(Cl)c(F)cc1F 30959,n1(CC)cc(C(=O)NCC2CCC(NC(C3CNC(=O)N3)=O)C2)c2ccccc12 30960,N1(C(C(CC#C)C)=O)CCc2ccccc2C(NC(=O)C(C)(C)C(F)F)C1 30961,N1(C(c2c(CC)nccc2)=O)CC2(CCN(C(C3CCN3CC)=O)CC2)C1 30962,c1(NC(CNC(c2c(C)cccn2)=O)C(C)C)ncc(C#N)cc1Br 30963,C(=O)(CCN(OC)C(=O)CC1CNC(=O)O1)NC(CCCC)CCC 30964,c1(OC)cc(C(=O)NCC2CCCCN2C(c2nccnc2Br)=O)ccc1O 30965,C1(C)(CNC(C2(N(C(C(CN(C)C)O)=O)C)CC2)=O)CC2(CC2)C1 30966,C(CC(=O)OCC(C)(C)C)N(CCCNC(=O)OC(C)(C)C)C(=O)Cc1cccs1 30967,Cc1ccc(F)c(NC(=O)CCc2ccc(NC(c3cc(C)cc(Cl)c3)=O)[nH]2)c1 30968,N1(C(CN(C)CC)=O)CCC2C(CCCN2C(c2cc3nc[nH]c3cn2)=O)C1 30969,N1(C(C(C2CCCC2)OCC)=O)C2CCC1CN(c1ccnc(C)n1)CC2 30970,c1(C(=O)NCCCCNC(C(c2nc(F)ccc2Cl)C)=O)c(F)ccc(F)c1N 30971,C1(C(N2CCC(C(C)(C)NC(CCSCC)=O)C2)=O)COc2cc(Cl)ccc2C1 30972,C1(CNC(C=CCCC)=O)CCCC1NC(c1snnc1CC)=O 30973,N1(C(C(C)(C)C2CCC2)=O)CCC(NC(=O)CC=CC(=O)O)CC1 30974,CCC(CC(=O)NC(CCN(C(=O)C(C)Cc1ccccc1C)C)C(C)C)SC 30975,c1(C(N2CCCC(NC(COCCOCC)=O)C2)=O)ccc(O)cc1C 30976,c1(SC)cccc(C(=O)NC2(C)CCN(C(=O)C(C)(C)CC(F)F)C2)c1[N+](=O)[O-] 30977,N1(C(=O)CCC2CCC2)CCC2(CC1)CC2CNC(C1(CCF)CC1)=O 30978,CC1(C)CC(CNC(c2cncc(Cl)n2)=O)N(C(=O)CCC2COC(C)(C)O2)C1 30979,c1(C(=O)NC(C2CCCCN2C(=O)Cc2cocn2)C)nn(C)c2c1COCC2 30980,C(=O)(C(C)(F)C(=O)NC1CC(CNC(c2cc(Cl)cc(Cl)c2)=O)C1)OC 30981,N1(C(CNC=O)=O)CCN(C(C2CCCC23CCC3)=O)C2CCC12 30982,C(C1=CCN(C(C2CCC3CC3C2)=O)CC1)NC(c1ccnn1CC1CCC1)=O 30983,C1(NC(c2ccsc2Cl)=O)CN(C(=O)C(F)=CC2CC2)CC12CCOCC2 30984,N1(C(=O)COCCF)CCN(C(C23CCCC2C3)=O)C2(CC2)C1 30985,C1(NC(COc2cccc(CC)c2)=O)CC(NC(=O)CNS(N)(=O)=O)C12CCC2 30986,c1(C(N2C3(CNC(CC(CC)O)=O)CC(C2)C3)=O)cc2cc(C)cc(C)c2[nH]1 30987,C(CS(=O)(=O)CC(=O)NC1CC1CNC(c1nc(C)c(C)nc1C)=O)OC 30988,N1(C(C(C)(C)OC)=O)CCC(NC(=O)CCc2cocn2)C2(CCC2)C1 30989,c1(C(=O)NC2C(NC(C(CC(C)C)NC(C)=O)=O)CC2)cc2ncccc2s1 30990,Cc1ccc(F)c(C(=O)NC(C2CCN(C(=O)CC3NC(=O)NC3=O)CC2)C)n1 30991,N1(C(c2cc(C)cc(F)c2)=O)CC(C)CN(C(C2COC3COCC23)=O)CC1C 30992,CC1CCCCCC1NC(=O)C=CC1CCCN1C(=O)C=Cc1cc[nH]c1 30993,N1(C(C(CC=CC)NC(=O)C=CC(C)(C)SC)=O)CCC2(C=CCO2)CC1 30994,C=C(CNC(c1cc(C)c(I)s1)=O)c1ccc(C)c([N+](=O)[O-])c1 30995,C12(CC(=O)NCCNC(c3c(CCC)onc3C)=O)CC3CC(CC(C3)C1)C2 30996,Cc1ccc(C(=O)NC(C)(C)CNC(=O)CC2CC(O)C2(C)C)c(F)c1Br 30997,CC1CC(NC2CN(Cc3ccccc3)CCC2O)C(=O)N1c1ccccc1 30998,C#Cc1cc(C(=O)NCC2CN(C(=O)Cc3sc(C)cc3C)C2)cc(N)c1 30999,C(=O)(C(C)(CC)CC#C)NC12CCC(C(=O)NCCSCC#C)(CC1)C2 31000,c1(SC)ncc(C(=O)NCCOC2CCN(C(C3C4COCC34)=O)C2)n1C 31001,c1(C(N(CC=CC(=O)N(C2(COC)CC2)C)C)=O)ccc([N+](=O)[O-])o1 31002,C(C)(C)(C(=O)NCCC(C)(C)NC(=O)C(C)Sc1nnnn1C1CC1)OC(C)=O 31003,c1(C(N2CC(C)C(NC(=O)C(c3ccc(F)c(F)c3)O)C2)=O)nc(Cl)ccc1N 31004,O=C(C1CCCc2nccn21)NCCNC(=O)CC12CNC(=O)C(C1)C2 31005,c1(C(N2CCC(C(=O)OCC)CC2)=O)c[nH]ccc1=N.C1CC1Cl 31006,N1(C(C(CC=C)N(C)C)=O)CCC(C2CC2)C1CNC(=O)Cc1ccc(F)cc1 31007,c1(C(=O)NC2C(NC(C(CC)(C)O)=O)C2)c(SC)cccc1F 31008,c1(C(N2CC3(CCN(C(C4C(OC)C4)=O)C3)C2)=O)cc2n(n1)CC(C)NC2=O 31009,CC1CN(C(C2C3(CC3)C23CC3)=O)CC2(CCN(C(=O)CC3OCCO3)C2)O1 31010,N1(C(CSCC#C)=O)CCC2(CC1)CN(C(=O)Cc1nonc1C)C2 31011,C12(C(N3CCCC(CNC)C3)=O)CCC(C(F)(F)F)(C1)OC2 31012,C12(CNC(=O)CC3CCN(C(C4CC(O)C(F)C4)=O)C3)CCC(CC1)C2 31013,N1(C(C2CC(=O)C2)=O)CCC2(C=C(C(=O)NOCC(F)(F)F)C2)C1 31014,CCCC(C)=CC(=O)NC(C(=O)NCC(O)COCC)C1CCC1 31015,c1(OC)nc(=NCC(C)(C(C)C)NC(=O)C(=O)Nc2ncc[nH]2)[nH]c2[nH]cnc12 31016,C1(NC(C2(Br)C(C)(C)C2)=O)CCCN(C(c2ccc(F)o2)=O)CC1 31017,c1(C(=O)NCCCC(CO)NC(CCc2cnc(C)s2)=O)cccc2nccn12 31018,Cc1cc(C(=O)NCC(C)NC(=O)COc2cccc(O)c2)ccc1F 31019,C(CCCCCCC)NC(C=CC(=O)NC1C(CNC(CC(C=C)C)=O)C1)=O 31020,c1(CNC(C(c2cnccn2)C)=O)ocnc1-c1cn(C(c2nncs2)C)nn1 31021,C(=O)(C(=O)CCC(C)C)NC1CCN(CC(=O)Nc2c(SC)cc(C)cc2)C1 31022,N1(C(c2cc(CC)on2)=O)CC(NC(c2coc(Cl)n2)=O)Cc2ccccc21 31023,N1(C(c2cnc(OCC)s2)=O)CC(C)CN(C(c2oc(C)nc2C)=O)C(C)C1 31024,c1(CCNC(=O)C(=O)NCC2(F)CC3(CNC3)C2)ccc(Br)cc1Cl 31025,N1(C(CC(C)SC)=O)CCCCC1C(=O)NCCCC1CC1 31026,CC1(C)CC(NC(=O)COCCF)CN1C(=O)Cc1nc[nH]n1 31027,C(c1cc(C(F)(F)F)ccc1Cl)=CC(N1CC(CNC(=O)CCF)OCCC1)=O 31028,C#Cc1cc(C(=O)NC2(CNC(=O)C(F)(CC)C(=O)OCC)CCC2)ccc1Cl 31029,CC12CCN(C(c3c(O)cc(Cl)cc3Cl)=O)CC1C2(F)F 31030,C1(N(C(C(C2CCN(C(C3CC(=C)C3)=O)C2)F)=O)C)CCCCC1(C)O 31031,n1(CCCC)nc(C(=O)NCC2(F)CC(NC(=O)C(F)=CCCF)C2)ccc1=O 31032,C1(C(N(C2CC(C#N)C2)CC(=O)NCCc2c(C)ocn2)=O)CC(=O)NC(C)C1 31033,Cc1cc2[nH]c(=O)c(C(=O)NCCC3CN(C(C4(Cl)CC4)=O)CC3C)cn2n1 31034,Cn1c(C2CC2)nn(CC(=O)NC2CC2CNC(=O)Cn2cnnc2O)c1=O 31035,N1(C(c2cccc(CCC)c2)=O)CCCC(F)(C(=O)NCc2cnsc2)C1 31036,O(NC(=O)C(F)(CNC(=O)CCC(N)=O)C(C)C)CC(C(C)C)O 31037,C(C(=O)N=c1cc(C)o[nH]1)CC(=O)NC(CNC(c1ccc(=NC)[nH]c1)=O)CO 31038,N1(C(CC(C)OC)=O)CC(CNC(=O)CCc2cncc(Br)c2)C(C)C1 31039,CCCC(C(O)c1ccccc1)NC(c1sccc1Cl)COC 31040,C(C(C(=O)N1CC(C)(CSC)C1)C(C)(C)C)NC(C=CC(CC)C)=O 31041,C1(C)(C(N2CCN(CCCNC(c3c(C)ncnc3)=O)CC2)=O)CCCCC1C 31042,CC(C(=O)N(CCNC(c1cnsc1)=O)CC1CC1)NC(c1ccco1)=O 31043,Cc1ccc(S(=O)(=O)NC2CN(C(c3cccc(C)c3Cl)=O)CC2F)c(F)c1 31044,c1(C2C(C(N(CCc3cc(OCC)ncc3)C)=O)C2)cc(C)cc(Br)c1 31045,CCCC(C)CCCC(=O)NC(CNC(c1ncc(OC)cn1)=O)C(C)(C)C 31046,S(=O)(=O)(CCC(=O)NC1CCC(CNC(=O)COC2CCCOC2)C1)N(C)C 31047,C1(C)(C(=O)OC)CC(CC(=O)OCC(=O)N(c2ccc(OC)cc2)C(C)C)CC1 31048,N1(C(C#C)=O)CCCC(C(=O)Nc2c(C(N)=O)cccc2C)CC1 31049,N1(C(c2c(C)nn(C)c2Cl)=O)CC2(CCN(C(=O)CCc3cncc(O)c3)C2)C1 31050,C1(CSC)COCCN1C(=O)C(n1cc(COC(=N)O)nn1)C 31051,c1(C(N(C2CCCN(C(=O)C(C)=C3CC3)CC2)CC)=O)ncc(OC)cc1F 31052,O=C(N=c1c(Cl)c[nH]cc1I)C1CC12CCN(C(c1ccccc1I)=O)CC2 31053,N1(C(C2(COC)CC2)=O)CCCC(O)(CNC(C23CCCC2C3)=O)CC1 31054,CC(CC(=O)N1CCN(C(=O)CCc2ccc[nH]2)C(CCO)C1)C(F)(F)F 31055,c1(C(N2CCOC(CCOC)C2)C(=O)NCCC(=O)OCC)cc(C)nc(C)n1 31056,CC1C(NC(c2cc(F)ccc2F)=O)CCCN1Cc1cnon1 31057,N1(C(c2nc(C#C)sc2)=O)CCCN(C(c2cccc(=O)n2C)=O)C(C)C1 31058,c1(C(N2C(CN(C(C(C)OCCC(C)C)=O)C)CCC2)=O)ccccc1C(C)O 31059,C(=O)(CCCC(=O)N1CCC(C(C)NC(c2ncoc2C)=O)C1)NCCC 31060,N1(C(c2c(C(C)C)occ2)=O)CCCC(NC(C23CCC(O)C2CC3)=O)CC1 31061,c1(C(N(CC(CC)NC(c2cc(OC)ccc2O)=O)C)=O)cnn2cnnc2c1 31062,N1(C(C2(OC)CCSC2)=O)CC(OC)CC(NC(=O)CSCCN(C)CCO)C1 31063,C123CCC(CC1)(C2)n1cc(nn1)N3.Cc1nnn(CC(N2CC(SC(F)F)C2)=O)n1 31064,c1(OC)c(C(N2CC(CO)(NC(c3ccc(=O)oc3)=O)C2)=O)cnn1C 31065,Cc1c(C(=O)NC2(CNC(C3CC4(C3)CC4(F)F)=O)CCCCC2)cncc1F 31066,n1(CC(=O)NC)ccc2ccc(NC(=O)C(N3CCC(CCF)(CO)C3)=O)cc12 31067,n1(CC(=O)N(C(C)CNC(C2CSC2)=O)C)cc(C2CC2)nn1 31068,CN1CCN(C(=O)CC(C)(C)C(C)(F)F)CCN(C)CCC1 31069,N1(C(CCC2C(C)C2)=O)CCCC1CCc1cccs1 31070,C(CN=c1ccc(S(=O)(=O)NC2CCCCC2O)c[nH]1)SCC(C)C 31071,CC1(C)CCN(C(C2CC2(C)C)=O)C(C(=O)Nc2ccc(F)c(O)c2)C1 31072,c1(CC(=O)N(CCCNC(CC2C(CC)C2)=O)CC)ccc(OC)c([N+](=O)[O-])c1 31073,C1(N(C(CCC2CC(NC(CCOCCC)=O)C2)=O)C)CCSCC1 31074,c1(C(=O)NC(CC=C)C(=O)N(C2CC(O)C2)C)ncc(C)cc1C 31075,CC(CCCNC(C1(C2CCCO2)CCCC1)=O)NC(c1ccon1)=O 31076,CC1CN(C(c2sccc2F)=O)CC(C)CN1C(c1cnn(C)c1C(F)(F)F)=O 31077,C1(C(N(CCCNC(C(C)NC(CC)=O)=O)C)=O)CC(OC)C(OC)C1 31078,N1(C(Cn2ncc(C#C)c2)=O)CCCC(COC)(NC(=O)CSCCC#N)C1 31079,C(=O)(C(O)CC(N)=O)N(CC(N1CCCC(CC=CC)C1)=O)CC 31080,C1(NC(CNC(CC(C)C)=O)=O)CCC(C)N(C(=O)C=C2CCOCC2)C1 31081,C1(CNC(c2n(C(C)(C)C)ncc2)=O)CCCC(NC(C2C3CCCC23)=O)C1 31082,C1(CNC(C(COC)O)=O)CCN(C(C2CC(c3cccc(F)c3)C2)=O)C1(C)C 31083,N1(C(C2CCN(C(c3c(OC)ccs3)=O)C2)=O)CCc2c(O)noc2C1 31084,c1(C(=O)NC(C(=O)NC(CN(C(CCOC(C)C)=O)C)C)C)ccccc1Cl 31085,C(=O)(C1CCc2c(Cl)cccc21)NCC1CCC(C)(C)CN1C(C1(CO)CC1)=O 31086,CC1=NOC(=O)C1CC(N1CCOC(CCCNC(C2CS(=O)(=O)C2)=O)C1)=O 31087,c1(C(=O)OC)ccc(CNC(=O)C(N2CCN(c3ncc(C)s3)CC2)=O)cc1C 31088,Cc1ccc2c(C(=O)NC3(CCNC(=O)CC(C)P(C)(C)=O)CC3)onc2c1 31089,N1(C(=O)CCc2ccon2)CCC2CN(C(=O)CCc3ccc(CO)cc3)C2C1 31090,C(C)(C(=O)NCC(C)N(C(=O)CNS(=O)(=O)N(C)C)C)(C(C)C)OC 31091,N1(C(CNC(C)=O)=O)CCC(C)(C(=O)NCCc2cccc(OCF)c2)C1 31092,c1(CNC2CCCN(S(C(C)C(F)F)(=O)=O)C2)cnc(N)c([N+](=O)[O-])c1 31093,C#CCC(C)(C(=O)NC1CN(C)CC1O)NC(C1CCCCN1C)=O 31094,C1(C)(C(=O)NCC(N(C(Cc2nc(CC)sc2)=O)C)C2CC2)COC(=O)C1 31095,Cc1ccc(N)c(C(N2CCCC2C(C)NC(=O)Cc2cccnc2)=O)c1 31096,C1(CCC(=O)NC)CN(C(=O)N(C)CCOCCOC)CCC1C 31097,n1(CCOC)ncc(C(=O)NC2(COC)CN(C(C3(C)CCSCC3)=O)C2)c1C 31098,c1(C(=O)NCc2scc(CNC(c3cc(C)ns3)=O)n2)cc(O)nc(C2CC2)n1 31099,CC(C)C(O)C(C)C(=O)NCC1(F)CN(C(c2ncn3c2CCC3)=O)C1 31100,c1(C(N(CC(C)NC(C(C2CC(F)(F)C2)OC)=O)C)=O)coc(C#N)c1 31101,c1(C(C(=O)OCC)=O)c[nH]c(=NCC(C)N(C)C(C2CCC(C)C2)=O)c(C)c1 31102,c1(C2C(CC(=O)NC(CO)C3CC3)(C(F)(F)F)C2)ccccc1C1CCC1 31103,c1(CCC(=O)NC(CN(C)C(c2ccc(Cl)s2)=O)(C)C)ncc(F)cn1 31104,c1(OC)ccc(C(N2CCCC(NC(=O)C(F)(F)C(F)F)C2C)=O)c(N)c1F 31105,N1(C(Cc2ccc(OC)cc2F)=O)CCN(C(C2(C)CCOC2)=O)CC2(CC2)C1 31106,c1(C(N(C2CCCC(NC(CCCC#CC)=O)C2)C)=O)cc(C)[nH]c(=NC)n1 31107,c1(C(CC)NC(=O)N(CCO)CCCS(C)(=O)=O)ccc(OC)c(F)c1 31108,C(=O)(C1CCc2nccn21)N1CCN(C(CCC2C(C)C2)=O)CC1CO 31109,c1(C(N2CCC(CNC(=O)C(c3ccc(F)cc3)F)C2)=O)ccc2c(c1)CCN2 31110,CC1=C(C(=O)N2CCCC2CCNC(c2ccc(F)c(F)c2F)=O)CCS1(=O)=O 31111,CC(CNC(C1CC1(C)C(F)F)=O)C(F)C(=O)NCC1CSC1 31112,C#Cc1ccc(C(=O)NC2(C(N3CCC(CO)C3(C)C)=O)CC(O)C2)nc1 31113,N1(C(CC2(OCC)CC2)=O)CC(C(=O)NC2COCC2F)C2(CCC2)C1 31114,c1(N2C(C(N3CCCC(C(=O)OC)C3)=O)CC3CC32)ncnc2c(Br)c[nH]c12 31115,C1(C)(C(NOC2CCCN(CC)C2)=O)CC(O)CN1C(=O)C=C(C)C(F)F 31116,C1(CNC(C2C(CCC)C2)=O)(CO)CC12CCN(C(c1cnnn1C)=O)CC2 31117,CC1(C)CC(NC(C2CC3CCC2CC3)=O)CN1C(C1CC(CCO)C1)=O 31118,c1(C(N2CC(N3CCN(C)CC3)C2)=O)ccc(F)c(C(=O)OC(C)(C)C)c1 31119,[N-]=[N+]=NC1CN(C(c2ccc3cc[nH]c3c2)=O)CC1NC(C1CC2CCC2C1)=O 31120,C1(C)(C(N2CC(N(C(c3c(SC)cn(C)n3)=O)C)C2)=O)CCCS1(=O)=O 31121,N1(C(C2(C#N)CCCO2)=O)CCC(C2CC2)(NC(c2cc(F)cnc2O)=O)C1 31122,N1(C2CN(C(C=CC(=O)N(C)C)=O)C2)CCN(C(C23CCCCC2C3)=O)CC1 31123,C(=O)(CCC(C)(C)F)N1CCCC(CN(C(c2nncn2C2CC2)=O)CC)C1 31124,C(CN=c1[nH]c(=NCCc2c[nH]c(=N)s2)[nH]c2cc(C)ccc12)C=NCOCC 31125,C=CC(CC)CC(=O)NCC1CN(C(C2CC3(CCC3)CO2)=O)CCN1C 31126,c1(C(=O)NC(C2CCN(C(C3(F)CC3C)=O)C2)C)ccnc(N2CCC2)c1 31127,C(C1(C)OCCc2ccccc21)NS(c1c(CC(=O)OC)cc(Br)c(F)c1)(=O)=O 31128,C1(C)(CNC(CSCC#C)=O)CN(C(c2cccc(O)c2C)=O)C(C)(C)C1 31129,C1(NC(=O)C2=COCCC2)CCN(c2ncc(Br)c(O)n2)CC12CCC2 31130,N1(C(C(C)c2cccs2)=O)CCCC(CCNC(=O)COc2ccccc2)C1 31131,N1(C(Cc2n(C)cnn2)=O)CC2CC(NC(c3cc(Br)co3)=O)CC1C2 31132,N1(C(C2C(C)(Br)C2)=O)CCC2(CCN(C(c3cn(CC4CC4)nn3)=O)C2)C1 31133,Cc1nc(C(=O)NC2C3CN(C(=O)C=CC4CCC4)CC23)c(=O)[nH]c1C 31134,c1(C(=O)NC2CCCN(C(C(=Cc3ccco3)C)=O)C2)c(N)cc(F)cc1Cl 31135,C1(C(=O)OC)CCCC1C(=O)N(CCCN(C)C(C1CCSC1)=O)C 31136,C(=O)(CS(=O)(=O)CC(C)C)NC1CC2CC(NC(C(C(=C)C)(C)C)=O)CC2C1 31137,c1(C(=O)NC(CC)(C)CNC(C2(C)CCOCC2)=O)nc2ccccc2cc1C 31138,Cc1cc(C)c(NCC(N2CC(CNC(=O)CCC3CNC(=O)N3)C2)=O)c(C)c1 31139,C1(C(=O)Nc2cc(Cl)ccc2Br)COC2(CCN(Cc3ccc(Br)cn3)CC2)C1 31140,c1(C(=O)NC2(COC)CN(C(C3CCC(CN(C)C)O3)=O)C2)c(Cl)nn(C)c1Cl 31141,C1(NC(c2cc(OC)n[nH]2)=O)CC2CCC(C1)N2C(C1CCCC1C(C)C)=O 31142,N1(C(c2nc(CC)sc2)=O)CC2(C1)CN(C(C1CC1C(C)C)=O)C2 31143,C1(NC(C(C)(C)C2CC2)=O)CN(C(C2CCC3(C2)N=N3)=O)CCC12CCC2 31144,CCCCCC(O)CC(=O)N1CCC(NC(c2c(Cl)ccc(F)c2F)=O)C(F)C1 31145,c1(C(C(=O)NCC2(C(=O)NC(c3cccs3)C)CC2)C)ccccc1 31146,C1(C(=O)OC)(C(C)C)CCN(C(C2(c3ccc(C)cc3)CC2)=O)C1(N)C 31147,C(C(F)(F)CCC(=O)NNC(=O)c1cnccn1)n1cc(C(COC)(C)O)nn1 31148,c1(C(N2CC(CN(C(CCOCC)=O)C)C2)=O)nc(COC)n[nH]1 31149,C12(CNC(=O)Cc3cc[nH]c3)CCCCC1CN(C(c1ccc(O)nc1Cl)=O)C2 31150,N1(C(CC=C)=O)CCCCC1CN(C)C(C1(n2cccn2)CCOCC1)=O 31151,C1(CNC(c2n[nH]c(C)c2C)=O)CN(C(C2CS(=O)(=O)C2)=O)CC1(F)CO 31152,C1(F)(C(N(CCCNC(c2ccc(COC)s2)=O)C2CC2)=O)C2CCCCC12 31153,c1(NC(C)C)ccc(NC(=O)C(=O)NCC2CNC(=O)C2)cn1 31154,C1(C(N(CC(CNC(CCCOC)=O)C)C)=O)CC(C(=O)OC(C)(C)C)=NO1 31155,N1(C(CN(CCC#C)C)=O)CCC2(COC(CNC(=O)CC3OCCCO3)C2)C1 31156,c1(CC(N2C(C(=O)OCC)C3C=CC2C3)C(=O)NC)cc2ccccc2o1 31157,N1(C(C2N(C)CCOC2)=O)CC2(CC(NC(C3(CC(F)F)CCNC3=O)=O)C2)C1 31158,N1(C(C(C)(C)CF)=O)CCC2(CC1)CCN(C(=O)CC1(c3ccon3)CCC1)C2 31159,n1(CCC)cc(C(=O)NC2CCCC2(C)CN(C)C(c2csc(O)n2)=O)c(C)n1 31160,O=C(COCc1ccccc1)N1CCC(S(=O)(=O)Nc2ccccc2)C1 31161,C(=O)(C(C)(C)CC(=O)N1CCCC(N(C)C(C2CCCC2F)=O)CC1)OC 31162,C1(C(=O)NC2C(CNC(c3c(C)ncn3C)=O)CCCC2)CCCCN(C)C1=O 31163,N1(C(C2CCC2(F)F)=O)CCC(F)(CNC(C2(c3cccs3)CC2)=O)C1 31164,C(=O)(CC(C)CC(=O)NC(CNC(=O)CCn1cc(C)cn1)CO)OC 31165,N1(C(CCC=C)=O)CC(NC(=O)C(C)N2CCC2)CCC1C 31166,C1(NC(CN(C(=O)OC)C)=O)CCN(C(=O)CN(C2CCC2)C)C1 31167,C(CN=c1[nH]c(Cl)nc2ccccc12)NC(C(C(C)C)NC(C)=O)=O 31168,C(C(C(C)(C)C)NC(C1(C)COC(=O)N1)=O)NC(Cc1cn(C)nc1)=O 31169,c1(C(N(C)CC2CCC(NC(CC3C(OC)CC3)=O)CC2)=O)cc([N+](=O)[O-])c[nH]1 31170,C1(CCC)(NC(C2CC2c2ccco2)=O)CCCN(C(=O)C(COC)N(C)C)C1 31171,c1(C(C)C)cncc(C(=O)NCC2CC(NC(=O)CCc3cccn3C)C2)c1 31172,c1(C(N(CC(CC)NC(c2cccnc2)=O)C)=O)c(C)oc(C)c1C 31173,N1(C(C2C(CC)C2)=O)CCC2(CCCN2C(=O)CSCc2cccnc2)C1 31174,c1(C(N(CC(C)O)CCNC(C2(C)CC=CC2)=O)=O)ccc(-c2cnn[nH]2)cc1 31175,C1(C(=O)NCCS(=O)(=O)NC)CC2CC1CN(C(=O)CCc1cscn1)C2 31176,N1(C(C2C(C)(C)COC2)=O)CC2CC(C1)CN(C(C1(C#N)CCC1)=O)C2 31177,c1(CC(=O)NC(C(C)NC(CC(=O)OCC)=O)C)cc(=O)n(CC(C)C)[nH]1 31178,N1(C(Cc2c(C)ncs2)=O)CC2CC1C2NC(C1CC(n2cccn2)C1)=O 31179,C1(NC(C(C=C)(C)C)=O)CCN(C(=O)Cn2cncc2C(=O)OC)CC1C 31180,N1(C(C2ON=C(CC)C2)=O)CC2CCC(C1)CC(NC(C1CC13CC3)=O)C2 31181,c1(C(=O)NC(CC)CNC(=O)Cc2ccns2)c(NC(=O)C(C)C)cccc1F 31182,CC(CNC(=O)COC(F)(F)F)CNC(=O)C(F)C1CCCC1 31183,C1(NC(c2cc(-c3ccns3)on2)=O)COCCN(C(c2ccccc2)=O)C1 31184,N1(Cc2cc(-c3ccc(-c4ccccc4)cn3)n[nH]2)CC(CN(C)C)CC1(C)C 31185,c1(C(N2C(CNC(C3CCCCCC3)=O)C3CCC2C3)=O)ccc2n[nH]cc2n1 31186,c1(C(=O)NC(CN(C(C2(COC)CC=CCC2)=O)C)C)ccc2ccccc2c1 31187,C1(NC(CCSCC)=O)CC2CCC1N(C(c1cc(C(N)=O)cs1)=O)C2 31188,O=C(C1=COCCO1)N1CCN(C(c2ccc(-c3ccco3)[nH]2)=O)C(CO)C1 31189,C1(CNC(C=CCC)=O)CCC(NC(c2cc(C(=O)OC)on2)=O)C1 31190,Cc1nc(Cl)nc(N2CC3CN(C(C4CCS(=O)(=O)C4)=O)CC3C2)c1C#N 31191,C(C(C(=O)NCCC1(O)CCN(C(=O)C=CCO)C1)C(C)(C)C)OCC=C 31192,C1(NC(CCOCCOC)=O)CN(C(c2ccsc2)=O)CC1C 31193,CC(C)CC(C)(C)C(=O)NCC1CC(C)CN(C(=O)C(Cl)=CCl)C1 31194,C1(C(=O)NCC(C2CCCC2)OC)CC(=O)CN1C(c1nn(C)cc1Cl)=O 31195,C1(C(N2CC(CNC(Cc3c(OC)nccc3)=O)C2)=O)CCc2ncncc2C1 31196,C1(C2CC2)(C(=O)NCC(CC)(CC)NC(c2cnn(C)c2C)=O)CC=CC1 31197,N1(C(c2cc(OC)c(O)nc2)=O)CC2(CCN(C(c3nc(C)n(C)n3)=O)C2)C1 31198,CCCCCC(O)CC(=O)NC12CC1CN(C(=O)CC(N1CCCCC1=O)C)C2 31199,c1(CC(C)C)nccc(C(=O)NC(C)CC2CN(C(c3ccccc3F)=O)C2)n1 31200,N1(C(c2sc(C)c([N+](=O)[O-])c2)=O)CCC2(CCOC2=O)CC1 31201,C1(CCC(=O)NC(COCC)C(C)C)CCCCN1C(c1cncs1)=O 31202,C1(C(N2CC(C)(C)C2c2cccnc2)=O)(COC)CCCNC1 31203,C1(C(=O)NCCC(CNC(=O)CNC(=O)C2CC2)O)CC(c2ccccn2)=NO1 31204,C(N=c1[nH]c2c(c(=NCCC3CC=CC3)[nH]1)CCCC2)C1CCC(=O)N1 31205,C(CCCCC(=O)NCCC(O)C1CCCC1)N(C(C=CC(=O)OCC)=O)C 31206,CCCC(CNC(C1CCC(=O)N1C)=O)CCO 31207,c1(CC)c(C(=O)NCC(C)N(C)C(c2cccc(-n3ccnc3)c2)=O)nnn1C 31208,C(=O)(C(O)CC(F)(F)F)N(CCNC(c1c(Cl)n[nH]c1C1CC1)=O)CC 31209,c1(-c2scc(C(N(CCCNC(C(CC)SC)=O)CC)=O)n2)cccc(C#N)c1 31210,c1(CC)cnc(O)c(C(=O)NCC(C)(C)NC(c2cc(COC)ccc2Cl)=O)c1 31211,C(CO)(CCC(C)C)NC(CSCCNC(Cc1scc(C)c1)=O)=O 31212,c1(C(N2CCC(CC=C)(NC(C3C4CCCC34)=O)C2)=O)ccc2c(c1)CCN2 31213,c1(CNCc2ccc(COC)s2)ccc(CN(C)C)cc1 31214,C1(O)(C(C)NC(c2cccc(C3CC3)n2)=O)CCN(c2nnc(C(N)=O)s2)CC1 31215,C1(NC(CCCC#C)=O)CCCC12CCN(C(c1cc(N)nc(Br)c1)=O)C2 31216,c1(C(N2CC(OC)(CNC(=O)C(C)C(C)(F)F)C2)=O)cc(S(C)(=O)=O)co1 31217,N1(C(COCCCOC)=O)CCCN(C(=O)CN2CCC(C)CC2)CC1C(C)C 31218,CC1(C)C(CC(=O)NC(C2CCCCC2)C(=O)NCc2ccc(O)cc2)C1(C)C 31219,CC1CC(NC(c2nncs2)=O)CCN1C(=O)CCN1CCOCC1 31220,N1(c2nnc(COC)s2)CCC2(CCC2)C(NC(=O)C2Cc3ccccc32)C1 31221,CC(C)C(C)C(CNC(C1(Br)CC1)=O)NC(C1(C(F)(F)F)CC1)=O 31222,C(=O)(C(=O)C(F)(F)F)N(CC(C)NC(C1(C)CCCO1)=O)C 31223,N1(C(CCC(=O)NCC)=O)CCCCC(C2CN(C(c3coc(Br)n3)=O)C2)C1 31224,N1(C(Cc2c(C)non2)=O)CCC(C2CCCCN2C(=O)COCCF)CC1 31225,Cc1cc(Br)cc(C)c1COC(=O)CCc1cccs1 31226,Cc1cc(CN2CCOC(C(N3CCC(CO)C(O)C3)=O)C2)c(C)cc1Br 31227,N1(C(c2cccn(C)c2=O)=O)CCCC(NC(=O)CCc2cnn[nH]2)C(F)C1 31228,CCCCCCN(C(=O)CCC=C(C)C)CCCC.C1(=O)C(C)N1 31229,N1(C(c2ncn(C3CNC3)n2)=O)CCOCC12CNC2 31230,c1(C(N2CC(C)(c3cn(-c4ccc(Cl)nc4)nn3)C2)=O)nccc2cccnc12 31231,C(=O)(CCCCCNC(=O)CC1CC1(C)C)NC(c1nccs1)(C)C 31232,c1(CNC(C(CC)O)=O)ncc(C(=O)NCCC23CC(CCO2)C3)cn1 31233,c1(C(N(C)CCOCCNC(C2CCS(=O)(=O)N2)=O)=O)cc(Cl)n[nH]c1=N 31234,c1(OCCC(=O)N(CC(C)O)CCNC(C(CC)F)=O)cccc(C)c1C 31235,C(=O)(C1=C(C)CCOC1)NCCN(CC(C)O)C(c1cnc(CC)[nH]1)=O 31236,C1(C(=O)NC2CN(C(=O)C(=CC3CCCC3)C)C2)(OC)CCCOC1 31237,CS(=O)(=O)CC(=O)N1CCCC1CC1CCCN(C(=O)Nc2ccc(Cl)cc2)C1 31238,C(=O)(C1=CCC(F)(F)CC1)NCC1(C)CCC(NC(CC(CC)C)=O)CC1 31239,N1(C(c2c(C)scn2)=O)CC2C3CCC(C2C1)N(C(c1cccnc1O)=O)C3 31240,C(CCS(=O)(=O)NCC(N1CC(O)(CNC(=O)C(C)=C(C)C)C1)=O)OC 31241,N1(C(c2ccn(CCCC)n2)=O)CCC2CN(C(C3(n4cnnn4)CC3)=O)CC12 31242,c1(C(N(C(C)CCNC(C2(O)CCOC2)=O)C)=O)cccc(Cn2cccn2)c1 31243,c1(CC)cc(C(N2CCC2C(=O)N(C)C)=O)ns1 31244,c1(C(N2CCC3(CN(C(c4c(N)nccn4)=O)C3)C2)=O)cc2c(Cl)cncc2o1 31245,c1(OC)cc(N)c(F)cc1C(=O)NC1CC(C)(NC(c2cc(O)nc(Cl)c2)=O)C1 31246,C#Cc1ccc(C(N2CCC(O)(C(C)CNC(c3ccc(Cl)s3)=O)C2)=O)cc1F 31247,C1(C(N(CC)CC2CC2)=O)CCCN(C(=O)CN2CCC(C)CC2)CC1 31248,C1(C(N2CC(C(C(=O)NCC3(c4ccno4)CCC3)O)C2)=O)COCCC1(F)F 31249,c1(C(=O)NC2CCN(C(C3N(C(C)C)CCC3)=O)C(C)C2)nnc2n1CCCC2 31250,C12(NC(C3CCC4(CCC4)O3)=O)CCCC1N(C(c1cnccc1Cl)=O)CCC2 31251,N1(C(C(=O)N(CCNC(C(CC)(F)F)=O)C)CC)CCc2ccccc21 31252,CC1CC(C(=O)NCC2(C(=O)NCC(F)Cl)CC2)=NO1 31253,C1(NC(C=C2CCC(C)CC2)=O)CC2(NC(=O)C=C3CCCC3)COC1C2 31254,C(C)(CCCC(C)C)NC(CC(CNC(C(COC)(C)OC)=O)C1CCC1)=O 31255,c1(OC)ccccc1CN1CCC(CNC(c2cc(C#N)cs2)=O)C1 31256,c1(C(=O)NC(C(=O)NC(C2(OC)CCC2)C)Cc2ccoc2)ccc(F)cn1 31257,c1(C(N(c2cc(I)ccn2)C)=O)cccc(Oc2ccccc2)c1 31258,C1(NC(C2(CC)CC2)=O)CC=CCC1C(=O)N(CC(F)(F)Cl)C 31259,C1(NC(c2cc(Br)cs2)=O)CCCN(Cc2ccc(I)c(O)c2)CC1 31260,c1(C2(NC3(c4nnnn4CC4CC4)CCN(C)C3)CC2)ccc(F)c(Cl)c1 31261,N1(C(c2ncn(CC)c2)=O)CCC(C)C1CNC(=O)C=CCCC(C)C 31262,c1(C(=O)NC(CC(C)NC(c2cccc(C(C)=O)c2)=O)C)cc(C)c(C)nn1 31263,C1(NC(C2CCC3(CN(S(=O)(=O)CC4CC4)C3)O2)=O)CCc2ccccc2O1 31264,c1(N(C(C(C(C)N)(C)O)=O)C)cccc(S(C)(=O)=O)c1 31265,CC(F)(C(=O)N1C2CCC1CN(C(c1ccc3cnnn3c1)=O)C2)C(F)(F)F 31266,C(C)(C(=O)N(CCc1cn(CC(C)O)nn1)C1CC1)(C1CC1)OC 31267,N1(C(CN(CC(=O)NC(C)CCC=C(C)C)CC=C)=O)CCCCCC1 31268,C1(NC(c2c(C)cc(F)nc2)=O)CCC2CC1CN2c1nc(Cl)ncc1Cl 31269,C(=O)(C(CO)N(C)C)N(CC(=O)NC1(CC(=O)OCC)CC1)C1CC1 31270,C(CCCC(CO)NC(=O)COC(F)F)NC(Cc1cccc(OC)c1)=O 31271,C1(COC(C2C(C)C(=O)C2)=O)(CF)CCOCC1 31272,N1(C(C(CC)SC)=O)CC(=O)NCC1C(=O)NC(COC)C(=O)OC 31273,c1(C(=O)NC2CC(C(N3CCCC(OC)C3)=O)C2)ccc(Cl)c(C)c1F 31274,C1(C(N2CCC(N(CC(N)=O)C)C2)=O)CC(C(C)=NO)C1(C)C 31275,N1(C(C)=O)CC2CCC(NC(c3ccnc(C(N)=O)c3)=O)(C2)C1 31276,c1(SC(C(=O)NCCCCN(C(C(C)=CC2CC2)=O)C)C)ccc(C)cc1 31277,c1(C(=O)NCCN(C(CC(C)O)=O)CC(C)O)cnc2c(c1)NCC2 31278,c1(CC)nc(C)c(C(=O)NC(C)CNC(c2nnsc2SC)=O)o1 31279,c1(C(N(C)CC2CC(F)CN2C(C2CCCO2)=O)=O)c(F)ccc(F)c1F 31280,C1(CNC(C(c2cccs2)SC)=O)CCC(C)(C)CN1C(=O)C=Cc1nc[nH]n1 31281,N1(C(COC)=O)C2CCCC1CN(C(=O)CCN1CCN(S(C)(=O)=O)CC1)C2 31282,c1(C(N2CC3(C(=O)NC4CCCC4(F)F)CC2CO3)=O)ccc2[nH]ccc2n1 31283,C12(C(N3CCCC(N(C(=O)C4=CSCS4)C)C3)=O)CC3CC(C(=O)N1)C2C3 31284,c1(C(N2CCN(C3CCOC3=O)CC2)C(=O)NCCC#N)cnc2c(c1)COC2 31285,c1(C(N2CCCC(C(=O)Nc3ccc(Cl)cc3CO)C2)=O)cc2ccoc2cn1 31286,c1(OCC)cnc(C(=O)NC2COCC2NC(=O)CCc2ccco2)c(Cl)c1 31287,CCC(COC)C(=O)N(CCNC(=O)C(c1ccc(Cl)cc1)C)C1CC1 31288,c1(CC)cc(C)c(C(=O)NC23CC2CN(C(=O)CC(C)NC(N)=O)C3)o1 31289,C1(NC(=O)NC(c2n(C)ncc2)C(=O)OCC(F)(F)C(N)=O)CC(O)C(F)C1 31290,C=CC1(c2ccccc2)COCCN1C(=O)C(=O)N1CC(Nc2ccc(Br)o2)C1 31291,N1(C(c2ccc(OCOC)cc2)=O)CC(NC(=O)CC2C(C)C2(F)F)CC(F)C1 31292,C1(C)(CNC(C2C(C)(C)C2)=O)CCN(C(c2cnn(C3CC3(F)F)c2)=O)C1 31293,c1(C(=O)NC2CCC(C)(NC(COC)=O)CC2)ccc2ncccc2c1F 31294,C1(C(=O)NC2CCCC2CF)COC2(C1)CN(C(=O)Cn1ncnn1)C2 31295,CCCC(=O)N(CCN(C(=O)Cn1cccc1)CC)CC 31296,C1(C(=O)OC)(C(=O)NCC(C)O)CCNC1 31297,Cc1cc(NC(C2CCN2C(=O)Cc2ccc(Cl)s2)=O)cc(Br)c1 31298,Cc1ccc(F)c(C(=O)NCC2C=CCN2C(=O)C=CCN2CCOCC2)c1Cl 31299,c1(C(CC)C)nc(C)cc(=NC(C)CC(C)NC(=O)C(C)(C(C)C)OC)[nH]1 31300,N1(C(C2CCC(F)(F)CC2)=O)CCN(C(C2CCC2(F)F)=O)CC(O)C1 31301,N1(C(Cc2c(C)cccc2C)=O)CCN(C(c2cscn2)=O)CC(CO)C1 31302,c1(C(=O)NCC2CC(NC(COCC)=O)C2)ccccc1SC(C)C 31303,CCCCCCCC(F)C(=O)N1CCOCC12CCCC2 31304,C(=O)(CCN=C(NCC(C1CCCCO1)(C)C)NC1CC=CC1)N(C)C 31305,CC1(C)CN(C(C2(CNC(c3cc(CO)ccn3)=O)CCCO2)=O)CCC1CO 31306,Cc1scc(C(=O)NCC(C)(O)CNC(c2cccn2C2CCCC2)=O)c1N 31307,C(=O)(C(CC(C)C)N(C)C(C)=O)NCC(CC)(C)NC(c1ccccc1OC)=O 31308,C(=O)(C(C)(O)C(C)C)N(CCCN(C)C)CCNC(c1ncc(OC)nc1)=O 31309,Cc1oc2cc(C(=O)NCC3CC3NC(c3nccc4n[nH]cc34)=O)[nH]c2c1C 31310,c1(C(=O)NC(C2CCOC2)C)ccc(CNC(c2coc(N(C)C)n2)=O)cc1 31311,C1(C(=O)NCC(CC)(CC)NC(C2C(C(F)F)C2(C)C)=O)CCCS(=O)(=O)C1 31312,C1(NC(c2n(CC)cc(Cl)c2)=O)CC2CN(C(C3(O)CCC3)=O)CC2C1 31313,CCC(C)(C(=O)NCC1CCN(C(=O)CC2CCCC(C)(C)C2)CC1)C(N)=O 31314,C1(C(=O)NCCC2CN(C(C(C)OCCC#C)=O)C2)CC2CCC1O2 31315,c1(C(N(C(C(=O)N(CC(C)OC)CC)C2CC2)C)=O)ccc2c[nH]nc2c1 31316,Cc1ccc(N)cc1C(N1CCCC(CO)(NC(=O)Cn2nnnc2C)C1)=O 31317,N1(C(C2CC(Cc3cn(COC)nn3)C2)=O)C2CCCC1C(C(=O)O)C2C(C)=O 31318,CCC(C(=O)N1CCC(C)(NC(=O)CN2CCN(C)C(=O)C2)C1)C(F)(F)F 31319,c1(C(=O)NC(CC(CC)C)C(=O)NCCOC)noc2ccc(Br)cc12 31320,C1(N(CCNC(CCCC)=O)C(c2csc(-c3ncc[nH]3)n2)=O)CCCCCC1 31321,C(C)(C(=O)N1CC(C(O)C(=O)NCCn2ccnn2)C1)OCCCC 31322,C(=O)(C(O)CC(N)=O)N1CCC(C(=O)NCCn2cccn2)(OC)C1 31323,N#Cc1c[nH]c(C(N2CCC(C(N3CCN(c4ccccc4)CC3)=O)CC2)=O)c1 31324,C1(NC(CC2(C=C)CCC2)=O)CCCN(C(c2cccnc2C(F)F)=O)CC1F 31325,N1(C(C(c2cnn(C)c2)NC)=O)CCc2ncc(C(F)(F)F)cc2C1 31326,c1(C(=O)NC2C3CC(OCC)C(C3)C2)noc2c1CC(F)(F)CC2 31327,CCCC(O)C(=O)NCC12CC(CN1C(=O)CC(C)N(C)C(=O)OC(C)(C)C)C2 31328,C1(C(C)(C)C)(CNC(CC(C)c2ccco2)=O)CCN(C(c2cccnn2)=O)C1 31329,c1(NC(=O)CCC2CCCN2c2ccn3nccc3c2)cc(Br)c(O)cc1Br 31330,CCC(CCC(=O)N1CCC(C)C1C(N1CC(OCC(N)=O)C1)=O)OC 31331,C1(OCC=C)CCCCC1N=c1cc(C)[nH]c(=NCCOc2ccccc2F)[nH]1 31332,N1(C(c2c(C)cno2)=O)CCC(C2CCN(C(=O)CC3COC(C)(C)C3)C2)CC1 31333,C1(CC(=O)NC(C)CO)C2CCC1CN(C(c1cc3ccoc3s1)=O)C2 31334,c1(OCC(=O)NC(C)CNC(c2cncs2)=O)cccc(Br)c1C#N 31335,C(C(C)(C)CC(=O)N1CC(NC(=O)CC(c2c(C)noc2C)C)C(C)C1)OC 31336,c1(CCC)c(C(=O)N(C2CCCN(C(=O)C(F)=C(C)C)C2)C)nnn1CC 31337,c1(NC(C(C)OCC=C)=O)nc(Cl)ncc1OC 31338,CC1(CC(=O)O)CCCN1C(c1ccc(OC2CCOC2)cc1)=O 31339,Cc1ccc2c(C(=O)NC3CCC4CCN(C(c5cccs5)=O)C3C4)n[nH]c2c1 31340,N1(C(C(C)C)=O)CCCCC1C(C)NC(=O)CCCc1nccs1 31341,C(=O)(C(CC)CC(F)F)NC(CNC(CCCOCCOCC)=O)CC(F)(F)F 31342,N1(C(c2nc(=N)[nH]cc2)=O)CC(F)(F)CC1C(=O)NC1C(O)C2CCOC12 31343,C1(C(CNC(C2C(OCC)C2)=O)(C)C)CCCN1C(=O)C(=O)Nc1ccccc1 31344,C1(C)(C(=O)NCC(C2CCCCC2)NC(Cc2c(C)con2)=O)CCCCO1 31345,N1(C(CCCC#C)=O)CCC(NC(=O)C=Cc2ccc(C(N)=O)cc2)CC1C 31346,C1(CC=C)(NC(c2ccnn2C(C)C)=O)CCCN(C(c2n[nH]c(CC)n2)=O)C1 31347,CC1(C)CN(C(=O)Cc2ccccc2Br)CC1NC(c1cnnc(O)c1)=O 31348,c1(NC(CCCC=C)C)ncc(S(=O)(=O)NCC2CCCCN2CC)cc1Cl 31349,c1(CC(C)NC(c2c(C)nc(COC)s2)=O)cc(F)c(F)cc1Br 31350,C(=O)(C#CC1(C)CCCO1)NC1CCC(NC(c2cc(C)cc(Cl)c2N)=O)CC1 31351,C1(COCC(=O)OCC)CN(N2CCCCC2C)C1 31352,Cc1cc2c(C(=O)NCC3CC(=O)N(C)C3=O)cccc2o1 31353,c1(NC)sccc1C(=O)NCc1cc(C(N2CCC(N(C)C)C2)=O)on1 31354,C(=O)(C1=CCC(C(F)(F)F)OC1)N1C2C(NC(n3cnnn3)=O)C(C2)C1 31355,N1(CC)CCCCC(N=c2[nH]c(=NC3CC(CO)C3)[nH]c3c(F)cc(F)cc23)C1 31356,C(=O)(C1=CCS(=O)(=O)C1)N1CCC(NC(C(C(=C)Cl)(C)C)=O)C(F)C1 31357,C(C)(CSC)(C(=O)NCCCC(F)(F)F)NC(c1cn(CCC)nc1)=O 31358,N1(CC(=O)OCCCCCF)CCN(C(c2cnco2)=O)CC1 31359,C1(C#N)(C(=O)NCC(CC)(CC)NC(=O)Cn2cc(C(C)O)nn2)CC12CCC2 31360,N1(C(CC(C)(C)C2CC2)=O)CCN(C(C2C3CN(CC(F)F)CC23)=O)C(C2CC2)C1 31361,C1(CC)CN(C(=O)CCNS(=O)(=O)C(F)F)CCC1NC(C1(CCOC)CC1)=O 31362,N1(C(=O)NC2CC(O)C23CCOCC3)CC2CC3CCCN3C2C1 31363,c1(CC(C(=O)NC(CNC(COC(CC)C)=O)(C)C)O)ccncc1Br 31364,CC1(C)COC(CC(=O)NC(C(=O)N2CC(C(C)(C)C)C2)c2cccs2)C1 31365,C1(CCCNC(C2C(C(=O)OC)C2)=O)CCCN1C(C1CCC(=O)C1)=O 31366,C1(C(=O)NCCSCC)C2CC3C(C2NC(C2(C)C(C)(C)C2(C)C)=O)C13 31367,N1(C(C2CCC(=O)OCC2)=O)CCCC2(CC(NC(c3cccs3)=O)C2)C1 31368,n1(CCC)cc(C(=O)NC2CC23CC(NC(=O)CS(=O)(=O)NCC)C3)c(C)n1 31369,C1(NC(c2c(C)n[nH]c2)=O)COC2CN(C(c3ocnc3C)=O)CC12 31370,c1(CCC)ncc(NC(=O)C(C)(C)CN(C(=O)C=CC2CCOC2)C)cn1 31371,c1(CCCC)nc(C(N2CC(CO)(NC(c3nc[nH]c3C(F)(F)F)=O)C2)=O)cs1 31372,C#Cc1ccc(C(N2CC3CC(NC(C45CCCC4CCC5)=O)C3C2)=O)nc1 31373,n1(CC(=O)N(C(C2(n3cnnn3)CC2)C)CCNC(CCO)=O)cnc(=N)[nH]1 31374,N1(C(C(C)NC(CC)=O)=O)CC(F)(F)CC1CNC(c1cccc(C)n1)=O 31375,c1(CNC(=O)Nc2c(C3CCN(C(=O)OC(C)(C)C)C3)n[nH]c2)c[nH]ccc1=N 31376,c1(-c2cc(C)no2)cccc(CNC23CC(C(=O)NC(C#N)C(N)=O)(C2)C3)c1 31377,S(=O)(=O)(c1ccc(Br)cc1NCC1OCC1(C)C)N1CCCC(CCC)C1 31378,c1(SCC)nccnc1C(=O)NCC(C(C)C)NC(C1(CC)CCC1)=O 31379,CC1C(NC(C2CCC2)=O)CC2CCC1N2C(=O)CC1CC(F)(F)C1 31380,C1(C(=O)NCCCCNC(c2c(C)n(C3CCOC3)nn2)=O)CCCS(=O)(=O)C1 31381,c1(CN(C(=O)Cc2ccnnc2)C(c2nn[nH]n2)C)cccnc1 31382,c1(C(=O)NCC2(F)CCC(NC(C3CCS(=O)(=O)N3)=O)C2)ccc2nn[nH]c2c1 31383,Cc1ccncc1CC(=O)NC1CN(C(=O)Cc2ncc(Cl)s2)CC1C 31384,c1(C(N2C(CNC(C3C(CN(C)C)C3)=O)CCC2)=O)ccc2ncc(=O)[nH]c2c1 31385,C1(c2cn(CCCN(C)C(c3cncc(OCC#N)c3)=O)nn2)COCC1(C)C 31386,C1(CNC(C2CCN(C(C)=O)C2)=O)CCCN(C(c2n[nH]cc2C(C)(C)C)=O)C1 31387,C(N=C(NC1CCS(=O)(=O)C1)N1CCn2c(cc3c(Cl)cccc23)C1)C1C(C)(C)C1 31388,C(=O)(CCC(C)OC(c1ccc(C2CCC2(C)C)cc1)=O)OCC 31389,CCCCC(C(=O)N1CC(C)(C#N)C1)NC(=O)CCN(C)CC 31390,c1(C(=O)NCC(O)CNC(C2CC3CC3C2)=O)ccc(S(=O)(=O)C(F)(F)F)cc1 31391,C1(CNC(CN2CC(C)C2)=O)CC2CN(C(C3(C(C)(C)C)CCCCC3)=O)CC12 31392,c1(C(N2C(C(N(C)CC3CCCO3)=O)COCC2)=O)ccc(O)c(F)c1 31393,CC1SCCC1NC(C1(CCNC(C2CC3(CC3)C2)=O)CCCC1)=O 31394,c1(OC)ccccc1CC(=O)NCCNC(c1cc(O)cs1)=O 31395,C1(O)(CNC(C=C(C)C2CC2)=O)CCN(C(=O)C(c2cc(C)cc(F)c2)C)CC1 31396,C1(F)(CNC(C(F)=C(C)C)=O)CCCN(C(=O)CCCC2CCC2)CC1 31397,CCC1=NOC(C(=O)NCCN(C(=O)CCc2ccncc2Br)C)C1 31398,C(C)(CCC(=O)NC(CSc1nc(-n2ccnc2)no1)C(=O)NC(C)C)SC 31399,C1(C(CNC(CC(C)F)=O)(C)C)CCN(C(c2cnn(C)c2C(F)(F)F)=O)CC1 31400,C1(CNC(CCSCCCC)=O)CCCCN(C(C2(C)CSC2)=O)C1 31401,C(CC(=O)N(C(C)Cc1cnc[nH]1)CC)N(CC=C)C(C1CN(C2COC2)C1)=O 31402,N1(C(c2cncc(COC)c2)=O)CC(NC(c2ccncc2OC)=O)CC(O)C1 31403,N1(C(C2C(C)(C)CCCC2)=O)CC23CCCC2(C1)CN(C(c1csc(S)n1)=O)C3 31404,N1(C(c2c(C)ncc(N)c2)=O)CC2CCCC(C1)N2C(=O)C(F)(F)C1CCCC1 31405,C(=O)(C1=CS(=O)CCC1)NC(C1(O)CN(C(C2(OC)CCCCC2)=O)C1)C 31406,Cc1cc(C)c(C#N)c(NC(C2CCCN(C(c3ccc(Cl)nc3)=O)C2)C)n1 31407,c1(OC)ccc(C=CC(=O)NC2CCN(C(C3(C)CC3(F)F)=O)CC2O)cc1Cl 31408,c1(C(=O)NC2C(NC(C3(OC)CCC3)=O)COC2)sc([N+](=O)[O-])cc1Cl 31409,c1(C(=O)OC)cc(C(=O)NC2CN(C(=O)CSCCC(C)C)CC2C)n(C)n1 31410,c1(OC)cnc(F)cc1C(=O)NC1COCC1NC(=O)C=CC1CCCC1 31411,C(=O)(C(C)CC(=O)OC)N1CCC(N2CCC(NC(CNC(CC)=O)=O)C2)CC1 31412,N1(C(C2CCC(C)(CC)O2)=O)CCC2CCN(C(=O)C(CC)(CC)OC)CC12 31413,c1(C(N2CCN(CC3CN(C(=O)CSC4CC4)C3)CC2)=O)nccn2nccc12 31414,c1(-c2onc(C3CC(C)(C)C3)n2)cc2occc2s1.c1(CC(C)C)ccccc1Cl 31415,C12CCN(CC1)C2=O.c1(C(C)NC(=O)CN(CCO)CCN(C)C)cnn[nH]1 31416,c1(C(N2C(CNC(=O)COCC3CCOC3)C=CC2)=O)nccc2cc[nH]c12 31417,c1(CCC(=O)NCC2(O)CN(C(=O)C=CC3CCCO3)C2)sccc1Br 31418,c1(C(=O)Nc2ccc(-c3ncn(CCCO)n3)cc2)cc2cncn2c(O)n1 31419,N1(C(c2c(C(C)=O)nccc2)=O)CC2(CCCCN2C(C2(CC(F)F)CC2)=O)C1 31420,C12(NC(COC)=O)CC(CNC(C3(O)CCSCC3)=O)(C1)OC21CCC1 31421,C1(NC(C(C2(NC(c3cc(SC)oc3)=O)CCC2)O)=O)CCCCC1CC(=O)O 31422,c1(OC)c(C(N2CCC(CNC(C3CC3C(=O)NCCO)=O)C2)=O)ccnc1Cl 31423,C1(C(=O)NCC(CC)NC(=O)CC2CCCO2)(OC)CCS(=O)(=O)C1 31424,N1(C(=O)NCCN(C2CCC3(CC3)N2)CC)CCCc2ccccc21 31425,c1(CC(=O)NC2C(NC(Cn3c(C)ccn3)=O)COC2)ccc2cccnc2c1 31426,c1(C(=O)OC)nn(C)c(NC(C2CN(C(C3CN(C)C3)=O)CCS2)=O)c1Cl 31427,CCCCN=C(NCC1(CCl)CN(C(=O)OC(C)(C)C)C1)NC1CCS(=O)(=O)C1 31428,N1(C(C2CN(C(CCC)C)C(=O)C2)=O)CCC2C(C1)CN2C(C1CC(O)C1)=O 31429,C1(C(N2CCN(C(=O)CN3CCCOC3=O)CC2CF)=O)CCOC2(CCC2)C1 31430,Fc1cc2nc(-n3nc(C4CCOC4)nc3CC3=CCCC3)[nH]c2cc1F 31431,C1(C(=O)NCCC(C)NC(=O)COc2cccc(Br)c2)CCN(C)C(=O)C1 31432,N1(C(C2(C)CCSCC2)=O)CCC(F)C(NC(C2(n3cccn3)CCC2)=O)C1 31433,C(=O)(C(C)CC(=O)c1ccccc1F)NCC1CC(NC(C(C)C)=O)C1 31434,N1(C(c2ccc(NC)c(F)c2)=O)CCC2CCN(C(C3CC=CC3)=O)CC12 31435,c1(C(N2C(C(N3CCC(CN(C)CC)C3)=O)C=CC2)=O)ncccc1Cl 31436,N1(C(=O)NC)CCC(C(=O)NCC(O)CNC(c2sccc2-n2cnnn2)=O)C1 31437,CCC(CCOC)C(=O)N1CC2CC(C1)C2NC(=O)CC1C(=O)NN=C1C 31438,c1(NC(C)=O)cccnc1C(N1CCOC(C(C)NC(=O)CCNC(N)=O)C1)=O 31439,C(=O)(CC1=CCN(C)CC1)NC(CCC)C(O)C(=O)NCC1CCOC1=O 31440,C1(CN(C(=O)Nc2cnco2)CC)CCCN(C(=O)OC(C)(C)C)C1 31441,Cc1nc(C)c(C(=O)NCC2CCOC2C(=O)Nc2ccc(C(C)C)nc2)s1 31442,CC(CC1CCCO1)C(=O)N(CCCOCCNC(c1csc(O)n1)=O)C 31443,C1(CN(C2CCC(O)(c3cccc(F)c3)CC2)C=O)CCCC(F)(F)C(=O)N1 31444,C1(C(N(CC=CC(=O)N(C(C#C)C)C)C)=O)CC(OC)(OC)C1 31445,C1(CC)CCN(C(c2cc(C)oc2C)=O)C1CNC(=O)C=CC1CCOC1 31446,C(=O)(C(C)(C)C(F)F)NC1CCC(F)(CNC(c2ccc(C(C)C)s2)=O)C1 31447,C1(NC(CCC(C)N(C)C)=O)CCN(C(C2CC(=C(F)F)C2)=O)CC1O 31448,c1(C(N2CC3CC(NC(C(=O)N(C)C)=O)C3C2)=O)ccc2c(c1)CCCCN2 31449,O=C(CCC(F)(F)F)NCC12CC1CN(C(c1cncc(O)c1)=O)C2 31450,CCC(CNC(C1CCOC(C)C1)=O)(CC)NC(=O)Cc1ccnnc1O 31451,C1(C(N2CCC(C(C)C(=O)N(C)Cc3cc(C)[nH]n3)CC2)=O)(CC)CNC(=O)C1 31452,CN1CC(F)CC1C(N1CC(OCCNC(C2CC2[N+](=O)[O-])=O)C1)=O 31453,C1(COC)(CNC(C2C(C)C2C)=O)CCN(C(=O)Cc2cnc(C)[nH]2)CC1 31454,C1(CNC(C(CC)(C)COC)=O)CC2CCC(C1)N2C(=O)C1=NOC(C)(C)C1 31455,C1(O)(CNC(c2c(CC)occ2)=O)CCCN(C(=O)C(C)(C)C2(C)CC2(F)F)C1 31456,C1(C(=O)NC(CC)CNC(C2C3(CC3)C23CC3)=O)CCc2c(ncn2C)C1 31457,C1(NC(c2ccnc(C(C)C)n2)=O)CC2CC1N(C(=O)Cc1nc[nH]n1)C2 31458,N1(CC(N2C(c3ccc(OCC)cc3)CCC2)=O)Cc2c(O)n[nH]c2C(F)(F)C1 31459,c1(C(=O)NCC2(CCNC(CCC(C)OC)=O)CC2)cc2c(ncn2C)[nH]1 31460,Cc1c(C(=O)NC2CN(C(C3SC4C=CC3CC4)=O)C(C)(C)C2)cccc1C#N 31461,C1(CNC(=O)NC(c2n[nH]c(C3CC3)n2)C)CC(C(F)(F)F)CO1 31462,C1(C(=O)N(C)CC2(C)CCC2)(CC)CN(C(=O)C(C)NC(=O)C2CC2)C1 31463,Cc1sc(Cl)nc1C(=O)NC1CCCC1NC(=O)C(F)=C1CCC1 31464,C#Cc1ccccc1CC(N1CCOCC1CNC(C1CN2CCC1CC2)=O)=O 31465,N1(C(C(CCC)NC(CC(C=C)CCC)=O)=O)CCC2(CCC(OC)C2)C1 31466,c12cccc(c1)C(=O)N2.C1(CNC(c2cn(CC)cn2)=O)CCCN1CC 31467,C(C1CN(C(c2cc[nH]c2)=O)CC1C(=O)Nc1cnc(CO)nc1C)=CC 31468,c1(COC(C)=O)ccc(C(=O)NC(C)(C)CCCNC(=O)CC2CCOCC2)cc1 31469,C(=O)(N=c1cc(-c2cncc(Br)c2)o[nH]1)N(CCN1CCCC1=O)CC 31470,c1(CC)ccc(N)c(C(N2CCN(C(c3cnc(C)nc3)=O)C(C3CC3)C2)=O)c1 31471,N1(C(c2c(C)cn(C)n2)=O)CC(C(=O)NCC2CC(C)(O)C2)CCC1C 31472,CC1CCN(C(c2sccc2F)=O)CC1NC(c1cc(F)c[nH]1)=O 31473,Cc1cc(C(=O)NC2CC(CCNC(C3CCC(C(N)=O)C3)=O)C2)cc(N)c1O 31474,C(CC(CC)C(=O)N1CCCC1C(C)(C)NC(=O)CCCC1CCOCC1)=CC 31475,C12(N(C(CSc3n[nH]c(=N)s3)=O)CC3CC3)CCC(CN(C(=O)C3=COCC3)C1)C2 31476,c1(C(=O)OC)ccccc1C(=O)N(CC(C)N(C(=O)C(C)Cc1ccco1)C)C 31477,N1(C(c2ccc(N(C)C)nn2)=O)CC(C2CN(C(c3ccc(N)cc3Cl)=O)C2)C1 31478,CC(C)(CCC(=O)NCC(=O)NCC(F)(F)F)c1ccccc1 31479,C(=O)(CCCC(C)C)NCC1(CNC(c2c(SCC)cccc2)=O)CC1(F)F 31480,C(=O)(C(F)CC(C)C)N(C(CCNC(C1(CC=C)COC1)=O)C)C 31481,CC(O)C(O)CNC(=O)CCC1CCC(NC(C2CCO2)=O)C1 31482,c1(NC(N2CCCC(NC)C2)=O)cccc2c1ccn2CC(=O)NC 31483,C1(C)(CC)C=C(C(=O)NCC(C)N(C)C(c2ncc(Cl)cc2F)=O)C1 31484,C(=O)(C=CS(C)=O)NCC1C(NC(C=CC=CC)=O)COC1 31485,C1(C)(C(N2CC(CNC(c3ccc(C(C)=O)nc3)=O)C(O)C2)=O)CCCS1(=O)=O 31486,N1(C(C(C2CCCC2)OC)=O)CC(CNC(=O)C=CC(F)F)CC1(C)C 31487,C(=O)(C1Cc2ccccc21)N1CC2CN(C(=O)C=Cc3cccs3)CC2C1 31488,c1(NC(C(=O)N(CC(C(C)O)O)C)=O)ccc(Cl)nc1O.C1(C)CC(=O)N1 31489,C(=O)(CS(=O)(=O)CCOC)NC(CN(C(c1cc(CS(C)(=O)=O)on1)=O)CC)C 31490,CC(C)CCCC(=O)NCC1(F)CCC(NC(C2CCC(C)(C)OC2)=O)C1 31491,N1(C(=O)OC(C)(C)C)CCC(CC(=O)OCc2c[nH]nc2-c2cnn(C)c2)C1 31492,CC(C)C(C)(CNC(c1ncoc1C1CC1)=O)NC(=O)CN1CC2CCC1C2 31493,c1(CN2C(CNC(c3c(C)cc[nH]3)=O)CCC2)ccc(C(F)(F)F)cc1Br 31494,c1(C(=O)NCC2CCCN(C(C3C(C)(CC)C3)=O)C2)noc2cc(Cl)ccc12 31495,c1(C(N(CC(C)NC(=O)C(O)CN(C)C)CC)=O)cccc(NC(C)=O)c1 31496,C(C(C(=O)NC1(CNC(=O)C=CCF)CCCCCC1)C(C)(C)C)OCC=C 31497,C(=O)(CCCC(N)=O)NC(C1CCN(C(c2ncccc2O)=O)CC1)C(C)C 31498,CC(CF)CC(=O)NC1CCCC1NC(=O)CCn1cccc1 31499,c1(N(C2CC3(CNC3)C2)C(=O)Cc2cc(O)nnc2O)cc(F)c(F)cc1Br 31500,c1(C(N2C(CNC(CC(CC)SC)=O)CC2)=O)ccc(Cl)c2ccccc12 31501,CC(CCCNC(c1cc(Cl)c[nH]1)=O)NC(=O)COCC(c1ccccc1)C 31502,Cn1nc(C(F)F)cc1S(=O)(=O)NCCc1cccc(Cl)c1 31503,C(C(=O)NCC(C)=CCC)(C1CCOC1)NC(C1(N(CC=C)C)CC1)=O 31504,C1(C(=O)NCCN2CCOCC2)(CNC(CN(C2CCSC2)C)=O)CCCC1 31505,C(=O)(CCC(F)(F)F)N1CC(NC(=O)CSC2CCC2)C(C(F)F)C1 31506,C(=O)(C(C)(C)C(C)(C)O)NC1C=CC(CNC(C(C)c2cc[nH]n2)=O)C1 31507,Cc1nc2ccccc2cc1C(=O)NC1CC2CC1N(C(=O)C(C)(C)C)C2 31508,c1(C(N2C(CN(C(C3CN(C(N)=O)C3)=O)CC)CCC2)=O)nc(OC)c(C)s1 31509,O=C1CCC(CC(=O)NCCCn2cc(-c3ccccc3F)nn2)C(=O)N1 31510,C(=O)(CC1OCCc2ccsc21)NCC1CCN(C(C2C(C)(C)C2(C)C)=O)C1 31511,C1(NC(=O)NCC2(C)COC2)CCOC2(CCOC2)C1 31512,C1(N(C(C2C(C(=O)OCC)CC2)=O)C)CCN(C(c2cnc[nH]2)=O)C1 31513,c1(CN(C2C3CNC2C3)CC(=O)OCCCC)ccc(OC)cc1 31514,Cc1[nH]nc(C(N2CC3C(NC(=O)C(C)(C)n4cc(Cl)cn4)C3C2)=O)c1F 31515,C1(COC)(CNC(c2ccc(C(N)=O)o2)=O)CCN(C(=O)C=C(C)Cl)C1 31516,c1(CC)ncc(CNC(C2(CCNC(=O)C=CC3CC3)CC2)=O)[nH]1 31517,c1(OCC(=O)N(CC(C)N(C(CCC#CC)=O)C)C)ccc(C(C)C)c(C)c1 31518,C#Cc1ccc(C(=O)NCC2(C)CCC(NC(c3cc(OC)nn3C)=O)C2)cc1 31519,c1(C(=O)NCC2(F)CN(C(C3CCC4(CC4)C3)=O)C2)cc(=O)c2ccncc2o1 31520,c1(OC)ncc(C(C2N(C(c3cnn(C)c3)=O)CCC2)=O)c(C)c1Br 31521,CC1(C)CN(C(c2cccc3ccoc23)C(=O)NC2CCC2)c2cccc(Cl)c21 31522,N1(C(c2cc(C3(C)CC3)n[nH]2)=O)CCCCC1CN(C(C1CCOC1=O)=O)C1CC1 31523,c1(CC)nnsc1C(=O)NCC1(C(N2CC(C)(F)C2)=O)CCCO1 31524,N1(C(C2(CSC)CC2)=O)CC(C2(NC(c3cnc(S)n3C)=O)CC2)C1 31525,Cc1cccn2cc(C(=O)NCC3C(O)C(O)CN3C(C3(F)CCOC3)=O)nc12 31526,c1(CN2CCCC(NC(c3ccnc(OC)c3F)=O)CC2)ccc(C#N)cc1F 31527,N1(C(CC(C=C)(C)C)=O)CCC2(CC1)OCCCC2NC(=O)C1=COCCO1 31528,Cc1nc(C#N)c(NCCC(N2CCN(C(=O)C(C)(C)C(N)=O)C3CC23)=O)o1 31529,C1(C(N2CCC(C(C)(C)NC(C(C)=CC)=O)C2)=O)CCc2[nH]nc(O)c2C1 31530,N#CC1CCCC(C(=O)NC(Cc2ccco2)C(N2CC(F)CC2CO)=O)C1 31531,c1(C(=O)NC2CC(CNC(C(CC=C)C)=O)C2)ccc(Cl)cc1-c1ccccc1 31532,Cc1ccc(C(=O)N(C)CCN(C(=O)C(C)OCCN(C)C)C)c(Cl)c1 31533,C1(OC)CCC(C(=O)NCCC2(NC(=O)Cc3csc(SC(C)C)n3)CCC2)C1 31534,O=C1OC2CC(C(=O)NCC3CCCN3C(c3cnc4[nH]ncc4c3)=O)CC2O1 31535,C(C)(CCCCNC(c1ccc(F)cn1)=O)NC(C(N1CCSCC1)C)=O 31536,Cc1ccnnc1C(N1CC(CNC(=O)CNC(C2CCOCC2)=O)C(C)C1)=O 31537,c1(C(C)C)nc(NCC2(CO)CC=CC2)cc(=NC2CC3CCC(C2)N3C)[nH]1 31538,N1(C(CC2C(=O)NC(=N)S2)=O)CC(NC(C2CCC3(CCC3)C2)=O)CC(O)C1 31539,c1(OC)cccc(C(=O)NC2CCCCC2NC(=O)CNC(c2cscn2)=O)c1 31540,CCC(C(=O)NCC(O)CCNC(=O)Cc1csc(C(C)C)n1)NC(C)=O 31541,n1(CC)nc(C(N2CCOC(CN(C(=O)C(C)CCOC)C)C2)=O)cc1C1CC1 31542,C12(NC(c3ccc(C)c(F)c3)=O)CCOCC1CN(C(=O)CC(C)N(C)C)C2 31543,C(=O)(C#CC(C)(C)C)N1CCCC(C(C)NC(=O)C(C)(C)N(S(C)(=O)=O)C)C1 31544,c1(C(N(CC(=O)NC(C)CN=[N+]=[N-])C)=O)ccncc1F 31545,Cc1ccc(F)c(C(N2CC(NC(c3c(C)nc(C)nc3C)=O)C(C)C2)=O)c1Cl 31546,c1(C(=O)NC2CC(CC(=O)Nc3ccc(Cl)c(O)c3)C2)cnc2c(Br)cccc2c1 31547,c1(C(N2CCC(CNC(C(CCC#C)O)=O)C2(C)C)=O)ccc2occc2c1 31548,n1(CCOCC)cc(C(N2CC(NC(c3cc(C4CC4)cs3)=O)C2)=O)nn1 31549,c1(OC)ccc(C)c(C2CCCN2c2nnc(-c3ncc[nH]3)n2CC2CC2)c1 31550,c1(C(N(C2CCN(C(c3cncn3C)=O)C2)CC)=O)c2c(nn1C)CCCC2 31551,c1(CN2C(C(=O)NCCCOCCC)CCC2)cc(C(F)(F)F)ccc1C 31552,C=CC(C)(C)CCNC(=O)C(CN(C)C)NC(c1ccnc(CO)c1)=O 31553,C1(CC(=O)NC(C2(O)CCCCC2)C(=O)N(C2CC(F)(F)C2)C)CC2CCC1C2 31554,n1(CCOCC)nc(C(=O)NCC23CC2CN(C(=O)C=C(C)C)C3)ccc1=O 31555,c1(CNC(CCN(C(=O)Cc2ccsc2)C)=O)cncc(F)c1 31556,CCC(C)CC(=O)C(=O)N1CC(C(=O)NCCCCCCF)C(F)(F)C1 31557,c1(OC)ncc(N2CCC(CN3CCOCC3)C2)cn1 31558,c1(C(=O)OC)ccc(-c2nc(Br)ccc2C)cc1C 31559,c1(CC)c(C(=O)N(CC(C)NC(=O)C(c2ccc(Cl)s2)=O)C)cnn1CC 31560,N1(C(c2ccc(F)c(Cl)c2)C(=O)NCCCCCC)CC(C)OC2(CCCC2)C1 31561,c1(COCCNC(C(c2n[nH]cc2Cl)N(CC(=C)C)C)=O)ccc(OC)cc1 31562,Cc1cccc(CCC(N2CCN(C(=O)C(O)C(C)(C)C)C(C)C2)=O)c1Br 31563,CN1CCN(C(=O)CC2(O)CCCCC2)C(CNC(c2ccc(C3CC3)o2)=O)C1 31564,C(N=c1[nH]c(=NCC2(OC)CCC2)[nH]c2cc[nH]c12)c1n(CCC)cnc1 31565,CC1CN(C(C2CC(n3ccnc3)C2)=O)CCC1NC(c1ccc(O)nc1)=O 31566,C(=O)(C(F)Cc1cnc[nH]1)N(CCC(C)NC(COCCOCCOC)=O)C 31567,N1(C(CCCCSC)=O)CC2CCCN(C(=O)CCc3cc(C)[nH]n3)C2C1 31568,C=CCCCCCCCCC(=O)NC1CC2CC1N(C(C1CC1(F)F)=O)C2 31569,c1(C(=O)NCC2N(C(c3cncc(CC)c3)=O)CCOC2)cc(Cl)c(F)cc1F 31570,C1(C(=O)NCC2(C(N3CC(F)(COC)C3)=O)CC(C)(C)C2)(CO)CCC(=O)N1 31571,C(N=c1[nH]c2cc(F)ccc2o1)C1CCN(C(c2cccc(OCC)c2)=O)C1 31572,Cc1cc2[nH]c(C(N3CCC(C)(NC(C4CCC5(CCC5)C4)=O)C3)=O)cc2s1 31573,C1(C(=O)NC(c2ncccn2)CC)(NC(=O)CC2CC2(C)C)CCCC1 31574,N1(C(CCc2cncc(C)c2)=O)CCC2CN(C(=O)C(C)NS(C)(=O)=O)CC2C1 31575,C(=O)(C(F)(CNC(C1CCCCC1)=O)C(C)C)NC(C#C)C(C)OC 31576,CC(CN=c1cc[nH]c(C#N)n1)(C1CC1)NC(C1CCC2CCCCC2C1)=O 31577,Cc1nn(C)c(NC(=O)C(C)C(C)(C)c2ccccc2)c1Br 31578,N1(C(C)C)CC(NC(=O)CC2CN(C(c3cc(CO)n(C)n3)=O)CC2C)CC1=O 31579,C1(C(=O)NC(CCC)CO)Cc2nccnc2CN1C(=O)Cc1ccc(F)cc1 31580,CCC(C)C(O)C(C)C(=O)N1CCC(CCC(=O)NCCSCCOC)C1 31581,c1(C(=O)NC2CCN(C(CN(CCOC)C)=O)C2C)ccnc2[nH]c(C)nc12 31582,C12(C(=O)Nc3nccs3)CCC(CC1)NC2 31583,C(=O)(CC(F)(F)C(F)F)NC1C(NC(CC(n2c(C)cc(C)n2)C)=O)COC1 31584,C(=O)(C(C(C)(C)C)OC)NCC1(NC(c2cc(CC(C)C)[nH]n2)=O)CCC1 31585,C(=O)(C(C)(F)C(=O)NCCCOCCNC(C1(C)CCC1)=O)OC 31586,C1(OCC(=O)NCCC)CCN(C(=O)Cn2c(N)cnc2C)CC1 31587,c1(CC)noc(C)c1CNC(=O)C(C)(C1CC1)N(C(=O)CCc1cn[nH]c1)C 31588,C(=O)(CCCCc1cnc[nH]1)NCC(CC)NC(=O)C(O)C1CC1 31589,C=CC1CN(C(=O)C(CC(C)C)OC)CC1NC(=O)CCN1CCC(O)CC1 31590,Cc1cccc(C(C)C)c1C(=O)NC1CC2CCC1N2C(=O)C(C)n1cncn1 31591,N1(C(c2c(CC=C)cccc2)=O)CC(C)CCC1CNC(=O)CN(C)C(N)=O 31592,c1(C(=O)NCC(CCOC)NC(c2cnc(CC(C)C)s2)=O)ccn(C)c(=O)c1 31593,c1(CC)noc2ncc(C(N3CCC4C(NC(c5c[nH]nc5C)=O)CC34)=O)cc12 31594,c1(C(C(=O)NCCC2CC2)N(C(C)COC)CCOC)ncn(C)n1 31595,c1(C(C(=O)NC2CC2)N(CCN=[N+]=[N-])CC)ccc(C2CC2C)o1 31596,C1(CC)C=CCCN1C(=O)CCC1(C)CCCN1C(=O)COCCCOC 31597,c1(OC)cc(C(=O)NCC2CCCN2C(=O)C=C(C)C(F)F)c2ccccc2n1 31598,c1(SC)cc(C(N2CC(N(C)C(C3CC(O)CN3C)=O)C(O)C2)=O)n(C)n1 31599,c1(NC(=O)CSCCC(O)c2cccs2)ccccc1COCC(F)(F)F 31600,C1(NC(c2nn(C)c3c2CCC3)=O)COC2(CCN(C(c3ncnn3C)=O)C2)C1 31601,C(=O)(CC1=NN(C)C(=O)C1)N1C(C(=O)NC2CCC3(C(C)C)C2C3)CCC1 31602,C1(C(=O)NC2C(NC(=O)COC3CC(F)(F)C3)CCCC2)CCC(F)(F)CC1 31603,CCCCC(C(=O)NC1(NC(C)=O)CC=CC1)NC(=O)C(O)CC(C)C 31604,N1(C(c2c(C)cns2)=O)CC=CC(C(=O)NOCCOC(C)C)C1 31605,C1(CC=C)(NC(C2CC2OC)=O)CC2CCC(C1)N2C(=O)CC1CC=CCC1 31606,C1(C(N(CCC#C)CCO)=O)CCN(C(c2occc2CC)=O)C(CC)C1 31607,c1(CN=C(NCC(O)CF)NC2CCC2)ccc2c(c1)CCO2 31608,c1(COC)cccc(C(=O)NCC2CCC(F)(CNC(=O)CC3CCCO3)C2)c1 31609,N1(C(C2CC(=O)NC(=O)C2)=O)CCOC2(CCC(NC(C3CC(=O)N3)=O)CC2)C1 31610,c1(C(=O)NC2C(CNC(=O)COC(F)F)C2)cc2ccc(Br)cn2n1 31611,c1(SCC(N2CC(OCCNC(C3(c4cccs4)CC3)=O)C2)=O)ccccn1 31612,c1(C(N(C)CC2COCCN2C(C2CC(C#N)C2)=O)=O)cnc(S(C)(=O)=O)s1 31613,N1(C(CCSCC(C)C)=O)CCCC(C)(NC(=O)Cc2ccc(Cl)cc2)C1 31614,Cc1cc(CC(=O)NC(C)CNC(C2(c3cccc(Cl)c3F)CC2)=O)ccc1O 31615,C1(SC)C(C(=O)NCC(CNC(COC(CC)C)=O)(C)O)C1(C)C 31616,C=CCCN=C(NCC1(OC)CCSC1)NC1CCCC(OC)C1 31617,N1(C(C(c2cnccn2)C)=O)CCc2[nH]nc(CNC(=O)C=CBr)c2C1 31618,c1(C(C)(C)C)ccc(C(=O)NC2(CNC(C3CCCOC3)=O)CCC2)[nH]1 31619,N12Cc3ccccc3CC1C2=O.c1(NC(C2C(N)C2)=O)cccc(C(=O)NC)c1 31620,c1(C(=O)NC2C(NC(c3cscc3F)=O)C2)ccc(-c2ccco2)[nH]1 31621,c1(CNC(C2CC(NC(CC(C)C(F)F)=O)C2)OC)cc(N)cc2ccccc12 31622,N1(C(c2ccc(C)cn2)=O)CC2CCN(C(=O)CC34CCCC3C4)C(C2)C1 31623,c1(C(N(C)CC2CCCN2C(C2OCC2(C)C)=O)=O)c(C(F)(F)F)cnn1C 31624,CC(C)CC(CNC(c1cnn(C)c1)=O)NC(=O)C(N1CCN(C)CC1)(C)C 31625,CC1(C)CC(CNC(c2ccco2)=O)CN1C(c1ccccc1C1CCCC1)=O 31626,C1(C(=O)NCC2(F)CC(C(=O)OCC)C2)CCN(C)C1(C)C 31627,c1(OCCC)ccccc1C=CC(=O)NC(C)CC(C)NC(=O)CCSCC 31628,C(=O)(C(CNC(=O)CC1CCC(=O)NC1)C(C)(C)C)N1CC(CN(C)C)C1 31629,N1(C(CC2CCCN(C)C2)=O)CCN(C(=O)C(F)=CC2CC2)C(CC(F)(F)F)C1 31630,C1(OCC(=O)NC23C(CN(C(C4C(OC)CC4)=O)C2)C3)CCC(F)(F)CC1 31631,c1(NC(=O)OC(C)(C)C)ccc(C(OC(F)(F)F)=O)o1 31632,N1(C(c2cnccn2)C(=O)NCCSC)Cc2cc(Cl)c(Cl)cc2C1 31633,c1(C(=O)Nc2scc(CC(N3CCC(C(F)(F)F)C3)=O)n2)nc2ccccn2n1 31634,CC(C)CC(C(=O)NCC(C)N(C)C)N(C(=O)CC1(O)CCCCC1)C 31635,N1(C(CN(C)S(N)(=O)=O)=O)CCn2nc(CNC(C3(F)CCC3)=O)cc2C1 31636,C1(O)(CNC(c2cccn2C(F)F)=O)CCCN(C(=O)C=CCN2CCCC2)C1 31637,N1(C(N)=O)CCCCC1C(=O)NC1C=CCN(C(C2CCC2)=O)C1 31638,c1(CN)cccnc1.Cc1occc1COC(F)F 31639,C(CCC(O)C(=O)NCC(C)(C)C(C)O)NC(c1n(C)cc(Cl)c1)=O 31640,C1(C(=O)OC(C)(C)C)(CN2CCCC2)CC=CCC1.c12ncc(s1)NC2 31641,C1(C(=O)NCCCOC(=N)O)C2CCC(C2)C1NC(=O)CCCn1ccnc1 31642,Cc1c(C(=O)N(C(C)CNC(=O)Cc2cnco2)C)cc(O)cc1N 31643,CC(C)CC(C(=O)NCCCNC(=O)C(C)(C)C1CCCO1)NC(=O)NC1CC1 31644,N1(C(CSCC=C)=O)CCC2(CC1)CN(C(C1C3CCC(C3)S1(=O)=O)=O)C2 31645,c1(COC(Cc2c(C)cc(O)cc2)=O)cc(=O)oc2cc(O)c(Cl)cc12 31646,c1(C(C2CNC2)=O)ccc(-c2cccc(C(=O)NC)c2)cc1.c1(CN)ccccc1 31647,c1(C(=O)NCC(CC=C)NC(c2cnn3cnnc3c2)=O)ncc2[nH]ncc2n1 31648,C1(NC(Cc2ccc(C)o2)=O)CC12CC(NC(C1(CF)CC(F)(F)C1)=O)C2 31649,CC1(F)CCCN(C(C2CCOCCN2C(=O)Cc2ccc3c(c2)CC3)=O)C1 31650,C(=O)(C(C#N)C(C)(C)C)NCCc1c(C(N2CCC(C(C)C)C2)=O)c[nH]n1 31651,C1(C(=O)NC2C(C)(C)C2)CCOCC1NC(=O)C(C)(F)c1ccon1 31652,Cn1cnc2ncnc(N3CC(C)(CNC(c4cnc(C(=O)O)cn4)=O)C3)c12 31653,Cc1[nH]nc(C(N2CCC3CCC23CNC(=O)CC(F)(F)F)=O)c1[N+](=O)[O-] 31654,Cc1nc(N2CCN(C(=O)C(C)OCC3CCCO3)CCC2C)c(C)c(C)n1 31655,N1(C(C(C(=O)OC)C)=O)CCC(CNC(=O)C(=Cc2ccccc2Cl)C)CC1C 31656,c1(CNC(=O)Cc2cnco2)cccc(NC(=O)CC2C=CCC2)c1 31657,C(C(C)C(=O)N1CC(C(C)NC(C2CCCC2C(F)(F)F)=O)C1)OC(C)=O 31658,c1(CC)[nH]c(C(=O)NC2CC(NC(=O)C#CC(C)C)C2)c(C)c1C(=O)OC 31659,N1(C(CCCc2cc(C)no2)=O)CCC2(CCCN(C(C3CCC(O)C3)=O)C2)C1 31660,c1(C(N(C)C(=O)OCCOC(c2cc3sccc3s2)=O)=O)c2ccccc2nn1C 31661,C=C(CNC(=O)C(F)C(C)CNC(=O)C=Cc1ccco1)C1CCOCC1 31662,c1(C(N2CC(CNC(CC3N(C)CCC3)=O)C2)=O)ccc2c(O)nc(S)nc2c1 31663,C1(NC(C(C)OCC(C)C)=O)CCCCCN(C(=O)CCCC2CCCCC2)C1 31664,c1(-c2cn(C(C(N3CC(COC)OCC3)=O)C)nn2)ccnc(F)c1OC 31665,N1(C(C2C(C)CCO2)=O)CCC(NC(=O)CN2C(C)CCC2C)CC1C 31666,c1(OC)cc(C(N2CCN(Cc3ccc(C)s3)CC2)C(=O)NC(C)(C)C)ccn1 31667,N1(c2cc(NC(=O)OC)ncn2)CCC2C(CCN2CC2(c3cccs3)CC2)C1 31668,CN1CC2CC1CN2C(=O)CCC(=O)Nc1ccccc1.C12=CC=C(C=C1)C2NC 31669,C(=O)(C1OCCn2ccnc21)NC1C(NC(c2cc(CO)on2)=O)C1 31670,N1(C(COCCC=C)=O)CCC(NC(c2nn(CC)cc2Cl)=O)C(F)C1 31671,C1(CNC(C2CC(=C)C2)=O)CCC2CN(C(c3ncoc3C3CC3)=O)CCC2C1 31672,c1(C(=O)NCC2C(NC(=O)CN3CCS(=O)CC3)COC2)cc([N+](=O)[O-])n[nH]1 31673,Cc1cnc(F)cc1C(N1CCN(C(=O)CCC[N+](=O)[O-])C(C)C1)=O 31674,C1(C(=O)NCCN(CCCC)C)CCC2(CC2)N1C(C1(N(C)C)CC1)=O 31675,c1(C(N2C(C(C)(C)NC(c3cnn(C)n3)=O)CCC2)=O)ccccc1O 31676,C(=O)(C(C(C)C)NC(=O)CC1CCCCO1)N(CCC#C)CCOC 31677,C(CSCc1ccccc1)(C(=O)N(C1C=CCC1)C)NC(C)=O 31678,C1(C(N(CC(CN(C(C(CC)C)=O)C)O)C)=O)CCC2CCCCC2C1 31679,Cc1ccc(F)c(C(=O)N(CCCCN(C)C(C2(C)C=CCCC2)=O)C)c1Cl 31680,N1(C(C2C(NC(C(CC)OCC)=O)CC2)=O)CCCCC1CO 31681,c1(C(=O)NC(C2(O)CN(C(CC(C)OC)=O)C2)C)ccnc(C2CC2)n1 31682,C(=O)(C1CCCc2cc(O)ccc21)N(C1CCN(C(C2(C)CCCC2)=O)C1)CC 31683,c1(Cn2cc(CC3CN(C(C4CC4N4CCCCC4)=O)C3)nn2)ccc(Br)cc1 31684,C12CCCCCN1C(=O)CN1CCN(CC1)N(CC1CCC1)C2=O.CC 31685,C(=O)(CC1=CCCCC1)NC1CCCN(c2ccc(C(C)C)nc2Cl)C1 31686,O=C(C1CCCc2nn[nH]c21)N1CCC(OC2CN(CC(Cl)=CCl)C2)CC1 31687,C=CC1(C(=O)NCCC2CCOC2)CCN(C(=O)Cc2ccc(C)s2)C1 31688,C12(CC(=O)N(C3CN(C(=O)CN4C(=O)CCC4=O)C3)C)CCC(C)(C1)OC2 31689,C1(O)(C(=O)NC(C)(CNC(=O)CCN2CCC(O)CC2)C2CC2)CCCCCC1 31690,C1(NC(C2NC(=O)OCC2)=O)CCCN(C(c2cnc(S)n2C2CC2)=O)CC1 31691,O=C(CC(O)CNC(=O)Cc1ccccc1F)NCC1CCN(C2CC2)C1 31692,C(=O)(C(C)(O)C(F)(F)F)NCC1(C)CCN(C(=O)Cn2ccnc2)CC1 31693,C(CC(=O)Nc1cc(C)cnc1C)(CC(C)C)NC(CC(COC)(C)C)=O 31694,N1(C(Cc2cc(C)sc2C)=O)CCCC(CO)(CNC(C2OCCC2(C)C)=O)C1 31695,Cc1ccc(F)c(CC(=O)NC2CC2NC(=O)CCCC2CC2)c1 31696,N1(C(C2C(=O)NCC2)=O)CCCC2(CCN(C(=O)CN3CCn4nccc43)C2)C1 31697,C(=O)(CC1C(=O)Nc2ccccc21)N1CCC(OCCCNC(COC)=O)CC1 31698,C1(NC(C(CCOCC)NC(=O)CS(=O)CC)=O)CCCC2(CC1)CC2 31699,N1(C(CCC#C)=O)CC(C(=O)N(c2ncccc2C)CC)CC(F)C1 31700,C1(CCO)(NC(=O)NC2CC2C(=O)NC(=O)C#CC2CC2)CCCCC1 31701,c1(C(N2CCN(C(COCCC)=O)CC2)=O)cnc([N+](=O)[O-])cc1C 31702,N1(C(CC(C=C)(C)O)=O)CC(C2CN(C(=O)CC3CCC(C)(C)O3)C2)C1 31703,Cc1nc2c(s1)CN(C(c1ccc(N(C)C)cn1)C(=O)Nc1ccccc1C)C2 31704,C1(NC(c2c(OC)nn(C)c2)=O)CN(C(c2cn(C3CCC3)nn2)=O)CC1(C)C 31705,C1(N(CCCC)C(C23CC(C2)C3)=O)CCN(C(=O)Cc2csc(COC)n2)CC1 31706,N(C(=NCC(C)C#N)NCC(c1cccc(F)c1)O)C(C=C)C 31707,c1(C(N(CC(CNC(CC(CC)C2CC2)=O)(C)C)C)=O)cnc2ncccn12 31708,C1(CSCCc2cccc(F)c2)CCc2nnc(C(F)F)n2C1 31709,c1(-n2cc(C3N(C(C(COC)NC(C)=O)=O)CCC3C)nn2)cccc(O)c1Cl 31710,C1(C(N2CC3C(NC(C4C=CCC4)=O)C(C3)C2)=O)COc2ccccc2O1 31711,N1(C(C(CC)NC(N)=O)=O)CCN(C(=O)CCc2ccc(Cl)nc2)CC1CC 31712,N1(C(CC#C)COC)CCN(C(=O)OCc2cnn(CCC(C)C)c2C)CC1 31713,CCC(CN(C)C)CC(=O)NCCN(C(C1COCC2(CC2)O1)=O)C1CC1 31714,C1(C(=O)NC2CCC(CNC(C3(C)CC3C)=O)CC2)(NC(C)=O)CCCCC1 31715,N1(C(C(CC)C#N)=O)CC(C(=O)NCC2(O)CCN(C)C2)CC(C)C1 31716,c1(C(N2CC(C)N(C(c3cccnc3)=O)CC2)=O)cc2c(F)c(Cl)ccc2[nH]1 31717,C12(NC(CCCC(=O)N(C)C)=O)CCCC1(F)CN(C(C1CCC(O)CC1)=O)C2 31718,C1(CNC(CSSC)=O)CCN(C(=O)C(C)Sc2ccc(N)cc2)C1(C)C 31719,c1(C(=O)Nc2nc(C3CCC(F)(F)CC3)cs2)ccc2c(c1)NS(=O)(=O)C2 31720,c1(C(=O)NC2C(NC(c3cncc(CC)c3)=O)CCC2)ccc([N+](=O)[O-])nc1 31721,c1(CNC(c2n(C=C)ccn2)c2nnnn2CC2CC2)ccc2c(c1)OCCO2 31722,N1(Cc2cc(C(=O)OCC)on2)CC(NC(C2(CC)CC2)=O)CCC1C 31723,CCC(O)C(C)C(=O)N(C1CCCCC1NC(=O)CC(C)SC)C 31724,c1(C(=O)OC(c2ncc(Br)cn2)C)cc(Cl)c(N)c([N+](=O)[O-])c1 31725,c1(C(=O)NCC2N(C(C(C)n3ccnc3)=O)CC=C2)nn(C)c(Cl)c1Cl 31726,N1(C(C2(C)CCCCO2)=O)CCOC2(C1)CN(C(=O)Cn1ccnn1)C2 31727,C1(CCC(=O)N(CC(C)NC(C2CSC2)=O)C)CC(C)(C)CO1 31728,C(C)(C(=O)N1CC2(C)CC1(C(=O)NCC1C=CCCC1)C2)(C(C)C)OC 31729,C1(CCN2CC(CN(CC)CC3CCCC3)OC(C)C2)CC1C1CCCCC1 31730,Cc1oc(-c2ccccc2)nc1C(=O)N(C)CCNC(C1CC(C)OC1=O)=O 31731,Cn1nc(CNC(=O)C(C)(C)NC(C2CCCCN2C)=O)n(C)c1=O 31732,N1(C(C(C)C)=O)CC=CC1CNC(=O)CCC1(OCc2ccccc2)CCC1 31733,Cn1cc(CC(=O)NC2COCC2NC(c2cnns2)=O)cn1 31734,CC1CN(C(=O)C=CI)CC2(CCN(C(=O)CC3(O)COC(C)(C)C3)C2)O1 31735,C(=O)(C(F)C(F)(F)F)NC(CC=C)CNC(=O)CCc1nnc(S)n1C 31736,C12(NC(=O)CSCc3ccccc3)CCCC1N(C(=O)COc1cn[nH]c1)CC2 31737,C(CC1=CCCCCC1)NC(C(C)NC(C(C)NC(=O)C1CC1)=O)=O 31738,C(CCCC(=O)NC(C)CCC(C)C)NC(C(COCC)C)=O 31739,c1(OC)c(C(=O)NC2CCN(C(c3cc(C(C)(C)C)[nH]c3C)=O)C2)ncnc1C 31740,c1(C(=O)NCCC2CCC(NC(C3(CC=C)CC3)=O)C2)[nH]nc2ncnc(O)c12 31741,C12(NC(C=CCOC)=O)CCCC1N(C(=O)Cc1ccc(C)cc1OC)CC2 31742,N1(C(Cc2n(C)ccn2)=O)CCCC(C2CN(C(c3cc(Cl)ncc3F)=O)C2)C1 31743,Cc1ccc(C(=O)C(=O)NC2CC(NC(=O)C(C(C)C)N3CCN(C)CC3)C2)cc1 31744,C=C(C)C1CC(=O)N(C2CC2)C(C)C(=O)NO1.c1(C(C)C)c[nH]ccc1=O 31745,c1(C(=O)NCCNC(c2c(C)cc(C)nc2C(C)C)=O)c(C)c(Cl)cc(C)c1N 31746,C1(N(C(COCC(=C)C)=O)C)CCCN(C(c2cscc2C(N)=O)=O)CC1 31747,C(C(=O)NCC(=O)NC(C)CCOC)(C(C)C)NC(C(CC)C)=O 31748,c1(C(=O)NC(CC=C)CNC(c2c(C)ncn2O)=O)cc(Cl)ccc1OC 31749,C(=O)(CC(C(F)F)NC(c1ccnc(C)n1)=O)NCCOCCC=C 31750,C1(C(=O)NC2(CO)CN(C(CN(CCCCCC)C)=O)C2)CC=CCC1C 31751,N1(C(Cc2cnc(C)o2)=O)CC2CC(NC(c3c[nH]cc3Br)=O)CC1C2 31752,CC1CCCn2ncc(C(N3CCC(NC(c4cc5ncccn5n4)=O)C3)=O)c21 31753,Cc1cccn2c(C(=O)NC3(C)CC(NC(=O)C(F)CC4CC4)C3)cnc12 31754,C12(C(N3CC(CNC(c4ccc(C)cc4F)=O)C(C)C3)=O)CCOC1CCOC2 31755,C1(CNC(c2cc(OC)n(C)n2)=O)CC2(CC2)CN1C(=O)CCCc1cncs1 31756,Cc1oc2ccccc2c1C(N1CCCOC(CCNC(=O)C2=CCOC2)C1)=O 31757,N1(C(CC)=O)CCN(CCNC(=O)CC2(O)CCCOC2)CC1 31758,C(CN=C(NCCC(C)(C)O)NC(c1cccs1)C)n1ncc(C)c1 31759,N1(C(c2csc(C)n2)C(=O)NC(C(=O)OC)C)CCN(c2ccccc2O)CC1 31760,c1(C(=O)NC(C2CN(C(c3c(Cl)cc(C)s3)=O)C2)C)c(C)nc(C2CC2)nc1O 31761,c1(C(C(=O)NCCCOC)N(CC(CC)CC)CC)sc(Br)nc1Cl 31762,CC1CN(C(C2CC23CC3)=O)CC(C)N(C(=O)C(C)Cc2ccccc2)C1 31763,C1(C(=O)NCC(CC(C)C)C)CN(C(C2CN(C)CC(C)O2)=O)CC12CCC2 31764,C1(C(N2CCSCC2)=O)(CC)CCCN1C(=O)Cn1cnnc1O 31765,c1(CC)cc(Br)cc(C(=O)NC2CCN(C(=O)Cc3nc[nH]n3)CC2F)c1N 31766,Cc1c(C(=O)NCCC2(CNC(c3ncccc3Cl)=O)CC2)cccc1F 31767,CC12CCOC(C(=O)NCC3CC(C(=O)NCCCN4CCC4)CO3)(C1)C2 31768,C1(CC)CN(C(=O)CCN(C(c2ccnn2C(F)F)=O)C(C)C)CC1O 31769,c1(C(=O)OC)cn(C)nc1OCCCOC1C=CCN(C(=O)OC(C)(C)C)C1 31770,c1(N(C(C(N)=O)C2CCCO2)C)ccc2nc(O)[nH]c2c1 31771,c1(OC)ccc(NC(=O)CC2CC(NC(=O)C(OC)OC)C2(C)C)c(O)c1 31772,c1(CC)cccc(OCC(N2CC(=C(F)CNC(=O)Cc3ncc(C)s3)C2)=O)c1 31773,C(=O)(CC(O)CC(C)(C)C)NCC(CNC(CCCc1ccc(C)c(C)c1)=O)O 31774,c1(C(N(C)Cc2c(CNC(C3C(C)CCO3)=O)cccc2)=O)c(Cl)cncc1Cl 31775,c1(C(=O)NCCOCCCNC(CCCC(CC)C)=O)c(F)ccc2n[nH]cc12 31776,C1(C(=O)NCCC2(O)CN(C(C3COC4(CCC4)C3)=O)C2)CCCCC(F)(F)C1 31777,Cc1cc([N+](=O)[O-])cnc1N1CC2CCN(C(=O)Oc3ccccc3)CC2C1 31778,C1(N(C(C(C2CCCC2)NC(C)=O)=O)C)CCN(C(c2ccc(C(C)=O)[nH]2)=O)C1 31779,c1(CC(N2CC(CC=C)(NC(=O)CC3CCC(O)C3)C2)=O)sc(C)cc1C 31780,Cc1cc(C#N)cnc1C(=O)NC1(C)CCCN(C(c2nc(Cl)cs2)=O)C1 31781,C12(C(=O)NC(CNC(c3ccnc(C)c3C)=O)(C)C)CCOC1CCOC2 31782,N1(C(COC2CCN(C(CC3CCCN(C)C3)=O)C2)=O)CC2CC2C2CC12 31783,C1(C(=O)NCC2(NC(Cn3c(N)cc(C)n3)=O)CC2)CN(C)CCN(C)C1 31784,C1(NC(C2CC(C)NC(=O)C2)=O)CN(C(=O)CC2CC(F)(F)C2)CC12CCCC2 31785,C(=O)(C1(C)CCOc2ccccc21)N1CC(OCCNC(C(C)(C)C2CC2)=O)C1 31786,C#CCCCC(=O)NCC1CC(NC(=O)CC2(OC3CCCCC3)CC2)C1 31787,c1(C(N(C2CN(C(C(C)OC)=O)C2)C)=O)c(NC(C)=O)c[nH]c1C 31788,c1(C(N2CCC(N(C(=O)CC3CCC(=O)NC3=O)CC)C2)=O)cc(O)cc(C#N)c1 31789,CC1CN(N(Cc2ccc(F)cc2Cl)Cc2ccnn2C)CC1F 31790,N1(C(C(COCC)C)=O)CCC(C)C(CC(N2CC(F)(F)CC2CO)=O)C1 31791,CCC(CNC(C1CC1C1CCCC1)=O)(CC)C(=O)N1CCN(C)CC1CO 31792,CCCC(CC)CC(=O)N1CC(NC(=O)COc2cc(Cl)ccc2C)C2(CC2)C1 31793,C1(C(N(CCOCC=C)C)=O)CN(C(=O)Cc2ccc(C)nc2)CC12CC2 31794,C(CCCC(C)(F)F)(C(=O)NCC1CCOC1)N(C)CCN1CCCC1=O 31795,CCC(CC)C(C)C(=O)N1CCC2(CC2C(=O)N(C(C)CO)CC)C1 31796,C1(NC(C(C(=O)OC)OC)=O)CCN(C(C2CCOC2)=O)CC1F 31797,C(COC(C)C)(C(=O)NCCNC(=O)CCCC1CC1)NC(C(C)NC(C)=O)=O 31798,C#Cc1ccc(C(=O)NCC(O)CCNC(=O)C(C)(CC)C(=O)OCC)c(C)c1 31799,CCC(CNC(=O)Cc1cscn1)NC(=O)C(N)=O 31800,Cc1ccc(C(=O)NC2C(Cl)(Cl)C23CC3)cc1Br 31801,N1(C(C(C)CC2CCCCC2)=O)CCC(O)C(NC(=O)C=CC2CC2)C1 31802,C(C(C)(F)CNC(=O)Cc1ccccc1)NC(COCC(C)C)=O 31803,C12(NC(C(OCC)OCC)=O)CCC(CN(C(=O)Cc3cc(C)cs3)C1)C2 31804,C1(CC(=O)NCC(=O)NCC)N(C(c2cc(C)[nH]c2C)=O)CCC1(C)C 31805,Cc1cnc(F)cc1NC(=O)NC1(CN(C)C)CCN(C)CC1 31806,c1(C(=O)NC(C2CCOC2)CNC(c2ccc(C)nc2)=O)c[nH]cc(F)c1=O 31807,C(=O)(CC1=NNC(=O)C1)N1C2CN(C(C(C)OCc3cccc(C)c3)=O)C(C2)C1 31808,c1(C(N2CC(CC(N3CC(C#N)C3)=O)C3(C2)CC3)=O)c[nH]c2ncccc12 31809,c1(C(N(C(CNC(Cc2c(C)ccc(F)c2)=O)C)C)=O)cccc(S(C)=O)c1 31810,CCC(C(=O)N(CCNC(=O)CC(c1ccc(Cl)cc1)O)C(C)C)C(C)(C)CC 31811,Cc1ncc(N)cc1C(N1CC(C2(NC(=O)Cn3cc(Cl)cn3)CC2)C1)=O 31812,C1(C(N2CC(C)C2c2ccccc2)=O)N(C(=O)C2=CCCCC2)CCC1(C)C 31813,CCC(CC)CC(=O)N1CCCC(C2CCCN2C(c2c[nH]c(=N)nc2C)=O)C1 31814,Cc1cc(C(=O)NC2CCC(CC(=O)NC3(C4CC4)CCCC3)CC2)ccc1O 31815,C1(NS(CC)(=O)=O)CCCN(c2nnc(-c3nn(C)cc3Br)n2C2CC2C)C1 31816,c1(OC)cccc(NC(C2(O)CCN(C(c3ccc(O)c(F)c3)=O)C2)=O)c1C 31817,N1(C(C23CC(NC(c4c(CCC)nco4)=O)(C2)C3)=O)CCC(O)CC12CC2 31818,CCC(O)CC(=O)N1CCCCC1Cn1cc(C2C3CCCCC23)nn1 31819,N1(C(CC2(C(=O)OC)CC2)=O)CCN(C(C2CSCCS2)=O)CC(C)(C)C1 31820,c1(CCC(=O)NC23CC(C2)N(C(c2ccncc2)=O)C3)cc(F)cc(F)c1 31821,N1(C(c2c(CC)[nH]c(=N)s2)=O)CC(F)(F)CC1CCNC(C12CC(CO1)C2)=O 31822,C1(CCN(C(=O)COC(c2ccccn2)=O)C)CCCCN1C(=O)C(C)(C)C 31823,CCC(CC)C(=O)N(CCCOCCNC(C1(Cc2cnn[nH]2)CCCC1)=O)C 31824,N1(C(c2ccn(C)c2)=O)CCC(NC(=O)CC2(O)CCC2)CC1 31825,c1(CC)nc(C)c(CNC(=O)C=CC(C)NC(=O)C(C)C(=O)OC)o1 31826,c1(SCC)ccc(NC(C2CN(C(=O)C3=C(C)OCC3)CCN2C)=O)cc1C 31827,N12CCC(O)(CC1)CNC(=O)c1scnc1CC2=O.c1(CNC=O)nccs1 31828,C(=O)(C(F)C(C)(F)F)N(CCCNC(CCC(=O)NCCCN(C)C)=O)CCO 31829,N1(C(c2nc(C)oc2)=O)CC(CCNC(C2CC3C=CC2C3)=O)C(C)C1 31830,C1(NC(C(CC)OCC)=O)CC2(C1)CC(CNC(c1cn(CC)nn1)=O)C2 31831,C1(C(N(CCCC(=O)NCCOC(C)C)C)=O)CCCC(C)C1 31832,C1(NC(C(CCO)N(C)C)=O)CN(C(C2CCC=CCCC2)=O)C2(CCC2)C1 31833,c1(OCC)cc(C(=O)N(CC(O)CNC(=O)CCc2cc[nH]n2)C)on1 31834,N1(C(c2c(C)noc2)=O)CC(C)CN(c2cc(O)ncn2)C(C)C1 31835,C1(NC(C(C)OCC#C)=O)CCN(C(c2cnc(C(C)(C)C)nc2)=O)C1C(C)C 31836,c1(C(N2CC(NC(COCCCCC)=O)C3C2C3)=O)csc(=NC2CC2)[nH]1 31837,C1(SCc2cc(CC)n[nH]2)CCN(C(=O)CN(C)CCc2noc(C)n2)CC1 31838,N1(C(C=CCC)=O)CCC(C2CC2)(CNC(c2ccc(Cl)s2)=O)C1 31839,Cc1ccn(C)c1C(=O)NC1CC1NC(C1(C2CCCCC2)CCOCC1)=O 31840,Cc1cccnc1CNC(C1COCCC1NC(=O)COCCF)=O 31841,N1(C(c2cc(C3(C)CC3)n[nH]2)=O)CCC2(CCC(NC(C3(CO)COC3)=O)C2)C1 31842,C(=O)(C1CCc2c(Cl)cccc21)NCC1N(C(c2n(C(C)C)ncc2F)=O)CC1 31843,c1(C(C)(C)C)ccoc1NC(C1(NC(=O)CSC2CCCCO2)CCCC1)=O 31844,C1(NC(C2CC(C)OC2C)=O)CC2(C1)CC2N=c1cnc(F)c[nH]1 31845,C1(CC)CN(CC)CCN1C(C1C(CNC(=O)C#CC(C)C)C1(C)C)=O 31846,CCCCC(C(=O)NC1CC(CCO)C1)NC(=O)C=CCCC(C)C 31847,C1(NC(C2CC2CF)=O)CC2CC1N(C(=O)Cn1ccccc1=O)C2 31848,CC1N(C(c2cccc(CNC(=O)Cc3ccc(O)cn3)n2)=O)CCOC1(C)C 31849,c1(C(=O)NCC(CC)NC(=O)C(C(C)C)N(C)C)cc(Cl)ccc1[N+](=O)[O-] 31850,C1(CNC(N2CCC(N(C(C)C)CC#N)CC2)=O)CCCC1S(C)(=O)=O 31851,C1(C(=O)NC(C(=O)NC)C(C)C)CC12CCN(C(=O)C(O)C(F)(F)F)C2 31852,N1(C(C(CSC(C)(C)C)NC(C)=O)=O)CC2CC(NC(=O)CSC(F)(F)F)C(C2)C1 31853,CCC(C#N)C(=O)N1CCCC1C1(NC(=O)C(F)CN(CC)CC)CC1 31854,N1(C(CCC=C(C)C)=O)CC(F)(F)CC1C(=O)NCCc1ccc(C)s1 31855,c1(C(N2CCC(C)(CNC(C(CCSC)O)=O)C2)=O)sc2nnc(S)n2c1C 31856,c1(NC(=O)NCC2CC2Nc2ccc(C(F)F)cn2)ccc(Br)cn1 31857,C(C)(C(CC(=O)NCc1ccc(C#N)s1)NC(C1CCC(C)(C)C1)=O)OC 31858,C(=O)(C(C)(C)C(=O)N(C)C)NC(CNC(C(C)SCCCC)=O)CCOC 31859,n1(CC)cc(C(N2CCN(CCO)C(C)C2)=O)c(=O)c2cc(Br)ccc12 31860,c1(C(N(C2CC(NC(c3cc4sccc4s3)=O)C2)C)=O)nccc2ccn(C)c12 31861,c1(NC(C(=O)N(C(c2ccc(F)c(Cl)c2)CN)CC)=O)ccc(C)c(C)c1 31862,CC(C)CC(F)(F)C(=O)NC1CC2(C1)CC2NC(=O)CCN1C(=O)CN(C)C1=O 31863,C(CCCCC(=O)NC1CCC(CCNC(c2cncc(CO)c2)=O)C1)N(C)C 31864,C1(NC(c2c(CC)cccc2)=O)CCN(C(c2c[nH]ccc2=O)=O)CC1C 31865,c1(C(=O)NC2CC(C(F)(F)F)C2)ccc(C(F)NC(=O)CC2CC2)cc1 31866,CC1CCN(C(c2ccnc(-n3cncn3)c2)=O)C1CNC(=O)C(C)CO 31867,C(CC(C(=O)NCc1ncc(C(N2CCOC(C(C)C)C2)=O)cn1)OC)OC 31868,C(CC(=O)NCCCCCNC(C1CS(=O)(=O)C1)=O)(C1CC1)NC(=O)OC(C)(C)C 31869,Cc1ccncc1CC(=O)NCC1(C)CCC(NC(=O)CCc2cccs2)C1 31870,N1(C(C(N2CCOCC2)C)=O)CCC2(CCN(C(=O)C3=CC4C=CC3C4)C2)C1 31871,C1(CNC(C2CCC(CCC)CC2)=O)CN(c2ncnc(=N)[nH]2)CCC1(C)C 31872,N1(C(C(C)C2CCCC2)=O)CC(CC(=O)NC2CCCCCC2F)CC1(C)C 31873,c1(CN(C(C(C2CN(C(CCNC(=O)NC)=O)C2)OC)=O)C)cnc(C)s1 31874,c1(OC)ncc(-c2cncc(C(=O)NCC3CCCC3CO)c2)c(SC)n1 31875,c1(CC(=O)NCC2CCCN(C(=O)C(c3ccc(F)cc3)O)C2)cccnc1Cl 31876,O=S(=O)(C1CCC(C(F)F)CC1)NCc1ccc(OC2CCOC2)cc1 31877,CC(C)CC(O)CC(=O)N1CCCCCC1C(N1CC(N(C)C)C1)=O 31878,c1(C(=O)NCC(C)CNC(c2c[nH]cc(Cl)c2=O)=O)cccc2c1oc(=O)n2C 31879,C1(NC(COCCC=C)=O)CCCCCC1C(=O)Nc1cc(C)ccc1OC 31880,C(=O)(C1OC(=O)c2ccccc21)N1CCC2(C(NC(c3c(C)occ3)=O)C2)CC1 31881,C1(C(C(N2CC(=C(CNC(C(C3CCOCC3)C)=O)F)C2)=O)F)CCCCCC1 31882,CC(C)CC(C(=O)NOC1CCOCC1)ONNCc1ncccn1 31883,CC(C)C(O)C(=O)NC1(CF)CCN(C(=O)CCc2csc(Br)c2)C1 31884,C1(CCCCCNC(c2cnccn2)=O)CCN(C(C2CCC(F)C2)=O)CC1 31885,CS(=O)CCC(=O)NC1CC1NC(c1cccn1CCc1ccccc1)=O 31886,c1(C(=O)NC2CCCN(C(C3CC(SC)C3)=O)C2)n[nH]c2cc(C)ccc12 31887,c1(CNC(C=CC(CC)C)=O)cccc(C(=O)NCCCc2nnnn2C)n1 31888,CCC(CCCC(=O)NCCN(CCO)CC)NC(c1nc(C)c(C)s1)=O 31889,CC1CNC(=O)CN1C(C1CC12CCN(C(=O)CN1CC3CC3C1)C2)=O 31890,N1(C(CC(COC)(C)C)=O)CC2CC(O)C1C2NC(=O)CCC1CCCO1 31891,N1(C(CC2(CSC)CC2)=O)CCC(C2(NC(=O)C(c3cnccn3)C)CC2)CC1 31892,Cc1nsc(N2CC(F)(F)CC2CNC(c2cn(C3CCC3)nc2C)=O)c1C#N 31893,c1(CC(=O)NCC(CNC(C2N(CC)CC2)=O)O)sc(C2CCC2)nc1C 31894,N1(C(CC(C(=O)OC)C)=O)CCC2C(C1)CN2C(=O)Cn1cc([N+](=O)[O-])c(C)n1 31895,C=C(Cl)C(C)(C)C(=O)NCC1(NC(=O)C(C)OCC(C)C)CCCCCC1 31896,CC(CC(F)(F)F)C(=O)N1CCC(C(=O)NCc2cc(O)ns2)C12CCC2 31897,C1(C(=O)NCC(C)CN(C(=O)CSCc2cccnc2)C)C2COCC12 31898,c1(CCC)cnnc(C(=O)NC2CCC2NC(=O)CCC(C)C)c1 31899,c1(C(=O)NC(CNC)C(C)(C)C)cc2cccnn2c1 31900,N1(Cc2c(C)c(I)nn2C)CCCC12CCCSC2 31901,C1(CC)(NC(=O)CC(C)C2CC2)CCCN(C(=O)CN2CCC(F)(F)C2)C1 31902,C12(CNC(c3cc(Cl)no3)=O)CCCC1CN(C(C13CCC(CF)(C1)OC3)=O)C2 31903,C1(CSC)CC(C(=O)NC2(CNC(C3(C)CCC3)=O)CC2)C1 31904,CCC(C)(CC)C(=O)NCCOC1CN(C(C2COC(C)(C)O2)=O)C1 31905,N1(C(CCNC(=O)OC)=O)CC(C)(NCC2=NOCC2)CC1(C)C 31906,C(C(F)(C(=O)NCCC(O)C(C)C)C(C)C)NC(C(=Cc1ccccc1)C)=O 31907,C1(=O)C(O)CCCN1C(=O)C=C(C)C(C)(C)C.C1(CCC)CCC(C)(CC)CC1 31908,C(=O)(C1COc2ccccc21)NCC1CN(C(CCCC)=O)C2C(O1)CCC2 31909,N1(C(C2C(C)(C)C(NC(=O)CCCC3CCC3)C2)=O)CCC2(CC1)CC2C#N 31910,N1(C(CCOC)=O)CCC(C2CCC2)(CNC(=O)CC=C(Cl)Cl)CC1 31911,C1(C)(C(=O)NC2(CNC(C(COC)(C)C)=O)CCCCCC2)CC(C)OC(C)C1 31912,C1(NC(c2ccc(F)s2)=O)CC(O)CN(C(=O)C2=CCCS2)C1 31913,CCC(C)C(C)C(=O)N1CC(F)CC1CN(C)C(c1ncc(OCC)cc1Cl)=O 31914,c1(CC)cc(NC(C2(F)CCN(C(c3cc(Br)ccc3F)=O)CC2)=O)ccc1F 31915,C(C1CN(C(=O)C(C)C2CCC2)CC1C(=O)NC(C)C(F)(F)F)=CC 31916,c1(N(C)CC2CC2)nc(N2CCCC(Cc3ccns3)CC2)c2c(n1)CSC2 31917,C(=O)(C(CCC1CCC1)NC(c1cnc(C2CC2)o1)=O)Nc1c(C)csc1 31918,N1(c2nc(C)cc(OCC)n2)Cc2nccn2CC(NC(c2coc(C)c2)=O)C1 31919,Cc1ccc(S(N)(=O)=O)cc1C(=O)Nc1cn(C2CN(C(=O)CC3CC3)C2)nn1 31920,c1(C(=O)NC(CNC(c2c(C)ccnc2)=O)(C)C(C)C)onc2c1CCCC2 31921,CC(C)(C)C(O)CNC(=O)NCC(COC(=O)Nc1ccccc1)(C)F 31922,S(=O)(=O)(c1ccc(Br)cc1NC(C)CCSC)NC(C=C)COC 31923,CC1CC(NC(=O)CCCN2CCCCC2)CN(C(c2coc(C#N)c2)=O)C1 31924,C(=O)(C=C1SCC(=O)N1C)N1CCC2(CC(CCCc3c(C)cc(Cl)nc3Cl)C2)C1 31925,Cc1nc2cc(C(=O)NCC3CN(C(C4CCOC4)=O)CC3C)cc(Br)c2o1 31926,Cc1noc(C(=O)OCC(=O)NC2CCC(C)(C)C2)c1I 31927,Cc1cc(C(N2CCN(C3COCC3NC(=O)CC3(C)CC3)CC2)=O)oc1C 31928,N1(C(c2n[nH]c(C3CC3)c2Cl)=O)CC2(CCN(C(C3CC34CC(F)(F)C4)=O)C2)C1 31929,CCC(C)CC(=O)C(=O)N1CCCC(CN(C)C(c2cc(O)n(C)n2)=O)C1 31930,N1(C(C2OCCN(C(=O)CN3CCOCC3)C2)=O)CCCC2(COC2)C1 31931,C(=O)(C(C(C)CC)c1ccco1)NCCC1CCCC1.CCCC(=O)NC 31932,Cc1cc(C(N2CCOC(CCNC(C3CC(C)(F)C3)=O)C2)=O)n2nccc2n1 31933,C1(C(CNC(c2c(C)cco2)=O)(C)O)CCCN(C(=O)Cc2c(C)noc2Cl)C1 31934,N1(C(Cc2c(C#C)cccc2)=O)CCN(C(=O)CC2CC(=C)C2)C(C)C1C 31935,CCC(CCCC(=O)NCc1nncs1)NC(C1CCC(O)C1)=O 31936,c1(C(=O)NCCCN(C(=O)CC2CCN(C)C2=O)CC)cc(OC)c(Cl)s1 31937,N1(C(C2Cc3nccn3C2)=O)CC2CCN(C(c3cc(O)cs3)=O)C2C1 31938,CC1(C)COCCC1C(N1CC2CC(NC(c3cnoc3C3CCC3)=O)C2C1)=O 31939,c1(C(N2C(CNC(CCOCC(C)C)=O)CC3(CC3)C2)=O)nsc2ccccc12 31940,c1(C2OCCC(OCC)C2)ccc(OCCN(C)Cc2cc(Cl)ccc2C)cc1F 31941,n1(CC)nncc1C(=O)NC12CC(CNC(=O)C(C3(O)CCCC3)F)(C1)C2 31942,C1(CC)CCC(NC(=O)C(Cn2ccnn2)NC(=O)C(C2CCOCC2)C)CC1 31943,c1(C(=O)NC(CNC(c2c(C)nn(C)c2C(F)(F)F)=O)C)ccc(C#N)nc1O 31944,c1(C(=O)NCC2OCCC2C(=O)NCCn2cnnn2)cc(F)cnc1O 31945,c1(NC(C2C(NC(C3C(C)(C)OC(=O)C3)=O)C3CCC2C3)=O)cc[nH]c2nccc1-2 31946,Cc1cccnc1C(=O)NCC1(C(=O)NCC(c2nccs2)C)CC2(CC2)C1 31947,n1(C(C)C)ncc(F)c1C(=O)NC1CCCC1CNC(=O)CCc1cnn(C)c1 31948,C1(CNC(CCN(C(=O)C(C)N(C)C(C)=O)CC#C)=O)CC2CC1CC2O 31949,N1(C(C2(SCC)CCC2)=O)CCC(N(C(=O)Cc2cccc(CO)c2)CC)CC1 31950,Cc1cnc2n1CCC(C(=O)NCCN(C(=O)C1=CCCS1)C)C2 31951,N1(C(C23OCC(C)(C2)C3)=O)CC=C(CNC(=O)Cc2cccnc2)CC1 31952,N1(C(c2ccnc3c2CCC3)=O)CCN(C(C2CCC(O)C2)=O)C2(CCC2)C1 31953,C1(NC(CSCCCC)=O)CC2CCC(C1C)N2C(C12CC(CO1)C2)=O 31954,c1(NCC2CN(C(C3CCc4nccn4C3)=O)C2)ncc([N+](=O)[O-])cc1F 31955,CC1CCN(C(=O)CN2CCCCCC2)CC1NC(=O)CC1CC=CCC1 31956,CC(CC(C)(C)C)C(F)C(=O)N1CCOC2(C1)CN(C(=O)C(C)(F)C(C)(C)F)C2 31957,c1(CC(=O)N(C(CCNC(C(COC)COC)=O)C)C)cnn2ccccc12 31958,C1(OCCCNC(C(C)c2ccsn2)=O)CCN(C(c2c[nH]ccc2=O)=O)CC1 31959,CCCC(C)(O)C(=O)NCC(C)(C)CNC(c1ccnc(Cn2cnnc2)c1)=O 31960,N1(C(C2CCC(=O)CC2)=O)CCC2CCCC12C(=O)NOCC1CCOC1 31961,C(=O)(C(C)(C)C(N)=O)N1CCC(CN(C)C(C2CCC2(C)C)=O)C1 31962,C1(CC(N2CC(C)(NC(=O)CCCC3CCOCC3)C2)=O)CCCCC1O 31963,N1(C(c2cncc(N)c2)=O)CCC(C2CC2)(CNC(c2ocnc2C(F)F)=O)C1 31964,CC(C)CCCC(C)C(=O)N(C1CCN(C(=O)C=CCO)CC1)CC1CCCO1 31965,c1(C(=O)NC2CN(c3ncc4sccc4n3)CC2F)cc(Br)cc2[nH]ccc12 31966,Cc1ncccc1CC(=O)NC1CC(NC(=O)CC2COC(C)(C)C2)C1 31967,C1(OCC(N2CCN(C3CC(C)OC3=O)CC2)=O)CCC(F)(F)CC1 31968,C(CC(CC)C(=O)N1CCN(C(=O)Cc2ccco2)CC1)=CC 31969,C#CC(CC(C)C)NC(=O)CN(C(=O)CSc1cn[nH]c1)CCOC 31970,c1(C(=O)NC2(C(F)F)CC(NC(c3ccc[n+]([O-])c3)=O)C2)cnc2n1CCCC2 31971,c1(C(N2CC3CN(C(c4scc(OC)c4)=O)C3CC2)=O)[nH]cc2c1CCS2(=O)=O 31972,CC(=O)C(C)(C)CC(=O)N1CC=CC1(C)C(=O)N(C1CC(C)(C)C1)C 31973,N1(C(C2(SC)CC2)=O)CC2CC1CC2NC(=O)Cc1c[nH]nc1C 31974,c1(C(=O)NCC(CC=C)NC(c2ccc(F)c(F)c2)=O)ccc(C#N)c(C)n1 31975,c1(C(=O)NCC(CNC(C=Cc2ccc(C)s2)=O)C)ccn2cnc(C)c2c1 31976,C1(NC(C(C)OCCC#C)=O)C2CCN(C(c3sc(Br)cc3C)=O)C12 31977,c1(CC(=O)NCC2N(C(C(CCOC)C)=O)CC=C2)cn2c(C)csc2n1 31978,N1(C(C(C)OCC#C)=O)CCCC1C(C)(C)C(=O)N(C)CCN(C)C(=O)C1CC1 31979,Cc1ccnc(C(=O)NCC(C)(C)CCNC(=O)CN2CCOCC2)c1 31980,N1(C(COC(C)(C)C)=O)CCC(C(C)(O)CNC(c2scnc2C2CC2)=O)CC1 31981,c1(C(N2C(CNC(Cc3ccc(C)cc3)=O)CC(F)C2)=O)cc(N)ccc1C 31982,N1(C(C2CC(=C)C2)=O)CCC(C2CCN(C(=O)C3=CC4CCCC34)CC2)CC1 31983,c1(NC(CC2N(C(C(CC)=O)=O)CCOC2)=O)nc(O)ccc1[N+](=O)[O-] 31984,C1(C(=O)NC(C(=O)N(CCC(=O)OC)C)C2CCCC2)CCC(=O)N1 31985,C1(CC)(CNC(=O)C(Cc2ccoc2)NC(=O)CSCCC#N)CCCC1 31986,C(CC(C(=O)NCCc1csc(C)n1)NC(=O)C=CC1CCCN1C)OC 31987,c1(CCCCC)ccc(C(N2CC(C(C)NC(C3CCOC3CC)=O)C2)=O)o1 31988,N1(C(C(C)OC)=O)CC2CN(C(=O)C(C3CCCCC3)C)CC2(C)C1 31989,CC1(NC(C2CCC(C)(O)CC2)=O)CCN(C(=O)C(O)CC2CCCCC2)CC1 31990,c1(NC23CCC(NC(N4CCC5(CCOC5)C4)=O)(CC2)C3)ncnn2ccc(Br)c12 31991,CC(Cc1nncn1C)N=c1[nH]c2c(c(=NCC3C4CCCCC34)[nH]1)CSC2 31992,c1(C(N(CC(C)N(C(c2cc(C)n(C)n2)=O)C)C)=O)ccc2ccccc2c1O 31993,Cc1cn2c(n1)CC(C(=O)NCCCCCNC(c1ccnc(C)c1O)=O)CC2 31994,C(=O)(C(O)CC1CC1)NC(C1CCCC1)CNC(=O)Cn1cnnn1 31995,c1(C(C)C)ccc(C(CNC(C2CC(C)(C)C2)=O)NC(=O)Cn2ccnn2)cc1 31996,C1(C(=O)Nc2cnc(OCC)c(Cl)c2)COCCC1C1CCNCC1 31997,C(=O)(C(C)S(=O)(=O)C(C)C)N1CCC(NC(c2cc(C)c(OC(F)F)cc2)=O)C1 31998,Cc1cc(C(=O)NCCOc2ccc(F)c(F)c2)c2ccc(Br)cc2n1 31999,C(=O)(CCCCSC)NC(CNC(C(C=C)OC)=O)(C)c1ccccc1 32000,c1(C(=O)NC2(CO)CN(C(CNS(C)(=O)=O)=O)C2)cc(OC)cc2c1OCC2 32001,C(=O)(CC(F)(F)C(F)F)NCC(CC=C)C(=O)N1CC2CC2C1 32002,C1(CCNC(C2CC(C)(F)C2)=O)CCN(C(=O)C(C2CCCO2)C2CC2)CC1 32003,C(=O)(C(C)CC(F)(F)F)NCCCC(C)NC(C1(N2CCOCC2)CCCC1)=O 32004,C#Cc1cncc(C(=O)NC23CC2CN(C(c2ccc(C)nc2C(C)C)=O)C3)c1 32005,C1(C(=O)OC)CCC(OC(=O)CCCSCC(N)=O)CC1 32006,C1(C(C)C)COCCN(C(=O)C(c2ccccc2)NC(=O)C(F)C(F)(F)F)C1 32007,C1(C(N(CCCCCNC(=O)CCCn2ccnc2)C)=O)CC2CCC1C2 32008,C1(NC(C(CC)SC)=O)CCCCC12CCN(c1ncnc(C)c1OC)CC2 32009,N1(C(CSCCOC)=O)CCC=C(C(=O)NC2(CCCN(C)C)CC2)C1 32010,c1(C(=O)NC(C(C)NC(C(COC)C)=O)CO)c(C)ccc(Cl)c1N 32011,c1(C(C(=O)NCCCC2CC2)N(C(C)C)C2CC2)ccc(C(F)F)cc1F 32012,C1(CC(=O)NCC(C)CNC(c2cc(Cl)c(Cl)[nH]2)=O)CCCC(F)(F)C1 32013,CCC1=NOC(CC(=O)NC2CCCC2NC(c2cnc(CC(C)C)[nH]2)=O)C1 32014,c1(N(C)C)cccc(N2CCN(CN3CC(SC(C)(C)C)OCC3)CC2)c1 32015,N1(C(C(CC)C#N)=O)CC(C2CCCN(C(=O)Cc3ccn(C(C)C)n3)C2)C1 32016,CCC(CC(C)C)C(=O)NC(CNC(c1cn(Cc2cccs2)nn1)=O)C1CC1 32017,C1(C(N2CC(C(N3CCC(CCOC)C3)=O)(CC)C2)=O)COCC(C)O1 32018,c1(C(=O)NC2C3CN(C(C4C(C)=CCS4)=O)CC2C3)cc2cccc(C)c2o1 32019,c1(NC(N(CCCC2CCCC2)Cc2ncc(C)o2)=O)cncc([N+](=O)[O-])c1 32020,C(CCCCNC(=O)CCC1(N(C)C)CCC1)N(C(=O)CC1CC1(C)C)C 32021,CC1(C)CCC(C(=O)NCc2ncoc2CNC(=O)CC2CC3CCC2C3)CC1 32022,C=CCN=C(NCC1CCCN1CCOC)N1CCC(C)(OC)C1 32023,C(=O)(C(CCC(C)C)NC(=O)C(=C1CCCCC1)F)NC(C#C)C(C)C 32024,n1(C(=O)NCC23CC(CN2C(=O)COCC2CC2)C3)cc(Br)c(O)nc1=O 32025,n1(CC)nc(C(=O)NCC2(C)CCCN2C(c2c(C)cnn2C)=O)cc1O 32026,Cc1oc(C(C)C)nc1C(=O)N(CC(O)CN(C(=O)C=Cc1ccncn1)C)C 32027,c1(C(N2CCSCC2c2ccc(Cl)cc2)=O)cnc2c[nH]nc2c1 32028,C1(NC(c2ccon2)=O)CCC2CCN(C(=O)C#CC3CCCCO3)C1C2 32029,C(C)(CN=c1cc(C)nc(C(F)(F)F)[nH]1)NC(c1c(CCC)n(C)nc1)=O 32030,C(=O)(C1CCCc2scnc21)NCC1CN(C(CCCCC(=O)NC)=O)CC1C 32031,CCCCCC(C)CC(=O)N1CC(CNC(C2(C)CC3(CCC3)C2)=O)C1 32032,C(=O)(CC1=CCCC1)NCc1c(CNC(C2C(=O)NCC2)=O)cccc1 32033,C(=O)(CC(C)C(=O)NC1C=CC(CNC(C2CC2C(F)F)=O)C1)OC 32034,C1(C=O)CC2(CCN2CC(C)(C)C)C1(C)C.c1(C(C)C)nc(CCO)cs1 32035,C1(CNC(c2ncc(OC)cn2)=O)CC(C(F)(F)F)CCN1C(=O)C(C)O 32036,N1(C(C(CC(C)C)F)=O)CC2CCN(C(c3cnn4ccsc34)=O)CC12 32037,c1(CN(C(CNC(C2C(C)C2)=O)C)C(c2cccc(CF)c2)=O)cccc(Cl)c1 32038,C1(C(N(C(CNC(CC=CC)=O)C)C)=O)CCc2nncn2CC1 32039,C1(C(=O)NCCSCCC=C)C(CNC(=O)CN2CCCC2)C1(C)C 32040,CC1CN(C(c2cc(Br)cnc2O)=O)CC1(C)CNC(=O)C1=COCCC1 32041,c1(CC(=O)NCCC(=O)NCCC(C)C)ccc(F)cc1F 32042,C(=O)(CCC(=O)c1ccc[nH]1)NC(C1CCN(C(COCCOCC)=O)C1)C 32043,N1(C(CC(c2c(C)n[nH]c2C)C)=O)CCN(C(=O)Cc2nnc(O)s2)C(CO)C1 32044,N1(C(c2ncc(C)cn2)=O)CC2CCC1C(CNC(c1ccc(F)c(Cl)c1)=O)C2 32045,N1(C(CC(C)OC)=O)CC2(C1)CN(C(C1CCn3nncc3C1)=O)CCO2 32046,C(=O)(C(C)CC(C)C)NCC(CNC(c1cccc(C(=O)OC)n1)=O)(C)O 32047,CN1C(=O)CC(N2CC(CNC(=O)NCCS(C)(=O)=O)C2)C1=O 32048,c1(C(N2CC(O)CC(NC(=O)C(F)F)C2)=O)ccc2c(c1)CCO2 32049,C=CCCCCCC(=O)N1CCCC1(C(=O)NCC1CN2CCC1C2)COC 32050,c1(NC(N2C(C)CCC(C(=O)OCCOCCO)C2)=O)ccc(S(C)(=O)=O)cc1 32051,c1(CSC(C)C(N2CCCC2CN(C(=O)Cn2cc(Cl)cn2)C)=O)ccccc1 32052,C1(=O)CCCCCNC2C(C)CN1C2.c1(NC(=O)CC2CC(F)C2)ccccc1 32053,N1(C(CCC(C)(F)F)=O)Cc2ccccc2CC1CNC(=O)CCOC1CCC1 32054,c1(C(C)=O)ccc(Cl)cc1NC(C1CCCN(Cc2ccc(Br)[nH]2)C1)=O 32055,c1(C(c2ccccc2)N(CCOC)C)ncccc1S(=O)(=O)NC1CNC1 32056,Cc1ccn(CC(C)(O)C(=O)NC2CC(NC(=O)C(C)(C)N3CCC3)C2)c(=O)c1 32057,CC1CCc2[nH]nc(C(=O)NC34CCCC3CN(C(=O)CCCC(N)=O)C4)c2C1 32058,N1(C(c2c(CC)c[nH]n2)=O)CC=CC(NC(=O)COC)C1 32059,c1(C(N2C3CC(CNC(CC(C)(C)O)=O)C2CC3)=O)ccc2c(n1)CCC2=O 32060,C1(NC(c2c(CC)non2)=O)CC2(C1)CC(C(=O)Nc1ccc(C(C)C)cn1)C2 32061,c1(N2C(c3cn(CCCCCC(=O)OC)nn3)CCC2)ccc(F)c(F)c1O 32062,C1(C(=O)NCC(C)(C)NC(=O)CC2CC(C(F)F)C2)(NC(C)=O)CCCC1 32063,c1(C(N2C(C(=O)NCCOc3ccc(C)cc3)CC(=C)C2)=O)ccc(C#N)cc1 32064,Cc1cc(C(=O)NC(C(N2CCCC(O)(C(N)=O)C2)=O)C2CCCC2)c(O)nn1 32065,C(c1ccncc1)=C(C)C(=O)N(CCCNC(C1CCCCC1C)=O)C 32066,c1(CN2CCCC(CNC(c3ccc(C#C)cc3)=O)C2)ncnc2c1ccn2C 32067,C1(CNC(c2c(CC=C)cccc2)=O)CCN(C(C2CC(F)CN2C)=O)C12CC2 32068,N1(C(COC2CN(C(c3c(C)ocn3)=O)C2)=O)CC2C(CO)C2C1 32069,CC1CN(C(C23CSC(C2)C3)=O)CC(C)C1NC(=O)C=Cc1cnn(C)c1 32070,Cc1csc2nc(CC(N3CC(NC(C4(C(N)=O)CC4)=O)CCC3C)=O)cn12 32071,C1(C(=O)NC(CN(C(=O)CC2(C)CC2)CC)C)COCCN1C=O 32072,c1(C(N2CCC2c2c(F)cccc2F)=O)ccc2ncccc2c1 32073,N1(C(Cn2c(C)nnn2)=O)CC(NC(c2cc(O)nc(Cl)c2)=O)CC(F)C1 32074,c1(N2C(=O)CC2)ccc(NC(=O)C(CNCC2CCC(=O)C2)CC2CC2)cc1 32075,C1(C(=O)NCC2(C)CN(C(=O)Cc3ccc(F)cc3)C2)C2CCC(F)C12 32076,c1(CC)cc(C(N2CCCC(O)(CN(C(=O)C(C)(F)F)C)C2)=O)ccc1O 32077,C(=O)(C1=CC2C=CC1C2)N(CCCCCNC(=O)CCC1CCCOC1)C 32078,N1(C(c2ccc(C(N)=O)o2)=O)CC2(CC(NC(=O)CCc3csnn3)C2)C1 32079,C12(C(=O)NCc3ccc(C)cc3C)C3CCC(CC13)C2(F)F 32080,c1(C(=O)NCCCC(C)NC(c2c(OC)noc2C)=O)ccc2ncsc2c1 32081,c1(SCC)ccc(NC(=O)NCC2(OCC)CCOC2)o1 32082,C1(C)(CC)C=C(C(=O)N2CC3CC3(C(N3CCC(N4CC=CC4)C3)=O)C2)C1 32083,C(CCC(C)C)(C(=O)NOCCCCC)NC(C(C=C=C)C)=O 32084,C1(C(=O)NCC2N(C(CCc3cccc(C)c3)=O)CCOC2)CC(C(C)C)=NO1 32085,CCCCC(C)C(=O)N1CC(NC(c2cccc(F)c2OCC)=O)C(C)C1 32086,c1(C(=O)OC)ncc[nH]c1=NC1CCCC(NC(C2CCOCC2)=O)C1 32087,C1(NC(c2c[nH]nc2-c2ccoc2)=O)COC2(C1)CN(C(=O)CC1CCC1)C2 32088,C(=O)(C(CNC(=O)CC1CSC1)CC(C)C)NC(C#C)(C)C1CCC1 32089,CC1(CCNC(=O)CC2CCC(=O)O2)CCN(C(c2cnoc2C2CCC2)=O)C1 32090,N1(C(c2nc(OC)c(C)s2)C(=O)NCC2CCOC2)CCCC2CCC(C)CC12 32091,C(C(CC(F)(F)F)NC(c1cnc(O)o1)=O)NC(CCC1CCC(=O)NC1)=O 32092,N1(C(CCN(C(c2ccoc2C2CC2)=O)CC)=O)CCCC(CN(C)C)C1 32093,c1(CC)c(C(=O)NCCC2(NC(c3cc(N)ccc3C)=O)CC2)cccc1C 32094,N1(CC(=O)NCCC(C)(C)NC(C(N2CCCCCC2)C)=O)CCCCC1=O 32095,c1(C(=O)NCC2(NC(c3c(CC)nccc3)=O)CC2)cc(O)ccc1C 32096,N1(C(C2NC(=O)CC(C)C2)=O)CC(C(=O)NC(C)(C)C(N)=O)C(C2CC2)C1 32097,c1(COC(=O)NC(c2c(C)sc(Br)n2)C(=O)OC(C)(C)C)cc(F)c(O)c(F)c1 32098,c1(C(=O)NCC(C)C#N)cnc(CNC(C2CC2(Cl)Cl)=O)nc1 32099,c1(C(=O)NCCOCCC#C)ccc(Br)cc1CBr 32100,CC1(C)OCCOC1C(=O)NCCC1CCN(C(=O)CN(C2CCCC2)C)CC1 32101,CCC(C)(C)CCCC(=O)NC1C(C)CN(C(c2cnn(CCF)c2)=O)CC1C 32102,CC(C)(CCCNC(=O)C1CC1)C(=O)NC1CCOC12CCCC2 32103,C(CN=S(C)(C)=O)N(C)C(c1csc(C(=O)OC(C)(C)C)n1)=O 32104,CN1CCC(C2(C(N3CC(CNC(c4ccc(Cl)o4)=O)C3)=O)CC2)CC1 32105,C1(C(N2C(CC(=O)OC)CCC2)=O)CCCN(C(C2CC2(Cl)Cl)=O)C1C 32106,C#Cc1cccc(C(N2CCSCC2C(=O)N(C)C(C)C2CC2)=O)c1 32107,C(=O)(C1=C(C)NC2=NCCCC2=C1)NCC1N(C(COCCCCC)=O)CC1 32108,CCC(CNC(=O)C=Cc1cnccn1)(CC)C(=O)NCCC1CCCC(C)C1 32109,N1(C(C2CN(C(c3n(C)nnc3)=O)CC(F)C2)=O)CCN2CCOCC2C1 32110,c1(CC(=O)N(C2CN(C(c3nonc3N)=O)CC2F)C)cncnc1O 32111,C(=O)(CC(O)C(C)CC)NC1(C(=O)NC(C=C)COC)CC1 32112,c1(CC)ccc(C(=O)NC2CN(C(=O)CSC(F)(F)F)CC2C(F)F)cn1 32113,c1(N2CCC(C)(CO)C2)ccc(S(=O)(=O)NC(CO)C2CCC2)cc1Br 32114,C1(C(=O)NCC23CC2CN(C(=O)CC2CCCCC2)C3)C2CCCCCC12 32115,c1(C(=O)NC(CNC(C(C)=CC)=O)(C)C2CC2)cc(C)c(-c2ccc(Cl)cc2)s1 32116,C1(C(=O)NC(C2CN(C(=O)CCC=CBr)C2)C)(CO)CCCCO1 32117,n1(CCS(C)(=O)=O)ccc(=NC(=O)C2COC(C)(C)C2)[nH]1 32118,c1(C(=O)NCC(C)N(C)C(C(C)C(N2CCCCC2)=O)=O)[nH]ccc1C1CC1 32119,c1(C(C(=O)NCCCCNC(C(SC)SC)=O)F)ccccc1 32120,CC(=O)CCCC(C)C(=O)N1CC(C)CC1C(N1CCC(NC(C)=O)CC1)=O 32121,C(=O)(C(C(C)C)n1cncn1)N(CC(CNC(C(CC)n1cncn1)=O)(C)C)C 32122,C(=O)(C(O)CC(F)F)NCCCN(C(CCc1cnc(C)o1)=O)C 32123,c1(NC(C2CN(C(=O)Cc3ccccc3O)CCC2O)=O)ccc(F)c(Br)c1F 32124,C1(CNC(=O)NC(c2ccc(SC)cc2)C)CCCCC(F)(F)C1 32125,N1(C(c2cc(CCC)[nH]n2)=O)CCC(C)C(NC(c2ncc(N(C)C)cn2)=O)C1 32126,C1(O)(CC(=O)N(C2C(OC)CN(C(CN(C(=O)OC)C)=O)C2)C2CC2)COC(C)(C)C1 32127,C1(C(=O)NC2CCN(c3ccc([N+](=O)[O-])cc3)C2)CCCC2(C1)CC2(F)F 32128,CCCCC(O)C(=O)NCCC(C)NC(=O)C(=O)NCC(F)(F)F 32129,C(C(C)(C)CNC(C1(Cl)CC1(F)F)=O)N(C(=O)CCCc1cccs1)C 32130,c1(C(N2CC(C)(NC(C(C=C=C)C)=O)C2)=O)ccc(C(=O)N(C)C)nc1C 32131,c1(C(C)NC(=O)NCC(C)(C)C(F)F)ccc(-c2ccccc2)c(F)c1 32132,C(C)(CCCNC(=O)C(F)(F)c1nccs1)NC(C(C)NC(C)=O)=O 32133,C12(C(=O)NC(CCCCC)C)CCC(CN(C(c3n[nH]c(C)c3O)=O)C1)C2 32134,Cc1c(C=CC(=O)N(C)CC2CCCN2C(C2CCOCC2)=O)cnn1C 32135,Nc1ccc(-c2cn(CCCNC(c3cnc(C4CC4)o3)=O)nn2)nc1 32136,C1(CNC(c2coc(O)n2)=O)CC(O)CN1C(=O)Cc1ccsn1 32137,C(=O)(CCC(=O)NC1CC1)N(CC(C)N(C(=O)C(Cl)=CCl)C)C 32138,CCC(CC)(CC)C(=O)NC1CC2CC1N(C(C1CC1c1ccccc1Cl)=O)C2 32139,c1(OCCC)c(Cl)cc(NC(c2cnc(OC)c(F)c2)=O)cc1Cl 32140,Cc1c(NS(C)(=O)=O)cccc1N=c1cc(N)nc(-c2ccccc2)[nH]1 32141,CC(C)S(=O)(=O)CC(=O)NCC1(CNC(C2CCCO2)=O)CCC1 32142,c1(C(=O)NCCCC(C)NC(=O)C(C)C#N)cncc(C(=O)OC(C)(C)C)c1 32143,C1(CNC(CCCC=C)=O)CC2CCC1N(C(=O)Cc1cc(C)cs1)C2 32144,C1(CNC(C2CCC(C)(C)C2)=O)(CO)CCN(C(=O)CC2SC(=N)NC2=O)CC1 32145,C1(SCC(=O)NCCN(C(c2cn(C(F)(F)F)cn2)=O)C2CC2)CCOC1=O 32146,c1(CN2CCC(NC(c3cc(Cl)ccc3Cl)=O)C(O)C2)cncc2ccccc12 32147,C1(NC(C(CC(C)C)N(C)C)=O)COC2(C1)CN(C(=O)Cc1ccncc1Cl)C2 32148,CC1(C)CC(C(=O)NCC(O)CC2CCC2)N(C(=O)C=Cc2ccco2)C1 32149,C1(CCNC(=O)Cn2cccc2)CCCN(C(c2sc(Cl)cc2Cl)=O)C1 32150,c1(C(N2CC(CC(C#C)C)C2)=O)cc(F)c(C)cc1Cl 32151,N(C1CCc2ccccc21)C(C12CC(Nc3nccc(Br)n3)(C1)C2)=O 32152,C1(C(=O)NCCCN2CCC2)CCC(NC(C2CCCS2)=O)CC1 32153,C(=O)(C(F)(F)C(C)O)NC(CN(C(c1c(C(=O)OC)nn(C)n1)=O)C)C 32154,Cc1cn2cc(C(=O)NCC3(NC(=O)C(C)N(C)C)CCOCC3)ccc2n1 32155,c1(C(=O)NC23C(CN(C(C(C=C)(C)CC)=O)C2)C3)ccc([N+](=O)[O-])c(N)n1 32156,N1(C(c2ccc(C)cc2)=O)CCCN(C(=O)C(CO)c2ccccc2)C(CO)C1 32157,C1(COC)CN(C(=O)C=C(C)C(C)(C)C)CCN1C(C1CCC12CCC2)=O 32158,C1(C(N2CC(=C)C2)=O)CC(=O)CN1C(=O)CCc1cccn1C 32159,C1(NC(CC(CCC)(C)C)=O)CC(C2CCN(C(=O)C(C)c3ccco3)CC2)C1 32160,C1(N(C(CN(C)CC)=O)C)CCC2CN(C(c3ocnc3C)=O)CC12 32161,C(CC(=O)N(CC(O)CN(C)C(C1CC(CCO)C1)=O)C)OCC(C)C 32162,Cc1csc2c(CC(N3CC(C4(NC(=O)C(C)CN(C)C)CC4)C3)=O)cccc12 32163,CCC(C(=O)N1CC2(CC2)CC1CNC(c1cn(CCCF)nn1)=O)C(C)C 32164,c1(C(N(CC(C)CNC(=O)CCn2cnccc2=O)C)=O)ccc(N)c(Cl)c1O 32165,CCC(C)CCCC(=O)N1CC(NC(=O)CC2CN3CCC2CC3)C(C)C1 32166,Cc1c(C(=O)NC(C)C(CO)NC(=O)C2=NOC(C)(C)C2)nc2sccn12 32167,c1(SCC)ccc([N+](=O)[O-])cc1C(=O)NC1C2CC(C1)N(C(=O)C#CC1(C)CC1)C2 32168,CC1(C)c2ccc(O)cc2CCN1C(C1CCCS(=O)(=O)C1)=O 32169,C1(c2ccccc2)(CC(=O)NCC2CCN2C(=O)Nc2ccccn2)CCCO1 32170,c1(C(=O)NCC(CC)NC(c2cnccn2)=O)nonc1N 32171,Cc1nc2c([nH]1)CC(C(=O)N(C)CCNC(c1ccc(C(C)C)o1)=O)CC2 32172,Cc1ncc(C(N2CCCC2CC(=O)NCc2cnn(C(C)C)c2)=O)c(=N)[nH]1 32173,Cc1ccc(CC(=O)NC(C)CNC(C2CCCC(C)O2)=O)c(Br)c1 32174,Cc1cc(N2CCC(NC(C3CCCC3(C)C)=O)C(F)C2)nc(S(C)(=O)=O)n1 32175,c1(C(=O)NC2CC(CNC(C(C)(O)C3CCC3)=O)C2)cc(Cl)nc(Cl)c1 32176,C=C(C)CC(C(=O)NC1CN(C(C2CC(C)(C)CN2C)=O)C1)OC 32177,c1(C(=O)NCC2CCCN(C(C(C)(C)CC#N)=O)C2)cc(F)cc2nc[nH]c12 32178,C(=O)(C1CCCc2cncn21)NCCCCNC(C(C)N(CC(F)(F)F)C)=O 32179,Cc1nc(C(N2CCC(C(=O)NC(C(=O)OC)C3CC3)C2C)=O)c(C)s1 32180,C#CCC(C)(C(=O)NCC1CNC(=O)C=CC(=O)O1)NC(C)=O.C(C)(C)(C)O 32181,c1(C(=O)NC(C2CCOC2)C)c[nH]nc1CNC(C1CC1c1ccsc1)=O 32182,C1(NC(C)=O)CCCC(NC(c2cc(-c3ccccc3)[nH]n2)=O)CC1 32183,N1(C(C(C=C)O)=O)CC(C(N2C(C(=O)OC)CC2C)=O)CC(C)C1 32184,Cc1coc(C(=O)NC(C)(C)C(C)NC(c2cc(C(C)C)no2)=O)c1C 32185,C1(C(=O)NCC2N(C(C(c3cccc(Cl)c3)CC)=O)CCC2)CCC2CC2C1 32186,CCCCCCCCCCC(=O)NC(C)CN(C(=O)C(c1ccc(Cl)cc1)O)C 32187,c1(C(N2CCC3CCC(C2)N3C(C2CCCO2)=O)=O)cc2cccc(F)c2o1 32188,c1(C(N2CC(N(C(C=CC(C)C)=O)C)C(F)C2)=O)cc2nccn2c(O)n1 32189,C1(CNC(CCC(C)C)=O)CC2CCC(C1)N2C(=O)COCc1cccnc1 32190,c1(C(C(=O)NC2(C=C)CNC2)(F)F)ccccc1Br 32191,c1(C(N2C(C#C)CCC2)C(=O)NC2CC(F)(F)C2)cccc2[nH]ncc12 32192,c1(C(N2CC(CN(C)C(c3n[nH]cc3F)=O)OCC2)=O)cnn2ccn(C)c12 32193,CC1(CNC(c2[nH]ccc2CNC(C2OC3CCC2C3)=O)=O)CCCCO1 32194,CCCCC(CNC(C1CC(OC)(OC)C1)=O)NC(=O)CC1CCC(=O)N1C 32195,C1(CNC(=O)CCC2CCC(=O)N2)CN(C(C2CC2(F)F)=O)CCC12CCC2 32196,c1(C(=O)NCC2(COC)CN(C(=O)C(C(C)C)NC(N)=O)C2)cncc(N)c1 32197,c1(CC(=O)N(CC(CNC(C(C)n2ccnc2)=O)F)C2CC2)cccc2cn[nH]c12 32198,CC1(C)C(C(=O)NCC(P(C)(C)=O)c2ccccc2)(CO)C1(C)C 32199,C(=O)(C#CC(=O)NCC1(F)CN(C(=O)C=Cc2cncn2C)C1)N(C)C 32200,C1(CN(C(CC(C)C2CCCO2)=O)C)CCN(C(=O)C(C)(C)n2ccnn2)CC1 32201,c1(C(N2C(C)CN(C(CNC(C)=O)=O)C(C)C2)=O)ncnc2c1ccn2C1CC1 32202,c1(-c2cc(C)cc(OC)c2F)cccc2[nH]nc(C(=O)Nc3conc3C)c12 32203,Cn1ccc(S(=O)(=O)NCC(C(=O)O)NCCC(C)(C)N2CCOCC2)c1 32204,C#CCCCC(C)C(=O)N(C1CC(C#N)C1)CC(=O)NCC1CCC(=O)NC1 32205,N1(C(C2C3CN(C)CC32)=O)CCC2C(CCN2C(c2ccc(F)cc2Cl)=O)C1 32206,C1(NC(C(C)OC)=O)CCN(C(c2cnc(-c3ccccn3)nc2)=O)CC1O 32207,N1(C(C(c2n(C)cnc2)O)=O)CCN(C(c2cocn2)=O)C(CO)C1 32208,c1(OC)cc(C)cc(C(=O)NCC2CC(O)CN2C(=O)CC(=O)N(C)C)c1C 32209,c1(C(=O)NC2CC3(CC(CNC(C(CC#C)(C)C)=O)C3)C2)cc(C)c(C)nc1C 32210,c1(C(N2CC(CC(=O)NOCC(C)C)(OC)C2)=O)sc(O)nc1C 32211,c1(OC)nccc(C(=O)NC23CC(CNC(=O)C(CCSC)NC(N)=O)(C2)C3)n1 32212,C1(CNC(C2CCN(CC)CC2)=O)CC2(C1)CN(C(=O)C=CC(=O)NC1CC1)C2 32213,Cc1c(C(=O)NC2COCCN(C(C3CCC(=O)N3)=O)C2)cccc1F 32214,N1(C(C(CNC(=O)COC2CCOCC2)O)=O)CCC2(CC1)CSC2 32215,C12(NC3CCN(c4ccccc4)C3)CC(CO)C(CO1)C2 32216,c1(CC)nc(C(C)NC(=O)C(F)N(C(C2(C(=O)NC)CC2C)=O)CC)n[nH]1 32217,C1(OC)CC2CC(C(=O)NC3CC(CNC(c4ccc(CN(C)C)o4)=O)C3)CC12 32218,C1(CNC(c2ccc(OC)cn2)=O)(OC)CCN(C(C2CCCS2)=O)CC1 32219,Cc1nc(N(C)CCN(C)C)cc(N2CCOC(Cn3ccnc3C)C2)n1 32220,C(=O)(C1=C(C(=O)OC)C(c2ccc3cnccn23)NC(=O)N1C1CC1)OC 32221,N1(C(C2N(C)CC(O)C2)=O)CCOCCC1C(=O)NCCCN=[N+]=[N-] 32222,c1(C(c2nnnn2CSc2ccccc2)NCC(COC)C)sc(C)c(Br)c1C 32223,c1(OC)cnc(NC(C2CC23CN(Cc2cc(C)[nH]c2C)C3)=O)c(F)c1 32224,N1(C(C2(COCC)CCOCC2)=O)CCN(C(=O)C(C)n2ccnc2)CC12CC2.NO.C 32225,C(=O)(C1=NOC2COCC12)N1C2C(C(N3CCC(CCO)CC3)=O)C(C2)C1 32226,C(CC(=O)N1CCN(C2CCC2)CC1)(C(C)OC)NC(C(COC)COC)=O 32227,N1(C(C2C(C=C)C2)=O)CCC(O)C(NC(=O)Cc2csc(-c3ncccn3)n2)C1 32228,CC(CC(N)=O)C(=O)NCC(C)(C)CCNC(C1CC(=O)N(c2nccs2)C1)=O 32229,Cc1cc(F)sc1C(=O)NC1(c2ccccc2)CCN(C(C2CNC(=O)C2)=O)C1 32230,N1(C(C(C)CN(C)C(C2CC2C(F)F)=O)=O)Cc2ccnn2CC1C 32231,Cc1ccc(N(CCCNC(=O)C2=CC3CCCC23)C(C)C)c([N+](=O)[O-])c1 32232,CN1CCC(C)(C(=O)NCCC2(CNC(=O)C(F)CC3CCCCC3)CC2)C1 32233,C=C(C)CC(C(=O)N(C(CC)C(=O)NC1(C)CCC(C)C1)C)NC(C)=O 32234,c1(CC(=O)NCC2CCCC2NC(c2cccc(F)c2O)=O)cc(Cl)ccc1Cl 32235,CC1CN(c2nc(C3CCOCC3)ns2)CCC1NC(c1ccnc(O)c1)=O 32236,c1(C(=O)NC(C2CCN(C(C3C(CC)C3)=O)C2)C)ccc(Cl)nc1 32237,N#CC1CCCC(CC(=O)N(C2CCCCCC2)CCC23CC(CO2)C3)C1 32238,C1(CNC(C(C)OCCCC)=O)CCCCN(C(=O)CC2(CSC)CC2)C1 32239,N1(C(C2CCN(C)C(=O)C2)=O)CC2(CCN(C(c3[nH]ccc3C3CC3)=O)CC2)C1 32240,CCC(C(=O)N(CC(C)NC(=O)Cc1cccc(C)c1F)CC)C(C)(F)F 32241,C1(C(=O)NCC(C)NC(=O)CC2(CO)CC2)CC2C(C1)C2(C)C.C(C)(C)(C)OC(=O)N 32242,C1(NC(CN(CCOC)C)=O)CN(C(=O)C(c2ccc(Cl)cc2)C)CC12CC2 32243,N1(C(c2cn[nH]c2)=O)CCCC(C2CN(C(C3COCCC3(F)F)=O)C2)C1 32244,C(CC(C)C)(C(=O)N1CC(N2CC(NC(=O)CC3(CSC)CC3)CC2=O)C1)OC 32245,c1(C(=O)NC2(C)CCN(C(c3ccon3)=O)C2)cncc(N=[N+]=[N-])c1 32246,N1C2CCC1CN(C(=O)C(=O)NCC)CC2.c1(N(C)S(N)(=O)=O)ccc(N)cc1 32247,C(=O)(N=c1[nH]nc(Br)s1)NC1CCCN(C(c2nc(CN(C)C)no2)C)C1 32248,C1(CCNC(CCN(C)CC)=O)CCCCN1C(c1ocnc1C1CC1)=O 32249,c1(C(=O)NC2C(NC(CC3OCC(C)(C)OC3)=O)C2)ccc(Cl)c(Cl)c1O 32250,c1(C(N2CCCC(N(C(c3cnco3)=O)CC)C2)=O)cnn2cccc(Cl)c12 32251,c1(C(=O)NCC2(NC(C(CC)NC(N)=O)=O)CCCCC2)cn2cnnc2cn1 32252,n1(CC)cc(Cl)c(C(=O)NCC2(OC)CCN(C(=O)Cc3cnn(C)c3)C2)n1 32253,C#CC1CC1C(=O)NC1CC(N(C(=O)CC2CCN2C(=O)OC(C)(C)C)C)C1 32254,N1(C(c2c(C)nsc2)=O)CC2(CC(C(=O)NCC(C)(O)C3(C)CC3)CO2)C1 32255,c1(C(N2CCN(C(C(C)N(CC)CC)=O)CC2C(F)F)=O)nc(O)nc(O)c1F 32256,CC(C)(C)CC(F)C(=O)NCC(C)(CO)NC(=O)CN1CCCC(CO)C1 32257,CC1(C(N2CC(C3CCCO3)C2)=O)CN(C(C2CCC(=O)C2)=O)C1 32258,Cc1cc(C(C)C)ccc1C(=O)NC1C2CC1N(C(c1cncnc1C)=O)C2 32259,N1(C(c2cc(C(C)C)on2)C(=O)NCCOC)CCC2CC12C(=O)OC.C=C(C)CN 32260,c1(CC(=O)NC2CC(NC(c3ccnnc3O)=O)C2)cc(F)cc(F)c1Br 32261,N1(C(CC(C=C)(C)C)=O)C(C)CC2CN(C(C3COCC(C)O3)=O)CC12 32262,C(C(F)(F)CCC(=O)NC(C(C)O)C(F)(F)F)n1cc(-c2cc(C)[nH]n2)nn1 32263,Cc1c(S(N)(=O)=O)cnc(NCCCc2ccc(Br)cc2)c1Br 32264,c1(C(=O)NC(CCCC)CNC(c2cc(OC)cnn2)=O)c(F)cc(F)cc1Cl 32265,c1(C(=O)NCC(C)CNC(=O)C(C)NS(C)(=O)=O)cccc2cncn12 32266,C1(C(=O)NC(C#C)C2CC2)C2CC3C(C2NC(=O)CCCCN(C)C)C13 32267,c1(CC(C(=O)OC)Nn2cc(C3CCCCC3)nn2)ccc(OC(F)F)cc1 32268,c1(CN2CC(NC(c3c(C)ccc(Br)c3)=O)C(C#N)C2)ccc2nc[nH]c2c1 32269,C(C(=O)Nc1cncnc1C)(C(C)(C)C)NC(CCSCCCC)=O 32270,N1(C(COc2cccc(OC)c2)=O)CC2CC(NC(=O)C(C#N)C(C)C)C(C2)C1 32271,c1(C(N(C(C)C)CCNC(c2cc[nH]c2)=O)=O)nccc2ccn(C)c12 32272,C1(NC(C=C(C)Cl)=O)CN(C(c2snnc2C)=O)CC1C 32273,C1(CCC)CN(C(C2C(C)C2C)=O)CC1C(=O)NCCC(=O)OCC 32274,N1(C(C(CCCC)O)=O)CCN(C(C2CC(OC)C2)=O)C2(CCC2)C1 32275,C1(C)(C(=O)NCC(=C2CN(C(CCCOC(C)C)=O)C2)F)CCCS1(=O)=O 32276,C1(C(=O)NC2(C)CC(NC(=O)CC3CC3(Cl)Cl)C2)COCCN1CC(F)F 32277,c1(C(N2C(C(N(C(=O)Cc3cnccc3C)CC)CC)CCC2)=O)cnc(C)nc1 32278,CC1CC2CC1CN(Cc1ccc(OCCCl)cc1)C2 32279,N1(C(C2N(C(C(COC(C)=O)C)=O)CCC2C)=O)CC2(CCN(C)CC2)C1 32280,C1(C(=O)NCc2ccc(CN(C(C(C)C#N)=O)C)cc2)CC2(CC(=O)N2)C1 32281,O=C1C=C2CN(C(=O)CC3CN(C(c4n[nH]cc4I)=O)CCO3)CCC2S1 32282,C1(CCNC(=O)CCCN2CCCC2)CC(F)(F)CN1C(=O)Cn1cnnc1 32283,c1(C(C(=O)N(CCNC(C(C)n2cccn2)=O)C2CC2)C)ccnn1C 32284,C(c1cnc2ccccc2n1)=CC(N1CCC(CC)(NC(C2CC2C)=O)CC1)=O 32285,S(=O)(=O)(c1ccc(NC2CCOC(C(C)C)C2)cc1Br)NCC(C)(C)OC(C)C 32286,c1(C(N2CCCC(CN(C(C(C(=C)Cl)(C)C)=O)C)C2)=O)cn2cc(C)ccc2n1 32287,C12CCCCN1C2=O.CCCCCCN(CCC(C)C)C(=O)OC(C)(C)C 32288,c1(C(=O)Nc2n[nH]cc2C(=O)O)ccc(-c2ccccc2)c(F)c1 32289,C1(CNC(CC=C(C)C)=O)CC2(CCN(C(c3cn(C(C)C)cc3C)=O)C2)CO1 32290,CCC(C(C)(C)O)NC(c1cnn(CCNC(C2CCC(=O)C2)=O)c1)=O 32291,C(=O)(CCCCC(N)=O)NC(C(=O)NC1CCCN(C)C1)CO 32292,C(N=c1[nH]c(=NCCSCC)[nH]c2cc[nH]c12)C1N(CCC)CCCC1 32293,C#Cc1ccnc(C(N2CCN(C(=O)C(CC)CC=C)C(C(C)(C)C)C2)=O)c1 32294,C1(F)(CNC(C(CCCC)C)=O)CCCN(C(=O)Cc2ccc3occc3c2)CC1 32295,CC1(C)CC(CNC(=O)C(F)=C2CCC2)N(C(=O)CC2CC3CC3C2)C1 32296,C(=O)(CCC(C)S(C)(=O)=O)NC(CNC(c1c(C)nn(C2CC2)c1Cl)=O)C1CC1 32297,CCC(C)C(C(=O)NCC1(C(N2CCC(O)CC2)=O)CCCO1)N(C)C 32298,c1(C(N2CC(O)(CCNC(CC(=C=C)C)=O)C2)=O)cnc2scc(C)n2c1=O 32299,CC(c1ccccc1Cl)=CC(=O)NC1CC(NC(c2cc(C)nc(C)n2)=O)C1 32300,Cc1ccc(O)c(C(=O)NCCNC(=O)CCc2ccn(C)n2)n1 32301,c1(C(N2CC(=O)NC2)=O)cc2n(n1)CCCN(Cc1cc(F)ccc1[N+](=O)[O-])C2 32302,N1(C(C(C)OCC=C)=O)CC(COC)(NC(=O)CC(C)OC)C1 32303,c1(C(C(=O)NCCCSC)N(CC=C)CC#N)nn(NC(C)=O)nc1C 32304,N1(C(c2ccc(CCC)[nH]2)=O)CC(NC(c2cccc(N)c2)=O)CC1(C)COC 32305,C1(C(=O)OC)C2CC1N(C(=O)C(C1CCN(C(=O)C(C)(C)Cl)C1)F)C2 32306,c1(NCC(CC)CO)nc(N2CC(C(F)(F)F)C(C)C2)nc2c1ncn2C(C)C 32307,N1(CC)CC(C(=O)NC2CN(C(c3ccnc(NC4CCC4)c3)=O)C2)NC1=O 32308,C(CCCCCC(=O)NC1CC(CC(=O)OC)C1)n1cc(-c2c(C)ncs2)nn1 32309,N1(C(COC)=O)CCCC2(NC(c3ncc(C(F)(F)F)s3)=O)CC2C1 32310,C(CC(=O)NOCCC(C)O)(C(F)(F)F)NC(C1(COCC)CC1)=O 32311,c1(C(N2CCC(C)(NC(c3nc(C)c(C)[nH]3)=O)CC2)=O)cnc(O)c2ccsc12 32312,C(CC(C(=O)NC1(CO)CCC1)NC(=O)Cc1ccc(C)s1)=CC 32313,c1(C(=O)NCC2=CCN(C(C3CC=CC(O)C3)=O)CC2)cccc2ccoc12 32314,C(CNC(c1cc(OC)cs1)=O)(CCC)NC(C(C)=C(CC)C)=O 32315,C12(C(N(CCN(C)C(C3(n4ccnn4)CC3)=O)C)=O)CC(C1)C(C)(C)O2 32316,C1(F)(C(=O)NCC2CC(NC(CSc3n(C(C)(C)C)cnn3)=O)C2)CCCCC1 32317,N1(C2CN(C(CCC3(C)CN(C(C(C)N(C)C)=O)C3)=O)C2)CC2(CCOCC2)C1 32318,O=C1CN(Cc2ccnc(F)c2)C(=O)N1CCOc1cccnc1 32319,N1(C(C2CC(=O)N2)=O)CCC(C2CCCN(C(c3ccn(O)c(=O)c3)=O)C2)C1 32320,Cc1cnc(N(C23CC(N)(C2)C3)C(C23CCC(CC2)CC3)=O)nc1C 32321,C(=O)(CCCCCF)NC1(C)CN(C(=O)CC2CCCC(C(F)(F)F)C2)C1 32322,C1(CCN)CCCN1N(C)CCCC1CC1 32323,N1(C(c2cc(CCC)[nH]n2)=O)CCCC(N2CCN(C(C3CCOC3)=O)CC2)C1 32324,Cc1ccnc(C(C)(C)C(=O)NC(C)CN(C(=O)C(F)OC(F)(F)F)C)c1 32325,N1(C(c2c(C)c(F)ccc2)=O)CCCC2CN(C(=O)C3=CCCS3)CCCC12 32326,C#CCCCCC(=O)NC1CC1CNC(c1ccc[n+]([O-])c1)=O 32327,c1(CN(C(=O)C=CC2CC2)C)cccc(O)c1 32328,N1(C(C(OCC)OCC)=O)CCC(C(=O)NC2CCC2C(F)(F)F)C(O)C1 32329,C(=O)(CCC(C)(C)N(C)C)NC(CC)CC(=O)NCC1CCC(C2CC2)O1 32330,C1(C=O)CCCN1N(C)C.N1(CCN(C=O)C)CCCC1=O 32331,c1(C(N2C(C)CC(NC(=O)COc3ccsc3)C2)=O)cc(F)cc2nc[nH]c12 32332,CN1CCCC1C=CC(=O)NCC1(O)CCN(C(c2cscn2)=O)C1 32333,c1(-n2c(C(c3ccccn3)NC3CSC3)nnn2)ccc2c(c1)CCC2 32334,C1(C(N(C2CN(C)C2)C)=O)CC12CCN(C(c1cscc1Cl)=O)CC2 32335,C(=O)(CCCCCC#N)NCc1ccc(C(N2CCC(C#CC)C2)=O)cc1 32336,N1(C(C(Cn2ccnn2)NC(CCCOC)=O)=O)CC2C(C1)C2(C)C 32337,c1(C(N2CCCCC(CNC(C(=O)NCC)=O)C2)=O)cc(C)nc2ccnn12 32338,N1(C(Cc2c(C)ccs2)=O)CC(C2CN(C(c3cc4ncccc4s3)=O)C2)C1 32339,C12(C(=O)NC(COC)CO)CC1CN(C(=O)C(C)=NOCC#N)C2 32340,c1(C(N2CCCC(N(C(=O)C(F)C(F)(F)F)CC)C2)=O)cc(C)nc(Cl)c1N 32341,C1(C(=O)NC2(CC)CN(C(=O)Cc3cn(C)nc3C)C2)CCCCN1N=O 32342,C1(C)(C(N(C2CC(C#N)C2)CC(=O)NCCCC2(C)CC2)=O)CCOC1 32343,C(C(O)C(=O)NC1CCC1CNC(=O)C(=O)NCCCC)=CC 32344,Clc1ccc(CCCCN(c2ccccc2)c2ccccn2)cc1Cl 32345,C(CC(=O)NOC1CCC1)C1CC(NC(C2C(C)C2)=O)C1 32346,C1(O)(CNC(CCc2onc(CC)n2)=O)CCN(C(c2snnc2C2CC2)=O)C1 32347,N1(C(C(C(=C)Cl)(C)C)=O)C2CCCC1CN(C(C1COCCC1C)=O)C2 32348,CCCCC(C)C(=O)N1CCN(C(c2cc(CC)no2)=O)C(C(C)C)C1 32349,N1(C(C(C)(C)NC(C)=O)=O)CC2(C(=O)NCC(F)Cl)CC1CO2 32350,c1(SC)nc(N2CCC(NC(=O)C=C3CCSCC3)C(F)C2)cc(C(F)F)n1 32351,C(=O)(C1=COCCC1)N(C)CC1CCN(C(c2c(C)n[nH]c2)=O)C1 32352,N1(C(C=CC=CC)=O)CC(NC(C2(COC)C=CCC2)=O)C(O)C1 32353,C1(NC(N(C(C)C)C)=O)CCC(C(C)O)CC1.C1(C)C(=O)O1 32354,Cc1cnc(C)c(C(=O)NCC2CCCN2C(=O)CCCNS(C)(=O)=O)c1 32355,c1(-c2nc(-c3scc(C)n3)nn2C2CCOC2C)cc(Cl)ncc1Cl 32356,C1(CNC(CC(CCC)CC)=O)CCCC2(CN(C(c3ccnnc3)=O)C2)O1 32357,c1(OC)ccoc1CNC1CC(C(N2CCCC2C2CCCC2)=O)C1 32358,C12(NC(Cn3c(C)ccn3)=O)CCC1CN(C(c1cc(O)nc(C3CC3)n1)=O)C2 32359,S(=O)(=O)(C1COC(C)(C)C1)NCC1(NC(NOCCOCC)=O)CC1 32360,CCN=C(NCc1ccccc1C(C)(F)F)NC1CCN(C2COCC2O)CC1 32361,C12(NC(CC3(OCC)CCC3)=O)CC1CN(C(=O)CSCCc1ccccc1)C2 32362,O=C(N=c1cc(C2CCCC2)[nH][nH]1)C1CCOC(c2ccccc2)C1 32363,N1(C(C(=O)NCC)=O)CC(CNC(C2CCC(N(C)C)CC2)=O)C(O)C1 32364,C12(C(=O)NC(CC=C)CC(F)F)CCCCC1C2(F)F 32365,Cc1cc(C(=O)NCC(O)CN(C(=O)C(C)C(=O)N2CCOCC2)C)sc1C 32366,C1(N(C)C(c2cncc(C(F)(F)F)c2)=O)CC2CC1N(C(C1CS(=O)(=O)C1)=O)C2 32367,c1(CSCC(=O)N(CC(C)(C)NC(C2C(OCC)CC2)=O)C)ccccc1Cl 32368,N1(C(c2ccc(C(N)=O)nc2)=O)CCN(C(=O)C2=CCSC2)C2CCCCC12 32369,N1(C(C2N(C(c3c(C)oc(CO)c3)=O)CC(=O)NC2)=O)CCOC2(CCC2)C1 32370,C#Cc1ccc(C(=O)NC(C)C(C(C)C)NC(=O)CN(C)CCC)c(F)c1Cl 32371,C1(CNC(C2(COC)CCC2)=O)CCC(C)(C)CN1C(c1ccc(C)nc1)=O 32372,C(C1=NOC2CC12)NCC1CC(NC(=O)OC(C)(C)C)C1 32373,C(=O)(C1Cc2ccccc21)N(C1CCN(C(C2(Cl)CC2(F)F)=O)CC1)C 32374,Nc1[nH]c(=O)c(Cl)nc1C(=O)N(CCCNC(C1CC(O)C(F)C1)=O)C1CC1 32375,Cc1nc(C(=O)NC2C=CC(CNC(=O)CSC(C)C)C2)c2ccnc-2[nH]1 32376,N1(C(C(C2CN(C(C3CC=C(C)CC3)=O)C2)O)=O)CCC(C)(O)C(O)C1 32377,N#Cc1cnccc1-c1cnc(C(F)(F)F)cc1C(=O)Nc1cc(O)nc(O)n1 32378,CC(CF)CC(=O)NCC1CN(C(c2cnn(-c3cccc(F)c3)c2)=O)C1 32379,n1(CC)ccnc1C(=O)NCCC1CN(C(=O)CC2(c3ccccc3)CC2)C1 32380,C1(CC(C)C)C(=O)N1.C1(NC(C(C)C)=O)CN(Cc2ccccc2)CC1C#N 32381,N1(C(=O)Nc2cccc(-c3nccc(C)n3)c2)Cc2c(F)cccc2C(C)(C)C1 32382,C12(NC(=O)CC3COCCOC3)CCCC1CN(C(c1cc(O)nc(O)n1)=O)C2 32383,CC1CCCCN1CC(=O)NCC1CCCC1C(N1CC2CC2(CO)C1)=O 32384,C=CCC(CC)C(=O)N1CCCC(N2CCNCC2)C1=O.C1CC(C2CC2)CN1 32385,Cc1cc(C(N2CCC(C)(CCNC(C3CC4CC3C4)=O)CC2)=O)ccc1O 32386,C12(C(N3CCC(O)(C(C)NC(C(=C(C)C4CC4)F)=O)C3)=O)CC3CC1C2C3O 32387,c1(CNC(CN(C(C2CC2C2(C)COC2)=O)CC)=O)nc(C)cc(C)n1 32388,c1(C(C(=O)NC(C(C)C)CNC(c2nnsc2C(F)F)=O)C)cc(F)cc(F)c1 32389,N1(C(C2N(C)C(=O)CC2)=O)CCCN(C(=O)C2=CCOCC2)CCC1 32390,c1(C(=O)NCC(CNC(C=CCOC)=O)OC)cn2ccnc2cn1 32391,N1(C(C(C)OC)=O)CCCC(N(C)C(c2ccc(-n3cncn3)cc2)=O)C1 32392,c1(CNC(C2CC(=O)NCC2)=O)ccc2c(c1)CN(C(=O)COC1CCC1)C2 32393,c1(C(=O)NCC(CNC(C(C2CCCOC2)OC)=O)C)c(F)ccc(F)c1F 32394,c1(C(=O)NC2(C)CN(C(c3c(O)cc(C)nn3)=O)C2)cc(F)cc2nccnc12 32395,c1(CC)ccc(CNC(c2cc(C)no2)c2nnnn2CCOCC2CC2)nc1 32396,C1(C)(CN(C)C)CCN(C(C2CCC(NC(=O)C(C)(C)F)CC2)=O)C1 32397,C1(N(c2ccc3occc3c2)C(CCC#C)=O)CCCC12CCNCC2 32398,c1(C(=O)NCC(CNC(C2(COC)CCOCC2)=O)C)nc(C)ccc1OC 32399,C1(NC(Cc2c(C)n(C)cn2)=O)C2CC3C1C3C2C(=O)NC1C(O)C2CCOC12 32400,C(=O)(C(Cc1ccc(O)cc1)C(F)(F)F)NCCCC(C)NC(C(C)=CCC)=O 32401,C(=O)(C1=CCCOC1)NCC1CC(NC(C2CC(OCC)C2)=O)C1 32402,Cc1cc(C(=O)Nc2nc(C(=O)Nc3c(Cl)cnn3C)cs2)cnc1O 32403,CC1C(C(=O)NC2CCN(C(=O)C=Cc3cnc[nH]3)C2)OC2CCCCC12 32404,CC(=O)CCCC(=O)NC12CCC(C1)N(C(=O)C(C(C)(C)C)OC(C)(C)C)C2 32405,C1(C(N2C(CNC(=O)C(=O)NC3CC3)C(O)C(O)C2)=O)CCCC(F)(F)CC1 32406,CCC(F)(F)C(C)(C)C(=O)N1CCC(C(C)NC(C2(C#N)CC3CC3C2)=O)C1 32407,c1(C(N2C3CCC(NC(c4cnc(Cl)s4)=O)C(C3)C2)=O)cnc(O)c([N+](=O)[O-])c1 32408,C(=O)(CCNC(c1cnsc1)=O)NC1C(C)C1 32409,c1(NC(C(CCCC)NC(=O)C(F)CC2CCOC2)=O)ccc2c(c1)CCC2 32410,CC(C(C)CO)NC(c1ccccc1)C1CC1c1ccc(Br)s1 32411,Cc1cc(NC(=O)CC2CCN(C(c3cc(Cl)ccc3O)=O)C2)nc(Cl)c1 32412,N1(C(C(C)N=[N+]=[N-])=O)CC(NC(c2ccc3nc(O)[nH]c3n2)=O)C(S(C)(=O)=O)C1 32413,c1(OC)ccc(CC(=O)NCC2(NC(=O)CCc3cc(Cl)no3)CC2)cc1 32414,c1(C(N2CC(NC(C3(OC)CCCOC3)=O)C2)=O)cc2c(C)c(F)ccc2[nH]1 32415,Cc1cn2ccc(C(=O)NC3CC(CNC(C4CC4(F)Cl)=O)C3)cc2n1 32416,N1(C(C2(C)CC2(F)F)=O)CCC2(CCN(C(c3cnc(NC4CC4)s3)=O)C2)C1 32417,N1(C(c2c(C(C)C)nns2)=O)CCCCC1CCN(C)C(C1COCCO1)=O 32418,c1(OC)cc(NC(C2CC2NCc2ccnc(-c3ccccc3)c2)=O)c(C)cn1 32419,N1(C(C)(C)C(=O)NCCc2nnc3n2CCNC3)C(=O)c2ccccc2C1=O 32420,c1(OC)ccc2c(c1)C(=O)CCN2C(=O)Cc1c(C)nc(C)nc1O 32421,N1(C(C(CC)n2cncn2)=O)C2CCC1CN(C(=O)C=CC1(C)CCOCC1)C2 32422,C1(COC)CN(C(=O)CCc2cnc(O)[nH]2)CCN1C(=O)CS(C)(=O)=O 32423,C(=O)(CN=c1[nH]c(C)cs1)NCC1CN(C(C(C)OC)=O)CC1C 32424,c1(C(N2CC(O)(CCNC(C3(F)CCOC3)=O)C2)=O)cc(F)ccc1Br 32425,C1(CNC(C2ON=C(C)C2)=O)C(C)CCCN1C(=O)CCC(C)C 32426,N1(C(c2c(C)cc(CNC(C3CC34CCCC4)=O)o2)=O)CCCC2C(=O)NCC12 32427,N1(C(C(C)OCCC(C)C)=O)CCCN(C(=O)C=Cc2cnc[nH]2)CCC1 32428,C1(C(N2CCC(O)(CNC(=O)CC3(C)CCOCC3)C2)=O)(COC)CC=CCC1 32429,C1(CC(=O)N(CCC)CCNC(=O)C2=C(Cl)CC2)CSc2ccccc2O1 32430,C1(NC(CC(C)C(F)F)=O)COC2(C1)CN(C(C1CC=CC1)=O)C2 32431,N1(C(=O)NCC(C)OCC=C)CC(c2ccc(Br)cc2)C(C)(C)C1 32432,c1(CC)nc(Cl)nc(N2CCC(NC(C3CCC(NC(C)=O)CC3)=O)CC2)c1Cl 32433,N1(C(Cc2ccn(C(C)C)n2)=O)CCC(C)C1CNC(=O)CC(C)C1CC1 32434,c1(C(=O)NCC2(CC(=O)Nc3cncc(CO)c3)CC2)c[nH]ccc1=O 32435,CC(C)CC(C)(CNC(C1CC12CCCC2)=O)NC(=O)C=C(Br)Br 32436,n1(CC)nc(C)c(C(=O)OC)c1C.n12nnnc1C(C(C)(C)C)NCC2 32437,O=S(=O)(c1ccc(F)c(Br)c1F)Nc1cccc(-c2ccccc2)c1 32438,C#CCC(CO)NC(C1(CNC(=O)CCOC2CC2)CCC1)=O 32439,C1(C(=O)NC2CCN(CC)CC2)CC2(C1)CN(C(=O)CC1CC(C)=NO1)C2 32440,C(CC(O)C(=O)NCC1CCN(C(=O)CSc2cccc(F)c2)C1)SC 32441,C1(NC(c2ccc(C(C)C)cc2O)=O)CN(C(=O)CCS(C)=O)C2(CCC2)C1 32442,c1(OC)cc(C(=O)NC(C)CCN(C(=O)CC2CNC(=O)C2)C)cc(Cl)c1 32443,c1(OC)cc(F)cc2cc(C(=O)NCC(C)(N)CO)[nH]c12 32444,C12(CNC(C(CC=C)NC(C)=O)=O)CCC(CC1)N2C(=O)C(F)(F)COC 32445,c1(C(C(=O)Nc2ccc(OC)cc2)N(C2CCOCC2C)C)cc(C)ccc1Br 32446,c1(OCC(=O)NC2CC(N(C(C3(O)CN(C)C3)=O)C)C2)cccc(NC(N)=O)c1 32447,CC(C)C(C)C(=O)NCC(C1CC1)NC(c1ccc(OC(F)(F)F)cn1)=O 32448,N1(CC(=O)NCCCN(C(C2C(C)COCC2)=O)C)CCCc2sccc2C1=O 32449,c1(C(N2CCCC(CC(=O)OC)C2)C2CC2)cccc(C(F)(F)F)c1F 32450,CC1=C(C)CC(C(=O)NCCC2(C(=O)NC3CNC(=O)C3(C)C)CC2)CC1 32451,NS(=O)(=O)c1ccsc1C(N1CC(O)(CCNC(=O)CC2COCCO2)C1)=O 32452,c1(CC(=O)NC(CC)CN(C(=O)C=CS(C)=O)CC)c[nH]c2ccc(C)cc12 32453,CCC(C)(C)C(O)C(=O)N1CC(C2(NC(=O)C(C)CSC(F)(F)F)CC2)C1 32454,CCC(CC(=O)N1CCC(C)(NC(=O)CCCNC(=O)OC)C1)OC 32455,C1(C(C)NC(C2CCN2S(C)(=O)=O)=O)CCN(C(C2(O)CC2)=O)C1 32456,C(=O)(C(C)(C)CCC)NCC(=O)N(CCCNCC(=O)OCC)C1CC1.C(C)(C)C 32457,N1(C(C2(C)CN(Cc3ccc(C)nc3)C2)=O)CCC2SC(=O)C=C2C1 32458,c1(C(N2C(C)CC(CCNC(c3ccnn3C)=O)CC2)=O)cccc2c1CCO2 32459,Cc1cc(S(N)(=O)=O)cc(C(=O)N(C(C)CNC(=O)CCCCC#N)C)c1C 32460,N1(C(C2CC(O)CN2Cc2cccc3c2OCC3)=O)Cc2cccc(Br)c2C1 32461,Cc1ccc(C2(C(N3CCCC(N(C(=O)C(C)N4CCC4)C)C3)=O)CCC2)cc1 32462,C(=O)(N=c1[nH]sc2c(Br)cccc12)NC1(C(F)(F)F)CCC(=O)NC1=O 32463,CCC(F)(F)CC(=O)N1CCCC(NC(=O)CCCn2cccn2)C1C 32464,c1(-c2[nH]c(=N)sc2)ccc(C(=O)NCC2(NC(C3CCOC3C)=O)CCC2)cc1 32465,c1(CC(=O)NCC2N(c3c(F)cnc(C)n3)CCOC2)cc(F)ccc1[N+](=O)[O-] 32466,CCN=c1ccc(C(=O)NC2CC2NC(c2ccc(C(F)(F)F)s2)=O)c[nH]1 32467,N1(C(C2CCN(C(c3cc(OCC)c(Cl)nc3)=O)CC2)=O)CCCC(F)(F)CC1 32468,C(C(=O)N=c1cc[nH]c(C)c1F)C1CC(NCc2c(N(C)C)nc(F)cc2)C1 32469,C1(NC(=O)NC2(CC)CCNC2=O)CC2(CC(OC)C2)C1 32470,C(=O)(C(C)S(N)(=O)=O)N1CCN(CC(=O)Nc2ccc(C(C)C(F)(F)F)cc2)CC1 32471,C=CCC(CC(F)F)C(=O)N1CCN(C(=O)CCC(CC)CC)C(CC(F)F)C1 32472,N1(C(C2C(C)(C)C2)=O)CCC2(CCN(C(c3cnc(C(N)=O)cn3)=O)CC2)C1 32473,c1(C(=O)NCC(CNC(c2csnn2)=O)CO)ccc(-n2cncn2)cn1 32474,N1(C(c2ncn(C)n2)=O)CCC(OCCCNC(C23CCC2C3)=O)CC1 32475,N1(C(C=CC(C)=O)=O)CCC(CC(C)(C)NC(=O)Cc2nccn2C)CC1 32476,CC1CN(C(=O)CSCC=O)CC1CNC(=O)C(F)(F)c1ccncc1.CC#N 32477,c1(C(=O)NC2CC(NC(C(C3CCCC3)OCC)=O)C2)cc(C(=O)OC)[nH]n1 32478,c1(C(=O)NCC(CC)NC(C2CCN(C)C2)=O)nncc2ccccc12 32479,Cc1ccc(O)c(C(=O)NC(c2cnn(C)c2)C(N2CCC3CC23)=O)c1 32480,c1(OC)ncnc(C(=O)NCCCOCCNC(C2CCNC2=O)=O)c1F 32481,Cc1ccc2ncc(C(N3CCC(C)C3CNC(=O)C(C)(C)CC(F)F)=O)n2c1 32482,C1(NC(c2c(C)nn(C)c2F)=O)COC2(CCN(C(=O)CS(=O)(=O)N(C)C)C2)C1 32483,CCCC(CCNC(C1CCC1CNC(C1(OC)CCOC1)=O)=O)CCC 32484,CCCC(CCC)CC(=O)NC(c1cn(C)nn1)C(N1CCC(O)CC1)=O 32485,C(CCCCCC(=O)NC(C(=O)OC)C1CCC1)NC(c1n(CC)ccc1)=O 32486,c1(N2CCC=C(C(=O)NCc3cc(C)c(O)c(C)c3)C2)ccnc(S(C)(=O)=O)n1 32487,C1(CCC)(NC(c2cccc(N(C)C)n2)=O)CCCN(C(=O)C(C)C(F)F)C1 32488,c1(C(=O)NC2CC(CNC(COC(CC)(C)C)=O)C2)cc(NC2CC2)ncc1Cl 32489,N1(C(Cc2c(C)nc[nH]2)=O)CC(NC(=O)C2=CCOCC2)CC12CCOCC2 32490,n1(CC(N2CCC(CNC(CCC(=C)C)=O)(OC)C2)=O)ccc2c(C)cccc12 32491,c1(C(=O)NC2C(CNC(C(C)c3ccsc3)=O)C2)ccc(Cl)c(F)c1O 32492,C1(C)(NC(CN(C2CCC2)C(C2C(C(C)C)CCC2)=O)=O)CN2CCC1CC2 32493,Cc1cnccc1C(C)C(=O)NCCN1CCC(NC(=O)C(N)=O)CC1 32494,c1(COC)cccc(C(=O)NC(C)C(C)NC(C2(C(F)(F)F)CC2)=O)c1 32495,n1(CC)cnc2c(NC(CNC(C3(C(F)F)CCOCC3)=O)CO)nc(Cl)nc12 32496,c1(C(=O)NCCOCCCNC(C2(C(=O)NC3CC3)CC2)=O)csc(Cl)c1 32497,C1(C(=O)NCC(CC)NC(=O)CSCC(C)C)CCOC1C(C)C 32498,C1(O)(C(N2CC(C)SC2)=O)CCCC(C)CC1 32499,C(=O)(C(C)(C)C(=O)NC1CN(C(=O)CC(=O)OC(C)(C)C)CC1C)NC 32500,c1(CN(CCOC)CCNC(c2coc(CC3CC3)n2)=O)nn(C)c2c1CCC2 32501,Cc1c(C(=O)NC2CCCC(NC(c3occc3F)=O)C2)ccn1C(C)C 32502,Cc1cccc2c1CC(C(=O)N(CC(C)CNC(=O)C(O)C1CCC1)C)N2 32503,c1(CNC(c2cc(C(=O)OC)n(C)c2)=O)ccc([N+](=O)[O-])cn1 32504,c1(C(N2CC(COC)CC23CCC3)=O)cnc2ncccc2c1 32505,c1(C(=O)NC2C(NC(c3c(CC)ncs3)=O)C2)cc(O)nc2cc(OC)ccc12 32506,N1(C(c2cc(C)n(C)n2)=O)CC(N(C(=O)CSCc2ccccn2)C)C(C)(C)C1 32507,N1(C(C)=O)CC2CC1CN(C(=O)C(C(C)C)NS(=O)(=O)c1cnn(C)c1)C2 32508,C1(CCC)CN(C(c2cc(Br)c(Br)o2)C(=O)NCc2nnn(C)n2)CCO1 32509,N1(C(C2CC(=C)C2)=O)CC(CNC(=O)C=Cc2cc(Cl)sc2Cl)OC(C)(C)C1 32510,C1(NC(CCC(=C)Cl)=O)CC12CCC(NC(c1ccsc1)=O)CC2 32511,CC1CC(=O)NCC1C(=O)NCC1CN(C(C2SCCCS2)=O)CCCO1 32512,N1(C(=O)OC(C)(C)C)CCCC(CCCCNc2cccc(CO)n2)C1 32513,C(=O)(CCC(=O)NC(CNC(c1sc(N(C)C)nc1Cl)=O)C1CCC1)OC 32514,C1(CNC(C2CCCC(C(N)=O)C2)=O)(NC(c2cc(F)n[nH]2)=O)CCCCCC1 32515,C1(NC(C#CC(C)C)=O)CCCC2CN(C(c3coc(C(C)(C)C)n3)=O)CC12 32516,C1(C(N2CC(C)(CNC(=O)CC3CCC3)OCC2)=O)OCC2CCCC1C2 32517,CC1CC(NS(=O)(=O)c2ccccc2COC)c2nccn21.N1C(=O)CCC1=O 32518,N1(C(C2(CC#C)CCCCO2)=O)CCCCCC(NC(c2ccoc2Cl)=O)C1 32519,C(CC(C)N=c1nc(C#N)[nH]cc1Cl)NC(CCCCC(=O)NC)=O 32520,c1(C(=O)NC23CC2CN(C(=O)CCCn2cncn2)C3)ccn2ccsc12 32521,N1(C(Cn2ccc(C)n2)=O)CCC(NC(=O)Cc2ccccc2Cl)C(C)C1 32522,N1(C(C(CC)C)=O)CCN(C(=O)CCCCCF)C(CC(=O)NC)C1 32523,Cc1cnc(N(C)Cc2csc3ccccc23)c(S(=O)(=O)NCCCCO)c1 32524,N1(C(C(C2CCCO2)NC(CCS(N)(=O)=O)=O)=O)CCC2(COC(=O)N2)C1 32525,c1(CCC(=O)NCC2N(C(c3cc(C)nn3C)=O)CC=C2)ccccc1[N+](=O)[O-] 32526,C1(NC(c2cnnn2C2CCOCC2)=O)CCN(CCOCCO)C1 32527,C1(CCC(=O)NCC(CC)NC(C2CSCN2C(C2CCC2)=O)=O)CCC(=O)N1 32528,CC(C)=C=CC(=O)NCCC1(C(=O)NC(C)CC(F)(F)F)CC1 32529,C(c1ccnc2ccccc12)=CC(=O)NC1CCCC1NC(C1CC2CC2C1)=O 32530,S(=O)(=O)(c1cncc(Br)c1)NC1CN(C(c2coc(Cl)n2)=O)CC1F 32531,C(CCCCCNC(=O)CCOCC(C)(C)C)N(C)C(C1(CF)CC(=O)C1)=O 32532,c1(C(N2CC(CCNC(CS(CC)=O)=O)C(C)C2)=O)ccc(C)cc1C 32533,c1(CCC(=O)N(C)CCOCCN(C(=O)CCC2CCOC2)C)cccnc1 32534,CC1CCC(C(=O)NC2(CCNC(=O)CCNC(=O)C(C)(C)C)CCC2)S1 32535,c1(OC)ccc(S(=O)(=O)N2CC3CN(Cc4ccc(C)c(F)c4)CC3C2)cc1 32536,C1(C(N(C(CCNC(C(C)(C)SC)=O)C)C)=O)CCCN(C(=O)OC(C)(C)C)C1 32537,N1(C(c2c(CC)nns2)=O)CCC(C)(C)C1C(=O)NCCc1ccc(C)cc1 32538,c1(C(=O)NCCCNC(C(C)OCCC=C)=O)ccc(F)c2[nH]ccc12 32539,c1(C(=O)NCC2(O)CN(C(c3ncnc(C)c3C)=O)C2)cc(F)cc(Cl)c1N 32540,CC1CN(C(C2CNC(=O)O2)=O)CC(C)N(C(=O)C2=NNC(=O)C2)C1 32541,C1(C(=O)NC(CC(=O)NC)c2ccccc2)CCCN(C(c2ccccc2Cl)=O)C1 32542,c1(OC)ccc(CCN(C(=O)C(N2CCN(CC(C)(C)C)CC2)=O)C)cc1OC 32543,Cc1ccc(C23COC(C2)C3C(=O)NCC(C(C)C)NC(c2cn(C)cn2)=O)cc1 32544,N1(C(c2c(C#C)c[nH]n2)=O)CC(F)(F)CC1(C)CNC(c1c[nH]cc1C1CC1)=O 32545,C=C=CC(C)C(=O)NCC(C)N(C(C1COC(=O)N1)=O)CC 32546,Nc1cc(C(=O)NCC2CC(NC(c3nc(C4CC4)cs3)=O)C2)cc(F)c1 32547,c1(OC)cc(C(=O)NCC2CCN(C(C3CCC=CCC3)=O)C2)cc(C2CC2)c1 32548,Cc1c(C(=O)NCC23CC(NC(=O)Cn4cc(Cl)cn4)(C2)C3)cccc1Cl 32549,c1(COC)nn[nH]c1C(=O)NCCCN(C(c1ccc(C(N)=O)s1)=O)C1CC1 32550,N1(C(C(C)(C)C)=O)CCc2cc(CNC(N3CCC4CCC34C(=O)O)=O)ccc21 32551,N(C1CCCn2ccnc21)C(C(C1CCCN(C(=O)CCC(C)(C)C#N)CC1)C)=O 32552,C1(n2c(C(c3cnc(COC)[nH]3)NCc3sncc3Br)nnn2)CCCCCC1 32553,C12(CNC(c3n(CC)ncc3)=O)CC(CO1)N(C(=O)C(C)OCC(F)(F)F)C2 32554,C1(C)(CNC(c2c(OC)nsc2OC)=O)CN(C(=O)CCC(N)=O)C(C)(C)C1 32555,C(CN=c1cc[nH]cc1S(=O)(=O)NCC1(CO)COC1)OC 32556,C(=O)(C(=O)C(C)(C)CC)NC(COCC)C(=O)NCC1(CO)CCCO1 32557,Cc1cc(C(N2CC(F)CC2C(=O)NCC2CC(=C3CC3)C2)=O)nc(O)n1 32558,C(=O)(C(C(C)(C)C)c1cc[nH]n1)N1CCCC(CNC(CSCCC)=O)C1 32559,C1(C2CCCO2)(C(N2CCN(C(C=C(C)c3ccsc3)=O)CC2)=O)CCCO1 32560,N1(C(=O)OC(C)(C)C)CC2(CCOCC2)C1C(F)(F)F.C12CCCC1NC(=O)N2C 32561,C1(C(=O)NC)CC(F)(F)CN1C(C(=O)NCc1cccs1)C1CC1(C)Br 32562,C(=O)(CC1=NNC(=O)C1)NC(C)(CNC(C1CC(CC2CC2)C1)=O)C1CC1 32563,C1(C2(C)CC2)(C(=O)NC(C2C(C(N(CC#C)CC#C)=O)C2)C)CC1 32564,c1(N(C)Cc2c(C)cccc2F)cccc(S(=O)(=O)N2CCC(C(C)O)C2)n1 32565,CCC(CC(=O)NCCc1ccc(CNC(=O)C=CBr)cc1)C(F)F 32566,C1(CC(=O)N(C)CCNC(c2c[nH]ccc2=N)=O)CCCNC(=O)C1 32567,c1(C(=O)NC(c2cc(F)ccc2F)C)cnn2c1OCC1(COC1)C2 32568,N1(Cc2ccn(C)n2)CCOCC1CNS(=O)(=O)CC1CCC1 32569,C1(CCC)C(=O)NCCN1C(=O)C(C)(CSC)NC(C1C2CC(=O)CC12)=O 32570,c1(OC)ccc(C(C)C(=O)NCC(c2ccccc2OC)N)cc1OC 32571,N1(C(C(c2cc(C)c(F)cc2)=O)=O)CC2CN(C(=O)C(O)O)CC2C1 32572,Cc1ccc2c(c1)C(C(=O)NC1CCC(NC(=O)CNC(C3CCCC3)=O)C1)C2 32573,c1(OC)ccc2cc(C(N3CCN4CCCCC4C3)=O)ncc2c1 32574,C1(CNC(C(C)CNC(=O)Cc2ccc[nH]2)=O)CC12CCOCC2 32575,c1(C(C(=O)NCC(C2CC(C)(C)C2)C)N(C)C)c(F)cccc1F 32576,c1(C(N2CCN(C(CSCC)=O)CC2C2CC2)=O)ccc(Cl)c(OC)c1F 32577,CCC(C(=O)N(C)CCOCCN(C(=O)C(C)C1CCC1)C)C(C)C 32578,Cc1ccc(C(N2CCC2C(=O)NCCCS(C)(=O)=O)=O)c(O)n1 32579,N1(c2cc(CCC)nc(Cl)n2)CCCC(C2CC2NC(C2(C)CCCO2)=O)C1 32580,c1(NC(C2C(C(N(C(c3cccnc3)(C)C)C)=O)C2)=O)cc(Br)cc2[nH]ncc12 32581,c1(C(=O)NC2CCC(C)(OCC)CC2)ccc(F)c2c1CCC2.C12CC1C(=O)N2 32582,CC1(C(N2CCN(C(=O)CNC(c3ccc(=N)[nH]n3)=O)CC2)=O)CCCS1(=O)=O 32583,C1(C(=O)NCC(C)(C)NC(c2ccc(CC(C)C)s2)=O)Cc2cccnc2C1 32584,Cc1cc(C(=O)NC2(CCNC(C3CCN(CC(F)(F)F)C3)=O)CC2)nc(C)c1 32585,C1(NC(Cc2nc(C)[nH]n2)=O)CC2CCC1(N=c1[nH]nc(C3CC3)o1)C2 32586,C1(NC(C2(C)CCNC2=O)=O)CCCN(C(=O)CC2CC(F)(F)C2)CC1 32587,c1(OCCn2cc(CCN(C(=O)COC3CC3)C)nn2)cccc(Br)c1[N+](=O)[O-] 32588,N1(C(C2N(C(CC(CC)SC)=O)CCC=C2)=O)CCC(C)=C(F)C1 32589,C1(CNC(CC(C)(C)C)=O)CC(C)(C)CN1C(C1CCC(C(F)F)CC1)=O 32590,Cn1ncc2nc(Cl)nc(NC3CCCC4CN(C(=O)C(C)(C)CO)CC34)c12 32591,C1(C(=O)NC(C(=O)NC)C)CC12CC(NC(=O)Cc1cn[nH]c1)C2 32592,C1(C)(C(=O)NCc2c(C(N3CC(c4c(C)nn[nH]4)C3)=O)cco2)CCN(C)C1 32593,c1(N2CCN(C(C(=O)N(CC#C)CC=C)C)CC2)ncnc2scc(C)c12 32594,c1(C(C(=O)NC(C(C)C)CNC(C2CC3CC3C2)=O)(C)F)ccccc1F 32595,c1(OC)cccc2c1CNC(C(N1CCC(n3cc(Cl)cn3)C1)=O)C2 32596,C(=O)(CC(Cl)Cl)NC1(C(=O)NCCC2(COC)CC2)CSC1 32597,O=S(=O)(C=Cc1ccccc1)NCC12CC1CN(S(=O)(=O)c1ccc(O)cc1)C2 32598,c1(C(=O)NC2CCC(NC(c3c[nH]nc3C3CC3)=O)CC2)ccc(F)c(O)c1F 32599,CCCCCCC(CC)C(=O)N1CC(C)(NC(c2cccc3c2ccn3C)=O)C1 32600,c1(OC)ncc(C(=O)NCC(C2CC2)NC(C2CCC(C(N)=O)N2C)=O)cc1Cl 32601,N1(C(C2C(=C)C2C(=O)OC)=O)C(C(=O)NCCOCCC)CCC12CC2 32602,Cc1nc2ccc(C(N3CC(NC(C4CCC(=O)O4)=O)C3)=O)cc2n1C 32603,c1(C(C)C)nc2cc(Cl)ccc2c(=NCc2cc(Cl)c(Cl)n2C)[nH]1 32604,n1(CCC)ccc(C(N2CC(NC(=O)CCC3CC3(F)F)C2)=O)n1 32605,N1(C(c2sc3cc(C)sc3c2)=O)CCC(C2CCN(C(=O)CC#N)CC2)C1 32606,C1(O)(CNC(C(=O)NCC2CC2)=O)CCCN(C(c2ccc(O)cc2Cl)=O)CC1 32607,C1(CNC(C2(N)CC2)C)CNCCC1c1ccccc1 32608,N1(Cc2c(OCC=C)cccc2)CC2CN(C(C3CC4CCC3O4)=O)CC12 32609,C1(C(=O)NC(CCCN(CC)CC)C)C2CN(C(c3ccc(F)cc3)=O)CC12 32610,n1(C2CN(C(C3(Cl)C(C(C)=O)C3)=O)C2)cc(C(c2ccccc2)NC=O)nn1 32611,CCC(F)(F)CC(=O)N1CCC(CCN(C)C(C23CC(C(F)F)(CO2)C3)=O)CC1 32612,N1(C(C2C(C)(C(F)F)C2)=O)CCN(C(=O)CCC2CC2)CC12CC2 32613,c1(-c2onc(COC)n2)cccc(CNC(=O)CC2(C(=O)O)CCCC2)c1 32614,N#Cc1cccc(Cl)c1NC(C1CN(Cc2nc(Cl)ccc2Cl)CCO1)=O 32615,Cc1cnn(C)c1CC(=O)NCC1(F)CC(NC(C2(C(F)(F)F)CCO2)=O)C1 32616,Cc1cnc(C=CC(=O)NCCC2CCCCN2C(C23CC(F)C2C3)=O)[nH]1 32617,C=C(Cl)CCC(=O)N1CC(CCNC(C2CC3CCC2C3)=O)(OC)C1 32618,C1(C)(C(N(C)CC2N(C(CCC(C)C#N)=O)CCCC2)=O)CCCCNC1=O 32619,c1(CNC(N)=O)ccc(C(N2CC(O)(CNC(=O)CC3CCSCC3)C2)=O)cc1 32620,c1(C(N2CCN(C(c3cn4c(n3)CCC4)=O)C3CC23)=O)ccc(F)c(Br)c1 32621,C(=O)(C1=CC(C)(C)C1)NC(C(c1c(OC)cccc1)NC(=O)CN(C)C1CC1)C 32622,C1(CNC(C=CCCC(C)C)=O)CCN(C(=O)C2=CCOCC2)CC1C 32623,c1(C(N2CC(O)CC(NC(CN=S(C)(C)=O)=O)C2)=O)cnc2ncnn2c1O 32624,C=CC(CC)CC(=O)N1CCC(C2CCCN2C(=O)CN2CCCCC(=O)C2)C1 32625,c1(CC)nn(C)c(CC)c1C(=O)NCC=C1CCN(C(=O)C(C)S(C)(=O)=O)CC1 32626,c1(NCC(N2CCCC(CS)C2)=O)ccc[n+]([O-])c1 32627,N1(C(C=CC(CC)C)=O)CCN(C(c2cnncc2O)=O)C(C)C1C 32628,C1(C2=CCCCCC2)(C(N(CCCNC(c2c(C)onc2CO)=O)C)=O)CC1 32629,C1(N(C(CCN(C(=O)CC=C(C)C)CC=C)=O)C)CCCC(O)C1 32630,c1(C(=O)NC(C2CCCN(C(c3csc(O)n3)=O)C2)C)cc(C#N)c(O)nc1N 32631,N1(C(C2N(C(C)=O)CCC2)=O)CCC12CN(C(=O)CCCn1ccnn1)C2 32632,N1(C(C2=CCC(NC(C(C(C)C)=O)=O)C2)=O)CCn2ccnc2C1 32633,N1(C(C(C(=O)OCC)OC)=O)CCC(O)(CC(=O)NC2CCN(C(C)=O)C2)CC1 32634,c1(CC(=O)N(CC(=O)NC(C)Cc2ncn(C)n2)CC#C)cccc(C)n1 32635,Cc1c[nH]c(C(=O)NCCOCCC(=O)NCC(C)C(C)C)c1C 32636,c1(C(=O)NC(c2ccccc2Cl)C(F)(F)F)cc(O)cc([N+](=O)[O-])c1 32637,c1(CC(N2CC(N(C(C(C=C)O)=O)C)C(C)(C)C2)=O)cnc2ccccc2c1 32638,C1(C(=O)NC2C=CCN(C(c3ccccc3Br)=O)C2)CC2CC(O)C(C1)C2 32639,C=CCCCC(C)(C)CNC(c1cn(CCNC(=O)C(F)CC2CCOC2)nn1)=O 32640,N1(C(C(CC)(C)COC)=O)CC2C1CCCN2C(c1cc2ccsc2n1C)=O 32641,Brc1ccc2c(c1)ncn2CC1CCCCCCN1 32642,C1(C(=O)NCCCC(C)NC(c2cc[nH]c2)=O)CC(S(C)(=O)=O)C1 32643,C12(CC(=O)NCC3(COC)CCCC3)CCC1CN(C(=O)C1=CCCCC1)C2 32644,c1(CN2C(C(N3CC4CCC(C3)O4)=O)CC3CC32)ccc(Cl)cc1OC(F)(F)F 32645,c1(C(=O)NC(CC)CN(C(=O)Cc2ccoc2C)C)occ(C)c1C(=O)OC 32646,C(=O)(CC(C)c1ccco1)N(CCC(C)NC(=O)CCc1ccncc1)C 32647,N1(C(CC2CCN(C)CC2)=O)CC2(NC(C3COC(=O)N3C)=O)CCCC2(F)C1 32648,c1(OC)cc(OC)c(C(N2CC(NC(=O)C(C)CF)C(O)C2)=O)c(N)c1 32649,Cc1cc(Br)c2ncnc(N3CCCC(c4n[nH]c(C)n4)C3)c2c1 32650,Cn1cc(Cl)cc1C(c1nnnn1CCN1CCOCC1)NCC1CC(C)(C)CO1 32651,c1(C(=O)OC)cc(C(=O)NCc2cccc(-c3ncc(C)o3)c2)c(C)s1 32652,N1(C(c2ccc(CSC)o2)=O)CC2CCC(C1)N2C(=O)CCC1CCCO1 32653,n1(CC)nnc2c1CCC(C(N1CCC(C(C)NC(c3c[nH][nH]c3=N)=O)C1)=O)C2 32654,C1(CCNC(CCN(C(COC(C)C)=O)CCCO)=O)CC=CCC1 32655,CC1CC(NC(c2ccc(Br)c(O)n2)=O)CN(C(C2CCC(=O)C2)=O)C1 32656,N1(C(C(C=C)(C)C)=O)CCC(NC(c2ccc(OC)cc2OC)=O)C(C(C)C)C1 32657,C(=O)(C(F)(F)CCn1ccnn1)NC(CC(C)NC(=O)CC1CC(O)C1(C)C)C 32658,C1(NC(C(C)=C2CCCC2)=O)CCN(C(=O)C=Cc2ccncc2)C1C 32659,C1(NC(COC)=O)C2CCCN(C(=O)CN3CC(C)(C)C3)C2C1(C)C 32660,Cc1cccc(-c2cc(C(=O)N(C(C)CNC(C3(C(C)(F)F)CC3)=O)C)on2)c1 32661,C12(C(=O)NCC3CC4(CCC4)CO3)CC(CN(C(c3nn[nH]n3)=O)C1)C2 32662,n1(CC)nc(C)c(C(N2CC(NC(C3(O)CCSC3)=O)C(CC3CC3)C2)=O)c1Cl 32663,C1(N2CCOCC2)(C(N(CCN(CC)CC)CC)=O)CCCC1 32664,C(C)(CO)(C(=O)N(CCC(O)CO)C)NC(C1C(C(C)C)C1)=O 32665,C1(CNC(=O)C=Cc2ccoc2)CC2CCC1N2C(=O)CCc1cccc(F)c1 32666,c1(CC(=O)NCCCCNC(C2C3CC3C3CC23)=O)cnc2ncccn12 32667,N1(C(c2n(CCC)ncc2)=O)CCN(C(=O)CS(=O)(=O)N(C)C)CC(CO)C1 32668,Cc1ncnc(O)c1CC(N1CCC1CNC(C1(O)CC(F)(F)C1)=O)=O 32669,C1(C(=O)NCCC(C)NC(C2(CCF)CC2)=O)OCC2COCCC12 32670,C(CCC(N)=O)(C(=O)N1CC(C)(c2cn(CC3CCCO3)nn2)C1)N(C)C 32671,Cc1c(C(N2CC(O)(CCNC(C3CCN(CC(C)C)C3)=O)C2)=O)c(Cl)nn1C 32672,N1(C(CCC(NN(C)C)=O)=O)CCC2(C=C(C(=O)N3CC(F)(C#N)C3)C2)C1 32673,C1(CC(=O)NCC(C2CC2)NC(c2cc(C(=O)OC)on2)=O)CCC12CCC2 32674,n1(C(C)C)ccc(CC(N2CC(NC(c3ccsc3Br)=O)C2)=O)n1 32675,Cn1cc(CCC(=O)N2CCC2CNC(c2nc(Cl)cs2)=O)nn1 32676,CCC(C)N(OC)C(=O)C(CC(C)C)ONC(=O)CC1(C)CCOC1 32677,N1(C(C(CCF)NC(=O)CC2CCC(O)C2)=O)CCOC2(CCC2)C1 32678,N1(C(CC2N(C(=O)CCc3cnco3)CCCC2)=O)CC(C2CC2(F)F)C1 32679,c1(C(=O)NCCNCC(C2CCCO2)O)cncc([N+](=O)[O-])c1 32680,c1(C(N(CCNC(c2c(CC)onc2)=O)C(C)C)=O)cc2cccn2cn1 32681,N1(C(c2c(C)cns2)=O)CC(CNC(c2cncc(-c3cc[nH]n3)c2)=O)C(C)C1 32682,c1(CC(=O)NCC2CN(C(c3c(Cl)ccc(N)c3)=O)C2)noc2ccc(F)cc12 32683,C(CC(C)C)(C(=O)OC1CCC1C(=O)NCc1ccncc1OC)OC 32684,C(=O)(CCC(C(C)C)NC(c1cc(C(C)C)[nH]n1)=O)NC(C(=O)NCC(C)C)C 32685,C(=O)(C#CC1CCCOC1)NC1CC2CN(C(c3n(C(C)C)ccc3)=O)CC21 32686,c1(C(N2CCC(CC(N3CCC(NS(=O)(=O)NCC)C3)=O)C2)=O)cn(C)cc1C 32687,c1(C(=O)NC2CN(C(COCCC#C)=O)CC2C)cc(C(N)=O)ccc1F 32688,C1(NC(CCOCCC)=O)CN(C(c2cnc(S)n2C2CC2)=O)CC1OC 32689,C(C(C(=O)N1CC2CC2(CO)C1)C(C)C)NC(C(C=C)C)=O 32690,c1(N2C(CNC(=O)Cc3cnsc3)CC2)cc(C2CC2)ncn1 32691,C1(C(=O)NCCC(C)NC(C2CC(=O)N(C)C2)=O)CC(C)(C)C1C(F)(F)F 32692,N1(c2c(C)cncn2)CCOC2(CCCN(C(=O)C(F)C(C)(C)O)C2)C1 32693,CC(O)C(C)(C)C(=O)N(CC(C)(C)CNC(c1cnc(C2CC2)nc1)=O)C 32694,C1(C(N2CC3C(C(=O)Nc4c(OC)nsc4)C3C2)=O)CC2(CCC2=O)C1 32695,N1(C(C2CCCN(CCC)C2)=O)CC(C2CN(C(=O)CN(C(=O)COC)C)C2)C1 32696,N1(C(c2cnc(-n3cccn3)s2)=O)CC2(CC(C(F)(F)F)C2)C1 32697,N1(C(C(C)NC(CC)(C)C)=O)CC2(CC(CNC(=O)Cc3ncc(C)s3)C2)C1 32698,c1(C(=O)NCC(CNC(C(C)CN2CCCCC2)=O)CO)cccc(N)c1F 32699,N1(C(C(C)N(C)C)=O)CCN(C(=O)CC2(O)CCC2)CC1c1ccnn1C 32700,C=CCC(C(=O)NCC1CCCO1)NC(=O)CC1OCCO1 32701,c1(CC)c(C(=O)NC2(CO)CN(C(=O)C3=CCCCC3)C2)sc2ccccc12 32702,CC(C)CC(C)CC(=O)N1CC(C)N(C(=O)CC2CC(C)(C)CO2)CC1C 32703,Cc1ncc(Cl)c(C(N2CCC(O)(CNC(C3CC4COCC4C3)=O)C2)=O)n1 32704,Cc1cc(C(=O)NC2CCC2CNC(C2(N=[N+]=[N-])CC2)=O)cnc1C(F)F 32705,c1(C(=O)NCC2C3(CN(C(c4nc(C)sc4)=O)C3)CC2)cc2n(n1)CCCC2O 32706,c1(C(=O)NC(C2(O)CCN(C(C3CC(C#N)C3)=O)CC2)C)ccc2c[nH]nc2c1 32707,c1(C(=O)NC2(C(=O)NCCC(O)C3CC3)CCCC2)cccc2[nH]ccc12 32708,c1(OC)nccc(C(N2CC(NC(=O)C(C)C)C(C)C2)=O)n1 32709,CC1CCC(C)(C)N1C(C1(C)CCN(C(=O)C(C2CCCCC2)C)CC1)=O 32710,c1(C(C)O)ccc(C(=O)NCCN(C2CCCC2)C(=O)CC2CCC(C)C2)cc1 32711,CC1CCN(C(C2CC(O)(C#N)C2)=O)C(C)C1NC(C1CN(C(N)=O)C1)=O 32712,c1(C(=O)NCC23CN(C(c4cc(C)on4)=O)C(CC2)C3)nc2cc(F)ccc2s1 32713,C1(C(C(C)NC(=O)N(C)Cc2ccco2)(C)C)Cc2ccccc2O1 32714,CC(C)(O)C(F)C(=O)NCC1CN(C(C2CC(=O)N2)=O)C1 32715,c1(C(N2CCN(c3nc(C)cc(SC)n3)CC2C)=O)ccnc2c1OCO2 32716,c1(CC)ccccc1-c1cn(CC2CCCC2NC(c2cnnn2C)=O)nn1 32717,c1(C(=O)NC(CNC(c2ccc(C)nn2)=O)C2CCC2)c(C)nn(C(C)C)c1C 32718,c1(CN(C(CCC)=O)C)cnn2c1CN(C(=O)C(C)SC)CC2 32719,CC1CCC(NC(c2cccnc2O)=O)CN1C(=O)CC1(NC(C)=O)CC1 32720,CC(CN=c1[nH]c(=NCC2CC23CCC(F)(F)CC3)[nH]c2c1CCCC2)C1CC1 32721,C1(OC)CCC(C(N2CC3CC3(NC(=O)C=C(C)C(F)F)C2)=O)CC1 32722,C1(CNC(C(C)(C)CO)=O)CCC2(CO1)CC(NC(C13CCC(CC1)CO3)=O)C2 32723,C1(CNC(C(n2cc(CC(O)CO)nn2)C)=O)CCC(C2OCCO2)CC1 32724,N1(C(c2nc(C(C)OC)sc2)=O)CCCC1(C)CNC(c1ccnn1C)=O 32725,CC1(C)CC(C(N2CCN(C(=O)C=Cc3ncc[nH]3)C(CO)C2)=O)C(C)(C)O1 32726,C12CCCC(C1)NC2=O.C1(CC#N)CN(C(=O)CO)C1 32727,C1(n2cc(CNC(CCSC)=O)nn2)CCN(C(=O)OC(C)(C)C)CC1 32728,c1(C(=O)NCC2C(NC(c3c(N)n(CCO)nc3)=O)CC2)cccc2sccc12 32729,c1(C(=O)NC(C(C)NC(C2(CCOC)CCCC2)=O)C)ccc2cnc(C)n2c1 32730,CCCCC(O)CC(=O)NC(C(N1CCCC(C)C1)=O)C1CC1 32731,N1(C(C2CCC(=O)N2)=O)CCCN(C(c2cc(-c3cccnc3)no2)=O)CC1 32732,C1(NC(CC(COC)C)=O)CC2CC1CN(C(c1ccncc1Br)=O)C2 32733,C(c1ccc(C(F)F)o1)=CC(=O)NCC(CCNC(Cc1cn(C)nc1)=O)O 32734,N1(C(c2cc(OC)n[nH]2)=O)CCc2nc(C(N3CCC(OC)CC3)=O)cn2CC1 32735,C=C(C)C1OCCC1CNC(=O)C(C1CCCCC1)NC(C1CN(C2CC2)C1)=O 32736,N1(C(C(N2CCCC(C)C2)=O)=O)CCCC(C)(CNC(c2ncccc2Cl)=O)C1 32737,CC(CCCc1ccccc1)C(=O)N1CCC(N(C(=O)C2=C(Cl)CC2)C)CC1 32738,c1(OC)cc(C(N2C3CCC2C(NC(=O)C=Cc2ccoc2)C3)=O)c(Cl)cc1Cl 32739,Cc1ccc(F)cc1C(N1CCC1CNC(C1(F)CCCN(C)C1)=O)=O 32740,C(=O)(C1=NOC(CNC(=O)CC(C)n2ccnc2)C1)NC1(C(COC)O)CC1 32741,Cc1cc(CC(=O)NC2COCC2NC(=O)CC(C)F)ccc1CO 32742,C1(C2=CCOCC2)(CNC(c2cc3c([nH]2)CCCC3)=O)CC1 32743,C(=O)(C(CCC1CCC1)NC(=O)C(c1cnn(C)c1)=O)NCc1ncc(C)[nH]1 32744,c1(CC)c[nH]nc1CNC(c1ncoc1CNC(C12CC(CO)(C1)C2)=O)=O 32745,Cc1ccc(CC(=O)NC2CC(NC(=O)C(C)(C)OC(C)C)C23CCC3)cc1O 32746,c1(CC)nc(C)c(C(=O)NC2(C)CCN(C(=O)CCC(C)SC)C2)c(C)n1 32747,C1(COC)(CNC(=O)C(C)=CCNC(c2cccnc2OC)=O)CCC(=O)N1 32748,c1(CC)nc(C)c(CC(=O)NC(C)CNC(=O)CC2CS(=O)(=O)CCO2)c(C)n1 32749,c1(OC)ccc(CC(=O)NCCC2CCCC2(C)C)c(O)c1 32750,N1(C(C2N(CCCC)CCCC2)=O)CC(NC(c2cc(C)[nH]c2C)=O)C(C)(C)C1 32751,C(=O)(C1=CCCN(C(=O)CC=C(Cl)Cl)C1)N1CC(C)(OC)C1 32752,C1(C)(C(N(C(N(CC(C)O)C(C)C)=O)C(C)C)=O)CCN(S(C)(=O)=O)CC1 32753,c1(C(=O)NC(CC)CNC(=O)C=CS(C)=O)cnc2cnc(Cl)cc2c1 32754,N1(C(c2c(C)coc2)=O)CCC2(CCN(C(=O)CC3COCCOC3)C2)C1 32755,c1(C(=O)NCC(C)(C)Nc2nccn3nnnc23)cncc2nc[nH]c12 32756,C=C(Cl)C(C)(C)C(=O)NCC(C1CCCN(C(c2ncncc2F)=O)C1)(C)O 32757,C(CC(O)CNC(c1n[nH]cc1Br)=O)NC(=O)COCC1CCCC1 32758,c1(CC)conc1CC(=O)N(CC(O)CNC(c1sncc1C)=O)C 32759,C1(NC(c2cc(F)c(Cl)cc2F)=O)CCCCCN(C(c2cc(CO)[nH]n2)=O)C1 32760,C=CCC(CC(F)F)C(=O)NC(CNC(c1cc(CC)cc(N)c1)=O)C(C)(C)C 32761,c1(C(N2CC(CNC(c3ccc(C)s3)=O)C3C2C3)=O)cc(F)c(C#N)c(F)c1 32762,CC1CN(C(=O)CCCF)CCC1CNC(c1cc(Cl)ccc1Cl)=O 32763,c1(CN(C)C(C2CC(CNC(=O)Nc3ccco3)C2)=O)cnc[nH]1 32764,C(CCCCCC(=O)NCC=C(C)C)NC(c1n(CC)nc(C)c1)=O 32765,c1(C(=O)NC(C2CCCN(C(=O)CCNC(=O)CO)C2)C)ncnc(O)c1F 32766,CC(CO)(C1CCC1)NC(=O)NC1CCC1OC(C)(C)C 32767,C1(C(C)C(=O)NCC(C2CC2)C2CC2)CCN(C(=O)COC2CCCOC2)C1 32768,N1(C(c2nc(CC)sc2N)=O)CC(CNC(=O)CCN2CCCCC2)C2(CC2)C1 32769,C=Cc1ccc(C(=O)NC(C)CC2CCN(C(=O)C(CC)NC(N)=O)CC2)cc1 32770,C1(CCC(=O)N(CC(C)N(C(CCCC)=O)C)C)CCCC(O)C1 32771,N1(C(=O)C2=CCCSC2)CCN(C(=O)COc2cccnc2)C2CCCCC2C1 32772,C=C(Br)CCC(=O)N1CCN(CCCNC(c2snnc2C)=O)CC1 32773,c1(C(N(CCNC(c2n(C)ncc2N)=O)CCO)=O)cc(Cl)cc(C(F)(F)F)n1 32774,N1(C(CCC)=O)CC2CCC(C1)C(NC(=O)C1=CC(C)(CC)C1)C2 32775,C1(N(c2cc(C(=O)OC)ncn2)C(=O)C(F)(F)Cl)CC2CCC(C1)N2 32776,C1(NC(C2(OC)CCCCC2)=O)CCN(C(c2cc(Cl)c[nH]2)=O)CC1C 32777,n1(CC)ccnc1C=CC(=O)NCCC1CN(C(C2CC(CC(=O)OC)C2)=O)C1 32778,S(=O)(=O)(c1cc(C)c(-c2ccccc2C#N)cc1C)NC(CC)CCN(C)C 32779,CC1=C(CNC(=O)CC2C=CC(NC(=O)C(c3ccccc3)O)C2)COCC1 32780,c1(C(N2CC3C(NC(C=CCOC)=O)CC(C3)C2)=O)ccc2cc(Cl)ccc2n1 32781,c1(C(=O)NCCN(C(=O)C2=CCCO2)CC)cccc2nccn12 32782,Cc1nnc(CCC(=O)NC2(CCNC(c3ccc(Cl)cc3)=O)CCC2)n1C 32783,C(=O)(CCC(C)(C)NC(c1cccc(F)c1N)=O)N(CC(C)(O)C1CC1)C 32784,N1(C(c2cn(CCC)nc2C)=O)CCC(C)(NC(c2n[nH]c(C)c2C)=O)CC1 32785,C(CCO)(C(C)(C)O)NC(c1ccn(CCNC(c2ccc(CC)s2)=O)c1)=O 32786,CCC(O)C(F)(F)C(=O)N1CC(F)(CNC(=O)C(C)(C(=O)OC(C)(C)C)OC)C1 32787,c1(C(N2C(C)CC(NC(=O)CC(C)(F)F)C2)=O)ncc2cc(Br)ccc2n1 32788,N1(C(CC(CC)C2CC2)=O)CCC2C(NC(c3c(C)nn(CC)c3Cl)=O)CC12 32789,Cc1cc(Cl)ccc1C(N1CC(CNC(C2(n3cncn3)CC2)=O)C2(CC2)C1)=O 32790,c1(C(=O)NCC23N(C(C(C)=C4CCC4)=O)CC(C2)C3)ccc(C)cc1N=[N+]=[N-] 32791,c1(C(=O)NCCCNC(c2c(C)ccc(OC)n2)=O)nccc2c1NCCC2 32792,c1(NCC2(NC(Cc3nc(C)sc3)=O)CCCCC2C)ncc([N+](=O)[O-])cn1 32793,CC(C)(C)CC(=O)NC1CCOC1C1CCN(C(c2ncn(C3CC3)n2)=O)CC1 32794,c1(N2C(C(=O)Nc3c(OC)c(F)ccc3)CCCC2)ccnc2ccnn12 32795,c1(COC)nc(N(C)NCC(C(C)C)N(C)C)cc(N2CCC(CCCO)CC2)n1 32796,N1(CC(=O)NCC(CNC(C2(N(C)C)CCCSC2)=O)(C)F)C(=O)CCCC1=O 32797,c1(CCC)ccccc1C(=O)NC(C)C(C(C)C)NC(c1ccc(O)nn1)=O 32798,C1(C(=O)NC(CNC(c2c(C)cc(CC)o2)=O)(C)CO)CCCCCN1C 32799,CC1OCCCC1C(N1CCC(N2CCN(C(=O)C(C)(C)C3CC3)CC2)C1)=O 32800,Cc1cc(=NC2CN(CC3CC3)C2)[nH]c(N2CCc3n[nH]cc3C2)n1 32801,CCC(CC)CC(=O)NCC(C1(O)CN(C(=O)CCF)C1)(C)C 32802,C(C(C)C)(C(O)C(=O)NCC=CC(=O)NCC1CCC(C)(C)CC1)OC 32803,C1(C(=O)NCc2occ(C)c2)CCC(C)N(C(C2OCCOC2C)=O)C1 32804,N1(C(C=C(C)Cl)=O)CCC2(CCCCN(C(C3CCOC(C)C3)=O)C2)C1 32805,Cc1cc(N)cnc1C(=O)NCC(C)NC(c1cnsc1C)=O 32806,CC1CC(NC(c2cnc(-c3cccnc3)s2)=O)CN(C(=O)CC2CC=CC2)C1 32807,C(C)(C)(CCC(=O)NCCCCOC(C)C)NC(C(COCC)C)=O 32808,C1(CNC(C(C)OCC=C)=O)CCN(C(C2CC2c2cccc(Cl)c2)=O)CC1 32809,C1(NC(c2cnn(C(C)(C)C)n2)=O)CCC(C)(CNC(=O)C=Cc2ncc[nH]2)C1 32810,C12(CCNC(=O)C=Cc3cnc[nH]3)CCC1CN(C(c1cc3sccc3[nH]1)=O)C2 32811,N1(C(C(CC=C)C)=O)CCC2CN(C(c3ccccn3)=O)C(C)C12 32812,C(CCC(C(=O)N1CCN(CC(C)O)CC1)NC(=O)CC(C)n1cccc1)OC 32813,C1(C(N2CC(N(C)C(c3cnn(C)c3)=O)C(C)(C)C2)=O)(OC)CCCCCCC1 32814,C1(C(=O)NC(C(C)C)CNC(=O)CC2CCN(C)C2=O)CC(=O)OC1(C)C 32815,C1(C(=O)NC(C2N(C(c3c(CC)c[nH]n3)=O)CCC2)C)CSc2ccccc2O1 32816,CC1(C)OCC2CC12C(N1CCCC(NC(c2ccnn2CC2CC2)=O)CC1)=O 32817,n1(CCN(CCCC)CC)cc(C(O)CC)nn1 32818,N1(C(CS(CCOC)(=O)=O)=O)CCC2(CC1)CN(C(C1CC1OC)=O)CCO2 32819,C1(C(=O)OC)C(C(=O)OC)C2CCC1N2CC1CC(C(F)(F)F)C1 32820,CCCC(CNC(=O)CCC1CCCCC1)NC(c1sncc1C)=O 32821,C1(NC(c2ccc(C)cc2C)=O)CN(C(=O)Cc2csc(C)n2)C2(CCCC2)C1 32822,C1(NC(c2nc(CCC)sc2)=O)CC2CCC1C(NC(c1cc(C#N)cs1)=O)C2 32823,c1(C(CN(C(c2cccs2)C)C2CC2)=O)ccc2c(c1)CCCN2 32824,c1(C(N(CCC)CCNC(=O)CN2CCOCC2)=O)ccc(O)cn1 32825,CCCC(C)(c1nnnn1CCC1(C)CC1)NC1CCC1(C)C 32826,C1(NC(CCn2c(C)cc(C)n2)=O)CC2CCC(C1)N2C(c1ncccc1C)=O 32827,c1(CC)oc(C)cc1C(=O)N(CCCC(=O)NCCC(F)F)C 32828,c1(C(=O)NC2CCCN(C(=O)CCCF)C2)cc2nc(F)ccc2o1 32829,Cc1sc(=O)n(CCNC2CCC(C)N(C(=O)NS(=O)(=O)C(F)(F)F)C2)c1C 32830,N1(C(=O)CCCc2ccccn2)CCC2CCN(C(=O)CC34CCCC3C4)C2C1 32831,c1(C(=O)NC(C)C(CO)NC(c2ccc[nH]2)=O)cccc(-c2cnco2)c1 32832,C(=O)(C1CCCc2nnn(C)c21)N1CCCN(C(c2c(C#C)c[nH]n2)=O)CC1 32833,N1(C(c2cc(C)nn2C)=O)CC2CCN(C(=O)CC3CCCCCCC3)CC2C1 32834,CC1(C)CCOC1C(=O)NC1CCCN(C(=O)CNC(=O)N(C)C)C1 32835,c1(C(N2CCC(CC=C)(NC(c3cn[nH]c3)=O)C2)=O)cc2c(O)ncnc2cn1 32836,Cc1cc(NC(=O)CC2C(NC(C3C(C)(C)C3(F)F)=O)CC2O)cc(CO)c1 32837,C(=O)(C1Cc2ccc(C)cc21)N1CCN(C(c2cc(CC)c(C)s2)=O)CC(O)C1 32838,N1(C(C(C=C)O)=O)CC2(CCN(C(c3c(C)oc(C)c3C)=O)CC2)C1 32839,N1(C(CN(C)CCO)=O)C2CCC1CC(CNC(c1cnn(C)c1C(F)F)=O)C2 32840,C(=O)(C(C(C)(C)C)OC(c1n[nH]c(C)c1-c1ccc(F)cc1)=O)NC 32841,C(=O)(C(F)CC(C)C)N(C1CCN(C(=O)CN(S(=O)(=O)CC)C)CC1)CCC 32842,C=CC(CC)CC(=O)N1CCC(C)C(NC(=O)C=Cc2cnc(OC)nc2)C1 32843,C1(NC(CCn2ccc(C)n2)=O)C2CC3CN(C(C4OCCCO4)=O)C1C3C2 32844,C1(C(N2CC(NC(=O)C=C3CCCC3)C2)=O)CC12CCCc1ccccc12 32845,C1(NC(CN(C2CC2)CC)=O)CC(NC(c2cc(SC)ccc2C)=O)C12CCC2 32846,C(=O)(CC(O)CCSC)NC1CCN(C(c2ccc(CC)nc2)=O)C1 32847,C12(NC(c3nc(C(C)(C)C)oc3)=O)CCCN(C(=O)C3=CCC3)CC1C2 32848,c1(CNC(C2CCCCO2)=O)cccc(Cn2cc(CNC3CCOC3)nn2)c1 32849,c1(NC(C(C)SC)=O)c(CN(CC(c2ccccc2)(C)C)C)cccc1F 32850,c1(-c2n(C)ncc2)cccc(C(=O)NC2CC(NC(=O)C=CC(F)F)CC2O)c1 32851,CC1(NC(=O)CNc2nccs2)CN(C(C2CC(O)(c3ccccn3)C2)=O)C1 32852,N1(C(c2nc(C)sc2)C(=O)NCc2ccon2)CCC(C(N)=O)CC1 32853,c1(C(N2C(C(=O)NCC3COCCO3)CCC2)=O)cc([N+](=O)[O-])cs1 32854,c1(OCC(=O)N(C2CCN(C(C(C)=CC3CC3)=O)C2)CCO)c(C)cccc1Cl 32855,C1(C)(C(=O)NCCCN(C(C2CCc3ncnn3C2)=O)CC)CC(C2CC2)=NO1 32856,N1(C(C(C)(C)OCC)=O)CCN(C(c2c[nH]cc2CC)=O)CC(O)C1 32857,O=S(=O)(c1ccc(NCc2ccc(Cl)nc2)c(F)c1)N1CC=C(CO)CC1 32858,c1(C(=O)NCC2C(C)CN(C(C3CCC3)=O)C2)ccn2ccnc2n1 32859,Cc1onc(-c2cccc(F)c2)c1C(=O)NC(C)CNC(c1coc(Cl)n1)=O 32860,c1(NC(C2C(CNC(Cc3n(C)ccc3)=O)C2)=O)cnc2[nH]cnc2c1 32861,c1(C(c2cccs2)NC(=O)NCCc2cn(C)nn2)cc(Cl)ccn1 32862,c1(-c2cn(CC3N(C(CC(CC)C(F)F)=O)CC3)nn2)ccc2nccnc2c1 32863,C(=O)(CCS(=O)(=O)c1ccc(OC)cc1)NCCNC(C(CCCC)(C)F)=O 32864,c1(C(N2CC(CNC(c3occ4c3CCOC4)=O)C2)=O)ccc2c(c1)CCOC2 32865,c1(C(N(C(CNC)C)C)=O)cc(F)c(O)c(Cl)c1.Cc1cc(CC=O)on1 32866,N1(C(Cc2cc(C)no2)=O)CCCC(C2CC2NC(c2cc(C(N)=O)cs2)=O)C1 32867,c1(C(=O)NC2CN(C(C3CCN(C)C3)=O)CC2F)cccc2c1CCC2 32868,N1(C(CC23C(C)(C)C(CC2)CC3)=O)CCCC(C2(NC(=O)C(O)C3CC3)CC2)C1 32869,c1(C(N(C(C)CNC(=O)CC2(OC)CCOCC2)CC)=O)n[nH]c2c1CCCC2 32870,c1(C(N(CCCCN(C(C(COC)OC)=O)C)C)=O)ccc2c(c1)C(C)C(C)O2 32871,C1(C(N2C(C(=O)NCCCc3ccco3)CCC2C2CC2)=O)CC2(C1)CC(O)C2 32872,C1(C(N2CCC(N(C(=O)CN3CSCC3=O)C)CC2)=O)C(C2CC2)C1(F)F 32873,c1(NC(CCC)CC(N2CC(C)(C)OCC2CC)=O)ccc2c(c1)ncn2C 32874,CCC(C(F)F)NC(=O)CCOCCOCCC1CC1 32875,CC(C)C(C)C(CNC(=O)C(=C1CCCCC1)F)NC(c1cc(=O)n(C)o1)=O 32876,N1(C(CC2ON=C(C)C2)=O)C(CC(=O)NC(C)(C)CC(C)(C)O)C2CCCC12 32877,C(=O)(C1=CC2(CCOC2)C1)NCC1(NC(c2c(C)ncnc2)=O)CCCCCC1 32878,Fc1cc(N2CCOCC2)ccc1NCCN.c1cn2ccsc2n1 32879,N1(c2c(C)c(NCc3c[nH]ccc3=N)ncn2)CCOc2cc(Cl)ccc2C1 32880,c1(C(=O)NCCC(C)N(C)C(c2cnsc2)=O)cccc(N)c1 32881,C1(C(N2CC(O)(CCNC(c3scc(C)c3Cl)=O)C2)=O)CCn2nnnc2C1 32882,C1(NC(Cn2ncc(C)c2)=O)C2CC1N(C(=O)CC1CC3(CCC3)C1)C2 32883,CC(=O)C(C)(C)CC(=O)NC(C1CN(C(C2CS(=O)(=O)C2)=O)C1)C 32884,C1(C(=O)NCCCN(CCO)C(C2CCC2n2cccn2)=O)(COC)CCCO1 32885,C1(CC=C)(NC(=O)CC(C)CF)CCN(C(=O)C=Cc2ccccc2)CC1 32886,c1(SCCNC(=O)CO)nnnn1C1CCCCC1 32887,C1(C(N2CCC3OCCC3C2)=O)CC2CCCC2N1C(C1CC=CCC1)=O 32888,N1(C(c2csc(C)c2C)=O)CC2(C1)C(NC(=O)Cc1cn[nH]c1)CCS2(=O)=O 32889,C(=O)(C(C(C)C1CC1)N1CCC(OOC(F)F)CC1)N(C1CCOC1)C(C)=O 32890,C(=O)(CCCN(C)N=O)NC1(CC)CCCN(C(=O)CCc2ccc(F)cc2)C1 32891,N1(C(=O)NCC(=O)NC2CC2)CC2CC1CN2C(c1csc(Br)n1)=O 32892,c1(CC(C)C(=O)N2CCC(C(C)(C)NC(C3CCOC3)=O)C2)ccc(Cl)cc1Cl 32893,CC1(C(N2CC(NC(c3ccoc3CC(N)=O)=O)CC(F)C2)=O)CCCC1(F)F 32894,C#Cc1ccc(NC(=O)C(C(C)NC(C2CC(C)CCO2)=O)C(C)C)c(C)c1 32895,CC(F)(F)C(F)C(=O)NCc1ccc(C(=O)NOCCCCCC2CC2)s1 32896,Cc1ccc(CNC(C23CC(C(=O)O)(OC2)C3)=O)c(NC(C)(C)C)c1 32897,C1(NC(C2(COC)CC2(F)F)=O)C2CC(CN(C(=O)CN(C)C(N)=O)C2)C1CO 32898,C1(CNC(C=CC(=O)OCC)=O)CC(C(=O)N2CCC(CO)(OC)C2)=NO1 32899,C=CCC(CNC(C1CC1C#N)=O)C(=O)NCCOCCN(C)C 32900,CCCCC(C)CCC(=O)NCC(O)CCNC(c1cc(C)nc2ccnn12)=O 32901,C1(c2cn(CCC=C(C)C)nn2)CN(C(C2(N(C)C)CCCOC2)=O)CCO1 32902,C(=O)(C(C)CCCc1ccccc1)NC1CN(C(CCC(=O)OCC)=O)C(C)C1 32903,c1(OCC)ccc(C(=O)NC(C)C(=O)NC2CCN(C(=O)C(N)=O)C2)cc1 32904,N1(C(c2c(C)nc3sccn32)=O)CCC2(CCC(NC(=O)C3=COCCC3)C2)C1 32905,N1(C(c2n(CC)nnc2)=O)CCN(C(=O)CCc2ccc(Cl)s2)CC1C 32906,c1(C(N2CCCC(c3onc(C)n3)C2)C(=O)NC(C)C)sc(C#N)cc1C 32907,C1(C)(COC)CC(NC(c2c(C)cccc2F)=O)CN1C(c1ccoc1Cl)=O 32908,N1(C(c2ccc(CNC(CCC=C)=O)cn2)=O)C(C)CCC1(C)C 32909,C1(OC)CC2(C1)CN(C(c1csc(CNC(C3(CF)CC3)=O)c1)=O)C2 32910,c1(C(=O)NC(CCNC(c2ccn(CC)n2)=O)C)ccc(C2CNC(=O)C2)cc1 32911,CCC(C)C(C(=O)N(C)CCOCCCNC(=O)C(c1cccc(F)c1)F)OC 32912,C(CC1=CCN(C(c2cc(N)nc(Cl)c2)=O)CC1)NC(C1N(CC)C(=O)CC1)=O 32913,C(CC(O)CC(=O)NCCC1(O)CCCN(C(c2cn[nH]c2)=O)C1)SC 32914,N1(C(c2ccccc2)=O)CCCC(C2CCCN(C(C3CC(O)C3)=O)C2)C1 32915,N1(C(COCC)=O)CCCC(C)(CNC(=O)C2=CCCC2C)C1 32916,C=C(C)CCC(=O)N(CCCNC(C1CCN1CC)=O)Cc1cccnc1 32917,c1(CN2C(CO)CC(OC)C2)ncc(Br)cc1Br 32918,c1(-c2cn(CCC(=O)N(C)CC3CC4(CC4)C3)nn2)ccc(Cl)c(F)c1 32919,C1(C(=O)NCC(=O)NCC#C)CC1C1CN(C(C2CC(C(C)C)C2)=O)C1 32920,CC1=CN2C(C(=O)NCCCCN(C)C(C3CC4CC4C3)=O)(C=C1)CC2 32921,N1(C(C(OC)OC)=O)CC2CC(NC(c3conc3C3CCC3)=O)CC1C2 32922,Cc1ccc(C(=O)NC(C)CCNC(=O)COCC2CCOC2)c(N)c1F 32923,c1(C(N(CCCCNC(CCS(=O)(=O)NC)=O)C)=O)cnc2c(c1)CCCO2 32924,C1(NC2(CS(C)(=O)=O)CC2)CCN(C(c2coc(-c3csc(C)n3)c2)C)CC1C 32925,c1(C(C)F)ccc(C(=O)NCC(C)N(C(=O)CSCC(N2CCCC2)=O)C)cc1 32926,C(=O)(C(O)C(F)(F)F)NCC1(CO)CC(C)C1.C(=O)CC(C)(C)C 32927,CCC(Cc1ccccc1)C(=O)N1CC(C)(NC(=O)CCC(=O)NC)C1 32928,N1(C(C(=O)NCc2ccc(F)cc2)C2CC2Cl)CCCC2CC(O)CCC12 32929,Cc1nc(O)ccc1C(N1CCC(C)C1C(=O)Nc1cnn(CCF)c1)=O 32930,C1(NC(C=CCC)=O)CCN(C(c2c(OC)noc2C)=O)CC12CCC2 32931,c1(OC)ccc(C(N2CCCC2C(C)(C)NC(C2CN(C)CC2O)=O)=O)nn1 32932,CCCC(F)C(=O)NCCOCCCN(C)C(C1CCC1C#N)=O 32933,C(C(=O)NCC1CCN(C(C2CCOCC2(C)C)=O)C1)(c1ccccc1)=C(C)C 32934,CC(C)CC(CC(C)C)C(=O)NCCC(C)N(C(=O)CCc1ncc(F)cn1)C 32935,CN1CC(CC(=O)NCc2nccc(O)n2)CCC1C(F)(F)F 32936,c1(SCC(N2C3CC(N(C(C=CC)=O)C)CC2CC3)=O)nc2ccc(C)cc2[nH]1 32937,C1(CNC(C(C)(C)SC)=O)CN(C)CCN1C(c1cc(Cl)sc1Cl)=O 32938,Fc1conc1CNC1CCCC1Cc1nc(-c2ccc(Br)s2)no1 32939,CC(F)(F)C(C)(C)CC(=O)N1CC(NC(c2cccc(O)n2)=O)CC12CCC2 32940,C(=O)(C1Cc2ccccc21)NC(CCC(C)C)C(=O)NC1CCCC1CF 32941,c1(CN(CCC(=O)N(CC)CC)CCC)cn(C2CC2)nc1C 32942,N1(C(CC2CCC(=O)C2)=O)CC2(CCC(CNC(c3ccoc3)=O)O2)C1 32943,C1(C(=O)NCC2(NC(c3cnc(-c4ccco4)s3)=O)CC2)CCC2(CC2)C1 32944,C1(O)(CN(C(C2CCN(C)C2)=O)C)CCN(C(=O)CCc2cnn[nH]2)CC1 32945,c1(NC(c2ccn(C(C)C)n2)c2nnnn2CCC2CC2)cccc2[nH]ccc12 32946,C1(C)(COC)CC(NC(C2CN(C)C2)=O)CN1C(=O)CCc1nncs1 32947,CCCC(CCC)CC(=O)N(C(C)C(=O)NCCCCCO)C1CC1 32948,c1(C(=O)NC2(CNC(C3C(CC)C3)=O)CC2)cncc(Cl)c1C 32949,N1(C(c2c(CC)noc2)=O)CC2CC(C)N(C(c3cn(C)nc3Br)=O)C2C1 32950,c1(OC)cc(F)cc(C=CC(N2CCC2CNC(c2c[nH]c(C#N)c2)=O)=O)c1 32951,c1(C(N2CC3(CC(NC(C4(F)CCOC4)=O)C3)C2)=O)ccc2nc(O)oc2c1 32952,C#Cc1cc(F)c(CN2CCN(C)C(CO)C2)c(F)c1 32953,N1(C(C2(C)CC2)=O)CC2CCCC2(NC(=O)CSCc2csc(=N)[nH]2)C1 32954,C1(OCC)CC2(CCN(C(=O)CC=CC(C)(C)C)C2)C1.C12C(C1(C)C)NC2=O 32955,c1(NC(C2C(NC(C(C)Sc3ccccn3)=O)C2)=O)ccnc2ncnn12 32956,CC(C)(Cc1ccccc1)C(=O)N1CCCC1CNC(c1c[nH]ccc1=O)=O 32957,C1(C)(CNC(CN(C)CC)=O)CCCN1C(=O)Cc1cc(C)no1 32958,C(=O)(N=c1c(Cl)c[nH]cc1Br)C1C=CC(NC(c2c(C)noc2)=O)C1 32959,C(=O)(CC(F)(F)Cl)NC(C(CO)NC(CCCNC(=O)OC)=O)C 32960,Cc1cc(C(=O)NC2C3CC2N(C(=O)C(C)OCc2ccncc2)C3)cc(C)n1 32961,N1(C(c2ccc(CC)cc2O)=O)CCC2(CC(NC(=O)C(C)OCOC)C2)C1 32962,Cn1nncc1CC(=O)N(CCN(C(CC(=O)NCC(F)(F)F)=O)O)C1CC1 32963,c1(C(N2CCC(CNC(C3C(OCC)C3)=O)C2)=O)ccc(-c2ccc(Cl)s2)cn1 32964,C1(NC(c2ccsn2)=O)C2CC3C1C3C2C(N1CC(n2cccn2)C1)=O 32965,N1(C(c2c(OC)noc2C)=O)CCCC(NC(=O)CCCCN(C)C)CC1 32966,C(=O)C(O)C(F)(F)F.C1(CCC2C(=O)CC2(C)C)COCCN1N(C)C=O 32967,c1(-c2n(CCN(C)C)ccc2)ccc(C(=O)NCc2ccccc2)nn1 32968,c1(N(C)CCn2cccn2)ccnc(NCC2CC2(F)F)n1 32969,C1(N(C(C2(CC)CCC2)=O)C)CC2CCC(C1)N2C(c1occ2c1CCC2)=O 32970,C1(OC)CC(CO)(NC(=O)CC2C=CC(NC(=O)CCCC3CC3C)C2)C1 32971,C=CCCCCCCCCC(C(=O)NC1CCC1)N(C)CCc1cnn(C)c1 32972,N1(C(C2C3(CCN(C(c4c(CC)ncs4)=O)C3)C2)=O)CCc2c(C)cccc2C1 32973,N1(C(C2(NC(C)=O)CC2)=O)CCC(NC(=O)Cc2nocc2C)C1 32974,c1(C(C(=O)NCCCC)N(C)C)cn(CCCN2CCC(C(=O)N(C)C)C2)nn1 32975,c1(N2CCC(CNC(C(C)CN3CCOCC3)=O)C2)cccc(O)n1 32976,S(=O)(=O)(c1ccc(Br)cc1)NCC(=O)NCCNC(c1cccc(CO)c1)=O 32977,N1(C(C2C(C)CCS2)=O)CC(C2CN(C(=O)CCCCC(N)=O)C2)C1 32978,N1(C(c2cnc(Br)s2)C(=O)NCCSC)CCCC(n2ccnc2C)C1 32979,N1(C(CCCCSC)=O)CC(NC(c2nc(C3CC3)ncc2Cl)=O)C(C2CC2)C1 32980,c1(CC(=O)NC(CC)CN(C(=O)C(C2CC2)SC)C)cc(F)ccc1C 32981,N1(C(c2ccc(CSC)cc2)=O)CCCN(C(=O)COC(F)(F)F)C(CO)C1 32982,N1(C(c2ccn(C(C)(C)C)n2)=O)CCOC(CCNC(c2nocc2Cl)=O)C1 32983,C(C(C(C)(C)C)NC(C1(C)CCCO1)=O)NC(=O)Cc1csc(C(F)(F)F)n1 32984,CCC(C)(C)CCNC(=O)C=CC(C)(C)NC(=O)C(C)C(F)F 32985,c1(C(C)OC)ccc(CNC(=NCc2snnc2C)NC2CCC2)cc1 32986,Cc1c(CNC(C)(CCc2ccsc2)c2nnnn2C2CCCC2)cccc1Br 32987,N1(c2nc(=N)nc(N3CCCC(CCN(C)C)CC3)[nH]2)CCCC(C2(C)CC2)C1 32988,C(CCF)(C(=O)NCCN(CC)CC)NC(C(CC)NC(=O)CCC)=O 32989,C(=O)(C1=C2CCCN=C2NN1)NC(CCCOC)c1cccnc1 32990,C1(C(N2CCC(=CCNC(C(CCC)NC(N)=O)=O)CC2)=O)CCCS(=O)(=O)C1 32991,C1(COC)CN(C(c2cc(C#N)[nH]c2C)=O)CCN1C(=O)C1=C(Cl)CCC1 32992,C1(OC)CCn2cc(C(=O)NCC3CCC(NC(=O)CC(C)(C)C)CC3)nc2C1 32993,C(c1cncnc1O)=CC(N1CCC(C(C)NC(=O)CC(F)(F)F)C1)=O 32994,N1(C(Cc2cc(C)[nH]n2)=O)CCOCC(C)(CNC(C2CCC2C(C)(C)C)=O)C1 32995,N1(C(c2n(C)cnc2)=O)CCOC(C2CN(C(C3CC=CCC3)=O)C2)C1 32996,C1(CC)CCC(C(N2CC(N(C)C(c3ccc(-c4ccccn4)s3)=O)C2)=O)C1 32997,N1(C(C(C)N(C(C(CCCC#C)C)=O)CC)=O)CC2CCC1C(O)C2O 32998,c1(C(N(CCCCNC(C(CCC)O)=O)C)=O)cc(F)cc2c1NCCC2 32999,C1(C(N(CC(CNC(C(C)C2(O)CCC2)=O)(C)C)C)=O)CCCC1P(C)(C)=O 33000,c1(C(=O)NCCN(CCOC)C(c2nnn(C)c2C)=O)cc2ncn(C)c2cn1 33001,c1(CN2CCC(N(C(=O)CCCN3CCCCC3)CC)C2)ccc2nonc2c1 33002,Cc1cc(C(=O)NCCC2(NC(=O)CCC(=O)N(C)C(C)C)CCCC2)c(C)cn1 33003,Cc1nn(C2CCCCC2)c(C)c1S(=O)(=O)Nc1cc(Br)nn1C 33004,CC(C(C)(C)C)=CC(=O)NCCCOCCC(=O)NCC1=CCCC1 33005,c1(CNC(=O)NCC(c2cccc(OC)c2)(C)C)cc2nc(F)ccc2o1 33006,S(=O)(=O)(c1cccc(C#N)c1)N1C2CC(NC(c3cn(C)nc3)=O)CC1CC2 33007,[N-]=[N+]=NC1CCC(C(=O)NC2CCN(C(c3cc(-c4cccs4)on3)=O)CC2)C1 33008,C(c1cnc2ccccc2n1)=CC(=O)NC1C2CN(C(C(C)(C)CF)=O)C1CC2 33009,c1(C(=O)NCCCOCCN(C)C(c2ccccn2)=O)cc(Cl)cs1 33010,Cc1cc(C)c2cc(C(=O)NCC(CO)NC(c3ccncc3Cl)=O)[nH]c2c1C 33011,C1(C(=O)NCCC2COCCN2C(=O)C(O)CCSC)(CC)CCC(O)CC1 33012,C(=O)(CCC(C)C)NC1(c2ccccc2)CN(C(CC2C(CC)C2(F)F)=O)C1 33013,C(c1cccc(F)c1)=CCC(=O)NC1COCCC1NC(c1cccnc1)=O 33014,c1(OC)ncnc(C(=O)NC2CC23CC(NC(=O)C(F)(F)C(O)C2CC2)C3)c1F 33015,Cc1cc(=NCC2CCCN(C(C3(F)CC4(CCC4)C3)=O)C2)[nH]c(C2CC2)n1 33016,N1(C(CC2CCC(NC(COC3(C#C)COC3)=O)CC2)=O)CCC(O)C(C)C1 33017,N1(C(C(CC=C)C)=O)CC(NC(c2cccc(C(F)F)n2)=O)C2(CCOCC2)C1 33018,c1(C(N2CC(C=C)C(NC(c3[nH]c(C)nc3C)=O)C2)=O)nn(C)c2c1C(O)CCC2 33019,N1(C(C2(C)COC2)=O)CCCC2CN(C(=O)C(C#N)C3CC3)CC12 33020,N1(C(C2C(C)CC(=O)N2)=O)CCC2(C1)CN(C(=O)CC1CCCC(F)(F)C1)C2 33021,c1(CNC(=NC)N(C)Cc2conc2CC)cccc2c1OCCO2 33022,c1(CC)ccc(NC(=O)C(CC2CCCC2)NC(C2CCC(COC)O2)=O)cc1 33023,CC(CC(C)(C)C)C(=O)N1CC2(CCN(C(=O)C(C)NC3(CO)CCCC3)C2)C1 33024,C1(C(=O)NCC(C(C)(C)C)NC(=O)C=Cc2ccc[nH]2)CC2CCC1CC2 33025,n1(CCCC)ncc(C(=O)NCC2(Nc3nnc(C(C)(C)C)s3)CC2)c1C 33026,N1(C(CNC(CCC)=O)=O)CCC(C(C)C)CC1CNC(=O)C(F)(F)C(F)F 33027,C(=O)(C(C)(O)C(F)(F)F)N1CC(C(C)C)C(C(N2CCC(C)(C)C2C)=O)C1 33028,C(=O)(C(C)CC(F)(F)F)NCC1CN(C(c2c(C(C)C)ncs2)=O)CC1(F)F 33029,N1(C(CC2N(C)CCC2)=O)CCC(CC(N)=O)(NC(=O)Cc2nccn2C)CC1 33030,CCC(CC)CCCC(=O)NC(CNC(C1CC(=O)N(OC)C1)=O)CC(C)C 33031,N1(C(C(CC(C)C)=O)=O)CCc2nc(O)cc(C(=O)NCCc3nccs3)c2C1 33032,C(=O)(CCCS(N)(=O)=O)NCC1C(NC(c2ncc(C)cc2C)=O)CCCC1 33033,N1(C(C2(Nc3ccccc3)CC2)=O)CCOCC(NC(c2ccsc2)=O)C1 33034,c1(C(=O)NCCC(C)NC(c2c(OC)cncc2)=O)cc(Br)c(C)nc1O 33035,C(=O)(C(CC(C)(C)C)OC)NC1C(OC)CN(C(=O)CSC2CC2)C1 33036,c1(CC(N2CCC(NC(=O)CC3CN4CCN3CC4)C2)=O)cc(F)c(F)cc1F 33037,Cc1nc2sccn2c1C(N1CCC(C)(CNC(C2CC3CC3C2)=O)C1)=O 33038,C1(CCNC(CC(C)(C)C)=O)CN(C(C2CC2c2cccc(F)c2)=O)CCCO1 33039,N1(C(C)=O)CC2OC(=O)N(C3CCN(C(c4cc(O)n(C)n4)=O)CC3)C2C1 33040,C1(NC(=O)C2=CCCC2)C2CC3C1C3C2C(=O)NCc1cccc(F)c1O 33041,C(=O)(C(C(C)C)n1cc(Br)cn1)N(CCNC(=O)CSC(C)(C)C)CC 33042,CC(=NOCC#N)C(=O)N1CCN(CCNC(c2oc(C)cc2C)=O)CC1 33043,N1(C(CCC)=O)CC(OC)CC1(C)CNC(c1ccc(C)nc1O)=O 33044,C1(C(=O)NCc2c(C)noc2)CCC(NC(=O)C(C)(C)C2CCC2)CC1 33045,C1(O)(C(C)NC(=O)CCNS(C)(=O)=O)CCN(C(=O)CSC(F)(F)F)CC1 33046,C1(OC)(CNC(c2sccc2Br)c2nnnn2CCCF)CCCOC1 33047,C(C(C)(O)CC(=O)N1CC2(CC2)CC1CC(=O)N(CC(C)CO)C)OC 33048,N1(C(COCc2c(C)ncs2)=O)CCC(C)C(NC(C2CC(C)(C)C2)=O)C1C 33049,c1(C(=O)NC2CC(NC(c3c(S(N)(=O)=O)ccs3)=O)C2)cnc2c(c1)CCCO2 33050,c1(C(=O)NC(CN(C(CSCC)=O)C)C)cc(C)c2nc(C)nn2c1 33051,C#CC1(C)CCCN(C(=O)C(=O)NC(c2cccc(C(F)(F)F)c2)COC)C1 33052,N1(C(C2CC(OC)C2)=O)CC(NC(c2cc(C)cc(O)n2)=O)C2(CCC2)C1 33053,N1(C(c2n(CC)ncc2)=O)CC2CC(C1)CN(C(=O)COC1CC1)C2 33054,C1(CC(=O)NC(CCC)CNC(c2cn(C(C)C)cn2)=O)CCCC(F)(F)C1 33055,C1(N(C(CCc2c(C)n[nH]c2C)=O)C)CCCCN(C(C2CCOC2)=O)C1 33056,C1(COC)(NC(c2cnn(C)c2F)=O)CCN(C(=O)CC2CCCO2)CC1 33057,N1(S(=O)(=O)CCCl)CC2CCC(C1)N2Cc1ncccc1F 33058,CC(C)CCC(C(=O)N(CC(O)CO)C)NC(=O)CCc1cccnc1 33059,Cc1cc(Cl)c(C(=O)NC2CC2NC(=O)Cn2cnc([N+](=O)[O-])c2)c(Cl)c1 33060,CCCC(C)CCCC(=O)N(CC(O)CN(C(=O)Cc1nonc1C)C)C 33061,C1(CC(=O)OC)CCCC2(CN(C(=O)CCc3cnn(C)c3)C2)O1 33062,c1(C(C(=O)NC)N(CCCCN2CCCCC2C)C)cc2c(Br)cccc2o1 33063,c1(C(N2CC(CNC(C(C)(C)C3CCC3)=O)C3C2C3)=O)cccc2c1CCC2=O 33064,C1(C(=O)NCCN(CCC)C(c2c[nH]c(=N)s2)=O)COCCN1CC(F)F 33065,C1(CNC(=O)Cn2cncn2)CN(C(C2CC3CC(=O)C2O3)=O)CC1(F)F 33066,c1(C(N(CCNC(=O)C(C)OCC(F)(F)F)CC)=O)cn2nc(C)cc2[nH]c1=O 33067,c1(CC)ccc(C(=O)NC(C)C(C)NC(c2ccc(C3CC3)nc2)=O)cc1F 33068,Cc1cc(C(N2CCC3(CC3C(=O)NCCCC3CCCCC3)C2)=O)nc(C)n1 33069,CN1N=C(C(=O)N2CC3CCOCC3(NC(=O)CCc3cnc[nH]3)C2)CCC1=O 33070,C(=O)(CCC(F)(F)F)NCCN1CCN(C(c2ccnc(C(C)(C)C)n2)=O)CC1 33071,N1(C(c2cc(C(C)=O)oc2C)=O)CCCN(C(C2(OC)CCCCC2)=O)CC1C 33072,N1(C(=O)C2CC2)CC2CN(C(=O)Cn3ccc(C(F)F)n3)CC2C1 33073,Cn1cnc2c1CCCC2C(=O)NC1CCN(C(=O)CN2CSCC2=O)CC1F 33074,C1(NC(C(C)N(C(=O)CN2CC(=O)NC2=O)C)=O)CN(C)NC1=O 33075,c1(C(=O)NCC(C(C)C)NC(C(CC#C)C)=O)cccc(S(=O)(=O)C(F)F)c1 33076,C1(CCNC(c2cc(C)nnc2)=O)CN(C(C2C(C)(C)OC2(C)C)=O)CC(C)O1 33077,C(CC(CNC(=O)C(C1CCCCC1)OC)NC(=O)CC1CC(OC)C1)OC 33078,c1(SC)cc(Br)ccc1C(N1CCC1CNC(=O)C#CC(=O)N(C)C)=O 33079,N1(C(C2(CC)CCCC2)=O)CC2CC1CN2Cc1ccc(OC(F)F)c(OC)c1 33080,C(=O)(C(C(C)C)NC=O)N(C1CCN(C(=O)C(c2ccccc2)SC)CC1)CC 33081,c1(C(=O)NCC2C(NC(C(C)OCC=C)=O)CC2)c[nH]c2c(C#N)cccc12 33082,N1(CC(=O)N(CCCN(C(c2c(NC)cnnc2)=O)C)C)C(=O)CC(C)(C)C1=O 33083,c1(C(N2CCC(NC(C3N(N=O)CCC3)=O)C2)=O)cc(C2CC2)cc(F)c1 33084,Nc1cc(Cl)ccc1C(N1CC2(C1)CN(C(c1coc(C(N)=O)c1)=O)C2)=O 33085,CCCCC(O)C(=O)N1CCCC1C(C)NC(c1ccncc1C)=O 33086,c1(C(C(=O)NC2C(NC(c3cn(CCC)nc3)=O)CC2)C)ccc(C#N)cc1 33087,c1(CN(C)Cc2nc(CCC)sc2)cccc(I)c1 33088,C1(OC)CN(C(c2ncn(C)c2C)=O)CC1NC(C1(OC)CC(CF)C1)=O 33089,Nc1c(F)ccc(F)c1C(N1CCCOC(CNC(C2CC2C2CCC2)=O)C1)=O 33090,c1(CC2(C(=O)NC(C3CN(C(Cc4nnc(C)o4)=O)C3)C)CC2)ccc(F)cc1 33091,Cc1nc(NC(CNC(C2CC3CC3C2)=O)C(C)C(C)C)[nH]c(=N)n1 33092,C1(NC(C)=O)CCC(C(=O)NCCN2CCCC2=O)OC1 33093,Cn1nc(-c2cn(CC3CCN(C(=O)C(Br)Br)C3)nn2)cc1N 33094,c1(C(N(C2CN(C(C3(S(C)(=O)=O)CC3)=O)CC2F)C)=O)ncnc2c1ccn2C 33095,CC1(CNC(c2cc(C(F)F)no2)=O)CCN(C(C2(C3CCCO3)CC2)=O)CC1 33096,c1(C(N(CCC(C)NC(c2ccoc2C2CC2)=O)C)=O)csc(C(N)=O)n1 33097,c1(-c2nc(C(C)SCC)nn2CC)cnn2c1CC(C)CC2 33098,c1(CC(C)C)ccc(C(=O)NCC2CC2NC(=O)CC(C)CF)cc1 33099,c1(C(=O)NC2(CC=C)CC2)ccc(CNC(=O)CC(Cl)Cl)nc1 33100,C1(NC(C(N2CCNC2=O)C)=O)C2CC1N(C(C1CCSC1)=O)C2 33101,C1(NC(CCCC#CC)=O)CN(C(c2ccc(CC)[nH]2)=O)CC2(CCOCC2)C1 33102,C(c1cccc(F)c1)=C(C(=O)NC1C=CCN(C(c2c(CC)onc2C)=O)C1)F 33103,Cc1cccc(C(O)C(N2CCOC(CNC(=O)CCc3nnc(C)s3)C2)=O)c1 33104,N1(C(c2cc(OC)nc(C)c2)=O)CCC(N=c2nn[nH]n2C)C(C)C1 33105,C1(C(=O)NC2CC(F)(CNC(C(C)OCCC#C)=O)C2)CCC(C(=O)OC)CC1 33106,C1(C(=O)NCCC2OCCN(C(c3n(CC)ncn3)=O)C2)CCCCC12CCC2 33107,C(CC(O)CC(=O)NCCCN(C(=O)CCCC(N)=O)Cc1ccccc1)SC 33108,c1(CC(C)C)cc(C(=O)NCC(C)NC(=O)CCc2cccnc2F)cc(O)n1 33109,c1(C(=O)NCCN(C(c2csc(C(=O)OC)c2)=O)CC)ccc(CC(C)C)nc1 33110,CCCCC(C(=O)N1CCCOC(CNC(=O)CCc2scnc2C)C1)N(C)C 33111,Cc1ccc(C(N2CCC(N(C(=O)C(O)Cn3cncn3)C)C2)=O)cc1 33112,Cc1scc(CNC(=O)C(C2CC2)NC(=O)C(C)NC=O)c1C 33113,c1(N2CCC(CC)(CO)C2)nc(=NCC(C)(C)SC)[nH]c2ncn(C)c12 33114,C1(Cn2cc(C(C(C)(C)C)O)nn2)CCCN(C(=O)C(c2cscn2)N(C)C)C1 33115,c1(OC)cccc2c1OCCC2NS(=O)(=O)c1c(Br)cc(C(=O)O)cc1Br 33116,c1(OC)ncccc1C(=O)NCCCC(=O)NC(C)Cc1cnccn1 33117,N(C(=NC(C)C)N1CCCCC(S(C)(=O)=O)C1)C(C#C)C(C)(C)OC 33118,N1(C(c2c(OC)cc(C)cn2)=O)CC(NC(=O)C2=CCCC2C)C(N=[N+]=[N-])C1 33119,CC1CCC(C2CC2)CN1CCCCOCF 33120,C(=O)(C#CC1CCCOC1)N1CC(CNC(c2cc(NC(C)=O)c(F)cc2)=O)C1 33121,c1(C(N(C)CC2CCN(C(=O)Cc3cncc(F)c3)C2)=O)cnc(N)c(N)c1 33122,Cc1ccc(C(=O)N(C)CC2CCCN2C(=O)CC2CC(CF)C2)cc1N 33123,c1(C(N2CCC(O)(C(C)NC(=O)CN3CCC(O)CC3)C2)=O)ccc2c(c1)CC2 33124,C#CCCC(C(=O)NC1CCCC(C)(C)C1)NC(C1CC2(C1)CC(C)C2)=O 33125,N1(C(C2CC(=O)N2)=O)Cc2ccc(CNC(c3ccc4nn[nH]c4n3)=O)cc2C1 33126,c1(C(=O)NCC2N(C(c3c(C)con3)=O)CC(O)C2)ccc2nc[nH]c2n1 33127,N1(C(C2CCC(CC)C2)=O)CCCN(C(c2cnn(CC)c2)=O)CCC1 33128,N1(C(CCC=C)=O)CCOC(CC(=O)N(C2CC2(C)C)C)C1 33129,C12(NC(C3CCc4cnnn4C3)=O)CCCC1N(C(=O)C=Cc1cscn1)CC2 33130,N1(C(c2n(CC)cnn2)=O)CC2CCCC2(NC(=O)Cc2n[nH]c(C)n2)C1 33131,C1(NC(C(C)SC)=O)CCN(CCNC(c2ncoc2C)=O)CC1 33132,C1(NC(C(C)NS(CC)(=O)=O)=O)CN(C(C2CCS2(=O)=O)=O)CCC1C(F)(F)F 33133,C(CC(C(=O)NC1CCN(C(C)=O)C1)NC(C1CCCSC1C)=O)=CC 33134,CC1(NC(C2CCCOC2)=O)CN(C(=O)C=Cc2ncco2)C1 33135,C1(F)(CNC(c2c(C)nco2)=O)CCCN(C(c2ccnn2C2CCC2)=O)C1 33136,CCC(C)C(CO)NC(=O)C(CC1CC1)NC(c1cc(C#N)cs1)=O 33137,CCC(C)CCCCC(=O)NOCC(=O)NC(C)C(=O)NC 33138,C(=O)(C(C)(C)CO)NC(C)C(C)NC(=O)CCOc1cccc(Br)c1 33139,C(=O)(CCCCC1CCCCC1)N(CCCN(C(CCCNC(=O)OC)=O)C)C 33140,C1(NC(CC(CC)C)=O)(CC)CCN(C(=O)CC23CCC(CC2)CC3)CC1 33141,Cc1cc(C(=O)NC(CC2CC2)C(=O)Nc2ccccc2CCO)ccn1 33142,C1(N(C(c2csnn2)=O)CCSc2nc(C3CC3)cs2)CCN(CC)CC1 33143,CC1CC(NC(c2ccns2)=O)CN1C(c1cc(Cn2cccn2)on1)=O 33144,c1(C(=O)NCC(CNC(=O)CCSC(F)(F)F)OC)cc(C(C)(C)O)ccn1 33145,N1(C(Cc2c(C)ccs2)=O)CCOC2(C1)CN(C(=O)CCC1CC(C)(C)CO1)C2 33146,n1(CC#C)c(C)cc(C(=O)NCC2(OC)CCN(C(=O)CC3CC3(C)C)C2)c1C 33147,N1(C(c2n(C(C)C)ncc2)=O)CCOC2(C1)CN(C(=O)C(C)CS(C)=O)C2 33148,CCC(C(=O)OC)C(=O)NCC(CC)NC(C1(c2cc[nH]n2)CCC1)=O 33149,c1(COC(C(=O)N(C2CCN(C(C3(OC)CC3)=O)C2)CCC)C)ccncc1 33150,N1(C(C2(CC)CCOC2)=O)CCCC(C)(CNC(c2csc(CC(C)C)n2)=O)C1 33151,c1(OC)ccc(CCC(=O)NC2CN(C(=O)CN(C)CCO)C3CC23)c(OC)c1 33152,C(=O)(CC1OCCc2ccccc21)N(CCCNC(c1csc2nnsc12)=O)C 33153,C1(OC)CC2CCC(C1)N2C(=O)CCCN(C)C(C1(C)CNC(=O)C1)=O 33154,c1(C(N(C2CCCN(C(C3C=CCC3)=O)C2)C)=O)cc(Br)cc2nc[nH]c12 33155,N1(C(COCCCOC)=O)CC2(C1)SCCC2NC(=O)C(O)P(C)(C)=O 33156,O=C(C1=CCCCO1)NCCC(O)CNC(C1(c2cc(Br)ccn2)CC1)=O 33157,c1(C(=O)NCC2(NC(C(C)Cc3ccco3)=O)CCCC2)cn(C)nc1C1CC1 33158,c1(NC(C2CN(C(C3C=CCS3)=O)CC2C(F)F)=O)nccnc1-n1ccnc1 33159,CCC(C#N)(CC)C(=O)N1CC2CC1(CNC(=O)Cn1nc(C)ccc1=O)C2 33160,c1(C(=O)NC(CCC)CNC(C23CCCC2CCC3)=O)cc(C)cc(C)c1C 33161,N1(C(C(C)N(C(=O)CC(C)CC)CCC)=O)CC(CO)C(C)(C)C1 33162,C1(NC(CC(CC2CC2)NC(c2cc(C)[nH]n2)=O)=O)CC2C(O)C(O)CC12 33163,c1(NC(C2CCN(C(c3cn(CCC(C)C)nn3)=O)CC2)C)nccc(C#N)n1 33164,C(C)(CCC(=O)NC(c1nnc(O)n1C)C)NC(CCOCC)=O 33165,c1(C(N(C(C)CNC(C2CC2F)=O)C)=O)cc(Br)nn1C 33166,N1(C(CCSC)=O)CCCC2(CCN(C(c3c(N)cc(Cl)cc3Cl)=O)C2)C1 33167,CN1N=CC(CC(N2CCOCC2CCNC(=O)CCC(N)=O)=O)C1=O 33168,C1(CC(C)C)(CC)CCN(C(C2(O)CC2)OC(c2cccnc2)=O)C1 33169,c1(C(=O)NC(CC(C)NC(c2cc(Cl)cnc2O)=O)C)csc(S(N)(=O)=O)c1 33170,Cc1ccc(CCC(N2CCN(C(C34CSCC3C4)=O)C3CC23)=O)c(C)c1 33171,c1(CNC(=O)NC(c2ccccc2)CCO)cc(C(F)(F)F)cnc1O 33172,c1(C(N2C3CC(CNC(C(CCC)(C)C)=O)C2CC3)=O)cc2n(n1)C(C)CCC2 33173,c1(C(C(=O)NCC(C)NC(CCOc2ccc(C)cc2)=O)O)ccc(F)c(F)c1 33174,C(CC)(CCC(=O)OC)NC(c1cccc(-c2cc(F)ncc2O)c1)C(=O)OC 33175,C(CC(=O)NC(C1CN(C(c2nc[nH]c2C(F)(F)F)=O)C1)C)(C(F)(F)F)OC 33176,N1(C(C2C3CCC(F)C23)=O)CC2CCCC2(C(N2CCCCC2CO)=O)C1 33177,c1(C(=O)OC)nc(COC(=O)CC(c2ccc(F)cc2)C)n(C)n1 33178,N1(C(CC(C=C)(C)O)=O)CC(NC(c2cnn(C(C)C)c2)=O)C(N=[N+]=[N-])C1 33179,C1(C)(CNC(CC2C=CC(NC(CC(C)SC)=O)C2)=O)CC(C)=NO1 33180,N1(C(C(C)SCC)=O)CCCC12CCCN(C(C1(C)CCCCCC1)=O)C2 33181,C1(N(C(CCc2onc(C)n2)=O)C)CCN(C(c2coc(C)c2)=O)CC1C 33182,Cn1cc(C(=O)NCC(O)CCNC(c2ccn(C3CC3(F)F)n2)=O)ccc1=O 33183,C(=O)(CC(C(F)(F)F)n1cccn1)NC(C(CC)C)CO.C12=CC=C(C=C1)C2=O 33184,c1(OCCNC(=O)NCC2CCOC(c3ccccc3)O2)c(Cl)cccc1Cl 33185,CCCC(C(=O)NC(C)CC)NC(=O)CC1CC2CC2C1 33186,C1(NC(c2cnc3[nH]nnc3c2)=O)CC2CN(C(c3occc3Cl)=O)CC2C1 33187,n1(C(C)(C)C)ccc(S(=O)(=O)NNC(=O)c2cc(-c3ccc(F)cc3F)on2)n1 33188,c1(NC(C23CC(NC(c4ccc(CC)cc4)=O)(C2)C3)=O)c(C=O)c(C)nn1C 33189,C1(C(=O)NOCC(N)=O)(CC=C)CCN(C(=O)C=CCOC(C)=O)C1 33190,c1(C(N2CC(C)C(CNC(C3CCC(C)(C)CC3)=O)C2)=O)ccc(S(N)(=O)=O)o1 33191,c1(C(=O)NC(CCCC)CNC(=O)CCCCC(C)C)coc2cc(F)ccc12 33192,c1(OC)cc(C#N)ccc1-c1c[nH]nc1C(=O)Nc1ccc2c(c1)OCO2 33193,C1(C(=O)NC2CC(CNC(c3cn(C)c(=O)cn3)=O)C2)CCCC1S(C)(=O)=O 33194,CC1CCC(CO)(NC(C2(N)CC2)=O)c2ccccc21 33195,C(CS(=O)(=O)CC(=O)N(C1CN(C(=O)CCc2ccncn2)CC1(C)C)C)OC 33196,C1(NC(=O)CCc2nncs2)CC2CC1CN(C(c1noc3c1CCCC3)=O)C2 33197,C(=O)(C1c2c[nH]nc2CN1C(=O)C(CO)N(C(=O)C1CC1)CC)N(C(CC(C)C)CO)C 33198,C(CCNC(=O)CCc1cccnc1F)(C(C)(C)C)N(C(=O)CC(C)(C)C)C 33199,C1(N(C(c2c(C)nco2)=O)C)CCCC(NC(=O)C(c2cc(Br)co2)=O)C1 33200,N1(C(C(CCC)OCC)=O)CCC2(CC1)CC2C(=O)NC(CC(C)C)c1ccco1 33201,N1(CC)CCN(C(C(=O)NC(C)C(=O)OC)c2csnn2)CC1(C)C 33202,C12(NC(C(CC3CC3)NC(c3nc[nH]n3)=O)=O)CCCCC1OCC2 33203,N1(C(C=CC(C)C)=O)CCC(NC(C2CCS(=O)(=O)C2)=O)C12CCC2 33204,CCCC(C(=O)NOC)NC(C1CC1OC(C)=O)=O 33205,C1(NC(C2(C)CC2F)=O)CC2CCC1CC2NC(C1CCC(=O)N(C2CC2)C1)=O 33206,c1(N(C)C(N2CCCC(C(O)C(=O)OC(C)(C)C)C2)=O)cccc(O)c1 33207,Cc1nc(N2CCC(CNC(c3cncs3)=O)C(C)C2)c2ccsc2n1 33208,C1(C)(C(N(CC#C)CC=C)=O)CC(O)CN1C(c1cnnn1CC)=O 33209,C1(C(N2C(C(=O)O)CCC2)=O)COC2(CCC2)CO1.C12CCC(CC1)C2 33210,C1(C2(O)CN(C(c3oc(SC)cc3C)=O)C2)(CNC(C(C=C=C)C)=O)CC1 33211,c1(OC)cc(CNC2CC2C(N2CC(OC)CC2CO)=O)c(Cl)cn1 33212,N1(C(Cc2ccc(C(=O)OC)s2)=O)CC(C)CN(C(=O)CNC(C)=O)CC1C 33213,c1(N2C(CCNC(c3n[nH]cc3Cl)=O)CCC2)cc(C(F)F)ncn1 33214,c1(C(N2CCN(C(=O)C=CBr)C(CC3CC3)C2)=O)cccc2nonc12 33215,C1(CNC(CSCC)=O)N(C(c2cc(C(C)(C)C)on2)=O)CCCC1(C)C 33216,C1(C(=O)NCCCCN(CCCNC(C(C)OCC)=O)C)CC(=O)N(OC)C1 33217,N1(C(C(CC)NC(C)=O)=O)CCCN(C(c2ncccc2C(=O)OC)=O)CC1C 33218,C1(CNC(CSCC=C)=O)CC(C)N(C(c2cn(C)c(O)n2)=O)C1 33219,C1(CCC)CCCN1S(=O)(=O)CCC1CCOCC1 33220,C1(C(=O)NC(C(=O)NCCC)CC)C2CCC(C2)C1NC(=O)CCCC(=O)NC 33221,N1(C(CC(C)n2cccn2)=O)CCC(N(C(=O)Cc2ccc(Cl)s2)CCO)CC1 33222,c1(C(=O)NCC2CCN(C(c3c(C)nc(C)o3)=O)C2)c(C)cc(F)cc1Br 33223,N1(CC(=O)NCc2ccsc2)CCC(C2CNC2)CC1 33224,N1(C(C(c2ccc(N)cn2)C)=O)CC2CC(C1)N(C(=O)CC1CCCC1O)C2 33225,C1(C(=O)NCC(CCC)(C)O)CCC2(CC2)N1C(C1CC2CCC2C1)=O 33226,Cc1ccc(NC(C2CN(C(c3sc(Cl)nc3Cl)=O)CCC2(F)F)=O)c(C#N)c1 33227,Cc1cc(CNC(C2(CCNC(=O)COCCCF)CC2)=O)c(C)s1 33228,C1(NC(c2n(C)c(S)nc2)=O)CC(O)CN(C(=O)CCCc2ccc(Cl)cc2)C1 33229,C(=O)(C(O)C(C)(C)C)N1CC(C(C(=O)NC2CC(C(=O)NCC)C2)OC)C1 33230,C1(C(=O)Nc2ccc(CCC(=O)NC)cc2)C2C=CC(C2)C1C(C)C 33231,Cc1ccc(C(C)C(=O)NCC2CN(C(=O)C=Cc3cn(C)cn3)CCO2)cc1 33232,n1(CCC)cc(C(=O)NCc2c[nH]nc2C2CCN(C(=O)C(F)OC)C2)cn1 33233,Cc1cnc(C(=O)NCC2CCCN(C(c3cncnc3C)=O)C2)cc1C 33234,C1(CNC(C(C)N(CC)CC)=O)(CO)CCCN(C(c2nc(C3CC3)cs2)=O)C1 33235,Cn1ccnc1C1CC1C(=O)NCC1(O)CN(C(c2ccccn2)=O)C1 33236,c1(C(N2CCC(C)(NC(C(C)n3ccnc3)=O)CC2)=O)ccc2sncc2c1 33237,N1(C(CS(C)(=O)=O)=O)CCC2CCC12CNC(=O)CCOc1ccc(F)c(Cl)c1 33238,CCC(F)(C(=O)OC)C(=O)NC(C)CNC(=O)COc1ccc(Cl)cc1 33239,N1(C(C2N(C(=O)CN3CCC(C)C3)CCC(C)C2)=O)CCCC(C2(C)CC2)C1 33240,N1(C(CCNC(=O)NC)=O)C2CCC1CC(NC(=O)CC1(CSC)CC1)C2 33241,C12CC(C(O)C1)N(CC)C2=O.c1(CN2C(C(=O)NC)CCC2)cccnc1 33242,Cn1cnc2cc(CC(=O)NCC3CC(NC(=O)C=C4CC4)C3)ccc12 33243,C(C(=O)N(CC(C)(C)CNC(c1nocc1C1CC1)=O)C)(C(C)C)SCC 33244,C12(C=CCN1C(c1occc1C)=O)C(=O)OC2.C=CC(C1CCC1)COCC 33245,CN1N=C(C(=O)N(CC(C)(C)C(=O)NC2CCC(=O)N(CCO)C2)C)CCC1=O 33246,C1(CC(=O)NCC(C)N(C(c2nnn(C(C)(C)C)n2)=O)CC)CCCC(C)(C)O1 33247,C1(C)(C(N2CC(CNC(c3c(COC)noc3)=O)C(O)C2)=O)CC2(CCC2)C1 33248,c1(C(=O)NCCC(=C)CNC(=O)C(C)(C)C(=C)Cl)cc2nc(C)cc(C)n2n1 33249,C1(C(N2CCC(N(C(=O)C(C)(C)C3CCCCO3)C)C2)=O)C(C)(C)OC1(C)C 33250,N(C1CCc2c(F)ccc(Br)c21)CC(=O)Nc1n(CC)ncc1 33251,N1(C(c2c(C)ccnn2)=O)CC(F)(F)CC1CNC(=O)C(N1C(=O)CCC1=O)C 33252,n1(CC)cnnc1C(=O)NC(C1CCCC1)CNC(=O)C(C)NS(=O)(=O)CCC 33253,c1(NC2(CNC(C3C(C)(COC)C3)=O)CCCC2)nc(C)nc(O)c1C 33254,c1(C(=O)NC(CNC(c2cc(C)ncc2)=O)(C)C)cc(N2CCCC2)nc(Cl)c1 33255,CCS(=O)(=O)CC(=O)NC1(CNC(C2CC2(C)C)=O)CC1 33256,N1(C(C=C(CCN(C)C)Cl)=O)CCOC2(C1)CN(C(C1CCCN1N=O)=O)C2 33257,c1(C(N2CC(=C(CNC(C3C(=C)C3)=O)F)C2)=O)n[nH]c(C(C)(C)C)n1 33258,C1(C(N2CCC(CNC(C(C)(C)Cc3cnn[nH]3)=O)CC2)=O)CN2CCN1CC2 33259,N1(C(c2c(CC)csc2)=O)Cc2ccccc2C(NC(C2CCNC2=O)=O)C1 33260,C(=O)(C1CSc2ccccc21)N(C)CC1CCN(c2ccc(C(C)=O)cn2)CC1 33261,Cc1ccc2[nH]cc(CC(N3CC(NC(C4(C(N)=O)CC4)=O)CC(O)C3)=O)c2c1 33262,c12ccc(cn1)CNC1CCCC1NC(=O)O2.c1(O)ccccc1.C1(SC)CC1 33263,C1(C(=O)NCC2(C(N)=O)CN(C(c3ccc(F)c(Cl)c3)=O)C2)CC2C(C1)C2(C)C 33264,C1(Cc2cn(CC(C3CC3)NC(C(C)OCC3CC3)=O)nn2)(OC)CCCCC1 33265,C1(NC(C=CC(CC)=CC)=O)CCCN(C(=O)CCc2ccncc2)CC1F 33266,c1(CC)cnc(O)c(C(=O)N(C)CC2CCCN2C(c2n[nH]cc2OC)=O)c1 33267,N1(C(C2CC3CC3C2)=O)CCC2(C1)c1[nH]cnc1CCN2C(C1(O)COC1)=O 33268,CC(C)CC(CNC(c1cocc1C(N)=O)=O)C(=O)NC(C)CC1CCC1 33269,c1(OCCC)cccc(C(=O)NC2CN(C(=O)C(C)=C3CCC3)CC2C)c1 33270,CCCC(CCCNC(=O)CC1CCCCCO1)NC(=O)CNC(=O)C(C)(C)C 33271,N1(C(c2scc(CNC(c3c(C)ocn3)=O)c2)=O)C2CCC1COC2 33272,Cc1cc(C(=O)N(C2CCN(C(c3cnc(N(C)C)o3)=O)CC2)C)c(C)nc1C 33273,c1(C(N(C2CC(NC(C3CCC(C)CC3)=O)C2)C)=O)cccc2nncn12 33274,C1(F)(CNC(CCOCCOC)=O)CCN(C(c2cnc(S)nc2)=O)C1 33275,N1(C(C2C3(CN(C(c4c(C)nn(C)c4C)=O)C3)C2)=O)C2CCC1CN(C)C2 33276,c1(C(C)C)cccc(C(=O)NCC(O)CNC(=O)CSC2CC2)c1N 33277,CC1(C)Cn2[nH]c(=NC(=O)NC(C3CC(F)(F)C3)C(=O)O)cc2CO1 33278,CN1CCC(NC(C2CCC(NC(C3(N(C)C)CCCC3)=O)C2)=O)C(C)(C)C1 33279,c1(C(c2n(C)nnn2)NCC(C)(C)OCCO)cc(Br)c(Br)o1 33280,C(=O)(CC(C)(C)C)NC(C)C(N1CCC(N(c2cc(Cl)ncn2)CCO)CC1)=O 33281,N1(CC)CCOCC1CC(=O)N(CCC(C)NC(=O)CN1CCN(C)CC1)C 33282,C(CCN=C(NCC(N1CC(C)OC(C)C1)(C)C)NCC(C)F)SC 33283,c1(C(=O)NC2C(NC(C=C(C)Cl)=O)CCC2)cccc(-n2ccnc2)c1 33284,c1(C(N(C(CC)CNC(=O)C(F)OC(F)(F)F)C)=O)cccc2nsnc12 33285,C(CCC(=O)NCCCN(C(=O)C(C)CN(C)C(=O)OC(C)(C)C)C)=CCC=C 33286,C1(C(N2CCC(N(C(c3cn(C)nc3O)=O)CC)C2)=O)CCc2nnc(O)n2C1 33287,c1(C(N(CCCN(C)C(C2CCC(CCO)CC2)=O)C)=O)cc2sccc2[nH]1 33288,N1(CC)CCC2(CC1)CC2C(N1CCC1(C)CC)C(=O)NC1CC2(CCC2)CO1 33289,C1(CNC(c2c(C)nc(O)[nH]2)=O)CN(C(=O)CC2CCC3(CCC3)O2)CCN1C 33290,N1(C(c2c(C)cn(C)c2)=O)CC(C)CN(C(=O)Cn2cnc(Br)c2)CC1C 33291,C(=O)(C(C)(O)CC)N1CC(CCO)(CNC(CCCOCCOCCCC)=O)C1 33292,C1(NC(C2C(CCC)C2)=O)CN(C(c2ccc(-n3cnnn3)cc2)=O)C(C)(C)C1 33293,C(CCS(C)=O)(C(=O)N1CC2C(NC(c3ccc(O)cn3)=O)C2C1)N(C)C 33294,c1(CC)onc(C(=O)NCC2CCC(N(C(=O)CC3CCOC3=O)C)CC2)c1C 33295,C1(C(=O)NCCn2ccc(C(N(CC)CC3CCCO3)=O)c2)C2CCC(C2)C1C 33296,C(=O)(C1CCCc2ncnn21)N1C(C)CC(NC(C2(OC)CCS(=O)(=O)C2)=O)C1 33297,Cc1nccnc1-c1cn(CCOCCNC(=O)CCNC(c2ccco2)=O)nn1 33298,c1(C(=O)NC2CCC(CCNC(CC(C=C)C)=O)C2)c(C)nc2sccn12 33299,c1(C(=O)NC2C(C)CN2C(=O)C=Cc2ccco2)ccnc(OCCO)c1 33300,C(CC1=CCOCC1)NC(=O)CC1CC(O)CN1C(c1cc(CO)on1)=O 33301,N1(C(CCOCC)=O)CCC(NC(c2cc(-c3ccccc3)[nH]c2C)=O)CC1C 33302,C1(CNC(CCc2cnc(C)s2)=O)CN(C)CCN1C(=O)CCc1cnc[nH]1 33303,N1(C(C(CC=C)(C)O)=O)CC=C(C(=O)NC(c2nc[nH]n2)CO)CC1 33304,CC(=Cn1ccnn1)C(=O)NCC12CCC(CN(C(c3cccnc3O)=O)C1)C2 33305,N1(C(Cc2cc(C)on2)=O)CC2(CCN(C(=O)CCC3CCCC(O)C3)CC2)C1 33306,c1(OC)cncnc1C(=O)N(C(C)C(=O)NC1CCCCC1F)C1CC1 33307,C1(COC)CCN(C(C)C(=O)NC(C)CCN2CCCCC2)CC1 33308,c1(C(=O)NCC(CNC(C2N(C(C)=O)CCC2)=O)O)cc2c(O)ccc(F)c2[nH]1 33309,c1(C(N(C(CNC(c2c(OC)n[nH]c2)=O)C)C)=O)cc2c(nn1)CCCC2 33310,C(=O)(C(C(C)(C)C)NC(c1ccnc(CNC(c2cnc(Br)s2)=O)c1)=O)NC 33311,CCN=c1[nH]cc(C(=O)NC2COCC2NC(c2nc(C)oc2C)=O)s1 33312,c1(CN2CC3N(C(C4CN(C)C4)=O)C(C3)C2)c[nH]c2ncc(Br)cc12 33313,N1(C(C2C(C)(C(F)F)C2)=O)C(C(N2CC(N3CCCCC3)C2)=O)CCC12CC2 33314,C1(NC(C2C(=C)CC2)=O)CCSC12CN(C(c1cnn(C3CCC3)n1)=O)C2 33315,CC1(C(=O)NCC2CCCCN2C(c2ccn(C3CCC3)n2)=O)CC2CCC1C2 33316,CCC(CC(F)(F)F)C(=O)NC(CC)(CC)CCNC(=O)CNC(=O)CC(C)(C)C 33317,N1(c2n(CC=C)c(C(O)CCOC)nn2)CCC(C)CC(C)C1 33318,C1(NC(c2c(C)con2)=O)CN(C(=O)Cc2ccns2)CCC12CCC2 33319,Cc1cc(C(N2CCN(Cc3ccccc3N(C)C)CC2)=O)nc(C2CC2)n1 33320,Cc1nc2sn(CC3CC(OC(F)F)C3)c(=O)c2c(C)c1C 33321,C1(NC(c2cnc(C)o2)=O)CCOC12CCN(C(c1cc(Br)c[nH]1)=O)CC2 33322,N1(C(c2nc(CCC)sc2)=O)CC2ON=C(CNC(c3nc(C)oc3C)=O)C2C1 33323,CC(C)CC(CNC(C1(F)CC1)=O)NC(C1(C(=O)C2CC2)CC1)=O 33324,CCCC(C)(O)CC(=O)N1C2CCC1C(CNC(=O)CC1(C(F)(F)F)CC1)C2 33325,N1(C(=O)CCc2nccs2)CCCCC1C(N1CCOC2CC12)=O 33326,c1(CC(=O)NC(C(C)NC(c2cc(C)c(C)nn2)=O)C)ccc2ncsc2c1 33327,c1(C(C(=O)N(C)CC2N(C(CN(C)CC)=O)CCC2)O)cccc(C)c1 33328,N1(CC(N2CCC(NC(=O)Cc3nc[nH]n3)(CO)C2)=O)CCS(=O)(=O)CC1 33329,N1(C(CC(=O)NC2CC2)=O)CCC(C(=O)NCc2cccc(F)c2)C12CCC2 33330,N1(C(CC(CC)OC)=O)CCCCC2(CCN(C(=O)OC(C)(C)C)C2)C1 33331,c1(NC(CN2CCCC(C(C)NC(C(C)C)=O)C2)=O)ccc(F)c(Br)c1 33332,c1(C(CC)(C)NC(=O)NC2(Cn3cnnc3)CC2)ccc(F)cc1 33333,Cc1cc(CN2CC(F)(F)CC2C(=O)Nc2nc(Cl)nc(Cl)n2)cnc1Cl 33334,C=CC(CCC)CC(=O)NC12CCC(NC(=O)C(O)CC(F)(F)F)(CC1)C2 33335,N12CCC3CN(CCC13)C(=O)CCC(=O)O2.c1(C(=O)O)ccsc1C(F)F 33336,N1(C(CC(C)(C)n2cc(-c3cnn(CCF)c3)nn2)=O)CC(C(=O)O)OCC12CC2 33337,C(C)(C)(CCCNC(=O)C(C)(C)C1CCCN1C(C1CCCO1)=O)OC 33338,CCCCCC(O)CC(=O)N(CCCCN(C(=O)CCc1ccccc1N)C)C 33339,C1(OC)CC(CC(=O)NCCC2CN(C(=O)CC(C)C)CCO2)C1(C)C 33340,N1(C(c2scc(C)c2Cl)=O)CCC2(CC1)OCCC2NC(C12CC(F)C1C2)=O 33341,C(=O)(CCC1=NNC(=O)CC1)NCCC(=O)NC1(C)CC(NC(=O)CO)C1 33342,S(=O)(=O)(c1cc(F)cc(Br)c1)N(C(=O)C(C)Oc1ccc(F)cc1)C(C)C 33343,N1(C(C(CSC)O)=O)CCC=CC1C(=O)N(CCO)CC1CC1 33344,c1(N2CCCC3(NC(c4ncc(F)cc4F)=O)C(C2)C3)ncc2cccnc2n1 33345,C(C)(C)(CCCCNC(C1(n2nccn2)CC1)=O)NC(C(CSC)OC)=O 33346,c1(C(N2CC=CC(NC(c3c(C)ccc(C)c3)=O)C2)=O)nn(C)c2c1CCCC2 33347,c1(C(=O)NCC2C(NC(c3c(CC)occ3)=O)CC2)cncnc1C1CC1 33348,c1(C(=O)NCCC(CNC(c2n(C)nc(C3CC3)c2)=O)O)ccc(F)cc1O 33349,C1(C2CCN(c3scc(C4CNCC(C)O4)n3)CC2)CCCN(CCO)C1=O 33350,N1(C(CCC=C)=O)CCc2ccccc2C1CCNC(=O)CCc1nnc(C)o1 33351,N1(C(C(COC)C)=O)CC(NC(c2cc(=O)n(C)o2)=O)CC12CCCCC2 33352,C1(C2CC2)(CNC(C(C(C)O)NC(C)=O)=O)CCN(C(=O)C2=C(C)OCC2)C1 33353,C=CCN=C(NCC(C1CCCCC1)(C)O)N1CCCC(CCC)C1 33354,c1(NC(N(CC(O)CO)CC)=O)cccnc1Sc1cnc(C)nc1 33355,CCC(O)C(C)C(=O)NC1CCC(CNC(c2cccc(C#N)c2)=O)CC1 33356,N1(C(c2c(SC)csc2)=O)CCCC(NC(=O)CC2CC2(C)C)C1 33357,C(=O)(CS(=O)(=O)C1CC1)NC(C(C)C)CCN(C)C(c1ccncc1N(C)C)=O 33358,Cc1cncc(C(=O)NCC=CCNC(c2cnc(C(C)C)n2C)=O)c1 33359,CCC(C)(C(=O)N1CC(O)(CCNC(=O)Cc2ncc(F)cc2F)C1)C(N)=O 33360,CN1CC(C(=O)NCC(C)(C)NC(=O)C=CC(F)F)CCC1=O 33361,N1(C(c2ccc(Br)o2)=O)CCC2(CCN(Cc3cccnc3Cl)C2)C1 33362,c1(C(=O)Nc2c(OC)cc(N3CCS(=O)(=O)CC3)cc2)nc2ncc(Br)cn2n1 33363,C1(C(N2C(C3(C(=O)NC(c4nc[nH]n4)CC)CC3)CCC2)=O)CC(F)C(=O)N1 33364,C1(CNC(C2N(CC)CC2)=O)CCC2(CCC2)CN1C(=O)C(Cl)=CCl 33365,c1(CC)nnsc1C(N1CC(CC(C)NC(c2cnn(CC(F)(F)F)c2)=O)C1)=O 33366,c1(OCC(NOCCCC(=O)OC)=O)cccc(C#N)c1 33367,C1(CCNC(c2cscn2)=O)CCN(C(c2cc(O)ncc2F)=O)CCC1(F)F 33368,c1(NC(CC2(C)CC2(Cl)Cl)=O)ccnc(-n2cc(-c3ncoc3C3CC3)nn2)c1 33369,Cc1cc(Cl)nc(N)c1C(=O)NCC1CC(C)CCN1C(C1CCCN1C=O)=O 33370,C(=O)(CCCCCN(C)C(C1CC12CCCCC2)=O)NCC1CN(CC)C(=O)O1 33371,Cc1ccc(CNC(C2C3CN(C(=O)CCc4ccoc4)CC23)=O)c(O)n1 33372,c1(C(=O)NCCCC(C)NC(=O)C2CC2)cccc(OCc2ccccc2F)c1 33373,CCCC(C#N)N(C)CCOCCN(C)C(C12CSCC1C2)=O 33374,C1(C(N(CCCNC(c2ccnn2C(C)C)=O)CC)=O)CCCC(CF)C1 33375,C(c1ccoc1)=CC(N1CCC(NC(=O)C(Cl)(Cl)Cl)C1)=O 33376,C1(CC)CC(CC(=O)NCC2CC(C)N(C(=O)C(C3CCC3)OC)C2)CCO1 33377,N1(C(Cc2cc(C)ns2)=O)CCCN(C(=O)CCC(CF)CF)C(C)C1 33378,c1(N2CC(C)C(CO)CC2)nccc(=NCCc2cccc(N)c2)[nH]1 33379,N1(C(CN(CCCCCC)C)=O)CC(NC(=O)C=CC(C)(C)C)C2(CCC2)C1 33380,c1(C(=O)N(C2(CCOCC=C)CCC2)C2CC2)nccc(Oc2ccccc2F)n1 33381,c1(C(N2CC(NC(c3c(C)n(C)nc3)=O)C(C)C2)=O)cnc2sccc2c1 33382,C(C(CC(F)(F)F)NC(c1cccc(O)c1Cl)=O)NC(C(CC)N(CC)CC)=O 33383,N1(CCC)C(=O)CCC1C(N1CCCCC1CCNC(c1ncncc1Cl)=O)=O 33384,C#Cc1cc(C(=O)NCC(C)(F)CNC(=O)CC2CCCS2(=O)=O)cc(N)c1 33385,C1(C(N2CCC(C)(NC(c3cc(C)c(C)o3)=O)C2)=O)CCCC2(CCC2)O1 33386,N1(C(c2nc(CC)oc2)=O)CC2CC3CC2C1C3NC(c1ccnn1CCF)=O 33387,C1(CNC(c2cnnn2C2CC2)=O)CN(C(C2C3(CC3)C23CC3)=O)CC12CC2 33388,CC1CC(C(=O)N2CC(O)(C3CCCN3C(=O)C#CC3CCC3)C2)=NO1 33389,CC1CN(C(=O)C(c2ccc(Cl)cc2)O)CC1NC(=O)C(C)C1CCOC1 33390,C1(CNC(CC=CC)=O)C=CCN1C(=O)CCc1ccc(C)s1 33391,c1(C(C(=O)N(CCOCC=C)C)NC(=O)C(C)SC(C)C)ccccc1 33392,c1(CCCCC)ccc(C(=O)NCC(CCOC)NC(=O)C(C)=CC(C)(C)C)o1 33393,C1(NC(c2c(CC)noc2C)=O)CC2CC(NC(=O)C(C3CCOCC3)F)C2C1 33394,Cc1cccc(C(=O)NCC2CC(C(=O)N3CC(CS(C)=O)C3)=NO2)c1C 33395,Cc1ccc(CNC(C2C(O)CCN2C(C2CCC(C)(C)OC2)=O)=O)c(O)n1 33396,N1(C(C(C#N)C2CC2)=O)CCOC2CN(C(c3c(F)cccc3F)=O)CC12 33397,N#CCS(=O)c1ccc(C(=O)NC(C)(CNC(c2cnsn2)=O)C2CCC2)cc1 33398,c1(C(N2C3(CNC(CC4C(C)CCCC4)=O)CC(C2)C3)=O)cc(F)ccc1N 33399,C(=O)(CC(C(F)F)NC(c1coc(SC)c1)=O)N1CC(F)(CC)C1 33400,N1(C(c2cncc(OC)n2)=O)CC(C(=O)NCC(O)C(C)(C)C)CC(C)C1 33401,N1(C(C(C)=C2CC2)=O)CC(N(C(=O)Cc2c[nH]nc2C)C)C(C)(C)C1 33402,N1(C(c2cc(C)[nH]c2C)=O)C2CCC1CN(C(c1cccc(C3CC3)n1)=O)C2 33403,CC1=C(C)CC(C(=O)NCC2COCCN2C(c2csc(C)c2C2CC2)=O)CC1 33404,N1(C(C(C2CCOC2)NC(c2nc(CCC)oc2)=O)=O)CCC12CCCC2 33405,c1(CC)ccc(CCC(=O)N(C(C)CNC(c2coc(Br)n2)=O)C)cc1 33406,c1(COCC)nc(C(=O)N(C(CNC(c2ccc(Cl)o2)=O)C2CC2)C)cs1 33407,c1(CN(CC(C)CS(C)(=O)=O)C)c[nH]c2cccc(Br)c12 33408,Cc1ncnc(C(N2CCC(CO)(NC(=O)C(F)C3CCOC3)CC2)=O)c1C 33409,C(C(O)CC(=O)N(CCC(=O)OC)OC)NC(C(CC)C(C)C)=O 33410,C1(C(=O)NCCn2c(C)cnn2)CCC(C)(C)N(C(=O)COCCCN(C)C)C1 33411,C1(O)(CCNC(C=CC(C)(C)SC)=O)CCN(C(=O)CC2C=CCCC2)C1 33412,c1(C(N2C3C(NC(c4c(Cl)ccc(SC)c4)=O)C(C3)C2)=O)c(N)ccc(F)c1C 33413,C1(C(=O)NCC(C)NC(c2nc(Cl)cs2)=O)CCC2C(C1)C2(F)F 33414,C12(NC(CNC(C)=O)=O)CN(C(C3(Br)CC3)=O)CC1CS(=O)(=O)C2 33415,C1(NC(c2c(OC)noc2C)=O)CC2CC1CN(C(c1ccccn1)=O)C2 33416,C1(NC(CSCCCC)=O)CC2CC(C1)N(C(C1CC(=O)N1)=O)C2 33417,C(=O)(C1=CCOCC1)NC1CCC(N(C(=O)CC2CC=CCC2)C)C1 33418,C1(CN(C(c2cscc2C)=O)CC)CCCN(C(C2CC(N3CCC3)C2)=O)C1 33419,C1(C(=O)NCC2(CNc3ncc(C)cn3)CCCC2)(OCC)CCOCC1 33420,C(=O)(CCCC(C)NC(=O)COC(C)C)NCC(COC)(C)O 33421,Cc1ccc(C=CC(N2CC(NC(c3cc4c(s3)CCC4)=O)C(C)(C)C2)=O)cn1 33422,N1(C(CC(C)OC)=O)CCC2(CC1)CC(NC(c1cc(Cl)c(O)cc1C)=O)C2 33423,Cc1cn2cc(C(=O)NCC3CC(F)(F)CN3C(=O)C(C)N(C)C)cc(F)c2n1 33424,c1(C(=O)NCC(C)NC(c2c(OC)ncc(Br)c2)=O)cnc2ccnn2c1 33425,C(=O)(CC(O)CC(C)(C)C)NCC1C2CN(C(c3nc(OC)nc(O)c3)=O)CC21 33426,C1(CC#C)(C(=O)NC2CC(N(C(=O)CC(C)CN(C)C)C)C2)CCCOC1 33427,C1(CC=C)(NC(C2CC(N(C)C)C2)=O)CN(C(c2cc(C3CC3)on2)=O)C1 33428,C1(CC#C)(C(=O)NC2CC2)CCCC1.C(C(C)O)CC 33429,Cc1cc(C(N2CCCCC2CN(C)C(C23CC(CC(F)F)(C2)C3)=O)=O)ncn1 33430,C1(C(=O)NC(CNC(c2cccc(SCC)c2)=O)CO)NC(=O)OC1(C)C 33431,CCC(C)C(C(=O)NC(CCO)CC(C)C)NC(=O)Cc1c(C)cnn1C 33432,N1(C(C(CC)NC(N)=O)=O)CCN(C(=O)CC2(C#N)CC2)C(C2CCCCC2)C1 33433,C(N=c1cc(NCC(CC)(CC)CC)nc(C(C)C)[nH]1)C1CCN(C(=O)OC)C1 33434,c1(C(C)C)ncc(C(c2nnnn2CC(F)F)NCC2CCCCC2)[nH]1 33435,N1(C(C(OC)OC)=O)CCCC(O)(CCNC(C23CC2COC3(C)C)=O)C1 33436,c1(C(N(C(C)CNC(=O)CCCC2CC2)CC)=O)cc(Br)c(OC)s1 33437,N1(C(CC(C)F)=O)CCC(NC(=O)COc2cccc(F)n2)C(CO)C1 33438,c1(C(N2CC(Cn3cc(C(C)O)nn3)OCC2)=O)nccc2cc(Br)ccc12 33439,CC1=C(C(=O)NC(C)CC2CCN(C(C3(C)CCCO3)=O)CC2)C(C)(C)CCC1 33440,c1(CC(c2ccccn2)NC(C(NS(N)(=O)=O)C2CC2)=O)ccc(Cl)cc1 33441,C(=O)(CC(C)C(F)F)NCCC(C)NC(c1cccc(CCN(C)C)c1)=O 33442,Cc1ccc2c(C(=O)NCCCNC(=O)C(C(C)C)c3cnn(C)c3)n[nH]c2c1 33443,c1(CN2CCC(NC(Cc3cc(C)no3)C(=O)OC(C)C)C2)ccc(I)c(O)c1 33444,CN1CCN(C(c2cc(Cl)cc(Cl)n2)=O)CC1CNC(=O)C(F)n1cccn1 33445,C(C1CCCc2cccnc21)c1n(-c2c(OC)cccc2)nc(-c2cc[nH]n2)n1 33446,c1(OCCC(=O)N(CCn2c(C)ncc2)C(C)C)cc(F)ccc1F 33447,c1(NC(C(n2c(C)nnn2)Cc2ccccc2)=O)cc(F)cc(Cl)c1 33448,N1(C(C(C)(N(C(C(N2CCOCC2)C)=O)C)C2CC2)=O)CCn2ccnc2C1 33449,c1(CNC(C2(NCCC)CCC2)=O)ncoc1CNC(=O)CC1C(OC)CC1 33450,n1(CC(=O)NCC2COCC2NC(=O)C(O)CC(F)F)cc([N+](=O)[O-])ccc1=O 33451,C1(C(=O)NC(C)CC(C)NC(c2sccc2F)=O)(Cc2cnn[nH]2)CCOCC1 33452,C12(C(=O)Nc3c(CCC)cccc3)CC(CO)(CN1C(=O)CSc1nc[nH]n1)C2 33453,c1(C(N2C3CN(C(C=C(C)C4CC4)=O)C(C3)C2)=O)cc2scc(C)c2[nH]1 33454,C1(COC)(NC(=O)C(C2CC2)SC)CCCN(C(C2(O)COC2)=O)C1 33455,CC(C)C#CC(=O)NC12CC1CN(C(c1ncn(C(C)(C)C)n1)=O)C2 33456,c1(C(=O)NC(C)CN(C(=O)Cn2cnnn2)C)ccccc1-c1ncc[nH]1 33457,N1(C(COCCC)=O)CC(C(=O)NCC(C)(C)C(=O)OC)C(F)C1 33458,N#Cc1cnc(NC(C2(F)CCN(Cc3cc(Cl)c(Cl)cc3O)CC2)=O)c(Br)c1 33459,C#CCCCC(C)C(=O)NC1CCCCN(C(c2ccc3nccn3c2)=O)C1 33460,C1(C(N(C2CCC(CNC(C=CC=CCC)=O)CC2)C)=O)CCOCC1(C)C 33461,CCC(CN(C(=O)C(C)OCOC)C)NC(=O)C=CC(=O)OC(C)(C)C 33462,c1(C(=O)OCC)cc(COC(C23CCC(C(F)F)(CC2)CC3)=O)ccc1[N+](=O)[O-] 33463,c1(CN(C(=O)CCC2(NC(c3cc(Cl)no3)=O)CCCC2)C)cccnc1 33464,c1(C(=O)NCC(CC)NC(=O)C(C)OCCC(C)C)ccnn1CCOC 33465,c1(CNC(=O)Cc2cnc[nH]2)cc(F)c(CO)c(F)c1.C12COCCN1C2=O 33466,N1(C(c2cccn(C)c2=O)=O)CC2CN(C(c3cnns3)=O)CC(F)(F)C2C1 33467,CC1CCCCN1CC(=O)N(C(=O)COc1ccc(C(N)=O)cc1)C1CC1 33468,c1(C(=O)NC2C(CC)COC2)ccnc(CNC(=O)Cn2cnc(C(N)=O)n2)c1 33469,c1(CC)nn(C)c(C(=O)N(C)CC2CCCCN2C(c2cnn(CC)c2)=O)c1Cl 33470,c1(OC)cc(Cl)c(Cl)cc1C(=O)NCCC(C)NC(C1C=CCC1)=O 33471,C1(NC(COC(CC)(C)C)=O)CCC2(CC2)N1C(=O)CN(C(=O)COC)C 33472,C1(C)(OC)CCN(C(C2CC(=O)CN2C(=O)CC2(OC)CCC2)=O)CC1 33473,C1(C(N2C(CNC(=O)C#CC(C)C)CC(OC)C2)=O)Cc2ccc(C)cc2S1 33474,c1(C(=O)NCCCC(C)(C)NC(c2c[nH]c(=NC)o2)=O)c[nH]c2c(Cl)cccc12 33475,C=C(Cl)C(C)(C)C(=O)NCC(O)CCNC(=O)CC1(N(C)C)COC1 33476,C1(CNC(CCSCCC)=O)CC2(CO1)CN(C(=O)CCC=C(C)C)C2 33477,c1(CC)c[nH]cc1CNCCN(C)CCN1CCOC1=O 33478,CC1SCCCC1C(=O)NCCN(CCCN(C)C)C(=O)CC1(C)CC1 33479,C(=O)(C(C)(C)NC(C)=O)N1CC(C(C(=O)NCCCN(C)C)OC)C1 33480,CC1=NS(=O)(=O)NC=C1C(=O)N1CC(CCNC(C2CCCC3CCCN23)=O)C1 33481,c1(C(=O)NCC2CCCC(CNC(=O)CCc3cnco3)C2)cc([N+](=O)[O-])c[nH]1 33482,C12(C(=O)NCC(CCNC(C=C(CCC)CCC)=O)O)CC1CCC2(F)F 33483,Nc1nc(C(=O)NC2CC(NC(C3(CF)CC3(F)F)=O)C2)cnc1Br 33484,C1(NC(c2cc(F)c(F)c(F)c2)=O)CC1C1CCCN(C(c2coc(Br)n2)=O)C1 33485,C1(NC(=O)CCc2cc(F)ccc2Br)CN(C(C2(F)CC2)=O)CC(F)(F)C1 33486,N1(C(C(C(C)C)n2cnnc2)=O)CCN(C(=O)C(N)=O)CC(O)C1 33487,CC1CN(C(=O)CCc2cn[nH]c2)CCC1NC(=O)CCc1cnn(C)c1 33488,c1(CC(N2CC(CC(=O)Nc3cc(Cl)ncc3Cl)C2)=O)ccc2c(c1)CCO2 33489,c1(C(N2CC(N(C)C(c3cc(F)cnc3O)=O)C(F)C2)=O)c(F)ccc(F)c1Cl 33490,c1(C(N(C(C)CCNC(=O)C=CC2C(C)C2(Cl)Cl)C)=O)n[nH]c2c1CCCC2 33491,c1(CC)nnc(C)cc1C(=O)NCC1CN(C(c2cnc3n2CCC3)=O)CCO1 33492,C(=O)(C1COc2ccc(Cl)cc21)NC1C(NC(c2c(CC)occ2)=O)CCC1 33493,N1(C(C2CCC(CNC(C3CC4CCC4C3)=O)CC2)=O)CCC(O)C(F)C1 33494,C1(C(=O)NCCC2CCCN2C)(NC(C(C=C)O)=O)CCCCC1 33495,N1(C(c2c(OC)cccc2F)=O)CCc2ccccc2C(NC(=O)C(C)(F)F)C1 33496,c1(C(=O)NCC(C)N(C)C(C2(CS(C)(=O)=O)COC2)=O)cnc(O)n1C 33497,C(=O)(C1c2c[nH]nc2CN1C(C1CCOC1(C)C)=O)NCc1c(C)cc(C)nc1 33498,C1(CC(=O)N(CCCNC(c2c(C)cncc2)=O)C)CC2CCC1CC2 33499,c1(N(C)Cc2c(C)ccc(Cl)c2)nc2c(c(=NCCC3CC3)[nH]1)SCC2 33500,CCC(C)CCCCC(=O)NC1CCCC12CCN(C(c1nnccc1C)=O)C2 33501,N1(C(Cc2ccn(C)n2)=O)CCCC(C)(C)C1CNC(=O)Cc1ccsn1 33502,CC(C)(C)CCC(=O)NC(Cc1cc[nH]n1)C(=O)NC1CCC2(CCC2)C1 33503,c1(NC(c2cnc(OCC)c(-c3ccsc3C#N)c2)=O)c(Cl)cccc1[N+](=O)[O-] 33504,Cn1ccnc1C(=O)NC1(C2CCCN2C(=O)CCSCc2nccn2C)CC1 33505,C1(CNC(CCc2ncc(C)[nH]2)=O)CC(NC(c2sc(C)cc2Cl)=O)C1(C)C 33506,n1(C(C(=O)OC)C)cc(CCCCC(=O)N(C)CC2CCC2)nn1 33507,C1(C(=O)NCC(CNC(c2cn(C(C)C)nn2)=O)C)CCCC(=O)O1 33508,C1(NC(C(C(C)C)SCC)=O)CC2(CCN(C(C3CCCN3N=O)=O)C2)C1 33509,Cc1nc(C(N2CCC(NC(C3CCC(=O)N(C4CC4)C3)=O)C2)=O)c(C)n1C 33510,C1(NC(C(C(C)NC(CC2(OC)CCC2)=O)C)=O)C2CCCC1COC2 33511,C(=O)(C(O)CCS(C)=O)N(CCC)CCNC(c1sccc1OC)=O 33512,C1(CC)C(NC(=O)C(c2cn(C)nc2C)C)CCN1C(=O)C=CC1CCC1 33513,Cc1nn(CC(=O)NC2CC2NC(C2(C)CC(C)(C)C2)=O)c(C)c1Cl 33514,c1(C(=O)NC2(CNC(CP(C)(C)=O)=O)CC2)cc2cc(Cl)cnc2[nH]1 33515,c1(CC(=O)NCC(C)(O)CNC(=O)CCc2cnc[nH]2)c(F)cccc1F 33516,C1(C(N2CC3C(NC(C4CC5COCC5C4)=O)(C3)C2)=O)CC2(C1)CC(F)(F)C2 33517,c1(CC)ccc(C=CC(=O)NCC2CCCN(C(C3CC3C(=O)OC)=O)C2)cc1 33518,C12(CCCCCCC1)C(=O)N2.c1(CC)cc(C(F)(F)F)cnc1C 33519,N1(Cc2cn(CC(C)C)nn2)CC(=O)N(Cc2ncnn2C)C1=O 33520,C(=O)(CCCC(=O)NCCC1(NC(=O)C(C)NC(C)=O)CCCC1)OCC 33521,C1(NC(CCSCC)=O)CC(NC(c2ccc(OC)cc2C(F)F)=O)C12CCC2 33522,c1(-c2ccn(CC)n2)nc(C(=O)NC(CO)C(=O)OCC)ccc1F 33523,c1(C(=O)NCCCN(C(=O)Cc2nc[nH]n2)CC)cc2ncccc2s1 33524,c1(OC)cccc(OC)c1C(N1CCC(C(=O)Nc2ccc(C)cc2Br)C1)=O 33525,C1(C(N(C2CC(C#N)C2)CC(=O)NCC(C#C)OC)=O)CCOC1(C)C 33526,c1(C(C)CNCc2cc(CO)no2)ccc(C(F)F)cc1 33527,C1(C(C)C)C(C(=O)NCCN2CCNC(=O)C2)CCN1C(=O)CC1CCSC1 33528,C(=O)(CCCN=[N+]=[N-])N1C2(C(=O)NC3CN(CCC)C3)CC2CC1 33529,C1(C(N2CC3(CCN(C(c4ccc([N+](=O)[O-])o4)=O)C3)C2)=O)CC2CC(O)C(C1)C2 33530,C(CCCCCN(C)C(C1CCC(CO)CC1)=O)NC(CCNC(=O)NC)=O 33531,CCCCC(CC)C(=O)N1CCC(=CCNC(C2CC3CC3C2)=O)CC1 33532,N1(C(CC(CC#C)NC(=O)CC2CCCCC2O)=O)CC(=O)NC2(CC2)C1 33533,N1(C(c2cccc(C)c2)=O)CCN(C(c2ccn(CCO)c2C)=O)C2CCC12 33534,c1(C(N(C2CN(C(C(CO)NC(C(C)C)=O)=O)C2)C)=O)ccc2c(c1)CCN2C 33535,C1(O)(CC(=O)NCC2(C)CCCC2)CCN(Cc2ccc(F)c(C(F)F)c2)CC1 33536,C(=O)(CC(C)(C(F)F)N(C)C)NC(CN(C(c1ccc(C)cn1)=O)C)C 33537,Cc1cc(CC(N2CCCC2CNC(c2ccn(C)n2)=O)=O)ccc1Cl 33538,C1(C(=O)NCCC2CCN(C(CCC=CCC=C)=O)C2)CS(=O)(=O)CCO1 33539,c1(CC)cc(C)c(C(=O)NC2COC(C3CCNCC3)C2)o1 33540,CC1(NC(=O)C(c2cccs2)=O)CCN(C(c2ccc(OCC3CC3)cc2)=O)C1 33541,c1(SC(C(=O)NC(CNC(c2cc(CCC)on2)=O)C)C)ccc(F)cc1 33542,C1(C(=O)NC2CN(C(C3CC(CF)C3)=O)CC2C(F)(F)F)SC2C=CC1CC2 33543,C(=O)(CC(C)(C(F)F)N(C)C)NC1C(O)CCN(C(CC=CC=C)=O)C1 33544,N1(C(CCC=CC)=O)CCCC1(C)CCC(N1C2COCC1C2)=O 33545,N1(C2CCN(C(C3CC34CCOC4)C(=O)NCCC)CC2)CCN(CC)CC1=O 33546,C12(CNC(Cc3cccc(C)c3)=O)CCCN(C(=O)CC3(C#N)CCC3)CC1C2 33547,C1(CC#C)CN(C(=O)COC2CN(C(=O)CN(C)C(C)C)C2)CCO1 33548,c1(COCCOC)noc(-c2cnn(-c3cnccn3)n2)n1 33549,C(C(CC(F)(F)F)NC(=O)C1=NOC(C)C1)NC(C(NOC)=O)=O 33550,c1(CNC(c2nc(CC)oc2C)=O)ccc2c(c1)CN(C(=O)C(=O)N1CCCC1)C2 33551,N1(C(C(C)OC)=O)CCC(N(CC(C)C)C(=O)C=CC2CCCCC2)CC1 33552,c1(CC)cccc(CC(=O)N(CC(CC)NC(=O)CCn2ccccc2=O)C)c1 33553,N1(C(C2N(CCC)CCOC2)=O)CCCCC(NC(c2cccc(N)c2)=O)C1 33554,C(=O)(CCC(C)(C)NC(N1CC=CC1)=O)N(CC=C)CC=C.C(C)C 33555,c1(OC)cncc(C(=O)N(CCCCCNC(C2CN(C)CCO2)=O)C(C)C)n1 33556,C1(NC(=O)Cc2ccon2)(CF)CCN(C(C2CCCCC2O)=O)C1 33557,C(=O)(C#CC1CCCO1)NC(CNC(c1c(SC(C)C)cccc1)=O)(C)CO 33558,N1(C(=O)NC2C(C(N)=O)CCCC2)CCOC2(CCS(=O)(=O)C2)C1 33559,Cc1cc(O)nnc1C(=O)NCC1(C)CCN(C(=O)CC2CCC(C)C2)CC1 33560,C=CC(C)(C)CC(=O)N1CCCC1CC(N1CCCC(F)(F)C1)=O 33561,C1(NC(c2[nH]c(=NC)sc2)=O)CN(C(c2ccnnc2S)=O)C2(CCCCC2)C1 33562,C1(CNC(=O)C(c2ccc(Br)cc2)F)CC1C1CCOCC1 33563,CCCCS(=O)(=O)CC(=O)NC(C)CN(C(C1CCCN1C1CC1)=O)CC 33564,N1(C(CCCCN(C)C)=O)CCC2(CCCN2C(=O)Cc2cccs2)CC1 33565,N1(c2nc(C)c(Br)cn2)CC(NC(c2ncc(Cl)s2)=O)CC(C)(C)C1 33566,N1(C(c2c(OC)oc(C)n2)=O)CCC12CN(C(C1CC3CCC1O3)=O)C2 33567,Cc1cc(C(C(=O)NC2CC(F)(F)C2)N(CC(=O)N(C)C)C)cc(C)c1Cl 33568,Cc1ccc(C)c(OCC(N2CC(O)(CNC(c3csc([N+](=O)[O-])c3)=O)C2)=O)c1 33569,C1(n2cc(C(CSCC)C)nn2)CN(C(=O)Cn2cccn2)CC1C 33570,Cc1ncc(C(F)(F)F)cc1C(=O)NC1CCCCN(C(C2(C(F)F)CC2)=O)C1 33571,c1(CNC(C2(NC(c3c(CC)ocn3)=O)CCC2)=O)oc(C)nc1C 33572,c1(C(=O)NCC2(NC(c3c(C(C)C)nns3)=O)CC2)cc(C2CCC2)nn1C 33573,c1(C(=O)NC2CCC(NC(c3cn(CC(N)=O)nn3)=O)CC2)ccc(O)nc1Cl 33574,CCC(C(=O)NCCC(O)CN(C(=O)CC1(C#N)CCCCC1)C1CC1)C(F)(F)F 33575,N1(C(C(=O)N(C)C)=O)CCN(C2CCN(C(=O)C=CC3CCOC3)CC2)CC1 33576,Cc1nc(C(=O)NC2CC(CCC(=O)NC3(CN(C)C)CC3)C2)c(C)o1 33577,C1(CNC(=O)C=CCn2cncn2)CCC(CNC(=O)Cn2cnnc2)CC1 33578,Cc1nn(C2CCOCC2)cc1C(=O)NCC1(NC(=O)C=CS(C)=O)CCCC1 33579,c1(C(N2CC(O)(CNC(=O)C3CC3)C2)=O)ccc(-n2cccc2)cc1Cl 33580,CCCCCC(C)CC(=O)NC1CCCCC1NC(=O)CN1CCNC1=O 33581,N1(C(C2(C)CCN(C)C2)=O)CCN(C(c2cc(Cl)c(Cl)s2)=O)CC(CO)C1 33582,C(=O)(C#CC1CCCO1)N1CCCC(CN(C(=O)CCOC2CCCC2)C)C1 33583,c1(C(C)(F)F)cc(S(=O)(=O)Oc2cccc(C(C)(C)C)c2)c(C(C)(C)C)s1 33584,C(=O)(C(C)C(F)(F)F)NCCC1N(C(CCOc2cccc(C)c2)=O)CCSC1 33585,C1(NC(C=CC=CC)=O)CCCC12CN(C(c1cccc(C(F)(F)F)n1)=O)C2 33586,c1(C(=O)NC2(C)CCCN(C(c3cc(C)on3)=O)C2)cc2cnccc2o1 33587,c1(C(N2CCC(c3ncc(C(=O)O)s3)C2)C)cccnc1 33588,C(CCCOC)(C(=O)N1CC(F)(F)C1)NC(c1nn(CC)nc1C)=O 33589,c1(C(N(C)CC2CCN(C(c3cn(CCO)nn3)=O)C2)=O)cc2cnccc2o1 33590,N(C(=NCCCCc1ccc(Cl)s1)NCc1ccccc1Cl)CC1CC(=O)NC1 33591,C1(N(CC(=O)N(CC(C)C)CC)C)CCOC1 33592,N1(C(C(N2CCC(C)C2)=O)=O)CCC(O)(C(=O)N(c2ccccc2)C)CC1 33593,C1(C(=O)NCCCCCO)(CC)CCCN(C(=O)COCC(F)F)C1 33594,c1(C(=O)OCC)nc(=NC2CC(F)(CNC(=O)C(C)COC)C2)cc[nH]1 33595,Cc1c(Cl)cc(C(=O)NCCCC(=O)N(CCCN)C)cc1Br 33596,CCC(C(=O)N1CC(N(C)C(c2csc(C)c2OC)=O)C1)C(C)C 33597,C1(CC)CN(C(=O)CCCC(N)=O)CCN1C(=O)C(CC)SC 33598,C1(C(=O)NCC2CCC(NC(=O)CCCC3OCCO3)C2)C2CCC1CC2 33599,CCC(C(=O)N1CC(CN(C)C(c2cccc(NC(=O)C3CC3)c2)=O)C1)C(C)O 33600,C#CC1(NC(=O)CCCC(C)NC(c2coc(C(N)=O)c2)=O)CCCCC1 33601,C1(NC(c2ccccc2-c2nc[nH]n2)=O)CN(C(C2CC2(F)F)=O)CC1C(F)F 33602,C(=O)(C1=C(Cl)CCCC1)N1C(CNC(C2(COC)CCCO2)=O)CC(F)C1 33603,C1(NC(c2nc(C(C)NC(CC(C)C)=O)oc2)=O)CCN2CCC1C2 33604,C(CC(O)CCC(C)(C)C)NCCc1cn(CCOC)nn1 33605,CCC(C)C(C(=O)NC1COCCN1C)N(C(=O)CCCNC(C)=O)C 33606,N1(C(=O)CCc2cccnc2)CC2CC(NC(=O)C(F)(F)CC3CC3)C1C2 33607,C1(CNC(C(CCOC)C)=O)CCC2(CN(C(C3CCOC(C)C3)=O)C2)O1 33608,C(=O)(CCc1ccc[nH]1)N(C(C)C(=O)NC(C)C(=O)NC)CC 33609,c1(CC)ccc(C(=O)NCC2(NC(=O)Cn3ncnn3)CC2)c(O)c1 33610,c1(OC)ccc(C(F)(F)C(=O)NC2CN(C(=O)C(O)CC3CC3)CC2F)cc1 33611,N1(C2CCN(C(c3cnc(C)n3C)=O)CC2)CCN(C(C2C=CCC2)=O)CC1=O 33612,C#Cc1ccc(CCC(=O)NC2CCC2CNC(=O)CCC2(C)CC2)cc1 33613,Cc1cc(Nc2ccc(NC(C3CCC(=O)C3)=O)c(C)c2)cc(=O)o1 33614,CC(C)(CS(N)(=O)=O)C(=O)N1CCN(C(c2ccn(C3CC3)n2)=O)CC2(CC2)C1 33615,C(C(CC(C)C)C(=O)NC(C)(C(=O)NCc1csnn1)C1CCC1)OC 33616,C=CC(C(=O)N(C1CCN(C(c2cnccn2)=O)C1)CC)NC(=O)OC(C)(C)C 33617,C(N=c1nnc(C)c(C)[nH]1)C1CCN(C(c2ccc(C)c(F)c2)=O)CC1C 33618,N1(CC(=O)NCC(CC(C)C)NC(C2CCC23CCC3)=O)CCc2sccc2C1 33619,N1(C(c2cc(C(C)=O)sc2)=O)CCN(C(=O)C(F)(F)C2CCCC2)CC1C1CC1 33620,c1(N(CCOC)C)nc(=NCCc2nc3ccc(F)cc3[nH]2)[nH]c2cc[nH]c12 33621,c1(CC)cnccc1C(=O)NCC(C)NC(=O)C(C)C(C)C 33622,C(CC(C)C=O)=CC.C1(OCCCC)CCN(C(C2(n3cc(Cl)cn3)CC2)=O)C1 33623,C1(C(=O)NCC(C)NC(c2cc(Cl)ncc2N)=O)CCc2cc(F)ccc2O1 33624,CC1CC(NC(=O)Cc2ccc(F)cc2)CN1C(=O)CC1CCS(=O)(=O)C1 33625,CCCC(CCCNC(=O)CSc1ccccn1)Nc1ncncc1I 33626,Cc1cccc(C)c1NC(=O)C(c1cc(Br)ncc1F)N1CCC(C(F)F)CC1 33627,C(=O)(CC(CC)CCC)N1C(C(C)NC(C(C#C)(C)C)=O)CCC1 33628,CC(C)CCC(F)C(=O)NC1CC1CNC(c1cc(C(N)=O)n(C)n1)=O 33629,c1(CNCCC(=O)N(C2CCCN(C(CSC)=O)C2)C)nc2ccccc2s1 33630,Nc1nc(C(N2CC(NC(c3cnns3)=O)CC(O)C2)=O)cnc1Br 33631,C(=O)(C(C)(F)CCCC)NC(CC(=O)NCCCC(C=C)(C)C)CC 33632,c1(CN(CC(C)C)N(C)CC2CCCO2)nnc2n1CCOCC2 33633,c1(C(N2CC3(CC3C(N3CCC(c4cn[nH]c4)CC3)=O)C2)=O)cccc(Cl)c1Cl 33634,c1(C(=O)NC(CC)CN(C)C(C2(CF)CCC2)=O)c(C)nc2sccn12 33635,C1(CNC(C2CCCN(C(N(C)C)=O)C2)=O)CCCCN(C(c2cncs2)=O)C1 33636,CCCC(CC)C(=O)N1CC2C(CC(=O)NC3CCN(C(C)=O)CC3)C2C1 33637,N1(C(c2nc(CCC)sc2)=O)CC(CNC(=O)C=CC2CC2)C2CC12 33638,Cc1cccc(-c2cccnc2C(N2CCN(CCO)CC2)=O)c1C 33639,N1(C(c2nccc(CC)c2)=O)CCN(C(c2cncc(C)n2)=O)C2CCCCC12 33640,CC1(C)CC(C(N2CCC2C2CCCC2)=O)CCN1C(=O)Cc1cn[nH]c1 33641,C1(NC(C(C)CC(F)(F)F)=O)C2CC3CN(C(=O)C4=COCCO4)C1C3C2 33642,CC1CCN(C(=O)C(=O)N(c2cnn(C)c2)CC(C)C)CCS1 33643,c1(NC(C2C(C)CCCC2)=O)cnc2ccc(F)cc2c1 33644,CC1CCN(C(c2cc(O)nn2C)=O)C1CNC(c1ccc(C2(C)CC2)cc1)=O 33645,c1(C(C)(CO)NC(C2CCN(C)C2)=O)cccc(CNC(=O)NC(C)(C)C)c1 33646,c1(NCCC2(COC)CC2)ncnc(N(C(CO)CC(C)C)C)c1C 33647,C1(CNC(C(CCCOC)C)=O)CC2COCC2N1C(C1CCOC1C)=O 33648,c1(C(N(CC)CC2CCCN(C(=O)CC(C)(C)OC)C2)=O)cnc(C)c(N)c1 33649,Cc1cnc(C(N2CCC(CO)(NC(=O)OC(C)(C)C)C2)=O)cc1C 33650,C1(C(=O)NC2COCCN(C(CN3CCC(C)(C)C3)=O)C2)CCCC2(CCC2)O1 33651,Cc1cc(F)cc(C)c1C(N1CC(NC(c2[nH]cnc2C#N)=O)C1)=O 33652,c1(CNC2C(OC)CS(=O)(=O)C2)nc2ccc(Br)nc2[nH]1 33653,N1(C(c2nc(CC)oc2C)=O)CC(NC(c2cnc(C)c(C)c2)=O)CC12CCC2 33654,Cc1cc(CNC(=O)C(C2CCC2)NC(=O)Cc2ccccn2)on1 33655,c1(CN(c2cc(OC)ncn2)c2ccccc2)n[nH]c2c1CCCC2 33656,C1(C(=O)NCC23C(CN(C(c4c(N)non4)=O)C2)C3)COc2ccccc2O1 33657,C#Cc1ccc(C(=O)NC2(COC)CCN(C(=O)C(C(C)C)NS(C)(=O)=O)C2)nc1 33658,C=CCCCC(=O)NCC(CC=C)NC(=O)C(=C1CCCCC1)F 33659,c1(C(N2CCC(C)(NC(=O)Cc3cccc(O)c3)C2)=O)oc2ccccc2c1Cl 33660,N1(C(c2nc(CC)oc2C)=O)CCC2CN(C(c3cn(C)nc3OC)=O)CC12 33661,C=C(C)CCC(=O)N(CC(C)(C)NC(=O)CC(C)CN(C)C)C 33662,C(=O)(C(C(C)O)NC(=O)Cc1cn[nH]c1)NCC1(C(C)C)CCCC1 33663,C1(NS(=O)(=O)CCOC2CCOC2)CCCC12CCCO2 33664,C(=O)(C1=CCCCO1)N1CCN(C2CCCN(C(CSC)=O)C2)CC1 33665,c1(C(=O)NC2C(C)N(C(=O)Cn3ncnn3)CC2)cc2c([nH]1)CCOC2 33666,CC(C)(CCC(=O)N(C1CCC1)C1CC1)NC(=O)CC1CC=CC1 33667,CCCCC(N)C(=O)NCc1ccc(F)nc1F 33668,Cc1nncc(C(N2CC=C(CNC(C3CCO3)=O)CC2)=O)c1C 33669,C(C)(CNC(C1CCNC1=O)=O)(CO)NC(C(C)=CC1CC1)=O 33670,C1(OC)CCCCCC1Nc1ccc(-c2ccc(C)nc2O)cn1 33671,c1(C(N2CCC(NC(C3N(CC)CCC3)=O)C2)=O)nc2ccc(C)cn2c1N 33672,C(CC(C(C)(C)C)NC(=O)CN1CCNC1=O)N(C(C1(OC)CC1)=O)C 33673,c1(-c2cc(C(=O)NC(c3c(OC)cccc3)CO)[nH]n2)ccc(C)c(C)c1 33674,C=CC(CC)CC(=O)N(C1CCCN(C(=O)C(O)C2CC2)C1)CC 33675,c1(C2(NC(CCc3nnc(C)o3)=O)CCCC2)ccc(OCc2cccs2)cc1 33676,CC1(C(=O)NCC2CC(NC(=O)CCc3cnoc3)C2)CC(C#N)C1 33677,c1(OC)ccc(N(C)Cc2cc(C)c(-c3cc(C(F)F)ccc3F)cn2)cc1C 33678,C1(N(C)C)(C(=O)NCC(O)CCNC(=O)CCC2CCC2)CCOCC1 33679,C12(NC(C3CC3(F)F)=O)CCC(C1)N(C(c1cc(Cl)ccc1-n1cccc1)=O)C2 33680,c1(NS(C)(=O)=O)cc(C(=O)Nc2cn(CC3(C4CCOCC4)CC3)nn2)ccn1 33681,C1(OCC)CCC1C(=O)N(C1(C(=O)N(CCCO)C2CCC2)CC1)C 33682,C(C(=O)NCc1cccs1)(C(C(C)C)OC)N1CCCC(C(=O)OC)C1 33683,C(=O)(C1=NOC2(C1)CN(C(=O)OC(C)(C)C)C2)N(CCO)CC=C(C)C1CC1 33684,c1(N(C)Cc2ccoc2)ccc(S(=O)(=O)NC2CC3CCC(C2)S3)cc1F 33685,c1(C(=O)NCCCN(C(C(CSC)O)=O)C)ccc2c(c1)CC(=O)NC2 33686,CN1CCN(c2nnco2)CC1CNC(c1cc(O)nn1C)=O 33687,C1(NC(C(C(=C)Cl)(C)C)=O)CN(C(=O)C(C)CC(=C)C)C2(CCC2)C1 33688,C1(C(N(CCNC(CSC)=O)CC2CC2)=O)CCCC2CCCN12 33689,N1(CC)CC(C(N2CC3CC2C3NC(=O)CSc2n[nH]c(C)n2)=O)CCC1=O 33690,N1(CC)CCCCC1C(=O)N(C1CCN(C(=O)CCSc2ccccc2C)C1)C 33691,c1(C(=O)NCCC23C(CN(C(CCOCC)=O)C2)CC3)sc2ccccc2c1C 33692,c1(C(=O)NCC(C)CNC(=O)CCn2cc(Cl)cn2)ccc([N+](=O)[O-])c(O)c1 33693,c1(NC2CN(C(c3c(OC)cc(I)cc3)=O)CC2C)nc(C)c(C#N)cc1Cl 33694,c1(C2(COc3cncc(C(=O)OCC)c3)CC2)ccc2c(c1)OCCCO2 33695,N1(CC)CC(C(=O)NC(C)CC2CN(C(C3CCCN3CC)=O)C2)CC1=O 33696,c1(CC(N2C(C)CC(CNC(=O)Cc3cnc[nH]3)CC2)=O)c[nH]c2cccnc12 33697,N1(C(c2nc(C)n(C)c2)=O)CCCC(NC(c2[nH]ncc2C#N)=O)CC1 33698,CCCC(CC)C(=O)NCc1cccc(C(=O)NCC2CCN(CCC)C2)n1 33699,N1(C(c2nc(CCC)oc2)=O)CCCC2(CCCN2C(c2cc[n+]([O-])cc2)=O)C1 33700,N1(C(C(c2ccc(OC)cc2)C)=O)CC(C2CCN(C(=O)C(O)C3CC3)CC2)C1 33701,c1(CCC)cc(C)ccc1N(C(=O)CCCn1ccnc1-c1ccc(C)nc1)C 33702,CC(C)(C)C(C(=O)NC12CC(NC(c3csc(=N)[nH]3)=O)(C1)C2)N1CCCC1=O 33703,CC1CN(C(C2CCCN2C)=O)CC(C)CN1C(=O)CCc1ccco1 33704,CN=c1ccc(C(=O)N(CCC(C)NC(C2CC2C(F)F)=O)C)c[nH]1 33705,c1(NC(C)=O)ccnc(C(N2CC(CO)(NC(C3CCC4CC34)=O)C2)=O)c1 33706,C1(CCC(=O)NCCC(C)N(C(C(C)=C(CC)C)=O)C)CCC(=O)NC1 33707,C1(C(=O)NCC2(COC)CN(C(C(C=C)C)=O)C2)CCC2(CCC2)C1 33708,C(=O)(C(O)CC(C)(C)C)N1CCC(N(C)C(c2cc(-n3cnnc3)ccn2)=O)C1 33709,N1(C(C2(CNC(c3cc(C)sn3)=O)CCC2)=O)CC(C)(C)OC(C)(C)C1 33710,Cc1cnc2c(C(=O)NCC(CO)NC(C3CC34CCCCC4)=O)cnn2c1 33711,CS(=O)C=CC(=O)NCC1C2CN(C(C3CC(O)(c4cccnc4)C3)=O)CC12 33712,c1(C(N2C(C3CCN(C(C=C(COC)C)=O)C3)CCC2)=O)ccc(N)cc1C 33713,CC1Cc2cccc(C(=O)N(C(CNC(c3ncc[nH]c3=O)=O)C3CC3)C)c2O1 33714,c1(-c2n(Cc3ccc(OC)cc3)nc(-c3ccc(Cl)s3)n2)cncc2nc[nH]c12 33715,c1(C(=O)NCCSCC(=O)O)ccc(-n2cc(-c3cncc(CO)c3)nn2)cc1 33716,c1(CNC(N(C(C(=O)OCC)C)C)=O)ncncc1C 33717,C1(C(=O)NCC2CCCC2C(C)C)(NC(COCCC)=O)CC(F)(F)C1 33718,S(=O)(=O)(c1ccc(-c2cc(Cl)c(Cl)c(Cl)c2)cc1Cl)NCc1ccc(OC)nc1 33719,C(c1cccc(F)c1Cl)=CC(=O)NCCCCCNC(Cc1cn(C)nn1)=O 33720,c1(C(=O)NC(c2ccnn2C)C(=O)NC(CCOC)COC)cc(C)ccc1C 33721,c1(C(N2CC3(C(NC(CCCOCCOC)=O)CC3)C2)=O)cnc2c[nH]nc2c1 33722,C1(O)(C(C)NC(=O)CC(C)c2ccco2)CCN(C(=O)CCn2ccnn2)C1 33723,CCCC(CCCNC(=O)CC1COCC1(C)C)NC(c1cnc[nH]1)=O 33724,C1(NC(C(CC)CC)=O)CCC(C)N(C(=O)C(c2cccc(Br)c2)C)C1 33725,c1(C(=O)NCc2ccc(Br)cc2F)cc(Br)cc([N+](=O)[O-])c1 33726,Cc1cccc(Br)c1C(C(=O)N(CC(C)(F)F)C)NC(c1nn(C)cc1C)=O 33727,c1(N2CCN(C(C34CNCC3(F)CCOC4)=O)CC2)ccc2c(c1)C1(CC1)C(=O)N2 33728,Cc1cccc2c1OCCN(C(=O)C(C)(N)CC(C)C)C2 33729,CCCS(=O)(=O)C(C)C(=O)NCC1CC2(C1)CN(C(C1CC1(C)C)=O)C2 33730,C1(CNC(C2(CC)CCCC2)=O)CC2(C1)CN(C(=O)Cc1cc(C)on1)C2 33731,c1(C(=O)NCC(CNC(c2ccc(CCCCC)o2)=O)C)cc(CC)ccc1N 33732,c1(C(N2CCC(C(O)C(F)F)C2)C(=O)NCCCC2CC2)ncc(Cl)s1 33733,N1(C(C2C(CC)OCC2)=O)CCC(F)(CNC(C23CC2C3)=O)CC1 33734,CC(CC(F)(F)F)C(=O)NCCNC(C1CCCN(C(=O)C#CC2CCC2)C1)=O 33735,C=CC1(C(=O)NCC(C2CC2)N(C)C)CCN(C(C2CC(=C3CC3)C2)=O)C1 33736,C1(NC(CN(CC#C)C(c2ccc(N)c(SC)c2)=O)=O)CCCCCC1CC1CC1 33737,C1(COC)(NC(=O)COC(C)C)CCN(C(=O)COCc2ccncc2)CC1 33738,c1(NC(=O)CCNC(C2CCC2)=O)cnc(C2CC2)o1.C12CC1CNC2=O 33739,Cc1ncc(CC(=O)NCC(C2CC2)NC(=O)C(C)N2CCC2)[nH]1 33740,c1(NC)ccc(C(F)(F)F)cc1C(=O)NC1CN(C(C2COC(=O)N2)=O)C1 33741,C(=O)(N=c1cc2ccccn2[nH]1)C1(C)C=CCN1C(c1cc(Cl)cs1)=O 33742,c1(OC(C)(C)C)ccc(C(=O)NC2CCN(C(c3coc(Br)n3)=O)CC2)cn1 33743,c1(C(N(CC(C)NC(=O)CC#N)C)=O)cnoc1C1CCOCC1 33744,N1(C(CSC(C)(C)C)=O)CCN(C(=O)C(F)C(C)(F)F)CC1c1cn[nH]c1 33745,Cc1cc(C(=O)NCC(C)(CO)NC(=O)C=Cc2nccs2)ccc1Cl 33746,C1(CCNC(=O)CCCN(C)C)(OC)CN(C(=O)CCc2nc(C)no2)C1 33747,O=C1CCc2c(C(=O)Nc3cc(Cl)c(Br)c(Cl)c3)cccc21 33748,c1(C(c2ccco2)=O)nn2c(c1CNCC(O)COc1ccc(Cl)cc1)CCC2 33749,c1(C(N(CC(C)(C)CNC(C2(CF)CCOCC2)=O)C)=O)c(F)cncc1Cl 33750,CN1C(=O)CCC(c2nc(C3(c4ccccc4F)CC3)no2)C1c1cccc(Cl)c1 33751,N1(C(COCC(C)C)=O)CCC(C)(CCNC(C2CC(C)C2)=O)C1 33752,Cc1nn(C)c(C)c1C(N1CC2CC1(CNC(C1CC1c1ccccc1)=O)C2)=O 33753,C1(CCNC(c2cc(C)on2)=O)CCN(C(C2CCCN2C=O)=O)CC1(F)F 33754,C12C(C1(C)C)C(=O)N2.C1(CCNC(C2CC(N(C)C)C2)=O)CC(F)(F)C1 33755,N1(C(c2cc(CC)oc2)=O)CC(C(N2CCCC(COC)C2)=O)C2(CC2)C1 33756,Cc1ccnc(C)c1CNC(=O)C(C1CCCO1)NC(=O)Cn1ncnn1 33757,C1(CC)CN(C(C2(NC(=O)CC(C)CN(C)C)CCOCC2)=O)CC(=O)N1 33758,c1(CSC)cccnc1C(N1CCOC(CNC(C2CCC(=O)N2C)=O)C1)=O 33759,S(=O)(=O)(c1cccnc1N1CCC(NC2CCCOC2C(C)(C)C)CC1)NC 33760,CCCCC(F)C(=O)N(C1CCCN(C(c2c[nH]c(=N)c(C)c2)=O)C1)CC1CC1 33761,CCC(C)(C)C(=O)C(=O)N1CC=C(C(=O)NC(CCO)C2CC2)C1 33762,c1(C(=O)NC2C(CNC(c3c(CC)c[nH]c3)=O)CCCC2)cn(C)c(=O)cn1 33763,c1(C(N(C(CNC(C2CCC(=O)O2)=O)C2CC2)C)=O)cc2ccccn2n1 33764,C1(C)(C(=O)NCC(CCOC)NC(=O)CCCn2cccn2)CC(=O)N(C)C1 33765,c1(CC)cccc(N(C)C(c2cc(CNC(=O)CC3CC=CCC3)no2)=O)c1 33766,C(=O)(C(S(C)(=O)=O)C1CC1)N(C(C)CNC(c1ccc(Cl)o1)=O)CC 33767,C1(OC)CCCC(CNC(=O)CN(CC(C)C)C(=O)Cn2cncn2)C1 33768,C1(C2CCCC2)(C(=O)NC2C3(CCN(C(c4cc(Cl)nnc4O)=O)C3)C2)CCC1 33769,C(=O)(C(O)C(C(C)C)OC)N(C)CC1CCCN(C(c2cc(CC)n(C)n2)=O)C1 33770,CC1COCCCN1C(C1CN(C(C2CCCC2)=O)C(C)(C)C1)=O 33771,Nc1cnc(Cl)c(C(N2CCOCC(NC(c3ccc(F)s3)=O)C2)=O)c1 33772,c1(C(N(C2(COC)CC2)C)=O)cccc(-n2cc(CNC=O)nn2)c1.C(C)(C)(C)S 33773,c1(C(N2CCC(CN(C)C(C3CCCN3C=O)=O)CC2)=O)cc(O)c(O)c(O)c1 33774,Cc1ccc(Br)cc1C(N1CCC(CO)C(C)C1)C(=O)NCCCF 33775,C1(C(C)NC(=O)NC(C#C)C2CCC2)(OC)CCC1 33776,C1(CC(N2CCC(C(=O)NCC3(O)CCCOC3)(CC)C2)=O)CCC(C)(C)CC1 33777,c1(CCC(=O)Nc2cccc(NC3CCCC3)c2)ccc(Cl)c(Cl)c1 33778,N1(C(CCC(=C)C)=O)CCN(C(=O)C(C)CCC)C(c2cn[nH]c2)C1 33779,c1(C(=O)NCC(C)(C)OCC)cnc(CNC(COCCOCC)=O)[nH]1 33780,c1(C(=O)NCC2CN(C(=O)CCc3cncs3)C2)cccc2cncn12 33781,C#Cc1cc(C(=O)NCCNC(C2CC[Si](C)(C)CC2)=O)cc(F)c1 33782,N(C(=NCCOc1ncccc1Cl)NC1CCCC1)C1CCC(C)C1 33783,C1(c2nn(CCC)c(-c3ccc(C)nc3)n2)CCC(F)(F)CC1 33784,c1(C(N(C(C2N(CC)CCC2)=O)C)C)sc(OC)nc1C 33785,c1(Nc2ccc(OC)cc2CC(N)C(=O)O)nc(C)nc2scc(CC(C)C)c12 33786,C1(NC(CSC(C)C)=O)COCCC1NC(c1cccnc1-n1nccn1)=O 33787,c1(CNC(=O)NCC2C(NC(=O)OC(C)(C)C)CC2)ccc(Cl)o1 33788,C=C1CCN(C(c2nscc2C)=O)C(C(=O)NCCC2CC=CCC2)C1 33789,Cc1ccc(C(=O)NCc2cc(NC(=O)OC(C)(C)C)sc2C)c(O)n1 33790,c1(C(=O)NCC2(F)CN(C(COCCCC)=O)C2)cccc(C(=O)N(C)C)c1 33791,c1(C(N(C(CNC(CC=C)=O)C)CC)=O)cnc(Br)c(N)n1 33792,N1(C(C(c2ccccc2)NC(C=CC(C)(C)C)=O)=O)CC2(CNC(=O)C2)C1 33793,c1(CC(=O)N(CCn2cc(CC(O)CO)nn2)CC)cc(Cl)cc2c1OCC2 33794,CC1(C)OCCOC1C(N1CCC2C(NC(=O)CNC(N)=O)CC12)=O 33795,N1(C(c2ccc(C)[nH]2)=O)CCN(C)C(CNC(=O)C(c2cccnc2)O)C1 33796,N1(C(C(C)Sc2nncn2C)=O)CC(NC(=O)CC(C)(C)C)CCC1C 33797,C1(CNC(C(CC)(CC)CO)=O)CN(C(=O)C=C2CCC(C)C2)C2COCC2O1 33798,C1(C)(OC)CCCN(C(=O)C(C)(CNC(c2ncoc2C)=O)CC)C1 33799,CN1CCOCC1CC(=O)NCc1ccc(CN(C)C(C2CC2C(N)=O)=O)cc1 33800,CCC(CC(C)C)C(=O)NCCN(c1ncc([N+](=O)[O-])cn1)CCOC 33801,N1(C(C(C(CC)C)OC)=O)CC2CCC(C1)N2C(=O)C(N1CCN(C)CC1)(C)C 33802,c1(C(=O)NC2C(Cn3cc(CN(C(C)=O)C)nn3)CCC2)cc(F)cnc1O 33803,C(=O)(C(CC(C)C)NC(c1c[nH]c(C#N)c1)=O)NC(C(CC)CC)C 33804,C1(C(=O)NCC2C(C)CN2C(=O)C2=COCC2)CCC(C2CCC2)CC1 33805,C1(CC(=O)NCC(CNC(=O)CCc2nccs2)F)CCCCC12CC2 33806,N1(C(C(CC)c2ccccc2)=O)CC(CNC(=O)CC(C)(F)F)C2(CC2)C1 33807,c1(Cc2cn(C(COCC)C(=O)NCC3COC(CO)C3)nn2)cccc(O)c1 33808,c1(C(=O)NC2CCCC(NC(CNC(=O)NC)=O)C2)cc(C)cc(F)c1 33809,c1(CNC(C2(CC(C)C)CC2)=O)ccc(CN(C)C(C2C(F)(F)C23CC3)=O)cc1 33810,c1(C(N2CCCC(CNC(=O)NC)C2)=O)cc(C#N)c(Br)s1 33811,CC1CCN(C(=O)OC(C)(C)C)C1C(=O)NCC1CCC(CC(C)(C)O)CC1 33812,N1(C(C(=O)NCc2ccc(C)cc2)=O)CCC(NC23CC2CNC3=O)C(C)C1 33813,C1(COC)(CNC(=O)Cc2c[nH]nc2O)CCCN1C(C1CNC(=O)N1)=O 33814,c1(C(=O)NCC2N(C(CC(C=C)C)=O)CC(O)C2)c[nH]c2ccncc12 33815,c1(OC)ccc(O)c(C(C)NCc2ccccc2Cn2cc(Cl)cn2)c1 33816,Cc1ccc(CCC(N2CC(C)(NC(c3cc(Cl)c(Cl)[nH]3)=O)C2)=O)cc1Cl 33817,C(CCC(C)NC(=O)C(N1CCOC1=O)C)NC(C(C)SCCCC)=O 33818,Cc1nnc2n1C(C(=O)N1CCN(C(c3csc4nnsc34)=O)C(C)C1)CC2 33819,N#Cc1cnn(CC(=O)OCCOc2ccc(Cl)cc2)c1 33820,FCCN=C(NCCNc1ccccn1)N1CCCC2(CCCNC2=O)C1 33821,C1(CNC(C2N(C)C(=O)NC2)=O)C(O)C(O)CN1C(c1ccc(F)cc1)=O 33822,c1(OC(C)C(N2CCN(C(=O)Cn3cccc3)CC2C)=O)cc(Cl)cc(Cl)c1 33823,O=C(C1=CCCC1)N1CCCC1CCCCNC(C12CC(CN1C1CC1)C2)=O 33824,C1(CC(N2CCC(NC(=O)CC3CC=CC3)(CF)C2)=O)CN2CCN1CC2 33825,C=CCCC(C(=O)Nc1ccc(C)nc1)NC(c1cc(C)n(CC)n1)=O 33826,N1(C(c2ncc(OCC)nc2)=O)CCCC(NC(=O)CCc2csc(C)n2)CC1 33827,Cc1cccc(C(N2C(C(=O)NCC=CC3CC3)CCC2C2CC2)=O)c1F 33828,c1(CN2CCC(N(C(C=CC(C)C)=O)C)CC2)ccc([N+](=O)[O-])cc1O 33829,C(CCCC(=O)NC1(C)CCN(C(=O)C2=COCC2)C1)OCC 33830,c1(C(N(CC(C)NC(CC(=C)Br)=O)C)=O)ncccc1S(=O)(=O)CC 33831,N1(C(c2cncc(COC)c2)=O)CCC2(CC1)CC2NC(C1CC2C=CC1C2)=O 33832,c1(N2CC(C)(C)C(NC(=O)CN3C(=O)CCC3=O)C2)nc2c(F)cc(Cl)cc2s1 33833,N1(C(c2c(CC)con2)=O)CCC(NC(=O)CCCN(C)C)C1c1ccccc1 33834,Cc1ccc(C#N)cc1NC(=O)C(C)N(C(=O)CSc1nc[nH]n1)C1CC1 33835,C(CC(C)C(=O)NCC1CC1NC(c1ccnnc1C)=O)=CCC 33836,Cc1cc(Cl)c(Cl)cc1C(=O)NCCN(C(=O)CC1(C)CC1F)C1CC1 33837,N1(C(c2cc(CCCCC)[nH]n2)=O)CCCOC(CNC(=O)C=CC=C(Cl)Cl)C1 33838,c1(OCC=C)cc(Cl)ccc1C(=O)NCC1(C(F)F)CCN(C(=O)C(C)OC)C1 33839,C1(C(C)C)CNC(=O)CN1C(C1CCC(N(C(=O)COC2CC=CC2)C)CC1)=O 33840,C(CC(CC)C(=O)N1C(CC(=O)NCc2cnc(C)n2CC)C2CCCC12)=CC 33841,C1(CCCNC(C2CCC(CC)O2)=O)CC2CCC(C1)N2C(c1coc(Cl)n1)=O 33842,N1(C(C2(C(C)=O)CC2)=O)CC2(CCN(C(=O)Cc3nnc(C)o3)C2)C1 33843,C12(CNC(c3cncc(C(N)=O)c3)=O)CCCC1N(C(=O)C=CC1CC1)CCC2 33844,c1(OC)ccc(C(F)(F)C(N2CC3CC3(CNC(=O)C(C)C3CCC3)C2)=O)cc1 33845,O=C(C1=NOC2(CCN(S(=O)(=O)C3CCCC3)C2)C1)N1CCc2ncncc2C1 33846,C#CC1CCCCN1C(=O)C(c1cn(C)nn1)NC(C1CCS1(=O)=O)=O 33847,CCC(CC(=O)N1CC(CO)(NC(=O)CS(=O)(=O)NC)C1)CC(F)(F)F 33848,C1(C(N(CC(CC)(C)OC)C)=O)(C(C)C)CCN(C(c2coc(C3CC3)n2)=O)C1 33849,C1(CC(N2CCC(NC(COCCN(C)C)=O)(CO)C2)=O)CC2CCC1CC2 33850,c1(C(N(CCCNC(=O)C2=NNC(=O)CC2)C)=O)ccc2nc(Br)nn2c1 33851,S(=O)(=O)(c1cc(C(=O)NC(C2CCN(C(=O)C3=COCCC3)C2)(C)C)co1)NC 33852,N1(C(C(C)OCCCC)=O)CC2CC2(C(=O)NC2CC3CCC2O3)C1 33853,C1(NC(c2c(C)cc(F)cc2)=O)CC2CC(NC(=O)C(C)(C)C3CCC3)CC2C1 33854,c12[nH]c3ccccc3c1CC1(CC)COCC(CCCNC2=O)CNC1=O 33855,N1(C(C(Cc2ccccc2)OCC)C(=O)NCCOC)CCC(S(N)(=O)=O)C1 33856,c1(NC2CCN(CC)CC2OC)cc([N+](=O)[O-])cc(CC)c1O 33857,C1(C)(C(=O)OC)CC(NC(=O)C=CC(C)NC(=O)C(c2cnn(C)c2)C)C1 33858,CCC(O)(CC)CCN=C(NCc1ccc2[nH]c(C)cc2c1)NC(C)C 33859,N1(C(c2ccc(F)c(C)c2)C(=O)NCC=C)CCOCC(C)(F)C1 33860,c1(C(=O)NCC2(COC)CN(C(CNC(CC)=O)=O)C2)cc(Cl)c(OC)cc1Cl 33861,C1(NC(C(CC=CC)NC(=O)CN2CCCCCC2)=O)CCC2(CCC2)CC1 33862,c1(C(=O)NC2CC(CNC(c3sccc3Cl)=O)C2)ncc(Cl)nc1Cl 33863,Cc1c(I)c(C(=O)OCc2cc(C3CC3)on2)nn1C 33864,O=C(CCS(=O)(=O)Nc1ccccc1)NC1CCN(C(=O)C=C2CC2)CC1O 33865,Cc1cc(C(=O)N(CCCNC(=O)CC(=O)NC2CC2)CC2CC2)ccc1O 33866,C(C)(C(CO)NC(c1ncoc1CCC(F)(F)F)=O)NC(C(C)N(C)C)=O 33867,c1(-c2cn(CC(=O)OC)nn2)cc(CN2CCC=C(CCO)C2)ccc1OC 33868,c1(C(=O)OC)c(C)ccc(C)c1C(=O)NCCC1CNCC1C 33869,c1(C(N2CCN(C(C(CC)C)=O)C3C2CC3)=O)cnc2c(c1)CCC(=O)N2 33870,CC1CCN(C(=O)C=C(Cl)Cl)C1C(=O)NCc1ccc(Sc2nc[nH]n2)o1 33871,N1(C(C(C)SC)=O)CC2CC3CC2C1C3NC(c1cc2sc(C)cc2[nH]1)=O 33872,CC1CCC(c2cn(CCC3CCCCN3)nn2)CC1 33873,c1(C(N(CC)CC2CCOC2)=O)n[nH]cc1CNC(=O)C(C)=CC1CC1 33874,C(=O)(C(F)CC(C)(C)NC(=O)CCC1CCOCC1)N(C)Cc1nccs1 33875,Cc1ccc(C=CCNC(C)CCCc2cccnc2)cn1 33876,Cc1c(N)ccc(C(=O)NC2CCOCC2NC(c2n[nH]c3c2COC3)=O)c1C 33877,N1(Cc2nc(C(C)OC)sc2)CC2CC1CN2C(C1CCCN(C(C)=O)C1)=O 33878,N1(C(C(CCC)CC)=O)CC2(CNC(=O)C(F)OC(F)(F)F)CC1CCO2 33879,CC1CC(C(N2CCC(NC(c3coc(Cl)n3)=O)C(C)C2)=O)CC(=O)N1 33880,c1(NC(=O)Cn2cc(-c3ccc(OC(F)F)nc3)nn2)cncc(OC(F)F)c1 33881,C(c1ccc(OC)cn1)=CC(N1CCC(CNC(CC=CC)=O)C1)=O 33882,CCCC(C(=O)N(CC(C)NC(C1(n2ccnc2)CCCC1)=O)C)C(C)C 33883,CCCC(C(=O)OC)C(=O)NC1CCC(CNC(=O)CC=CC(C)(C)C)CC1 33884,C1(NC(=O)CC2CSC2)CC(O)CN(C(c2cnn(-c3nccs3)c2)=O)C1 33885,C1(C(=O)NC(c2ccccc2)C(=O)NC(C2(O)CCC2)C)CCCOC1 33886,N=c1nc(N2CCC(C3CC3)C2)[nH]c(=NCc2ccc3c(c2)CCCC3)[nH]1 33887,Cc1cc(C)c(C(=O)NC2CCN(C(C3COCC3(C)C)=O)C2C(C)C)c(=O)o1 33888,Cc1n[nH]c(=NCC(C)(C2CC2)NC(=O)C(C)Cc2ccccc2C)s1 33889,C(CC(F)F)(C(=O)N1CCC1C(=O)N(C)C)NC(c1cc(CC)on1)=O 33890,C1(NC(c2sc(CC)c(C)c2)=O)CC2CCC1N2C(=O)COCC1CCCCO1 33891,C1(NC(c2c(C)cnn2C)=O)CC2CCC1C(NC(=O)C(C)OCCC(C)C)C2 33892,C1(C(=O)NCCCN(C)C(C2CSCN2C(C2CCCC2)=O)=O)CC2CCC1O2 33893,CCC(F)(F)CC(=O)N1CC2(CNC(c3nccn3C(C)C)=O)CCC1C2 33894,CCC(CC(=O)N1CCC1COC)NC(=O)CCc1ccccc1O 33895,c1(CC)ncc(Cl)c(C(=O)NC2(CC)CCN(C(C3CCOC(=O)N3)=O)CC2)n1 33896,C1(O)(CCNC(c2c(CC)occ2)=O)CCN(C(=O)CC2CCC(C)(C)O2)C1 33897,CC1(C)OC2CC(C(=O)NC3(c4nnnn4CCSC)COC(C4CC4)C3)CC2O1 33898,C1(C(N(CCN(C)C)Cc2c(F)cccc2Cl)=O)C2(CCC2)C12CCC2 33899,c1(C(=O)NC(CC)C(=O)OC)cc2n(n1)CCN(C(c1ccc(OC)nn1)=O)C2 33900,N1(C(c2c(C)ncn2C)C(=O)NCCCSC)CC2CCCCC2C1C 33901,O=C1NCCc2cc(F)c(NC(C3CC(=C4CCC4)C3)=O)cc21 33902,c1(CC)nc(C)ncc1C(=O)NCC1(F)CCN(C(=O)CCC2CCCO2)CC1 33903,N1(C(C2=C(C)CCCC2)=O)C(C)CC2CN(C(c3ccnc(C)c3C)=O)CC12 33904,N1(C(c2ccc(CCCCC)o2)=O)CC2C(C(=O)NC(C)C)C2C1 33905,C1(NC(C23C(C)(C)C(CC2)CC3)=O)CCCC2CN(C(c3cc(Br)co3)=O)CC12 33906,C1(CC)CN(CCNc2ccc3c(c2)O3)C(C)CO1.c1(OC)ccccc1C 33907,Cc1nccc(C(=O)NCCCN(C)C(C2CNC(=O)N2C)=O)n1 33908,N1(C(COCCOC)=O)C(C(=O)N(CCCC(=O)OC)C)CCC12CC2 33909,C(=O)(CCCC(=O)N1CCOCC(CNC(=O)C(C)CC(F)F)C1)OCC 33910,C1(O)(C(N2CC(O)(CNC(C3(C)CCC(C)C3)=O)C2)=O)CCCC(C)(C)C1 33911,CC(C)C(C)C(CNC(=O)CCc1ccon1)NC(c1cnc[nH]c1=N)=O 33912,CC1OC(C)(C)OC1(C)C(=O)NC12CC(NC(c3c[nH]cc(F)c3=O)=O)(C1)C2 33913,C(CC(N)=O)(C(=O)NCC1CCC2(CC1)CC2)NC(c1cccc(C)n1)=O 33914,Cc1cc(Cl)c(C(=O)N(C(C)(C)NC(c2cc(F)ccc2C)=O)CCO)cc1F 33915,C#CCC(C)(C(=O)NC1CN(C)CC12CC2)NC(=O)CSCC(F)F 33916,c1(CO)cnc2ccc(Br)cn12.c1(OC)ccc2cc1CN1C(CCC1)C(=O)N2 33917,c12ccc(cc1)oc2=O.C(=O)(C(C)=NOCC#N)N1C(c2c(C)ccs2)CCC1 33918,N1(C(C2=NOC(C)C2)=O)CCC2(CC1)CN(C(c1cn(C)cc1C(F)(F)F)=O)C2 33919,c1(NCc2c(C)noc2)[nH]c(=NC(C)COCCN(C)C)nc2c1ncn2C 33920,N1(C(=O)CCCn2cccc2)CCOC(c2ncc[nH]2)C1.c12ocnc1c(=O)[nH]o2 33921,c1(OCC)ccc(C(=O)NCC2(CNC(C3(C)CC3(C)C)=O)CCCC2)cn1 33922,c1(C(=O)NC(CC)CNC(C2CC3(CCC3)C2)=O)ccc(F)c(C)c1O 33923,CC(C)CC(C)CC(=O)NC(CNC(=O)Cn1cc(CN(C)C)nn1)CC(C)C 33924,c1(C(N2CCCC(CNC(C3(COC)CC(=C)C3)=O)C2)=O)cc(=N)[nH]c(Cl)n1 33925,C=CCC(CC(=O)NCC1CC(COC)C1)NC(=O)CN1CCNC1=O 33926,C(=O)(C#CC1CC1)N1C(C(N(C2CC2)CC2C(=O)NCC2)=O)C(O)CC1 33927,N1(C(CNC=O)=O)Cc2ccccc2C(NC(C23CCC(CF)(CC2)CC3)=O)C1 33928,N1(C(c2cc(C)c(C)o2)=O)CCN(C)CC1CNC(c1nocc1C1CC1)=O 33929,Cc1nc(C(=O)NCCCN(C)C(C2(C)CCCCNC2=O)=O)ccc1[N+](=O)[O-] 33930,C1(N(C(c2ccccc2O)=O)CC)CC(F)(F)CN1C(=O)Cc1sc(O)nc1O 33931,Cc1c(NCc2cscc2Cl)ncnc1N1C2CCCC1CC2 33932,C1(N(C(CC=C)=O)CCC)CCN(C(=O)C(C)C=C)C1 33933,N#CCCCC(=O)NC1C=CCC(C(N2CCN(c3ccccc3)CC2)=O)C1 33934,C1(NC)CCC(NC(=O)CCN(CCO)C(=O)OC(C)(C)C)CC1 33935,C1(NC(CCOC)=O)CC2(C1)CC(NC(c1cncc(-c3cnn(C)c3)c1)=O)C2 33936,CCC(CC(=O)NCC(C)CNC(c1nccc(C)c1N)=O)C(F)F 33937,C(=O)(N=S(C)(=O)C1CC(O)C1)c1nc2n(c1)CC(C(=O)OC(C)(C)C)CC2 33938,C1(CC)COCCN1C(=O)CC1CC1CNC(c1cc(-n2cccn2)ccn1)=O 33939,N1(C(CCCCC=C)=O)CC2(CCC2)CC1CNC(=O)CCc1cc(C)n(C)n1 33940,C1(OC)CC(CCNC(=O)C(F)C(C)C)N(C(C2CC(F)CN2C)=O)C1 33941,C1(NC(CNC(=O)CC2CCCC2)=O)CCCCN(C(c2ncsc2Br)=O)C1 33942,CC(C)C(C)(C)CNC(c1conc1C(C)NC(c1ncc(F)cn1)=O)=O 33943,Cc1cc(C(=O)NC2CCN(C(c3ccc(CN(C)C)[nH]3)=O)CC2)cc(F)c1C 33944,c1(OC)cccc2c1CC(C(N1CC(N(C(=O)CCSCC(C)C)C)C1)=O)CO2 33945,C#CCC(O)C(=O)NCCN(CC(C)O)C(C1CC(=C2CCC2)C1)=O 33946,C1(C(=O)NC(C(=O)OC)C(C)C)CC2CN(C(=O)Cc3cccnc3C)CC2C1 33947,CC(CC(=O)NCCN(C)C(c1cnc2sccc2c1)=O)P(C)(C)=O 33948,N1(C(CC)=O)CCC(C2CCN(C(c3cc(F)c(Br)c(F)c3)=O)C2)CC1 33949,C(=O)(C(C)S(N)(=O)=O)N1CCC(NC(c2ccc(C)cc2)=O)C1C 33950,c1(-c2c(SC3(C(=O)OC)CCC3)ncnc2)ccccc1S(=O)(=O)NC 33951,C(C(C)CC(=O)N1CC2C(CNC(c3ccncc3SC(C)C)=O)C2C1)OC 33952,C1(CS(=O)(=O)NCC2CC(=C3CC3)C2)CC2C(C1)C2(F)F 33953,C(=O)(C1CCc2scnc21)N1CC(C(C)NC(c2ccn(C)c2)=O)OCC1 33954,N1(C(COC)=O)CCc2nc(CNC(C3CCC4C(C3)C4(F)F)=O)sc2C1 33955,C1(NC(c2n(C)ncc2)=O)CC2CC1CN2C(c1ccncc1F)=O 33956,c1(CCC(c2n(CCC)nnn2)NC(c2nnnn2C)C)ccc(F)cc1 33957,c1(N2CCC(CSCC)CC2)cc(C)c(S(=O)(=O)NC2CCCC(C)C2)cn1 33958,N1(C(COCC=C)=O)CC(NC(C2CCCCC(=O)N2)=O)CC12CCOCC2 33959,N1(C(c2cc(OCC)n[nH]2)=O)CCC2(CCCN(C(=O)CC3(CO)CC3)C2)C1 33960,C1(NC(c2cncnc2C2CC2)=O)CCCN(C(C2CCCC3(CC3)C2)=O)CC1 33961,C1(O)(CNC(c2ccc(F)c(CO)c2)=O)CCCN(C(c2cnn[nH]2)=O)C1 33962,c1(C(N2CC(O)(C3CCCN3C(C3(C4CCCO4)CC3)=O)C2)=O)ccnc(Cl)c1 33963,C(=O)(C(C)(C)O)NCCN(CC(C)(C)CC1CCOCC1)CCOC 33964,c1(OCCNC2(c3ccc(-c4cn(CCCC)nc4)cc3)CC2)c(C)cccc1F 33965,CC(C)CC(CC(C)C)C(=O)N(C)CC1CN(C(C2OCC2(C)C)=O)CC12CC2 33966,C1(NC(C=Cc2cc(OC)ns2)=O)CC2CCC(C1)N2C(=O)Cc1c[nH]nc1C 33967,c1(C(N2CCC(COC)(CNC(=O)C(F)CC3CC3)C2)=O)cn2c(n1)CCC2 33968,CC(C)CCC(C)N=c1[nH]c(=NC2COC3(CCN(C(C)C)CC3)C2)[nH]c2cc[nH]c12 33969,CP(C)(=O)CC(=O)NCCNC(c1cc(Cl)sc1Cl)=O 33970,N1(C(C2(CC)CC2)=O)CCC2(C1)CN(C(=O)C(C)(C)n1cnc(C)c1)CCO2 33971,C1(N(C(=O)CSc2nnnn2C2CCCC2)C)CCC(NC(C2(C)CC2F)=O)CC1 33972,c1(CN(C)Cc2nn(CC)nc2C)ccc(C)cc1C 33973,C12(CNC(C3CCCC(NC(c4nc(C(C)C)oc4)=O)C3)=O)CCC(CC1)OC2 33974,c1(CC(C)C)ccc2cc(C(=O)NC3CCNCC3)[nH]c2c1 33975,c1(C(=O)NC2CCCCN(C(C3C(OC)CCCC3)=O)C2)cc2c([nH]1)CCOC2 33976,N1(Cc2ccc(OC(C)=O)cc2)CCC2CN(c3ncc4sccc4n3)CCC12 33977,c1(C(=O)NC2CCN(C(c3c(OC)ccs3)=O)C2)ccc(C2CC2)c(OC)c1 33978,N1(C(C2(CC#C)CCCOC2)=O)CC2(CCN(C(=O)CC3CCCC3)CC2)C1 33979,C1(CNC(CN(C)S(N)(=O)=O)=O)CN(C(=O)CCc2ccsc2Cl)CC1O 33980,C1(C(N2CC(CCNC(c3c(C)c[nH]n3)=O)OCC2)=O)CC1C1(C)COC1 33981,C(C(=O)NC1CC2(C1)CC2C(=O)NCC1(C#N)CC1)(C(C)C)NC(C)=O 33982,CC1CCC=C1C(=O)N1CCN(C(CNC(=O)CCC2CCCC2)C(F)F)CC1 33983,c1(CC(=O)NC2C3(CN(C(c4n(C)cnc4)=O)C3)CC2)cccc([N+](=O)[O-])c1 33984,Cc1csc(C(=O)NC2CN(C(=O)CCc3ccc[nH]3)CC2F)c1Cl 33985,c1(CCC)cc(=NC2CCCC(NC(C3(C)CC3)=O)C2)[nH]c(Cl)n1 33986,N1(C(CCCC(C)=O)=O)CCN2C(=O)C(NC(c3ncn(C)c3C)=O)CC2C1 33987,CC(C)(C)C(C)(O)C(=O)N1CCCN(C(c2coc(C(F)(F)F)n2)=O)C(CO)C1 33988,c1(SC)ccnc(NC2CCCCC2NC(c2cn(C3CCOC3)cn2)=O)n1 33989,C1(C(N(CC)Cc2ccc(O)cc2)=O)CCCN(C(c2cnoc2C)=O)CC1 33990,c1(C(N(CC(C)N(C(=O)Cn2ncc(O)nc2=O)C)C)=O)cc([N+](=O)[O-])nn1C 33991,C1(NC(c2c(C)n(C)nc2)=O)C(C)CN(C(=O)CC(C2CC2)C2CC2)CC1C 33992,C1(CNC(c2c(C)cc(O)nn2)=O)CN(C(c2ccc(F)cn2)=O)CCC1(F)F 33993,CC1(C)CN(C(=O)NCc2ccccc2)CCC1C(=O)OCCSCCCN 33994,C1(CNC(c2c(C)scn2)=O)CC(NC(=O)Cc2sccc2Cl)C1(C)C 33995,c1(OC)cc(NC(=O)C(=O)N(CCCN(C)C)C)c(Br)cc1Br 33996,C(c1cccc(F)c1F)=CC(=O)NC1CCCC(CNC(C(C)O)=O)C1 33997,CCC(C(C)C)C(C(=O)NCCC)N1CCC(N2CCC(O)CC2)CC1 33998,C1(C(N(C)CCN(C(=O)C=CC(=O)NC2CC2)C)=O)CC(=O)N(C2CC2)C1 33999,C1(CC)CN(C(=O)C(F)OC(F)(F)F)CC1C(=O)N(C)Cc1ccc(F)cc1 34000,Cc1ccc2c(C(=O)N(C)CCN(C)C(C3SC4C=CC3CC4)=O)c[nH]c2c1 34001,N1(C(CNC(C)=O)=O)CCN(CCN(C)C(C2CC2Cl)=O)CC1 34002,C1(NC(N(C)C)=O)CC(CNC(c2coc(N(C)C)n2)=O)C12CCC2 34003,N1(C(Cc2cccc(C)c2)=O)CCN(C(=O)Cc2ccccc2F)CC(CO)C1 34004,C1(NC(CCOCCOC)=O)CCN(C(C2(c3ccc(C)nc3)CC2)=O)CC1F 34005,N1(C(C=Cc2cn(C)nc2)=O)Cc2ccccc2C1CNC(c1cnns1)=O 34006,c1(SC)nc(N2CC3CC2CN3C(=O)C=Cc2ccccc2)c(Br)c(C)n1 34007,c1(OC)cccc(-n2cc(CNC(=O)CN3CC(C)(C)C3)nn2)c1C 34008,c1(OC)ccc(CC(=O)NC2CC(NC(c3csnn3)=O)C23CCC3)c(F)c1 34009,c1(C(=O)NCC2CC(F)CN2C(=O)C=CC2CCCC2)cc2cc(Cl)cnc2o1 34010,C1(CNC(CNC=O)=O)CC(O)CN1C(=O)CCN1CCOCC1 34011,n1(C(C)C)cnc(CN2CCCC2C(=O)NCC2(F)COC2)c1 34012,N1(C(CN(CCC)C)=O)CC2CCCC2(C(=O)NC2(CC3CC3)CCC2)C1 34013,C1(C(=O)NC2CN(C(C3(SC)CC3)=O)CC2CC2CC2)CC(C)(C)OC1(C)C 34014,N1(S(=O)(=O)c2cccc(Br)c2)CCC2(CCCC2N2CCNCC(F)(F)C2)CC1 34015,C1(CCNC(C2(Cl)C(C(C)=O)C2)=O)CCCN(C(c2[nH]nnc2C(F)F)=O)C1 34016,N1(C(CC(C)C(F)F)=O)CC2(CCN(C(=O)C=Cc3ccn(C)c3)C2)C1 34017,C1(CCOC)(NC(c2ccon2)=O)CCN(C(C2CCOC2C)=O)C1 34018,C#CCCCC(C)C(=O)NC1CC(F)(CNC(c2cc(F)c(F)cc2F)=O)C1 34019,N1(C(CN(CC)Cc2ccccc2)=O)CCCCC1CNc1cnccn1 34020,C1(C(=O)OC)COC2(CCC2)CN1CCC(C)F 34021,N1(C(=O)Cc2ccc(Cl)s2)CC2CCCC(N=c3cnc(F)c[nH]3)C2C1 34022,N1(C(c2ncc(F)cc2F)=O)CC2CCN(C(C3CC4CCC3O4)=O)C2C1 34023,C12(CNC(c3ccc(Cl)cn3)=O)CC1CN(C(c1cccc(=O)o1)=O)C2 34024,N1(C(C2(SCC)CC2)=O)CC(NC(c2cnc(CC3CC3)s2)=O)C2(CC2)C1 34025,N1(C(CC(CNC(c2ccc(Cl)o2)=O)O)=O)CC2(CCCC2)C1 34026,c1(C(=O)NC2CC(NC(CCCC)=O)C23CCC3)cc2cnc(Cl)cc2s1 34027,c1(N(C)Cc2cccc(C(F)(F)F)n2)ccc(S(=O)(=O)NCC2(C)CCCS2)cn1 34028,c1(CCC)nc(=NCCCCC(C)NC(=O)C=C2CCCCCC2(F)F)s[nH]1 34029,c1(C(=O)NC2CCC(CNC(c3cc(C)oc3)=O)C2)ccc([N+](=O)[O-])n1C 34030,C12(NC(C(C)OCC=C)=O)CCCC1(F)CN(C(c1[nH]nc([N+](=O)[O-])c1Cl)=O)C2 34031,N1(C(c2c(COC)nn(C)c2)=O)CCC(C)C(NC(=O)COC(C)C)C1C 34032,c1(NC(CC2CCN(C(CC=CC=C)=O)C2)=O)cccc(CC(=O)OC)c1F 34033,C1(C(N2C(CNC(CC(C)SC)=O)C(O)CC2)=O)CC2CCC(C1)C2=O 34034,CC1CN(C(=O)CCCOC(C)(C)C)CCCN1C(=O)C(C)C#N 34035,C1(N(C)C)(C(=O)NCC(CNC(=O)C(F)=C2CCCC2)CO)CCCOC1 34036,C#CC1(NC(C2C=CC(NC(=O)CCCOCCC)C2)=O)CCCCC1 34037,N1(C(C2(C)CCCCNC2=O)=O)CCOC2(CCN(C(=O)C=CCF)C2)C1 34038,C=CC(C)(O)CC(=O)NCC(C(=O)NCc1sc(C)cc1C)OC 34039,c1(OCCC)ccc(Cl)cc1CC(N1CC2C(NC(=O)C3=C(Cl)CC3)C2C1)=O 34040,c1(N(C)Cc2ccc(C(N)=O)cc2)ccnc2cc(F)cnc12 34041,c1(OC)ccc(CNC(C(C)(C)OC)c2nnnn2CC(F)F)cc1C#N 34042,O=C1CCCC(CNC2COCCC2c2ccc(F)cc2)C1 34043,C1(C(=O)NC2CC(CNC(C3(F)CC4(CCC4)C3)=O)C2)CC2(C1)CC(F)(F)C2 34044,c1(C(N(CC(C)NC(C=CC(=O)OCC)=O)C)=O)ccc(C2CCC2(C)C)cc1 34045,C1(C(=O)NC2CCC(NC(c3ncc(C)cn3)=O)C2)Cc2ccc(Br)cc2C1 34046,C(=O)(C(C(=O)NCCCN(C)C(c1cn(C)c(=O)n1C)=O)C(C)C)OCC 34047,N1(C(C)=O)CCCC1CC(=O)N(CC(C)(C)CNC(C1(C(F)F)CCC1)=O)C 34048,C#Cc1ccc(CCC(=O)NC2CCN(C(c3cnn(C)c3)=O)C23CC3)cc1 34049,c1(C(=O)NC(CCOC)CNC(c2c[nH]nc2C)=O)c(Cl)c([N+](=O)[O-])nn1C 34050,N1(C(C2CC23CCOC3)C(=O)NC(C)C)CCc2ccc(F)c(F)c2C1 34051,C1(C(C)CNC(C2(F)CCC2)=O)CCN(C(c2ccc(O)nc2)=O)CC1 34052,C1(NC(c2c(CC)onc2)=O)CCCN(C(c2coc(Cl)c2)=O)C1C 34053,CCC1=NOC(C(=O)NC2CC2NC(c2cn(CCO)nn2)=O)C1 34054,C1(NC(c2ncn(CC)n2)=O)CN(C(c2sccc2CC#N)=O)CC1C 34055,CC(C(C)c1nc(-c2cnn(C)c2)nn1CC1CCCC1(F)F)C(C)(C)C 34056,CCCCC(C(=O)N1CCSCC(C)C1)NC(C1CC2(CC(=O)C2)C1)=O 34057,c1(OC)ncnc(Cl)c1NC(=O)CC1(Nc2ccc(C)cc2Cl)CCC1 34058,C1(CNC(CCC(=C)C)=O)CN(C(C2CC2C(=O)OCC)=O)CCC12CCC2 34059,C1(CNC(c2cc(C)cc(O)n2)=O)CC2CCC(C1)N2C(=O)CC(O)CN(C)C 34060,Cc1ccc(Cl)c(C(=O)NC23CC2CN(C(c2ccc(C4CC4)nc2)=O)C3)c1 34061,CC1(C)OCCC1(O)C(=O)NC1CCC(CC(=O)NC2CC23CCC3)CC1 34062,c1(C(N2CCC(N(C)C(c3csc(C(F)(F)F)c3)=O)C2)=O)cc(F)cc(F)c1 34063,N1(C(c2nc(C)oc2C)=O)CCCC2(C1)C(NC(=O)C(C)NC(N)=O)CCN2C 34064,c1(C(=O)NC2(C)CN(C(C=CCOC)=O)C2)ccc(S(=O)CC#N)cc1 34065,CC1(NC(C23CC(CN2C(c2cc(N)cc(F)c2)=O)C3)=O)CN2CCC1CC2 34066,c1(CN(C(=O)C(CCc2ccccc2)C(=O)O)CC)cc(Cl)cc(Cl)c1 34067,C1(NC(C(C)OCCN(C)C)=O)CCSC12CN(C(=O)C(F)=C1CCCC1)C2 34068,N1(C(=O)OC(C)(C)C)CC(C(=O)OCC#CC(=O)NCC(F)(F)F)OC(CO)C1 34069,c1(C(C)NC(c2c(C)n(C)cn2)=O)ccc2c(c1)CN(C(=O)C(F)C(C)C)C2 34070,Cc1c(C(N2CCCC2C2(C(=O)NCCCC3CCOCC3)CC2)=O)cnn1C 34071,c1(OC)cnnc(C(=O)NCC(O)CC(=O)NCC(C)SC)c1 34072,C1(NC(C2(CCO)CC2)=O)CCCN(C(C2(C(F)(F)F)CCOCC2)=O)CC1F 34073,N1(C(CC=C)=O)CCCC2(C1)CN(C(=O)CC1OCCOC1(C)C)CCO2 34074,C(N=c1ccc(-c2ccncc2)c[nH]1)c1cc(C)nc(O)c1 34075,C1(NC(CN(C(=O)CN(CC(C)(C)C)C)CCC)=O)CCOC(CC)C1 34076,c1(CC(=O)NCC2(CNC(CCOCCN(C)C)=O)CC2)nn(C)cc1Br 34077,Cc1nsc(C(=O)NCC2CCCN(C(=O)C(C)(C)C3CCC3)C2)c1N 34078,CCC(C)CCC(=O)NCc1ccc(C(N2CC(OCCF)C2)=O)s1 34079,CCC(CC(=O)Nc1cnn(CC2CC2)c1)N(C(=O)CC1(C)CC1)C 34080,C1(CN(C(C(C)OCC)=O)C)CCCN(C(c2ccc(CC3CCC3)cc2)=O)C1 34081,N1(C(CS(CC)=O)=O)CC(CNC(=O)C(F)(F)c2nccs2)CC(C)C1 34082,C1(C(N(C(CN(C)C(=O)OC(C)(C)C)(C)C)C)=O)CC(C2CC2)=NO1 34083,C=CC(C)(CC)OC.c12c[nH]nc1COC2=O 34084,N1(C(c2cnn(C)c2)C(=O)NC(C(=O)OC)CC(C)C)CCCC(C2CCC2)C1 34085,N1(C(CN(C(C)C)C)=O)CC2CCC(NC(c3cnn4ccncc34)=O)C2C1 34086,C1(NC(C(=O)N(C)C)=O)CCC2CCN(C(c3ccccc3SCCO)=O)C1C2 34087,c1(OC(C)C)cncc(C(=O)NCC2CN(C(=O)Cc3cc(Cl)cs3)C2)c1 34088,C1(C)(CNC(C2CC(CCC)C2)=O)CCN(C(=O)Cc2ncoc2C)CC1 34089,C(=O)(CS(=O)(=O)C(C)C)N1C(COC)(CNC(=O)C=CC(C)(C)SC)CCC1 34090,c1(N2CC3(CN(C(c4c(OC)nccc4)=O)C3)C2)ncnc2scc(C)c12 34091,C1(NC(=O)NC2C=CCCC2)CCC=CCC1 34092,Nc1nc(Cl)ccc1C(N1CC2CC2(CNC(=O)CCC2CC2(Cl)Cl)C1)=O 34093,N1(C(=O)Oc2ccc(Cl)cc2)CCC2COCCC12 34094,CCC(C)(C)C(C)OC(C1CCCN1C(=O)OC(C)(C)C)=O 34095,C#CC1(NC(C2CC(NC(c3csc(F)c3)=O)C23CCC3)=O)CCCCC1 34096,N1(C(c2nc(COC)oc2)=O)C2CCC1CC(NC(=O)Cc1ccc(Br)cc1)C2 34097,C1(O)(COC)CCN(c2nnnn2NC(c2ccc(Cl)cc2)c2ccsc2Br)C1 34098,C1(C#N)(C(=O)NCC(C)NC(c2cccnc2C(F)(F)F)=O)CC1(C)C 34099,Cc1csc(Cl)c1C(=O)NCCCN1CCN(C(=O)CSc2ccncc2)CC1 34100,c1(Cn2cc(CNc3cc(C)cc(C)c3)nn2)ccc2c(c1F)OCCO2 34101,Cc1c(C(=O)NCCC(C)(C)NC(C2CC2(C)C(F)F)=O)cnc2ncnn12 34102,n1(CC(C)C)cccc(C(=O)N(CCCCNC(C2CC(C)(F)C2)=O)C)c1=O 34103,c1(CN(c2c(C)ccs2)C)nc(C(C)O)nn1-c1ccc(Br)nc1 34104,O=C(C(c1cccs1)=Cc1cccs1)NCCC1CCC(C(F)(F)F)O1 34105,C1(CC(=O)N(C(COC)C)C)CCN(C(=O)CC=C(Cl)Cl)C1(C)C 34106,C(=O)(C1=CCCCCC1)NC(CC#C)C(=O)NC1C=CCCC1CO 34107,c1(NC(N2CC(NC(C(F)=CC)=O)CC2(C)COC)=O)ccc2ccccc2c1 34108,N1(C(C(C)SCC)=O)CCC2CCCC12C(=O)N(C)CC1CC(F)C1 34109,C(=O)(C(C)(CNC(c1nn(C)cc1Cl)=O)CC)NCCOCC 34110,N1(C(CN2CC(C)C2)=O)CCC2C(C1)CN2C(=O)C(N1C(=O)CCC1=O)C 34111,c1(C(N2CC(C)N(C(C3CC(C(C)C)C3)=O)CC2)=O)cc2occc2n1C 34112,CC1C(NC(=O)C(C)(C)c2ncco2)CCCN1C(C1C(C)(C)C1(C)C)=O 34113,C1(CC)CCC(C(=O)N(C)CC2CCCN2C(c2cnsc2)=O)CC1 34114,c1(C(=O)NCC2CCCN2C(C2CC(CF)C2)=O)cc2c(F)c(Cl)ccc2[nH]1 34115,c1(C(=O)NC(COC)CNC(c2cnn(CCO)c2)=O)cnc(Cl)n1C 34116,C(=O)(C1=CCCCC1C)N1CCCC(C(=O)NCC(C2CC2)SC)CC1 34117,N1(C(C2CCN(c3n(C)ccn3)C2)=O)CC2(CCN(C(c3cnsn3)=O)CC2)C1 34118,C(=O)(CCCS(=O)(=O)NC(=O)Nc1nc(C)no1)OC 34119,C1(NC(COCCCCCC)=O)CCC2(CC1)CN(C(=O)Cc1nccn1C)C2 34120,C1(CNC(C(C2CN(C(c3cc(OCC)n[nH]3)=O)C2)OC)=O)CCCCN1C 34121,C1(F)(C(=O)OC)CCN(C(=O)COC)C1.c12ccc(cc1)OC(=O)N2 34122,N1(C(CC2C(NC(C3(C)C(C)(C)C3)=O)CCC2)=O)CC(CO)C2(CCC2)C1 34123,c1(C(=O)NCC(C)CNC(=O)C(C)Cc2ccccc2F)cccc(N)c1Br 34124,C1(NC(=O)NCc2ccc(S(C)=O)cc2)CCC(F)(F)C(C)(C)O1 34125,c1(C(=O)NCC(CCOC)NC(C2CC3CC3C2)=O)oc(COC)nc1C 34126,CC1CCCCN1CCC(=O)NCC1CC1NC(c1ccc(SC(F)F)cc1)=O 34127,C(=O)(C(CC(C)C)NC)N1C(C(N2CCCC(CCC=C)C2)=O)(C(C)C)CCC1 34128,N1(C(c2ccc(CC)cc2)=O)CCCCCC1CNC(=O)C(C)(CC)CO 34129,C(=O)(C1=C(SC)CCCC1)N1C(CN(C(C(CC)CC)=O)C)CCCC1 34130,N1(C(c2ccn(CCC)c2)C(=O)NC(C)C(=O)OC)CC(CO)C1(C)C 34131,c1(C(N2CC3C(NC(c4cnc5sccn45)=O)(C3)C2)=O)c(F)ccc2n[nH]cc12 34132,N1(C(C=COCC)=O)CC(NC(c2cc3n(n2)CCC3)=O)C(C)(C)C1 34133,c1(CC(=O)NCCNC(C2CCSCC2)=O)noc2ccc(Br)cc12 34134,N1(C(C2N(C)CCN(C(C(c3cnn(C)c3)C)=O)C2)=O)CCCC(C)(C)CC1 34135,C1(CC(C)(C)C#N)C(=O)N1.N1(CCS(C)=O)CCC(SC(F)(F)F)CC1 34136,Cc1c(C(=O)NCC2CC2CNC(C2(CC(F)F)CC2)=O)cnn1C1CCCC1 34137,c1(-c2cnc(C3N(C)CCC3)s2)nc(C2CCCCC2)nn1CCCO 34138,C1(C(=O)Nc2c(C)cccc2CO)CCN(C(=O)CNC(=O)C2CC2)C12CCC2 34139,c1(NC(C2C(NC(c3cc(-c4ccco4)on3)=O)CCC2)=O)ccc(Cl)cc1Br 34140,C1(C(N2CCCC(Cn3cc(C(CC)O)nn3)C2)=O)CCc2nc(O)[nH]c2C1 34141,c1(NC(C)=O)ccc(NC(c2nnnn2C(C)(C)C)(C2CCCCC2)CF)cc1 34142,CC(C)C(C)C(C)CC(=O)NC(C)CC1CCN(C(=O)Cn2cnc(=N)[nH]2)CC1 34143,CCCC(O)C(=O)NCC(C1CCN(C(C2(C)CCNC2=O)=O)CC1)O 34144,N1(C(C(CC)CCOC)=O)CC(C(N2CCCN(C)CC2C)=O)C2(CCC2)C1 34145,C1(NC(C(COCC)(C)C)=O)COC2CN(C(=O)C(F)C(C)(F)F)CC12 34146,C(=O)(C1CC(=O)c2ccccc21)N1C(C)(CNC(C(C)NC(N)=O)=O)CCC1 34147,Cc1cc(C(=O)N(C2CN(C(C3(C)CCCCCC3)=O)CC2(C)C)C)nc(C)c1 34148,C=CC(C)(CC)C(=O)N(CCCNC(=O)CNC(=O)COc1ccc(F)cc1)C 34149,Cc1cncc(C(=O)NC2CCCC2NC(=O)CCF)c1Cl 34150,c1(C(=O)NCC(C)(Cn2cccn2)NC(=O)C(F)=CC2CC2)cc(Cl)ccc1O 34151,C1(NC(C2CN(CCOC)C(=O)C2)=O)CN(C(=O)C(F)=C(C)C)CC(C)(C)C1 34152,Cc1oc(Cl)nc1C(=O)NC1(CCCC(=O)NC2CC(C(F)F)C2)CCC1 34153,CC1CC(NC(=O)C(C)S(N)(=O)=O)CN(C(=O)C(C)(C)F)C1 34154,N1(C(c2n(C(C)C)ccn2)=O)CCC2CCN(C(c3ccnc(S)c3)=O)CC2C1 34155,N1(C(c2c(C)[nH]cc2)=O)CC(NC(C2CCC(N(C)C)CC2)=O)C2CC12 34156,C1(NC(C2CCC3CC23)=O)CN(C(c2cnc(Br)s2)=O)CC12CC2 34157,C1(NC(CN(C2CCCC2)C)=O)CC(F)CN(C(c2c[nH]nc2C(C)(C)C)=O)C1 34158,N1(C(CNC(=O)OCC=C)=O)CCOC2(CCCN(C(=O)CC3CC3)C2)C1 34159,C(=O)(CCC(=O)NCC1(CNC(C2CC2C(F)F)=O)CC1)c1cn(C(C)C)nc1 34160,CC(C)CC(C)(O)C(=O)NC(C)CCNC(c1ccn2ccnc2c1)=O 34161,C(=O)(C(C)(C)Cc1cnn[nH]1)N1CC(CNC(c2cc(COC)[nH]n2)=O)(OC)C1 34162,c1(CNC(C2(C)CCN(C(c3cc(C(C)=O)cn3C)=O)C2)=O)ccn(C)c(=O)c1 34163,CC1=CC(O)CN(C(=O)N(C)C)C1.c12nc(cs1)C(C)N2 34164,C1(CNC(=O)CN2CCOCC2)CC(F)(F)CN1Cc1ncc(Cl)cn1 34165,c1(C(N2CC3N(C(CN(C)S(N)(=O)=O)=O)C(CC3)C2)=O)cc2ccc(Cl)cn2c1 34166,c1(CC)ncc(C(=O)NC(CO)C(C)NC(c2ccncc2C)=O)c(O)n1 34167,Cc1cc(C(=O)NC2CCCC23CN(C(=O)C(F)C(F)(F)F)C3)cc(N)c1Cl 34168,C1(NC(CC2CC(=C)C2)=O)CCCC1NC(=O)C(C)(C)C1(C)CC1(F)F 34169,C(=O)(C(F)C(C)(F)F)N(C1CCN(C(C2(CC=C)CC=CC2)=O)C1)CCC 34170,c1(OC)cc(C2CCN(C(C3(C)CCN(C(C)=O)C3)=O)CC2)cnc1OC 34171,C1(C(=O)NCCN(C(=O)C(C)N2CCC2)CC)CCC(NC(N)=O)CC1 34172,c1(CC)noc(C(=O)N(C2CCN(C(C3(CO)CC3)=O)CC2)CC)c1C 34173,c1(C(=O)NCC(C)CNC(=O)Cc2cccc(F)c2O)cnc2c(c1)nnn2C 34174,c1(NC(c2cccc(OCCCl)c2)C(=O)NC(CC)C)cn(C2CC2)nc1C 34175,CCC(O)C(C)(C)C(=O)N1CCN(C(=O)C(C)(Cl)Cl)CC(O)C1 34176,c1(C(=O)NC2C(C(=O)NC(CC=C)C(=O)OCC)CC2)cc(C)nc(O)n1 34177,c1(CNCc2cccc(C(=O)OCc3ccccc3)c2)cc(CCO)cc(Br)c1 34178,Cc1ccsc1C(N1CCCC1CCNC(=O)C(C)SC(F)(F)F)=O 34179,C1(C(=O)NCc2cc(OCC)c(OC)cc2)CC2(CC(=O)CCS2(=O)=O)C1 34180,N1(C(CCCCC=C)=O)CCCCC12CN(C(c1cn(CCC3CC3)nn1)=O)C2 34181,O=C(C1Cc2ccccc21)N1CCC(N2CCN(C(C3(CO)COC3)=O)CC2)C1 34182,N#Cc1cnc(N(C(=O)CC2CCCO2)CC2CC2)c(Br)c1 34183,N1(C(c2c(C(=O)NCCCOC)c[nH]n2)=O)CCC(CCOC2CC2(F)F)CC1 34184,N1(C(CN(CC#C)C(C2CC=CCO2)=O)=O)CC(O)CC1CC 34185,c1(C(N2CCC(Cn3cccn3)C2)C(=O)NCC=C)nn(C(C)C)nc1Br 34186,Cc1cc(Br)cc(C(=O)NC2(CCO)CN(C(C3CC(C)CO3)=O)C2)c1C 34187,N1(C(C2(CF)CCN(C(CC(C)(C)OC)=O)C2)=O)CCCCC(C)C1 34188,C1(C)(C(N2CC(NC(c3c(C)occ3C(F)(F)F)=O)C2)=O)OC(C)(C)OC1C 34189,C(=O)(C1CSc2ccccc21)NCCC1(C)CCN(C(C2CC(O)C2)=O)C1 34190,C1(CNC(CCCC#CC)=O)CC12CCN(C(C1CC3CCC(C1)N3C)=O)CC2 34191,C1(C(=O)NCC(COC)NC(CC2N(CC)CCC2)=O)CCc2cnnn2C1 34192,N1(C(C(COC)C(F)(F)F)=O)CCCC2(NC(=O)CS(C)(=O)=O)CCCC12 34193,N1(C(c2cnc(C3CCC3)o2)=O)CCN(C(c2cnn3c2OCC3)=O)C(CO)C1 34194,c1(CC)ncc(C(=O)NC2CC3CN(C(c4ocnc4C(F)F)=O)CC23)c(O)n1 34195,CC1(C)CCCC(C(N2CC3(CC(CNC(=O)Cc4cn[nH]c4)C3)C2)=O)C1 34196,C(C(=O)NCC1CC(C)N(C(=O)CN(c2ccccc2)C(C)=O)C1)(C(C)C)OC 34197,c1(C(=O)NCC(=CC(=O)NC(CC=C)CO)C)n[nH]c(C)c1Cl 34198,C1(NC(c2coc(C(F)F)c2)=O)(CF)CCN(C(c2cncnc2)=O)C1 34199,C(C1=NCC(c2ccccc2)O1)Nc1cnccc1 34200,C1(CCNC(C(C)(C)OCC)=O)CN(C(c2coc(N(C)C)n2)=O)CC1C 34201,N1(C(C(C2CCCCCC2)OC)=O)CCCC(C)(NC(c2csc(Cl)c2Cl)=O)C1 34202,CC1CC(NC(=O)CC(C)(C)F)CN(C(c2cncnc2)=O)C1 34203,c1(C(N(CCNC(C2(C)C(C)CCC2)=O)CC2CC2)=O)cnn2c1CCC2 34204,c1(NC(C2CC3CC3N2C(=O)CCN2CCOCC2)=O)cccc(C(F)(F)F)c1 34205,N1(C(CC=C=C)=O)CC2CC1C2NC(c1ccccc1)=O 34206,N1(C(c2n(CCOC)ncc2)=O)CCCC1(C)C(C)(C)CNC(=O)C(F)C1CCC1 34207,c1(C(N(CCCOCCNC(C2CCC(F)C2)=O)C)=O)nnn(C)c1N 34208,C1(C(F)(F)F)(OC)CCCN(C(C(=O)NC(C)C)c2nccs2)C1 34209,c1(OC)ncccc1-c1cn(CCCNC(=O)C(C)(C2CC2)OC(=O)C2CC2)nn1 34210,C1(C(=O)NC2CC(NC(c3c(C)nsc3)=O)C2)C2CN(C(=O)OC(C)(C)C)CC12 34211,CCC(CCOC)C(=O)N1CCC(CN(C)C(C2COC(=O)N2C)=O)C1 34212,C(=O)(C(C)(C)CC(F)(F)F)N(CCNC(C(CCC)N(C)C)=O)CCC 34213,N1(C(C(c2cccc(Cl)c2)CC)=O)CCN(C(c2ccc(Cl)cc2N)=O)CC1C 34214,c1(C(=O)NCC2N(C(c3c(CC)nn[nH]3)=O)CC(O)C2)cnc(C)cc1Cl 34215,C1(C(=O)NC)COCCN1C(c1cccc(-c2cc[nH]n2)c1)=O 34216,c1(C(=O)NCC2(O)CCN(C(C3C(c4cc(C)on4)C3)=O)C2)cccc(=S)n1O 34217,c1(C(N2CC(C(=O)NCc3c(OC)c(F)ccc3)C2)=O)cc(F)c(F)cc1Cl 34218,c1(C(=O)NC(C2(O)CN(C(C(CC)N(C)C)=O)C2)C)cc2nccnc2cc1C 34219,C=Cc1cncc(C(=O)NC(C2CCOC2)CNC(c2c(C)cnnc2O)=O)c1 34220,N1(C(C(C2CCN(C(c3cnn(C4CC4)c3)C)C2)F)=O)CCC2(COC(C)C2)C1 34221,c1(C(=O)NCC2CCN(C(CN(C(COC)=O)C)=O)CC2)ccc(Cl)cc1Cl 34222,C1(NC(C2CCC=CO2)=O)CN(C(=O)COc2ccon2)CC12CCOCC2 34223,c1(OC)c(F)ccc(F)c1C(=O)NC1CC1CNC(=O)CC1CCC2(CCC2)O1 34224,C1(C(=O)NCC2N(C(C(CC(C)C)O)=O)CCCC2)CCc2n[nH]cc2C1C 34225,c1(CN2CC(C)CC(NC(CC=CCC)=O)C2)coc2ccccc12 34226,C(=O)(C(F)(CNC(c1ccc[n+]([O-])c1)=O)C(C)C)NCc1nc(C)sc1C 34227,N1(C(c2c(C)con2)=O)CC(NC(c2cccc3cnsc23)=O)C2(CCC2)C1 34228,C(C(CC(C)C)C(=O)Nc1cnc(C)c(C#N)c1)NC(C1(OC)CC1)=O 34229,N1(c2nc(Cl)nc(C)c2F)CCC2(CC1)OCCC2NC(=O)Cn1nnnc1C 34230,c1(CN2CC(OC)C(CNC(=O)CCOC(C)C)CC2)ccc2nc[nH]c2c1 34231,C1(CNC(c2scnc2Cl)=O)CCCC1NC(=O)C(Cc1ccccc1)C1CC1 34232,N1(C(CC2CC(=C)C2)=O)CCN2CCOCC2(CNC(=O)C(C)CCCOC)C1 34233,c1(CNC(CN(C)C(N)=O)=O)c[nH]nc1NCC1(C(=O)NCCO)CC1 34234,CC(C)CCC(F)C(=O)NC(C)(CNC(c1cccc2nccn12)=O)CO 34235,Cc1cc(C(N2CCCC(NC(C3(C)C=CCCC3)=O)C2)=O)ncc1Cl 34236,CC1OC(=O)NC1C(=O)NCC1(CNC(=O)CCC2CCCCC2)CC1 34237,c1(SC)cc(N(C2CCN(C(c3cnoc3)=O)C2)C)nc(SC)n1 34238,N1(C(c2csc(C)c2C)=O)CCC2CCN(C(c3cc4sc(Cl)cc4[nH]3)=O)CC12 34239,Cc1noc(C)c1C(C)C(=O)NCCC(C)NC(=O)C(C)C1CCCO1 34240,c1(NC(C2C(N(C(=O)C=CCN3CCCCC3)CCN)C2)=O)cnncc1Cl 34241,N1(C(C2N(C(C3C(C)CCCC3)=O)CCCC2(C)C)=O)CC23CCC2(COC3)C1 34242,c1(C(=O)NCCC(C)N(C(C(c2cncnc2)C)=O)C)cnc2cnn(C)c2c1 34243,CC(N=c1cc[nH]cc1S(=O)(=O)NCc1ccc2c(c1)CCCC2)c1cccs1 34244,Cc1ccc2c(c1)CC(C)N(C(=O)NC(C)CCC1CCCC1)C2 34245,C(=O)(CC(C)C1CC1)NC1(CNC(COCC(C)C)=O)CC1 34246,C1(CC(N2CCC(c3nccc(O)n3)CC2)=O)CCC2(CC1)CC2 34247,N1(C(Cc2c(C)noc2)=O)CCC2C1CCCN2C(C1CCCCO1)=O 34248,C(CC(O)C(=O)NC1(c2ccccc2)CN(C(c2cc(C)on2)=O)C1)OC 34249,c1(C(C(=O)NCCC(=O)OCC)N(c2ccccc2)C)nc(Cl)sc1Cl 34250,C=CC(CC)C(=O)NCC1(C(=O)NCC2CC2Cl)CCC1 34251,C(CC(C(=O)NC(CCO)c1ccco1)NC(C1CN(C(C)=O)C1)=O)SC 34252,S(=O)(=O)(c1ccc2c(c1)CCN2CC)N1C(C(=O)OC(C(CCCC)O)=O)CCC1 34253,c1(C(N(S(C)(=O)=O)C)=O)cccc(-c2cncc(Nc3ncccc3Br)c2)c1 34254,c1(C(=O)NCC2N(C(C=NOC)=O)CCC2)cccc(C#N)c1 34255,N1(C(C(C)O)=O)CCC(C2CC(NC(=O)CCc3ccn(C)n3)C2)CC1 34256,C1(CNC(C2CC(C#C)(O)C2)=O)CC(C(=O)N2CCCN(C(N)=O)CC2)=NO1 34257,N1(C(c2c(C)nc(C)o2)=O)CC2CCN(C(=O)CC3CCCNC3=O)CC12 34258,c1(C(=O)NCCN(C(c2c(C)ccc(C)c2)=O)C)nc2ccccc2cc1C1CC1 34259,C(=O)(C(C)(C)S(C)(=O)=O)N1CC(CNC(c2c(OC(C)C)cccc2)=O)C1 34260,C(=O)(C1=CCCC1P(C)(C)=O)N(C1CCN(C(c2cncc(NC)n2)=O)CC1)C 34261,C1(NC(C2(CC)CCOC2)=O)CCCCCC1NC(=O)C(F)(F)c1csc(C)c1 34262,Cc1ccccc1C1(C(=O)NCC(C)CNC(C2(C)CSC2)=O)CC1 34263,N1(C(COCCCC#C)=O)CCC(F)(F)C(CNC(c2sccc2COC)=O)C1 34264,C(N=c1cc2n([nH]1)CCCC2)(c1cccc(OC)c1)c1nnnn1CC(F)F 34265,C(=O)(C(C#N)C(C)C)N1CCCC(NC(Cc2c(C)cnn2C)=O)C1 34266,C1(C(C)C)CN(C(C2(C(F)F)CCCC2)=O)CCN1C(c1csc(C2CC2)n1)=O 34267,c1(C(N(CC(CC)NC(C(CC=C)NC(C)=O)=O)CC)=O)cc(F)ccc1C 34268,N1(C(CCN(CCC)C)=O)CC=C(C(C)(C)C(=O)NC2CC(C3CC3)C2)C1 34269,C=CCC(CNC(=O)C(C)SC)NCC(=O)NC(=O)CC1(N(CC)CC)CCC1 34270,C1(OC)(CNC(c2cnoc2C)=O)CCN(C(=O)C2=COCCC2)CC1 34271,N1(C(c2c(SCC)cncc2)=O)C2CCC1C(CNC(=O)Cn1ccnc1C)C2 34272,N1(C(CC2C=CC(NC(=O)CC3CCCOCC3)C2)=O)CCC12CCSCC2 34273,c1(CCSCC(=O)NC(=O)Cc2ccccc2)ccccc1-c1nn[nH]n1 34274,C1(CNC(C=CC2N(C)CCC2)=O)CN(C)CCN1Cc1ccccc1 34275,C=CC1CN(C(=O)COCC(F)F)CC1NC(=O)CCc1ncc(F)cn1 34276,c1(C(=O)NCC2CCN(C(c3n(C)ccc3)=O)C2)n[nH]c2ccc([N+](=O)[O-])cc12 34277,N1(C(c2cn(CCNC(C3C(C)CC3)=O)nc2)=O)CC2(C)CC1CCO2 34278,N1(C(C2N(Cc3ccc(OC)c(I)c3)CC(OC)C2)=O)CCC2(CC1)CN(C)C2 34279,NS(=O)(=O)c1ccc(C(N2CC(NC(=O)CCN3C(=O)CCC3=O)C(O)C2)=O)o1 34280,C1(NC(CC2CC(OCC)C2)=O)CC2(CC2)CN1C(=O)CNC(=O)CCC(C)C 34281,Cc1nscc1C(=O)NC(C)(CNC(=O)CCC1CCC(C)O1)C1CC1 34282,C1(C(=O)NCCC(C)N(C)C(c2cn(C)nn2)=O)CCC(C)(C)C1 34283,C1(NC(Cn2nc(C)n(C)c2=O)=O)CC12CCN(C(C1OCCC1(C)C)=O)CC2 34284,N1(C(c2cc(C)oc2C(F)(F)F)=O)CCN(C(c2cnc(O)o2)=O)CC(C)(F)C1 34285,Cc1cc(NC(=O)NC2(c3ccccc3)CCOC2)cnc1C 34286,CCC(C(=O)NCC1(C)CCCN1C(=O)C1=NOC(C(C)(C)C)C1)C(C)C 34287,c1(CCC(=O)NC(C2CCN(C(c3c(C)nn(C)c3)=O)C2)C)c(Cl)cccc1Cl 34288,CCCN=C(NCc1ccc(NC)c(Cl)c1)NCC1CCN1C(=O)OC(C)(C)C 34289,C1(C(=O)NCC2C3CN(C(=O)CSc4ccccc4)CC23)C2CCC3C(C2)CC13 34290,C1(NC(C(n2c(C)ncc2)C)=O)CN(C(=O)Cc2cnsc2)CC12CCC2 34291,C(=O)(C1=C(C)OCCS1(=O)=O)NC1CN(C(C(CC)CC(F)F)=O)CC1C 34292,c1(C(=O)NC2CC3(C2)CC3NC(c2ncccc2F)=O)cc(F)c2cn[nH]c2c1 34293,C1(CC)CCC(C(N2CCCC(CNC(c3nnn(C(C)(C)C)n3)=O)C2)=O)CC1 34294,C1(NC(c2c(C(C)C)scn2)=O)CN(C(c2c[nH]ccc2=O)=O)CC2(CCC2)C1 34295,C(C(C)C(=O)NC(C(=O)NCCCC1CCOC1)C1CCCC1)OC 34296,C1(NC(COC(CC)CC)=O)CC12CCN(C(C1CCCC(=O)C1)=O)CC2 34297,Cc1cc(Br)ccc1CC(=O)NC1CCC1NC(C1CCCCN1C)=O 34298,c1(-c2cn(CCC3(C(=O)OC)CCOCC3)nn2)ncc(Br)cc1C(=O)O 34299,C1(C(=O)NCCCCC2CN(C(c3c(C)cc(C)[nH]3)=O)C2)CC12CCCOC2 34300,c1(OC)cc(C(=O)NC2CCN(C(c3cc(C)c(C)[nH]3)=O)C2)c(N)c(Br)c1 34301,C=CCC(C(=O)N1CC(C(=O)N(CCCN(C)C)CC)CC(C)C1)C(C)C 34302,C1(C(CC)=O)CCCC1OC(=O)CC 34303,Cc1nc2ccnn2c(C)c1C(=O)NC1CC(C)(NC(=O)CCn2cncn2)C1 34304,C1(C(N(CC(=O)NCC)C)=O)CCCN(C(=O)COC2CC2)CC1 34305,N1(C(CCC(=O)OCC)=O)CCC2(CCCN2C(=O)Cn2cc(C)cn2)C1 34306,CCCC(C(=O)NCCCOCCNC(C1CCc2nncn2C1)=O)S(N)(=O)=O 34307,N1(C(C(F)=CCC)=O)CCCC(NC(=O)COCC2CCCO2)C1C 34308,N1(C(c2nc(F)ccc2Cl)=O)CC(C2(N=c3[nH]nc(C4CC4)o3)CC2)C1 34309,C1(C(=O)NC2C(NC(c3ncsc3Cc3ccccc3)=O)C2)COC2(CCC2)C1 34310,C(=O)(C(CNC(=O)Cn1cccc1)CC(C)C)NC1CC(OC)C1(C)C 34311,N1(C(c2c(C)noc2C)=O)CCCC(F)(C(=O)NCc2cncnc2)C1 34312,N1(C(C(C(C)(C)O)F)=O)CC2OCCN(C(c3c[nH]c4nccc-4c3)=O)C2C1 34313,C1(C(F)(F)F)(C(=O)NC(CCNC(Cc2c(C)scc2)=O)C)CC2CCC1C2 34314,CC(C1OCCc2sccc21)NCC(=O)NCC1CCC1 34315,N1(C(CC2(C)N(C(c3cnc(CC)o3)=O)CC2)=O)CC(=O)NC(C)C1 34316,c1(C(N(C2CCN(Cc3cc(F)cc(F)c3F)C2)C)=O)ccncc1[N+](=O)[O-] 34317,N1(C(C(C(C)(C)C)SC)=O)CCCC(C2CN(C(=O)CN3CCOCC3)C2)C1 34318,N1(C(c2c(CC)nn(C)c2)=O)CC2CC1CN(C(c1nocc1Cl)=O)C2 34319,Nc1cc(Cl)nc(Cl)c1C(N1CC2CC2(NC(=O)CC(F)(F)F)C1)=O 34320,C(CC(C)C(=O)NC(C)CC1CN(C(=O)CCc2conc2C)C1)=CC 34321,CC1CN(C(C2CCCN2C=O)=O)CC1NC(C1(N(C)C)CCC1)=O 34322,CC1OCCC1(C)C(N1CCC(C(=O)NCC(C2CC(C)(C)C2)O)CC1)=O 34323,C1(CSc2nnc(-c3sccc3)o2)CCN(C2CCCCC2)C1=O 34324,C1(OC)CCCN(C(C2CCOCC2)C(=O)Nc2nnn(C)n2)CC1 34325,c1(CSCC)ccccc1C(=O)NC(CN(C)C(C1(C)CC=CC1)=O)CC 34326,c1(C(N(CC(C)NC(C(CNC(C)=O)(C)C)=O)C)=O)cc2sccc2cn1 34327,c1(NCCCCN(C)C2CC2)[nH]c(=NCC2(C3CC3)CCCO2)nc2sccc12 34328,c1(C(N(C(c2ccccc2)CNC(c2onc(C)n2)=O)C)=O)ccc(O)nn1 34329,c1(C(=O)NC2C(CNC(C(CC)CC3CCCC3)=O)C2)ncc2ccccn12 34330,C1N=C2C=CN=C(N2)Nc2cnccc21.N1(C(C)C)CCN(CCO)CC1 34331,c1(CN(C(C2CCCN(C(c3coc(C)n3)=O)C2)=O)CC)ccc(O)cc1 34332,N1(CCSc2ccc(C(C)C)cc2)CCCN(C(=O)C(C)C#N)CC1 34333,c1(OC)cc(C(=O)NCC(Cl)=CCl)sc1Br 34334,N1(C(CC(C)(C)O)=O)CC2(CC(C(=O)Nc3ccc(F)c(F)c3)CO2)C1 34335,c1(CC(=O)NCCCCC(C)NC(c2cc(C(N)=O)[nH]n2)=O)cccc(F)c1O 34336,C(=O)(CC(C)CC(F)(F)F)N1CC(C)C(NC(c2cc3cc(Cl)ccn3n2)=O)C1 34337,C1(CCC(=O)N(C2CCOC2)C)CCCN(C(c2cccc(F)c2)=O)C1 34338,N1(C(c2c(C)cccn2)=O)CC(C)CN(C(c2ccc(F)c(N)c2F)=O)C(C)C1 34339,N1(C(c2ccccc2)C)CCCC(C)(C(=O)N(CC2(C(F)(F)F)CC=CC2)CC)C1 34340,c1(C(N(C2CCC(NC(c3ccncn3)=O)CC2)C)=O)ccc(S(N)(=O)=O)cc1 34341,c1(NC(C(=O)NCC)=O)ccc2c(c1)CN(C(=O)CCc1ccc(C)cc1)CC2 34342,C1(NC(COCCC)=O)CN(C(=O)CCc2scnc2C)CCC1F 34343,C1(NC(CCC=C)=O)CN(C(=O)COc2ccon2)CCC1C 34344,C(C(CO)(CO)NC(c1cccnc1)=O)N(C)C(C1CNC(=O)N1C)=O 34345,C(=O)(CCCCc1ccccc1OC)NC(CC)(C)C#N 34346,N1(C(CN(C)C2CC2)=O)CCCC(C)(C(=O)NC(C)(C)C(O)CO)C1 34347,c1(CC(=O)N(C2CCCN(C(c3cccnc3)=O)CC2)CC)c(F)cncc1Cl 34348,C1(C(=O)NCCCCNC(CN(CC(=O)NC(C)C)C)=O)CCc2nc(C)cn2C1 34349,C(=O)(C(C(CC)CC)OC)N1CC(N(C(=O)C(c2cnn(CC)c2C)=O)CC)C1 34350,c1(C(=O)NC2C(NC(C=CCOC)=O)C2)cccc2oc(C)cc12 34351,c1(C(N(C2CCC(NC(c3c(C)ocn3)=O)C2)C)=O)cnc2c(cnn2C)c1 34352,C1(NC(CC(C(C)C)NC(c2c(C)ccnc2C)=O)=O)CC(C2CCCC2)C1 34353,C1(C(=O)NCC#CCNC(C(CC)C2CCOCC2)=O)(OC)CCC(C)(C)C1 34354,C1(COC)(NC(=O)CCC=C(C)C)CCN(C(=O)C(c2ccccc2)SC)C1 34355,c1(C(=O)NC(C(C)(C)OC)C)ccc(CNC(=O)Cn2cc(C#N)cn2)nc1 34356,c1(C(N(CC(=O)OC)CC)=O)cnc(CNC(c2ccnn2CC)=O)nc1 34357,N1(C(C(C2SC(=N)NC2=O)C)=O)CC2OCCN(C(C3CN(C)CCO3)=O)C2C1 34358,C(c1cccc(C)c1)=CC(N1CC(C(C(=O)N(C2(CC)CC2)C)O)C1)=O 34359,N1(C(c2cc(C(C)C)no2)=O)CCN(C(=O)CCCNS(C)(=O)=O)CC2(CC2)C1 34360,C1(NC(c2cc(CC)ncc2)=O)CCN(C(=O)Cc2cncnc2)CC(C)(C)C1 34361,N1(C(C(C)=CC)=O)CC(CNC(C2CNC(=O)C2)=O)C(F)(F)C1 34362,c1(COC)nn(C)cc1C(=O)Nc1cccc(-c2nc(C)co2)c1 34363,N1(C(c2nc(CCC)oc2)=O)CCC(CC)C1CNC(C1CC(F)C1)=O 34364,N1(C(C2CCOC2)=O)CCCOC(CC(N2CC(NC(=O)NC)C2)=O)C1.CCS 34365,N1(C(C(C=C)c2ccccc2)=O)CCN(C(c2cnn(C3CC3)c2)=O)CC1CO 34366,n1(CC)nc2c(c1C(=O)NC(C)CCN(C)C(C1CC1C(F)F)=O)CCCC2 34367,c1(OC(C)C(=O)NC(C)(C)CO)cccc(C(F)(F)F)c1 34368,CCCCC(C)(F)C(=O)NCC(C)N(C(=O)CN1CCOCC1)C 34369,N1(C(CCN(C)CC)=O)CCC2C(NC(c3nn(CC)cc3Cl)=O)C2CC1 34370,N1(C(=O)COC2CCCC2)CC2CCC(NC(=O)COCCCF)(C2)C1 34371,C1(NC(c2ccc(SC(C)C)cc2)=O)CC2CC1CN2C(=O)CN(C)CCO 34372,c1(C(=O)NCC(CN(C(CN(CC)CC)=O)C)O)ccc(-n2cncn2)c(F)c1 34373,N1(C(c2ccn(C)n2)=O)CC2(CCCC2NC(C2C(C)(C)OC2(C)C)=O)C1 34374,c1(C(N(CC(CC)NC(=O)CCNS(C)(=O)=O)CC)=O)cc(CC)cc(F)c1 34375,C(=O)(C1CCCc2n[nH]cc21)NC(Cc1cccc(OC)c1)(C)C 34376,c1(CC(=O)NCC(CC)NC(=O)COc2cn[nH]c2)csc(C(C)(C)C)n1 34377,CCCCC(CC)(c1nnnn1CCCSC)NCC1CCCC(CO)C1 34378,c1(N2CCC(C)(NC(c3cc(SC)oc3)=O)CC2)ccn2ccnc2n1 34379,c1(C(=O)NC2(CCOC)CCN(C(c3cnn(C)c3)=O)C2)cc(C)cnc1C 34380,c1(C(N2C(CC)C(NC(c3cnn(CC)c3C)=O)CC2)=O)ccc(=N)[nH]c1Cl 34381,N1(C(c2ccccc2)=O)CCN(C(c2cnc(-c3ccccn3)nc2)=O)C2CC12 34382,C1(CNC(CC2CC(SC)C2)=O)CCCCC1NC(c1nnccc1C)=O 34383,N1(C(C2(CC=C)CCCCC2)=O)CC2CC(CNC(C3C=CCCC3)=O)C2C1 34384,c1(C(=O)NCCC(=C)CNC(c2ncccc2C)=O)nn(C)nc1Br 34385,C1(CNC(c2n(CC)nc(C)c2)=O)CCCCN(C(C23CC(O)C2C3)=O)C1 34386,c1(CC(=O)NCC2C(NC(C(c3ccccc3)OC)=O)COC2)ccncc1C 34387,C1(C(=O)NCC23OCC(NC(c4c(C#C)c[nH]n4)=O)(C2)C3)CCCCN1N=O 34388,CC(C)CCCCCCC(=O)N1CCC2C(NC(=O)C(O)CN(C)C)C2C1 34389,c1(N2CC(C(=O)NC)OCC2)ccc(S(=O)(=O)NCc2csc(Br)n2)c(Cl)c1 34390,C=CC(F)(F)C(=O)NCC1CCN(C(=O)CC2(O)CCC2)CC1 34391,Cc1cc(Cl)cc(C)c1OCC(=O)NC(C)CCCNC(=O)C(C)(C)F 34392,CCC(C)CCC(=O)NCC(C)(CO)NC(C12CC(C)(CCO1)C2)=O 34393,C(=O)(NNC(=O)C(O)c1ccccc1OC(F)(F)F)c1c(C)cccc1Cl 34394,C(=O)(C(CCNC(=O)CN1CCCC1)OCC)N1CC(=CCC)C1 34395,C(=O)(CCCCC(=O)NCC1(C)CCN(C(c2cnccn2)=O)C1)OC 34396,c1(C(N(C2CCCC2)CCNC(CC#N)=O)=O)ccncc1C(F)F 34397,N1(C(CSC)=O)CCN(CC2CCCN(C(=O)C(C)CF)C2)CC1 34398,CCC(CNC(=O)C(=O)Nc1cc(Cl)ccc1C(F)(F)F)CC(F)F 34399,C1(C(=O)NCC(C=C)(C)C)CN(C(=O)CCc2ccnn2C)CC1F 34400,N1(C(CC=C)=O)CC(C)(C)CCC1CNC(c1cccc(OCCOC)c1)=O 34401,c1(CN(C)C(=O)NCc2cc(-c3ccccc3)[nH]n2)noc(C2CCC2)n1 34402,CN1CCOCC(NC(C2CCCN(C(=O)COC3CCCOC3)C2)=O)C1 34403,c1(C(=O)NCC2(CNC(C3C(C)N(C)CC3)=O)CC2(F)F)cncc2n[nH]cc12 34404,C1(C(=O)NCC2N(C)CCN(C(C(C)S(N)(=O)=O)=O)C2)CCc2nncn2C1 34405,C1(C)(NC(C=CCOCCOC)=O)CCN(C(=O)CCc2cc(Cl)no2)C1 34406,C1(OC)C2CCN(C(c3cc(C(F)F)cc(C)c3)C(=O)NC3CC3)C2C1(C)C 34407,C1(OC(C)=O)CCN(C(C2CC(NC(c3ccns3)=O)C2)=O)C1 34408,C1(NC(c2cc(C)c(Br)o2)=O)(CO)CCCN(C(c2nocc2C2CC2)=O)C1 34409,c1(CNC(C(n2cc(CCOC)nn2)C)=O)cccc(C#N)c1 34410,C12(C(=O)NC(C)CN=[N+]=[N-])CCN(C1)S(=O)(=O)C2 34411,c1(OC)cc(C)c(C(N2CCC(C)(CCNC(C3CCC(=O)N3)=O)C2)=O)c(C)c1 34412,C1(F)(C(N(CCNC(C2(N(C)C)CCCOC2)=O)C2CC2)=O)CC2(CCC2)C1 34413,Cc1ccc(-c2ccccc2)c(NC(c2cc(C(=O)O)c(C)[nH]2)=O)c1 34414,N1(C(C2C(CCOC)C2)=O)CCC(C)(C)C1CC(N1CC(S(C)=O)C1)=O 34415,c1(C(N(CCCNC(=O)C=C(C)C)CC)=O)cc(F)c(F)c(O)c1F 34416,c1(C(=O)NC(C(=O)N(CC#C)CC)C2CCCO2)c[nH]c(=NC)s1 34417,c1(C(=O)NC2CC(C(C(=O)NCC(CCC)O)F)C2)c(C)n[nH]c1C 34418,Cc1c(Cl)cnn1CC(=O)NCC1CCCN1C(c1n[nH]c(C2CC2)n1)=O 34419,S(=O)(=O)(CC(=O)N1CC(N(C(=O)C(C)OCC2CCCO2)C)C1)NCC 34420,N1(C(C(C(C)C)C)=O)CCC(CNC(c2ccccc2-n2ccnn2)=O)C(C)C1 34421,c1(CCC)c(C(=O)N(CCCOCCNC(=O)C=C2CCC2)C)cnn1C 34422,C(=O)(C(C)(CC)OC)NC1C(C(N(CCC)CCN(C)C)=O)C1(C)C 34423,C(=O)(C1Cc2ccccc21)N1CC(CC)(NC(c2cnn(C)n2)=O)C1 34424,c1(CCC)cc(C(=O)NC(C)CC(C)NC(c2cccnc2F)=O)nn1C 34425,N1(C(c2scc(C(C)=O)c2)=O)CCC(C2CN(C(=O)CC3CCCCO3)C2)C1 34426,c1(C(=O)NCC(CN(C(CNS(NC)(=O)=O)=O)C)O)cnc(O)c(C)c1 34427,N12CCCN(CC1)C1CCN(C1)C(=O)C2.Cc1ccccc1NC(=O)C(C)(C)Br 34428,N1(C(c2cc(OC)n(C)n2)=O)CCN(C(C2CCNC2=O)=O)C(C2CCCC2)C1 34429,Cc1ccc(N2CCCC3(NC(C4CCCC(F)(F)C4)=O)CC3C2)c([N+](=O)[O-])c1 34430,c1(C(=O)NCC(CO)NC(c2n(CC)ncc2)=O)c(F)cc(C)cc1F 34431,CC(C)CC(F)(F)C(=O)N1CCC1C1CCN(C(c2c[nH]nc2[N+](=O)[O-])=O)CC1 34432,Cc1cnn(C)c1C(=O)N(C)CC1(CNC(C2COCC(C)O2)=O)CC1 34433,c1(C(N(C2CCN(C(c3cc(C)ns3)=O)C2)CCO)=O)nc(=O)n(C)[nH]1 34434,N1(CC(COCC(C)C)O)CCC(CNC(=O)C(F)Cc2ccccc2)C1(C)C 34435,c1(C(N(CC(=O)NC(C)C(O)C(C)C)CC)=O)ncnc(O)c1F 34436,Cc1ccc(O)c(C(=O)NC(C)(C)CN(C)C(C2CC2(C)C(C)C)=O)n1 34437,C1(NC(c2cc(C(C)=O)[nH]n2)=O)CN(C(c2ccnc(Cl)c2O)=O)CCC1C 34438,C1(CNC(=O)COC2CC2)CCC(CNC(c2csc(C(F)(F)F)c2)=O)CC1 34439,CC(C)CCCCCC(=O)NCC1(C(C)(C)O)CN(C(C2CC(C)N(C)C2)=O)C1 34440,c1(C(=O)NCCC(C)N(C(CC2(CC)CCOCC2)=O)C)ccc2cnoc2c1 34441,CC(CN(C)C)CCC(=O)N1CCCC(C(=O)NCC2CC3OC2C2CC32)CC1 34442,C(N=c1nc(C2CCOCC2)[nH]s1)C1CN(C(C(C(C)C)OC)=O)C1 34443,c1(C(N(CCNC(C(c2cn(C)nc2)O)=O)C2CC2)=O)c(Cl)ccc2c1OCO2 34444,c1(CC)cc(C(=O)N(CC(O)CN(C(=O)C=CC2CC2)C)C)ccc1Br 34445,C1(CC(=O)NCC2COC(=O)C2)COCCN1C(c1ccc(CO)s1)=O 34446,c1(C(=O)NC(C2CN(C(c3ccc(C)n3C)=O)C2)C)n[nH]c2ccc(Br)cc12 34447,c1(C(C)NC(=O)NCC(c2ccc(C)cc2)(C)CO)cc(C)cnc1F 34448,C12(C(=O)NCCNC(CC(CC)(C)C)=O)CCC(C)(C(=O)O1)C2(C)C 34449,C12(CNC(c3cc(OC(CC)C)ncc3)=O)CCC1CN(C(=O)C=CSC)C2 34450,c1(C(=O)NC(C2(O)CN(C(=O)Cc3cncs3)C2)C)cc([N+](=O)[O-])n(C)n1 34451,CC1(C)CC(C(=O)NC2CCCC(O)C2O)CCN1C(=O)C1=CCSC1 34452,N1(C(C(CC=C)NC(N)=O)=O)CC2CC(C(=O)NCCOC3CCCC3)(C2)C1 34453,CCC(CC(=O)NC12CC1CN(C(c1cocc1C)=O)C2)c1ccccc1 34454,c1(NC(C)CCNC(C2CCOC3(CCC3)C2)=O)cc(=O)n2ccccc2n1 34455,N1(C(c2c(OCCOC)nccc2)=O)CC(CNC(=O)C(C)COC)C2(CC2)C1 34456,Cc1cccc2nc(C(=O)NC(C)CNC(=O)C=Cc3nccs3)cn12 34457,N1(C(c2cnc(COC)s2)=O)CCCC(CNC(=O)COCCCF)CC1 34458,C1(C2=CCCCCC2)(C(=O)NCC(CNC(C=Cc2cccc(C)c2)=O)C)CC1 34459,C#CCCCCC(c1nnnn1CCCC=C)NCCc1ccc(Br)c(C)c1 34460,Cc1cc(CNC(C(N2CC(C(F)(F)F)C(C)C2)=O)=O)ccc1F 34461,c12cc(C)ccc1CO2.Cc1cccc(C(CO)NC(=O)C(=O)NC2CC2)c1 34462,Cc1oc(CNC(c2ccn(C(C)C)n2)=O)nc1C(=O)NCC(O)CF 34463,C1(C(=O)NCC2(NC(COCc3ncc(C)o3)=O)CCC2)CCC2(CC2)C1 34464,N1(C(CCC#C)=O)CC(C(=O)NC(CO)C2(O)CC2)CCC1C 34465,C(=O)(CS(=O)(=O)CCO)NC1C2CCN(C(CC3CCC(C)(C)CO3)=O)CC21 34466,c1(C(=O)Nc2nnc(NS(C)(=O)=O)s2)c(Br)ccc(Br)c1N 34467,C(C(C)(C(C)C)NC(=O)C(N)=O)NC(C(c1cccnc1)OC)=O 34468,CC1CC(C)(C)CCC1NCCC(C)(c1nnnn1C1CCC(F)(F)CC1)SC 34469,O=CN1CCOCC1C(=O)NC1CN(C(=O)Cn2nc(O)ccc2=O)CC1F 34470,c1(OC)cc([N+](=O)[O-])ccc1CCN=C(NCC(O)COC)NCCSC 34471,c1(C(N(CC(CNC(COC)=O)O)C)=O)ccc(Oc2ccc(SC)cc2)cc1 34472,C12(C(=O)NCc3cn(C4CN(C(CSCC=C)=O)C4)nn3)CCCCC1C2 34473,c1(C(N2CC(C)C(NC(=O)CCC3CC3(Cl)Cl)C2)=O)csc2c(O)ccnc12 34474,N1(C(C(CC)(F)F)=O)CC2CC(O)C1C2NC(c1cc(C(F)F)ncn1)=O 34475,c1(CNC(C(C2CC(CC)C2)N(C2CC(C)(C)C2OC)C)=O)ccc(F)cc1F 34476,N1(C(C2(CC#C)CCC2)=O)CCC(C#C)(C(=O)NC2CC2C2CCCCC2)CC1 34477,C1(NC(Cc2cc(C)on2)=O)COCCN(C(=O)C(C2CC(F)(F)C2)O)C1 34478,N1(C(c2cn(CC)nc2C)=O)CCC(F)(CNC(=O)Cc2nnc(O)s2)CC1 34479,N1(C(C2(C)N(C(CN(C(=O)OC)C)=O)CC=C2)=O)CCC2(CC1)CC2 34480,C1(F)(CNC(c2cnc(C3CCOC3)s2)=O)CC(CNC(C2CCCCO2)=O)C1 34481,Cn1nc(C(F)F)c(CN2CCC(O)CC2C(=O)Nc2cncc(F)c2)c1Cl 34482,CC(CNc1ccccc1)C(=O)NC1COCC1NC(C1(N(C)C)CC1)=O 34483,C#Cc1cn(C)nc1C(N1CCCC(CNC(=O)COC(C)CC)CC1)=O 34484,c1(OCC(=O)N(CC(C)O)CCNC(C2CCC(=O)O2)=O)ccc(Br)cn1 34485,c1(N2CCCC(C(C)NC(=O)C=CBr)C2)cc(Cl)nc(-c2ccccn2)n1 34486,N1(C(CC(CC)(C)C)=O)CCCN(C(c2cnccn2)=O)CC1C(C)C 34487,c1(C(=O)NC(C2CN(C(=O)C3=COCC3)CCO2)C)cc(Cl)cc(Br)c1 34488,c1(N(c2ncnc(COC)c2F)C2CNCC2C#N)ncnc2c(C)csc12 34489,Cn1cc(C(=O)NCC(C)(C)CC2CN(C(=O)C3CC3)C2)nn1 34490,c1(CC)ccc(F)cc1C(N1CCN(C(=O)Cc2ccc3c(c2)CC3)C2CC12)=O 34491,C1(CC(=O)NC2CN(C(c3c(C)cc[nH]3)=O)C(C)C2)CC2(CCCC2)CO1 34492,C1(F)(CNC(c2ccn(C3CCCCC3)n2)=O)CN(C(C2CC2(F)Cl)=O)C1 34493,N1(C(CN(C(C(C)C2(O)CCC2)=O)C)=O)CCN(C(C2COCC2(C)C)=O)CC1 34494,c1(CNC(C2(OC)CNC2)C)ncc(C(C)(C)C)[nH]1 34495,c1(C(C)NC(=O)C(=O)NC(CNC(=O)OC(C)(C)C)C(C)C)ncccc1C 34496,c1(C(=O)NC(CNC(CC(CC)SC)=O)C)ccc2c(c1)CCN2C(C)=O 34497,N1(C(CCOCC#C)=O)CCC(C(=O)NCC(O)COCC)C12CC2 34498,C1(N(c2ccc(C(N)=O)cc2)C)CC2CC1CN2S(=O)(=O)C1CC1 34499,CCCC(C(=O)N1CCC(NC(=O)CNC(=O)C(C)(C)C)C12CCC2)C(C)C 34500,C1(CNC(C=CCCC=C(C)C)=O)CC(F)(F)CN1C(=O)C(c1ccc(Cl)s1)=O 34501,C(=O)(C1=CCN(C(=O)Cn2ncnn2)C1)NCC(COC)(O)CO 34502,CC1CN(C(=O)CCNC(N)=O)CC1NC(c1nc(Cl)cs1)=O 34503,N1(C(CC(C)(F)F)=O)CCC2(CCC(CNC(=O)C=Cc3cscn3)O2)CC1 34504,C1(NC(c2cc(C)c(F)nc2)=O)CCC(F)(F)C(C)(C)C1 34505,CC1C(NC(=O)CC2CCC=CCC2)CCCN1c1ccnc(C2CC2)n1 34506,C(=O)(C(C(C)(C)C)OCC(=O)NCC)C1C(C(=O)OCC)CCCC1.C(C(=O)N)N 34507,C(=O)(CCCCC(C)C)N1CC2C(S)C2C1.Cc1ccc(C2CNCCO2)cn1 34508,c1(C(N2CC3C(NC(=O)CC(C4CC4)C4CC4)(CC3)C2)=O)cn2c(n1)CCCC2 34509,C1(NC(CCC=C=C)=O)CCC2CCN(C(c3ccc(F)c(C)c3Cl)=O)C1C2 34510,c1(CC(=O)NCC2N(C(C=CC3(C)COC3)=O)CC(O)C2)cc(F)ccc1F 34511,c1(OC)ccc(Cl)c(C(=O)NCCC2(O)CN(c3nccc(C#N)n3)C2)n1 34512,C(CNC(=O)CC1CCCC1C)(CCNC(C1(CC(C)C)CCC1)=O)OC 34513,CC(O)C(F)(F)C(=O)NC1COCC1NC(c1cc([N+](=O)[O-])n[nH]1)=O 34514,N(C(=NCC1=CCCCC1)NCC1(C#N)CCC1)CC1N(CC)CCC1 34515,C(=O)(C(C)(C)C(C)O)NCCCNC(COCc1c(C)ncs1)=O 34516,N1(C(C(C)OCCC=C)=O)CC(NC(c2nocc2C(C)(C)C)=O)CC1(C)C 34517,N1(C(C(C)C2CC2)=O)CCN(C(=O)CN(C(c2ccco2)=O)C2CC2)CC1 34518,N1(C(CN(C(c2c(CCC)n[nH]c2)=O)C)=O)CC(N(C)C)C(C)C1 34519,Cc1ncc(C(=O)NC(C)(C)C(=O)NCCC2CCCCO2)cc1C#N 34520,N1(C(c2cc(C)c(F)cn2)=O)CCC2OCCN(C(=O)CC3CCCOC3)C2C1 34521,c1(C(=O)NCC2(CNC(c3ccc(NC)c(F)c3)=O)CC2)nn(C)cc1[N+](=O)[O-] 34522,C1(CN(C)C(C2CC(C#N)C2)=O)CCCN(C(=O)C(O)CF)C1 34523,N1(C(C2CC(C)(C)N2)=O)CCC(S(=O)(=O)C(F)F)C1 34524,C(=O)(CCC(C(=O)NCCCN(C)C(C1CC(C)(C)CO1)=O)N(C)C)OC 34525,c1(NC(C2C(O)CCN(CC#CC)C2)=O)ccc(N=Nc2ccccc2)cc1 34526,C1(C(=O)Nc2cccnc2C(F)(F)F)CN2CC3CC2(CO1)C3 34527,n1(C(C)C)cncc1C(=O)N(CCCNC(=O)CC1CCCO1)C 34528,N1(C(c2cc(OC)cc(C)c2)C(=O)NC(CC)C)CC(C)c2ccccc21 34529,C1(O)(CC(N2CC(CNC(C3(C(=O)OCC)CC34CC4)=O)C2)=O)CCCCC1 34530,c1(CNC2CC(OC)C(CN)C2)cnc2ncccn12 34531,N1(C(C2CCN(CC)CC2)=O)CCCC(CNC(c2cc(F)ccc2O)=O)C1C 34532,[N-]=[N+]=NC1CCC2(C(=O)NC(CNC(=O)Cn3nccn3)CO)CC12 34533,N1(C(C2ON=C(C)C2)=O)CCCC(C)(CNC(c2c(C)noc2C(F)(F)F)=O)C1 34534,C1(CNC(c2oc(CC)c(C)c2)=O)CN(C(=O)C(CC(C)C)N(C)C)CCCO1 34535,c1(C(=O)NCC2CC(OC)CN2C(c2csc(C(F)F)c2)=O)nnc(O)cc1O 34536,O=S(=O)(c1ccc(F)s1)Nc1ccc(OCC(F)F)nc1 34537,c1(OC2C(SC)C2)cccnc1.c1(COC(C2(CNC(C)(C)C)CC2)=O)cccs1 34538,C=CC(C)(CCOC)C(=O)NCCN(C(=O)C1=COCCO1)C 34539,c1(C(=O)NCCCC(C)NC(C2CC3CCC(C2)O3)=O)cccc2c1ncn2C 34540,C(C(O)CC(=O)NCC1CC12CC2)NC(=O)CCc1ncccn1 34541,C1(N(C(CC(C)CF)=O)C)CCC2(CC1)CCN(C(c1ccc(F)cc1O)=O)C2 34542,c12ccccc1CCC(=O)N2.Cc1nn[nH]c1COC(C1CC=CCC1)=O 34543,C1(NC(CC(c2ccc(C)cc2)C)=O)CCN(C(C2(C)CCC2)=O)C12CCCC2 34544,CC1(C)NC(=O)CC1C(N1CCC(C(=O)CNC2CCS(=O)CC2)CC1)=O 34545,CC(C)CC(CNC(=O)CCCC#N)C(=O)NCCCC1CC1C 34546,CC(C)CC(C)CC(C)C(=O)NC1(CN(C(=O)CCc2cncnc2)C)CC1 34547,C1(N(C(COCC=C)=O)C)CC2CCC(C1)N2C(C1(C(F)F)CCOCC1)=O 34548,C(=O)(CC(C)(C)C(F)(F)F)NCCOC1CN(C(C(CC)(O)c2ccccc2)=O)C1 34549,c1(CC)ccc(C(N2CCC(C)(CNC(=O)C(C)(C)CO)C2)=O)c(C)n1 34550,C1(CNC(C(CO)N(C)C)=O)CN(C(=O)CN2CCNC(=O)C2)CC(C)(C)O1 34551,c1(C(=O)NCC2C(C)CN(C(C3CCCCO3)=O)C2)cc(Br)c(F)cc1N 34552,CCCN=C(NCc1ccc(F)cc1Cl)NC1CN(C2CC2)CC1C 34553,C1(CCC#C)CCCN1C(=O)C(C1CCN(C(C2CC(=O)C2)=O)C1)C 34554,N1(C(c2cn(CC)nn2)=O)CCCCCC1CNC(=O)C(C)C(C)C 34555,c1(CN(C(C2CCC2NC(C2CCCSC2)=O)=O)CC)ccccn1 34556,CC1(CCO)CCN1C(=O)C(C1CCOC1)NC(C1CC(F)C1)=O 34557,Cn1ncc2ccc(CN3CCC(O)(C(=O)Nc4cc(C#N)ccc4Br)C3)cc12 34558,c1(C(N(CCNC(C2CCC(CC)C2)=O)C2CC2)=O)cc(N)cnc1C 34559,C1(NC(c2coc(C3CCC3)n2)=O)COC2(C1)CN(C(c1cc[nH]n1)=O)C2 34560,C1(NC(CC(COC)C)=O)CC1C1CCCN(C(c2cnn(C)c2Cl)=O)C1 34561,N1(C(c2cc(C)sc2)=O)CCCC(NC(c2n[nH]cc2Br)=O)C(F)C1 34562,C(=O)(C#CC1(C)COC1)NCC1CN(C(Cn2ccc(C)cc2=O)=O)CC1O 34563,N1(C(C2C(OCC)C2)=O)CCC(NC(=O)CCn2cccnc2=O)C(CO)CC1 34564,C1(NC(C2C(CNC(c3cccc(=O)o3)=O)C2)=O)C(O)C2CCOC12 34565,c1(OC)cc(OC)cc(CNC(C2CC3CCC2CC3)=O)c1 34566,C12(CNC(c3cc(CC)n(C)n3)=O)CC(CO1)N(C(=O)C(C)CO)C2 34567,C(=O)(CCCC(C)CC)NC1(C(N2CCCCC(CC)C2)=O)CCOCC1 34568,c1(C(N2CCC(C(N)=O)(C(=O)NCC3CC34CC4)C2)=O)n[nH]c2c1CCC2 34569,c1(C(N(C)CCN(C)C(C2CCCS(=O)(=O)C2)=O)=O)cncc2n[nH]cc12 34570,C=Cn1ncc(C(=O)NCc2ccc(C(=O)NCC3CCCCC3C)o2)c1N 34571,C1(C#CC(=O)N2CC(NC(C3(C(C)(C)C)CCCCC3)=O)CC2C)(CC)COC1 34572,C1(C2CC2)(NC(CCNC(c2nn(C)c(O)c2)=O)=O)CCOC1 34573,c1(OC)cc(NCC(C2CC2)N(C(=O)C(C)CC(F)(F)F)C)ccc1[N+](=O)[O-] 34574,CCC(CC)(CC)C(=O)NCC(CNC(c1cn(C)cn1)=O)C(F)(F)F 34575,N1(C(C(C)O)=O)CCC(n2cc(C(=O)N(CCC(F)(F)F)CC(=O)O)nn2)CC1 34576,C1(OCc2cn(CCCCC)nn2)CCCN(C(=O)CC2CCCC(O)C2)C1 34577,C=CC1CN(C(c2ncsc2C)=O)CC1NC(=O)C(C)(C)C1CC1 34578,C1(NC(c2c(C)ccn2C)=O)CC2(C1)CC(CNC(=O)CN1CCC(C)C1)C2 34579,CC1(C2CC2C(N2CCCC2C(C)(C)C(N2CC3CCC2CC3)=O)=O)COC1 34580,n1(CCNC(C(C2(O)CCC2)NC(C2COCCO2)=O)=O)cc(CO)nn1 34581,C(=O)(CC(CC)CCCC)NC(CC#C)CC(=O)NCC1(C)CC(C)=NO1 34582,CCC(CC(=O)NCC1(C(=O)NCc2ccco2)CCCO1)C1CC1 34583,Cc1nn2cc(C(N3CCC(N(C(=O)C(c4ccccc4F)C)C)C3)=O)nc2s1 34584,N1(CC(N2CCC(NC(=O)CC3CCSCC3)C2)=O)C(=O)CNC1=O 34585,N1(C(c2c(SC)nccn2)=O)CCC2(CCC(NC(=O)Cc3nccs3)CC2)C1 34586,CC1C(NC(=O)C(CCN(C)C)NC(=O)Cc2ncccc2F)CCCN1C 34587,n1(CCC)cc(CN2CCC(C(N3CCC3(C)C(=O)OC)=O)C2)cn1 34588,C1(CC)CCC(C(N2CCC2CC(=O)NCC(C)O)=O)CC1 34589,C(=O)(C1=Cc2ccccc2C1C)NC(C)CCCNC(=O)C1=C(Cl)CC1 34590,Cc1ccc(C(N2CC=CC(NC(=O)C(c3ccccc3)O)C2)=O)cc1F 34591,Cc1cc(C(N2CCOC(C(=O)NCCCCC3CCCC3)C2)=O)c(C)s1 34592,N1(C(c2cc(C)ncn2)=O)CCC(CO)C(NC(c2csc(C(F)(F)F)c2)=O)C1 34593,C(=O)(C1=CS(=O)(=O)CCC1)N1CCC(N(C(=O)C(C)CF)CC)CC1 34594,c1(C(C)=O)cc(Cl)c(NC(=O)COC(c2c(F)cc(F)cc2F)=O)c(Cl)c1 34595,c1(-c2cc(NC(N3CCCC(c4ncc(C)s4)C3)=O)no2)ccc(F)cc1F 34596,N1(C(C2CCCCC2)C(=O)NC(CC)(C)C)CCSC(C(C)C)C1.C1CN1 34597,C1(C(N(C(C)C(N2CCC2(C)CC)=O)CC)=O)CCC(F)C1 34598,N1(C(C)C(=O)N2CC(CCNC(=O)CCc3nncs3)C2)CCN(C)CC1 34599,c1(NC(N2CCC(C)(c3cn(CC4CC4)nn3)C2)=O)cnc2ccccc2c1 34600,C1(n2cc(C(=O)OCC)nn2)CCCN(N2CC(N3CC(C)(C)C3=O)C2)C1 34601,N1(C(=O)Cc2c(C)cnn2C)CCCC(C)C1CCNC(c1c(OC)scc1)=O 34602,c1(C(=O)NC2(CNC(=O)CCF)CCC2)cc(Cl)c2c(c1)OCCCO2 34603,N#Cc1ccnc(NCC(c2ccccc2F)NC(C2(C(F)(F)F)CC2)=O)n1 34604,c1(C(c2nnnn2C2CC2)NC2C(C=C)CCCC2)cccc2cnccc12 34605,C=CCC(CNC(C1C2CCCC12)=O)C(=O)N1C2CCC1CC2 34606,c1(C(N2CC(NC(C=CS(C)=O)=O)CC2(C)C)=O)ccc(Br)cc1C#N 34607,CCCCC(C(=O)N(C)CC1CCC(=O)N1)NC(c1n[nH]c(=N)[nH]1)=O 34608,NS(=O)(=O)CC(=O)N1CCCCC1c1n[nH]cc1C(=O)NCC1CCC(O)C1 34609,C12(CNC(C3C(CCC)C3)=O)CC1CN(C(=O)Cc1cncc(Br)c1)C2 34610,C(C)(CNC(c1cnc(C)s1)=O)(CO)NC(CSCCCC)=O 34611,Cc1cc2c(NC3CC3C(=O)Nc3cnc4[nH]ncc4c3)ncnc2[nH]1 34612,C1(NC(CCC=CC(C)C)=O)CCCN(C(=O)C=CC=Cc2ccccc2)C1C 34613,C1(NC(C2N(CC)CC2)=O)CCSC12CN(C(C1CCN(CC3CC3)CC1)=O)C2 34614,c1(SCC(N2CC(NC(c3ccnn(C)c3=O)=O)C(F)C2)=O)ccc([N+](=O)[O-])cc1 34615,N1(C(c2c(C)ccs2)=O)CCC2CN(C(C3COCCO3)=O)CCC12 34616,Cc1cc(NC(C2CN(C(=O)C(c3cncnc3)C)CC2(F)F)=O)c(C)cc1O 34617,C1(NC(C=CC(=O)OCCCC)=O)CC2(C1)CN(C(C1(C)CCC1)=O)C2 34618,N1(C(CC(C(C)C)C(C)C)=O)CCc2c(c(CNC(C3CC3F)=O)nn2C)C1 34619,c1(C(=O)NCCCC(C)NC(C2CN3CCC2CC3)=O)nn(C)c2c1CCCC2 34620,c1(C(N2C(C)CC(Nc3nccc(C(C)(C)C)n3)C2)=O)cn2ccccc2n1 34621,C(=O)(CC(F)(F)CC)NC(C(C)NC(C(CCC)NC(=O)OC(C)(C)C)=O)CO 34622,Cc1cnc(N)c(C(=O)NC2CC(CNC(c3cccc(Cl)c3F)=O)C2)c1 34623,Cc1nn2cc(C(=O)NCC(CC(C)C)NC(C3COC(=O)N3C)=O)nc2s1 34624,C#Cc1cccc(C(=O)N(C(C)CCNC(=O)COC2(C)CCCC2)C)c1Cl 34625,N1(C(C(CC)(C)C)=O)CC2CCCC(C1)N2C(=O)Cc1cccc2c1CCC2 34626,CC1CCN(C(c2cn3c(n2)CCC3)=O)CC1NC(=O)Cc1ccccc1Cl 34627,N1(C(C(CC)n2cncn2)=O)CC2CCC1CN2Cc1cccnc1 34628,c1(C(N(CCNC(c2nc(C(C)(C)C)sc2)=O)CC2CC2)=O)cc(C2CC2)ncn1 34629,C(=O)(C#CC1CCCCO1)NC1CN(C(c2cc(CC)c(F)cc2)=O)CC(F)C1 34630,N1(C(=O)OC(C)(C)C)CC2CCCN(Cc3cccc(F)c3Cl)C2C1 34631,c1(C(CC(=O)N(C2CCN(C(=O)COCC3CC3)CC2)CC)C)ccc(F)cc1 34632,C(=O)(C(C)(C)CCC(=O)N(CC(C)CNC(C1CC2C=CC1C2)=O)C)OC 34633,CCC(O)C(C)C(=O)NC1(CO)CN(C(=O)C=CC(C)C)C1 34634,Cc1ocnc1CC(=O)N(CCCCCNC(=O)CC(C)n1cccc1)C 34635,C(CCCC(C)NC(=O)CCCc1ccsc1)NC(C1C(C(C)=O)COC1)=O 34636,c1(CC(=O)NC2CCCC(CN=c3[nH]nc(O)s3)C2)cccc(Cl)c1Cl 34637,c1(OC)cccc(C(N2CCC(F)C(NC(=O)C(C(C)O)NC(C)=O)C2)=O)c1F 34638,N1(C(c2cc(C)nnc2)=O)CCCC(C)(CNC(=O)Cc2cc(C)n(C)n2)C1 34639,c1(NC(=O)OCC)ccc(C(=O)NCCC2CCC(NC(=O)CC(F)F)C2)cc1 34640,c1(C(=O)NCC(C)N(C(=O)C(C2CCC2)OC)CC)cc(C)ccc1OC 34641,n1(CC(=O)OC)cnc(C)c1C(=O)NCCCCNC(=O)C(C)Cn1cccn1 34642,N1(C(c2ncn(CC)n2)=O)CCC2CC12C(=O)NCCCc1c[nH]nc1C 34643,C1(C(=O)NCCOC2CN(C(CC3(C=C)CC3)=O)C2)CCS(=O)(=O)C(C)C1 34644,N1(C(C23CC(OC)C2C3)=O)CC(NC(=O)CCCN2CCCC2)C(O)C1 34645,CC(=O)CCN=C(NCCCCCN(C)C)N1CCC(C2CC2)C1 34646,N1(Cc2c(OC)cccn2)C2CCCC1CC(NC(C1(C)CCCN1)=O)C2 34647,c1(OC)cc(C)c(C)cc1C(N1CCC1(C)C(=O)Nc1scnc1C(N)=O)=O 34648,CC(C)(CCNC(C1CCC1C(C)(C)C)=O)NC(=O)OC(C)(C)C 34649,C1(C2CCN(C(c3coc(Cl)n3)=O)CC2)(NC(C2(C)CC2)=O)CC1 34650,C1(CCOCCC(=O)NCC(C)N(C)C)CCCNC1 34651,N1(C(CCOCCOC)=O)CC(O)CC1C(=O)NC1CCC(NC(C)=O)CC1 34652,c1(C(C(=O)NCC)N(C(C)COC)C)ccc(C(C)(C)C)o1 34653,c1(CC(=O)NC2CCN(C(C(CC)F)=O)C2(C)C)ccc2nc(O)[nH]c2c1 34654,N1(C(c2cc(COC)on2)C(=O)NCCCC)CCOC(c2n[nH]c(C)n2)C1 34655,C1(C(=O)NCC2CC(NC(C3CN(S(CC)(=O)=O)C3)=O)C2)CCC(F)(F)CC1 34656,CC(C)CC(F)C(=O)N(CCCCCNC(c1nn(C)cc1Br)=O)C 34657,Cn1cnc(C(N2CCCCC2CNC(C2CCCC2(F)F)=O)=O)cc1=O 34658,C12(NC(c3ccc(O)nc3)=O)CCCC1N(C(c1ccc3nccn3c1)=O)CC2 34659,N1(C(c2c(C)nc[nH]2)=O)CCOC(C(C)NC(=O)C(F)(F)c2ccsc2Cl)C1 34660,CC1CN(C(C2CCCN2C)=O)CCN1C(c1cc(Cl)ns1)=O 34661,Cc1c(CN(C(N2CCC2C2CCCCC2)=O)CC2CC2)oc2ccccc12 34662,C(=O)(C(CCSC)NC(=O)NC(C)(C)C)NC12CC(OC)C1C2 34663,c1(-n2cc(CN(CCN(C(C(C)OCC=C)=O)C)C)nn2)ccc2[nH]ncc2c1 34664,c1(C(=O)NC2CCCN(C(C3C(C(C)C)CCC3)=O)CC2)cnc2c(c1)CCC2 34665,Cn1ncc(=NC(=O)C2CC23CCN(Cc2ccc(C(=O)O)s2)C3)[nH]1 34666,c1(C(=O)NC2CCCC(NC(C3CC(F)C3)=O)C2)c(F)c(F)c(F)c(F)c1F 34667,N1(C(C2CC(C)CN2C(c2cn(C)cn2)=O)=O)CCC2(CCSC2)C1 34668,Cc1cnc2cc(C(N3CCCC3C(C)NC(=O)CC(F)(F)F)=O)nn2c1 34669,N1(C(C2(COC)CCCC2)=O)CCC(C2CC2)(NC(=O)C(O)C2CCCC2)C1 34670,C1(C2(O)CCOC2)(C(N(C)CC2CCN(C(c3ccc(C4CC4)o3)=O)C2)=O)CC1 34671,C1(NC(C2C(CNC(c3cc(C)n(C)n3)=O)C2)=O)CC(C2CCC2)C1 34672,C1(NC(COCCC)=O)CC2CN(C(C3CC(Cl)(Cl)C3)=O)CC2C1 34673,C1(NC(c2c(C)n[nH]c2)=O)CC2CCC1N2C(=O)C=CC1CCOC1 34674,C=CCC(CC(C)C)C(=O)NCc1ccc(C(=O)NC(C)C(C)n2cccn2)o1 34675,N1(C(C(C(C)C)CN(C)C)=O)CCN(C(=O)CCCC(N)=O)C2(CCC2)C1 34676,CC(CC(=O)N1CCC(C(=O)NCC(C)(C)N2CCCC2)O1)N(C)C 34677,C1(NC(C2(C(=O)OCC)CCCC2)=O)CCN(C(C2CCC(=O)N2C)=O)C1CC 34678,C1(NC(Cc2cc(C(N)=O)on2)=O)CCCCC1NC(=O)Cc1cncnc1O 34679,c1(CC)oc2ccccc2c1C(N1CC(CNC(=O)C(C)CSC)C(F)(F)C1)=O 34680,CC(CO)CCCNC(C1C(NC(=O)CN2CC3CC3C2)C1(C)C)=O 34681,Cc1nc(CC(=O)N(C)CC2(O)CN(C(C3(NC(N)=O)CC3)=O)C2)co1 34682,C(=O)(CCCCBr)NCC1N(C(c2c(C)nn[nH]2)=O)CC=C1 34683,c1(OC(C)C(=O)NCC2CCN2C(c2nn(C)cc2C(F)F)=O)cccc(F)c1 34684,CCCC(C)CC(=O)NCC1(O)CCCN(C(=O)CCc2nc(C(C)C)no2)C1 34685,C(=O)(CCCCCCO)N1CCC(O)(CNC(c2ccc(Cl)cc2C(F)F)=O)C1 34686,c1(C(N(C)CCNC(C2CS(=O)(=O)CC(=O)N2)=O)=O)cccc2cnnc(O)c12 34687,Cc1sc(Cl)nc1C(=O)N(CCC(C(C)C)NC(C1(C)COCCO1)=O)C 34688,c1(N2CCC(C(C)NC(C3(C)CCCCO3)=O)CC2)cc(=O)n(C)cn1 34689,C1(CC(=O)NCCCN(C(=O)CC=CC=C(C)C)CCC)CCC(C)C1 34690,c1(C(=O)NCCCCCN(C(=O)CC2CC2(C)C)C)cnn2c(Cl)cccc12 34691,Cc1cc(C(=O)NC2CC2NC(=O)COCc2nccn2C)cc(C)c1Cl 34692,CC1CN(C(=O)CSS(C)(=O)=O)CC1NC(=O)CCCc1ccsc1 34693,n1(CC)cc(Cl)c(C(=O)NC2CCC2NC(c2cnc[nH]2)=O)n1 34694,N1(C(c2n[nH]c(C)c2Cl)=O)CCCC(C)(CNC(=O)CC2CC(C)(C)CCO2)C1 34695,N1(C(c2cc(CCC)[nH]n2)=O)CCN(C(C2CCC(=O)N2)=O)CC1C(C)(C)C 34696,S(=O)(=O)(c1c[nH]c2nc(Cl)ccc12)NCC1CCC(CC)C1 34697,C1(CNC(CCNC(=O)OCC)=O)CC2(CCC2)CN1C(C1CC1(Cl)Cl)=O 34698,C1(NC(CCC2N(C)CCC2)=O)CC=C(C(=O)Nc2ccc(C3CC3)nc2)C1 34699,O=S(=O)(c1ccncc1)NC1C2CCC1CC(CO)C2 34700,CC(CS(C)(=O)=O)C(=O)N1CC2CC(NC(c3ccc(N(C)C)nc3)=O)C(C2)C1 34701,C1(CNC(c2ccc(C(C)(C)C)[nH]2)=O)CN(C(C2CCC3CC23)=O)CCC1(F)F 34702,CC(CCC(C)(C)C)N=c1[nH]c(N2CCOC(CC(F)(F)F)C2)nc(=N)[nH]1 34703,Cc1c(C(=O)NCC(O)CNC(=O)CC2CC3(CC3)C2)sc2nccn12 34704,c1(CC(=O)NC(CC)(C)CNC(=O)Cc2cccs2)ccc2scc(C)c2c1 34705,c1(CCC)nnc(S)n1CC(=O)NCCCCC(C)NC(c1cnc(S)n1C)=O 34706,CC(C)CC(C)(CNC(C1CC(OC(C)(C)C)C1)=O)NCc1ccc(F)cc1F 34707,C=CCC(C)(C)C(=O)NC1CCN(C(=O)CCCCC2CC2)CC1CO 34708,OC1COC2C(NC3CCCC4(C3)N=N4)COC12 34709,c1(C(=O)NC(C(=O)OC2C(OC(C)=O)C2)(C)C)cc(Cl)cc(Cl)c1 34710,CC1CC2(CCO1)CC2C(=O)NCCN1CCN(c2ccncc2[N+](=O)[O-])CC1 34711,N#Cc1ccc(CC(=O)NCC2CCN(C(=O)CCN3CCCC3)C2)cc1 34712,C(c1ccc(F)cc1)=CC(=O)NCC1CC(F)(CNC(C2(F)CC2(Cl)Cl)=O)C1 34713,N(C(=NCC(C)(C)CC#N)NCC1CCOC1)C(C)Cc1ccccn1 34714,c1(C(CCNC(c2cn(CC(=O)OC)nn2)C)O)ccc(Br)cc1.N1CCOCC1 34715,N1(CCOCC)CCN(C2CCN(C(=O)CC(N)C3CCOCC3)C2)CC1 34716,C1(CN(C(C(n2ccc(C(F)(F)F)n2)C)=O)C)CC(F)CN1C(c1ccns1)=O 34717,N1(C(c2cc(C)ncc2C)=O)CCC(C)(C)C(CNC(=O)Cc2cnoc2)C1 34718,N1(C(C(c2ccc(Cl)cc2)C)=O)CCC(Cn2cc(CC3CC3)nn2)C(F)(F)C1 34719,CN(C)N=Nc1ccccc1C(N1CCCC1Cc1ccc(C(F)F)cc1)=O 34720,C1(N(C)C)CCCN(C(=O)C(C)(N)C(F)F)CC1 34721,N1(C(c2ccc(OC)c(C3CC3)c2)C(=O)NC2CCCC2)CCOCC12CCC2 34722,C1(C)(C(=O)NC(CC=C)CNC(=O)CN2CC(F)(F)C2)CCCOC1 34723,C(=O)(C1=CC2CCCCC12)N1C(C(C)(C)NC(c2c(OC)cccc2)=O)CCC1 34724,c1(C(=O)NCC23C(CN(C(C4CC(C)(F)C4)=O)C2)C3)cccc2c1CCO2 34725,Cc1c[nH]c2ncc(C(N3CC4CCN(C(=O)C=CS(C)=O)C4C3)=O)cc12 34726,Clc1ccc(CNc2cnn(C3CCC3)n2)c(I)c1 34727,N1(C(C2CCC(COC)C2)=O)CCN(C(c2cnc(C)s2)=O)CC(O)C1 34728,C(C(O)CS(=O)(=O)c1cccs1)NC(c1ccc(-n2ncc(C(=O)O)c2)cc1)=O 34729,CC1CCN(C(C2CCC=CO2)=O)CC1NC(=O)CC1CCC(C(C)(C)C)CC1 34730,C12(C(N3C4CN(C(C5C(CC)C5)=O)CC3CC4)=O)CCCCC1CCCC2 34731,C#Cc1ccc(C(N2CCN(C(C3CC3C(C)(C)C)=O)CC2C2CCC2)=O)cc1 34732,c1(C(C(C)(C)C)NCCNC(=O)NCC2(N(C)C)CCC2)cccc(C)c1 34733,c1(C(N2CCC(F)(CNC(c3ncn(CC)n3)=O)CC2)=O)cc[nH]c2nccc1-2 34734,c1(C(N2CCC(O)(c3onc(C)n3)C2)=O)nc(C(F)(F)F)ccc1Br 34735,n1(CCNC(CC2(O)CCCN(C)C2)=O)cnc2ccc(F)cc2c1=O 34736,c1(NC(c2nn(C)cc2Cl)c2n(CCSC)nnn2)nnc(C)n1C 34737,C(CCOCCO)(C(=O)N(C(C(N)=O)C1CC1)C)NC(C=CCC)=O 34738,C1(C(N(CC(C)(C)CO)C)=O)(CN(C)C)CCCC1 34739,CCC(CC)(C(=O)NCCCN(c1cc(Cl)ncn1)C(C)C)c1ccccc1 34740,Cn1c(Br)cnc1NC(N1CCN(c2ccc(Cl)nn2)CC1)=O 34741,c1(OC)ccc2c(c1)CCC2(C)CNc1nc(OC)ncc1Cl 34742,C(=O)(C#CC1CCCCC1)N1CC(N(C)C(c2ccc(Cl)c(F)c2)=O)C1 34743,c1(OC)ccccc1C(=O)NC(CNC(=O)C(C1CCCC1)OC)CO 34744,Cn1cc(C(N2CCC(O)(CNC(C3CCC(=O)N3)=O)C2)=O)c2cc(F)ccc12 34745,Cc1cc(C(N2CCC(C)(C(=O)NCC3(C)CC4CCC3C4)CC2)=O)c(C)n1C 34746,C#CC1CCC(NC(c2csc(CNC(c3ccc(CO)cc3)=O)c2)=O)C1 34747,N1(C(C(N2C(CC)CCC2)=O)=O)CCOCC1CN(C(=O)Cc1ccsc1)C 34748,C(=O)(CCC(=O)NN(C)C)NC1C(CO)CCN(C(COCCCC)=O)C1 34749,c1(C(=O)NCC23CC2CN(C(C2CC=CC2)=O)C3)cccc2cccn12 34750,c1(C(=O)NCC(C(C)C)NC(C2CC2C#N)=O)ccc(SC(F)(F)F)nc1 34751,N1(C(CC=CC=C)=O)CC(NC(c2ccc(-c3cnn(C)c3)o2)=O)CC2(CC2)C1 34752,C1C(C)CN(C(=O)CCCC(Cl)Cl)CC1C.N12CCCN(CC1)C(=O)C2.CCC 34753,c1(C(N(CC(C)(C)NC(C2C(=C)C2)=O)C)=O)ccccc1-n1nnnc1C1CC1 34754,N1(C(CC2C(C)(C)CCO2)=O)CC=C(CNC(=O)Cn2cnc(C(N)=O)n2)CC1 34755,c1(CC(=O)NCC2C(NC(C(CC)O)=O)CC2)c(C)nn(CC(C)C)c1C 34756,CC(C)C(CC(=O)NCC1CC1C(C)C)NC(C1CC2CC(=O)C1O2)=O 34757,C(CCC(C)C(=O)NCC1(C(=O)NOCCCO)CCOC1)OC 34758,c1(C(N2CC(C(N3C(CC)CC(O)C3)=O)(CC)C2)=O)cnn2c1CCC2 34759,CC1(CNC(=O)C=CCO)CC(F)(F)CN1C(C1CCC2(CC2)C1)=O 34760,C1(NC(Cc2nc(C)[nH]n2)=O)CNCCOC1 34761,C1(NC(CC(=C=C)C)=O)CN(C(=O)CC2CCCOC2)C2(CCOCC2)C1 34762,c1(CCC)ncoc1C(=O)N(CCNC(C1CC1(C)C)=O)CC 34763,C(C)(C(=O)NC1(C)CCC(C)C1)(C(C)C)NC(C)=O 34764,c1(C(=O)NC2CC(CNC(=O)COC3COC3)C2)cc(Cl)ncc1F 34765,N1(C(CCNC(COC)=O)=O)CCOC(CNC(c2c[nH]nc2COC)=O)C1 34766,c1(C(N(C2CCN(C(C3CC34CC4)=O)CC2)CC(C)C)=O)ncncc1Cl 34767,c1(C(N2CCC(C3CC3)(NC(=O)CC3CCC3)C2)=O)ccc2cnnc(O)c2c1 34768,C(CC(C(=O)NC(c1cncc(F)c1)C)NC(=O)Cc1nc(=N)[nH][nH]1)=CC 34769,c1(C(N2CC(NC(c3n(CC)nnc3)=O)C3C2C3)=O)cnc(N)c(N)c1 34770,Cc1ccc(CNC2CC3(C2)CC(C(=O)NCc2ccc(C#N)cc2)C3)c(O)c1 34771,N1(C(CC(C)SC)=O)C2COCC1CC(NC(=O)C(C)=NOCC#N)C2 34772,c1(C2(OC)CC2)nnc(N(C(c2ccc(C(F)(F)F)cc2)C)C2CC2)n1CC(C)C 34773,C1(CCC)CN(C(C2CCC(C(C)C)N2C(=O)CCC(=O)C2CC2)=O)CC1C(N)=O 34774,c1(CC(n2cc(-c3cncc(F)c3)nn2)C)ccccc1F.c1(=O)c(=O)n1C 34775,C(=O)(C(O)C(C)(C)CC)N1CC(NC(CCC=CCC=C)=O)C2(C1)CC2 34776,C1(CNC(COCC)=O)(CNC(c2nonc2CC)=O)CCOCC1 34777,C1(C(C)NC(c2cc(Cl)c[nH]2)=O)CCCCN1C(=O)CCCc1ccccc1 34778,N1(C(C2C(NC(CCOC(C)=O)=O)CC2)=O)CCOC(C#N)C1 34779,c1(C(=O)NC(c2c(C(=O)NCC3C(OCC)CC3)con2)C)cc(O)nc(C)n1 34780,CN=S(C)(=O)c1cccc(CNC2CCN(C(=O)OC(C)(C)C)CCC2CO)c1 34781,C#Cc1ccc(C(=O)NCC(O)CN(C)C(c2ccc(CO)cc2OC)=O)cn1 34782,Cc1ccc2nc(N(CC(O)CN(C)C(c3c(C)nn(C)c3C)=O)C)sc2n1 34783,CC1(C)OCCOC1CC(=O)NCCOCCCNC(=O)CC1OCCCO1 34784,C12(NC(C(=C)F)=O)CCC(NC(=O)Nc3nnc(-c4ccc(Cl)cc4)s3)(CC1)C2 34785,N1(CC(C)OC)C(=O)CN(C(C)C=CC(F)(F)F)C1=O 34786,C1(CCC(=O)N(C)CCO)CCCN(C(c2cocc2C(N)=O)=O)C1 34787,C1(NC(C2(C)N(C)CCC2)=O)C2CCC(C2)C1C(=O)NC1COCC1O 34788,Cn1cnc(CNc2cccc(OCC3CCCCC3)c2)cc1=O 34789,c1(CNC2(C(c3ccccc3Cl)O)CCCC2)c(Cl)ccc(Br)c1F 34790,c1(C(=O)NCCCCCN(C(=O)CC2CCCC(F)(F)C2)C)cc(=O)n(C)cn1 34791,n1(C(C)C)cncc1C(=O)NCC1CCCC1NC(C1CC(N(C)C)C1)=O 34792,C1(C2CCN(C(C3(C)CC3C)=O)C2)(NC(c2n[nH]c(C)c2C)=O)CC1 34793,c1(C(=O)NCC2(OC)CN(C(C3(CC)CCCCO3)=O)C2)ccc(C)cc1Cl 34794,c1(NC(N(CCC(=O)OCC)CC)=O)ccc(C)cc1OCCCCCC 34795,C(=O)(C(CCC(C)C)N(C(C)(C)C)C(C)C)NC1(c2ccc(CC)cc2)CCC1 34796,N(C(=NCCC(=O)N(C)C)NC1CCOCC1F)Cc1n(CCC)ncn1 34797,C#CCCC(=O)N(CCC(C)(C)NC(C1CC(N(C)C(C)=O)C1)=O)C 34798,c1(OC)ccc(S(=O)(=O)NCC2(F)CCCN(C(=O)CC3CC3)C2)cn1 34799,C(CC(C(=O)N(C)Cc1nc(C)no1)NC(=O)CCCc1ncco1)OC 34800,c1(CC(=O)NCC(C)NC(CC(c2cccc(OC)c2)C)=O)ccc(F)c(C)c1 34801,CC(C(=O)NCc1ccc(CNC(=O)C=CCN2CCCC2)cc1F)S(N)(=O)=O 34802,C12(NC(N3CCN(C(c4ccc([N+](=O)[O-])cc4)C)CC3)=O)CCOC1CS(=O)(=O)C2 34803,N1(C(C(CC#C)(C)C)=O)CC2CCC1C(CNC(C1(c3ccn(C)n3)CC1)=O)C2 34804,N1(C(c2sccc2Br)=O)CCCC(O)(Cn2cc(C3(F)COC3)nn2)CC1 34805,c1(C(=O)NC(CC(C)NC(c2c(C#C)c[nH]n2)=O)C)noc2c1CCCC2 34806,Cc1nc(O)nc(O)c1CC(N1CCCC(CNC(C2(C(N)=O)CCC2)=O)C1)=O 34807,c1(C(C)=O)ncc(C(N2CC(O)(C(C)NC(=O)C(c3ccnn3C)C)C2)=O)s1 34808,N(C1CC2(CCC2)Oc2ccc(F)cc21)c1n(C)c(Cl)nc1 34809,C1(C(N2CC(C(C)(C)O)C2)=O)CN(C(=O)CCc2cncs2)CC2(CCC2)C1 34810,c1(C(=O)NCC(C)NC(=O)Cc2ccc(Br)cc2)nccc(C#N)c1F 34811,c1(CCNC(C(=O)NCC2CCCC2O)=O)c[nH]c2cccc(Br)c12 34812,c1(OCCCC)ccccc1OC1(C)N(C(=O)Nc2ccccc2)CCC1 34813,CCCCCCCCC(F)C(=O)NC1CCCN(C(=O)C2=CCCOCC2)CC1 34814,c1(C(N2CCCC(NC(c3c(C#N)nc[nH]3)=O)C2)=O)ccc2c(O)nncc2c1 34815,C=CC(C)CC(=O)NCCOCCOCCNC(C1CCCCO1)=O 34816,N1(C(CCC(C)OC)=O)CCCC(F)(C(=O)NC2CC(C)C2)C1 34817,C1(CC=C)CCCCN1C(C1CCN1C(=O)CC1CCOC1)=O 34818,N1(C(C(CC)(C)F)=O)CCC2(CC1)CN(C(=O)C1CC1)C2.C12CCCN(C1)C2=O 34819,O=C(C1=CC(O)CCC1)NCC(C1CCCC1)NC(c1cccc[n+]1[O-])=O 34820,C(c1ccccc1)=C(C(=O)NCC1C(NC(CCC=C)=O)CCC1)c1cccs1 34821,n1(CC)cccc1C(c1nnnn1C1CCOC1)NCc1cncs1 34822,c1(C(=O)NC(C(CO)NC(C(C(C)O)N(C)C)=O)C)nnc2n1CCCCC2 34823,Cc1coc(C(C)(C)C)c1C(N1CC(N(C(=O)C(F)C2CCOC2)C)C1)=O 34824,c1(C(=O)Nc2c(C(=O)NC3CC(F)(F)C3)ccc(Cl)n2)cc(Cl)c(F)c(Cl)c1F 34825,N1(C(C2(C)N(C(c3c(CC)noc3)=O)CCC2)=O)CCc2ncncc2C1 34826,C1(C(N(CC(C)NC(=O)CCc2cnc[nH]2)C)=O)CC2(C1)C(F)(F)C21CC1 34827,C(CO)(CC(F)(F)F)NC(C(c1n(C)ncc1)NC(=O)CC1OCCC1(C)C)=O 34828,C(=O)(CC1=CCN(C(C23CCC(OC)C2C3)=O)CC1)N(CCC=C)CC 34829,C1(C(C)NC(c2coc(Cl)c2)=O)CCCN(C(C2CCCCN2S(C)(=O)=O)=O)C1 34830,N(C1CCOc2ccc(Cl)cc21)C(c1cnc(C)n1-c1ccc(F)cc1CN)=O 34831,N1(C(C(F)=C(C)C)=O)Cc2nccn2CC(NC(=O)C(c2ccn(C)n2)C)C1 34832,C#Cc1ccc(C2(C(=O)NCC3CCN3C(c3coc(CO)c3)=O)CCC2)cc1 34833,N1(C(c2n(C(CC)C)ncc2)=O)CCN(C(=O)CC(C)(C)C2CC2)CC1C(C)C 34834,CC(C)S(=O)(=O)CCCN(C1CCCN(C(=O)C(=O)Nc2ccccc2)CC1)C 34835,CC(C)(Cc1cnn[nH]1)C(=O)N1CC(NC(C2CCC(C(F)(F)F)O2)=O)C(O)C1 34836,c1(C(N2CC(NC(C(C)n3cccn3)=O)C2)=O)cc(NC(C2CCC2)=O)on1 34837,c1(SCC(=O)N(CC(CNC(C2(C#C)CC2)=O)(C)C)CC)ccc(Cl)cc1 34838,S(=O)(=O)(c1ccncc1)NC1CCN(C(c2ccc(NC(C)C)cc2)=O)CC1F 34839,CC1c2c[nH]nc2CCC1C(N1CCC(CNC(=O)CC2=CCCC2)C1(C)C)=O 34840,N1(C(C(CCC)NC(C)=O)=O)CCN(Cc2cnc(OC)c(C)c2)CC1C#N 34841,c1(C(=O)NC(C)C(=O)NC(c2nc[nH]n2)CO)cc[nH]c2nccc1-2 34842,c1(C(=O)OC)ccc(SC)cc1.c12cc(sn1)C(C(=O)NCCCF)N2C 34843,C1(CC(N2CCC(O)(CNC(c3cnc(C(C)C)s3)=O)C2)=O)OCCCC1(C)C 34844,c1(C(=O)NCC(CC)NC(c2snnc2C)=O)cccc2cnsc12 34845,C1(CNC(C2CCC(CNC(=O)COCCCF)CC2)=O)CC2(CCC2)CO1 34846,Cc1ccc(C(=O)NCC2CCN(C(C34CCC3C4)=O)C2)cc1 34847,c1(C(=O)NC2C(SC)CN(C(=O)CN3CCSCC3)C2)nccn2cc(C)nc12 34848,N1(C(=O)CCN2CCCC2)CCC(C(N2CCCC(CN(Cl)Cl)C2)=O)CC1 34849,C1(C(N2CCN(CCN(C(=O)Cn3ccnn3)C)CC2)=O)CCCC12OCCO2 34850,C1(NCC2CC(C)N(C(CNc3nccc(OC)n3)=O)C2)CCCCCS1(=O)=O 34851,N1(C(C(CC)NC(N)=O)=O)CC(NC(=O)CCc2ccccc2C)CCC1C 34852,N1(C(c2cn(CC3CNC(=O)O3)nn2)=O)CCCC2CN(C(=O)CC3CC3)CC12 34853,C1(C(=O)NC(C2CCN(C(=O)CCc3cnc(C4CC4)o3)C2)C)C=CC=CC=C1 34854,C(C(F)(C(=O)N(C)CC1(OC)CCC1)C(C)C)NC(c1cc(=NC)[nH]cc1)=O 34855,C(=O)(C(CCN(C)C)NC(c1cnnc(O)c1)=O)N1CCC(CC)C1 34856,c1(CC(C(=O)NS(=O)(=O)C2(c3cncnc3)CC2)n2cnnc2)ccc(O)cc1 34857,C1(C(N2CC(C)C(NC(C3(C(F)(F)F)CC3)=O)C2)=O)CC1C1CCOCC1 34858,CCC(CN(C)C)C(=O)NC1CC(CNC(=O)C=CC(=O)OC(C)(C)C)C1 34859,c1(CC)nc(C)c(C(=O)NC2CCCC(N(C)C(c3cocc3C)=O)C2)o1 34860,N1(C(C)C(=O)N2CC(c3cnn(-c4ccccc4)c3)C2)CCCCC1=O 34861,C(=O)(C(C)CC(=C)C)NC1(CNC(c2cc(CCCCC)on2)=O)CCCCC1 34862,N1(C(CSC)=O)CCN(C(C2CCCN(C(=O)CC3(C)CC3(Cl)Cl)C2)=O)CC1 34863,Cc1nc(O)sc1C(=O)NC1COCCC1C(=O)N(C)CCN1CCCC1 34864,C12(C(=O)NCCCCCNC(C(CN(C)C)(F)F)=O)CCCN(C1)S(=O)(=O)C2 34865,c1(C(=O)NCCC(C)CO)ccc2ncc(-c3cc(F)c(F)cc3O)n2c1 34866,c1(NC(CN(C(CN(CC=C)CC)=O)C)=O)ncc[nH]1.C(=O)(COC)N(C)C 34867,N1(C(c2c(OC)nccc2)=O)CCCC(N(c2cnc(C#N)cn2)C)CC1 34868,c1(C(N(C2CCN(C(=O)C(C)(C)C)C2)CCC)=O)c2c(nn1CC)CCCC2 34869,c1(C(N2C3CN(C(=O)Cc4cn[nH]c4)C(C3)C2)=O)nc2cnccc2s1 34870,C(CC(C)(C)F)NC(C1CN(C(C2C(C(=O)OCC)C2)=O)C1)=O 34871,Cc1cncc(C(N)C(=O)NC(C)CC2CCNCC2)c1 34872,C1(C(N2CCC(NC(CC(C=C)CC)=O)C(C)C2)=O)CCC2(CC1)CNC(=O)C2 34873,CC1(C(=O)NCCCNC(=O)C(c2ccc(F)cc2)(C)O)CCC(O)CC1 34874,N1(C(COCC)=O)CCN(C(C2CCCCN2C(=O)CC)=O)CC1CCOC 34875,c1(C(N2CC(C=C)C(NC(=O)COc3cn[nH]c3)C2)=O)csc2ccc(F)cc12 34876,C(CCCCC(=O)NC1CCC(C(N)=O)CC1)N(C(=O)C(=O)C1CCCC1)C 34877,Cn1ccc2nc(N3CCC(CC(N4CCC(CO)C(F)(F)C4)=O)CC3)ncc12 34878,C1(OC(C)C)CC(CC(=O)Nc2ccc(C(F)(F)F)cn2)C1(C)C.C1CCC(=O)N1 34879,c1(NC(N=c2n(-c3c(OC)cc(Cl)cc3)[nH]nn2)=O)cccc2c1nc(O)n2C 34880,c1(C(N2CC(NC(C3(OC)CCOC3)=O)C(O)C2)=O)c(N)sc(C)c1C 34881,CC1=NOC(=O)C1CCC(=O)NCCOC1CCN(C(c2ocnc2C)=O)C1 34882,c1(CC)c(C(C)NC(c2nn(C)cc2C)=O)oc2ccccc12 34883,C1(NC(c2c(O)ncc(NC(C)=O)c2)=O)CCC2(CCCNC2)C1 34884,c1(C(N2CC(C(C)NC(c3cnc(CC)s3)=O)OCC2)=O)cc(O)ccc1N 34885,CC1CN(C(C2CC2c2ccc(Br)cc2)=O)CCN1S(=O)(=O)c1cccs1 34886,C=CCN=C(NCCC1CC(C(=O)NC)C1(C)C)NCC(C)(C)NC(C)=O 34887,Cc1cccc2nc(C(=O)NC(C)(C)C(C)NC(C3CNC(=O)N3)=O)cn12 34888,c1(C(=O)NC2CCC(NC(c3cc(C)sc3)=O)CC2)cnc2cn(C)nc2c1 34889,c1(C(=O)NCC(C(C)(C)C)NC(c2c(C)cc(CO)o2)=O)cc(C)c(O)c(N)c1 34890,CCC(CC)C(C)C(=O)N1CCC(C(=O)NCc2nnc(O)o2)(CO)C1 34891,c1(C(=O)NC(C2CCN(C(=O)Cc3n[nH]c(=N)s3)C2)C)cc(OC(F)F)n(C)n1 34892,C1(C(N(C(C)CC2CC2)C)=O)C2CC3C(C2NC(=O)C(C)C(F)F)C13 34893,c1(CCC)nsc(N)c1C(=O)NC1CC1NC(=O)Cn1cccn1 34894,N1(C(CCC2CC(NC(Cc3cc(C)sc3)=O)C2)=O)CCCCC1C 34895,Cc1ccc(C(CNC(c2occc2C)=O)NC(c2scc(C)c2C)=O)cc1 34896,O=C1CCCCn2nc(C(N3CCOCC(CNC(C4CCOC4)=O)C3)=O)cc21 34897,C1(NC(Cn2ncc(C#C)c2)=O)CN(C(=O)C(C)CC(F)F)C(C)(C)C1 34898,c1(CC)cnc(C)nc1N1CCC(CNC(=O)CN(C)CCOC)C1 34899,C1(CN(C)C(c2cc(CO)[nH]n2)=O)CN(C(c2cc(Cl)cn2C)=O)CCO1 34900,CC1CCC(C)(C(=O)NCC(=C2CN(C(C3CC4CCC3C4)=O)C2)F)CC1 34901,Cc1c(C)c(C)c(CSCCC(C)(F)F)c(C)c1C 34902,c1(C(=O)NCC2N(C(CCCC#C)=O)CC2)ccc(NC)c(C(F)(F)F)c1 34903,c1(C(=O)NCC(C(=O)NCc2ncc(C)[nH]2)C)cncc(C#N)c1 34904,Cc1ccc(CC(CO)NC(c2cnc[nH]2)=O)nc1 34905,c1(C(N2CC(CC)N(C(=O)CC3C=CS(=O)(=O)C3)CC2)=O)nccn2ccnc12 34906,C1(N(C)C(C23CSCC2C3)=O)CCN(C(=O)CCOc2ccccc2)CC1 34907,C1(N(C(=O)CCC2CCC2)C)CCN(C(=O)Cc2nccn2C)C1 34908,c1(C(N2CC(C)C(NC(c3csc(O)n3)=O)CC2)=O)cncc2c(O)nccc12 34909,C(CCC(C(=O)NCc1cccc(F)c1F)NC(c1cocn1)=O)OC 34910,n1(CC(=O)N(C2CCN(C(=O)C=CC(F)(F)F)C2)CCC)cnnc1O 34911,Cc1cc(C(=O)NC2CCC(C)N(C(C3SC4C=CC3CC4)=O)C2)ccc1O 34912,C1(CCC)CN(C(c2cc(F)ccc2F)=O)CCN1C(c1cc2[nH]ccc2s1)=O 34913,C1(C(=O)NCC(C)(C2CC2)NC(c2ccnnc2)=O)CC(C)(c2ccccc2)C1 34914,C1(CCC)CCCCC1NC(c1csc(CNC(C2(CO)CCCCC2)=O)c1)=O 34915,CC1(C(N2CCCN(C(=O)CC3CCCCO3)CC2)=O)COCC1(F)F 34916,c1(N2CC3(CN(C(c4c(C)cno4)=O)C3)C2)ccc2c(n1)CCCC2=O 34917,c1(CC(=O)NCC2CC2NC(c2cocn2)=O)cnc(C2CC2)[nH]1 34918,C(=O)(C1=C(Cl)CCCC1)NC(C)CNC(=O)C(C)(C)n1cnnn1 34919,c1(C(N2CCC(COC)(NC(C3(CF)CC3)=O)C2)=O)cc(Cl)cc(C(F)(F)F)n1 34920,N1(C(C(C(C)C)F)=O)CCC(C)(NC(=O)CCc2nnc(O)nc2O)CC1 34921,c1(OC)c(Cl)ccnc1NC(C1CC(NCc2cnccc2Br)C1)=O 34922,N1(C(C2C3(CC(NC(C4C(C)CCOC4)=O)C3)C2)=O)CCC(O)(C(N)=O)CC1 34923,C(CC(=O)NN1CCCC1C(=O)NCc1nc(C)sc1C)OC 34924,N1(C(=O)NC(C)C(=O)N(CC(F)(F)F)C)CCN(C2CCCC2)C(C)C1 34925,N1(C(CCSCCC=C)=O)CCN(C(C2CC2C(=O)OCC(CC)CC)=O)CC(C)C1 34926,C1(NC2C(OCCC(C)C)CCCC2)CC(C2CCOC2)C1 34927,N1(C(C2(C)CC(C)(C)C2)=O)CCCN(CCNC(C2CCCO2)=O)CC1 34928,CN1CCC(CC(N2CCCC(C(C)NC(C3CC3OC(C)(C)C)=O)C2)=O)CC1 34929,C(C(N=[N+]=[N-])C(=O)N1CCC(C)(NC(=O)CC2CCCCC2O)C1)OCC 34930,N1(C(CC2(OC)CC2)=O)CC2CC(Nc3ncnn4cccc34)CC1C2 34931,Cc1cc(F)ccc1CC(=O)NC(CNC(=O)CC1CCCC(=O)N1)CC(C)C 34932,C(C(O)C(=O)NCC(c1ccccn1)(F)F)NC(=O)CC1CCCCC1 34933,c1(C(=O)NC2(C(=O)NC(CC(=O)OCC)C)CCC2)c[n+]([O-])c(C)cn1 34934,C1(C)(CC(=O)NCCN(C(C2(c3cccs3)C(C)C2)=O)CC2CC2)CCCO1 34935,c1(NC(Cn2c(C)cnc2)=O)cccc(CNC(c2cncc(N)n2)=O)c1 34936,N1(C(CN(C)CC)=O)C2CCC1CC(O)(CNC(=O)C(C)OCOC)C2 34937,Cc1cc(C(=O)NCC2(NC(C3(F)CCCC3)=O)CCCCC2C)cc(C)c1N 34938,N1(C(C2N(C(Cn3ncc(CC)c3)=O)CCCC2CC)=O)CC2(CNC(=O)N2)C1 34939,c1(C(N2CC(C(C)C)N(C(C3CC(C)(F)C3)=O)CC2)=O)coc(S(C)(=O)=O)c1 34940,CCCCCC(C)CC(=O)NCC1(O)CCCN(C(C2(CC)COC2)=O)C1 34941,C(CNC(c1cncs1)=O)(C(C)C(C)C)NC(c1c(C)cn(C)n1)=O 34942,C=CC1(C(=O)NCC(C)(CC)NC(c2ccn(C3CC3)c2C)=O)CCCCC1 34943,C1(NC(C2CCCCC2)=O)C2CCC1N(C(c1ccc(C(F)F)cn1)=O)C2 34944,CC(C(C)(C)CC(=O)O)NC(=O)C(C)OCc1cn(Cc2ccccc2)nn1 34945,C12(NC(=O)CN3CCSCC3)CCC1CN(C(C1Cc3nncn3C1)=O)C2 34946,c1(C(=O)NC2(C)CN(C(=O)CCCCOCCO)C2)ncc2ccccn12 34947,C12(NC(C3CN(C(C)C)C3)=O)CC3CC(C1)CC(CNC(C14CSC(C1)C4)=O)(C3)C2 34948,C(=O)(C(C)(C)C(F)F)N1CC(CNC(c2cnc(CCC)[nH]2)=O)C(OCCSC)C1 34949,C1(C(C)NC(C2CNC(=O)C2)=O)CN(C(=O)CN2CCCCC2)CCO1 34950,c1(C(N2CC(O)(CN(C(C(C)O)=O)C)C2)=O)cn(C)nc1-c1cccs1 34951,CC(CC(=O)NCC(O)CNC(C1(F)CCCC1)=O)NC(=O)NC1CCCC1 34952,c1(C(=O)NCC(CNC(c2ccc(C(C)C)nc2)=O)(C)O)cc(CO)ccc1Cl 34953,N1(C(C(CCC)OC)=O)CCC(CO)(NC(=O)CCOc2ccc(F)cc2)CC1 34954,c1(CC)n[nH]cc1C(=O)NC1CCC(CCC(=O)NCc2ccco2)C1 34955,N1(C(c2c(CC)occ2C)=O)CC(C(=O)NCc2csc(C)c2C)CCC1(C)C 34956,C(CNC(C1CC(=O)NC1(C)C)=O)(C(=O)N=c1cc(C)n(C(C)C)[nH]1)OC 34957,C(=O)(C1=C(C)OCCC1)N1CCC(C(N(C)CC)=O)C1C(C)C 34958,c1(C(=O)NC2CC(NC(c3onc(C)n3)=O)C2)cccc(C(F)(F)F)c1Cl 34959,C1(C(=O)NC(C2CCN(C)C2)C)(CO)CN(C(C2CCN(S(C)(=O)=O)C2)=O)C1 34960,c1(N(C(=O)CCCC(F)(F)F)C2CCNCC2F)ncnc2n[nH]c(Br)c12 34961,Cc1cc(C(=O)NCCC2CCCN(C(=O)Cc3cnc[nH]3)CC2)cc(F)c1C 34962,C#Cc1ccc(C(N2CCCC2CNC(=O)CC(N2CCCCC2=O)C)=O)o1 34963,N1(C(C(C)C(C)(F)F)=O)CC2(CCCC2CNC(=O)C(C2CCOCC2)O)C1 34964,C1(C(N2C(CN(C(=O)C#CC3CCC3)C)CCCC2)=O)CC2(CCC2=O)C1 34965,CCC(CC(=O)N(C)CCOCCC(N1CC=CC1C(=O)NC)=O)OC 34966,Cc1ccccc1CCC(=O)NC1(CNC(=O)C(C)C#N)CCCC1 34967,CC(C)S(=O)(=O)C(C)C(=O)NCCN(C(=O)CCCCN1CCCC1)C1CC1 34968,c1(C(=O)NCCCCNC(=O)C(c2ccccc2)F)cn(C2COC2)nn1 34969,c1(OC)cc(Cl)ncc1C(=O)Nc1c[nH]nc1C(=O)Nc1cc(I)ncn1 34970,CC1CC2CN(C(c3cccnc3O)=O)CC2N1C(=O)CCCC1CCCO1 34971,C1(CC(=O)NCCCCNC(C(Cc2ccccc2)OC)=O)CCC(=O)N1C 34972,N1(C(Cc2cc(C)on2)=O)CCC(C)(CNC(=O)C(C2CCOCC2)C)C1 34973,c1(C(N2C(C3CCN(C(C(CC)=CC)=O)C3)CCCC2)=O)ccc2ccnn2c1 34974,CCC(F)(F)CC(=O)NCC1CC1NC(=O)C(c1ccnn1C)O 34975,c1(C(=O)NC2CCCC(C(=O)NC3CC3)CC2)cccn2nccc12 34976,C1(C2CC2)(C(=O)NCC(C)CNC(=O)C(=C2CCCCC2)F)CC=CC1 34977,C(=O)(C(C)(C)C(F)(F)F)N(C(c1c(Cl)ccc(OC)n1)=O)C1CC1 34978,c1(C(=O)NCCOC2CN(C(C3CC34CCCOC4)=O)C2)cn2cccnc2n1 34979,CCC(C)(CNC(c1cc(C)c(F)cn1)=O)C(=O)NOCC(O)C(C)C 34980,c1(SC)ccc(C(=O)NCCC2CCCCN2C(=O)C(Cl)=CCl)c(Cl)c1 34981,C1(C(N)=O)(C(=O)NCC2(CNC(=O)COC3CCC3)CC2)CC1 34982,CCC(C)CCC(O)CC(=O)NC1(C)CN(C(c2csnc2OC)=O)C1 34983,N1(C(c2c(CC)ccs2)=O)CC(CNC(c2cnnc(O)c2)=O)CC1(C)C 34984,C1(NC(c2ccc(F)cc2)c2n(CCCCCC)nnn2)CCCCC1S(C)(=O)=O 34985,c1(COC)ccc(C(=O)N(C(C)CNC(C2(CC#N)COC2)=O)C)o1 34986,N1(C(CC2ON=C(C)C2)=O)CCC2CN(C(c3[nH]cc(C)c3C)=O)C2C1 34987,Cc1nn(C)c(C)c1CC(=O)N(C1CN(C(C23CCC2C3)=O)C1)CCO 34988,Cc1nc(=NC(=O)CCNC(C2CCN(c3cccc(Br)c3)C2=O)=O)o[nH]1 34989,N1(C(CN(CCOCC#C)C(c2cnsc2)=O)=O)CCC1CC 34990,N1(C(CC=CCNC(c2c(CC)con2)=O)=O)CCC12CCCSC2 34991,C(C(C)(C)CCC=C)NC(CCC=C)(C)c1nnnn1CCSC 34992,C1(NC(C(C2CC2)OC)=O)CC2(CCN(Cc3cn4ccccc4n3)CC2)C1 34993,N1(C(CC(=C)Br)=O)CC(CNC(=O)CC(CC)C2CCC2)C(C)C1 34994,C1(NC(c2occc2CNC(c2ccccc2F)=O)=O)Cc2ccccc2C1 34995,O=C1CCN(C(c2ccc(N3CCOCC3)nc2)=O)c2cc(Br)ccc2N1 34996,C1(C2CCN(C(=O)CC(C)C(C)(C)C)C2)(NC(C)=O)CC1 34997,C=CC(C)(CC)C(=O)NCC1(CCNC(=O)C(C(C)C)c2ccncc2)CC1 34998,c1(C(=O)NC(CC=C)CNC(=O)C(C)(C)C)cc(S(N)(=O)=O)c(F)c(F)c1F 34999,c1(C(=O)NC(CCNC(CC2CCC(C#N)C2)=O)(C)C)cc(F)cc([N+](=O)[O-])c1 35000,C1(C2CCN(C(=O)COC(F)(F)F)CC2)(NC(c2c(F)ccc(C)c2)=O)CCC1 35001,Cc1nc(Cl)[nH]c(=NCC2(NC(C3CCC(C(F)(F)F)CC3)=O)COC2)c1Cl 35002,c1(C(C(=O)NCC)N(c2cccc([N+](=O)[O-])c2)CC)cnc2c(c1)c(C)nn2C 35003,C1(C(=O)NC23CC2CN(C(=O)CCc2ccsc2Cl)C3)CCCC1C1CC1 35004,Cc1[nH]c2c(C)c1c(=O)[nH]c1cccc(c1)[nH]c2=O.C(=O)(C(C)C)NC(C)C 35005,C(=O)(CC(C)(C)OC)N(CCCNC(c1csc(-c2cn[nH]c2)n1)=O)CC 35006,C(=O)(C(O)(C1CC1)C1CC1)N(CC(CC)NC(=O)C(C)(C)c1ccsc1)C 35007,Cc1cc(=O)cc(C)n1CCCC(=O)NCC(C)CNC(=O)C(C)n1cnnn1 35008,CCCC(C(=O)N1CC2CN(C(=O)CCCN3CCOCC3)CC2C1)C(C)C 35009,c1(C(C)NC(=O)CSC2C=CC(NC(C3(c4cccs4)CC3)=O)C2)ccccc1 35010,C1(CNC(C(C#C)(C)C)=O)CN(C(=O)CCn2ccnc2)CC(C)(C)O1 35011,CCCC(C)CCCC(=O)N1CC=C(CNC(=O)C(CC)OC)CC1 35012,C1(C(=O)NCC=CCNC(=O)CC2COC3CC2C3)(OC)CCCOC1 35013,N1(C(=O)CC2CCC(F)(F)C2)CCC2CN(C(c3ccc(Cl)cc3Cl)=O)CC2C1 35014,c1(C(=O)NCC2(CNC(=O)CCOCC3CC3)CCC2)occ2c1CCCC2 35015,c1(CC)noc(CC)c1CC(N1CC(NC(c2conc2C)=O)CC1C)=O 35016,C1(NC(C=CSC)=O)CCC2CC1CN2C(=O)CC1CCOC(C)(C)C1 35017,Cc1nc(C(C)C)nc(O)c1C(N1CC2(COC(CNC(C3CCO3)=O)C2)C1)=O 35018,C1(NC(C(C2CC2)SC)=O)CCCC1NC(=O)Cn1ccc(Br)n1 35019,CC(C)CC(F)(F)C(=O)N1C2CCC1CC(CNC(C1CC(C)CO1)=O)C2 35020,C#CCC(C)(C(=O)NCCC1CC1C)NC(c1cc(C#N)cs1)=O 35021,C1(C(N2C(C)CC2)=O)CCc2ncnc(C)c2C1.C1(N2CC(=O)N2)CCCC1.CO 35022,CCCCCCC(=O)N1CC(NC(c2oncc2C)=O)C(C(F)F)C1 35023,C(C1=CCN(C(=O)C(O)CN2CCCC2)CC1)NC(C(COC)O)=O 35024,CC1=C(C(=O)N2CC3(C(=O)NCC(O)CC4CCC4)CC2CO3)CCCO1 35025,CC1C(NC(=O)CCC2CCC(C)O2)CCCN1C(c1cn(C)c(=O)n1C)=O 35026,C(=O)(CC1c2ccccc2C(=O)N1C)NCCCCNC(CC1CC(SC)C1)=O 35027,Cc1ccc(-c2ccc(C(N3CCCC(N4CC(O)C4)C3)=O)cc2)cc1 35028,S(=O)(=O)(c1ccc(=NCCS(=O)C(C)(C)C)[nH]c1)NCc1nc(C)sc1 35029,c1(C(=O)NC2C(CNC(=O)C=CC3CCOCC3)CC2)cc(Cl)cc(F)c1F 35030,Cc1cc(C(N2CC(C)CCC2CNC(c2cn(CO)nn2)=O)=O)c(C)nc1C 35031,C(C)(C(O)C(=O)OCc1nnc(-c2ccc(C(F)(F)F)cc2)o1)OC 35032,C(=O)(C1=CC(C)CC1)NC(C)CCNC(c1ccn(C2CCC2)n1)=O 35033,C12(C(N3CCC(C)(C(=O)NC)C3)=O)COC(C1)C(NC(=O)CC(=O)NC1CC1)C2 35034,CC1CCN(C(C2(CF)CC2)=O)CC1NC(C1CCN(C2CC2)CC1)=O.C(C(F)F)O 35035,CC1CN(C(=O)Cn2cnc(C(F)(F)F)n2)CC1NC(=O)CC12COCC(C1)C2 35036,C12(COC)CC(OC(C)(C)C)(CN1C(=O)Nc1cccnc1SC(F)(F)F)C2 35037,C12(CC(=O)NC(CNC(C(C)(C)F)=O)C(C)(C)C)CC3CC(C1)CC(O)(C3)C2 35038,CCCC(C(=O)NOCc1cn(CCCN(C)C)nn1)N(C)C 35039,c1(C(N(C)CC2(NC(C3CCCCCCC3)=O)CC2)=O)c2c(nn1C)CCSC2 35040,c1(C(N(c2ncc(CCC)cn2)C2CC(N)C2)=O)cc(C(F)(F)F)ccc1F 35041,c1(C(=O)NC(CN(C(C(C)SCCCC)=O)CC)C)cnc(CC(C)C)[nH]1 35042,C1(CNC(c2ccc(COC)o2)=O)CC12CCN(C(c1ccc(F)o1)=O)CC2 35043,Cc1cnc[nH]c1=NCCCC(C)NC(=O)Cc1cnn(C(C)(C)C)c1 35044,c1(NC2C(C)CCN(C(C3CC3c3ccccc3)=O)C2)ncnc2sccc12 35045,C1(C(=O)NC(CCCCC)C)CN(C(C2(O)CCOCC2)=O)CC12CC2 35046,c1(C2C(C(=O)NCCCNC(C(C)(C)C3(C)CC3(F)F)=O)C2)ccc(F)cc1 35047,c1(C(=O)NCC2(CCNC(C3C(OC)C3C)=O)CC2)occc1CN(C)C 35048,N1(C(C2C(CN(C)C)C2)=O)CC2(C1)C(NC(C1CCC1)=O)CCS2(=O)=O 35049,C=CCC(C)(C)CC(=O)NC1CCCC1NC(=O)C=C(C)C1CC1 35050,CCC(CC(=O)NC(CCOCCO)C(=O)N1CC=CCC1)C1CC1 35051,c1(OC)cc(Cl)cc(N)c1C(=O)N(CCO)Cc1sccc1C 35052,C1(C(N(C)Cc2ccns2)=O)CCC(C2CC2)N1C(c1ccc(C#N)s1)=O 35053,c1(-c2cn(CC(N3CCC(C#N)CC3)=O)nn2)ccc2ccccc2n1 35054,CCCCCC(O)C(=O)NCc1cc(-c2ccc(C#N)cc2)nn1C 35055,C1(CN(C(=O)Cc2sccc2C)CC)CCCCN1C(=O)CN1CCC(F)(F)C1 35056,c1(C(N2CCC(CCNC(C(C)CC(F)F)=O)C2)=O)cccc2c1CC(=O)N2C 35057,C1(N(C(CC(=O)NCC#C)=O)C)CCN(C(=O)C(C)CSC)CC1 35058,N1(C(CC2CN(C)C2)=O)CC2CC2(C(=O)N(C2CCCC(O)C2)C)C1 35059,c1(C(C)C)ccc(C(=O)Nc2cccc(NC(=O)CCC3CNC(=O)N3)c2)cn1 35060,Cc1oc(-c2ccccc2F)nc1C(=O)NCC(O)CN(C)C(c1cncs1)=O 35061,C(=O)(NNC(=O)c1ccc(CO)cc1)NC(C)CC(N)=O 35062,Cc1c(CC(=O)NC2CN(C(=O)COCC(C)C)CCC2C)sc2ccccc12 35063,N(C1CCCc2c1cnn2Cc1ccccc1)C(c1cc(C)c(O)c(C)c1)C 35064,C(=O)(C1CCSc2ccccc21)N1C(C)CCN(C(c2cnn[nH]2)=O)CC1 35065,c1(C(N2C(C(N3CCC(C(C)(C)O)CC3)=O)CC2)=O)cc([N+](=O)[O-])n[nH]1 35066,C1(NC(C2CCC(NC(CCC3C(C)C3)=O)C2)=O)CC2CC1CC21CC1 35067,C(CC(C)C(=O)N1CCC(Cc2ccncc2C)CC1)=CC 35068,C(=O)(CC(C(F)(F)F)N1CCOCC1)N1CCC(F)(C(N2CCOCC2)C)C1 35069,O(NC(=O)C(C1CC=CCC1)NC(C1C2CCC(F)C12)=O)CC(C)(C)O 35070,c1(C(=O)OCC2CC(C)OC2C)cccnc1[N+](=O)[O-] 35071,N1(C(C2C(C)C2)=O)CC2(CCC2NC(=O)CCc2cc(Cl)cc(Cl)c2)C1 35072,c1(N2CC(C#N)C(NC(c3c(F)ccc(Cl)c3F)=O)C2)ncnc2cc(Br)sc12 35073,CCCC(C)CCCC(=O)NCC1CN(C(=O)Cc2cc(Cl)n(C)n2)CC1(C)C 35074,CC1CN(C(=O)Cc2cc[nH]c2)CC(C)CN1C(C1CC12CC(O)C2)=O 35075,Cc1cc(C=CC(N2CC(CCNC(=O)CSC(C)(C)C)C(C)C2)=O)on1 35076,C(C(C)S(N)(=O)=O)NC(C1(NC(C(C)=CC=C)=O)CC1(C)C)=O 35077,c1(OC)ccc2ccccc2c1NC(C1CNCCN1Cc1cncs1)=O 35078,C(=O)(CCC(C)(C)[N+](=O)[O-])N1CCC(CNC(C2(CC)CC2(F)F)=O)C12CC2 35079,N1(C(C(COC)OC)=O)CCN(C2CCCN(C(=O)C=C(C)C(C)C)C2)C(=O)C1 35080,C12(C(=O)NC(C)CCN(C)C(c3cccnc3S)=O)CCC(O1)c1ccccc12 35081,C1(NC(C2(CC)CCC2)=O)CN(C(=O)C(C)CSC)CCC1CO 35082,N1(Cc2nc(-c3ccc(CC)cc3)on2)CCC(CC(N)=O)C(F)(F)C1 35083,c1(CC)cc(C(=O)NC2CC2CNC(c2cncc(N)n2)=O)cc(O)n1 35084,CCC(C)C(=O)C(=O)NC1COCCC1C(=O)N(CCC(N)=O)CC 35085,N1(C(CNC(C2C(C)C2)=O)=O)CCC(C(=O)NCC2CC2Cl)(CF)C1 35086,c1(C(=O)NCC2C(N(C)C)CN(C(CC3C(CC)C3)=O)C2)c(Cl)ccnc1C 35087,S(=O)(=O)(c1c[nH]c(=NCCNc2cccnc2)cc1C)NCC1CCN(CC)C1 35088,C12(C(=O)NC(CC=C)CNC(C3CCO3)=O)CC3(F)CC(F)(C1)CC(F)(C2)C3 35089,Cc1cc(C(=O)NC2(CNC(=O)CCSc3nnnn3C)CCOC2)ncn1 35090,c1(C(=O)NC2CCCC(OC)CC2)c(F)cc(Cl)cc1Cl 35091,Cc1c(CNC(C2CC(CNC(C3(O)CCCC3)=O)C2)=O)cccc1F 35092,c1(OC)ccc(F)cc1CC(N1CC(NC(c2cn(C)cn2)=O)C(C)C1)=O 35093,c1(Cn2cc(CCCCNC(C(C)CCN(C)C)=O)nn2)csc2ccccc12 35094,c1(C(=O)NCC2(F)CN(C(c3c(C)c(Cl)ccn3)=O)C2)cncc2c1CCCC2 35095,N(C1CCOc2ccc(O)cc21)C(c1c(C)cco1)C 35096,Cc1ccc2c(c1)C(=O)N(C(C)C(=O)NCCNC(=O)CC1COCCO1)C2=O 35097,N1(C(C2(C#N)CC(C)C2)=O)CC=C(C(=O)Nc2cccc(C#N)c2)C1 35098,n1(CCOC(C)C)nc(Cc2ccccc2Br)nc1-c1cncn1C1CC1 35099,N1(C(CCC(C)C)=O)CC(CNC(=O)C(C2CCCCCC2)C)OC(C)(C)C1 35100,N1(C(c2ccc(C(C)C)cc2)=O)CCCC(C)(NC(C2CCC3CC2CO3)=O)C1 35101,CCCCC(CNC(c1cc(C)cs1)=O)NC(=O)CC(c1ccccc1)N(C)C 35102,C1(NC(CC2CC(C)(C)OC2=O)=O)CN(C(c2ccnc(O)c2)=O)C2(CCC2)C1 35103,Cc1noc(CN(C)C(=O)NCc2ccn(CC(F)(F)F)n2)n1 35104,C(CN=c1[nH]c(=NCC(=O)Nc2nccs2)c2ncccc2[nH]1)C1CC(C)C1 35105,C(CCCC(=O)N1CC(O)CC1C)NC(c1c(CCC)[nH]cc1)=O 35106,C1(C(N2C3CC(NC(C(CCC)C)=O)(C3)C2)=O)CC(C(C)C)=NO1 35107,C1(C(N(CC(C)(C)NC(COCCCC(C)C)=O)C)=O)CCCCC1(F)F 35108,N1(C2CCN(C(CC3C(C)C3)=O)CC2)CCC(NC(C2(N(C)C)CC2)=O)CC1 35109,N1(C(c2c(C)cc[nH]2)=O)CCC(C(C)(O)CNC(c2nocc2Br)=O)CC1 35110,c1(OC)nccc(C(N2CC(NC(c3nc(C)ncc3Br)=O)C(F)C2)=O)c1F 35111,CC1CC(NC(=O)Cc2c(F)cccc2Cl)CN(C(c2cccc(F)c2O)=O)C1 35112,N1(C(CC)C(N)=O)CCC(NC(c2c[nH]nc2C)=O)C(O)C1 35113,C(=O)(CC(C)C(=O)OC)N1CCC(NC(c2cc(CC)ncc2)=O)(COC)C1 35114,c1(NC(c2c(C(C)C)nns2)=O)ccccc1I 35115,c1(OC)cc(C(=O)NC2CC(NC(=O)C(OC)OC)C2)cc(C)c1 35116,C1(C(=O)NC(CC)CNC(c2ccc(C)cn2)=O)CC(O)CN1C(=O)N(C)C 35117,C1(C)(C(N(CC#C)CC=C)=O)CCCN1C(=O)CCn1cc(C(=O)OC)cn1 35118,c1(C(=O)NC2C3CN(C(c4ccc(C(C)=O)cc4)=O)CC32)c(F)cc(F)cc1Cl 35119,N1(C(C(CSC)(C)C)=O)CCC(CNC(C2CCCC(CF)C2)=O)C(O)C1 35120,c1(C(N(CC(CNC(C(C)SCCCC)=O)C)C)=O)ccc(-n2ccnn2)cc1 35121,c1(C(N2C(CC(=O)NCC(C)C3CC3)C3CCCC32)=O)cc2ccccc2o1 35122,CC1CCC=C1C(=O)N1CCC(C)(C)C1CC(N1CCSCC(C)C1)=O 35123,c1(COC)cccc(NC(C2CCC(NC(=O)CC(=O)OC)CC2)=O)c1O 35124,O=C(O)CCC(F)(F)C(=O)Nc1ccc(F)cc1-c1ccc(Cl)cc1 35125,c1(SCCN(C(=O)C(C(=O)OC)OC)C)cc(Cl)cc(Cl)c1 35126,N1(C(CCOCCC)=O)CCCC2CN(C(c3cccc(NCC)c3)=O)CCC12 35127,C=CCC(C)C(=O)N(C1CCCN(C(=O)C=C(CC)CC)C1)CCF 35128,c1(OC)cc(C(C)=O)ccc1OC(=O)CC(C)CC.c12cn(nn1)CCCS2 35129,C1(C(N2CCC(O)(CN(C)C)C2)=O)COCCN(C(=O)CSCC(N)=O)C1 35130,C1(C(=O)NCC2N(C(c3c(OC)nsc3)=O)C3C(C2)C3)Cc2ccccc2S1 35131,C1(NC(C(F)OC)=O)C(C)(C)CN(C(=O)CN2CC3CC3C2)CC1(C)C 35132,CCCCC(F)C(=O)NCC1COC(CNC(=O)Cc2csc(C3CC3)n2)C1 35133,C(=O)(C(F)(F)C(C)O)N.c1(-c2cn(-c3ccc(CC)cc3)nn2)cc(F)cc(Cl)c1 35134,c1(C(N(CCOCCOCCOC)C)=O)ccc(-n2cnnn2)cn1.C1CCO1 35135,C=C=C(C)CC(=O)NC1(CC=C)CCN(C(c2cnn(C(C)CC)c2C)=O)C1 35136,C(CC(C)(C)C(=O)NCC(N1CCOCC1)=O)NC(C=CC=CC)=O 35137,c1(NC(C2C3CN(C(CCCC(C)C)=O)CC32)=O)cc(Cl)c(Cl)cc1C#N 35138,N1(C(c2nc(CC)oc2)=O)CCC2(NC(=O)CCCc3cc(C)no3)CC2C1 35139,c1(OC)ccc(C(=O)NCCCN(C)C(c2c(F)cncc2Cl)=O)c(O)c1 35140,C1(C(=O)NCCC2CCCN2C(=O)CN2CCSCC2)CCCCCC1(F)F 35141,N1(C(C2CC(C)SCC2)=O)CCN(C(=O)Cn2cccc2)CC1CO 35142,c1(NCc2nc3ccc(OC)cc3[nH]2)[nH]c(=NCC2CC2)nc2ncn(C)c12 35143,c1(OC)c(C(=O)NCCNC(c2cnc(C)c(N)c2)=O)cccc1Br 35144,CCCCCCCCC(=O)N1CCCC1CNC(C1CCCCC1C(N)=O)=O 35145,Cn1cncc1CNC(C1(C)CCN1C(=O)COC(C)(C)C)=O 35146,C1(NC(C=C(C)C(C)C)=O)CCN(C(=O)C(C)SC(F)(F)F)C1C1CC1 35147,N1(C(CCN(C(C)=O)C)=O)CCC(CN(C(=O)C(F)(F)c2cnccn2)C)CC1 35148,CN1N=CC(CC(=O)N(CC(CO)(CO)NC(=O)CC2CCCC2)C)C1=O 35149,CCC(CC)CCCC(=O)N1CCC2CN(C(c3nn(C)cc3Cl)=O)C2C1 35150,N1(C(C(C)C(F)F)=O)CCC(C)(NC(c2cc(C3CC3)cc(F)c2)=O)CC1 35151,Cc1ccc(CCCC(=O)NC2CCCC2CNC(=O)Cc2cn(C)nn2)s1 35152,C1(C)(NC(CNS(CCOCC)(=O)=O)=O)CCCN1C(=O)COCCC(C)C 35153,N1(C(c2c(C)noc2)=O)CCN(C(=O)CCn2cccn2)CC1CO 35154,C(=O)(C1=CS(=O)(=O)CCC1)NC1CN(C(C(C2CC2)OCC)=O)CC1(C)C 35155,CCC(C)CC(C)C(=O)N1CCC(F)(CNC(=O)CC2(C(F)F)CC2)CC1 35156,c1(C(=O)Nc2cnn(CC(F)F)c2)noc2ccc(Cl)cc12 35157,N1(C(C2C(OC)C2)=O)CCCC1(C)CNC(=O)CCNC(=O)CC1CCC(=O)N1 35158,C1(CNC(C(N2CC(C)C2)C)=O)(CNC(C2(C)CCSCC2)=O)CC12CCC2 35159,c1(C(=O)NCC2(OC)CN(C(c3cc(C)ncc3C)=O)C2)ccn(O)c(=O)c1 35160,C1(C)(C(=O)NC2CCC(NC(c3ccc(CC)[nH]3)=O)C2)CCC(C)(C)CC1 35161,C(=O)(C(CO)C(C)(C)C)NCc1c(C(=O)NCC(C(=O)NC)(C)C)occ1 35162,C1(NC(c2c(CC)n[nH]c2)=O)CCCN(C(c2ccsc2-n2cnnn2)=O)CC1 35163,c1(C(=O)OC)cc(F)c(Br)c(S(=O)(=O)N2CC(Oc3ccc(C)cc3F)C2)c1 35164,O=C(CCCNC(c1cccnc1)=O)NCC1CN(C(c2cc(Cl)c[nH]2)=O)C1 35165,c1(C(COCC2CCC2)=O)c[nH]c(C(=O)NOCCCN(C(COC)=O)CC)c1 35166,N1(C(C2(COCC)CC2)=O)CC(C2CCCCN(C(=O)CC3COCCO3)C2)C1 35167,c1(C(=O)NC2CC(F)(CNC(c3cn(CC)nc3C)=O)C2)nnc(O)cc1O 35168,N1(Cc2c(C)cccn2)CC2(CN(C(c3ccc(Br)cc3CO)=O)CCO2)C1 35169,C(=O)(CCCCC(=O)NC1CN(C(=O)CSc2nnnn2C)CC(C)(C)C1)NC 35170,N1(C(COCCNC(C(C2CCCCC2)C)=O)=O)CCC2(CC(F)C2)C1 35171,N1(C(Cn2c(C)ccn2)=O)CCC(O)(CN(C)C(C2(C)CCCC2C)=O)CC1 35172,CC(C)CCCOCC(=O)NCC(C)N(C(=O)CC1CCN(C)C1)C 35173,N1(C(C(C)(C)NC(=O)NCC)=O)CC(N(C)C(c2nnccc2C)=O)C(C)(C)C1 35174,C12(C(=O)NC3(CNC(CCOCC)=O)CCOC3)CC(CO)(C1)OC2C 35175,O=C(CCCC(F)(F)F)NC1CC(O)CN(C(=O)COC2CCOC2)C1 35176,c1(OCC)oc2ccccc2c1C(=O)NCC(CC)NC(C1CC2(C1)CC2F)=O 35177,c1(C(N2C(C)CC(=O)N2)=O)ccc2cccnc2c1 35178,c1(C(C(=O)NCCC#N)N(CC)CC2CCCO2)nc2c(s1)CC(C)CC2 35179,CCCCCCC(C)C(=O)NC(C(=O)NC1CC(F)(F)C1(C)C)C(C)C 35180,C12(C(N(CCC(=O)NC(CC=C)C3CC3)C)=O)COCC1C2 35181,N12CCCCC1C2.c1(SCCn2cc(C(C(C)(C)C)O)nn2)ccnc(SC2COCC2)c1 35182,C1(CNC(C2C(COC)CC2)=O)COCC1NC(=O)COc1cccnc1 35183,CN=c1ccc(C(=O)NCC(C2CCN(C(=O)CC3CCC(C)C3)CC2)O)c[nH]1 35184,c1(OC)cc(C2(C(N3CCCC(C)(NC(=O)CCC(N)=O)C3)=O)CC2)ccc1C 35185,C(N=c1nc2sccc2c(N2CCC(SC(F)F)C2)[nH]1)c1[nH]n(C)c(=N)n1 35186,N1(C(=O)CC2CCCC2)CC(C2CCCN(C(=O)C(c3cccc(Cl)c3)O)C2)C1 35187,c1(C(=O)NC(Cn2c(CC)ncc2)C)ccc(Br)cc1N=[N+]=[N-] 35188,c1(NC(N2CCOC(C3CCCOC3)C2)=O)cc(F)c(N2CCC2)c(F)c1 35189,C1(F)(C(=O)OC)CN(C(=O)CONC(c2cccnc2)=O)C1 35190,N1(C(C(CC)OCC)=O)CC(N=c2nc(C(C)(C)C)[nH]s2)CC(C)(C)C1 35191,N1(C(Cc2c(C)nsc2)=O)CCCC2(NC(=O)COCCCC(C)C)CCCC12 35192,N1(C(C2CCN(CC#C)CC2)=O)CC=C(CNC(c2nncn2C)=O)CC1 35193,N1(C(=O)CSCc2ccncc2)CC2CCC(C1CO)N2C(c1ccncc1)=O 35194,c1(C(N2CCC(NC(C(C)OCCCC)=O)C2)=O)ncccc1C(F)F 35195,[N-]=[N+]=NCC(C(=O)NC1(C2CC2)CC1)NC(=O)Cc1cnoc1 35196,C12(NC(=O)COC3CC(F)(F)C3)CCN(C(c3cccc(O)c3Cl)=O)CC1C2 35197,C#CCCC(C(=O)NCC(C)C#N)NC(=O)CCCCCN(C)C 35198,n1(CC)nnc(C)c1C(=O)NC(C)C(C)NC(c1cnn(C)c1C(F)F)=O 35199,C1(NC(C(C)C)=O)CCCC12CCN(C(=O)C(C)CS(C)(=O)=O)CC2 35200,c1(OCC)ccc(Br)c(-c2nnc(CCC(N3CC(=O)NCC3C(C)C)=O)o2)c1 35201,O=S(=O)(c1cccc(F)c1F)N1CCC(OCc2ccc(F)cc2)CC1 35202,c1(C(=O)OCC(=O)NC(C2C(C)CCC2)=O)c[nH]nc1[N+](=O)[O-] 35203,N1(C(c2cnc(COC)s2)=O)CCN(C(=O)CC2CN(C)C2)C(C)CC1C 35204,N1(C(COCCC=C)=O)CC2(CC2)CC1CN(C(=O)CSCCC(F)(F)F)CC 35205,C(=O)(C(C)(C)CCOC)NC1CCCC(NC(C2(COC)CC(=C)C2)=O)C1 35206,Cn1ccc(C(N2CC(C(=O)NCC=CCl)CC2(C)C)=O)cc1=O 35207,C1(C(=O)NCC2CCN(C(CC3C(C)(C)C3)=O)CC2)CCOC2(CCOCC2)C1 35208,CC1(C)CC(O)(C(=O)NCC(C2CCCC2)NC(=O)CC2CCCOC2)C1 35209,C1(C(=O)NCc2cc(C(=O)NCC3(C)CC3)n[nH]2)(OC)CCC(C)C1 35210,Cc1cc(F)c(C(N2CC3CN(Cc4cncc(C)n4)C3C2)=O)c(F)c1 35211,Cn1nc(C(=O)NC2CCCC2NC(C2CCC3CC23)=O)c2c1CCC(C)(C)C2 35212,N1(C(C(CC)C)=O)CC2CCC(C(=O)NCCc3ncn(C)n3)(C2)C1 35213,Cc1nccc(C(=O)NCC2(NC(=O)CNC(C3CCCCC3)=O)CCOC2)c1N 35214,N1(C(C)C)CCCC1C(N1CC(C(C)NC(=O)Cc2nccn2C)C1)=O 35215,c1(CC(=O)NC2CN(C(CC(c3c(C)n[nH]c3C)C)=O)C2)c(F)cccc1Cl 35216,S(C1CCc2c(F)cc(F)cc21)C(=O)Nc1cccc(C)c1 35217,C1(NCC)CC2(CCC(C(N3CC4CCN(C(=O)OC(C)(C)C)CC4C3)=O)CC2)C1 35218,C(CC(CC)C(=O)NCCN(CCCN(C)C)C(c1cc(F)n[nH]1)=O)=CC 35219,CCCCCC(C)CC(=O)NC(CNC(=O)CN1C(=O)C(C)C(C)C1=O)CC 35220,CCC(C)C(O)C(C)C(=O)N1CCC(NC(C2CCC3CC23)=O)C1 35221,CCC(C)(C)C(C)CC(=O)NC1(CNC(=O)C=Cc2cc(Cl)ccc2Cl)CCC1 35222,C1(CNC(C2CCC(CC)O2)=O)CC(NC(c2cnc[nH]2)=O)CC1O 35223,N1(C(CC2CCCN(C(C)C)C2)=O)CC2CN(C(=O)Cc3cnnn3C)CC2C1 35224,N1(C(CC(COC)C)=O)CCCCC(CNC(=O)C=C2CCC(C)(C)CC2)C1 35225,N1(C(c2c(C)cccc2F)=O)CC(NC(=O)Cc2cc[nH]n2)CC2(CC2)C1 35226,CCCCCCC(F)C(=O)N(C)CC1CCCN1C(=O)CC12COC(CF)(C1)C2 35227,c1(C(=O)NCC2N(C)CCN(C(=O)C=C3CCC3)C2)cnn2ccn(C)c12 35228,C=CCCCCC(=O)N1CCC(OCC(=O)NC(CCF)C(=O)OC)C1 35229,C=CCC(CC)C(=O)NCC1CC(O)CN1C(=O)Cc1ccsc1 35230,c1(NC(c2nnnn2CC2CCOC2)(C2CC(=C)C2)C)cc(CO)ccc1OC 35231,Cn1nccc1C(=O)NCCC(O)CNC(c1c[nH]c(Br)c1)=O 35232,CC1CCN(CCC(=O)NCCCCCCNc2ccnc(OCCO)c2)CC1 35233,CCC(CCCC(=O)N1CCCCC1CCO)NC(=O)C(C)(C)SC 35234,Cc1nn(C)c(C)c1Cn1cc(CCNc2nccc(OCCO)c2F)nn1 35235,N(C(=S)N1CC(CO)CC(C)C1)c1ccc(OC)c(Cl)c1 35236,CC(C)CC(CNC(=O)C1=CCCCO1)C(=O)NC(C1(O)CCCC1)(C)C 35237,S(=O)(=O)(c1cc(NC(=O)NC2(C(c3cnsn3)=O)CC2)co1)NC(C)(C)C 35238,C1(C(N(CCNC(=O)C(C)(CC)C(F)F)CC)=O)CCc2ncnc(C)c2C1 35239,C(C1=NOC2COCC12)NC(CCN(C(=O)CCCn1ccnn1)CC1CC1)=O 35240,CC1CCC(CNC(=O)Cc2cc[nH]c2)N(C(=O)CN2CCC(CO)CC2)C1 35241,Cc1cccc(-c2cccc(NC(C3CC(C)N(Cc4ccccc4)C3)=O)c2)c1 35242,c1(C(=O)NCCOCCCNC(C2C(C)C2C)=O)cc(C2CC2)cnc1Cl 35243,C12(CNC(c3c(CC)noc3)=O)CCCN(C(c3c(C)coc3C)=O)C1C2 35244,c1(C(N2CC3(CCN3C(C3(F)CCCCC3)=O)C2)=O)ccc(Cl)c(F)c1F 35245,c1(OCCN(C(=O)C(=O)N(CCC(F)(F)F)CCN)C)ccc(Br)cc1 35246,C1(CC(NCP(OCC)(C)=O)=O)CN(C(c2cc(COC)on2)=O)CC12CC2 35247,N1(C(c2cc(C)ncc2)=O)CC2CN(C(c3ccc(Cl)cc3F)=O)C2C1 35248,N1(C(C(CO)N(C)C)=O)CCC2(C1)CN(C(=O)CS(=O)(=O)C(C)(C)C)CCO2 35249,N1(C(c2cnc(C(C)C)s2)=O)CC2CC1C2NC(=O)C(C)C1CC1 35250,c1(OCC)cc(C(=O)NCCC2CN(C(c3csnc3C)=O)C2)[nH]n1 35251,N1(Cc2c(OC)cco2)CCCC(NC(c2cnc(Cl)cc2I)=O)CC1 35252,C(=O)(C(C)(C)CC(F)F)NCc1c(C(=O)NCC(C#C)OC)con1 35253,c1(CN(C(=O)Nc2ccccn2)CC2CCN(C(=O)C(F)(F)F)C2)ccccn1 35254,C(=O)(C(O)C(F)(F)F)N1CCC(CCC2N(C(C=CC)=O)CCC2)CC1 35255,c1(OC)ncnc(C)c1C(=O)NCC1(CNC(=O)Cc2ccc(Br)cc2)CC1 35256,c1(C(N2C(CNC(COCC)=O)CC(C)CC2)=O)n[nH]c2cc(C)ccc12 35257,N1(C(C2(COC)CCC2)=O)CC2CCC1C2NC(=O)CCc1ccc(Cl)cc1 35258,C1(C(N(CC)Cc2occc2C)=O)CN(C(c2ccnn2C2CC2)=O)C(C)(C)C1 35259,C1(NC(C(CC=C)C)=O)CN(C(c2cnn(C)c2C(C)(F)F)=O)CC(F)(F)C1 35260,C(C1OCc2ccccc21)N(C1CC(n2nnnc2C(F)(F)F)C1)CC 35261,C1(NC(CCCCNC(C)=O)=O)CC2(C1)CN(C(=O)CC1C(C(C)=O)C1(C)C)C2 35262,c1(OC)ccc(C)nc1C(=O)NC1CC1CNC(c1ccc(C(C)C)cc1C)=O 35263,C1(NC(C2C(C)CCS2)=O)CCC(NC(=O)C(C)(C)c2ccc(Cl)s2)CC1 35264,c1(C(=O)NCC2CCCN(Cc3c(O)cccc3O)C2)cccc2sccc12 35265,N1(C(c2c(CC)[nH]cc2)=O)CCCC(NC(c2csc(S(N)(=O)=O)c2)=O)C(F)C1 35266,N1(C(C(C(CC)C)O)=O)CCCC2(C1)CN(C(c1nc(O)[nH]c(=O)n1)=O)CCO2 35267,c1(COC)cc[nH]c1C(=O)NC1(CNC(=O)C(C)NC(C2CCC2)=O)CCCC1 35268,C(c1cccc(O)c1)=CC(N1C2CN(C(c3cccnc3C(F)(F)F)=O)CC21)=O 35269,c1(CNCC2(C(=O)NC3C(CC)C3)CC2)sccc1Cl 35270,N1(C(C(c2ccc(Cl)s2)C)=O)CCC(NC(=O)Cc2ccc(O)c(Cl)c2)CC1C 35271,Cc1cc(C)n(CCC(=O)N(CC(C)(C)Cn2cc(C3COC(C)(C)C3)nn2)C2CCCN2)n1 35272,c1(CCN=C(NCCOC(CC)C)NCC2CC(F)(F)C2)ccc(S(N)(=O)=O)cc1 35273,c1(C(N2CC3(CN(C(c4ccc(C)s4)=O)C3)C2)=O)cc(N)cc(C)c1F 35274,c1(-c2ccc(N3CCN(c4ncc(Br)cn4)CC3)nc2)cccc2ncsc12 35275,CCC(C(=O)NCC1CC(C)CN(C(=O)C(n2nccc2C)C)C1)C(F)(F)F 35276,CN1CCN(C(C2CC(O)CN2C(=O)C(F)C(C)(F)F)=O)CC12CCC2 35277,N1(CC(C2CC2)OCC)CCC2(CCCCN(C(c3cn(C)nn3)=O)C2)C1 35278,C1(NC(C(c2ccc(F)cc2)OC)=O)CC12CC(NC(c1ccncc1F)=O)C2 35279,c1(CC)nnc(C(=O)NCC2(NC(C3CCOC3CC)=O)CC2)s1 35280,C(=O)(C(CC(N)=O)SC)NC(C1(OC)CCN(C(c2ccc(C(F)F)o2)=O)C1)C 35281,c1(OC)ccc(C(c2cccs2)NC(=O)NC(CCO)CC(C)C)cc1OC 35282,C(N=c1cc(NCCc2ccn(C(C)C)n2)nc[nH]1)C1CN(CCC)C(=O)C1 35283,C(=O)(CCCCN(C)C)NCC1C(NC(COC(C)=O)=O)CCC1 35284,CCCC(C(O)C(=O)N1CCc2c[nH]nc2C1)NC(=O)C=CC(F)(F)F 35285,N1(C(c2nc(CC)[nH]n2)=O)CC(NC(C2(C(C)C)CC2)=O)CC1C 35286,N1(C(C(CC)C#N)=O)CC(O)(C2CCN(C(=O)Cc3cn4ccsc4n3)CC2)C1 35287,CC(C)(C(=O)NCCC1CC(NC(=O)C(C2CC(F)(F)C2)O)C1)C(F)(F)F 35288,N1(C(C2N(C(CC3CCC(=O)N3)=O)CC2)=O)CCOCC(CO)C1 35289,c1(C(N2CC3C(N(C(C(C)NC(N)=O)=O)C)C3C2)=O)cc2cc(F)ccc2o1 35290,C(C)(C)(CCCC(=O)NC(C(C)C)c1nc[nH]n1)NC(c1ccc(OC)cc1)=O 35291,c1(NC(C2C3CN(C(C4CCC(C)CO4)=O)CC32)=O)nc2cc(F)ccc2s1 35292,C1(CC)CCCCCCN1C(C1CCOCCN1C(C1CCSCC1)=O)=O 35293,N1(C(c2cncc(C(C)=O)c2)=O)CC2CC(C1)N(C(=O)CC1CC=CCC1)C2 35294,C1(C(=O)NC(c2nocc2C(=O)NC(c2cccc(F)c2)C)C)CCCCC1O 35295,C12(CNC(C3(C)COCCO3)=O)CCC1CN(C(c1cc3occc3[nH]1)=O)C2 35296,C12(CNC(CC3CC(=O)C3)=O)CCC(C1)N(C(=O)CCCCN1CCCC1)C2 35297,c1(SCCC(=O)NC(CN(C(C(C)NC(=O)OC)=O)C)C)ccccn1 35298,C(CC(=O)NC1CCN(C(c2nc(Br)cnc2N)=O)C1)(C(F)(F)F)OC 35299,Cc1cc(C(C(=O)NC2CCOC2)N(C)C(c2ccc(Cl)c(Cl)c2)C)c(C)nn1 35300,C1(C(=O)NCC2C3CN(C(CCCCOC)=O)CC32)COc2ccc(O)cc2O1 35301,N1(CC(=O)NC(C)CN(C(=O)CCc2cscc2Br)C)CCCCCC1 35302,N1(C(c2c(C)nc(CC)s2)=O)CCC(NC(=O)CCN(CC)CC)C(CO)CC1 35303,c1(CC(=O)NC(C(C)C)CCN(C)C(C2CC(C)(C)C2)=O)ccccc1[N+](=O)[O-] 35304,Cc1cc(Br)ccc1CCNC(C1CC2CC2N1C(=O)CNC(=O)CC(C)C)=O 35305,c1(N(C)C)ccc(C(N2CCC2CNC(c2cnc(Cl)cc2N)=O)=O)c(F)c1 35306,c1(C(N2C3CN(C(=O)Cc4c(F)cccc4F)CC32)=O)cccc2c1OCO2 35307,c1(C(=O)NC(CC(C)NC(C2CC(CC)C2)=O)C)ccnc(C(F)F)c1 35308,c1(OC)cc(C(=O)NC(CNC(=O)CN2CC(C)C2)C2CC2)[nH]n1 35309,c1(NCC(C)(C)C)ccc(S(=O)(=O)NC2C(C)SCC2)c(Br)c1 35310,C12(C(=O)NC3(C(=O)OCC)CCC3)CC(C)(CN1C(c1nc(C)oc1C)=O)C2 35311,C1(C(=O)NCC23OCC(NC(C4(C)CC4)=O)C(C2)C3)COc2cc(Cl)ccc2C1 35312,CC1CNc2c(C(=O)NCCN(C)C(C3CCC(N=[N+]=[N-])CC3)=O)cnn2C1 35313,C1(N(C2CCOC2C)C(c2cccc(OC(C)=O)c2)=O)CCNCC12CC2 35314,C(C1CN(C(=O)CCN(C)CC2CC2)CC1C(=O)Nc1ccncc1)=CC 35315,O=c1c(-c2nc(CCO)nn2C(c2cccnc2)CCO)c[nH]cc1F 35316,N1(c2c(C(C)=O)cccn2)CCC(NC(=O)C(C)n2cnnn2)C(O)C1 35317,Cn1nc(C(N2CCOC(CC(=O)NCCOCC3CCCC3)C2)=O)cc1Cl 35318,c1(C(C)(C)C)cc(C(=O)NCC(O)CNC(=O)CCOCC(F)(F)F)cs1 35319,C1(C(=O)NC(C2CCOCC2)C#C)(CC)CCN(C(=O)CCc2conc2C)C1 35320,N1(C(C(CC)F)=O)CC2CCOC2(CNC(c2cc(OC(C)C)ccc2Cl)=O)C1 35321,N1(C(c2c(CC)ncs2)=O)C(CNC(c2cc(C(C)C)on2)=O)CC2CC12 35322,C(=O)(C1CCCc2cn(C(C)C)nc21)NCC(CNC(c1c(C)nns1)=O)F 35323,c1(OC)ccc(C(C)=CC(=O)NC2CCC2NC(c2csc(CO)n2)=O)cc1 35324,CC(C)C(C(=O)NC1CN(C)CCN(C)C1)C(C)NC(C1CC=CC1)=O 35325,c1(CC(=O)NC2CCCCN(C(C(CCCC)=O)=O)C2)csc2cccc(F)c12 35326,C1(NC(CCC(=O)NC)=O)(CNC(c2cccnc2N)=O)CCCCC1C 35327,N1(C(C2CCCSC2)=O)CCCCC2(CCN(C(C3CC3C(F)F)=O)C2)C1 35328,c1(C(=O)NC2C(CNC(=O)Cn3cnnc3O)C2)cc2ccc(Cl)c(F)c2[nH]1 35329,c1(C(=O)NC2CCCN(C(c3noc(CC)c3C)=O)C2)ccc(Cl)cc1OC 35330,Cc1ccc(S(=O)(=O)NC(C(Cc2ccccc2)N2CCOCC2)=O)cc1C 35331,C1(CNC(c2cnn(C)n2)=O)C(C2CC2)CCN1c1ncnc(Cl)c1F 35332,CC1(C)C(CC(=O)NCCC2COCCO2)CCN1C(C1CCCCCC1)=O 35333,C(C(C(=O)NCC1(NC(C2CC2(F)C(=O)OC)=O)CC1)N(C)C)OCC 35334,N1(C(C2CC(OCC)C2)=O)CC2CC2C1C(=O)NC(C)CCCO 35335,c1(C(=O)NC)ccc(CC(=O)NCCCOCCNC(C2CCCCS2)=O)cc1 35336,c1(C(=O)NC2CN(C(C3(C(C)C)CNC(=O)C3)=O)C2)nn(C)c(Cl)c1Cl 35337,c1(NCC2CN(C(c3[nH]cc(CC(C)C)c3)=O)CC2C)ncnc2c1nnn2C 35338,CON(C(=O)CCCCN(C)C(C1(C#N)CC=CC1)=O)C1CCOCC1 35339,N1(C(CC2CC(=C)C2)=O)CC2CCN(C(c3cc(N)cc(OC)c3OC)=O)C2C1 35340,c1(C(N(CC(CC)NC(C2(c3cccs3)CC2)=O)C)=O)cnc(O)n(C)c1=O 35341,O=C(C1=CCCSC1)NC1CCN(C(c2ncc(F)cn2)=O)CC1CO 35342,C12(C(=O)NCC3C(C(=O)OCC)CCO3)CC3CC(C1)CC(F)(C3)C2 35343,Cc1c(C(=O)N(C)CCC2CCCCN2C(=O)C#CC2CC2)cccc1CO 35344,c1(C(=O)NC(CCCC)CNC(c2ccco2)=O)cccc(OC)c1OC 35345,C(CC(=O)NC(=O)CC1CCCC1)NC1C(CNC(C)=O)C1 35346,c1(C(=O)NCCC(=C)CNC(c2cc(Br)c(C)o2)=O)cccc(CC)n1 35347,c1(C(=O)NCc2ccc(C#N)nc2)cc(F)c(Br)cc1F 35348,C12(C(=O)NCCN(C(CCCCSC)=O)CCOCCO)CCC(F)(CC1)C2 35349,C(=O)(C1=NOC2COCC12)N1C(C)CN(C(C(C)=NOCC#N)=O)C(C)C1 35350,Cc1ccc(NNC(=O)CNC(=O)CC2CCC(C#N)C2)cn1 35351,N1(C(c2ccc(NC(C)=O)nc2)=O)C2CCC1CN(C(=O)COC1(C)CCC1)C2 35352,c1(C(N2C(CN(C(=O)COCC3CC3)C)CCC2)=O)ccc(F)c2ccncc12 35353,C=CC(C)(O)CC(=O)NC1C2CC(NC(=O)Cc3nc[nH]n3)CC12 35354,c1(C(=O)NC(CNC(C2(C)CCC(C)C2)=O)C)cnn2ccccc12 35355,C1(C(N(CCO)CC)=O)CC12CCN(C(=O)Cn1ccnc1C)C2 35356,c1(C(N2CCCC(CN(c3ncncc3Br)C)C2)=O)cncc2c1CCCC2 35357,N1(Cc2ccc(CNC(=O)Cc3ccc(I)cc3)cc2)CCCS1(=O)=O 35358,CC1(F)CCC(C(=O)NC2CCCC2NC(c2ccc([N+](=O)[O-])o2)=O)CC1 35359,CC1(C)CCC(CO)N(C(=O)C(c2cc(F)c(F)c(F)c2)O)C1 35360,c1(C(=O)NCC2N(C(CN(S(CC)(=O)=O)C)=O)CC(O)C2)cccc(F)c1C 35361,CC(C)(C)C(O)C(=O)NCC1CN(C(c2ccnc(C(F)(F)F)n2)=O)CC1(C)C 35362,Cn1nc(C(=O)NC2CCC(NC(c3coc(CC4CC4)n3)=O)C2)cc1C#N 35363,N1(C(C2(CC)CC2)=O)Cc2cccc(CNC(=O)Cc3cn[nH]c3)c2C1 35364,c1(OCC)ccc(S(=O)(=O)NC(=O)Cc2cc(Cl)cs2)cc1[N+](=O)[O-] 35365,N#Cc1ccc(C=CC(=O)NC2CCCN(C(c3cn4ccnc4s3)=O)C2)cc1 35366,CC(C1COc2ccccc21)n1ccnn1.c1(NC)cc(CO)ncn1 35367,Cc1nc2cc(C(N3CC(NC(C4CNC(=O)N4)=O)C3)=O)ccc2n(C)c1=O 35368,CSC1=C(C(=O)NCC(C2CC2)N(C(=O)C(CO)c2ccccc2)C)CCCC1 35369,C1(C(=O)N(CCNC(c2c[nH]cc2C2CC2)=O)C2CC2)(COC)CC1(F)F 35370,C1(NC(=O)NCC(C)OC)CCN(C)C2(CC2)C1 35371,C1(NC(C(CC)NC(C)=O)=O)CCN(C(=O)CSCCC(C)C)C1C 35372,c1(C(N2CC3C(C(=O)NCCC(=O)OC)C3C2)=O)c(OC)cc(NC(C)=O)cc1I 35373,c1(C(=O)NCCCN(C(c2csc(C)c2)=O)CC)cc(C(C)(C)C)n[nH]1 35374,C1(NC(N(CCOC)CC2COC2)=O)C2CCC(C2)N1C(=O)OC(C)(C)C 35375,C12(C(=O)NCC(C)(C)CNC(C3(CO)CC3(F)F)=O)CC=CC(C1)OC2 35376,C=Cn1nccc1C(N1CCSCC1C(=O)N(C(CC)C1CC1)C)=O 35377,c1(C2C(C(N3C(C(=O)NCCC(=O)O)CC3)=O)C2)ccccc1OC(F)(F)F 35378,Cc1ncncc1C(=O)NCCn1cc(CNC(C2CC2(F)Cl)=O)nn1 35379,N1(CCNC(c2c(C)occ2)=O)CCC(NC(c2c[nH]c(=S)cn2)=O)CC1 35380,C1(NC(C(C)C2(O)CCC2)=O)CCCCCC1NC(c1cc(F)ccc1F)=O 35381,CC1CC(C(=O)NC2C3CCC2N(C(=O)Cc2ccon2)C3)=NO1 35382,C(CCC1CC1)(C(=O)NCC1(CNC(COCCCOC)=O)CCCO1)OC 35383,C1(NC(C=CC(=O)OCC)=O)C2CC(O)C1N(C(=O)Cc1csc(NC=O)n1)C2 35384,CC1(CNC(=O)C=Cc2ccco2)CN(C(=O)CCN2CCC(F)C2)CCO1 35385,C(=O)(C#CC(C)(C)CNC(C1(C)CC1(C)C)=O)NC1C(C)COC1 35386,CCCN=c1[nH]c2c(c(=NC(C)c3ccc(Cl)cc3Cl)[nH]1)CSC2 35387,c1(C(=O)NC2C(NC(=O)Cc3ccnnc3O)CCCC2)ccc([N+](=O)[O-])o1 35388,N1(C(C2(CC)CCNC2=O)=O)CCN(C(c2cc(=O)c(OC)c[nH]2)=O)CC(O)C1 35389,N1(C(C=CC)=O)CCC2(CC1)CC(NC(=O)C(C)Sc1nnnn1C1CC1)CO2 35390,CCC(C)(CCNC(=O)C(F)C1CCCC1)NC(c1ccsc1OC)=O 35391,C(=O)(C(C(C)OC)N(C)C)NCC1OCC(C(N(CCC#C)C)=O)C1 35392,C(C(C)(COC)C(=O)N(C(C)(C)CC(=O)NC(C1CCCO1)C)C)OC 35393,c1(C(C(N2C(C(N)=O)CC2)=O)NC(c2ccco2)=O)ccc(Cl)cc1Cl 35394,C1(C(N2CCC(CNC(CCS(C)=O)=O)C23CC3)=O)COc2cc(F)ccc2C1 35395,N1(C(c2cc(OCC)cc(F)c2)=O)CC2(CC(NC(=O)Cc3ccsc3)CO2)C1 35396,c1(C(N2CCC(N(C(=O)CS(=O)(=O)NC)CCC)CC2)=O)ccc2nccn2c1 35397,C1(OC)CC(NC(c2ccccc2C(N)=O)=O)CN(C(=O)CNC(N)=O)C1 35398,c1(C(=O)NCCC2(O)CN(C(C(COC)O)=O)C2)cccc2c1CNC2=O 35399,c1(NC2CCN(C(CC3C(=O)NC(=O)N3)=O)C2)ncnc2c1CCC2 35400,CC1C2C(CCN2C(=O)C=CCN2CCCC2)CN1C(=O)CCOC1CCOC1 35401,c1(C(N2CC(C=C)(CC(=O)NCCOC3CCOC3)C2)=O)ccc([N+](=O)[O-])[nH]1 35402,C1(C(=O)NC(C(C)NC(C2CC2c2cccc(F)c2)=O)(C)C)CCCC(=O)N1C 35403,C(=O)(C1=CC2CCCCC12)N(C)CC1CN(C(=O)CC(=O)OC(C)(C)C)CCO1 35404,c1(C(=O)NC2CC3CCC2N3C(=O)CC2CCOCC2)ccc(C(F)F)c(F)c1 35405,N1(C(c2cc(C)ncc2C)=O)CC2CCCC(C1)N2C(c1cccc(N)c1O)=O 35406,C1(C(=O)N)CCC12CCOCC2.N1(C(N(C)C)=O)CCCC(C(=O)NC2(C)CC2)C1 35407,C(=O)(C1CCCn2cnnc21)NC1C(NC(=O)CCN2CCCS2(=O)=O)CCC1 35408,C(=O)(C1CCCc2sccc21)NCC(CNC(c1c(CC)cccc1CC)=O)C 35409,N1(C(C(C)SCCCC)=O)CC(O)CC1CNC(=O)C(N1CCSCC1)C 35410,N1(C(C(C)Sc2nncs2)=O)CCn2c(nc3ccccc23)C1 35411,C1(CC(=O)NCC2CCCN2C(c2ncoc2-c2cccs2)=O)CCCS1(=O)=O 35412,C1(C(=O)NCc2ccc(C(F)(F)F)cc2)CCCN(C(C2(C3CC3)CC2)=O)CC1 35413,c1(NC(C2CN(Cc3c(Br)cn(C)n3)C2)=O)n[nH]c2c1CS(=O)(=O)C2 35414,N1(C(Cc2ncc(CC)[nH]2)=O)CC(CCNC(=O)CC(=O)NC2CC2)OC(C)C1 35415,C(C(C(F)(F)F)N1CCN(C(=O)CC2C=CCC2)CC1)NC(CN(C)CCO)=O 35416,c1(C(=O)NCC(c2ccccc2F)OC)cc2c(Cl)cncc2s1 35417,C1(C(N2CCC(CN(C(=O)CN3CCC(C)(C)C3)C)CC2)=O)CCCCC12CC2 35418,c1(C(=O)NCCC(C)NC(c2ccc(Cl)o2)=O)oc2ccccc2c1CO 35419,C(=O)(CCCCCN(C)C(C12C=CC(CC1)C2)=O)NCc1c(C)cc(C)s1 35420,C1(C(N2CC(C)(NC(c3cn4c(n3)CCC4)=O)C2)=O)CCC(S(C)(=O)=O)CC1 35421,C(=O)(C(F)C(F)(F)F)N(C(CC)CNC(=O)CC1CCS(=O)(=O)C1)C 35422,c1(CCC)ccc(C(=O)NC2COCCC2NC(C2CC(F)C2)=O)cc1[N+](=O)[O-] 35423,C(=O)(CC(O)C(C)(C)C)NC1CCC(NC(C2ON=C(C)C2)=O)CC1 35424,CCCCC(C(=O)NCC=CCSC)NC(=O)CCC(N)=O 35425,c1(CN(C2CCN(C(=O)CSC3CC3)CC2)C)nnc(-c2ccccc2)n1C 35426,c1(C(N2CCCC(CC(=O)Nc3nccc(C)c3)C2)=O)cc(Br)cnc1O 35427,c1(C(=O)NC2CN(C(C3(O)CCOC3)=O)CC2O)cc(F)cc(Cl)c1 35428,N1(C(C(C)(C)SC)=O)CCN(CCN(C(=O)C=Cc2cocn2)C)CC1 35429,c1(C(N2CCCCC(NC(=O)Cc3cn[nH]c3)CC2)=O)cccc2nsnc12 35430,C(=O)(C1=C(Cl)CCC1)NC(C1CCC1)CNC(C(C)Cn1cccn1)=O 35431,c1(C(N2CCN(C(=O)CC3CC(F)C3)C(C3CC3)C2)=O)ccc2c(c1)COCO2 35432,CCCC(C)(O)CC(=O)N1C2CCC(C2)C1C(=O)NCCCc1ccccc1 35433,N1(C(CCC(C)C)=O)CCOCC2(COCCN2C(=O)C2=CC3CCCC23)C1 35434,c1(CC)ccc(C(=O)NC2CCC(NC(C3(F)CCC3)=O)C2)[nH]1 35435,C(C(CC(C)(C)C(=O)OC)NCc1cn(-c2cc(C)cc(C)c2)nn1)OC 35436,C12(CNC(C(C(C)C)C)=O)CCC(CN(C(=O)CCCc3n[nH]c(=N)s3)C1)C2 35437,Cc1[nH]c(C(=O)NCCCO)c(C)c1C(=O)Nc1cnc(Cl)cn1 35438,C(=O)(N1CC(C)(O)CO1)C1C(C(C2(C)CC2)C)C1.C(=O)(C(C)(C)C)NC 35439,C1(S(N)(=O)=O)(C(=O)NCCNC(C(COc2c(CC)cccc2)C)=O)CCCC1 35440,c1(OC)cnc(F)cc1C(=O)NCC(C)(CO)NC(=O)C=Cc1ccc(O)cc1 35441,Cc1cccc(C(N2CC(CC(C)NC(=O)COC3(C)CCC3)C2)=O)c1Cl 35442,C(=O)(C1=NOC2(CCN(C(C3CCSCC3)=O)C2)C1)Nc1cc(C2(C)CC2)no1 35443,N1(C(C(C)n2cnnn2)=O)CCN(C(=O)C#CC2CCC2)C(CC(F)F)C1 35444,c1(C(=O)NC(CC)CNC(=O)CCc2ccc(F)nc2)cncc2cccnc12 35445,C1(C(=O)NCC2(NC(c3cc[nH]c3)=O)CCC2)CC12CCSCC2 35446,C(=O)(C(O)C(C)OC)N(C1CCN(C(C2(CF)CCC2)=O)CC1)CCC 35447,c1(C(=O)NC2CC3CN(C(CCC(N)=O)=O)C2C3)ccc(S(=O)(=O)NC2CC2)o1 35448,C#CC1(O)CN(C(=O)CN(C(=O)CC2CC3(CCC3)C2)C2CCC2)C1 35449,C1(CC)C(C(=O)NCC2(O)CCN(C(c3ccc(CO)cn3)=O)C2)CCN1C 35450,c1(C(C)=O)ccc(C(N2CCC(C3CCCN3C(c3csc(CO)n3)=O)C2)=O)o1 35451,c1(CC)nn[nH]c1C(=O)N(C)CC1(NC(=O)C(COC)OC)CC1 35452,c1(C(=O)NCC(CC)NC(=O)CCC(C)OC)ccc(N)c(CC(C)C)c1 35453,C(=O)(CCCCN(C)C(C1CC(F)C1)=O)NC(c1nnc(C)o1)C 35454,C(=O)(C1=NNC(=O)C1)NCC(CC(=O)N(C(CC(CC)C)C)C)O 35455,c1(CNC(C(C(C)O)NC(=O)CC(C)(C)O)=O)ccc(C#N)cc1 35456,c1(C(N2CCC(NC(c3ccccn3)=O)CC2C2CC2)=O)cncc2sccc12 35457,c1(C(=O)NCC(CC2CN(C(C3C(C)CCCC3)=O)C2)(C)C)nccc2occc12 35458,CC1(C)CC2(CC2C(=O)NCC2(NC(c3ccc(F)c(C(F)F)c3)=O)CC2)C1 35459,C(=O)(CCC(C)(C)F)NCC(CCNC(C1N(C(CC(C)C)=O)CCCC1)=O)O 35460,C1(CNC(=O)CSc2ccsc2[N+](=O)[O-])CCN(C(C2CC2F)=O)C12CCC2 35461,c1(CC(=O)NC(C2CCCN(C(=O)CC3(O)CC3)C2)C)ccc(F)c(F)c1 35462,C1(C(N2CCC(NC(C(CC)=CC)=O)C(C)C2)=O)CCCC2CCCN12 35463,CC1(C)CCCC(C(=O)NC2CCCC23CN(C(c2snc(Cl)c2Cl)=O)C3)CC1 35464,CC(C)(CCN=c1nc(-c2ccccc2)[nH]s1)NC(=O)Cn1cc(Cl)cn1 35465,c1(CC(C(=O)NC2CC(CNC(C3CC(OC)C3)=O)C2)C)ccc(F)cc1 35466,N1(C(CNC(=O)OCC=C)=O)CCC(C)C(NC(=O)C=CCOC)C1 35467,N1(CC)C(=O)CCC1CC(=O)N(C)CCOCCCNC(=O)CN1CSCC1=O 35468,C1(C)(CCC(=O)NCCCN(C(C)C)C(C2CC(F)(F)C2)=O)CCC(=O)N1 35469,n1(CCC(=O)NC2CCC(NC(c3ccc(CC)[nH]3)=O)C2)cc(Br)c(C)n1 35470,O=C1CCC(=O)N2CC(C(F)C2)N1.c1(C(N2CCCC2)=O)ccnn1C1CCC1 35471,C12(C(=O)NC3C(NC(CSCCC#N)=O)COCC3)CC3CC(CC(C3)C1)C2 35472,Cn1cc(C(C(=O)O)NC(=O)CN2CCC2n2cc(-c3cnn(C)c3)nn2)nn1 35473,c1(C(=O)NC2CC(O)(CNC(=O)CC3CCCS3(=O)=O)C2)cc2c(s1)CCC2 35474,CC(C)S(=O)(=O)CCCN1CC=CC(NC(c2coc(Cn3cccn3)c2)=O)C1 35475,C(=O)(CC(C)(C)NC(C1CCC(F)CC1)=O)NC(C=C)C1CCC1 35476,C=CC1CN(C(=O)Cn2cc(C3CCC3)nn2)CC1NC(c1cc(C)c(C)[nH]1)=O 35477,N1(C(C(C2CCOCC2)OCC)=O)CCC2C1CCCN2C(c1cnc(O)s1)=O 35478,C=C(Cl)CC1C(=O)NOC(C)C(=O)ON1CC.C1(CC(=O)OC)CN(C(C)=O)C1 35479,C1(CC=C)(C(=O)NCCC(O)C2CCCC2)CCN(C(=O)C=Cc2cocn2)C1 35480,Cc1ccc2n[nH]cc2c1C(=O)NC1CCN(C(c2cnc(O)c(Br)c2)=O)C1 35481,N1(C(CC(=C)C)=O)CC2CCC(N=c3ccc(C(=O)OC)c(OC)[nH]3)CC2C1 35482,N1(C(c2c(C)nc(CC)s2)=O)CC(CNC(c2ccsc2C#N)=O)CC1(C)C 35483,C(=O)(C1CCCc2c[nH]nc21)NC1(CNC(C23OCC(C)(C2)C3)=O)CC1 35484,c1(CC(=O)NC(C)CCNC(=O)C(C)C2CCCO2)ccc2nonc2c1 35485,C1(NC(C=COCC)=O)CC2CC(C1)CN(C(=O)COc1cc(F)cc(F)c1)C2 35486,C1(C(=O)NC(C)CCOC)(CC)CCCN(C(c2cc(CO)nn2C)=O)C1 35487,c1(C(=O)NC2C(NC(c3c(C)nc(COC)s3)=O)C2)cc([N+](=O)[O-])c(C)cc1C 35488,c1(C(=O)OC)ccc(C(=O)NC2CCC(NC(=O)CS(N)(=O)=O)CC2)nc1 35489,c1(CCC(=O)NC(CC)CNC(C2CCC(F)(F)CO2)=O)nc2ccccc2o1 35490,C(C1(C)COC1)=CC(=O)NCCN(C(C1C(C)(C(=O)OCC)C1)=O)CC 35491,N1(C(C2CCCN(CC)C2)=O)C2CCC(C2)C1CNC(c1ccc(O)nc1)=O 35492,N1(C(C2C(COC)C2)=O)CC2(COC(CNC(=O)Cn3nc(C)nc3C)C2)C1 35493,N1(C(C(C)(C)C2(O)CCC2)=O)CCCC(Cn2ccnc2)C1 35494,CCC(CC(C)C)C(=O)NCC1(O)CN(C(=O)Cc2ccn(CC(F)(F)F)n2)C1 35495,O=C1CCc2cccc(C(=O)NC3CCCC3CNC(c3coc(SC)c3)=O)c21 35496,C1(C)(NC(C2CN(C(c3c(CC)nns3)=O)CC(C)O2)=O)CCC(=O)NC1=O 35497,C1(N(C)C(C2(C(C)(C)C)CCC2)=O)CCN(C(=O)COc2ccsn2)C1 35498,c1(C(=O)NC2C(C(=O)NCc3c(C)nccn3)CCC=C2)ccn(C)c(=O)c1 35499,C1(C(=O)NC(C(=O)NC)(C)C)CC2CC1CC2NC(=O)C(CO)N(C)C 35500,N1(C(C(CC2CC2)NC(C2(CN(C)C)CC2)=O)=O)CCC(O)CC1 35501,C=C1CCN(C(=O)CC2CCCN2Cc2ccc(Br)cn2)CC1 35502,C1(CC)CN(C(=O)C=Cc2cccnc2)CCN1C(=O)COCC(=O)NC 35503,N1(C(c2c(C)ncs2)=O)CCCC2C1CCCN2C(C1CCC(N(C)C)CC1)=O 35504,c1(NC(C(C2CN(C(C(COC)O)=O)C2)OC)=O)cncc(N2CCCC2)n1 35505,N1(C(C2CCN(C(c3n(CC)ccn3)=O)C23CC3)=O)CCC(O)CC(C)C1 35506,N1(C(C(CCOC)OC)=O)CCN(C(=O)CCCSC)C(C)C1 35507,CC1CS(=O)CCN1C(C1CCCC(NC(=O)CCc2nccs2)C1)=O 35508,C12(C(=O)NCC(C(C)C)CO)COCC1CN(C(c1cc3ncccn3n1)=O)C2 35509,C(COC(C)C)(C(=O)NC(c1cccnc1)C)NC(CSCC)=O 35510,c1(C(C(=O)NCCC(=O)OCC)N(CC=C)C(C)C)ccc(C)nn1 35511,Cc1ncc(C#N)cc1NC(C1(O)CCN(C(c2ccoc2)=O)C1)=O 35512,N1(C(CCC(=C)Cl)=O)CCC2CN(C(C3(C)CCCNC3=O)=O)CC2CC1 35513,C1(CC)CN(C(=O)CC2CS(=O)(=O)C2)CCN1C(=O)COc1cnn(C)c1 35514,C(=O)(CC(C)CNC(=O)C(C)c1ccco1)NCc1n(CC)cnn1 35515,C(CC(C)C(=O)N1CCN(CCNC(=O)Cc2n[nH]c(=NC)s2)CC1)=CC 35516,CC(C)CCC(F)C(=O)NC1(CCC(=O)N(C)Cc2ccsc2)CCCC1 35517,c1(OC)ncnc(C(=O)NC2(C)CN(C(C3CCOC(=O)CC3)=O)C2)c1F 35518,N1(C(C2CCC(C)=CC2C)C(=O)NCC(=C)C)CCCC2OCCC2C1 35519,CCC(Cc1ccccc1)C(=O)NCC1(F)CN(C(=O)C(c2cnccn2)C)C1 35520,CCCC(CC)C(=O)NCC(O)CCNC(c1cc(=O)c(Br)c[nH]1)=O 35521,N1(C(CC2CC(=O)OC2)=O)CC=CC(C(=O)NC2CC(CO)C3CC23)C1 35522,CC(CC(C)NC(=O)CS(=O)(=O)NC1CC1)N=c1[nH]c(Cl)nc2ccccc12 35523,CC1(C(=O)NCC2CC(NC(C3CC(=O)N(O)C3)=O)C2)CS(=O)(=O)C1 35524,C1(CNC(C(CC)N(CC)CC)=O)CCN(C(c2cncc(N)n2)=O)C12CC2 35525,C(CC(=O)NCC(C)C1CCC1)(C1CC1)NC(C(C1CC1)SC)=O 35526,CCCC(C)(CCCC1CC1)n1nnnc1CN1CCCC(C2CCCCN2)C1 35527,N1(C(C2CC(O)(CC#C)C2)=O)CCCCC1CNC(c1ccnc(C(N)=O)c1)=O 35528,c1(C(=O)NC2CC(C)(NC(CC(=C)Br)=O)C2)c(O)nnc2c1CCC2 35529,C(C)(CCCNC(=O)CSCC(C)C)NC(C1(NC(C)=O)CCC1)=O 35530,C(=O)(NNc1cccc2ccsc12)C1N(C(=O)OC(C)(C)C)C(C)(C)CO1 35531,N1(C(c2cc(Br)cs2)C(=O)NCCSC)CC2CCCCN2c2ccccc21 35532,c1(C(=O)NC2C(C)CCN(C(c3csc4cncn34)=O)C2)cc2occc2n1C 35533,c1(C(=O)NC2CC(F)(CNC(C(N3CCOCC3)C)=O)C2)c(F)ccc(F)c1N 35534,N#CC1(C(N2CCN(C(C3(S(N)(=O)=O)CCC3)=O)CC2)=O)CC2CC2C1 35535,N1(C(C2OCCC(C)C2)=O)CCN(C(c2cc(O)cc(=O)o2)=O)CC1CF 35536,Cc1cc2[nH]c(=O)c(C(=O)NC3CCN(CC(=O)OC(C)C)C3=O)cn2n1 35537,CC(=O)CC(C)(C)C(=O)N1CCC(C)C(CNC(C2CN(C)CC(C)O2)=O)C1 35538,C1(C(N2CCC(C(C)OC)CC2)=O)CC2CCC1N2C(c1csc(C)c1)=O 35539,CN=c1[nH]c(=NCCCOC)[nH]c(=NC2CCOC3(CCC3)C2)[nH]1 35540,c1(C(N(CCCCN(C(CCn2c(C)ncc2)=O)C)C)=O)ccc(F)c(Cl)c1F 35541,c1(C(CNC2CCC(C(=O)Nc3c(Cl)cccc3I)CC2)O)cc2ccccc2s1 35542,N1(C(c2c(C)ccnc2)=O)CCCC(C)C1CNC(=O)C(F)C1CCOC1 35543,c1(C(N2CCN(C(c3ccc(C(C)=O)nn3)=O)C3C2C3)=O)c[nH]c2ccccc12 35544,N1(C(CN(C(COc2cc(C)on2)=O)CCO)=O)CC2(CCC2)C12CCC2 35545,C1(CNC(CC2C(C)CCO2)=O)CCCN(C(C2(c3ccc(Cl)cc3)CC2)=O)C1 35546,N1(C(COCCC#C)=O)CCC(C)(CC(=O)N(CC(C)C#N)C)C1 35547,C(=O)(C(C)C(O)CC(C)C)N1C(C)(CC(=O)Nc2c(F)ccc(C)c2)CC1 35548,c1(OC)ccc(CC(=O)NC(CNC(=O)Cc2ccnc(O)c2)C2CC2)cc1O 35549,C=CCC(CNC(=O)CC1CC2CC2C1)NC(c1cccs1)=O 35550,C=C(Cl)CC(C(=O)NC(c1nccn1C)C)NC(=O)Cc1ccn(CC)n1 35551,C1(NC(c2cc(C)sc2)=O)C2CC3CN(C(c4cc(C(F)F)nn4C)=O)C1C3C2 35552,Cc1ccc(C(=O)NCC(C)(CO)NC(=O)CC2CCC2(C)C)c(O)n1 35553,c1(OC)c(C(N2CCCCC(Cn3cc(C4CCC4)nn3)C2)=O)ccc(Cl)c1Cl 35554,c1(OCC)cc(C(N2CCC(=CCNC(=O)CCC3(C)CC3)CC2)=O)cc(F)c1 35555,Cc1ccc(Cl)c(C(=O)NCCNC(c2ccc(C(C)(C)C)cc2)=O)c1N 35556,N1(C(C(CSC)OC)=O)CCC(NC(=O)Cc2nc3ccccc3s2)C(C)(C)C1 35557,C1(NC(CCCN(C(=O)CC2CNC(=O)O2)C)=O)(CO)CC2CCCC12 35558,CCCCCC(O)CC(=O)NCC1CC2(CC2)CN1C(=O)C(O)CC1CC1 35559,N1(CCNC(c2nc(C(C)C)oc2)=O)CCCN(C(C2CC2(F)Cl)=O)CC1 35560,CC1CC(C(F)(F)F)n2nc(C(=O)NCC3CC4(CC4)CO3)cc2N1 35561,n1(CC=C)nnnc1C(c1cc(C(F)(F)F)cs1)NCC(C)OC 35562,Cc1nc([N+](=O)[O-])cn1CC(=O)NCCC(C(C)C)NC(C1CCOC(=O)N1)=O 35563,C1(NC(c2ccnc(Cl)c2F)c2n(C3(C)CC3)nnn2)COC2(CCC2)CO1 35564,c1(C(=O)NCC2(CNC(C(C(C)C)OC)=O)CC23CCC3)ccc(Cl)c(F)c1O 35565,O(C1CCCc2ccccc21)CC(=O)N(Cc1n[nH]c2c1CCCC2)C.CC(C)O 35566,C(=O)(C(O)CCCc1ccccc1)N(CCNC(C1CCCN(C)C1)=O)C1CC1 35567,N1(N2CCn3c(O)nnc3C2)CC2C(CO)C3CCC2(C1)O3.O=CNCCSC 35568,c1(NC(C2N(C(C3(SC)CC3)=O)CCC2)=O)ccc(C)c(F)c1F 35569,C1(NC(C2(C)N(C(CCc3c(C)noc3)=O)CCC2)=O)(CO)CC2CCCC12 35570,c1(C(=O)NCC(C)CNC(C23CC(C)(C2)C3)=O)cc2c(o1)CCCNC2=O 35571,C1(CNC(c2c(N)c(Cl)ncc2)=O)CCC2(CCC2)C1NC(c1ccoc1Cl)=O 35572,N1(c2nccn(CC#C)c2=O)CC(CC(=O)OCCOC)c2ccccc21 35573,Cc1cnnc(O)c1C(=O)NCC(C)CN(C)C(c1cscc1F)=O 35574,C1(C(=O)NCC2C3CN(C(=O)C(C)OC)CC23)(CC)CCCCC1 35575,n1(CC#C)cccc1C(=O)NCCCNC(=O)C(C)OCc1ccccc1 35576,C1(C(=O)NCC(CC(F)(F)F)NC(c2c[nH]c(=N)s2)=O)CC2CCCC(C1)C2 35577,N1(C(C(CC=C)NC(C)=O)=O)CCC(C)N(C(=O)CSC(C)(C)C)CC1 35578,CN1CCN(C(=O)CCc2cc(F)ccc2Br)C(CNC(=O)C(N)=O)C1 35579,c1(OC)ccc([N+](=O)[O-])cc1-n1cc(CN(C(=O)C(C2CCC2)OC)C)nn1 35580,CCCS(=O)(=O)CC(=O)NC12CCN(C(c3cc(C)c(C)o3)=O)CC1C2 35581,N1(C(C(C)=C2CC2)=O)CCC(C(=O)NCC(C)(C)C(C)C)C1C 35582,N(C(=NCCCSC)NCC1CC2CCC2C1)C(C#C)COC 35583,CCCCCCCCNC(=O)C(=O)NC1CN(C(=O)C(C)SC)CCC1F 35584,n1(CC2CCN(C3CCCN(C)C3=O)CC2)ncc(Cl)c(Cl)c1=O 35585,Cc1ccc(Cl)cc1C(=O)NCC(CO)NC(=O)CN1CCC(C)C1 35586,CC1CN(C(C2CC(O)(CNC(C3(O)CCC3)=O)C2)=O)CC(C)(C)C1 35587,CC1(NC(C23CC(CN2C(C2(CCN=[N+]=[N-])CC2)=O)C3)=O)CCOC1=O 35588,C1(CNC(C(c2ccc(C)o2)C)=O)CN(C(=O)C=Cc2cccs2)C(C)(C)C1 35589,C1(N(C)C(c2ccc(Br)o2)=O)CN(C(c2ccncc2)=O)CC1O 35590,c1(C(N2CCC(C(N(CCC(=O)OC)C)=O)C2)=O)ncc(F)cc1F 35591,C(N=c1nc(N2CCCC(Cn3ccnn3)C2)cc(C)[nH]1)C1(OC)CCC1 35592,N1(C(c2scc(OC)c2OC)=O)CCN(C(C2OCCO2)=O)CC2(CC2)C1 35593,c1(C(=O)NC2(CCC)CCN(C(CC=C)=O)CC2)cc2c(cnn2C)nc1C 35594,C1(CCC)CN(C(=O)CO)CCN1C(C12CC(NC(=O)CCC3CC3)(C1)C2)=O 35595,N1(C(C2CC(C)SCC2)=O)CC(NC(C2COC(C)(C)C2)=O)CC(C)(C)C1 35596,C=C(Cl)CCCN=c1ccc2cc(S(=O)(=O)N(C3CCC3)CC)ccc2[nH]1 35597,N1(C(c2c(CC)noc2)=O)CC(CNC(c2cccc(C)c2)=O)CCC1C 35598,c1(C(N(C(CC(=O)OCC)c2ccccc2)CCC)=O)ccc(CCOC)o1 35599,c1(C(=O)NCc2occ(C(=O)NCC(C(CC)C)C)c2)ccnc(C)c1N 35600,c1(C(N2C(CCNC(CCCCCC=C)=O)CCC2)=O)cc(N)c(F)c(F)c1Cl 35601,c1(C(N(CC(C)NC(=O)CCOCC(F)(F)F)CC)=O)cncc(Br)c1 35602,C(c1cn(CCCN(C)C(C2CCN(c3ccc(Cl)cn3)CC2)=O)nn1)=CC 35603,C1(C(=O)NCC(Cc2ccccc2)N(C(C(C)O)=O)C)CCC(F)CC1 35604,C12(C(N3CCC(NC(c4cc(C)cc(O)c4)=O)C3)=O)CCC(C)(CC1)OC2 35605,N1(C(C23N(C(C(CC)COC)=O)CC(C)(C2)C3)=O)CCC2CC1C(=O)O2 35606,C1(NC(C(N2CCSCC2)C)=O)CC(F)CN(C(c2cc(C3CCC3)on2)=O)C1 35607,Cc1ccc2sc(C(N3CC4CCN(C(=O)C(C)S(N)(=O)=O)CC34)=O)cc2c1 35608,N1(C(c2c(C)nc(C)o2)=O)CC2CCCC(C1)N2C(=O)C(C)n1ccnc1 35609,c1(C(N(C)CC2CCN(C(C3CN(C(C)C)C3)=O)C2)=O)cnccc1Cl 35610,C(=O)(CCC(=O)N1CC(CCNC(C2(SC)CCC2)=O)C1)Nc1nnc(CC)s1 35611,C12(C(N(CCN(C(C3CC3(C)C(C)C)=O)CC)CC)=O)CC(C)(C1)OC2(C)C 35612,CC1(C)CC(CC(=O)Nc2ccnc(C3CC3)c2)C(=O)O1 35613,C1(NC(=O)CCC(F)(F)F)CCCC2CN(C(=O)CC3CCOC3)CC12 35614,C1(C(=O)NC(c2ccc(F)cn2)CO)CC2c3ccccc3C1c1ccccc12 35615,Cn1nnc(CN(C(=O)Nc2cc(F)c[nH]2)CC2CC2c2ccco2)n1 35616,N1(C(c2c(C)occ2)=O)CCC2CC(CNC(C3CCC(C)CC3)=O)CCC2C1 35617,CC(C)CC(C(=O)NCCc1noc(=O)n1C)ONC(=O)C1(N(C)C)CC1 35618,C1(CC(C)C)(C(N(C2CC(NC(CCC=CC)=O)C2)C)=O)CCNC1=O 35619,C1(NC(c2cccc(F)c2OCCF)=O)CN(C(=O)COC(F)F)CCC1CO 35620,c1(C(CC)O)nc(C2CCC(=O)N2C)n(-c2nc(C)nn2C)n1 35621,N1(C(CCCCOCCC=C)=O)CCN(C(c2ccnc(C)c2)=O)C(C)C1C 35622,C1(F)(C(=O)OCC)CN(C(=O)C(=O)c2cccs2)CC1(C)C(F)(F)F 35623,N1(C(c2onc(CC)n2)=O)CC2(CCN(C(=O)Cc3cccs3)CC2)C1 35624,c1(C(=O)NC(CNC(C(C)NC(c2ccoc2)=O)=O)C)cc(Cl)c(Cl)n1C 35625,c1(NC(c2ccc(-c3cccc(C)c3)cn2)=O)ccc(F)c(Cl)c1F 35626,N1(C(CCC#C)=O)CCOCC(F)(CNC(C2CN(C3CCOC3)C2)=O)C1 35627,C1(C(=O)NCC(CC=C)NC(c2cc(CCC)oc2C)=O)CC2C=CC1C2 35628,CC(C(=O)NC(C(=O)NCC1(CO)CCC1)c1cccs1)OC1CCCC1 35629,C(=O)(CCCC(C)(C)C)N1CCC(CN(C(=O)Cc2cn3ccsc3n2)C)C1 35630,Cc1cc(O)nnc1C(=O)NC(C)CCNC(=O)C(C)(C)c1cscc1Cl 35631,c1(CC)c(NC2CCN(C(C3(F)CCOC3)=O)CC2C)nc(C)nc1Cl 35632,N1(C(c2nnn(CC)c2C)=O)CCC(C2(NC(=O)C3=C(C)CC3)CC2)CC1 35633,[N-]=[N+]=NCCCC(=O)NCC1(O)CC(CNC(=O)CCc2csc(=N)[nH]2)C1 35634,c1(CCC(=O)NCCOCCNC(c2cc(C)c(C)[nH]2)=O)cc2ccccc2o1 35635,C1(CN(C(=O)CSc2nncs2)C)CCCN1C(C1CCC(=O)O1)=O 35636,N1(C(C(CC)OCC)=O)CCC2(CCCN2C(c2cc(C(F)F)no2)=O)CC1 35637,n1(CC)nc(C)cc1C(=O)NCC1CC1NC(=O)C(C)(C)n1ccc(C2CC2)n1 35638,C1(CN(C)C(c2ccc(C3CCOC3)s2)=O)CCN(C(c2occc2F)=O)CC1 35639,N1(C(c2ncncc2Cl)=O)CCC(CNC2C(C)(C(F)F)C2)C(O)C1 35640,N1(C(c2c(C)nc(C)o2)=O)CC2(COC(CNC(c3csc(S)n3)=O)C2)C1 35641,N1(C(c2cnn(CCC)c2Cl)=O)CCC2CN(C(C3(C=C)CCC3)=O)CCC2C1 35642,C(=O)(CCS(=O)(=O)C1CCCC1)NCC(CCOC)NC(=O)COC(C)(C)C 35643,C=CCC(C)C(=O)NCC1(C(=O)NCCOC(C)=O)CC=CC1 35644,CC(C)(C(=O)NCC(O)CCNC(c1cnn(CC2CCCO2)c1)=O)C(F)(F)F 35645,Cc1c(F)ccc(C(=O)N(C2CCC(NC(C3CCCCC3C)=O)CC2)C)c1C 35646,C1(NC(C(C)OCCCCCC)=O)C=CCN(C(C2CC23CCC3)=O)C1 35647,Cc1cc(C)c(C=CC(=O)NC2(CO)CCN(C(=O)C3=CCCS3)CC2)cc1C 35648,C(=O)(C1=CCC2CCC1N2C(C1(CF)CC1)=O)N1CCC(C)(O)CC1 35649,N1(C(c2nscc2Br)C(=O)NCC2(C(=O)OCC)CC2)CC2CCC2(C)C1 35650,c1(C(=O)NC2CCC(NC(=O)C3=C(Cl)CCC3)CC2)c(Cl)ccc2ccoc12 35651,c1(NC(c2cc(CC)on2)=O)ccc(S(=O)(=O)N(CCOC)CC)cc1 35652,CCC(CC)CCCC(=O)N1CC2CCC1CC2NC(C1C=CC=CC=C1)=O 35653,N1(C(c2scc(CNC(C(C=CC)O)=O)c2)=O)CCc2c(cnn2C)C1 35654,CC(=O)CCN=C(NCC1CCCCS1)NCC(C1COC(C)(C)O1)O 35655,C12(CNC(C3CCN(C(C4CCNC4=O)=O)CC3)=O)CCC(CC1)O2 35656,C(N=c1nc(C(=O)OC)c(Cl)c[nH]1)C1CCCC(NC(C(CCC)(C)CC)=O)C1 35657,c1(OC)cc(C(=O)NC(CNC(C2CCCC23CC3)=O)C2CC2)c(F)cc1N 35658,C(=O)(C(C)C(O)CC)NCC(CC=C)NC(c1cncc(CO)c1)=O 35659,C1(CNC(C=Cc2n(C)cnc2)=O)CCN(C(=O)C=CC(=O)NC2CC2)C12CC2 35660,c1(C(=O)NC2CN(C(C(C)(C)OCC(F)(F)F)=O)CC2F)cc2sccc2[nH]1 35661,c1(C(=O)NCC2N(C(C3C(OC)C3)=O)CC(OC)C2)c([N+](=O)[O-])cnn1CC 35662,C1(CNC(c2c(C(C)C)noc2)=O)CN(C(C2CC3CC3C2)=O)CCC1C 35663,Cc1cc(C(N2CCOC(C(C)NC(C3CCCCO3)=O)C2)=O)cc(C)c1F 35664,C1(NC(C(CC#C)C)=O)CS(=O)(=O)C2CN(C(=O)CNC(=O)NC3CC3)CC12 35665,C1(C(=O)NC2CC(NC(C3CC4(CC4)C3)=O)C2)CCC12CCCO2 35666,c1(C(=O)NC2C(NC(c3nncc(OC)c3)=O)COCC2)cc(C)c(Cl)cn1 35667,S(=O)(=O)(c1cccc(C(=O)N(C)C)c1)N(C1CC(Nc2c(C)cncn2)C1)C 35668,C1(N(C)CC2(C(=O)NC3(CO)CCCC3)CC2)CCC(n2cc(C3CC3)nn2)C1 35669,N1(C(=O)CO)CCC2(CC1)CN(C(c1ccc3nn[nH]c3n1)=O)CCO2 35670,c1(C(=O)NC2C(NC(C3CCC(=O)NC3)=O)C2)ccc2c(c1)C(=O)CCO2 35671,C12(CC(C)(C)C1)c1nnnn1CCCCOCCN2.n1(C)cc(C2CC2)cn1.CO 35672,CC1CC(CNC(=NCCN2CCOCC2)NCC2CC2CF)CC(C)O1 35673,N#Cc1ccncc1NCc1cc(C(=O)NCc2ccc(Br)cc2Cl)ccn1 35674,C1(C2CCOCC2)(NC(C(CC(C)C)ONC(C2C(C)C2C)=O)=O)CC1 35675,C(C(C(=O)NCCN(C(=O)C(C)(C)n1ccnn1)C)C(C)(C)C)OCC=C 35676,C(=O)(CCCC(=O)NCc1ccc(C(=O)NC)nc1)N(CCCCN(C)C)CC 35677,Cc1c(C(F)(F)F)n[nH]c1C(=O)NC(C)CN(C(=O)Cn1cnc(Br)c1)C 35678,C(=O)(CCCCCC#N)NCC1(C(=O)NCC2(C)CCN(C)C2)CC1 35679,c1(C(=O)NCC#CC(=O)N(C)Cc2ccncn2)cccn(C)c1=O 35680,c1(C(N2CC(NC(C3(COC)CC3)=O)C(C3CC3)C2)=O)oc2ccccc2c1C 35681,c1(CNCC2N(CC(C)C)CCC2)n[nH]c2cc(F)ccc12 35682,c1(C(N2C(CN(C(C3C(C=C)C3)=O)C3CC3)CCC2)=O)nc2cccnc2s1 35683,CCC(CCC(=O)NCCN(C)C)NC(=O)CN(CC(C)(C)C)C 35684,C1(CC(C)NC(C=C(COC)C)=O)CCN(C(=O)C(N2CCCCCC2)C)CC1 35685,c1(OC2CCN(C(N3C(CC(C)C)COCC3)=O)C2)ccc(C#N)n1C 35686,C1(CNC(C(C)(CO)OC)=O)CN(C(=O)CCc2nnc(O)nc2O)CC1(C)C 35687,c1(C(N2C(C(=O)Nc3cc(OC)cc(C)c3)CC3CC32)=O)[nH]nc2ncccc12 35688,c1(C(=O)NCCCC(C)NC(c2cc(CC3CC3)on2)=O)cc[nH]c(=N)c1 35689,N1(C(C(CN=[N+]=[N-])NC(=O)C(C2CC2)C2CC2)=O)CC2CCC(O)C2C1 35690,n1(CNC(c2cc(OC)c(OCC3CCCO3)cc2)C#N)cnc2ccccc12 35691,c1(CC)ncc(C(=O)N(C2CCCCC2)Cc2cccnc2)c(C)n1 35692,c1(OC)nccc(C(=O)NCc2occc2C(=O)NC(c2ccccc2)C)n1 35693,C1(F)(CNC(CN(C2CC2)CC)=O)CCCN(C(=O)CS(C)(=O)=O)CC1 35694,c1(C(=O)Nc2cncc(C(=O)NCC(N)=O)c2)cccc2ccnn12 35695,c1(C(=O)NCC(CC)NC(c2cc(C(C)(C)C)ncn2)=O)ccc(CO)c(F)c1 35696,C1(CNC(c2n(CC=C)ccc2)=O)(CNC(C2SCCS2)=O)CC12CCC2 35697,N1(C(c2cc(N(C)C)ncc2)C(=O)NCC2CCOC2)CCCC(C)(C)CC1 35698,c1(CC(N2C(C)CC(NC(CC(CC)C3CC3)=O)C2)=O)ccc(O)c(C)c1 35699,C(=O)(CCCCCNC1CC1NC(c1ccc(Br)c(COC)c1)=O)OCC 35700,c1(CC(=O)N(CCOC)CCNC(C2CCC2)=O)cccc2cccnc12 35701,NC(=O)C1CN(C(C2CC3(C2)CC3(F)F)=O)c2ccccc21 35702,C(C)(CCC(=O)N1CCN(C2CCN(C(=O)C=C3CCC3)CC2)CC1)OC 35703,c1(NCc2cc(C(=O)OC)c(C)cc2)cc(Br)c(Cl)nc1OC 35704,C1(C(=O)NC(C)C)CCCCCC1NC(C1CC1(F)F)=O 35705,C(C)(C)(CC(=O)NC(C1CN(C(=O)CC2CCCS2(=O)=O)CCO1)C)SC 35706,c1(C(=O)NC(C)(C)CCNC(C2CCCCC2C(N)=O)=O)cc(N)ccc1Cl 35707,N1(C(CSc2cn(C)nc2)=O)CCC(CO)C(NC(=O)CCOC2CCC2)C1 35708,c1(OC(C(C)OC2CCCOC2)=O)cc[n+]([O-])cc1 35709,N1(CC(=O)NCC(C(C)C)NC(=O)CC2CCCCN2C)CCC(=O)NC1=O 35710,c1(C(N(CCCN(C(=O)C=CC2CCOC2)C)C)=O)cc(C(F)(F)F)cc(N)c1 35711,C(=O)(CC(C(C)C)NC(C1CN(CC)CCO1)=O)N(CC=C)C 35712,C1(C(=O)NC2C(NC(C=CC(=O)OCC)=O)CC2)CC(=O)N(c2cnn(C)c2)C1 35713,C1(C)(C(N2C(C(C)C)COCC2)=O)CCCN(C(c2ccc(Cl)o2)=O)C1 35714,C(=O)(CS(=O)(=O)CCC)N1CC(CCNC(CCC=CC)=O)OC(C)C1 35715,C1(N(C(=O)CN2CCSCC2)C)CCCC(NC(=O)C=CC2CCCC2)C1 35716,N1(C=O)CCCN(C(N)=O)CC1.Cc1ccc(CC(=O)NC2(C3CC3)CCC2)o1 35717,CC(C)C(N=[N+]=[N-])C(=O)N1CC2CC1C2NC(c1cncn(C)c1=O)=O 35718,C12(CNC(c3cc(C)ncn3)=O)CCC1CCN2C(=O)CNC(c1ccsc1)=O 35719,Nc1cc2[nH]c(O)nc2cc1C(N1CCCC2CC12)=O 35720,Cc1nc(NC(C2CC(C)CN2Cc2cnn(C)c2C)=O)cc(Cl)n1 35721,C1(CNC(C(CC=C)(C)C)=O)CC2CCC(C1)N2C(=O)CC1CC(C)C1 35722,Cc1nnc(N(C(=O)C(C)CC(N)=O)C2CCN(C)CC2)c(C#N)c1C 35723,c1(CN(C)C)ccc(C(=O)NC2COCC2CNC(=O)CN2CCCC2=O)o1 35724,C1(CC(=O)Nc2cnc[nH]2)CC2(CC2)CO1.C1(=O)CCC2CC(C2)N1C 35725,CC1=CC(C(=O)N(C(C)C(=O)NCC(c2ccsc2)C)C2CC2)SC1 35726,CC1CC2CN(C(=O)CCCCNC(=O)CNC(=O)CCC(CF)CF)CCN2C1 35727,N1(C(C2CCCN(C(C(C)CC3CC3)=O)C2)=O)CC2(COCC(=O)N2)C1 35728,N#Cc1ccc(C(=O)NC2CCCC2CNC(=O)Cc2cccc(F)c2)o1 35729,C(=O)(CCC1CCc2ccccc21)NCc1c(N(C)C)cc(C(=O)O)nn1 35730,C1(NC(=O)C=CC2CCCC2)CCN(C(C2CCCS2)=O)CC1F 35731,c1(NCCS(CCOC)=O)[nH]c(=NCCc2cn(C(C)C)nn2)nc2scnc12 35732,n12cnc(c1)C(=O)N(CCF)CC2.N#CCCSCC(=O)NCC1CC1 35733,N1(C(c2cc(CC)on2)=O)CCCN(C(=O)C(N2CCN(C)CC2)C)C(C)C1 35734,C(=O)(CC1=CCOCC1)N1CCC(N(C(=O)Cc2cccc(C#N)c2)CC)CC1 35735,C(N=c1cc(C)nc(-c2cccs2)[nH]1)C1OCCN(C(C(C(CC)C)OC)=O)C1 35736,Cc1ccc2cc(C(N3CCC4CCC(C3)N4C(=O)COCCF)=O)ccc2n1 35737,CCC(C)CCC(=O)NC1CC2(NC(c3cccc(N(C)C)c3)=O)COC1C2 35738,C1(SCc2n(C)ncc2)CCN(C(=O)C(=O)NCC(=O)OC(C)(C)C)CC1 35739,c1(C(=O)NCC(CC)(C)NC(=O)Cn2cccc2)cccc(C2CC2)n1 35740,c1(CC(N2CC(OCCNC(C(C)=CC)=O)C2)=O)ccc2ncccc2c1 35741,N1(Cc2ccc(CC)s2)CC2CC1(C(=O)O)CN2C(=O)OC(C)(C)C 35742,c1(C(C(=O)NCCC)N(c2ccccc2)CC2CCOCC2)ccc(CO)cc1 35743,C1(CCC)(C(=O)NCC(CCOC)NC(=O)CCCCSC)CCNC1=O 35744,N1(C(COCCC=C)=O)CC2ON=C(CNC(c3cccc4ncnn34)=O)C2C1 35745,CCCC(C)CC(=O)NCCC(C)NC(=O)CSc1cc(F)ccc1F 35746,c1(C(=O)NC(C2N(C(CCCC(=C)C)=O)CCC2)C)ccc2cc[nH]c2n1 35747,c1(OC)ncc(CN(C)C(=NCC2CCCNC2=O)NC2CCCC2)cc1Cl 35748,c1(N2CCN(CCO)CC2)ncnc2cc(N(c3c(Cl)cccc3Cl)C)ccc12 35749,n1(CC(=O)NC(CC)CN(C(=O)C(C)OC2CCOC2)CC)cnc(=N)[nH]1 35750,CN=c1[nH]c(=NCc2ccccc2OC(C)C)[nH]c(=NCCC2(C)CC2(Cl)Cl)[nH]1 35751,N1(C(C(COC)Cl)=O)CCC2(CCC2N2CC3CCC2C3)CC1 35752,C#CCCCCCC(=O)NC1(CCOC)CCN(C(=O)Cc2ccnc(C)c2)C1 35753,C1(NC(COCCC)=O)(CF)CCN(C(c2sc(C(C)C)nc2C)=O)C1 35754,N#Cc1cccc(C(=O)NC2CCN(c3ncnc4n[nH]cc34)CC2)c1Cl 35755,c1(C(=O)NCCC(C)NC(c2c(CC)nns2)=O)ccc(C#N)n1C 35756,N1(C(C(=O)NCCC)CC2CCC(F)(F)CC2)CCCC2CN(C)CCC12 35757,C1(NC(CC(C)F)=O)CC12CCC(NC(=O)CCc1cn[nH]c1)CC2 35758,C(C(C(=O)NCC1(C)CCCN1C(=O)CCc1ncccc1C)C(F)(F)F)OC 35759,Cc1ccc(C=CC(=O)NCCCNC(c2c(-c3cccs3)noc2C)=O)cn1 35760,c1(OC)ncc(Cl)cc1C(N1CCN(C(c2cc(C)co2)=O)CC1C(F)F)=O 35761,C(=O)(C(C)(C)CN(C(=O)Cc1ccsn1)C)NCCS(CC)=O 35762,N1(C(C2N(CC)CCC2)=O)Cc2ccccc2C(NC(=O)Cc2nnc(C)s2)C1 35763,CC1(C(N2CCC(O)(CCNC(C3CCC4(CC4)C3)=O)C2)=O)COC(=O)N1 35764,c1(OC(C)C(=O)NCC2CC(NC(c3coc(O)n3)=O)C2)cccnc1 35765,c1(C(N(C(CNc2ncc(C#N)cc2Br)C2CC2)C)=O)cnc2c(c1)ncn2C 35766,c1(NC(=O)NC(CC2CCCC2)CO)cccc2nc(O)nc(O)c12 35767,CC(C)CC(CNC(=O)CC1CCCCOC1)C(=O)NCC1(C)COCCO1 35768,N1(C(c2nn(CC)c(O)c2)=O)CCOCC(N(C(=O)CNS(=O)(=O)CC)CC)C1 35769,N1(C(C2(C)CCC2)=O)CC2COCCC2(NC(=O)CC2CCNC2=O)C1 35770,C1(C(=O)NCC(C2CC2)SC)CCN(C(=O)CC2CCCC(C)O2)O1 35771,C1(NC(CSCC#C)=O)CN(c2nnc(C(N)=O)s2)CC2(CC2)C1 35772,c1(C(=O)NCC2C(NC(=O)C=CC3CCC3)CC2)cnc2[nH]ncc2c1 35773,Cc1c(C(=O)NC(CO)C(=O)NCC2CSCCO2)ncn1C 35774,CC(C)C(S(=O)(=O)NC(C)(C)CSc1ccccc1)c1ccccc1 35775,N1(C(C(CCC)O)=O)CCC2(CC1)CC2C(=O)NC(c1ccc(Cl)cc1)C(=O)OC 35776,CN1CCC(C)(C(=O)NCC2CCN(C(=O)Cc3cn[nH]c3)CC2O)CC1 35777,c1(C(N(CCN(C(C2CC(=C3CCC3)C2)=O)CC)CC)=O)c(C)n[nH]c1C 35778,C(C(C(=O)NCC1CN(C(C2(C3CCC3)CC2(F)F)=O)C1)C(C)(C)C)OCC=C 35779,c1(C(=O)NC(C)C#N)ccc2c(-c3cscc3C#N)nn(C)c2c1 35780,N1(C(CC2CC(=O)C2)=O)CC=CC(NC(C23CSCC2C3)=O)C1 35781,C1(NC(C2N(C)CCC2)=O)CC2CC1N(C(=O)Cc1cccc(C3CC3)c1)C2 35782,Cn1cc(C(=O)NC2CCC(NC(C3(C)COC3)=O)CC2)c(C(F)F)n1 35783,C#CC1CN(C(=O)CCC2CCCCN2C(c2cc(Cl)no2)=O)CCO1 35784,C1(C(=O)NC2CC(C(C(=O)NC(C#C)CC3CCC3)F)C2)Cc2ccccc2C1 35785,C(=O)(C(C)(C)F)NC(C1CCCCC1)CNC(C(C)c1ccon1)=O 35786,N1(C(C#C)(C)C2CCC2)CCC(OCC(=O)NCc2ccccc2)C1 35787,c1(C(C(N2CC(C(C)(C)O)(CNC(CCOC)=O)C2)=O)C)ccc(N(C)C)cc1 35788,C12(C(=O)NC(C(C)F)C)CC(CCO1)N(C(C1CN(C)C(=O)N1)=O)C2 35789,CCC(C)(C)C(=O)NCC1C2CN(C(=O)CNC(c3cccs3)=O)CC12 35790,c1(C(N2CC(NC(C3(CC)CC3(F)F)=O)C2)=O)ccccc1S(C)(=O)=O 35791,CCCC(C(=O)OC)NC(=O)CC1CN(C(=O)C(C(C)O)N(C)C)CC1C 35792,c1(C(=O)NCC2CN(C(C3CCC(=O)NC3)=O)CC2O)[nH]cc2c1CCC2 35793,N1(C(Cn2nnc(C)n2)=O)CC=C(C(=O)N2CCC(OC3CC3)CC2)CC1 35794,C(=O)(CCCCC(F)(F)F)NC12CC(NC(CC(C=C)C)=O)(C1)C2 35795,C(CC(C(C)(C)C)NC(=O)CC1CN(C)C1)N(C(c1c(C)c[nH]c1)=O)C 35796,CCCCCCC(c1nnnn1C(C)(C)C)NC(c1ccc(F)cc1)C(=O)NC 35797,Cc1cnc(F)c(C(N2CCC(NC(c3cc(C(N)=O)ccn3)=O)C2C)=O)c1 35798,Cc1ncc(Cl)cc1NC(=O)CCN(C)C(c1nn(C)cc1Cl)=O 35799,CN1C(=O)OCC1C(=O)NC1CC(CNC(c2cccc(=O)o2)=O)C1 35800,c1(C(=O)NCCCN(C(C(C(=O)OC)OC)=O)C2CC2)cc2n(n1)CC(F)C2 35801,C12(C(=O)OC)CC1CN(C(=O)CC(O)CNC(c1cc(C3CC3)[nH]n1)=O)C2 35802,c1(C(N2C(C(N)=O)CCC(C)C2)=O)coc2c1CN(C(=O)CC1CCC1)C2 35803,C1(n2c(C(c3nn(C)nc3Br)NCC(CC(C)C)OC)nnn2)CCC(F)(F)CC1 35804,N1(C(CC2CC(OC)C2)=O)CCC(CCNC(=O)CCc2cc(C)[nH]n2)CC1C 35805,c1(C(=O)NCC(CC)NC(c2cnsc2C)=O)n[nH]c(C)n1 35806,C(=O)(C1=CCCCCC1)NC1CCC(NC(c2c(SC)n(C)nc2)=O)C1 35807,n1(C(C)C)ncc(C(N2CCCC2CN(C(=O)CSCc2ncc[nH]2)C)=O)c1N 35808,CC1=C(C(=O)NCC2CCC(N(C(=O)CN3CC(C)(C)C3)C)CC2)COCC1 35809,CCCC(C)CC(=O)NCC(O)CN(C(=O)COc1ccc(CC(N)=O)cc1)C 35810,N1(C(C=CC(=O)OCC)=O)CC2CC(NC(=O)Cc3cnco3)CC2C1 35811,C1(NC(c2cnsn2)=O)CN(C(C2CC(C(F)(F)F)C2)=O)CC1C1CC1 35812,N1(CCCOC)C(C)CN(C2=Cc3ncccc32)CC1C 35813,Cc1ccc(C=CC(=O)NC2CC2NC(c2cnc(C(C)(C)C)s2)=O)cc1Cl 35814,c1(C2(C(=O)NCC(C)CN(C(=O)C(C)C3CCC3)C)CCC2)ccccc1 35815,c1(OCC)ccc(NC(c2occc2CNC(C2(OC)CCOC2)=O)=O)cn1 35816,N1(C(C(CC)(C)COC)=O)CC(NC(c2cnn3ccccc23)=O)C2(CCC2)C1 35817,C1(NC(C2C(CCOCC)C2)=O)CCC(CNC(=O)CC(C)(C)O)CC1 35818,C1(C)(OC)CCN(C(=O)C(O)CCCNC(c2csnc2Cl)=O)CC1 35819,C1(C(N2CC(F)(NC(C3CC(OC(C)=O)C3)=O)C2)=O)CC(C2CC2)=NO1 35820,CC#CCC(C(=O)NCCC1(COC)CCN(C(C)=O)C1)NC(=O)OC(C)(C)C 35821,Cc1cc(F)cc(Br)c1C(=O)NC1CC2CCC1N2C(C1CCC(=O)C1)=O 35822,c1(C(N(C(CC(F)F)C(=O)NCC(O)(CO)CO)C)=O)ccnc2cc[nH]c12 35823,c1(C(=O)NCC2N(C(c3cccc(C)c3C)=O)CCCC2)cccc(S(C)=O)c1 35824,c1(C(=O)NCC(CC(F)(F)F)NC(CSC)=O)c(C)c(C)cc2ccccc12 35825,C#CC1(N(C(C2(C)N(C)CC(Oc3ccccc3)C2)=O)C)CCN(C(C)=O)CC1 35826,c1(CN(C)CCOCCNC(c2cc(Cl)c[nH]2)=O)ccc([N+](=O)[O-])cc1 35827,C1(S(C)(=O)=O)(NC(=O)NCc2c(OC)ccc(C(C)(C)C)c2)CC(O)C1 35828,c1(CCOC)nnc(NC(=O)CC2(CO)CC2)s1.CC(C)CN(C)C 35829,c1(C(=O)NC2CC(NC(C3CCCO3)=O)C2)c[nH]cc(F)c1=O 35830,N1(C(C(CC#C)C2CC2)=O)CCC2CCC(NC(c3conc3C3CC3)=O)C12 35831,CC1(C)CCC(C(N2CC3CC3(CNC(c3ccc(Cl)o3)=O)C2)=O)O1 35832,N1(C(c2scc(C(C)=O)c2)=O)CC(O)CC1CNC(=O)COC1CCOC1 35833,c1(C(N(C)CC2(O)CN(C(CC=CC=C)=O)C2)=O)cc(S(N)(=O)=O)cs1 35834,CCC1=NOC(C(=O)NCCC(O)CNC(=O)C(F)(F)CO)C1 35835,CC1(F)CN(C(=O)C(O)C2CCC2)CCN(C(c2c(Cl)ccnc2F)=O)C1 35836,c1(NC(C(=O)NCC(=C)Cl)=O)ccc(C(N2CCCC2c2ccco2)=O)cc1 35837,N1(C(CSC)=O)CC2CC(C(=O)NCCC(O)CO)C(C2)C1 35838,C1(Cn2cc(CN3CCCC(C)(SC)C3)nn2)CCCCN(C2CCC2)C1 35839,CCCCCCCCCC(=O)NC1CN(c2ncnc(Cl)c2F)CC1(C)C 35840,C(=O)(CCCCCNC(C1C(C)(C)C1(F)F)=O)NCc1nc(CC)sc1 35841,C12(C(N3CC(O)(C(C)NC(=O)CC4CC5CC5C4)C3)=O)CC(C)(C1)OC21CCC1 35842,C(=O)(C(CO)C(F)(F)F)NC(CCC=C)C(=O)NC1CCOC1C 35843,C(=O)(C(O)CC(F)(F)F)N(C)CCNC(C1CCC(Oc2ccncc2)C1)=O 35844,C1(C(N(CCCF)C)=O)CCCCN(C(C2(N(C)C)CC2)=O)C1 35845,CC1CC(=O)NC(C(N2CC(NC(c3cn(CCC(C)(C)C)nn3)=O)C2)=O)C1 35846,c1(-c2nc(-c3c(CSC(C)C)nccc3)nn2C2CC2)ccn(C(C)C)c(=O)c1 35847,c1(C(N2C(CC)CN(C)CC2)=O)ccc(S(=O)(=O)N(CC(C)C(F)(F)F)C)cc1 35848,c1(CN=C(NC(C#C)C(C)(C)OC)NC2CCC2)ccc(C#N)cc1Cl 35849,CCC(C)C(C(=O)NCC(C)(C)CNC(=O)CN(c1ccccc1)C)OC 35850,Cc1cc(C)c(C(=O)NC2CC23CC(NC(C2CCC(C)(C)O2)=O)C3)[nH]1 35851,C=C(CNC(C1CC1CN(C)C)=O)CCNC(c1ccoc1C)=O 35852,CCCCCC(CC)C(=O)NC(CNC(c1nocc1C)=O)CO 35853,c1(C(=O)NC(CNC(C(CC)n2nccc2C)=O)C2CC2)cc2cccnn2n1 35854,c1(C(=O)NC2C(NC(C(C)O)=O)COC2)cnc(C2CCC2)nc1O 35855,CCCC(C(=O)NC)NC(=O)CC1(N(C)C(C2CC(C)(C(=O)OC)C2)=O)CC1 35856,N1(C(CCNC(=O)C=CCl)=O)C(CNC(=O)Cc2cnc[nH]2)CC2CCCC12 35857,c1(NCCCN(C(C)C)CC)nccc(C)c1NC(c1ncccc1OC)=O 35858,C1(CC)CCCCN1C(=O)COCCNC(=O)CCC1CC1(C)C 35859,N1(C(CCS(C)=O)=O)CC(NC(c2cccc3c2CCC3)=O)C(C2CC2)C1 35860,C(C(C)C(C)C(=O)NCC1CN(C(C2CCC(=O)N(C)C2)=O)CCO1)OC 35861,C1(NC=O)C(F)(F)C12CC2.CC(C)(COC(C)(C)C)Cn1cc(-c2c[nH]cc2)nn1 35862,CCC(Cc1ccccc1C)C(=O)N1CC(NC(c2csc(CO)n2)=O)C(C)C1 35863,C1(CC(C)NC(CCC2CC(C)C2)=O)CCN(C(c2nccn2C)=O)CC1 35864,c1(C(=O)NCCN(C)C(C2CCCOC2c2cc[nH]n2)=O)cc(F)c(O)c(Cl)c1 35865,C1(NC(c2ccnc(CO)c2)=O)(CF)CCN(C(=O)CC2CCCC2(F)F)C1 35866,C1(C=O)(COC)CN(C(c2ccc(CO)o2)=O)C1.N(CC)CC1CC1 35867,N1(C(C2(C)N(C(Cc3c(C)ocn3)=O)CC=C2)=O)CCC(N=[N+]=[N-])C1 35868,N1(C(C(C)N=[N+]=[N-])=O)CC2CCCC2(CNC(c2cnnc(O)c2)=O)C1 35869,C(=O)(C(C)(C)CCCO)NCCC1CCN(C(C(C(C)(C)C)NC(N)=O)=O)CC1 35870,Cc1nocc1NC(=O)CNC(=O)CNC(c1ccc(F)s1)=O 35871,N1(C(CC2CC(=C)C2)=O)CCCC(O)(CN(C(=O)CCCn2cccn2)C)C1 35872,C1(C(=O)NC(C)CNC(C2CC(=O)N(c3nccs3)C2)=O)C2C3CCC(C3)C12 35873,N1(C(C(COC)NC(C2CCC(=O)C2)=O)=O)CC2(CNC(=O)C2)C1 35874,N1(C(=O)NC2CCCN(S(=O)(=O)Cc3ccccc3)C2)CC2CCCC(N)C2C1 35875,c1(C(=O)NCC(C)(C)Nc2nc(COC)nc(Cl)c2)ccc2c(c1)nc(O)n2C 35876,c1(OC)cc(C(=O)NCC23CC2CN(C(c2n[nH]cc2C)=O)C3)nc(Br)c1 35877,C1(C)(CNC(CN(C)C(N)=O)=O)CN(C(=O)CC2CCCC23CC3)CCO1 35878,C1(CNC(CCC(C)OC)=O)CN(C(c2nnn(C(C)C)c2C)=O)CC(C)(C)C1 35879,N1(C(CC(C)OC)=O)CC2CCN(C(c3nccc4[nH]ccc34)=O)C(C2)C1 35880,c1(NC(CCCN(CCOCC)C)=O)cccc(F)c1CNC(=O)COC(C)=O 35881,c1(C(=O)NCC2(C(N)=O)CN(C(C3C4CCCOC34)=O)C2)ccc(Cl)c(F)c1F 35882,c1(OC)cccc(C(=O)NC2CCCC(NC(c3nnsc3SC)=O)C2)c1F 35883,N1(C(CCc2cc(C)nn2C)=O)CC(NC(C2CC(F)(F)C2)=O)CC(C)C1 35884,C1(C(=O)NC(C2(O)CCN(C(=O)CC3CC3)C2)C)C2CCC1(c1ccccn1)C2 35885,c1(CC)ccc(C(=O)NCC(CO)NC(c2ccc(C)cc2C)=O)cc1C#N 35886,n1(CC)cncc1CNCc1cc(C)on1 35887,c1(COC)c(C(=O)NC2CCNC(C(=O)O)C2)oc2ccccc12 35888,c1(CN2CC3CN(C(c4c(C)nc(Br)s4)=O)CC32)c(F)cc(F)cc1Br 35889,CC1(C)CCC(C(N2CCOC(Cn3cncn3)C2)=O)O1 35890,CC(C)(CC1CCOC1)C(=O)NCC1CCN1C(=O)COCC1CCOCC1 35891,N1(C(CCC(C)SC)=O)CCC(NC(C2(C(F)(F)F)CC(F)(F)C2)=O)CC1C 35892,C1(NC(C2(OCC)CCSCC2)=O)COCCN(C(c2csnc2Cl)=O)C1 35893,N1(C(=O)CCN2CCC2)CCC2(CCCN2C(c2ccccc2Cl)=O)C1 35894,O=C(CC1=CCCC1)NC1COCCN(C(c2cc3n(c2)CCC3)=O)C1 35895,N(C1=NC2CC3CC3C2N1)S(=O)(=O)CCOc1cc(Cl)cc(Cl)c1 35896,C(C(C)(C)CNC(=O)C(CC1CC1)NC(=O)CCOC(C)=O)OC.C(C(C)C)O 35897,c1(C(=O)NC2CC(NC(C3(O)CCCC3)=O)C23CCC3)nnn2c1CSCC2 35898,C(=O)(C1=CCS(=O)(=O)C1)N(C)CC1CCCN1C(=O)CC1CCCC(=O)N1 35899,C#CCC(CC(=O)NC(c1cccc(C)c1)C)NC(c1ccc(O)nc1)=O 35900,c1(C(N2C(CNC(Cc3n(C)ncc3Cl)=O)CCCC2)=O)coc2c1COC2 35901,Cc1nn(CC(N2CCCC(C(C)NC(=O)Cn3nnc(=O)[nH]3)C2)=O)c(=O)o1 35902,C1(C(=O)NC(CC)C2CCC2)CC2C=CC1N(C(=O)CCNC(=O)CO)C2 35903,N1(C(C2CCC(C)O2)=O)CC(CNC(c2cc3ccccc3o2)=O)OC(C)(C)C1 35904,C1(NC(=O)CN(c2ccccc2)CCO)C2CN(C(=O)C(F)=C3CCC3)CC12 35905,N1(C(C(F)=CC)=O)CCC2(NC(c3cccc(Br)c3C)=O)CCCCC12 35906,c1(C(N2CCCC(C(=O)Nc3cnc(Cl)nc3)C2)=O)cnc2ccccn12 35907,N(C1CCc2cc(CNC(=O)Cc3cnc(C)s3)ccc21)C(C(CCC#C)O)=O 35908,C(CC)(CCC(=O)N(CCCC)Cc1ccc(OC(F)(F)F)cc1)NC(C)CC 35909,c1(C(=O)NC2CC3CN(c4nc(CC)nc(C)c4)CC32)ccc2ncsc2c1 35910,C1CC(N(C(=O)C(C)n2cccc2)C)C1.C(C(=O)OCCO)OCCOCCOC 35911,C1(C(=O)NC2COCC2NC(c2cnc(O)s2)=O)(OC)CCOCC1 35912,Cc1cc2ccccc2cc1C(=O)NCC1CCCN(C(C2CC2C#N)=O)C1 35913,C(CC)(CC(=O)NCC1(CO)CCCC1)NC(CC=C)=O 35914,S(=O)(=O)(c1ccccc1)NC(C(=O)NCCCNC(Cc1c(C)cnn1C)=O)C 35915,Cc1cc(F)ccc1C(=O)NC1CCCN(Cc2scnc2C)C1 35916,Cc1cc(C(=O)N(CCCCNC(c2ccc(CO)nc2)=O)C)c(Cl)cc1Cl 35917,N1(C(C(C2CCCN(C(C3CNC(=O)CN3C)=O)C2)C)=O)CC2(CO)CC2(CO)C1 35918,C(CC(=O)N(CC(C)CNC(c1csnc1C1CC1)=O)C)(C(C)C)OCC 35919,CC(=O)n1cc(CNC2CC(C(=O)NCCN3CCNC3=O)C2)c2cccnc12 35920,c1(OCC)nccc(C(=O)NCCC2(NC(c3ccc(F)c(C)c3)=O)CC2)c1F 35921,c1(C(N2C(CNC(Cc3c(SC)cccc3)=O)C=CC2)=O)cccc2c1OCO2 35922,C(c1cnn(C)c1)=CC(=O)NCC(COC)NC(c1csnn1)=O 35923,c1(C(=O)NC(C)C(CO)NC(c2cnc3cccnn23)=O)cccc2nn[nH]c12 35924,c1(C(=O)NCCN(C(CCC#C)=O)CCOC)cc(Br)c(OC)s1 35925,CCCCN=C(NCC1(O)CCC1)NCC1CCCCN1S(C)(=O)=O 35926,CC1CN(C(=O)CCCC2CCC2)CCC1NC(=O)CCc1cncc(Br)c1 35927,C(=O)(CC(C)COC(C1(CNC(=O)OC(C)(C)C)CC1(F)F)=O)OC 35928,C1(NC(c2cc(CC)sn2)=O)C=CCN(C(c2nonc2N)=O)C1 35929,c1(CN2C(C)CC(NC(C3(CF)CC3)=O)C2)cc(C(C)(C)C)cc(C(C)(C)C)c1 35930,c1(CC(=O)OC(C)CC=Cc2ccccc2)ccc(F)c(C(F)(F)F)c1 35931,CCC(C)CC(C(=O)NC1CN(C(C23CCC(C2)C3)=O)C1)NC(=O)OC(C)(C)C 35932,CCC(C)(C)OCC(=O)N(CC(C)CNC(C1(CO)CC1)=O)C 35933,N1(C(c2c(C)nccn2)=O)CCN(C(=O)CC2(O)CCOC2)C(CC2CC2)C1 35934,C1(NC(c2cccc(C#N)c2)=O)CC2CC1CN(C(c1cnc[nH]1)=O)C2 35935,N1(CC)CC2CCC1CN2C(=O)CC1CC(NCc2c(C)cc(C)nc2C)C1 35936,C1(N(C(c2cscc2Br)=O)CC)CCCN(C(=O)CC2CCCC(O)C2)C1 35937,C1(C2CCN(C(=O)CCOCC(F)(F)F)CC2)(NC(C2C(C)CCC2)=O)CC1 35938,CC1(CNC(C2CC(C(F)(F)F)C2)=O)CCN(C(C2(O)CC(F)(F)C2)=O)C1 35939,Cc1ncc2n1CCC(C(=O)NC1(CF)CCN(C(c3ccncc3Cl)=O)C1)C2 35940,C#CCCCCCC(=O)N1CCC2CN(C(=O)CSCC(C)C)CC12 35941,CCCCC(C)CCC(=O)NCCCN(C(C1CCC(OCC)CC1)=O)CC 35942,c1(C(N2C3C(NC(C4CC(OCC)C4)=O)CC(C3)C2)=O)sc2ccccc2c1Cl 35943,c1(OC)cccc(C(N2CCCNC(=O)C2)C(=O)NC(c2ccccc2)C)c1Br 35944,c1(OCC)ccc(C(N2CCC(NC(=O)CC(C)CC)C(C)(C)C2)=O)cc1C#N 35945,C12(CNC(C=CC)=O)COCCN1CCN(C(C13CCC(CC1)OC3)=O)C2 35946,CSC1=C(C(=O)NCCC2(CNC(=O)C(n3ccnc3C)C)CC2)CCCC1 35947,c1(CC)noc(C)c1C(=O)NC1CCCC(NC(c2ccn(C(C)(C)C)n2)=O)C1 35948,N1(C(c2cc(C)sc2C)=O)CC(NC(C2CC3C(C2)C3(F)F)=O)C2(CC2)C1 35949,C1(C(=O)NCC=C2CCN(C(C3(C(N)=O)CCC3)=O)CC2)CNc2ccnn2C1 35950,C1CCN(C(=O)C=CC(C)(C)SC)C1CNC(C1C2CC3C(C2)C13)=O.CC=C 35951,C1(N(C(C=Cc2ccc(SC)s2)=O)C)CN(C(C2(CCF)CCC2)=O)CC12CC2 35952,c1(C(C(=O)O)C2(C3CN(CCF)C3)CC2)ncccn1.C1(=O)CN1 35953,C1(CNC(C(=O)NCCNC(C)=O)=O)C2CCCC1N(C(c1[nH]cnc1C)=O)C2 35954,c1(OC)ncnc(OC)c1-c1nc(C2CCC(F)(F)CC2)nn1C 35955,CCCCCCCCC(=O)N1CCC(N(C(=O)CC2(O)CCOC2)CCC)CC1 35956,N1(C(C2(CC)COC2)=O)CCC2(CC1)CC2(CO)CNC(C1CCCO1)=O 35957,Cc1nc(C(=O)NCC(C)NC(C2(CC3CC3)CCC2)=O)c2ccccn12 35958,Cc1c(C(=O)NC2(C3CCCN(C(=O)CC4CC4)C3)CC2)oc2ccc(F)cc12 35959,c1(C(=O)NCC(CNC(CC(C=C)CC)=O)C)ccc2c(c1)OCCN2 35960,C1(NC(c2c(CC)noc2)=O)CC(CNC(c2cccc(F)c2)=O)C1(C)C 35961,c1(CC)cc(C(=O)NC2CCCC2CC(=O)NCCCC(C)(C)O)ncn1 35962,c1(C(=O)NC2C(NC(c3cc(C)nc(C)c3)=O)COC2)cc2nccn2c(O)n1 35963,C1(C(=O)NC2CCN(C(Cn3c(C)nnn3)=O)C2)CCc2nc[nH]c2C1 35964,N1(C(CC2COCC(C)O2)=O)CCCCC2(C1)CN(C(=O)CCn1cccc1)C2 35965,C1(NC(=O)CC2CC2C(F)(F)F)CCCCN(C(=O)C=Cc2ccccc2)C1 35966,CCCC(C(=O)NCC1(C)CCCN1C(=O)C(F)C(C)C)OCC 35967,C(C)(CC(C)(C)OC)(c1n(CC)nnn1)NCCSc1cncn1CC 35968,S(=O)(=O)(c1ccc(C2CC2)cc1F)N(C(C)C)C1CC1 35969,CCCC(C)(O)CC(=O)N1CC(CC(C)NC(c2cc(C3CC3)ccc2Cl)=O)C1 35970,N1(C(C(C)=C2CC2)=O)C2CCC1C(C(=O)NC(c1ccns1)C)C2 35971,c1(OC)cc2ncc(NC(c3cccc(-c4ccco4)n3)=O)c(Cl)c2cc1OC 35972,N1(C(C2(C)COC2)=O)CCN(C(=O)Nc2cc(Cl)cc(Cl)c2)C2CC12 35973,N1(C(c2nc3c(s2)CCCCC3)C(=O)NCC(F)F)CCC(C2CC(F)(F)C2)C1 35974,c1(C(=O)NCC(CN(C)C(c2ccnn2C(F)F)=O)O)coc2ccc(O)cc12 35975,CC(CCc1ccccc1)CC(=O)N1CCCC1CNC(=O)C=CC1CC1 35976,Cc1[nH]nc(CNC(=O)C(c2cccs2)NC(=O)C=Cc2cncs2)c1C 35977,c1(OC)cc(C(N2CCC(CC(=O)NCC(C)C#N)C2)=O)on1 35978,N1(C(C=NOC)=O)CC2CC(NC(C3(C4CCCO4)CC3)=O)C2C1 35979,C1(COC)CN(C(=O)C(C)(C)n2cccn2)CCN1C(c1cc2n(c1)CCC2)=O 35980,c1(C(=O)NCCC2N(C(CSc3onc(C)n3)=O)CCC2)c(C)cccc1C 35981,Cc1c(C(=O)N(C)CCOCCNC(=O)C(C)C(C)C)cnn1C1CCC1 35982,Cc1ccc(C(N2CCCC(C)(NC(c3cscc3F)=O)C2)=O)c(Cl)c1 35983,C1(NC(C2C(OCC)C2)=O)(CNC(c2cc[nH]c2C2CCC2)=O)CC(F)(F)C1 35984,N1(C(c2ccc(C(=O)OC)o2)C(=O)NC(C)C)CCOC(C2CC(F)(F)C2)C1 35985,C(=O)(C1CCCn2cncc21)NCCOC1CCN(C(c2nc(CC)oc2)=O)CC1 35986,n1(CC)ccc2nc(N(C(=O)C(O)C(C)(C)C)CC3CNC3)ncc12 35987,N1(C(CCC2C(C)(C)C2)=O)CCOC2(CCC(Nc3ncc(Br)cn3)CC2)C1 35988,N1(C(C)C)CCCC1CC(=O)N(C)CC1CCN(C(c2ccsn2)=O)C1 35989,C1(CC(=O)NCc2cccc(Br)c2)COCCN1C(c1cncc(CO)c1)=O 35990,c1(C(=O)NC(CC(C)NC(c2c(C)cn(C)c2)=O)C)ccc(Cl)cc1F 35991,[N-]=[N+]=NC1CN(C(c2c[nH]nc2-c2ccc(Cl)s2)=O)CC1NC(C1CCC1)=O 35992,Cc1[nH]c(C)c(C(=O)NCC2CN(C(c3cn(C(F)F)cn3)=O)CC2O)c1C 35993,c1(CC)onc(C)c1C(N1CCCC(C(=O)NCCCCC(=O)NC)C1)=O 35994,Cc1ncc(Cl)c(C(=O)NCCN(C(=O)C(c2cc(F)cc(F)c2)C)C)n1 35995,N1(C(C(C(CC)C)O)=O)CC(NC(C2OCC2(C)C)=O)CC(C)(C)C1 35996,c1(C(=O)NCCC(C)(C)NC(C(C)OC2CCOCC2)=O)ccc2c(c1)COC2 35997,c1(C(=O)NCC2N(C(C3CC(C)(C)O3)=O)CCN(C)C2)ncnc2c1ccn2C 35998,C1(CCC)(CO)CCN(C(=O)C(CNC(=O)C(C)(CO)OC)CC2CC2)C1 35999,c1(C(=O)OC)cc2c(N3CC(CNC(=O)COCC(F)F)CC3C)[nH]cnc-2n1 36000,c1(C(=O)NC(CNC(c2ccc(C)nc2O)=O)(C)CO)nccc2ccccc12 36001,C1(C(N2CCCC(=C)C2)=O)CC1C1CN(C(C2(C)CNC(=O)C2)=O)C1 36002,Cc1cc(F)ccc1CC(=O)NCC1CC2(CC2)CN1C(=O)C(C)CF 36003,O=C1NC(=O)C2C3CCC(CC3Nc3cccc(F)c3[N+](=O)[O-])C12 36004,CC(C)=C=CC(=O)NC(C)CN(C)C(c1ccc(CN2CCCC2)cc1)=O 36005,C(C(C(=O)N1CC(N(C)C)C2(CC2)C1)C(C)C)NC(c1c(C(C)C)nco1)=O 36006,C1(CNC(=O)Cn2cncn2)(NC(c2cc(Br)no2)=O)CCCC1 36007,C1(CCC)CN(C(=O)C(C(C)C)C2CCC2)CC1C(=O)NCC1(CCC)CC1 36008,C1(C(=O)OC)CN(C(=O)CCCn2cc(CC3(O)CC(C(=O)O)C3)nn2)CC1F 36009,C1(Cn2cc(CC(C(=O)OC)C)nn2)CCCCN(C(C2(F)CC2)=O)C1 36010,CC(CC(=O)NC1C=CC(CNC(c2cc(Cl)n[nH]2)=O)C1)n1cccn1 36011,c1(NC(C2CC2NCc2cnc[nH]2)=O)cc([N+](=O)[O-])c(Br)cc1Cl 36012,C#CCCCCCC(=O)NCCCN1CCN(C(=O)CC2CSCCO2)CC1 36013,Cc1nc(SCCC(=O)N(C2CCN(C(=O)Cc3c[nH]nc3C)C2)C)n[nH]1 36014,c1(C(=O)NCCCCNC(C2CCCN(C(CC)=O)C2)=O)cc(F)c(F)c(F)c1 36015,C1(C(N(C(CCC)Cc2ccccc2)C)=O)CC2CC(=O)C1O2 36016,C1(COCC)CCCN(C(=O)C(C2(C)CC2)NC(=O)CC2CN(C)C2)C1 36017,C(=O)(CCCCC(C)(C)C)N1CCC(NC(COCc2ncc(C)o2)=O)C1(C)C 36018,Cc1nc(C2CCCCC2)nc(O)c1CCC(=O)N1CC(NC(=O)CO)C1 36019,c1(C(N2CCC(NC(c3c(C=C)cnn3C)=O)C2)=O)c(Cl)ccc(F)c1F 36020,N1(C(CCOC)=O)CCC(C)C1C(=O)NCCn1cnnc1C 36021,C1(O)(C(=O)NC2CCN(C(C3CC(C(=O)OC)C3)=O)C(C)C2)CCC(C)(C)CC1 36022,N1(C(C(CN(CC)CC)F)=O)CCC(F)(NC(=O)CC2CCOC2C)CC1 36023,C1(NC(C(=O)N(C)C)=O)CCCN(C(c2coc3c2COC3)=O)CC1 36024,n1(CCC(=O)NC(CNC(=O)CCC2CC2CC2CC2)C2CC2)ccccc1=O 36025,N1(C(C2CC(=C)C2)=O)C2CCC(C(=O)NC(C3CCCCC3)(C)C)C1CC2 36026,N1(C(CCCOC(C)=O)=O)CC(F)(F)CC1CCC(=O)NC1CC1(F)F.CCO 36027,Cn1nc(C(=O)NCCC2CCC(NC(C3(CF)COC3)=O)C2)cc1Cl 36028,C1(NC(C2(CO)CN(C(C(SC)SC)=O)C2)=O)CC2(CCC2)C1O 36029,c1(OC)cc(C(=O)NCCN(C(=O)CCCc2cccc(Cl)c2)CC)cc(Cl)n1 36030,C1(C(=O)NCC2(OC)CC2)CCCCC1NC(=O)C(C)(C)C1CC1 36031,C1(C(=O)NC2CCC(NC(Cc3ccn(C(C)C)n3)=O)C2)CC2(CCO2)C1 36032,Cc1cccc2c1CC(C(N1CCC(NC(c3occc3Cl)=O)C1)=O)O2 36033,Cc1c(CN(c2ccc(-c3ccccc3)cc2)C2CCCCC2C)cccc1F 36034,c1(C(N(CC(C)NC(CC2ON=C(C)C2)=O)C)=O)cn(C)c(C)cc1=O 36035,N1(CCn2c(C)ncc2)CCCC(C(=O)NCC2=CCCCC2)C1 36036,c1(SC)ccc(C(=O)NC(C2CCCC2)CNC(C2C3CCCC23)=O)cc1 36037,N1(C(C(c2ccccc2)C)=O)CCCC1CCCNC(=O)CCc1cccnc1 36038,CN1CCC(C)(C(N2CCC2CNC(=O)C=Cc2ccccc2)=O)C1=O 36039,C1(NC(c2cc(OC)ncc2)=O)CN(C(c2nc(C)ncc2Cl)=O)CC2(CC2)C1 36040,C(=O)(CCCC(F)(F)F)NCC1(NC(c2c(SC)cnnc2)=O)CCCCC1C 36041,c1(CC)cc(C(=O)NCC2CCCN(C(=O)CC3CC(F)C3)C2)cc(O)n1 36042,N1(C(C2(COC)CCCO2)=O)CCCN(C(c2cnn(C3CC3)c2C)=O)CCC1 36043,C1(CNC(=O)Cc2ccc(Cl)s2)CN(C(C2CC3(CCCO3)C2)=O)CC12CCC2 36044,N1(C(CCC=CC)=O)CCOC(C)C1C(=O)NCCC(C)C(C)C 36045,[N-]=[N+]=NC1COCC1NC(=O)Cn1cc(CN2CC3CC3C2)nn1 36046,C1(C(c2n(CCOC)nnn2)NCC2(OC)CCCOC2)CC2(CCC2)C1 36047,n1(CC)cc([N+](=O)[O-])c(C(=O)NCC(O)CN(C(=O)CNC(=O)OC)C)n1 36048,N1(C(c2nc(O)cc(C(C)(C)C)n2)=O)CCC2CCC(C1)S2 36049,C1(C(=O)NC(CCC)C(=O)N(CCS(C)(=O)=O)C)CCCCC1(C)C 36050,Cc1ccnc2ccc(C(=O)NCC34CC3CN(C(C3CCC3(F)F)=O)C4)cc12 36051,N1(CCC(=O)NC(CNC(C2CN(C(=O)NC)C2)=O)(C)C2CCC2)CCCCC1 36052,C1(NC(C2CC(=C)C2)=O)(COC)CCCN(C(c2ccc(F)c(Cl)c2)=O)C1 36053,c1(CC)cc(C(N2CCC(C(C)NC(c3cn(C(C)C)cn3)=O)CC2)=O)nn1C 36054,C(=O)(C(C)CCC(C)(C)C)N.c1(C(C)O)ncc(F)cn1.C12CC(C(F)F)(C1)NC2=O 36055,CC(O)C(C(=O)N1CC(C2CCCO2)C1)NC(=O)COc1cccnc1 36056,c1(OC)nccc(N(C2CNCC2O)C(c2ncccc2N(C)C)=O)n1 36057,N1(C(c2n(CC#C)ccc2)=O)CC(NC(c2cc(CC)cc(F)c2)=O)C2CC2C1 36058,c1(C(=O)NC(C2(CNC(=O)Cn3cnnc3)CC2)C)ccc(CN(C)C)o1 36059,N1(C(c2ccc(C(C)=O)cc2)=O)CCC(CO)C(NC(c2cc(C)[nH]n2)=O)C1 36060,S(=O)(=O)(c1cccc(Cl)c1)N1CCC(C(=O)NCCOCCC)C1 36061,Cc1ccc(C)c(NC(C2(O)CCN(C(=O)Cc3cc(F)ccc3Cl)C2)=O)c1 36062,N1(C(C(C)C)=O)CC(C)(C)OCC1CNC(=O)C(C(C)C)n1cccc1 36063,C(=O)(C(F)C(C)(C)O)N(C)CC1OCCN(C(CC2C(C)C(=O)CC2)=O)C1 36064,N1(C(Cn2ncc(C)c2)=O)CC2CC1CN2c1cc(-n2cncn2)ncn1 36065,c1(NC(C)=O)c[nH]c(C)c1C(=O)NC(C)CCNC(C1(F)CCOC1)=O 36066,N1(C(c2cc(F)c[nH]2)=O)CCCOC2(COC2)C1 36067,Cc1nn(C)c(N2CCN(C(=O)C3CC3)CC2)c1CNC(=O)CNS(=O)(=O)C1CC1 36068,C(=O)(C(CC1CC1)OC)NCC(CNC(C1(c2ccno2)CC1)=O)OC 36069,C(=O)(CC(C(F)F)NC(=O)Cc1ncn(C)c1C)N1C(COCC#C)CCC1 36070,c1(CN2CCC(NC(c3cnc(OCC)nc3)=O)C2)ccc(F)c2ccccc12 36071,C(=O)(C(O)C(C)(C)C)NCC1(O)CN(C(C2(CC=C)CCC2)=O)C1 36072,Cc1cc(C2CCN(C(c3nccn3C(F)F)C(=O)NCCCF)C2)cc(C)c1 36073,C=CCC(C)(C)CC(=O)NCC1CCCC(NC(c2cncc(C)c2)=O)C1 36074,N1(C(C2C(CCOC)C2)=O)CC2(CC(NC(=O)C=CCN(C)C)CO2)C1 36075,n1(C(=O)NCC2CCN2C(=O)Cc2cnccn2)c(-c2cccs2)nnc1S 36076,C(c1c(Cl)nc2sccn12)=CC(N1CC(NC(C2CC3C=CC2O3)=O)C(O)C1)=O 36077,c1(C(=O)OCC)cccnc1N1CCC(NC(c2conc2CC)=O)CC1 36078,Cc1nc(O)nc(C)c1CC(N1CC=C(CNC(=O)CCCN(C)C)CC1)=O 36079,Cc1ccc(F)cc1C(N1CCC(C(F)F)(CNC(=O)Cn2cncn2)C1)=O 36080,CCCN=C(NCC1(C2CC2)CC1)NC1CCN(CC)C(C)C1 36081,CC1CCN(C(=O)CCn2cccc2)CC1NC(c1ccnc(OC(F)F)c1)=O 36082,Cc1ccnc(C)c1C(=O)NCC(C1CC1)NC(=O)CC1CC(C(F)F)C1 36083,c1(-n2c(COC(F)F)nc(C(C)SC)n2)cccc2nc[nH]c12 36084,C12(NC(c3n(C=C)nnc3)=O)CCN(C(c3c(Cl)cnn3CC)=O)CC1C2 36085,c1(C(N2CC(NC(C3CN(C)C(=O)C3)=O)C(O)CC2)=O)nccn2nccc12 36086,c1(C(=O)NCC2CCCN(C(C3CC(C)C3)=O)CC2)cn(C)c(=O)nc1O 36087,C(CCCCC(=O)N1CCOCC(CNC(C2CC23CC3)=O)C1)OCC 36088,C1(NC(C=C(C)C(F)F)=O)CCCCCC1C(N1CCC(C)C1)=O 36089,C1(CC=C)(C(=O)N(CC(C)C)C)CCN(C(=O)CCOC(C2CCCN2C)=O)C1 36090,C1(N(C(=O)C(F)Cc2ccccc2)C)CCCN(C(=O)OC(C)(C)C)CC1 36091,C1(NC(C2CC2C2CCCN(C(C3CC34CC4)=O)C2)=O)CCCCC12OCCO2 36092,C1(NC(C2C(C)=CCS2)=O)CN(C(c2csc(C)n2)=O)CC1(C)C 36093,C12(CNC(C3CC(=C4CCC4)C3)=O)CCC(C1)N(C(=O)COc1ccsc1)C2 36094,N1(C(C(C)c2cccs2)=O)CCC2(CCN(C(c3cnn(C)n3)=O)CC2)C1 36095,c1(SCC#N)cccc(C(=O)NCC(O)CNC(=O)CCN2CCCC2)c1 36096,Cc1cc(C(N2CCC2C(=O)Nc2cnc(Br)c(C)c2)=O)ccc1O 36097,CCCCC(F)C(=O)N1CCC(C(=O)NCC(=O)OCCOC)C12CC2 36098,c1(C(=O)NC2CCCN(Cc3ccc[nH]3)CC2)cn2c(Cl)cccc2n1 36099,c1(N(C)C)cnc(C(N2CCC(NC(c3ccncc3C(F)(F)F)=O)C2)=O)nc1 36100,C1(NC(CC(COC)C)=O)CC2CCC(C1)N2C(c1cnc(O)c(Cl)c1O)=O 36101,N1(C(c2c(C)nc(N)cn2)=O)CCC2CCN(C(c3sccc3F)=O)CC2C1 36102,CC1C(NC(C2C=CCC2)=O)CCN1C(=O)Cc1cn(C)nc1Cl 36103,C=CC(C)(CC)C(=O)NCC1CC1CNC(c1nc(N(C)C)nc(=N)[nH]1)=O 36104,C(=O)(CCCc1cccnc1)NC(CN(C(c1cnccn1)=O)CC)C 36105,N1(CC(=O)NC23CC(CNC(Cc4c(C)n[nH]c4)=O)(C2)C3)C(=O)C(C)C(C)C1=O 36106,c1(C(N2C(CNC(C3CC3C3CCCCC3)=O)CCC2)=O)nc2cnccc2s1 36107,c1(CC)nn(C)cc1C(=O)NC1CCN(C(=O)Cc2cnc[nH]2)C1C(C)C 36108,C12(NC(c3c(C)ccs3)=O)CCCN(C(C3(CS(C)(=O)=O)COC3)=O)CC1C2 36109,C1(C(=O)NCc2c(C(=O)NCCC(COC)O)nco2)OCCCC1(C)C 36110,CCCCC(O)C(=O)NCC1(C)CCN(C(c2ncccc2C2CC2)=O)C1 36111,N1(C(C2C(C(C)NC(Cc3c(C)scc3)=O)C2)=O)CCOC2CCCC12 36112,C(=O)(CN=c1ccc(Cl)n[nH]1)N1CC(NC(CC(CCC)O)=O)C(OC)C1 36113,C1(C(=O)OC)CC(C)(C)CN1C(CCC1CCCC1)C(=O)NC1CCCC1 36114,N1(C(C(C(C)C)c2cccnc2)=O)C2CCC1C(CNC(=O)C=C1CCC(C)C1)C2 36115,C(CCCCOCCc1cc(C(=O)OC)no1)NC 36116,c1(C(=O)NC(CCNC(c2c(CC)nns2)=O)C)cc(Cl)ccc1OC 36117,c1(C(=O)NCC(C2CCCCCC2)NC(CCOCC#C)=O)nnc(O)cc1O 36118,N1(C(CSC)=O)CC2CC3CC2C1C3NC(=O)CCc1ccc([N+](=O)[O-])cc1Cl 36119,Cc1snnc1C(=O)NCCOC1CCN(C(c2cnn(-c3nccs3)c2)=O)C1 36120,C1(NC(CN(C)CC)=O)(CC)CN(C(=O)CC(C)c2ccccc2)C1 36121,CCC(C)(COC)C(=O)NC1CN(C(c2cccc(F)c2C)=O)CC1F 36122,CC1Oc2ccc(C(=O)NC3CN(C(C4(C)CCCS4)=O)C3)cc2NC1=O 36123,N1(C(C23C(C)(C)OCC2C3)=O)CCC2CN(C(c3ccnc4ccnn34)=O)CC12 36124,c1(C(=O)NCc2ncoc2CCNC(C2(CCF)CCC2)=O)ccnc(S)c1 36125,c1(OC)ccc(Cl)c(C(=O)NC(C)CCN(C)C(C2CC(C3CCC3)C2)=O)c1 36126,c1(C(N2CC3CN(C(C4CCC(C)O4)=O)CC32)=O)cc2ccc(Cl)cc2[nH]1 36127,c1(C(C)C(N2CCCC2CNC(c2cnoc2C2CCC2)=O)=O)ccc(F)cc1 36128,c1(N(C)CC2C(C)C2)ccc(S(=O)(=O)N2CCCN(C)CC2)cc1Cl 36129,N1(C(CSCC)=O)CCC(NC(c2ccc3c(c2)CCO3)=O)C(F)(F)CC1 36130,n1(CC)ncc(C(=O)NCCn2cc(CNC(c3c[nH]c(=N)s3)=O)nn2)n1 36131,CCC(C)CC(C)N(C(=O)CCNC(c1cn(C)cc1C)=O)C 36132,c1(C(N2C(CNC(c3ccccc3F)=O)CC2)=O)cc2ccsc2c(=O)[nH]1 36133,c1(C(=O)NCC2CC(C)CN(C(=O)CCCC(C)(C)C)C2)nn(C)cc1[N+](=O)[O-] 36134,N1(C(CC(=O)NCC)=O)CCCCC1C(C)(C)CNC(c1cc(C)c(C)o1)=O 36135,c1(C(C)NC(=O)CN2CCN(C(C3(O)CC3)=O)CC2=O)ccc2n[nH]cc2c1 36136,C1(NC(C(CC)NC(N)=O)=O)CN(C(=O)C(C)OC)CC2CC12 36137,c1(C(=O)NCC(CN(C(C2CCN(CC(C)C)C2)=O)C)C)cc(S(N)(=O)=O)co1 36138,C(=O)(CC(C)C(F)F)NCC(CC)(C)NC(=O)CCc1nc(C(C)(C)C)no1 36139,CC1(C)CCCCCC1NC(C1COCCC1NC(C1CCCCC(=O)N1)=O)=O 36140,Cc1ccc(F)c(C(N2CCC(NC(c3ncsc3S(N)(=O)=O)=O)CC2)=O)c1F 36141,C1(C(=O)OC2(c3c(OC)ccc(F)c3)CC2)CC(O)C12CC(F)(F)C2 36142,CC(CC(=O)NCC1CCN(C(=O)OC(C)(C)C)C1)NC(=O)CN1CC(C)(C)C1 36143,C=C(Cl)CCC(=O)N1CCC(CN(C(c2ccn(CCF)n2)=O)C2CC2)CC1 36144,C(=O)(C(CC)CC(F)(F)F)N1C(CCCNC(C(C#C)(C)C)=O)CCC1 36145,O(C1CCCc2ccccc21)CC(=O)N(CCCNC(C1(O)CC1)=O)C 36146,Fc1cc(Nc2nccc(C(F)F)n2)cc(-c2csc(NCc3ccccc3)c2)c1 36147,c1(OC(C)C(=O)N(S(C)(=O)=O)CCO)ccc(F)cc1 36148,C1(C(=O)NC2CC(C)OC2=O)CN(C(C2CCC(O)C2)=O)CC(C)(C)C1 36149,N1(C(C2CCC(CC)CC2)=O)CCCC2CN(C(=O)Cc3ccsn3)CCC12 36150,c1(OCCC(N2CCC(C(=O)NCC3(n4ccnc4)CC3)C2)=O)ccccc1 36151,C1(NC(c2cc(OC)ncc2)=O)CC2CN(C(C3CCOC3)=O)CC2C1 36152,C1(C)(CNC(Cc2nnc(C)s2)=O)CCCN(C(=O)CC2COC3CC2C3)C1 36153,c1(CC(=O)N(C)CC2(CNC(C3C=CC(C(=O)OC)C3)=O)CC2)ccc(Cl)cn1 36154,CC(C)=C=CC(=O)NCC1(NC(=O)C(c2ccccc2)F)CCOCC1 36155,C12(CNC(c3n(COC)ncc3)=O)CCC(NC(c3cn[nH]c3)=O)(CO1)C2 36156,N1(C(C=CCOC)=O)CC2CCC1C(CNC(=O)C(CO)NC(=O)C(F)(F)F)C2 36157,N1(CC(=O)NC(c2ccc(-c3ccc(Cl)cc3Cl)nc2)C)CCc2[nH]nc(O)c2C1 36158,c1(C(=O)NC(CN(C(c2ccn(C3CCC3)n2)=O)CC)C)nc(C)sc1C 36159,C1(CC(=O)NCC(CC)NC(c2cnc(S)n2C(F)F)=O)C=NN(C)C1=O 36160,c1(C(=O)NCC(C)(C2CC2)NC(c2ccc[nH]2)=O)cccc(S(=O)(=O)CCO)c1 36161,C12(NC(CCc3n(C)cnc3)=O)CN(C(c3cccs3)=O)CC1CS(=O)(=O)C2 36162,Cc1cc(C)c(C(=O)NCC2(O)CC(NC(=O)Cn3ccnc3C(C)C)C2)o1 36163,C1(CNC(CCCOCC=C)=O)CN(C(c2cn(CCCC)nn2)=O)C(C)(C)C1 36164,c1(C(=O)OCCCNC(=O)CSC2CCCC2)cc(F)cc(Cl)c1 36165,CCC(C(=O)NC1CCC1C(=O)NC1CCOCC1O)C(F)(F)F 36166,C1(CCNC(C2(CCOC)CC2)=O)CN(C(c2c(OC)nn(C)c2)=O)CCO1 36167,N1(CCNC(CCCOC)=O)CCN(C(c2ccc(C(N)=O)s2)=O)CC1 36168,C(C1CCN(C(=O)CCCN=[N+]=[N-])CC1)=CC(=O)NCc1cccc(CC)c1 36169,N1(C(C(CC)C)=O)CCCC(C)(C(=O)Nc2cn(C)nc2C(N)=O)C1 36170,C1(C(=O)NCC(C)(C)OCCNC(C2CC2Cl)=O)Cc2ccccc2C1 36171,C1(C(N2CCC3(C(NC(c4ccoc4Cl)=O)C3)C2)=O)COC2COCC2O1 36172,Cn1ncc2c(N3C4CCCC3CC4)nc(=NCCC3CCC4(CC3)CC4)[nH]c12 36173,c1(CC(=O)NCC2(C)CC(NC(=O)Cc3ccsn3)C2)c(F)cccc1Cl 36174,n1(CCC(=O)NCC(=O)N(CCCOC)C)sc2ccccc2c1=O 36175,C(=O)(CCCC(C)CC)NC1(C#C)CC1.C(=O)(C1CN1C)OC 36176,N1(C(CSCC=C)=O)CCC2(CC(C(=O)NC3CC4CC3C(O)C4O)C2)C1 36177,C1(C(N(CC(=O)OC)C2CC2)=O)C2CCC(C2)N1C(=O)C(C1CC1)C1CC1 36178,C1(NC(c2cnn(C3CC3)c2)=O)CC2CN(C(=O)C3=COCCO3)CC2C1 36179,N1(C(c2c(N)cn(C)n2)=O)CC(NC(c2cc(C(C)(C)C)on2)=O)CC2(CC2)C1 36180,N1(Cc2ncc(C)s2)CCC(C(C)NC(c2ccncn2)=O)CC1 36181,C1(C(N2CC(N(C)C(c3ncoc3-c3cccs3)=O)C2)=O)C2CS(=O)(=O)CC12 36182,N1(C(c2ccon2)=O)CC2CCC(C1)N2C(=O)C(c1cccc(Br)n1)(F)F 36183,c1(C(N(CCCCNC(CN(CCC)C)=O)C)=O)cc(C#N)ccc1Br 36184,c1(SC)ccc([N+](=O)[O-])c(C(=O)NC2CC(CCNC(=O)CC(C)C(C)C)C2)c1 36185,C(=O)(CCC(=O)N1CCCCC1C(C)NC(C1CN(CC(C)C)C1)=O)NCCC 36186,C1(C(=O)NCCC)CCN(Cc2cccc(I)c2)CC1F 36187,C1(COC(c2ccn(CC(F)(F)F)n2)=O)CCCCN1Cc1nn[nH]n1 36188,C1(NC(CSC(C)C)=O)CC2(CCN(C(c3csc(C4CC4)c3)=O)CC2)C1 36189,CN1C2CCC1CN(C(C1COCCN1C(c1ccc(O)c(C#N)c1)=O)=O)C2 36190,Cc1cc(CC(=O)NCC2C=CC(NC(c3nccn3C)=O)C2)n(C)n1 36191,C1(C(=O)NCc2ccc(C)c(C)c2)N(C(=O)CCc2ccoc2)CC12CCCC2 36192,Cn1ncc(Cl)c1C(=O)NCC1C=CCN1C(=O)CCn1ccccc1=O 36193,C1(C(=O)NC2CC(C3CNC3)C2)CNc2ccnn2C1 36194,c1(CCC)ccc(C(=O)NC2CC(F)(CNC(C3(C)CCC(=O)N3)=O)C2)cc1 36195,c1(OC)cc(CC(N2CCC(C)(NC(c3cc(C(C)C)on3)=O)C2)=O)cc(Cl)c1 36196,N1(C(CC2(C=C)CN(C(c3cc(Cl)n[nH]3)=O)C2)=O)CC2(CC(O)C2)C1 36197,N(C1CCCn2cnnc21)C(C)C(=O)Nc1ccc(N2CCOCC2)cc1 36198,Cc1ccc(-c2nc(C(=O)NCC(C)(C)NC(C3CCC3F)=O)cs2)n1C 36199,Cc1ccc2cc1NS2(=O)=O.N1(C(=O)CC2CC2C)CC(C)NC(C)C1 36200,c1(CC(=O)NC2C(NC(C(C=C)O)=O)CCCC2)nn(C)c2ccccc12 36201,C1(OCCNC(=O)Cc2ccon2)CCN(C(=O)CCC2CC2(Cl)Cl)C1 36202,C(=O)(CC(CNC(=O)CN1CCC(=O)CC1)C1CCC1)NC(C=C)C1CC1 36203,C(=O)(CC(c1ccccc1)C1CC1)NC1C(NC(C(=O)NCC(F)(F)F)=O)CC1 36204,c1(CCC(N2CCC(NC(C3(F)C(C)C3)=O)C23CC3)=O)ccc([N+](=O)[O-])cc1 36205,C(=O)(CCS(=O)(=O)c1ccccc1)NC(CC)CN(C(=O)C(C)CC1CC1)CC 36206,CCCC(CC)CC(=O)NCC12CC(CN1C(c1cccc(C#N)c1)=O)C2 36207,C1(F)(C(N(CCC)CCNC(C2CC2C(F)(F)F)=O)=O)CC1C 36208,C(=O)(CCCN(C)N=O)NCCC1CC(OC)CN1C(=O)C(C)NC(C)=O 36209,C(=O)(CCCCN=[N+]=[N-])NCC(CN(C(C1(C2(C)CC2)CC1)=O)CC)(C)C 36210,N1(C(CN(C)C(C2(C)CCCS2)=O)=O)CCN(C(c2nccn2C)=O)CC1 36211,N1(C(C2N(C(C3C(C=C)C3)=O)CCOC2)=O)CC(C2CC2)(COCC)C1 36212,N1(C(c2ccc(C)c(F)c2)=O)CCCCCC(NC(C2(C)CC2(F)F)=O)C1 36213,C#CCCC(CCc1ccccc1)OC(c1ccc(Br)c(O)c1)=O 36214,N1(C(CCC2(NC(c3occ(C)c3)=O)CCCC2)=O)Cc2cccc(C)c2C1 36215,Nc1ncc(C(=O)NC2CC(NC(c3ccccn3)=O)C2)cc1-c1ccccc1 36216,c1(C(N2C(C(C)NC(c3sccc3Br)=O)CCC2)=O)cccc(=O)n1C 36217,CCCC(C(=O)NC(C)CN(C(=O)CC1(OC)CCOCC1)C)c1ccccc1 36218,N1(C(CCC(=O)N(C(C)C)C)=O)CCN(C(c2coc(C(F)(F)F)c2)=O)C(C)C1 36219,C1(C(N2CCC(N(C(c3c(Cl)ccc(OC)c3)=O)C)C2)=O)CCc2nccn2C1 36220,Cc1cc(C(N2CCCC2C2(NC(=O)CC3CCCOCC3)CC2)=O)cc(N)c1 36221,C(=O)(C1CCCn2c(C)cnc21)NCC1CCCN(C(CCC#CC)=O)CC1 36222,N1(C(C)C)CC(NC(=O)CCCNC(C2CS(=O)C2)=O)C(C)C1 36223,c1(NC(CN2C(C)CC2)=O)cccc(NC(=O)Cn2ncc(Br)n2)c1 36224,C1(COC2CCN(C(C(C)O)=O)C2)CCN(C(C2CC(F)C(=O)N2)=O)CC1 36225,CC1CC=C(C(=O)N2CCCC(CC(=O)NC3(C)CCCCC3)C2)CC1 36226,c1(CN2CC(CCC)C(C(=O)ON3CCCCC3)C2)ccc(SC)c(C)c1 36227,N1(C(C(CC(=O)OC)C)=O)CC2(CCCC2)C1C(=O)NCCC1(O)CCCCC1 36228,C1(C(C)C)CCN(C(c2cc(CNC(=O)C(C)n3cccn3)on2)=O)C1 36229,C=CCC(F)(F)CN(C(=O)C(C1CCN(C(=O)C(C)C2CC2)CC1)C)C 36230,c1(C(=O)NCCOCCCN(C(C2(CC)CC2)=O)C)cc2c(cc1Cl)CCCC2 36231,c1(C(=O)NC2CCC(CCNC(c3c(OC)csc3)=O)C2)cn(C)c(=O)cc1C 36232,Cc1ccc2c(c1)CC(N(C(=O)COc1nc(C(C)OC(C)C)no1)C)C2 36233,C1(CNC(c2ccc(N3CCC3)nc2)=O)CN(C(c2nccnc2Cl)=O)CCO1 36234,N1(C(C)=O)CC(C)OC2(CCN(C(c3c(C)nc(C(C)(C)C)nc3S)=O)CC2)C1 36235,c1(COCC)nc(C)c(C(=O)N(C)CCNC(c2nc(C3CC3)cs2)=O)s1 36236,C12(CNC(=O)CC3CC(F)C3)CCC(NC(C3CC4CCC4C3)=O)(CC1)CO2 36237,c1(C(N2CC(NC(C3CCCSC3)=O)C(F)CC2)=O)cnc2n1CCOC2 36238,C1(CNC(c2ccnc(CO)c2)=O)CC2CC2N1C(=O)COCC1CCOCC1 36239,C1(NC(c2cnc(OC)s2)=O)CCCN(C(=O)Cc2cccc(F)c2F)C1C 36240,c1(C(C)NC(C2CN(C)C2)=O)ccc(CNC(c2ccc(C#N)[nH]2)=O)cc1 36241,N1(C(COC(C)=O)=O)CCC2(CCCN(Cc3cc(Cl)c(O)cc3F)C2)CC1 36242,N1(C(C2(C)C=CCC2)=O)CC(C2CN(C(=O)C(C)(C)S(C)(=O)=O)C2)C1 36243,c1(CNC(C(C)SC(F)(F)F)=O)cnn2c1CN(C(=O)CC1COC(=O)C1)CC2 36244,C1(C(=O)NCc2ccc(C(N(CCCC=C)CC)=O)s2)CC(C)(C)CN1C 36245,C(=O)(CCCCC#N)N(CCC(C)NC(=O)CC1CCC(F)(F)C1)C 36246,C1(CNC(C(C#C)(C)C)=O)CCCC2(CCN(C(c3nc(C)oc3C)=O)CC2)O1 36247,c1(C(=O)NC(CN(C(C2CCCCC2)=O)CC)C)cc(F)ccc1O 36248,N1(C(C(C2CCC2)OCC)=O)CC(NC(=O)CCn2cc(C)cn2)C(C)C1 36249,n1(CC#C)cccc1C(=O)NC(C)CNC(c1cc(C2CCC2)no1)=O 36250,c1(CC(=O)NCCC(C)NC(CC(CC)OC)=O)cccc(F)c1F 36251,c1(OC)ccc(F)c(C(=O)NCC2CC3(CC3)CN2C(=O)CC2CNC(=O)C2)c1 36252,C1(NC(C(CC)CC(C)C)=O)CCCC12CCN(C(=O)CC1CC(F)(F)C1)CC2 36253,N1(C(c2c(C)[nH]cc2)=O)CCC(CO)C(NC(=O)Cc2cn(C)cn2)C1 36254,C(=O)(C(O)CCNC(C1CC1(C)C(F)F)=O)NCc1nnn(CC)n1 36255,C=CC1CN(C(=O)CCS(C)(=O)=O)CC1NC(=O)C(C1CC1)SC 36256,C1(c2n(C)ncc2)CN(C(=O)C(NC2=NCCS2)=O)CCO1.C(CCC1CCC1)N 36257,C=C(C)CC(=O)OCCN(C1CCCCC1)C(C1CCCN1C(C)=O)=O 36258,N1(C(C2CCCOC2)=O)CC2CCN(C(C3(O)CCSCC3)=O)CC12 36259,N1(C(C(C)(C2CC2)OC)=O)CCN(C(C23CC2COC3(C)C)=O)CC(O)C1 36260,N1(C(C(c2ccccc2)C)=O)CC(NC(c2c[nH]c(=O)cn2)=O)C(C)C1 36261,N1(C(C2(CC)CCCC2O)=O)CCC12CN(C(=O)CCCC1CCOCC1)C2 36262,CCCCCC(C)(C)C(=O)N(C)CCN(C(=O)Cn1cc([N+](=O)[O-])cn1)C 36263,C(CCCCCCCO)=CC(=O)NC1COCC1CNC(=O)CCCCCC#N 36264,C#CCC(CC(=O)NC1CC2(NC(c3cn(C)nn3)=O)COC1C2)c1ccccc1 36265,C(=O)(CC(C)C(C)C)NCC1(NC(c2cn(CC(CC)O)nn2)=O)CCOCC1 36266,c1(C(N2CC=CC(NC(C=CCN(C)CC)=O)C2)=O)cc[nH]c2nccc1-2 36267,C(c1cccc(C)c1)=CC(N1CC(NC(C(CC)Oc2ccccc2Cl)=O)C1)=O 36268,C1(C(=O)Nc2cccc(NC(c3cnn(C)n3)=O)c2)CC2(C1)CC2(F)F 36269,C1(C(=O)NC2(COC)CC2)CC12CC(NC(=O)CCC1CCCO1)C2 36270,c1(NC)ccccc1C(=O)NCCCN(C(=O)CN1CCCNC1=O)C 36271,C1(CNC(=O)COC2CCCC2)C(C2CC2)CCN1C(C12CCC(F)(CC1)C2)=O 36272,C(CC(CC)C(=O)NC(c1cnn(C)c1)C(=O)NC(COCC)C(C)C)=CC 36273,Cc1ccc(-n2nnnc2CNC(c2cnn(C3CNC3)c2)=O)cc1 36274,O(NC(=O)C(O)CNC(=O)C(O)C(F)(F)F)C(C=C)C 36275,n1(CC(=O)NCC(CC)N(C)C(c2cnc(C3CC3)s2)=O)nnc(C2CC2)n1 36276,c1(C(=O)NC2CC3(CC(NC(C4C(C(=O)OC)C4)=O)C3)C2)ccnc2[nH]cnc12 36277,N1(C(c2ccc(CCC)s2)=O)CCCCC(NC(C2CCN2C2CCCC2)=O)C1 36278,C(=O)(C1CCCc2ncc(C)n21)N1CCC(NC(CCc2nnc(CC)o2)=O)C1 36279,c1(OC)ccc(C(=O)C=CC(=O)NC2CCC(NC(=O)C=CCO)C2)cc1OC 36280,CC1CC(F)(F)CN1C(=O)C=CC(C)(C)NC(=O)C=CC1CCC1 36281,CCCC(C(=O)N1CCN(C(=O)Cc2ccc(OCC)cn2)CC1C)C(C)C 36282,C(C1CCOCC1)=CC(=O)NC1CC(NC(C2(C(N)=O)CCC2)=O)C1 36283,c1(C(=O)NCC2(F)CC(NC(CC(CN(C)C)O)=O)C2)ncnc2sccc12 36284,C=C=CC(C)C(=O)NC1(C)CC(NC(=O)CCc2nc(-c3ccoc3)no2)C1 36285,C(=O)(C(C)(C)CC#N)NC1C(NC(c2c(SC)cn(C)n2)=O)COCC1 36286,N1(C(CN(C(C)CNC(c2nn(C)cc2Cl)=O)C)=O)CCCC(C(N)=O)C1 36287,c1(C(=O)NCC2C(CNC(CNS(CC)(=O)=O)=O)C2)cc2oc(C)c(C)c2[nH]1 36288,c1(OCC)ccccc1C(=O)NC(c1cnc[nH]1)C 36289,C1(C(=O)NCCOCCN(C(C(C)=C(CC)C)=O)C)CCCC(=O)N1C 36290,c1(C(=O)OCCCC#C)nnc(C(F)F)s1 36291,C1(C(=O)NC2CCC(NC(=O)Cc3ccccc3F)CC2)(COC)CCOCC1 36292,C=CC(CCC)CC(=O)NCC1CCN1C(c1cc(F)c(N)c(F)c1)=O 36293,N1(C(C2CCN(C)C2=O)=O)CC2CN(C(c3cnc4ccsc4c3)=O)CC2(C)C1 36294,N1(C(C(F)=CC)=O)CCCCC1C(C)(C)CNC(=O)CC(C)N(C)C 36295,C1(C(=O)NCCNC(C2CN(C(c3ccc(C)o3)=O)C2)=O)CC12CCCCC2 36296,c1(C(=O)NCC2N(C(c3cc(COC)no3)=O)CC2)ccc([N+](=O)[O-])cn1 36297,CCC(CNC(C1(CCNC(=O)CCC2CCCC2)CC1)=O)CCO 36298,Cc1ccc(C(=O)NCC2(F)CCN(C(=O)CC3CC=CCC3)CC2)c(O)n1 36299,N1(C(C(C)SC)=O)CC(NC(C2CCC(C(F)(F)F)O2)=O)C(CO)C1 36300,C(=O)(C(COC)CC(C)C)NC1(CC=C)CN(C(=O)C(C)=CC(C)(C)C)C1 36301,C12(C(=O)NCC3(C)OCCN(C(Cc4nnc(C)o4)=O)C3)CCCCC1C2(F)F 36302,Cc1ncnc(N2CCC(CCNC(c3ccc(=O)n(CC4CC4)c3)=O)C2)c1F 36303,C1(C(C)Nc2cccc(COCCO)c2)CCCN(CC(c2ccccc2)O)C1 36304,c1(CC(=O)NC(CNC(C(C)OC)=O)(C)C)c(Br)ccc(Cl)c1F 36305,C(Cc1cnc[nH]1)(C(=O)N1CC(C)(CN(C)C)C1)NC(CN(C(C)=O)C)=O 36306,c1(C(N2CC(CNC(c3[nH]nnc3C3CC3)=O)C2)=O)cc2c(F)cc(F)cc2[nH]1 36307,c1(C(=O)NC2CC(CNC(C(CC)n3cncn3)=O)C2)cc(C)nc(O)n1 36308,C1(CC(=O)NCC(C2CCN(C(=O)C=Cc3cc[nH]n3)CC2)C)CCCCN1C 36309,C(=O)(C1COc2ccccc21)N(CCNC(CSCCC)=O)CC 36310,CC1CCC(CNC(c2coc(CNC(C3(C)CSC3)=O)c2)=O)N1C 36311,c1(C(=O)NC2(C)CC(NC(c3ncnc(C)c3C)=O)C2)cc2nc(=O)ccn2[nH]1 36312,N1(C(C(C(n2ncc(C)c2)C)NC(=O)OC(C)(C)C)=O)CCN(C)CC1(C)C 36313,CC1(C(=O)NCCCCCNC(=O)CNC(c2ccncc2)=O)CCC(=O)NC1 36314,C1(NC(CSCCC)=O)CC(C)CN(C(c2c[nH]nc2Br)=O)C1 36315,c1(CNC(NC(COC)C)=NCCc2cn3c(n2)SCC3)ccc(C#N)c(F)c1 36316,c1(C(=O)Nc2c(C(=O)OC)scc2)ccccc1N1CCNC1=O 36317,C=C=CC(C)C(=O)NC(CNC(c1cc(C)n(CC)n1)=O)CC 36318,n1(CCC(=O)NCC2CC(OC)CN2C(=O)Cn2cnnn2)ccc(O)nc1=O 36319,C1(NC(c2cncc(NC)n2)=O)CN(C(=O)CCc2cc(C)no2)C(C)(C)C1 36320,C(=O)(C#CC(C)(C)C)NC(CCNC(C=NOC)=O)(C)C.N1CCN(CCO)CC1 36321,CC1(CNC(=O)CC2CCSCC2)CCCN(C(C2CC3(C2)CC32CC2)=O)C1 36322,c1(N2CC(C)C(N(C)C)CC2)ccc(S(=O)(=O)NCc2ccnc(C#N)c2)cn1 36323,N1(C(CCC=CC)=O)CC(CNC(=O)COc2cc(C)ccc2C)OC(C)(C)C1 36324,Cc1cc2cc(F)ccc2n1CCNC1CC(C)S(=O)(=O)C(C)C1 36325,CC(C)CC(O)CC(=O)N1CC(C)C(C)(CNC(C2(C(C)C)CC2)=O)C1 36326,Cc1ccc(C(=O)NC2CCC(C)N(C(c3ccnc(F)c3F)=O)C2)cc1N 36327,Cc1ccc(CC(=O)NC2CC2CNC(C2C(C)(C)C2(F)F)=O)cn1 36328,C1(NC(c2cnc(C)s2)=O)(CNC(=O)Cc2cccc(F)c2)CCCCC1C 36329,N1(C(=O)NC(c2cc[nH]c2)C)CC2C(Cc3ccc(Cl)cc3)C2C1 36330,c1(C(N2CCCC(CN(C(C(CC#C)C)=O)C)C2)=O)c(C)nn(CCO)c1C 36331,CC1CCCN(C(=O)CC(C)(C)C)C1CNC(=O)CCc1cnccn1 36332,C1(CC)CCC2(CC1)NC(=O)N(C(=O)Cc1ccc(Cl)s1)C2=O 36333,Cc1cc(C(=O)N(CC(C)C(=O)NCc2nn[nH]c2C2CC2)C)n(C)n1 36334,c1(OC)cc(CC(N2CCC(NC(C3CCCOCC3)=O)C2(C)C)=O)ccc1C 36335,C1(CNC(CCC(=C)Cl)=O)CN(C(c2c(N)cc(Cl)cc2F)=O)CC2(CCC2)O1 36336,CCC1=C(C(=O)NCCN(C2CCCC2)C(C2CCCC(F)C2)=O)SCCO1 36337,Cc1cc(O)ncc1NC(C1CCC(C2CC2)N1C(c1nnn(C)c1N)=O)=O 36338,CC(C)C(CN(C)C)C(=O)N(C(CC(F)F)C(=O)N(C)CCC1CCCN1C)C 36339,C1(CNC(Cc2cccc(OC)c2)=O)CC(F)(F)C12CCC2 36340,N1(C(C(=O)NCC(c2cccs2)C)=O)CCN(C)CC2(C)CCCC12 36341,C1(CNC(c2n(C(C)C)ccn2)=O)CC(C)N(C(=O)C(N2C(=O)CCC2=O)C)C1 36342,N1(c2c(C#N)cccn2)CC2CCC1CC2C(=O)O 36343,Cc1cc(C(N2CC(NC(c3cc(C4CCCC4)[nH]n3)=O)C3CC23)=O)c(C)cn1 36344,c1(NCCCOc2c(C)cccc2)cc2[nH]nnc2cc1F 36345,C(=O)(C(CNC(c1oncc1CC)=O)CC(C)C)NC1(CC#C)CCC1 36346,C1(N(C(=O)CC2CCC3CC23)CC)CCN(C(=O)Cc2ccccc2F)CC1 36347,CC1CN(C(c2cc(CF)on2)=O)CC(C)C1NC(c1csc(C(F)F)n1)=O 36348,N1(C(C2CCOC2)=O)CCCC(Cn2cc(C3CC=CCC3)nn2)C1 36349,C=C=CCC(C(=O)N(C)CCO)NC(=O)OC(C)(C)C.c1(C(N(C)C)=O)cscn1 36350,C1(NC(CCCC=C)=O)CC2CC1N(C(=O)CCc1ccsc1Cl)C2 36351,N1(C(C(C(C)(C)C)n2cc(CC3(O)COC3)nn2)=O)C2CCC1CC(F)C2 36352,c1(OS(CC2C(C)(C)OCC2)(=O)=O)c(-c2ccccc2)nc2ncccn12 36353,C=Cc1ccccc1N(c1nccn1N)C(c1cscc1C)=O 36354,c1(C(N2CCN(C(c3cn(CC)nc3)=O)C(CO)C2)=O)cccn2c(O)nnc12 36355,CCC(C)(C)C(C)CC(=O)NC1CCC1CNC(=O)Cn1cnc(C#N)n1 36356,CCC(CCC(=O)N1CCC(C(C)=O)CC1)OC 36357,C(C(=O)NNC(=O)c1ccc(Cn2cccn2)o1)Oc1cccc(CC#N)c1 36358,C1(C(NOCCOC(C)C)=O)CC(NC(=O)CCC2CCCN2C)C1(C)C 36359,C1(CC(=O)NCC(CCOC)NC(=O)CN2CCS(=O)CC2)COC(C)(C)CO1 36360,C(=O)(C(F)CC(C)(C)NC(=O)CCC(N)=O)N1CCCC(CCC)CC1 36361,c1(C(=O)NCC2N(C(C3C(C)=C3)=O)CCC2C)cnc(F)cc1C 36362,C1(NC(CC2N(C)CCC2)=O)COCCN(C(=O)CCSCC(N)=O)C1 36363,c1(OC)ccc2[nH]cc(C(=O)NC(C)CC(C)NC(=O)CSC3CC3)c2c1 36364,N1(C(C(C)OCC(C)C)=O)CCC2(CCC2)C(NC(=O)CSC2CC2)C1 36365,C#CC1CN(C(=O)Cc2ccc(Cl)s2)CCN1C(c1cc(C(C)(C)C)[nH]c1C)=O 36366,C#CC1(C(=O)NCCC(=C)CNC(=O)CN2CCC(OC)C2)CCCCC1 36367,Fc1cc(F)c2[nH]c(=NC3CCCOC3)[nH]c(=NCC3(Cl)CC34CCC4)c2c1 36368,C(CCCC(C)(C)C)n1c(NC)nnc1-c1cccn1C.C1CCOC1 36369,c1(CNC(CC2N(C(CC(C)c3ccco3)=O)CC2)=O)ccc(O)cc1 36370,C1(NC(CCOC)=O)CC=C(C(=O)NCC2CC3C=CC2O3)C1 36371,N1(C(Cn2c(C)nc(C)n2)=O)CCC2(CC1)CCN(C(C1(C(F)F)CC1)=O)CC2 36372,N1(C(C(=O)NCC(=C)C)C(C2CCOC2)OCC)CCC2(CC1)NC(=O)NC2=O 36373,c1(C(N(C(CCNC(c2c(CC)ncnc2)=O)C)C)=O)ccc(C(C)C)nc1C 36374,CN1CCN(C(c2cc(CNC(=O)CCc3ccsc3)[nH]n2)=O)CC1CO 36375,Cc1nc(N)c2c(C)c(C(=O)NCc3ccc(CNC(=O)C(C)O)cc3)sc2n1 36376,N1(C(C(C)SCC)=O)CCc2sc(CNC(c3cc(F)c(C)cc3O)=O)nc2C1 36377,c1(CC)ncc(C(=O)NC2COCC2NC(=O)CCC2CC2(F)F)c(C)n1 36378,C1(C(=O)Nc2scc(C(=O)OCC)n2)C(C2CC2)CCN1C(C1CCCO1)=O 36379,C(C)(C)(C(=O)NC1CCC1C(=O)NCCCN1CCCC1C)SC 36380,C(=O)(CCCCCC(C)C)NCC(CC)NC(C12CC(CC(C)O1)C2)=O 36381,N1(C(=O)Nc2cc(C)c(C(F)(F)F)cn2)CCC(N=c2[nH][nH]c(=N)[nH]2)CC1 36382,c1(C(=O)NC2CCN(C(C3CCNC(=O)C3)=O)CC2)ccnc2ncccc12 36383,C1(CC)CN(C(=O)C(C2CCC2)NC(c2ccnnc2C)=O)CCO1 36384,N1(C(Cc2cc(C)no2)=O)CCC2CCN(C(C3CC3C(F)F)=O)C2C1 36385,c1(NC2(CNC(C3CC(CC)OCC3)=O)CCC2)ncc(S(C)(=O)=O)cc1Cl 36386,C#CCN(OC)C(=O)CC1(NC(c2ccn3ccccc23)=O)CCCCC1 36387,CCC(O)C(C)(C)C(=O)NCC1CCN(C(=O)CSCCC(C)C)C1 36388,Cc1c(C(=O)NC2CCC2CNC(C2COC(=O)N2)=O)[nH]c2c(C)cccc12 36389,C1(CC(=O)NC2C(C)CN(C(=O)CNc3nccs3)C2)Cc2cc(F)ccc2O1 36390,CC1(C)C(NC(C2CCOC2)=O)C(C)(C)C1NC(=O)CCc1cc(Cl)cs1 36391,c1(CNC(C(CCC)CC)=O)ccc2c(c1)CN(C(C1CCN1S(C)(=O)=O)=O)C2 36392,C#Cc1cnn(C)c1C(N1CCC(N(C(=O)Cc2cnns2)CC)CC1)=O 36393,C1(C2CCN(C(Cc3c(C(C)C)con3)=O)C2)CCCCN1C(c1cccs1)=O 36394,N1(C(C=CCC)=O)CCOC2CN(C(=O)CNS(=O)(=O)c3cccc(F)c3)CC12 36395,c1(NC(C(CC)(C)OC)c2nnnn2CCCF)ccc(C)c(S(C)(=O)=O)c1 36396,O=C1CCC(C(=O)NC2CC(NC(=O)CCN3CCCCCC3)C(O)C2)=NN1 36397,C(=O)(C(C)(C)CCCNC(c1cc2cccn2cn1)=O)N1CCC(C)(N(C)C)C1 36398,C#Cc1ccc(C(N2CC(C)CC2C(=O)Nc2cnn(C)c2)=O)cc1C 36399,Cc1nc[nH]c1CC(O)C(=O)NCC1CCN(C(C2C3CC4C(C3)C24)=O)C1 36400,C(C)(N=c1[nH]c(=NCC(CO)C2CC2)c2c(F)cccc2[nH]1)c1cc(C)on1 36401,C1(C(=O)NC(CC)CNC(c2snnc2C)=O)CCN(S(=O)(=O)NC)CC1 36402,C(=O)(C1=CC2C=CC1C2)NC1CCN(C(C(C)OC(C)(C)C)=O)C1C(C)(C)C 36403,C1(CNC(c2c(OC)n(C)nc2)=O)C(C2CC2)CCN1C(c1nnn(C)c1C)=O 36404,C1(C(N2CCC(CN(C(=O)COCC3CC3)C)C2)=O)CCc2n[nH]cc2C1 36405,n1(CC)ccnc1C=CC(=O)NC1CC(CNC(C2(SC)CC2)=O)C1 36406,C(CCCCNC(=O)Cc1ccnn1C)NC(C(C1CCCC1)OCC)=O 36407,Cn1cc(C(=O)NC2CCCN(C(=O)CCC3CC3(Cl)Cl)C2)c(O)n1 36408,NS(=O)(=O)c1ccc(C(=O)NC2(CNC(=O)C(F)(F)C3CC3)CC3CCC2C3)o1 36409,N1(C(C(CC)C)=O)CC(CNC(c2sccc2C)=O)OC(C)(C)C1 36410,Cc1cc(N2CCCC(C)(NC(=O)CCC(F)(F)F)C2)ccc1[N+](=O)[O-] 36411,C(=O)(C(O)CCC(F)(F)F)NC1CCCC(NC(c2cn(CC)nc2)=O)CC1 36412,N1(C(C(C)OCC(C)C)=O)CCOC(C(N2CCCC(C)(C)C2)=O)CC1 36413,c1(NC(C)=O)cnc(C)c(C(N2CCCC2CNC(C2OCC2(C)C)=O)=O)c1 36414,C(N=c1[nH]c(=NC2CCC(CCNCCO)C2)c2ncccc2[nH]1)C1(C)CCOC1 36415,c1(NC(C2(C(=O)O)CC2)=O)cc(F)c(NS(=O)(=O)C(F)(F)F)cc1F 36416,Cc1sccc1C(=O)NC(C1CCCN1C(=O)CSS(C)(=O)=O)C 36417,CC1CN(C(c2ccc3sccc3c2)=O)CC(C)CN1C(c1ncccc1Cl)=O 36418,N1(C(C(C)OCC)=O)CC(NC(=O)CCc2cnc(O)[nH]2)C2(CCOCC2)C1 36419,c1(OCC(=O)NC2CC(C)(NC(C(C(C)C)SCC)=O)C2)cc(C)ccc1F 36420,CCC(C)C(C)CCNCC(=O)NCC(=O)Nc1cccc(C(F)(F)F)c1 36421,c12cc(N(C)C)ccc1OC2=O.C1(N(CC)CC)CCS(=O)(=O)C1 36422,c1(SC)nc(N2CCCCC2CNC(c2cnc(C)s2)=O)cc(Cl)n1 36423,CCC(C)CC(C)C(=O)N(CC(=O)NC1C2CCN(CC2)C1C)C1CCC1 36424,c1(C(C)C(=O)N2CC(C(C)N)C2)c[nH]c2ccccc12 36425,C1(O)(CNC(c2cccc(F)c2)=O)CCCN(C(C23CCCN2CCC3)=O)CC1 36426,c1(C(c2n(CC(=C)C)nnn2)NCCc2cccc(F)c2)cc(F)c(F)cc1F 36427,S(=O)(=O)(C1CCN(C(C2CCS(=O)(=O)C(C)C2)=O)CC1)NC 36428,c1(OC)ccc(CN2CC3CC3(C(=O)Nc3ccc(C4CC4)nc3)C2)c(C)c1 36429,C1(C(C)NC(Cn2cc(C(=O)OC)nn2)=O)CCCN(C(C2(CO)COC2)=O)C1 36430,N1(C(c2coc(CO)c2)=O)CCCN(C(=O)C2=C(Cl)CCC2)C(CO)C1 36431,c1(CC)cc(C(=O)NCCCC(=O)NC(CO)(CO)CO)c(C)o1 36432,Cc1cc(C)c(C(=O)NCC(C)(C)NC(=O)COc2ccc(Cl)cc2)c(N)c1 36433,C1(O)(CNC(CNS(C)(=O)=O)=O)CCCN(C(=O)CC2CC3CCC2C3)C1 36434,N1(C(C(CC)OCC)=O)CCC(O)(CCNC(=O)CCc2nccs2)C1 36435,c1(C(N2CCN(C(CCC=C)=O)C(CC)C2)=O)cc2ccc(OC)cc2nc1C 36436,C1(NC(c2nc(C(C)=O)sc2)=O)CCC(C)(CNC(c2ccc(CO)s2)=O)C1 36437,C1(C(N(C2CN(C(c3cc([N+](=O)[O-])cn3C)=O)C2)C)=O)CCCCC(C)(C)C1 36438,c1(NC(c2cc(-c3c(OCOC)cc(F)cc3)[nH]n2)=O)c(C)cc(C#N)cc1Cl 36439,c1(OC)ccc(Cl)c(OC)c1C(=O)NCC1(C)CN(C(c2cc(C)nn2C)=O)C1 36440,N1(C(C(C)O)=O)CCCC1C=CC(N1CCCC(CF)C1)=O 36441,c1(CC)cncc(C(=O)NCC2CCC(NC(=O)CCc3cnn(C)c3C)C2)c1 36442,Cc1cncc(C(N2CCOC(CN(C)C(c3cc(Br)oc3C)=O)C2)=O)n1 36443,C1(C(N2C3CN(C(CC4(C)CC4)=O)CC2CCC3)=O)CCCC12NC(=O)NC2=O 36444,N1(C(C2CCOC2)=O)CCCN(C(=O)Cc2cscn2)C(c2ccccc2)C1 36445,C1(C(=O)NCCCCNC(CSCCC)=O)(N(C)C)CCCCC1 36446,C(CC(O)CC(=O)NC1CC2(C1)CC(NC(=O)CCc1nnc(C)n1C)C2)SC 36447,C1(NC(C(C)N2CCCC2)=O)CC2CCC1(C(N1CCCC1C)=O)C2 36448,c1(C(N2CC(C)(CNC(C(C(=O)NC)(C)C)=O)OCC2)=O)csc2ccccc12 36449,C1(NC(C2N(C(c3c(C)nsc3)=O)CC2C)=O)(CO)CC2CCCC12 36450,c1(C(N(C2CCN(C(c3cccc(F)c3I)=O)C2)C)=O)cc(F)c(Cl)cc1Cl 36451,C1(CC)(CO)CCN(C(=O)NCCNC(c2ncccc2N(C)C)=O)C1 36452,Cc1cc(C)c(C(N2CCOC(CCNC(=O)C(C)(F)F)C2)=O)c(O)n1 36453,C(CCC(C)CC(=O)N1CC(NC(c2cncn(C)c2=O)=O)C(F)C1)=C(C)C 36454,CC1(C)CN(C(C2(c3ccno3)CC2)=O)CCN(C(C2(C)CCC(=O)NC2)=O)C1 36455,c1(CNC2CC(NC(c3cn(CCC)nc3)=O)C2)cc(OCC)ncn1 36456,C#CCCCCC(=O)NC(C1CCOC1)CNC(C1(C(F)(F)F)CC(=C)C1)=O 36457,N1(C(C=CSC)=O)CC2CCC(CNC(C3C4CCCCCCC34)=O)(C2)C1 36458,C1(OC)CC(NC(=O)C(C)Cn2ccnc2)CN(C(C2(n3nccn3)CC2)=O)C1 36459,c1(C(=O)NC2C(NC(C3(CCN(C)C)CC3)=O)CC2)cccnc1C(F)(F)F 36460,c1(NCC2C(C)CN(C(c3ccc(=O)n(C)n3)=O)CC2)c(F)cccc1[N+](=O)[O-] 36461,c1(CC)ccc(C(=O)NC(C2CCCCC2)CNC(C2COC(=O)O2)=O)o1 36462,N(C(=NCc1cc(C)nn1C)N1CCc2ccc(Cl)cc2C1)C(C=C)C 36463,Cc1cccc(C2CC2)c1CNC(=O)C(N1CCCC(c2ccno2)C1)C 36464,N1(C(CN(C(C(CC=C)CC)=O)C)=O)CC(C)CC(C)(C)C1 36465,Cc1c(C(N2CCCC2CN(C)C(C2(O)CC2)=O)=O)sc2cc(F)ccc12 36466,C12(NC(c3nocc3Cl)=O)CCCC1N(C(c1ccc(OC(F)F)cc1)=O)CC2 36467,C1(CNC(C(C)(C)OCC)=O)CCN(C(c2coc3c2COC3)=O)CC1O 36468,C1(C(N2CC(CCNC(CC3(OC)CCC3)=O)C2)=O)CCN(c2ccncc2)C1 36469,c1(C(=O)NC(C2CCCN2C(=O)C=C(Cl)Cl)(C)C)cc(P(C)(C)=O)cs1 36470,Cc1cc(F)c(C(=O)NCC(O)CN(C(=O)Cc2c[nH]ccc2=O)C)cc1F 36471,Cc1cccc(-c2csc(C(=O)NC(C)C(N)=O)c2)n1 36472,Cc1[nH]c(C)c(C(N2CCOC(CNC(=O)CC(C)C(F)F)C2)=O)c1C 36473,c1(C(N2CCC(N(C(C3(OC)CCCC3)=O)C)CC2)=O)cc(S(N)(=O)=O)c(C)o1 36474,C1(CCNC(c2c(C)cc(C)s2)=O)CCCN(C(=O)C(N2CCC(C)C2)=O)CC1 36475,C1(c2n(CCCCCOC)ccn2)CCCN(C(c2cccc[n+]2[O-])=O)C1 36476,C1(CN(C)Cc2ccc(NC(N)=O)cc2)CN(C(=O)COCCCF)CC12CC2 36477,C#CC1(O)CC(C(=O)NC2CCOC(c3ccncc3)C2)C1 36478,N1(C(c2n(CC)nc(C)c2)=O)CCN(C)CC1CNC(=O)CC(C)c1ccco1 36479,N1(C(COC)=O)CCC(CNC(=O)C(c2cncnc2)C)C(F)(F)C1 36480,c1(CC(=O)NCCN(C(Cc2nc(CC)sc2)=O)CC(C)O)cncc(O)c1 36481,C(C(C(=O)NCC1CC(C)(NC(=O)CSc2nnnn2C)C1)NC(C)=O)OC 36482,C1(C(=O)NCc2cc(C)ncc2)COC2(C1)CN(C(C1CCC(=O)C1)=O)C2 36483,NC(=O)CCC(C(=O)N=c1ccn(CC(F)(F)F)[nH]1)n1cc2ccccc2n1 36484,C(=O)(N=c1[nH][nH]c2c1CN(C(c1ccc3[nH]c(C)cc3c1)=O)C2)SC(C)=O 36485,C1(C)(C(N(CCNC(C2CC3C(C2)C3(F)F)=O)CC)=O)C2CC3CC(C2)CC1C3 36486,C1(C(C)NC(C2CCN(CC)C2)=O)CCN(C(=O)CNC(C2CCCC2)=O)CC1 36487,C(=O)(C(C)(C)c1cccs1)NC(C1CC(NC(=O)CCc2ncc[nH]2)C1)C 36488,C1(NC(CC(=O)N(C)C)=O)CN(C(=O)CCCc2ncc(Br)cn2)CC1O 36489,c1(C(=O)NC23C(CN(C(Cc4ccc(C)s4)=O)C2)C3)ccc2ncc(=O)[nH]c2c1 36490,CCCC(C(=O)N1CCC1C(=O)N(CC(C)(O)C1CC1)C)OC 36491,CC1CCN(CC(=O)NCC2CCC(N(C)C(C3(C4CCC4)CC3)=O)CC2)CC1 36492,C(=O)(C(C(C)C)c1cnc(C)s1)NCCC1CC(NC(CC(C)C)=O)C1 36493,CC1CN(C(C2CCC(N(C)C)CC2)=O)CC1NC(c1nncs1)=O 36494,N1(C(C(C)c2ccsn2)=O)CCC2(CCC2)C(NC(=O)CCC2CC2)C1 36495,C1(O)(C(C(=O)NC2CC(NC(c3c(C)snn3)=O)C2)(F)F)CCOCC1 36496,N1(C(C2(CC)CN(C(C(CCC)NC(C)=O)=O)C2)=O)CCC2(CCCN2C)C1 36497,c1(C(N2CCC(OCCNC(CS(CC)=O)=O)C2)=O)cc(C(=O)OC)cc(O)c1 36498,c1(C(N2CCCC(NC(CC3C(CC)C3(F)F)=O)C2)=O)cc(S(C)(=O)=O)c(C)o1 36499,C1(C)(CNC(NCC(CC)(C)C)=NCC2CCOC2)CCCC1(F)F 36500,N1(CC(=O)NC2CCC(CNC(C3(N(C)C)CCC3)=O)C2)C(=O)CC(C)(C)C1=O 36501,C1(CC(=O)NC2(CC)CCCOC2)CC2(C1)CN(C(c1ncc(F)cc1N)=O)C2 36502,c1(C(N2CC(C)C(C(=O)NC3(C4CCCO4)CC3)C2)=O)cc2ncccc2[nH]1 36503,C(CC(O)C(F)(F)F)N(c1cc(F)cc(F)c1)C(=O)Nc1cccc(SC)c1 36504,Cc1cc(C(N2CCC(OCCNC(C3CC(F)C3)=O)C2)=O)n(C)n1 36505,c1(C(=O)NCCC2(NC(c3c(C)coc3)=O)CCC2)nn(C)c2ccc(F)cc12 36506,C1(CNC(C2(SCC)CC2)=O)CCN(C(C2C3CCCCC23)=O)CC1 36507,CC1=C(C)CC(C)(C(N2CC(O)(CNC(c3cc(F)c(O)c(F)c3)=O)C2)=O)CC1 36508,c1(C(=O)NCc2c(C(N(C(CCC)C)C)=O)scc2)cc(OC)n(C)n1 36509,C1(CC)COCCN(C(c2cc(CCNC(=O)C(C)SC(C)C)on2)=O)C1 36510,C1(C)(CC(=O)OC)CCN(C(c2ccc(C)c(I)c2)C(=O)NCC(C)C)CC1 36511,c1(C(=O)NCC(CC)(CC)NC(c2ccn(C)n2)=O)c(O)cc(F)cc1F 36512,C(=O)(C(O)Cc1ccccc1)NCCCN(C(=O)CC1CCCO1)C(C)C 36513,c1(-c2c(CC)nc(Cl)nc2C)ccc(S(=O)(=O)CC)cc1 36514,C1(NC(CC(C)(C)OC)=O)CN(C(C23CCC(N=[N+]=[N-])C2C3)=O)CC(C)(C)C1 36515,C1(CNC(CCC)=O)CN(C(=O)C2=CC(C)C2)CC(C)(C)C1 36516,c1(NCCc2c(C)cccc2)[nH]c(=NC2CC2c2ccccc2)nc2scnc12 36517,Cc1ccc(=O)n(CC(=O)N(CC(C)NC(=O)Cc2cc(Br)cs2)C)n1 36518,c1(CC)ccc([N+](=O)[O-])cc1C(=O)NC1(C)CN(C(=O)C(CC)C(C)O)C1 36519,C=CC(CC)CC(=O)NCCC1CSCCN1C(c1n[nH]c(C2CC2)c1Cl)=O 36520,c1(OC)nc(C(=O)NCC(C)CNC(=O)CCC(=O)c2ccccc2)cc(O)n1 36521,NS(=O)(=O)c1cc(CN2CCC3(C2)CC3(F)F)c(Cl)cc1F.C12(CC1)C(=O)NC2 36522,C(C(C)NC(c1cc(C)n(C)n1)=O)(C(C)C)NC(c1c(-c2cc(C)no2)ocn1)=O 36523,C(=O)(C(CC(F)F)C1CCC1)NC1CC(CNC(=O)CCn2cncn2)CC1O 36524,C1(F)(CNC(C(C)S(N)(=O)=O)=O)CCCN(C(C2NC(=O)OC2(C)C)=O)CC1 36525,c1(C(N2CCC(C)(CNC(CC3(C=C)CC3)=O)CC2)=O)ccc2oc(O)nc2c1 36526,N1(C(c2c(OC)cccc2)=O)CCC(C)C(CNC(=O)CCc2cccs2)C1 36527,CN1CCC(C(=O)N(CCNC(=O)C2=CSCCO2)CC2CC2)S1(=O)=O 36528,Cc1cc(C)n(C(C)CNC(N2CCCC2Cc2ccncc2)=O)n1 36529,c1(OC)cc(F)c(F)cc1NNC(=O)NC(c1ccc(C#N)cc1)C 36530,c1(C(=O)NC(C2N(C(C3CC(OC)C3)=O)CCC2)C)ncnc2c1CCC2 36531,CN1C(=O)OC2CN(C(C3CCN(C(C4CCO4)=O)CC3(C)C)=O)CC12 36532,C1(NC(C2(OC)CCOC2)=O)CCCC(CC(=O)N(C2CCOC(C)C2)C)C1 36533,c1(CC(=O)NC2CN(C(C(P(C)(C)=O)O)=O)CC23CC3)cc(Cl)cc2c1OCC2 36534,C(=O)(C(O)C(C)(C)C)N1C(C(=O)NCC2CC3C=CC2O3)CC(C)C1 36535,Cn1nnnc1SC(CNC(CCNC(=O)COC1CCOC1)=O)C1CC1 36536,c1(CC)c(C(N2CCCCC2CN(C(=O)CCc2nncn2C)C)=O)ccn1C 36537,C1(C)(CC(=O)N(CCCNC(C2(CC(F)(F)F)CC2)=O)CC)CCS(=O)(=O)N1 36538,C(CCCCC(=O)N(CC(C)O)CCNC(C1CC(O)CN1C)=O)OCC 36539,C(=O)(C(C)(C)CCSC)NC1C(CNC(C(CC)Sc2nc(=N)[nH][nH]2)=O)CC1 36540,C1(NC(CC2(N(C)C)CC2)=O)CCN(C(=O)CCC2(C)CC2)CC1F 36541,N(C1CCCc2ccoc21)C(C1N(C(=O)Cn2ncccc2=O)CCN(C)C1)=O 36542,C1(CNC(C2CC(CCC)C2)=O)CN(C(c2ncnn2C(C)C)=O)CCC1(C)C 36543,C(C(C)C(C)C)N(CCC(=O)NC1CC(NC(C(C)N(C(C)=O)C)=O)C1)C 36544,N1(C(C)C)CCCN(C(C2CCC(C(C)C)N2C(=O)C2=CCOCC2)=O)CC1 36545,CC1=CCSC1C(=O)NCc1ccsc1C(=O)NCCC(C)N(C)C 36546,C(=O)(CC1=NNC(=O)C1)NCC1N(C(c2c(C)cc[nH]c2=N)=O)CCCC1 36547,C1(O)(C(C)C)CCCN(C(=O)CCS(C)=O)C1.c12cn(nn1)CCC21CC1 36548,c1(N2C(CNC(c3cn(C(C)C)nn3)=O)CCCC2)ccc([N+](=O)[O-])cc1C#N 36549,c1(C(=O)NCC(C2CC2)NC(c2ccc(CC)c(N)c2)=O)cccc2scnc12 36550,c1(CNC(=O)NCC2CC(C(F)(F)F)CO2)cc2ncccc2s1 36551,C1(CNC(C(C)Cc2ccco2)=O)CN(C)CCN1C(c1cccc(=S)n1O)=O 36552,c1(C(N2CC(NC(C3C(=C)CC3)=O)C3(C2)CC3)=O)cc(Br)c(OC)cc1N 36553,c1(CC)cccc2[nH]c(C(N3CC(CNC(C4COCCO4)=O)C(O)C3)=O)cc12 36554,CC1=CCC(C(N2CC(O)(C(C)(C)CNC(=O)CC(C)(C)C)C2)=O)CC1 36555,c1(C(N2C3(C(N(C4CCCCC4)CCC)=O)CC(C2)C3)=O)cc2ccccn2n1 36556,C1(NC(COCC)=O)CC(OC2CC2)CN(C(c2cccc(C(C)(C)C)n2)=O)C1 36557,c1(C(CC)C)nccc(N2CC(C)(C)C2C2CCN(C(c3cncs3)=O)CC2)n1 36558,C1(CNC(CCN2CCN(C)CC2)=O)CCN(C(C2C=CCC2)=O)C12CCC2 36559,c1(C(=O)Nc2cccc(CNC(CCN(C)CCO)=O)c2)coc2ccccc12 36560,N1(C(C2CCC(CC)C2)=O)CCC(C=CC(=O)NC(CCO)C(F)F)CC1 36561,N1(C(C2CC(C#C)(O)C2)=O)CC(NC(c2cnn(CC(F)(F)F)c2)=O)CC1(C)C 36562,C(=O)(C(CC)CC=CC)N1CC(CN(C(CC2CC(=C)C2)=O)C)OCC1 36563,N1(C(CC2(COC)CC2)=O)CC2C(NC(=O)C(c3ncccc3F)(F)F)C2C1 36564,C1(C(N(c2ccsc2)CC)=O)CN(C(C2CCC3(CCC3)O2)=O)C2(CCC2)C1 36565,C1(C(=O)NCC2(CNC(c3cnc(C)nc3)=O)CCCC2)CCC(C)(C)CC1 36566,C(=O)(CCCCCCCCC)NCC(CNC(C1C(=C)CC1)=O)(C)C 36567,c1(C(N2CCC3(CCN(C(C45CC(F)(C4)C5)=O)C3)C2)=O)cnc2ncnn2c1O 36568,CCC(C)CC(C(=O)NC(C)C(C)SC)NC(c1cnc2n1CCC2)=O 36569,CCC(CC)C(C)C(=O)NC(C)(C(=O)NCC1=CCCCC1)C1CCC1 36570,C1(O)(CNC(c2cnc(N3CCOCC3)s2)=O)CN(Cc2cn(C3CC3)nn2)C1 36571,C1(CNC(c2c(C)scc2)=O)C(C2CC2)CCN1C(c1coc(C(C)C)n1)=O 36572,C1(NC(c2c(C#C)c[nH]n2)=O)CC2CC1CN(C(=O)CC1CCS(=O)(=O)CC1)C2 36573,C(=O)(C(C)C(C)(C)O)NCC(C)NC(c1ccc(OCC(F)F)cc1)=O 36574,CC1CCC(NC(=O)C(CC=CCl)c2ccccc2)CN1C(C1CCC1)=O 36575,C(CC#N)(C(=O)C(C)OC(=O)NC(C(=O)OC)C)NC(=O)OC(C)(C)C 36576,C1(C(=O)NCCN(C2CC2)CC)CC2(CC2)CN1C(C1CCCC(=O)C1)=O 36577,N1(C(C=Cc2cnc(C)s2)=O)CCCC2C1CCCN2C(=O)C#CC1(C)CC1 36578,CCC(C)(C)CC(=O)N(CC(C)N(C)C(C1CSCN1C(C)=O)=O)C 36579,C1(O)(C(=O)NC2(CNC(=O)Cc3cc(C)ns3)CC(OC)C2)CC2CCC1C2 36580,C#CCC(CC#C)NC(=O)C(Cn1ccnn1)NC(=O)CCC1CCC(=O)C1 36581,N1(C(c2c(C)cc(N)cc2)=O)CCC(F)(F)C(CNC(c2occ(C)c2C)=O)C1 36582,C1(COC)CC(CNC(=O)CCOCCCNC(=O)C(C)n2cncn2)C1 36583,C1(CC)(NC(=O)CC(c2ccc(SC)cc2)C)CCN(C(=O)C(C)(C)CO)CC1 36584,CC(CC(F)F)C(=O)N(C1CCC(NC(=O)C(C)N2CCC2)CC1)C 36585,N1(C(c2c(C(C)C)ccs2)=O)CC2CC1CN2C(c1n[nH]cc1Br)=O 36586,C1(CCOC)CCCCN1C(N1CCC(C)(O)C1)=O 36587,C1(N(C=O)Cc2nscc2Br)CCc2nncn2C1 36588,c1(C(N2CC(NC(C(CCC)(C)CC)=O)C(C)C2)=O)nnc2ccccc2n1 36589,CC1(C)OC(=O)CC1C(=O)NC1CCCN(C(=O)CSCC(F)F)C1 36590,N1(C(C(CCNC(C2(CC#C)CC2)=O)O)=O)CC2(C1)CC(C)(F)C2 36591,N1(C(CC(=C)C)=O)CCC2(CC1)CN(C(C1(C)C=CCCC1)=O)CC(C)O2 36592,C1(NC(=O)CCF)CCCCC1NC(c1coc(Br)c1)=O 36593,CCCC(C(=O)N1CC(CNC(c2cocn2)=O)(COC)C1)C(C)C 36594,C1(NC(=O)CC2CCCCC2)CC(F)CN(C(=O)C(F)F)C1 36595,C1(OC2CN(C(c3c(CC)nns3)=O)C2)CCN(C(c2ncoc2C)=O)CC1 36596,N(C(=NCCC(=O)NC)NCC1CCCCC1C1CC1)Cc1c(CC)cccc1 36597,C(CCN=c1cc(C)nc(CC)[nH]1)N(CC)CC.c1ccc(C(F)(F)F)cn1 36598,C1(NC(C2COCC2C(F)F)=O)CC2CCC1CN(C(C1CC1F)=O)C2 36599,N1(C(C(=O)NCC)=O)CCC2(CC1)COC(CNC(c1c(Cl)nn(C)c1C)=O)C2 36600,Cc1c(Cl)ccc(C(=O)N(C2CCCN(C(c3cccc(=O)n3C)=O)C2)C)c1O 36601,C1(NC(COC2C(CC)CCCC2)=O)CCN(C(c2cc(O)cs2)=O)C(C)C1 36602,Cc1nc(NCC2(O)CCCN(C(c3cnn4ncccc34)=O)C2)c(C)c(O)n1 36603,C(=O)(C(C)(c1ccccc1)OC)N(C1(CC(=O)NCC2(C(=O)OC)CC2)CC1)C 36604,Cc1nnccc1C(=O)NCc1cccnc1N1CCNC(=O)C1 36605,c1(C(=O)OCC)nnc(CNC(c2nnc(C)o2)C)s1 36606,n1(CC(=O)NCC(C2CC2)NC(c2ccccc2)=O)nc(Cl)ccc1=O 36607,CC1CN(C(c2scnc2C(F)(F)F)=O)CCN1C(C1CC2(CCOC2)C1)=O 36608,c1(CN2C(C3CCN(C(C(CC=C)C)=O)CC3)CCC2)ccc([N+](=O)[O-])cc1F 36609,c1(C(N2CCC(C)(c3cnn[nH]3)CC2)C(=O)NC(C)(C)C)cc(S(N)(=O)=O)cs1 36610,Cc1ccc2c(CC(=O)N(C)CCNC(C3CC4CCCCN4C3)=O)coc2c1 36611,c1(C(C)CNC(=O)Nc2ccnn2CC2CC2)ccc(Br)cc1F 36612,CC1CCC(NC(C2(NC(N)=O)CC2)=O)CN1C(c1n[nH]c2c1COC2)=O 36613,C1(CNC(CC=C)=O)CCC(CN(C)C(c2cc(C3CC(F)(F)C3)[nH]n2)=O)CC1 36614,C1(C(N(C2CCN(C(c3conc3C3(C)COC3)=O)C2)C)=O)COC(=O)N1 36615,c1(C(=O)NCC(CCCC)NC(=O)C(C)SCC)ccnc(F)c1OC 36616,c1(CSC)cc(C(=O)NCC23CC2CN(C(=O)CC(C)C2CC2)C3)ccc1F 36617,N#Cc1c(C(=O)NC2CC(NC(c3n[nH]c4c3COCC4)=O)C2)cccc1F 36618,N1(C(C=C(C)C)=O)CCCC(C)C1C(=O)C(C)N(C)C 36619,C1(C(C)NC(c2nc(CC)sc2)=O)CCN(C(c2cc(C3CCC3)[nH]n2)=O)CC1 36620,c1(OC)ccccc1C(=O)NCC1CC(NC(=O)C(c2ccccn2)O)C1 36621,C12(C(=O)NCC3(C)N(C(c4c(C)ccnc4)=O)CCC3)CCCN(CC1)C2 36622,Cc1cc(C(=O)NCc2cc[nH]c2C(=O)NCCc2cnn(C)c2)cc(C#N)c1 36623,N1(C(C2(NC(c3ccc(C)cn3)=O)CCOCC2)=O)CCCC(O)(CO)C1 36624,N1(C(CN(C(=O)Cn2nc(C)nc2C)CC#C)=O)CCCC(C)C1CO 36625,C1(C(N2CCN(C(=O)C3=COCCO3)C(C(F)F)C2)=O)CC2CCC1CC2 36626,C(CN=C(NCc1cc(O)cc(O)c1)NCc1cc(C)ccn1)N(CC)CC 36627,c1(CC(=O)N(C2CC(C(=O)NCC(C)Cc3cn[nH]c3)C2)C)cccn1C 36628,c1(C(=O)NCCCOCCN(C(=O)CC2COC(=O)C2)C)c(Cl)cnn1C 36629,c1(NC2(CNC(CC(=O)OC)=O)COC2)cc(Br)c(F)cc1OC 36630,C1(OC)CC(NC(C2CC=CC2)=O)CN(C(C2CCC(=O)N2C2CC2)=O)C1 36631,C1(C(=O)NC2CCC(NC(c3ccncc3O)=O)C2)CCCC1(F)F 36632,Cc1nn(C(C)C)cc1C(=O)NCC1(CNc2ccccn2)CCC1.C(=O)(C=CCF)N 36633,C1(C(=O)NCC(C)NC(CC2C(OCC)COCC2)=O)CC(=O)NC1(C)C 36634,N1(C(c2cc(OCC)no2)=O)CC2CCN(C(C3CC(SC)C3)=O)CC12 36635,c1(C(=O)NCCOc2c(OC)cc(C)cc2)cc([N+](=O)[O-])cc(O)c1O 36636,N1(C(Cc2nc(C)sc2)=O)CCCN(C(=O)Cc2cccc3nonc23)C(C)C1 36637,C(CCC(N)=O)(C(=O)NCC1CCN1C(=O)C=CCN1CCCCC1)NC(C)=O 36638,C(C(C(=O)N1CCCCC1CCNC(c1ncccc1C)=O)C(F)(F)F)OC 36639,C(=O)(CCC(=O)NN(C)C)NC1CC(C)CN(C(c2cc(O)ncn2)=O)C1 36640,c1(CC)nc(C)c(C(N2CC(C(=O)NC(C)(CO)C3CC3)(CC)C2)=O)o1 36641,C1(NC(c2cc(C)ns2)=O)CCCN(C(=O)C(CCCO)c2ccccc2)C1C 36642,CC1(C)CCCC(CC(=O)NCC2COCCN(C(=O)Cc3ccon3)C2)C1 36643,c1(C(=O)NCC2C(NC(COCC)=O)COC2)c(F)cccc1[N+](=O)[O-] 36644,N1(C(c2c(OC)n(C)nc2)=O)CCN(C(c2cc(O)cs2)=O)CC1C 36645,c1(C(N2CCC(c3c(C(=O)OCC)c[nH]n3)C2)=O)cc(C)n(C)c(=O)c1 36646,C(=O)(C(C)(O)CC(C)C)NC(CC(=O)NCc1snc(CC)n1)C(C)C 36647,C(=O)(C#CC1CCOCC1)NC1CCC(CNC(C(c2ccccc2)C)=O)CC1 36648,C(CC(C)C)(C(=O)NCC(C)CN(C(=O)CC1CCC(C)(C)CO1)C)NC(C)=O 36649,C1(C(=O)NC(C2CCCCC2)C#C)COCCN1C(c1ccnc(C)n1)=O 36650,CCCS(=O)(=O)c1ccccc1C(=O)NCCCCCNC(C1CC1F)=O 36651,Cc1nc(C(=O)NC2CC2CNC(=O)C=CC2CCCCCC2)c(C)n1C 36652,n1(COC)nccc1C(=O)NC1CCC1CNC(C1CCC(C(=O)OC)C1)=O 36653,C1(CNC(c2n(CCSC)nnn2)c2ccncc2)CC2CCC1CC2 36654,c1(OCC)ccc(C)cc1C(NC(=NCC1(C#N)CCOCC1)NC(C)C)C 36655,Cc1ccc(S(=O)(=O)N2CCC2C(=O)Nc2cc(C)cnc2Br)c(F)c1 36656,N1(Cc2ncc(CC)o2)CC2(C)CN(C(=O)CCC(C)OC)CC2(C)C1 36657,c1(C(=O)NCC2N(C(c3cnc(=N)[nH]c3)=O)CCCC2)ccc2c(c1)CCCS2 36658,C1(CC(=O)NCCC(C)(C)NC(CC(C)SC)=O)CCOC(C)(C)C1 36659,C1(C(=O)NCC=CCNC(c2cc(C3CC3)[nH]n2)=O)CCC(n2ccnn2)C1 36660,C1(CNC(C(C)(c2ccccc2)OC)=O)CC2CCC1N2C(c1cocc1C)=O 36661,C12(CNC(C3OCCN(C)C3)=O)CCC(CNC(C3CC3(F)F)=O)(CC1)CO2 36662,c1(CN(C(C(C)O)(C)C2CCOCC2)C=O)ccc(Br)cc1OC1CC1 36663,N1(C(=O)C(c2cccnc2)O)CCC(C(F)(F)F)C(NC(C2(F)CCC2)=O)C1 36664,C(=O)(NNC(=O)C1OCCC1Cn1cc(C)cn1)OCC 36665,Cn1ncc(C(=O)NC2CC3CC(C2)N(C(=O)C(C)(C)C)C3)c1S(N)(=O)=O 36666,CC(C)C(O)C(C)C(=O)NCCCC(C)(C)NC(c1cc(C2CC2)on1)=O 36667,c1(CC)ccc(C)c(C(=O)NC(C)C(C)(C)NC(=O)CN2CCSCC2)c1 36668,CC1CCc2nc(C(=O)NCC3CCCC3NC(=O)CC(C)(C)O)ccc2C1 36669,C1(NC(c2nc(-c3c(C)cccc3)sc2)=O)(CNC(=O)C(N)=O)CC2CCC1C2 36670,Cc1ccc(F)cc1CC(=O)NC(C)C(C)(C)NC(C1CC2(CCC2)CO1)=O 36671,n1(CC)nccc1C1OCCC1NC(=O)NCCc1ccccn1 36672,c1(C(N2CCC(NC(c3ccc(S(C)(=O)=O)s3)=O)C2)=O)cccc2nc(Cl)cn12 36673,C(=O)(N=c1[nH]nc(C2CC2)s1)N(c1ccccc1CCOC(C)(C)C)C 36674,C1(COC)(NC(=O)C=CC(F)(F)F)CCN(C(=O)Cn2cnc(=N)[nH]2)CC1 36675,Cc1nc(F)ccc1CNC(C1CCN(C(=O)C2CC3CC(=O)C2O3)O1)=O 36676,CCC(N=c1ccnc(NC2CCN(S(C)(=O)=O)CC2)[nH]1)C(C)C 36677,N1(C(CC=CC)=O)CC(NC(=O)C=Cc2ccoc2)CC(F)(F)C1 36678,CC(C(=O)N1CCCC1CCNC(c1c[nH]cc1C(C)(C)C)=O)C(F)(F)C(F)F 36679,CCCCCCCCC(C)C(=O)NC(C1CCN(C(C2(C)CCC(=O)C2)=O)C1)C 36680,N1(C(C(C)NC(CC)=O)=O)CC(=O)NCC1C(=O)NCC1(O)CCN(C)C1 36681,N1(C(CN(C)C)=O)CCCC(C)(C)C1CNC(C1(Cc2ccc(F)cc2)CC1)=O 36682,c1(CC(=O)NC2C(NC(c3cc(C(C)C)nn3C)=O)C2)cn2ccccc2n1 36683,C1(CNC(CCCOCC)=O)CCCC(NC(c2nnc(CC)s2)=O)C1 36684,c1(N2CC(CN(C(c3cc(C)no3)=O)C)OCC2)ncnc2scc(C)c12 36685,c1(N2CCCC(CCNC(CC3C(C)CCC3)=O)CC2)ncc([N+](=O)[O-])c(=N)[nH]1 36686,C1(C(N(CCCCNC(C(=O)NCC)=O)C)=O)COCC(C)(C)O1 36687,N1(C(c2ccn(C)c2)=O)CCC(C(C)(C)C(=O)NCc2ccncc2F)CC1 36688,CC(C)(C)CC(=O)NCC1CC(C(N2CCC(c3nc[nH]n3)C2)=O)CO1 36689,C1(C(=O)NCC(C)CN(C)C(c2cnn(C3CC3(F)F)c2)=O)OCC1(C)C 36690,C1(NC(c2ccc(OC)c(I)n2)=O)CCc2ncc(Br)n2C1 36691,c1(C(=O)NCCC2CN(C(c3c(CC)nccn3)=O)C2)cc2c(=O)[nH]ccn2c1 36692,n1(C(C)C)cnc(C(=O)NC(CO)C(C)NC(C2(N3CCOCC3)CC2)=O)c1 36693,C(=O)(C(C(C)C)C(C)C)NCCC1CCCN(C(CCC(=O)OC)=O)CC1 36694,Cc1cc(C(N2CCC(F)(CNC(C3CCCN3C3CC3)=O)C2)=O)nnc1C 36695,CN=c1[nH]cc(C(=O)NC2(CCCCNC(c3csnn3)=O)CC2)o1 36696,C(c1ccc(F)nc1)=CC(=O)NCC1CCCN(C(c2cncc(Cl)c2Cl)=O)C1 36697,C1(N(CCCC)C(=O)C=Cc2cscn2)CCN(C(c2cc(C)cs2)=O)CC1 36698,c1(OC2CN(CC(c3ccc(CC)cc3)O)C2)ccc(Cl)cc1[N+](=O)[O-] 36699,C1(C(N(CC(C)(C)N(C)C)C)=O)CCN(C(C2CC(C)(C)C2)=O)CC1 36700,N1(CC(COCC(C)C)O)C2CCC1CN(Cc1ccc(C3CC3)o1)C2 36701,C1(C2CCOCC2)(C(=O)NCC(C(C)(C)C)NC(C(C)CC(F)F)=O)CC1 36702,C1(CNC(C(CC=CC)NC(c2cc(CSC)on2)=O)=O)OC(=O)CC1(C)C 36703,Cc1cc(C)c(C(=O)NCCCCN(C)C(c2c(C(F)F)cnn2C)=O)c(S)n1 36704,C(=O)(C1=CC2(CN(C(C3C(C)(C)C3(F)F)=O)C2)OC1)N(CCCO)CCC 36705,C1(NC(C(CCC)=CCC)=O)CCCC(C(=O)NCCN2CCCOCC2)CC1 36706,C(C(F)(F)C(F)F)O.C1(COC)(NCC2CC2)CCC1 36707,C1(CC(=O)NCCC(CC)CO)CCN(C(C2OC3CCC2C3)=O)C1(C)C 36708,c1(CNC(=O)NCC(c2cccc(I)c2)C)ccc2cnccc2c1 36709,c1(C(C)=O)cccc(OC(C)C(=O)NCCCCC(C)NC(=O)CSC(F)F)c1 36710,c1(CC(=O)NC(C(N)CO)C(=O)O)cc(Cl)ccc1I 36711,CCCC(C(=O)NCC1CCCCN(C(=O)CCN2CCOCC2)C1)S(N)(=O)=O 36712,Cc1noc(C(F)F)c1C(=O)NCCN(C(=O)Cc1sccc1Cl)CC(C)O 36713,N1(C(CC2(NC(C)=O)CC2)=O)CCC(C(F)F)(CNC(C2CC(O)CN2C)=O)C1 36714,c1(CC(N2CC(O)(C(C)NC(C3CC(CCC)C3)=O)C2)=O)sc(C)nc1C 36715,c1(OCCOCCCNC(C(C)(C)NC(=O)OC)=O)ccc(Cl)c(C(=O)OC)c1 36716,c1(C(=O)OC)c(C)ccc(NC(C2COCCN2CC2CCCC2)=O)c1C 36717,c1(N(C)CCC2CCCCC2)nc2c(c(=NCC3CCC=CCCC3)[nH]1)COC2 36718,CCC(C)C(=O)NCC(=O)NCCN(C(C1CC(NC(=O)OC)C1)=O)CC 36719,N1(C(c2c(C)snc2)=O)C2CCC1C(CNC(=O)CCc1nc(C3CC3)no1)C2 36720,CC1(NC(c2c[nH]c(Br)c2)=O)CCN(C(=O)CC(F)(F)F)C1 36721,C1(C(=O)NCC23CC(NC(c4ccc(CC)s4)=O)(C2)C3)CC(C)(C)C1C(F)(F)F 36722,N1(C(CC(COC)C)=O)CCC2CCCC12C(N1CCCCC(N(C)C)C1)=O 36723,C=C(Br)CC(C)(C)C(=O)N1CC(CNC(=O)C(C)SCC)C(C)C1 36724,c1(N2CCC(C)OCC2)ccc(S(=O)(=O)NC2CCCC(C(F)(F)F)C2)c(Br)c1 36725,C(CC(CNC(=O)CCF)NC(=O)CNC(c1cccs1)=O)Oc1ccccc1 36726,N1(CC(=O)NCc2c(OC)cncc2)C(=O)NC(C)(c2ccc(F)cc2C)C1=O 36727,c1(-c2c(C(=O)NC(C)C(C)n3ccnc3)c[nH]n2)ccc2c(c1)CCCO2 36728,c1(C(N2C(CNC(c3c(C)nccc3)=O)CCCC2)=O)ccc(CO)c(Cl)c1 36729,c1(C(CNC(=O)CCc2ccon2)NC(C2C=CCC2)=O)ccc(Cl)cc1 36730,c1(C(C(=O)OCC)N(C(C)(C)C)CCNC(=O)N(C)C)ccc(Br)c(OC)c1F 36731,C1(N(C(=O)NC2CC3(C(C(=O)OC)C3)C2)C)CC(C)OC(C)C1 36732,C(=O)(C#CC1CCCCC1)N1CCCC(CCC(=O)NCC2(O)CCC(C)C2)C1 36733,C1(C(=O)NCCOCCN(C)C)CNC(=O)CN1C(=O)CCn1cccc1 36734,C1(C(=O)NC2CC(NC(C34CC(C3)C(C(F)(F)F)O4)=O)C2)CC2C=CC1C21CC1 36735,c1(C(=O)NC2CCC(C)(CNC(=O)C3=C(Cl)CC3)C2)cccn2cncc12 36736,Cc1ccc([N+](=O)[O-])cc1C(N1CCC2CN(C(C3(C#N)CC=CC3)=O)CC12)=O 36737,c1(C(=O)NCCC2(CNC(C(C)O)=O)CCCC2)nccc2cc[nH]c12 36738,CCCCC(F)F.C(=O)(C(C)CO)N(Cc1ccccc1)CC 36739,C12(C(N3CCCN(C(=O)COc4ccc(Cl)nc4)CC3)=O)CCCCC1C2(F)F 36740,C1(CC(N2C3CN(C(C4(C=C)CCC4)=O)C(C3)C2)=O)CCc2ccccc2C1=O 36741,C(c1ccc(C)cc1C)=CC(=O)NC1CCCC(CNC(CN(C)CC)=O)C1 36742,Cc1cc(F)cc(C(N2CC(N(C)C(C3CCOCC3)=O)C3(CC3)C2)=O)c1O 36743,C=CCC(Cc1ccccc1)C(=O)NCCCOc1c(F)cccc1F 36744,N1(C(C(C)SCC)=O)CCC(CNC(c2cnccn2)C2CCCC2)C12CCC2 36745,N1(C(C=Cc2cc(C)no2)=O)CC2CCC(N(C(=O)C3=CCCSC3)C)C2C1 36746,c1(C(N2C(C)(C(=O)NC)CC(O)C2)=O)nccc2[nH]ccc12 36747,C(CNC(=O)Cc1ccccc1)(C(C)(C)C)NC(CCN(C)CCO)=O 36748,C1(C(=O)NCCCN2CC=CC2)CCC(O)CN1C(c1cc(C(F)F)[nH]n1)=O 36749,N(C(=NCc1ccccc1[N+](=O)[O-])N1CCC(C)(F)C1)Cc1cc(C)on1 36750,c1(Nc2c(CNC(C3SCCCS3)=O)con2)ccnc(C2CCC2)n1 36751,C1(OC)(CNC(c2n[nH]c(C)c2O)=O)CCN(C(c2cn(C)nc2C(C)C)=O)C1 36752,CC1CC2(CCN(C3CCN(C)C3=O)CC2)CN1C(C1CC1(Cl)Cl)=O 36753,c1(C(OS(NCC(=O)OC(C)(C)C)(=O)=O)=O)cccnc1Oc1ccccc1 36754,N1(C(c2ccc(C)c(O)c2)=O)CCC2(CC1)CC(NC(C1CC=CCO1)=O)CO2 36755,c1(C(=O)NCCCN(C(=O)C(OC)OC)CCC)cc(C(N)=O)[nH]n1 36756,N1(C(CC2(OCC)CC2)=O)CCC(CN(C)C(c2cnc(C3CCC3)o2)=O)C1 36757,C1(NC(c2ccnc(F)c2Cl)=O)CC2CC1CN2C(c1ccc[n+]([O-])c1)=O 36758,C#CCCCCCC(=O)NC(C)(C)CCC(=O)N1CC2CC1C2CF 36759,C(=O)(CC(CNC(C1(OC(C)=O)CCC1)=O)C1CCC1)NCC(CC)C 36760,C(=O)(C(C)(C)CCCF)NCC(C(=O)NCc1c(C)cc(O)cc1)CC1CC1 36761,N1(C(CCOCC(C)(C)C)=O)CCCC(F)(C(=O)NCC23CCCC2CCC3)C1 36762,C1(CNC(C2CC3(C2)CC3F)=O)COCCN1C(=O)Cn1cnnc1O 36763,CC1CN(C(c2cncc(F)c2)C(=O)NC2(C)CC2)C12CCOCC2 36764,c1(C(=O)NC(CNC(C(c2c(C)nn(C)c2)O)=O)CO)cc(Cl)cc(Cl)c1 36765,CC(=O)C(C)(C)CC(=O)N(C1CCN(C(c2ccccc2[N+](=O)[O-])=O)C1)C 36766,C(CC(=O)N(C1CC(O)C1)C)(C(C)C)NC(c1ccc(OC)cn1)=O 36767,N1(CC)CCC(NC(=O)C(F)CC2CN(C(C3(CO)CCCO3)=O)C2)C1 36768,C1(C(C)C)CCC(C(=O)NCC(c2cccnc2)O)N1C(c1cc(Cl)ccn1)=O 36769,C1(CNC(=O)CCc2ccc(Cl)s2)CN(C(=O)C(F)=CCCF)CC12CCC2 36770,C(=O)(CCCCCNC(C)=O)NCC1CC(NC(COCCC)=O)C1 36771,C(=O)(C(C)C(C)(C)C)NCCCN(C(=O)C=Cc1cccc(CO)c1)CC 36772,c1(CC)ccncc1NC(c1cc(CNC(=O)C(O)c2ccsc2)on1)=O 36773,c1(CN2CC(F)CC(C(=O)NC(CCC)C(=O)NC)C2)ccc(F)c(NC)c1F 36774,C1(CNC(c2c(C)cn(C)n2)=O)COC(C)(C)CN1C(=O)CCCN1CCCC1 36775,N1(C(C(N)=O)=O)CC2CC1CN(C(c1cc(C(N)=O)co1)=O)C2.N1(C(=O)N)CCCC1 36776,C1(NC(C(=Cc2ccccn2)C)=O)C2CCC1N(C(c1cc(C(F)F)no1)=O)C2 36777,C1(C2CC2)(C(=O)NCC(c2ccccc2)CNC(C)=O)CC1 36778,CCCC(C)CC(C)(c1nnnn1C1CC1)NCCc1cn(C)nn1 36779,C(CCCC(=O)NCC1C2CCCC12)N(C)C(C1CCCN1C=O)=O 36780,c1(C(=O)NC2C(CNC(C=CC(C)C)=O)CCCC2)ccc2c(c1)B(O)OC2 36781,Cc1c(NCCCN2CCCN(C)CC2)nc[nH]c1=NCC1CC2(C1)CC(O)C2 36782,N1(C(C=CC)=O)CCC(CNC(=O)CC2CCNC2=O)C1C(C)(C)C 36783,c1(C(=O)OC)ccc(CN2CCCN(CCC3CC3F)CC2)c(C)c1 36784,C1(C)(COC(C(C(C)C)n2cncn2)=O)CCCN(C(=O)OC(C)(C)C)C1 36785,c1(NCCCCC(N)=O)[nH]c(=NCCCC2CC2(Cl)Cl)nc2scnc12 36786,c1(C(=O)NCC(CCC)NC(C2CCCN2CC)=O)c(OC)ncnc1C 36787,C#CCCCC(C)C(=O)N1CCOC(CC(=O)NC(c2n[nH]c(C)n2)C)C1 36788,C1(C(=O)Nc2cc(OC)c(O)cc2)CC12CCN(C(c1cc(O)n(C)n1)=O)CC2 36789,CCS(=O)(=O)CCN=c1[nH]c(N2CC3CCCCC3C2)nc2c1CCC2 36790,Cc1ccc(CC(N2CCC2CNC(=O)CN(S(C)(=O)=O)C)=O)c(Cl)c1 36791,C1(O)(C(C)NC(c2ccc(SC)s2)=O)CCN(C(=O)COC(C)(C)CC)C1 36792,C(=O)(C=C1SCC(=O)N1C)NC1CCN(C(c2n(CCC)ccc2)=O)CC1O 36793,CC1CC(C(=O)NC2(CCNC(=O)Cc3ccc(Br)nc3)CCCC2)=NO1 36794,C(=O)(C1CCc2ccccc21)N1CCCC(C(C)NS(C(CC)C(C)C)(=O)=O)C1 36795,c1(CC(=O)NCCC(C)NC(C2CC23CC3)=O)c[nH]c2ccc(Cl)cc12 36796,N1(C(=O)CC2CCCN(C(c3cnn(C(F)F)c3)=O)C2)CCC(CO)C(F)C1 36797,CC(CCCCNC(C1CCCC12CC2)=O)NC(c1conc1C(F)(F)F)=O 36798,c1(CC(=O)NCC2C(NC(=O)Cc3sccc3Cl)CC2)ccccc1Cl 36799,c1(CNC(c2cc(C)ns2)=O)nc(C)c(C(=O)NCC(C2CC2)N(C)C)o1 36800,CC1=NOC(C)(C(=O)NC(CO)C(C)NC(=O)Cn2nc(C)cc2C(F)F)C1 36801,C(C1=NOC(CC2CCOC2)C1)NCC(c1ccccc1)N(C)C 36802,C(CCC(=O)NOCC(=O)NCC12CCC(CC1)CO2)SC 36803,C(c1c(C)noc1C)=CC(N1CCC(N(CCC)C(C2CCCN2C=O)=O)C1)=O 36804,N1(C(CSCCCC)=O)CCN(C(c2cc3scc(C)c3[nH]2)=O)CC(O)C1 36805,N1(C(C(C(C)O)NC(=O)OC(C)(C)C)=O)CCCN(C(=O)C2CC2)CC1C 36806,Cc1cc(C(N2CC(CNC(=O)C(C)O)C(C)(C)C2)=O)cc(C(F)F)c1 36807,N1(C(C2(SC)CN(C(=O)C(C3CCOCC3)O)C2)=O)CC(C#N)(CCF)C1 36808,CC(CN=[N+]=[N-])NC(C1COCC1NC(=O)CC1(C)CCC1)=O 36809,C12(C(N(C)OC3CCCC3)=O)CC(C)(CN1C(c1cc(C(N)=O)co1)=O)C2 36810,Cc1ccc(CNC(c2nnnn2C(C)C)(C)CC2C=CCC2)c(F)c1 36811,c1(OC)ccc(CCNC(C2CC3(CC3)CN2C)=O)c([N+](=O)[O-])c1 36812,C1(CNC(COc2cc(C)on2)=O)CN(C)CCN1C(c1ccncc1Br)=O 36813,C1(CC)CN(C(c2cc[nH]n2)=O)CCC1NC(=O)Cc1ccccc1Cl 36814,CC(C)(CCCO)C(=O)NC1CCCCC1CNC(c1c[nH]nc1[N+](=O)[O-])=O 36815,C(=O)(C(CNC(C1(C)CC(F)(F)C1)=O)CC=C)N(CCOCC#C)C 36816,Cc1nc(N2CC3C(CNC(=O)CC(C)CC(C)(C)C)C3C2)c2cc[nH]c2n1 36817,c1(C(c2nnn[nH]2)NCC(N)=O)ccc(NC(C2CC23CC3)=O)cc1.C(C)(C)(C)O 36818,N1(C(C(CC)OCC)=O)CC(NC(=O)C(c2cnn(C)c2)C)CC12CCOCC2 36819,C1(C(N2CC(O)(CCNC(=O)COCC(F)(F)F)C2)=O)CCC(C2CCC2)CC1 36820,N1(C(C(=O)OCC)=O)CCC(C(F)C(=O)Nc2ccc(SC)cc2)CC1 36821,C(=O)(CC(C)c1ccco1)N(CCCN(C(=O)CC#N)C)C 36822,C=C(CNC(C1(CCF)CC1)=O)CCNC(c1csnc1OC)=O 36823,C1(N(C(C(c2ccccc2)C)=O)C)CCCCN(C(c2ccncc2Cl)=O)C1 36824,Nc1ccnc2c(C(=O)NC3CN(C(C4CCCSC4)=O)C3)cnn12 36825,C1(NC(=O)CC2(CNC(C3(Cl)CC3(F)F)=O)CC2)CCC(C(F)F)CC1 36826,c1(C(N2CCOCCC2C2CC2)C(=O)NC)ccc(S(=O)(=O)C(C)C)cc1 36827,c1(C(=O)NC2CCC(CNC(c3nccc(N(C)C)c3)=O)C2)cnc(N)c(Cl)c1 36828,N1(C(c2c(CCCC)ocn2)=O)CCN(C(=O)Cc2ccns2)CC1CO 36829,C(C(O)CC(=O)N1CCCC1C(=O)NCC1CC1)NC(=O)OC(C)(C)C 36830,Cc1c(C(=O)NCC2CCCN2C(=O)Cc2cn(C)nc2Cl)sc2nccn12 36831,c1(C(N2C(COC)CN(C(c3nc(Cl)sc3C)=O)CC2)=O)cc(C)cc(C)c1O 36832,O(C=CC(=O)NC(CNC(=O)CCCOC1CCOCC1)C(C)C)CC 36833,c1(C(=O)NCC2(O)CCN(C(CC)=O)C2)ccc(C#N)cc1C 36834,C(=O)(CC1CCC(C)(C)c2ccccc21)NCCCNC(C(COC)O)=O 36835,CN=c1[nH]ccc(C(N2CCCC(NC(C3(F)CC=CCC3)=O)C2)=O)c1[N+](=O)[O-] 36836,c1(SC)ncc(C#N)c(N2CCCC(C(N3CCCC(CO)C3)=O)C2)n1 36837,c1(NC(C(C2CCCCC2)NC(C=CCOC)=O)=O)ccc(C)c(CO)c1 36838,c1(CC)n[nH]cc1C(=O)NCC(N1CCC(C(=O)NCCOC)C1)=O 36839,C(CC(C)C)(C(=O)N1CCC(C)C(C(=O)NOC(COC)COC)C1)OC 36840,C=CCC(C(=O)N(C(C)CSC)C)NC(=O)C(C)N.C(C)=O 36841,N1(C(=O)CC2C=CCC2)CC2(CCN2C(c2cc(-c3ccncc3)on2)=O)C1 36842,C1(CC(N2CC(CNC(Cc3cccc(SC)c3)=O)C2)=O)CCC2(CCC2)CO1 36843,CCCC(CCNC(=O)C(C(C)OC)NC(c1cccn1CCC)=O)C1CC1 36844,Cc1cc(O)ccc1C(=O)NCC1CCCN(C(=O)CCC2CCCN2C)CC1 36845,Cc1nn(C(C)C)c(C)c1C(=O)NC(C1CCN(c2ncncc2Cl)C1)C 36846,CC(CC(F)F)C(=O)N(C)CC1CCCCN1C(=O)C(O)Cc1ccccc1 36847,N1(C(C2CC(=O)NC(=O)N2)=O)CCC(CNC(=O)Cn2cc(Cl)cn2)C(F)(F)C1 36848,c1(COCC(N2C(CNC(=O)CC3CCCOC3)CC2)=O)ccnc(O)c1 36849,Cc1nc(C2CC2)sc1C(=O)NC1(C)CCN(C(=O)C(C)NCCC(C)C)C1 36850,C1(CN(C(C2CC(OC)(OC)C2)=O)C)CCc2nc(C(F)(F)F)cn2C1 36851,N1(C(C2CC(=O)NC2)=O)CC2(C1)CN(Cc1cc(Cl)ccn1)C2 36852,N1(C(C(CC)NC(C)=O)=O)CCN(C(=O)Cc2nc([N+](=O)[O-])n[nH]2)C(C(C)C)C1 36853,c1(-n2c(C(C(C)(C)SC)NCC(C(C)C)OC)nnn2)ccc(F)cc1 36854,C1(C(C)NC(=O)CC2CC3CC3C2)CCN(C(C2(COCC)CCCO2)=O)CC1 36855,C1(NC(C(C2CCC(F)(F)CC2)OC)=O)CC2CCC1N2C(c1ccnn1C)=O 36856,N1(C(C2(C)CC(=O)C2)=O)CCC(C)(C)C(CNC(c2c(F)cccc2F)=O)C1 36857,N1(C(C(CCNC(CC(CC)C2CCC2)=O)O)=O)CC2CCC(C1)O2 36858,N1(CCC)CCN(S(=O)(=O)N(C)C)CC1.c1(C2CNC(=O)N2)c(F)cccc1F 36859,N1(C(C(CC)N(C)C)=O)CC=C(CCNC(=O)CC2CN3CCN2CC3)CC1 36860,c1(C(=O)NC2CCCC(NC)C2)cccc2c1OCCC2 36861,C1(C(N(C)CC2CCN(C(=O)Cc3nccn3C)C2)=O)CCC(C)(C)CC1 36862,C1(CN)CCN(C(=O)Cn2cc(CN3CCCCC3)nn2)C1 36863,CC(C)CC(C)CC(=O)NC(C)CCN(C)C(c1nncn1C1CC1)=O 36864,N1(C(c2c(C)nc(CC)s2)=O)CC2(CCCCN(C(C3CN(C)C3)=O)C2)C1 36865,C1(NC(CSc2c(C)n[nH]c2C)=O)CCN(CCc2nccc(CO)n2)C1(C)C 36866,c1(N(C)CCOCC(C)(C)C(C)(F)F)ccc(S(=O)(=O)NC2CC2)cn1 36867,N1(c2nccc(CC)n2)CCC2(NC(c3cn(C)nc3COC)=O)CCCC12 36868,c1(CC)cc(Cl)ccc1NC(c1nnnn1C1CCOCC1)(C1CC1(Cl)Cl)C 36869,c1(-c2nc(C)c(C(=O)Nc3cc(F)c(Cl)cc3F)cc2)ccc2c(C)[nH]nc2c1 36870,c1(OC)cc(SC)ccc1CNC(Cc1sccc1Br)C(=O)O 36871,C1(CNC(C=C(C)C)=O)CCC(CNC(=O)Cc2ccn(C)c2)CC1 36872,C1(OCCCCOC(c2cn(C3(C(=O)O)CC3)nn2)=O)C=CCCCC1 36873,C1(NC(CSCCCC)=O)CC(OC)CN(C(c2cc(C)nc(C)c2)=O)C1 36874,c1(C(N2CCCC(F)(CNC(C3C(C)(C)CC3)=O)C2)=O)n[nH]c2cc(Cl)ccc12 36875,N1(C(CCCCCOCC)=O)CC2CCC1CN2C(C1C(C)(C)C1(F)F)=O 36876,C1(NC(c2cccc(C)n2)=O)CC2CC1N(C(=O)C(F)(F)CCn1ccnn1)C2 36877,C(=O)(C(C)C(F)F)NC(=O)NC1(CN)CC1.c12ccc(o1)CN(CC)C2.C(C)(C)(C)O 36878,C1(C(=O)NCC(=O)N(C)CC)CCC(CNC(c2csc(=N)[nH]2)=O)O1 36879,C(=O)(C1CCCc2ncccc21)N1C2CC(CN(C(c3ccc(Cl)o3)=O)C2)C1 36880,c1(OCC)ncc(NC(=O)CC2CCCN(C(=O)C(C)C(C)C)C2)cn1 36881,CC(C)CC(F)(F)C(=O)NC1CN(C(c2c(Cl)nn(C)c2Cl)=O)CC2(CC2)C1 36882,C(=O)(CC(C)CC(=O)NCCC(C)NC(=O)Cc1ncn2c1CCCC2)OC 36883,N1(C(c2cc(C)sc2)=O)CCCC(NC(c2ccn(C)c2C2CCC2)=O)C1C 36884,N1(C(c2cn(C3CC3)cn2)=O)CCCC(F)(C(N2CCCCC2CO)=O)C1 36885,c1(C(N2CCC(N(C(c3c[nH]nc3SC)=O)CC)C2)=O)cn2ccc(C)cc2n1 36886,C1(NC(C=CCOCCOC)=O)CC(O)(CC2(C(=O)NC)CC2)C1 36887,C1(NC(CNS(NC)(=O)=O)=O)CCCC12CCN(C(c1ccc(OC)nc1C)=O)C2 36888,c1(C(N2CC(C)C(CNC(c3cn[nH]c3)=O)C2)=O)nc(Br)c2ccccn12 36889,N1(C(CCCc2onc(CCC)n2)=O)CCN(C(=O)C(O)CCSC)C(CC)C1 36890,Cc1ccc(C(=O)N(C2CCCC2)CCNC(=O)C(C)(C)C(N)=O)c(C)c1Br 36891,c1(-c2n(-c3ccc(C)cc3)nc(CCC(F)(F)F)n2)ccc(C(C)(C)C)c(F)c1 36892,C(=O)(C(F)CC1CN(C(=O)C(c2ccccc2)O)C1)N(CCSC)CC 36893,C12(CNC(=O)COc3ccon3)COCCN1C(=O)CN(C(C1CCOC1)=O)C2 36894,c1(C(N2CC(O)(CN(C)C(c3cccn3C)=O)C2)=O)cccc(F)c1F 36895,CC1CN(Cc2ccccc2)CCC1NCc1ccnc(C2CCCC2)n1 36896,N1(C(C(c2ccnn2C)C)=O)CCC=CC1C(=O)NOCC1CCCO1 36897,C1(NC(CCC#C)=O)CC2CC1CN(C(c1cc(C(F)F)no1)=O)C2 36898,c1(NC(C2(NC(C(C)OCC=C)=O)CCSC2)=O)c(C)ccn(C)c1=O 36899,c1(C(N2CC3CCC2CN3C(C23CCC2C3)=O)=O)cc2oc(Br)cc2[nH]1 36900,CCC(C)CC(=O)N1CCC(C(c2ccccc2Cl)N(C2CCCCC2)C)CC1 36901,c1(C(N2C(C(=O)NC(COC)C)CC(F)C2)=O)cc(Br)ccc1C(F)(F)F 36902,c1(CCCC(=O)NCC(CC=C)NC(C2(COC(C)C)CC2)=O)ccc(O)cc1 36903,c1(C(=O)NC2CC(=C)CN2c2nccc(C(=O)OC)n2)cc2sccc2s1 36904,N1(C(C(COC)(F)F)=O)CC2(CC(CNC(=O)Cc3ccccc3F)C2)C1 36905,S(=O)(=O)(c1cnc(NCC2(Br)CC2)c(Cl)c1)N1CCCC(C(C)O)C1 36906,CC1(C)CN(C(C2CCN(C(C3CC(O)C3)=O)C2)=O)CC1O 36907,C(C(=O)NC(C)(CNC(=O)C=Cc1cn[nH]c1)CO)(C(C)(C)C)SC 36908,c1(CC(=O)OCC)ncc(NC(=O)C(C(C)C)NC(=O)CC(C)C)cn1 36909,C12(C(=O)NCCC3N(C)CCC3)C(NC(C3CC4C=CC3C4)=O)C3CC1C2C3 36910,c1(C(C(N2C(CNC(c3c(C)nsc3)=O)CCC2)=O)C)cccc(OC(F)F)c1 36911,C1(CNC(Cc2cc(OC)ncc2)=O)CCN(C(C2CC=C(C)CC2)=O)C12CC2 36912,C12(CC)CCC(C(=O)NC3CCC(NC(C4(C)CC(F)C4)=O)C3)(CC1)CO2 36913,N(C(=NCC1CCC1)N1Cc2ccccc2C(F)(F)C1)Cc1c(OC)ccnc1 36914,N1(C(c2c(N)ncc(C)c2)=O)CC2CC3CC2C1C3NC(c1csc(C)c1C)=O 36915,c1(C(=O)NCCCC(C)NC(CCCCC)=O)ccccc1C#N 36916,CC1CN(C(=O)C=CC2CCCN2C)CC1(C)C(=O)Nc1ccc(F)c(CO)c1 36917,c1(N(C)CC2CCCN(C(C34CC(C)(CO3)C4)=O)C2)ncc(C#N)cc1F 36918,N1(C(c2sc(C(F)(F)F)nc2Br)C(=O)NCCCC)CC2(CCC2)CC1CO 36919,C(C(C)(C)C#CC(=O)NCC(O)CC(F)(F)F)NC(C1CCCC(OC)C1)=O 36920,C1(C(N(C)CCOCCCO)=O)CCN(C(C2(N(C)C)CCCCC2)=O)CC1(C)C 36921,C1(NC(C(CN(C(C2(CC)CCCO2)=O)C)C)=O)CCC(C#N)CC1 36922,Cc1c[nH]nc1C(=O)N(CCCNC(=O)C(Cc1ccccc1)N(C)C)C 36923,C1(OCC)CN(C(c2nccc(C)n2)=O)CC1CNC(c1ccc(SC)cc1)=O 36924,C(CCCC(=O)N1CCC(NC(=O)CSc2ccc(F)cc2)C(C)C1)(OC)OC 36925,N1(C(C(CC)N(C)C)=O)CCSCC1CCNC(=O)C(O)c1ccco1 36926,C(=O)(C1CCC(=O)c2ccccc21)N1CCCC(NC(CNC(CC)=O)=O)C1 36927,c1(CC(=O)NC2CN(C(C(C)C)=O)CC23CCC3)nn(C)c2ccccc12 36928,c1(C(=O)NCC2(C)OCCN(C(C3CN(C(C)=O)C3)=O)C2)cc2ncccc2[nH]1 36929,c1(CNC(C2(CCC)CCC2)=O)cc(C(=O)NCCCCCF)co1 36930,c1(CN(C(=O)Nc2cnoc2C(C)C)Cc2c(C)nsc2)cccc(Cl)c1 36931,C1(OC)CC(NC(c2cc(C)nc(O)c2)=O)CN(C(=O)C(C)Cc2cnc[nH]2)C1 36932,C(=O)(CC(O)C(C)C)NC1C(NC(C(CC#C)C)=O)CCCC1 36933,N1(C(C2(SC)CC2)=O)CC(CCC(=O)NC2(CC(C)C)CC2)C1 36934,N1(C(c2ccn(CC)n2)=O)C2CCC(C2)C1CNC(c1cc(C)c(C)o1)=O 36935,C(=O)(CC(F)(F)F)NCCC1(OC)CN(C(C2CCC(C(F)(F)F)C2)=O)C1 36936,c1(C(=O)NC2C(C)CN(C(=O)CCC(=O)N(C)C)C2)ccc2cncn2c1 36937,Cc1c(N)cc(C(=O)NCC(C)NC(=O)C(c2cccc(Cl)c2)O)cc1[N+](=O)[O-] 36938,c1(C(N2C(CNC(c3n(CC)ncc3)=O)CC2)=O)cc(C2CC2)nc2ccnn12 36939,C1(OC)CN(C(C23CC2CCN3C(=O)C(C2CCCCC2)=O)=O)CC1(C)C 36940,N1(C(C(CNC(C2C=C(C)CS2)=O)OC)=O)CCOC(C)(C)C1C 36941,c1(CNC(C2(CC)CC2)=O)ncoc1CCNC(C1CC(C)(C)O1)=O 36942,Cc1cc(O)ccc1C(N1CC=CC(NC(=O)Cn2ccc(Br)n2)C1)=O 36943,c1(C(=O)NC2C3(CC(NC(c4c(C)cc(Br)o4)=O)C3)C2)cc[nH]c2nccc1-2 36944,C(=O)(CCC(=O)OCc1csnc1C1CC1)OCC 36945,c1(CC(N2CCC(C(C)NC(=O)C(N)=O)C2)=O)cccc2ncccc12 36946,C(=O)(C(C)(C)CCCNC(=O)C(c1cnn(C)c1)C)N1C(CC)CCOCC1 36947,C(C(C)(Cn1cccn1)NC(c1c[nH]c(=N)o1)=O)NC(CSC)=O 36948,c1(C(N2CCC(NC(C(CCSC)OC)=O)C(F)C2)=O)cc2oc(C)c(C)c2[nH]1 36949,c1(CC(=O)OCC2(C)CCCO2)cccc(Cc2ccccc2O)c1 36950,CC1CCN(C(=O)C(c2ccoc2)NC(=O)COCCC(C)C)CC(C)O1 36951,CCCC(C)(C)C(=O)NC1C=CC(C(N2CC(=O)NC(C(=O)OC)C2)=O)C1 36952,N1(C(c2nncc(OC)c2)=O)CC(F)(F)CC1(C)CNC(c1ccc(Cl)cn1)=O 36953,CC1(c2ccc(-c3noc(CCNC(=O)OC(C)(C)C)n3)cc2)NC(=O)NC1=O 36954,c1(C(C(=O)NCCC2(C)CC2)N(C)Cc2cnc(CC)s2)ccc(C)cc1Cl 36955,C1(C)(CNC(CN(C(C)C)C)=O)COCCN(C(C2CCC(C)(F)CC2)=O)C1 36956,C(=O)(C(CO)C(C)(C)C)NC(CCC#C)C(=O)N(C)Cc1nccn1C 36957,C(=O)(C1CCc2c[nH]nc21)N1CC2(C(NC(=O)Cn3ncc(O)nc3=O)CC2)C1 36958,c1(C(=O)NC2CCCN(C(CC3(COC)CC3)=O)C2)cc2cc(F)cc(F)c2[nH]1 36959,C1(=CC(=O)NC2(CC=C)CN(C(c3ccc(CSCC)o3)=O)C2)CCC(C)CC1 36960,C1(O)(C(C)(C)OC)CC(NCCN(c2ccccc2)S(C)(=O)=O)C1 36961,C1(O)(CN(C(C(C)CF)=O)C)CCN(C(C2CCCC2C(F)F)=O)CC1 36962,CC(=O)C(C)(C)CC(=O)N1CC=CC(C(=O)NCC=CCCOC)C1.C 36963,CCC(C)CCN=c1[nH]c(=NCC2(CO)CC3CCC2CC3)c2ncccc2[nH]1 36964,CC1(C(=O)NCC2CCCC(CNC(C3CCC(=O)O3)=O)C2)CCC2CC2C1 36965,c1(CNC(c2c(C)cno2)=O)cccc2c1CCN(c1cc(O)nc(O)n1)C2 36966,c1(C(=O)NC2CC(CNC(C3CCC(CC)C3)=O)C2)ccc(OC2CCC2)nc1 36967,C(=O)(C1=COCCC1)N(CCNC(CS(CC)=O)=O)CCc1ccccc1 36968,C1(C(N2CC(=CCC)C2)=O)CN(C(C2CC(N(C)C)C2)=O)CC1F 36969,Cc1cc(C2(C(=O)NC3CCCN(C(C4(O)CCCCC4)=O)C3)CC2)cc(C)c1 36970,Cc1ccnc(-n2cc(CN3CCC(C(NOCCCC(F)(F)F)=O)C3)nn2)n1 36971,c1(C(N2C3C(NC(C(C)c4ccsc4)=O)C(C3)C2)=O)ccc2cccnc2n1 36972,N1(C(CSCCC=C)=O)CCCC(O)(CNC(=O)C(C(C)C)NS(C)(=O)=O)C1 36973,N1(C(CCCCC(N)=O)=O)CC(NC(=O)C(O)C2CCC2)CC12CCCCCC2 36974,C(CN=C(NCc1cccs1)N1CC(O)C(C)(C)C1)c1ncc(C)cn1 36975,c1(C(=O)NC(CNC(C2(OCC)CCC2)=O)C2CC2)scc(C)c1C 36976,CCCCC(O)C(=O)N(CC(=O)NC1(CC)CCCC1)C(C)C 36977,C=C(C)c1cncc(C(c2nnnn2CCCSC)NCC2(C#N)CCCC2)c1 36978,C(=O)(C#CC1(C)CCCO1)N(CCC(=O)NCC(CC)C(C)C)C(C)C 36979,c1(NC(COC2CN(C(c3cncn(C)c3=O)=O)C2)=O)cn(C)c(=O)nc1O 36980,c1(CN(C(C(CNC)(C)C)=O)C(C)C)cc(OC)c(OC)c(OC)c1 36981,C1(O)(CC)CCN(C(=O)C=CC(C)NC(C2CCCC2O)=O)C1 36982,N1(C(c2ccn(CCCC)n2)=O)CCC2(NC(=O)C=CC3CC3)CCCCC12 36983,c1(NC(C)=O)ccc(F)c(C(=O)NC2CCN(C(c3cnn(C)n3)=O)C2)c1 36984,C1(CNC(CCOCCC)=O)CCC2(CCC2)CN1C(=O)C(C)C(C)COC 36985,c1(CC(=O)NCC(C(F)(F)F)N2CCN(c3nnco3)CC2)ccc(Cl)cc1Cl 36986,C=CCC(CC=C)C(=O)N1CCC(C(=O)N(CCCCC)C)(CC)C1 36987,C1(NC(C(C)(C)OC)=O)CCC(C)C(C)C1 36988,c1(C(=O)NCC2(C(C)(C)C)CCN(C(c3onc(C)n3)=O)C2)cnc2c[nH]nc2c1 36989,N1(C(C=CC=CC)=O)CC(NC(c2ncc(F)cn2)=O)CC1c1ccccc1 36990,Cc1c(C(=O)NCC2CC(C)N(C(c3coc(C(F)F)n3)=O)C2)sc(Cl)c1Cl 36991,n1(CC(=O)NCCOc2c(C)cccc2F)ccc(=NC(=O)CN(C)C)nc1O 36992,c1(C(=O)NCC2N(C(CC=CC=C)=O)CCC2)cncc(F)c1C 36993,c1(CNC(C2C(C(=O)OC)OCC2)=O)ccc(OC(F)F)nc1Cl 36994,CCCC(C)(CC)C(=O)NC1CCN(CCNC(C2CC23CCSCC3)=O)CC1 36995,C1(C(N(C2CN(C(C(c3cccnc3)C)=O)C2)C)=O)C(C)(C)C1(C)C 36996,C1(NC(CCCCCC)=O)CC2CN(C(=O)C(=Cc3cccs3)C)CCN2C1=O 36997,CCC(CC)C(=O)NCC.C1(C)CC(CNC(=O)COCCOCCOCC)CO1 36998,c1(-c2nc(C(C)Nc3cc(S(C)(=O)=O)co3)[nH]n2)ccc2ccccc2c1 36999,c1(CC(=O)NCCC2C(C)CCCC2)cc(Br)ccc1Cl 37000,Cc1cc(C(=O)NCCCCC(C)NC(=O)CCC2(C)CC2)cc(N)c1 37001,N1(C(c2cc(C(C)C)on2)=O)CCC(C(=O)NC(C)(C)C(C)(C)O)CC1 37002,c1(C(N(CC(C)N(C(c2nc(C)oc2C)=O)C)C)=O)ncc(Cl)cc1Cl 37003,c1(OC)c(CN2CCC(CC(=O)Nc3cnc(Cl)nc3C)CC2)cc(Cl)cc1Cl 37004,N1(C(C2(CCC)CC2)=O)CCC2CCCN(C(c3cn(C)nc3C)=O)C2C1 37005,C1(C(=O)OCC)C2COC(C(N3CCCC3CNCC3CC34CCCC4)=O)CC12 37006,C1(C(=O)NCC2N(C(c3nc(C)sc3)=O)CCCC2)CC2CC1C1C2C1(F)F 37007,C#CCC(CC(F)F)C(=O)N1C(C(=O)NCC2(O)CCCCC2)CCC1C1CC1 37008,c1(SC)cc(C(=O)NCC2CN(C(=O)CCSC(F)(F)F)C3CC23)ccc1F 37009,c1(C(=O)NC(C2N(C(c3c(C(C)C)ncs3)=O)CCC2)C)cc2n(n1)CCC2 37010,c1(OC)ccc(Br)c(C(N2CCCC(O)(CNC(=O)C(C)SC)C2)=O)c1 37011,c1(C(=O)NC2C(NC(C(CC)O)=O)C2)ccc(C(F)F)nc1 37012,C1(OCC)CC(NC(=NCCF)NCC2CCSCC2)C12CCCCC2 37013,C1(C(=O)NC(C)C(CO)NC(=O)Cc2ccn(C)c2)(COC)CCCC1 37014,c1(C(=O)NC2C(CC(=O)NCCn3cc(Cl)cn3)CC2)ccc(C(F)F)o1 37015,c1(NC(c2cncc(CNC(c3cnn(C)c3N)=O)c2)=O)ccccc1N=[N+]=[N-] 37016,c1(N2CCC(c3onc(-c4nccc(C)c4)n3)C2)cc(Cl)ccc1Cl 37017,C1(NC(C(F)=C(C)C)=O)CCCC(NC(c2cc(Cl)n(C)n2)=O)C1 37018,c1(C(N2CC3CC2CN3C(c2nc3ccccc3o2)=O)=O)cccn2ncnc12 37019,CC1CCC(O)(C(=O)NC2CCCN(C(=O)C(C)CSC(F)(F)F)C2C)CC1 37020,C1(C2CCN(C(=O)CCc3cc(F)cc(F)c3)C2)(NC(C2C(CC)C2)=O)CC1 37021,c1(C(=O)NCC(CN(C(C2(OCC)CCC2)=O)C)O)c(C)nn(C)c1N 37022,CC(C)C(CC(=O)N1CCC(O)CC1)NC(c1cocn1)=O 37023,CCC(CC(=O)NC(C(=O)NCC1(CCOC)CCC1)C(C)O)OC 37024,CC(C)C1=NOC(C(=O)NCC2CC3CCC2N3C(C23CC(C)(CO2)C3)=O)C1 37025,CCC(C)C(O)C(=O)N1CCCN(C(c2[nH]c(-c3cccnc3)nc2C)=O)CC1 37026,c1(C(=O)NC(C)C(C)NC(c2cnnn2C)=O)c(Cl)c(Cl)cc(Cl)c1Cl 37027,c1(C(=O)NC(C)Cn2cc(Br)cn2)cc(S(=O)(=O)N(C)C)ccc1Cl 37028,N1(C(c2ccc(C)n2C)=O)CCCCC2(CCN(C(c3cncc(N)n3)=O)C2)C1 37029,CC1(C)CCCCCC1NC1CCCN(C2COC2)C1 37030,Cc1ccc([N+](=O)[O-])cc1C(N1CCN(C(=O)Cc2ccc(F)cc2)CC1C)=O 37031,C1(NC(C2C(C(C)C)CN(C(C3CSC3)=O)C2)=O)CCNC(=O)CC1 37032,CP(C)(=O)C(O)C(=O)N(C1CCCN(C(=O)C=CBr)C1)Cc1ccccc1 37033,CC1CNc2cc(C(=O)NC3CCC(N(C)C(C4CC(F)C4)=O)CC3)ccc2O1 37034,C(C(C(=O)NOC(C)(C)C(=O)OC)C(C)(C)C)NC(C(CCC)C#N)=O 37035,N1(C(c2cc(OC)n[nH]2)=O)CC(CNC(C2CCCN2C)=O)C2(CC2)C1 37036,C1(C(=O)NCCCCN2CCOC2=O)Cc2ccc(Br)cc2N1 37037,c1(N2CC3CN(C(Cc4cc(C)cc(C)c4)=O)CC3C2)nc2ccc(Cl)cc2s1 37038,C=C(C)C(CC(=O)NCC1CCC1NC(=O)Cc1ccc(F)cc1F)OOCC 37039,C1(NC(c2n[nH]c(O)n2)=O)CCN(C(C2CCCC(F)(F)CC2)=O)CC12CCC2 37040,C1(NC(C=C(CCC)C)=O)(COC)CCN(C(=O)CCC=C(C)C)C1 37041,c1(C(=O)NCCN(C(=O)C(F)C2CCC2)C2CC2)cc2ccccn2n1 37042,C(=O)(CCC1CC1(F)F)N(C)CCOCCN(C)C(C1CC1C(F)(F)F)=O 37043,C1(CC(=O)NCCOC2CCN(C(C(C)(C)CC3CC3)=O)C2)CCCCC(=O)N1 37044,Cc1nn[nH]c1C(N1CCCC1CN(C(=O)CC1(CS(C)(=O)=O)CC1)C)=O 37045,c1(C(=O)NC2CS(=O)(=O)CC2NC(c2cnccc2Cl)=O)cn2cnnc2cn1 37046,C12(NC(C(=O)NCC(COCC)O)=O)CC3CC(C1)CC(O)(C3)C2 37047,c1(OC)c(C(=O)NCC2CCCN(C(=O)C(C)S(N)(=O)=O)C2)ccc(Cl)c1C 37048,N1(C(C=CC2N(C(CC=CC(C)(C)C)=O)CCC2)=O)CCOC(C)(C)C1 37049,c1(C(N(C)CC2CN(C(c3ccncn3)=O)C2)=O)cc(N)cc(O)n1 37050,C1(C(N(CCOCCNC(c2c(C(C)C)scc2)=O)C)=O)CC2CCCC2C1 37051,C(=O)(C(C)(C)C(C)(F)F)N1CCN(C(c2cc(C)nc(O)n2)=O)C(CO)C1 37052,N1(C(CC(CC)CN(C)C)=O)CC2CCCC(C1)N2C(=O)C1=NNC(=O)C1 37053,N1(C(C=CC=CC)=O)C2CCC1(CNC(=O)CCCN1CCCC1)CC2 37054,c1(C(=O)NC2(CC(=O)N(CCOCCOC)C)CCCCC2)cnccc1C#N 37055,C1(C(N(CC(N2CC(OC(F)F)C2)=O)C2CCC2)=O)CCCC1O 37056,CC(C)CC(CNC(C1(C(F)(F)F)CC(F)(F)C1)=O)NC(c1ccccn1)=O 37057,C1(CC=CC)CCCN(C(=O)CC2CC2CNC(=O)C(C)SCC)C1 37058,C1(NC(c2c(OC)cnc(Br)c2)=O)CC2(CCN(C(c3c[nH]cc3C)=O)CC2)C1 37059,N1(C(CC(COC)C)=O)CC(NC(c2cccc(C)c2)=O)CC12CCC2 37060,c1(OC)cnn2c1CN(C(=O)Cc1ccc(-c3nn[nH]n3)cn1)CC2 37061,C1(C(N2CC(OCCNC(c3c(C(C)C)c[nH]c3)=O)C2)=O)CC(=O)NC(C)C1 37062,c1(CC(C)CN2CCCC2)cc(C(=O)O)cc(Cl)c1 37063,CC1CN(CC(=O)NCC2CCN2C(=O)CN(C)Cc2ccccc2)CC1 37064,Cc1cc(F)ncc1C(=O)NC(C)CC1CN(C(=O)CCOC2CCOCC2)C1 37065,N1(C(c2cc(COC)[nH]n2)=O)CC2CCC(C1)C2NC(c1cc(COC)cs1)=O 37066,c1(C(=O)NCc2nc(-c3ccc(F)cc3F)cs2)c(I)cnc(Cl)c1F 37067,c1(NC=O)ccon1.C1(C(=O)OCC)C(C(=O)NCC2(c3cc[nH]n3)CC2)C1(F)F 37068,c1(C(CC(=O)NC2CN(C(C3(C(=O)OCC)CC3)=O)CC2O)C)ccc(F)cc1F 37069,N1(C(c2[nH]nnc2C2CC2)=O)CC2(C=C(C(=O)NCC3(CCO)CCC3)CO2)C1 37070,c1(-c2cc(C)cc(O)c2)ccn2cc(C(N3CCCC3C)=O)nc2c1 37071,N1(C(CN(C)C)=O)CC2CCCN(C(c3ccc4oc(O)nc4n3)=O)C2C1 37072,Cc1ccc(OCC(=O)NC2CCC23CN(C(c2[nH]ncc2C#N)=O)C3)c(C)c1 37073,N1(C(CC(C)OC)=O)CCn2c(CNC(=O)CSc3nnnn3C)nnc2C1 37074,Cc1cccc(C(=O)NC2CCC(C)(CNC(c3cc(C(F)(F)F)no3)=O)C2)n1 37075,c1(C(CC)CC)cc(C(=O)NC2CC(CNC(=O)CN3CSCC3=O)C2)on1 37076,C=CC(CC)CC(=O)NCCN(C(=O)C(C)(C)CC)Cc1cccc(Cl)c1 37077,c1(C(N2CC(CNC(C=CC(=O)OCCCC)=O)C2)=O)cc(N(C)C)ccc1F 37078,c1(C(=O)NCCC(C(C)C)NC(c2nc(C)sc2)=O)c[nH]c2cc(F)ccc12 37079,c1(C(=O)NC2CN(C(C3(C=C)CCCCC3)=O)CC(C)C2)cc2ncccc2o1 37080,C1(F)(c2cc(C)cc(C)c2)CCN(C(=NCC(C)C)NCC2=CCCC2)C1 37081,c1(C(N2CC(N(C(c3cnc(COC)s3)=O)C)C2)=O)cc(C(C)C)ccc1O 37082,N1(C(C2CC3CC3C2)=O)CC2(C(=O)NCCCOCCO)CCC1CC2 37083,c1(NC(=O)NCCCO)cccc(SCC2NC(=O)NC2=O)c1 37084,c1(C(=O)NCC2COCC2NC(C2(C(F)F)CC2)=O)cn2cc[nH]c(=O)c2n1 37085,n1(CCC2CCC2)cc(CCCOC(N2CCOCC2)=O)nn1 37086,C(=O)(C1=CCCOCC1)NCC1(C)CCC(NC(=O)Cn2ccccc2=O)CC1 37087,c1(C(=O)NCCOCCNC(=O)CCc2ccc[nH]2)ccc(Cl)cc1Cl 37088,Cn1ccc(C2(C(N3CC(O)(CCNC(c4csc(C(F)F)c4)=O)C3)=O)CC2)n1 37089,c1(NC(C2CC3CCCCC3N2C(c2ccoc2)=O)=O)ccc2nc(O)[nH]c2c1 37090,N1(C(C2CN(C(N)=O)C2)=O)CCC(CC(c2ccccc2)O)C1 37091,N1(C(C2N(C(C)=O)CSC2)=O)CCCCCC(NC(c2csc3cncn23)=O)C1 37092,c1(C(=O)NC2CCN(C(C3CC(CC)(CC)C3)=O)C2)cc(C)c(Cl)cc1OC 37093,N1(C(CC2CC(OC)C2)=O)CCCC(C)C1CCNC(=O)CCC1CC(F)(F)C1 37094,C(=O)(CCCN=[N+]=[N-])NC1C(NC(c2nn(C(CC)C)c(C)c2)=O)COCC1 37095,N1(C(c2c(CC)noc2)=O)CCC(CCCCCNC(C2CC(C)CO2)=O)CC1 37096,c1(N2CCC3(CC(OC)C3)C2)nc(=NCc2cc(C)cs2)[nH]c2c1CCC2 37097,N1(C(C(C)OCC=C)=O)CC2CCCC(NC(c3cc(O)cc(=O)o3)=O)(C2)C1 37098,c1(NC(c2c(CC)ncs2)=O)ccc(C)c(C(F)(F)F)c1 37099,C1(NC(c2ccn(CC)n2)=O)CC2(C1)CC2NC(=O)CCc1ccc(C2CC2C)o1 37100,c1(C(=O)NCCC2CC(NC(c3cn(CCO)nn3)=O)C2)cc(Cl)ccc1O 37101,C1(CC=C)(NC(C2CC3CC3C2)=O)CCCN(C(C2CC(=O)N(C3CC3)C2)=O)C1 37102,C1(NC(Cc2c(C)n[nH]c2C)=O)CCCN(C(=O)CNC=O)CC1F 37103,c1(CC(C(N2CCC(C)(NC(CC3CC(OC)C3)=O)C2)=O)C)ccc(F)c(F)c1 37104,CCCCC(C)C(=O)N1CCN(C(=O)CCCOCC(C)C)CC1c1cn[nH]c1 37105,C1(C)(C(c2n(CCSC)nnn2)NCCC(=O)NC(N)=O)CCOCC1 37106,C(C(C)(C)CNC(c1nocc1Br)=O)N(C)C(C1C=CCCC1)=O 37107,C1(C(=O)NCC(C2CC(C)(C)C2)C)C2CN(C(=O)CC(C)(F)F)CC12 37108,C(=O)(C1=CC2C=CC(C1)C2)NC(CC(CC)C)C(=O)N1CCC12CC(O)C2 37109,c1(C2CCCN(C(C(=O)NC(CCCCCC)C)=O)C2)ccccc1[N+](=O)[O-] 37110,c1(CNC(C(C)n2cccn2)=O)ccccc1CN(C)C(C1C(F)(F)C12CC2)=O 37111,C(=O)(C1=CS(=O)CCC1)N1C(CNC(C=Cc2c(C)ccs2)=O)COCC1 37112,c1(OC)nccc(=NC2CCCOC3(CCCOC3)C2)[nH]1 37113,c1(N(CC(=O)NCC(CCCC)NC(=O)CC(F)(F)F)C)ncnc2[nH]cnc12 37114,Cc1ccc2oc(C(=O)NC3CN(C(=O)CCNC(=O)CO)C4CC34)cc2n1 37115,C(=O)(C(=O)C(C)(C)C)NCc1c(NC(CC2(OC)CCOCC2)=O)cccc1 37116,CC(C)CC(C)(CNC(C1(C(C)(F)F)CCC1)=O)NC(c1cnc2n1CCC2)=O 37117,C1(N(C(CC)=O)C)CCCC(NC(=O)C#CC(C)NC(=O)OC(C)(C)C)C1 37118,c1(NC(N)=O)cc(Br)cnc1N1CCCC(Cc2ccc(Cl)cc2)C1 37119,CCC(C)(C(=O)NC(CNC(=O)C=Cc1cccc(F)c1F)C(C)C)C(F)F 37120,C(=O)(C(CC)C(C)O)N(CC(CC1CN(C(C(CC)CC)=O)C1)(C)C)c1nccs1 37121,c1(CC)ccc(Oc2ccc(CNC(=O)CCC3CCC(=O)NC3)cn2)cc1 37122,N1(C(COCc2onc(CC)n2)=O)CCC2CC12C(=O)NCC12CCC(CC1)C2 37123,N1(C(C(N2CCC(C)CC2)=O)=O)C(CNC(=O)C=CC2CCC2)CC2CCCC12 37124,c1(OC(CC)C(=O)NC2CCCN(C(=O)C=CBr)C2)ccccc1F 37125,C1(NC(CCOCC)=O)CCC(CC(=O)NCCC2CCCC2)C1 37126,C(=O)(C(O)P(C)(C)=O)N1CCC(C(C)(C)NC(C(C)n2cncn2)=O)C1 37127,C1(NC(C=CCCC)=O)CCS(=O)(=O)C12CN(C(C1CN(S(N)(=O)=O)C1)=O)C2 37128,c1(C(N2CC(NC(c3cc(CCC)nn3C)=O)C(C)C2)=O)nc(C)c(C)[nH]c1=O 37129,c1(CCC(=O)NCC2C(C(=O)NC3C(CCOC)C3)CC2)nc(C(C)C)no1 37130,C1(c2nnnn2CCCSC)(NC(c2ccnn2C)CC)CN2CCCC2C1 37131,CCC(C(=O)NC1CC1NC(=O)CCc1sccc1Br)c1ccccc1 37132,Cc1cnc(C(=O)NCC2C(C)CCN2C(c2cc(C3CC3)n(C)n2)=O)cc1C 37133,c1(OC)ccc([N+](=O)[O-])cc1C(N1CCC12CN(c1ncccn1)C2)=O 37134,c1(C(=O)NC(CCN(C(C(CC)n2cncn2)=O)C)C)ccccc1C(C)=O 37135,N1(C(C(Br)=C(C)C)=O)CC(C)OC2(CCN(c3ncc([N+](=O)[O-])cc3Br)C2)C1 37136,CCCCC(C(=O)NC1CCN(C(C2CCCCS2)=O)C1C(C)C)N(C)C 37137,N1(C(C(C)SC(F)(F)F)=O)CC(CO)C2(C1)CN(c1ncnc3c1cnn3C)C2 37138,C1(CNC(C2CN(CC)C(=O)C2)=O)C(C)CCCN1C(=O)Cc1cc(C)no1 37139,c1(NCCOCCNC(C2CC3CCCC23)=O)ncc(F)c(-c2ccsc2)n1.O 37140,C1(NC(C2(CC#C)CC=CCC2)=O)CN(C(c2ccco2)=O)CC1S(C)(=O)=O 37141,c1(SCC(N2CC(C(C)NC(=O)CCOC3CCCCC3)C2)=O)n[nH]c(O)n1 37142,Cn1nc(NCC2CC3CC(OC(F)F)C3C2)c(C(F)F)c1Cl 37143,C(=O)(C1=NOC2(CCN(C(c3ccsn3)=O)C2)C1)N1CCN(C)C(=O)C1 37144,Cn1c(C(=O)NC(C)(C)CNC(c2c(F)cccc2Br)=O)cc2c1CCOC2 37145,C(=O)(CCCC#CC)NC1CCN(C(C(C)OCC#C)=O)C1 37146,n1(-c2ccn(CC)n2)nc(C2CCOCC2)nc1-c1cc(C)nn1C 37147,c1(CC)ccc(C(N2CCN(C(=O)C=C3CCC3)CC2CC(F)F)=O)c(O)c1 37148,c1(C(=O)NC2CCCC(NC(C3CC(CC4CC4)C3)=O)C2)cccc2ccsc12 37149,CC(CC(=O)N(C)Cc1ccc(F)c(C(F)(F)F)c1)C(C)(C)C 37150,N1(C(c2cc(C)c(Cl)s2)=O)CCCC(NC(=O)C(c2ccc(F)cc2)(C)O)CC1 37151,C1(C(=O)OC)CC(C(N2CC(OC)C(c3cccc(F)c3)C2)=O)CN(C(C)=O)C1 37152,C1(CC=C)(NC(=O)CC(C)(C)C)CCCN(C(=O)CSc2ccc(C)c(C)c2)C1 37153,CN1CCCC(CN2C(=O)NC(Cc3ccc(F)cc3)C2=O)C1=O 37154,Cn1c(Cl)nc2cc(C(=O)NC3C=CC(C)(C)CC3)ccc12 37155,CCC(C)(C)CC(=O)N1CCCC(CCNC(C2CCC3(CCC3)C2)=O)CC1 37156,C(C1=NOC2CN(C(=O)C=Cc3cncs3)CC12)NC(=O)COC1CCC1 37157,Cn1ncc2c(NCc3cnccc3Cl)[nH]c(=NCC34CCCC3C4(F)F)nc12 37158,C#Cc1cn(C)nc1C(N1CC2CC1CN2C(=O)CCCCN1CCCC1)=O 37159,c1(C(N2CC(CNC(=O)C=Cc3cn[nH]c3)C(O)C2)=O)cc(F)cc(F)c1 37160,C(=O)(CCC(N)CC1CCCCC1)NCc1c(C)noc1 37161,C(=O)(CCC(=O)NCC1(O)CC(C(=O)NC(CC2CCCC2)CO)C1)NCC 37162,C1(NC(C2CCC3(CCC3)OC2)=O)CC2CCCC(C1)N2C(C1CSC1)=O 37163,C1(CC=C)(C(N2CC(C#N)(SC)C2)=O)CCCN1C(C1CC1C1CCC1)=O 37164,C(=O)(CC(CC)CC)NC(CCCC)CNC(c1ccn(CC#N)n1)=O 37165,c1(C(=O)NCC2CC(OC)CN2C(=O)CC(C)F)cc(Cl)c2[nH]c(O)nc2c1 37166,N1(C(=O)C(O)c2ccsc2)CC2CC2(NC(C23CC(F)(C2)C3)=O)C1 37167,c1(C(C(=O)OC(C)C)NC(=O)NCCc2cn(CC)nc2)ccc(F)cc1 37168,c1(OC)c(Br)ccc(F)c1S(=O)(=O)N1CCC(O)(c2ccccc2Cl)CC1 37169,c1(SC)nc(C)cc(=NCC(CC(C)C)NC(=O)CC2OCCCC2(C)C)[nH]1 37170,C12(CC(N3C4(CN(CC(c5cnc[nH]5)=O)C4)CC3)=O)CC3CC(CC(C3)C1)C2 37171,c1(NC2C3(CC(NC(C4(N(C)C)CCC4)=O)C3)C2)ccc(C#N)nn1 37172,C1(C(=O)NC(c2cnn(C)c2)C(=O)NC)C=CCNC1 37173,N1(C(C=CC=CCC)=O)CCC(CCNC(c2cnc(N(C)C)nc2)=O)CC1C 37174,c1(N2CCC(NC(N(CC(C(=O)OC)C)C(C)C)=O)C2=O)c(F)cccc1F 37175,C1(CNC(C2CCCC(O)C2)=O)CC2C(C1)C2(F)F 37176,c1(COC)nc(-c2nc(Cl)cs2)n(-c2nccn2C)n1 37177,n1(CC)ncc(C(N2CCN(C(=O)C(O)C(F)F)CC2)=O)c1C 37178,C1(Cn2cc(C(CC)OC)nn2)CC(COC)CN1C(=O)CC1(C)CCOC1 37179,C1(C(N2C(C(=O)N(C)Cc3cncnc3)(CC)CCC2)=O)C2CC3C(C2=O)C13 37180,CCC(O)C(=O)NC1CC(F)(CNC(c2n[nH]cc2-c2cnn(C)c2)=O)C1 37181,C=CCC(C)(C)C(=O)NCC1CCC(NC(C2CC3CC2C3)=O)CC1 37182,C12(C(N3CCN(C(CCCNC(=O)OCC)=O)C4C3C4)=O)CCC(C)(CC1)OC2 37183,C1(NC(c2c(C)onc2)=O)C2CC1N(C(C1(n3cccn3)CCC1)=O)C2 37184,c1(NC)ccccc1C(=O)NC1CC1NC(c1cnc(Br)s1)=O 37185,C#Cc1cncc(C(=O)NCC(C(C)(C)C)NC(=O)Cc2ccsc2Cl)c1 37186,N1(C(c2c(CC)nnc(C)c2)=O)CC2(COC(CNC(=O)C=NOC)C2)C1 37187,C(C)(CC)(CCNC(=O)C(C)Cc1cnn(C)c1)NC(C(C)=C(CC)C)=O 37188,N1(C(C)C(=O)NCC2CC2NC(=O)COC2CCCC2)C(=O)CCC1=O 37189,c1(OC)nc(C)ccc1C(N1CC(O)CC1CNC(c1sc(F)cc1C)=O)=O 37190,C1(C(N(C2CC(SC)C2)C)=O)CCCCN(C(C2CCOC2(C)C)=O)C1 37191,C1(CNC(C(CCC)N(C)C)=O)CCN(c2ncc(Cl)cn2)CC1C 37192,Cc1sncc1C(=O)N(C(C(=O)NC(c1ccccc1)C)C1CC1)C1CC1 37193,C1(N(CC#C)C(C2CC(C)(C)C2)=O)CCN(C(c2cscc2C#N)=O)CC1 37194,c1(CC(N2CC(C(=O)NCC3CC(=C)C3)(COC)C2)=O)ccc(C)c(F)c1 37195,c1(C(N(CCC)CCNC(=O)C(O)C2CC2)=O)ccc(Br)c([N+](=O)[O-])c1 37196,C1(C=O)OCCCC1(C)C.C1CCCN(N(C)C)C1.CC1CC2N1C2=O 37197,Cc1cc(C(N2CCCC2C2CCN(C(C3CCOC3)=O)CC2)=O)cc(C)c1Cl 37198,c1(C(N2CCCC(C3CC3)C2C)C(=O)NCCOC)cc(OC)c(OC)c(Br)c1 37199,C1(C(=O)NCC2C=CC(NC(c3n(CC)ccc3)=O)C2)CCc2cnc(C)n2C1 37200,S(=O)(=O)(c1cc(Br)ccc1F)N1CCC(c2ccccc2)(C(=O)OC)C1 37201,Cc1nnc(CCC(=O)N(CC(n2cc(-c3ccc(F)cc3)nn2)C)C2CC2)n1C 37202,CC1c2cc(Br)ccc2CCN1CCSc1ccccc1F 37203,c1(CC(=O)NC2CC(F)(CNC(CCC(C)SC)=O)C2)ccc(C)c(F)c1F 37204,C(C)(C)(C(C)NC(=O)CC(C)C1CCCO1)NC(C)=O 37205,C1(CNC(C(C2CN(C(C(C)C#N)=O)C2)O)=O)CCNC(=O)C1 37206,CN1C(=O)OCC1C(=O)NC1CN(C(c2cn(Cc3ccccc3)cn2)=O)C1 37207,C1(NC(COCCCC)=O)CN(C(=O)CC(O)C2CCCC2)C2CCCC12 37208,C12CCCCC1OCCO2.C(=O)(CC(=O)NC)N1CC(=CCC)C1 37209,N1(C(CNC=O)=O)CCC(C2CCN(C(c3c[nH]c4c(Cl)cccc34)=O)C2)C1 37210,CCC(O)C(=O)N1CCCC1C(=O)NC(C)Cc1cn[nH]c1 37211,CC1(C)CCC(O)(C(=O)NC2COCC2n2cc(C(C3CCOC3)C)nn2)CC1 37212,c1(NC)nc(C)ccc1C(=O)N(C)CC1CCCC(NC(=O)Cc2ccsc2)C1 37213,CCC(CN(C)C)CC(=O)NC1CN(C(c2cc(C)nc(O)n2)=O)CC12CC2 37214,C12(NC(C(CC)=CC)=O)CC1CN(C(=O)Cc1sc(C3CC3)nc1C)C2 37215,CC1CN2CCN1C(C(=O)NC(C1CCN(C(=O)Cn3cccn3)C1)C)C2 37216,N1(C(c2cc3ccsc3n2C)C(=O)NCCCOC)CCCC(C2(O)CCC2)C1 37217,Cc1ccnc(C(N2CCC(C(=O)NOCC3CCOC3)(C(C)C)CC2)=O)c1N 37218,CCC(C(=O)OC)C(=O)NC1CN(C(=O)Cc2ccc(OC)cn2)C1 37219,c1(NC(=O)C(=O)N(CC(C)NC(=O)OC(C)(C)C)C)ccc2c(O)nccc2n1 37220,Cc1ccc2ncc(C(=O)NCC3CC3CNC(=O)Cc3cnnn3C)n2c1 37221,C(=O)(C=C1SCC(=O)N1C)NCC(C)N(C(C(C)CC(F)(F)F)=O)C 37222,N1(C(c2nn(C)c(Br)c2C)C(=O)NCCCSC)CCC2(CNC(=O)C2)C1 37223,N1(C(C(n2c(C)ncc2)C)=O)CCC(C(=O)NCCC2(C)CC2)C1C 37224,C(=O)(C1=C(SC)CCCC1)NCC(CC)NC(c1ccc(Br)o1)=O 37225,N1(C(C(c2ccc(N(C)C)cc2)C)=O)CC(NC(=O)CC2CSC2)CC12CCC2 37226,CC1(C)C2CCC1(CC(=O)NC1(CF)CCN(C(=O)CCC3CCCO3)C1)CC2 37227,C#Cc1ccccc1CC(=O)N(C)CCNC(c1cc(C2CC2)on1)=O 37228,C1(NC(CCSCC)=O)CC2(CCN(C(c3cnn(C(C)C)c3Cl)=O)C2)C1 37229,c1(NC2CCCN(C(C(C(C)C)SC)=O)CC2)cccc(F)c1[N+](=O)[O-] 37230,c1(NC2CC(C)C2)nc2cccnc2c(=NCc2nn(C)cc2Br)[nH]1 37231,N1(C(c2occ(C)c2C)=O)CCCC12CCN(C(=O)CC1CSC1)CC2 37232,C1(C(=O)NCCOCC(N)=O)(CC)CCN(C(=O)C(C)=C2CC2)C1 37233,c1(OC2(C)CN(C(C3CCC(C(N)=O)C3)=O)C2)cc(C(=O)NC)ccn1 37234,N#Cc1ccc(C(=O)NCC(CC2CC2)C(=O)NCCc2cncs2)o1 37235,C12(C(N(C(CC)CC)C)=O)CC(NC(=O)CN3CCCC3)(C1)C2 37236,N1(c2ccc(C)cn2)CC2C(C1C(=O)NCCc1ccccc1O)C2(C)C 37237,C1(C(N2C3C(NC(C(CCC)=CCC)=O)C(C3)C2)=O)CCC([N+](=O)[O-])CC1 37238,c1(C(=O)NC2C3CCN(C(c4c(CC)nc[nH]4)=O)C32)c(Br)ccc(OC)c1C 37239,c1(-c2n(CC)cnc2)cc(CN2CCOC(CN)C2)ccc1O 37240,c1(N2CC(C)OCC2)nc(=NCCOc2ccncc2)[nH]c2c1ncn2C 37241,C(c1ccc(C)cc1)=CC(N1C(CC)C(C(=O)N(C(C)CN(C)C(C)=O)C)CC1)=O 37242,c1(CNC(NCc2cc(C)on2)=NCc2cnn(CCF)c2)cc2occc2[nH]1 37243,c1(C(=O)NCC(C)(CC)NC(C=CCN(CC)CC)=O)ccnc2[nH]ncc12 37244,c1(CC)cnccc1C(=O)NCC(C1CCOC1)NC(c1ncc(F)cn1)=O 37245,c1(C(C)C(=O)N(C)C(c2ccc(Cl)cc2)C2CCCC2)ccc2c(c1)OCO2 37246,C1(C(=O)NC(Cn2cc(C(CC)O)nn2)C)CC(C(=O)OC(C)(C)C)=NO1 37247,C1(NC(C(C)=C2CCCC2)=O)CCC2CN(Cc3ccc(C(C)C)cc3)CC2C1 37248,Cc1ncc(CC(N2CCC(NC(=O)C(C)NC=O)C(C)C2)=O)c(O)n1 37249,c1(C(N2CCC(C)(CNC(C3CC(=O)N(O)C3)=O)C2)=O)cc2nc(=O)ccn2[nH]1 37250,N(C1CCCc2cc(OC)ccc21)C(c1n(CC)nnn1)c1c[nH]nc1C 37251,Cn1cc(I)cc1C(N1CCCC2CC12)C(=O)NCc1ccco1 37252,C1(C(=O)NC(CCC)(C)CC)CCCCN(C(=O)CC2CC(OC)C2)C1 37253,C(=O)(C(C)(O)CC(F)(F)F)N1CC(C)C(NC(c2ccc(C(F)(F)F)nc2)=O)C1 37254,C(C)(N=c1nc(NC(C2CCC2)C)c2c([nH]1)c(C)nn2C)c1ncc(C)cc1Br 37255,C(=O)(CCC(C)(C)C)NCC1OCCC(NC(CCN2C(C)CCCC2)=O)C1 37256,c1(C(N2CC3C(CNC(Cc4c(C)noc4)=O)(C3)C2)=O)cnc2c(c1)CCCO2 37257,C1(OC)CC(CCNC(=O)CC(F)F)N(C(=O)CCCOC(C)=O)C1.C(C)(=O)O 37258,CCC(CC(C)C)C(=O)N(CC(O)CNC(c1ccc(Br)c(Cl)c1)=O)C 37259,c1(C(C(=O)OCC2C(OC)CCC2)(C)C)ccc(C(F)(F)F)cn1 37260,C12(C(N3CCCCC(N(C)C(c4nocc4Cl)=O)C3)=O)CC1Cc1c[nH]nc12 37261,c1(C(=O)NCC2C(NC(CC3(C)CCCO3)=O)CC2)nccc(Cl)c1F 37262,N(C1CCCc2n[nH]cc21)C(C(CO)NC(CCC(C)(F)F)=O)=O 37263,CCCCC(CCCC)C(=O)N1CC(NC(=O)C(C)(C)NC(=O)C(F)(F)F)C(C)C1 37264,C=CCN=c1nc(N2CCS(=O)(=O)NC2)c2ccc(OC)cc2[nH]1 37265,Cc1c(C(=O)NCCCCCCNC(=O)CN2CCCC2=O)c(C(F)F)nn1C 37266,N1(C(c2cn(C(C)C)nn2)=O)CCC(C)(C)C1CC(=O)NC(C(F)(F)F)C1CC1 37267,C1(NC(C=CCNC(CC2ON=C(C)C2)=O)=O)CCC(C)(C)C(C)C1 37268,c1(C(=O)NC2C(NC(c3c(CC)nc(C)o3)=O)COCC2)cc(C)nc(C)c1 37269,c1(NC)ncccc1C(N1CCC(F)(C(N2CCC(CN(C)C)C2)=O)C1)=O 37270,C#CC1CN(C(C2CC3(C2)CC(O)C3)=O)CCN1C(c1cc(C2CC2)on1)=O 37271,C1(NC(C(C)n2cncn2)=O)CC1C1CCN(C(c2nnc(S)n2C)=O)CC1 37272,C1(C(N(C2CCC(O)C2)C)=O)CCOC2(CCN(C(=O)OC(C)(C)C)CC2)C1 37273,CC1CN(C(C(=O)NCc2ccco2)c2cnsc2)CC(C2CC2)O1 37274,CCC(N=c1nc(N2CCC3NC(=O)NCC3C2)c2[nH]ccc2[nH]1)c1ncc[nH]1 37275,N#Cc1ccc(CN2CCC(O)(C(=O)Nc3cc(Cl)ccc3I)C2)cn1 37276,N1(C(C(C(=O)N(C)C)(C)C)=O)CC2CCC1C1CN(C(=O)CNS(C)(=O)=O)CC21 37277,c1(C(=O)NCC2C(C)CCN(C(c3c(CC)noc3)=O)C2)ccc2c(c1)OCC2 37278,N1(C(CC2C(C)(C)C2(C)C)=O)CC=C(CC(=O)NC2C=CCCC2CO)CC1 37279,c1(CSC)cccnc1C(=O)NC(C)CC1CN(C(C2COCCOC2)=O)C1 37280,Oc1ccc(Cl)c(F)c1CN1CCC1C1CCCCC1 37281,C(=O)(C1=CCCCO1)N(C1CCCN(C(C(=CC2CCCC2)C)=O)C1)CC1CC1 37282,C1(N(C(=O)NCC2(C(=O)OC3CC(F)(F)C3)CC2)C2CC2)CCC(O)(C(F)(F)F)C1 37283,CC1(C)CC(O)(C(=O)NCC2CCCN(C(c3ccc(C(C)(C)C)s3)=O)C2)C1 37284,Cc1cccc([N+](=O)[O-])c1N1CCCC(C)(CNC(C2(CF)CCC2)=O)C1 37285,c1(C(=O)NCC(C(=O)NCc2onc(COC)n2)C)ccc(C)cc1 37286,N1(C(=O)CC2CCOCC2)CCCCC(C2CN(C(C3CCSC3)=O)C2)C1 37287,CCC(C)C(CC(=O)N(c1cccnc1)Cc1ccccn1)C1CCCO1 37288,N1(C(c2c(C(C)C)onc2)=O)CC2CCC2(CNC(C2CCS(=O)(=O)CC2)=O)C1 37289,N1(C(c2ccc(CC)s2)=O)CC=C(CCNC(C2CC2(F)Cl)=O)CC1 37290,CCCCCC(=O)N(C)CC1(CNC(=O)CC2CC(NC(C)=O)C2(C)C)CC1 37291,C1(CNC(C(C2CC(F)(F)C2)OC)=O)C(C)CCCN1C(=O)C1=CCN(C)C1 37292,C1(C(N2CC(F)(CNC(C3C(C)CC3)=O)C2)=O)CC2C=CC1C21CC1 37293,C1(CCO)(NS(=O)(=O)Cc2ccc(F)c(F)c2)CCS(=O)(=O)CC1 37294,C1(CC(C)(C)C)CN(C(c2scnc2C(F)F)=O)CC1NC(=O)C=CCF 37295,N1(CC)CC(C(=O)NCC(O)CNC(=O)Cc2ncc(C)[nH]2)c2ccccc21 37296,C(=O)(CC1=CCCC1)NC(C(=O)NCc1c(C)ncs1)c1cccs1 37297,C#Cc1ccc(Cl)c(C(N2CCCC2C(C)NC(=O)C=CCn2cncn2)=O)c1 37298,N1(C(CC(C)(C)NC(C2C(C(C)=O)C2(C)C)=O)=O)CCCC2CC1C2(C)C 37299,CCCCCCn1nnnc1C(CC1CCCCC1)NCC1CC1(Cl)Cl 37300,Oc1c(F)ccc(CN=c2ccnc(N3CCC(c4ccncc4)CC3)[nH]2)c1F 37301,Cn1nc2ccccc2c1C(N1CCCN(C(c2ccncn2)=O)C(CO)C1)=O 37302,N1(C(C2C3CN(C)CC32)=O)CCC2CN(C(C3(CO)CC3(F)F)=O)CC2CC1 37303,c1(C(CNCc2ccn(-c3cccc(OC)c3)n2)O)ccc(F)cc1F 37304,C1(CNC(c2cc(CC)nn2C)=O)CC2(CCN(C(=O)C=CC3CC3)C2)CO1 37305,c1(CNC2C(C(=O)OC)COCC2)nc2ccccc2n1CC(F)F 37306,C12CCC(C)(C)CN1C2.c1(CNC(CN2C(C)CCC2C)=O)ccc(C#N)cc1 37307,CCCCC(C)C(=O)NCc1n[nH]cc1C(=O)Nc1conc1C 37308,c1(C(=O)OC)cc(C(=O)NC2CC(NC(=O)C(C(C)O)N(C)C)C2)c(F)cn1 37309,N1(C(C(=O)NCC)=O)CCC2CN(C(c3ncnc(OC)c3F)=O)CCC2C1 37310,C12(CNC(c3n(C(C)C)cnc3)=O)CC(CO1)N(C(C1CCN(C)C(=O)C1)=O)C2 37311,Cc1ccc(C(=O)Nc2n[nH]cc2CNC(=O)CSCCC(C)C)cc1 37312,N1(CC(N)=O)CCCC(N=c2[nH]c(=NCC3CCSC3)c3[nH]ccc3[nH]2)C1 37313,C(=O)(CC(C)CCC(=O)NCC(CC(C)C)NC(=O)C=Cc1cnc(C)s1)OC 37314,C(=O)(CCCC(C)(F)F)NCCN(C(=O)CCOCC1CCC1)CC 37315,CC1(C)CC(NC(c2ccns2)=O)CN(C(=O)COCCO)C1 37316,C(c1cccc([N+](=O)[O-])c1)=CC(=O)NC(CN(C(=O)C(C)(C)C(F)(F)F)C)(C)C 37317,Cc1nc(CO)ncc1C(=O)NC(CNC(=O)CC1CC(F)(F)C1)C(C)C 37318,C12(C(=O)NC(COC)C(=O)OC)CC(C)(CN1C(=O)C(F)C(F)(F)F)C2 37319,c1(C(N2C(C)CC(CNC(c3cc(Cl)ccn3)=O)C2)=O)cc2ccccc2cn1 37320,N1(C(c2cc(COC)no2)=O)CCCOC(CCNC(C2(C)CC=CCC2)=O)C1 37321,C1(CC(=O)NCC(CC(=O)OC)O)CN(C(c2ccccc2O)=O)CC12CC2 37322,c1(C(N2C3CCC2CN(C(C2(N4CCCC4)CC2)=O)C3)=O)c[nH]c2nccc-2c1 37323,C1(C(=O)NC(CC)CN(C)C(c2sccc2CO)=O)CCn2cnnc2C1 37324,CC(C)C(CO)C(=O)N1CCC(NC(=O)Cn2nnc(C3CC3)n2)C1C 37325,C(=O)(C(C)CC(C)C)N1C(CCC(=O)NC(CC#C)CC#C)CCC1 37326,C1(C(=O)OC(C)(C)C)CCCC(NC(C2(SC3CCCOC3)CCC2)=O)C1 37327,C(=O)(C(O)CC(F)(F)F)NCCCN(C(C1(C)CC(F)(F)C1)=O)CC 37328,c1(C(=O)NC(c2cn(CC)nc2)C)cncnc1C1CC1 37329,Cc1nc(CN2CCCC2CC(=O)NCCc2cncn2C)oc1C 37330,C1(NC(=O)C=CC2CCCC2)CC2CCC1(NC(C1(F)CCCCC1)=O)C2 37331,c1(C(=O)NCC(C)N(C(C=CC(=O)OCC)=O)CC)nccc(C(F)F)n1 37332,C1(NC(C=CSC)=O)CC2(C1)CC(CNC(c1cc(C3CC3)nc(O)c1)=O)C2 37333,C1(CC(=O)NCC2(C)CC(NC(=O)CN3CC4CC4C3)C2)CCCCC1(F)F 37334,C1(CNC(C(CCSC)O)=O)CC2COCC2N1C(c1cnn(C(C)C)c1N)=O 37335,C1(NC(C23CCC(OC)C2CC3)=O)CCN(C(C2(C)CCCC2)=O)CC1(C)C 37336,C1(C)(C(=O)NC(C)Cc2ccco2)CCCCC1(C)C 37337,C(CC(O)C(=O)NCCn1cc(CNC(c2ccc(C(C)C)nc2)=O)nn1)SC 37338,C1(CC(=O)NCCN(C(c2cnsc2)=O)CC)CC(C)(C)CCO1 37339,c1(C(=O)NC2(C)CC(NC(c3c(C)ncc(C)c3)=O)C2)ccc2nn(C)cc2c1 37340,c1(C(=O)OC)cc(CN2CCC(C)(C)CC2)nc2ccc(F)cc12 37341,C1(C(N2CC(CNC(CC=C=C)=O)OCCC2)=O)CCOCC12CCCCC2 37342,C1(C)(C(=O)NCC2C(NC(C=CC=CC)=O)COC2)CC2CCC(C1)S2 37343,N1(C(c2ccc(Cl)cc2F)C(=O)NC(CC)(C)C)CC(C)OCC1(C)C 37344,N1(C(C2=CCCCC2C)=O)CCn2nc(CNC(=O)CCn3ccnn3)cc2C1 37345,C1(O)(C(C)NC(=O)Cc2ccn(C(C)C)n2)CCN(C(C2CNC(=O)N2C)=O)C1 37346,c1(C(N(CC(C)NC(c2ccnc(C(C)(F)F)c2)=O)C)=O)cncc(Cl)c1Cl 37347,c1(CCC(=O)NCC(CNC(=O)C(C2CCCCC2)O)OC)ccc(C#N)cc1 37348,c1(C(C(=O)NC2CC(F)(CNC(c3cc(CF)on3)=O)C2)O)cc(F)cc(Cl)c1 37349,C1(NC(c2ccon2)=O)CCCOC1C1CCN(C(=O)CN2CCCC2=O)CC1 37350,N1(C(C(C(=O)OCC)F)=O)CCC(C)(CNC(c2ncn(C(C)(C)C)n2)=O)CC1 37351,N1(C(C=CC=CC)=O)CCCC(CO)(NC(=O)C(C)C2CCOC2)C1 37352,c1(OC)nc(C(=O)NC(C)CCNC(c2coc(Cl)c2)=O)ncc1F 37353,CC1CN(C(c2cc(Cl)ccc2N)=O)CCN1C(=O)COCc1ccccn1 37354,C1(C)(C(N(C(C)CC(F)(F)F)C)=O)CC(O)CN1C(c1ccc(=N)[nH]n1)=O 37355,N1(C(c2cc3cscc3s2)=O)CCC(C2CCCN(c3ncncc3I)C2)CC1 37356,c1(C(=O)NC(C(=O)N2CCC(CC#C)C2)(C)CSC)cc(C)ncc1C 37357,N1(C(C(C)CN(C)C)=O)CCN(C(=O)CSCCN(C)C)C2CCC12.c1ncc[nH]1 37358,C1(C(N(CC(C2CC2)OC)C)=O)CCN(C(c2nc[nH]n2)=O)C1C 37359,Cc1ccc(F)c(C(N2CCC(F)CC2C(=O)NCC2CC(CN=[N+]=[N-])C2)=O)n1 37360,c1(C(=O)NC2CCCC2)occ2c1CCC2.Cc1cc(C(=O)N2CCC2)ccn1 37361,CC1CN(C(C2(C(C)(C)O)CC2)=O)CCC1C(=O)NCCC1CCC(C)(C)C1 37362,C1(CNC(C2(C)CCC2)=O)CN(C(=O)CC2CCCNC2=O)CCC12CCOC2 37363,C1(F)(C(=O)NCc2ccc(C(N)=O)s2)CCCN(C(C2C3COCC23)=O)C1 37364,c1(C2(C(=O)NCCC3CN(C(C(C)NC(C)=O)=O)C3)CC2)ccccc1F 37365,C1(C(=O)NCC2CC(NC(C3CCC(C)(O)CC3)=O)C2)Cc2cc(F)ccc2O1 37366,C1(C(=O)NCCN(C)C2CC2)CC(F)CCN1C(=O)CCC1CC1(C)C 37367,Cc1ccccc1-n1ccc(C(=O)Nc2ccc(C(=O)N(C)C)nc2)n1 37368,CCCCCCC(C)(CC)c1nc(Cc2ccc(C)nc2)no1 37369,N1(C(c2cc(OCC)n[nH]2)=O)CCC(C(=O)NC2(CC(=O)OCC)CC2)CC1 37370,c1(CCC)cnnc(C(=O)NC2CN(C(c3cc[nH]c3C3CC3)=O)CC2OC)c1 37371,c1(OC)cnncc1C(=O)NCC(O)CNC(C1(O)CCCCC1)=O 37372,C1(NC(=O)Cc2cscn2)CN(C(c2csc(O)n2)=O)C2(CCCCCC2)C1 37373,C(C(=O)NCC(C1C(=C)C1C(=O)OC(C)(C)C)=O)(C(C)OC)NC(COC)C(C)C 37374,C1(CNC(c2cc(CCC)nn2C)=O)CCCC2(CN(C(=O)CN(C)C)C2)O1 37375,Cc1nc(C2CCC2)sc1C(=O)NC(C1CCOC1)CNC(C1(F)CC=CC1)=O 37376,[N-]=[N+]=NC1CCC(NC(=O)NCC2CCN(C(=O)CCCCN3CCCC3)C2)C1 37377,CCCCCC(=O)N1CCC(C(=O)N(CCCCN(C)C)C)C1C 37378,C1(C(=O)NC2(C)CC(C(=O)OC)C2)CC(F)(F)CN1C(=O)C(C)COC 37379,c1(SC)ccc(C(=O)NC2(CNC(=O)C#CC3CC3)CCCCC2)cc1 37380,CCCCCC(O)C(=O)N1CC2CC1(CNC(C1CC1CN(C)C)=O)C2 37381,c1(N(C)CC2CCN(CC)C2)nc(N(CCCCOC)C)nc2ccsc12 37382,CCN=C(NCCc1ccsc1Br)NCC(c1ccoc1)O 37383,c1(C(=O)NCCN(C(=O)CC2(O)CCC2)CCOC)scc(C)c1C 37384,C(=O)(C1=CCCCO1)N1CCC(OCCNC(C2CC(Cl)(Cl)C2)=O)C1 37385,CC#CCCC(=O)NC1CCCC(NC(=O)CCOc2ccc(Br)cc2)C1 37386,c1(C(=O)NC2(CC=C)CCN(C(=O)C(CCO)NC)C2)oc2ccccc2c1C 37387,N1(C(CCCC#C)=O)C2CCCC1CC(CNC(c1ccccc1C)=O)C2 37388,c1(CCC(=O)NC2CN(C(C3(OC)CCSC3)=O)C(C)C2)c(C)nn(C)c1C 37389,C1(NC(=O)CC23COC(C2)C3)CCN(C(=O)C(c2ccccc2)F)CC1 37390,c1(C(N2CCCN(C(C3(C)CCC(=O)N3)=O)CC2)=O)cc2c(s1)C(C)(C)CCC2 37391,N1(C(C2=C(C)OCC2)=O)CC(NC(=O)C(C)CS(C)(=O)=O)C2(CCOCC2)C1 37392,C1(NC(C(C#C)(C)C)=O)CC2CCCC2N1C(=O)C(CCSCC)OC 37393,c1(OC(C)(C)C)ccc(F)c(Cl)c1.O1NC(=O)C#CC(=O)NCCC1 37394,C1(C2CCCN(C(c3cc4ccc(F)cc4s3)=O)C2)(NC(CC2C(C)C2)=O)CC1 37395,O=C(C1=CC2(CCOC2)C1)N1CCC(NS(=O)(=O)C2CC2)CC1 37396,N1(CC(=O)NC(C(=O)NC(CCCC)C)C2(C)CC2)CCCNC1=O 37397,N1(C(CSCC)=O)CCC2(CCCC2NC(c2c[nH]c3cccnc23)=O)C1 37398,c1(CCC(=O)NC2(C)CN(C(c3cc4n(n3)CCC4)=O)C2)cccc(Cl)c1Cl 37399,N1(C(C(C)NC(=O)C(F)(F)F)=O)CCC2CN(C(c3ccccc3C#N)=O)CC12 37400,c1(C(N(C(=O)COC(Cn2c(C)csc2=O)=O)C(C)C)=O)cccc2ccccc12 37401,C1(C)(CNC(COC(C)C)=O)CN(C(=O)CC2CCC(C)(C)O2)CCO1 37402,Cc1nc2c([nH]1)CN(C(C1CCCN1C(C1CC1Cl)=O)=O)CC2 37403,C1(C(=O)NCCCN(C(=O)CCN(S(C)(=O)=O)C2CC2)C)CCC(C2CCC2)CC1 37404,C1(C(=O)NC2(CC#C)CCC2)C=CCN1C(=O)Cc1csnn1 37405,c1(CC)cc(F)ccc1C(=O)NCCCN1CCC(NC(=O)CC(=O)OC)C1 37406,S(=O)(=O)(c1ccc(Cl)nc1)N1CC2(CC(C(=O)NCCc3c(C)ncs3)C2)C1 37407,C1(C(F)(F)F)(NC(C(N2C(CNC(C(N)=O)=O)CC2)=O)=O)CC2(CC2)C1 37408,C1(NC(CCn2ncc(C)c2)=O)CC2CC1N(C(=O)CCNC(=O)CO)C2 37409,Cc1cc(=O)oc(C)c1C(=O)NCCCCCCNC(=O)C(C)P(C)(C)=O 37410,c1(-c2ccc(NC(C34CNCC3C4)=O)s2)cccc2ccccc12 37411,c1(C(=O)NCCN(C(C2(C(=O)OC)C=CCC2)=O)C)cc2c(cc1Cl)NC(=O)C2 37412,c1(CNC(c2cc(F)ncc2F)c2n(CCSC)nnn2)nc2ccccc2s1 37413,N1(C(C(CC=C)CC)=O)CCC2(CCC2NC(c2nncn2C2CC2)=O)CC1 37414,N1(C(C(CO)OC)=O)CCCC(CNC(c2cc(Cl)n[nH]2)=O)C1 37415,Cc1cc(F)c(CNc2nccc(=NCC3CC34CCCCC4)[nH]2)c(Br)c1 37416,N1(C(C(C)OCC#C)=O)CCN(C(=O)CC2C(CC)C2(F)F)CC1 37417,C12(C(=O)NC3CC(C)(CNC(C=CC)=O)C3)CCCCC(=O)N1CCC2 37418,N1(C(C(C)SC)=O)CCCN(C(=O)CCc2nc(-c3cccs3)no2)CC1C 37419,c1(C(=O)NCC2(C)CCCN2C(c2c[nH]nc2[N+](=O)[O-])=O)cc(F)c(Cl)cc1F 37420,c1(C(=O)NC2C(CNC(CCC=C=C)=O)CCC2)ccc([N+](=O)[O-])c(N(C)C)c1 37421,Cc1ccc(C(=O)N(C)CCNC(C2CCOC2=O)=O)cc1OC(F)F 37422,C1(C(=O)NC)(CNC)CCCN1C(=O)CC(=O)OC 37423,c1(NC(C)=O)cnccc1C(=O)NC1CC(C)(NC(=O)C=CSc2nc[nH]n2)C1 37424,c1(C(N(CCN(C(C)C)C(C2CC23CC3)=O)C)=O)cccc2cc[nH]c12 37425,Cn1c(CC(=O)NCC(C2CC2)NC(=O)CC2(C(F)(F)F)CC2)nnc1S 37426,C(=O)(C(CCC1CC1)NC(N)=O)N1CC(CCC(C)NC(=O)C(C)C2CC2)C1 37427,N1(C(COC)=O)CC(NC(=O)NCc2cn(C3CCCCC3)nn2)OC(C)(C)C1 37428,N1(C(C(F)=CC)=O)CCCOC(CNC(=O)CC2COC(C)(C)CO2)C1 37429,c1(C(=O)NCC(CO)NC(=O)CC2COCCO2)ccc(-c2nnc(S)o2)cc1 37430,C1(C(N2CCC(C(C(=O)NCC(=O)OCC=C)C)CC2)=O)CCC(C)=C(C)C1 37431,c1(C(=O)NCC(CNC(C2C(C)=CCS2)=O)(C)F)cc(N)c(O)c(F)c1 37432,c1(OC)ccc2ccccc2c1C(=O)Nc1csc(-c2cc(SC)ccc2O)n1 37433,C(CCCC(=O)NCC1(CC)CC(NC(=O)CCc2ccncc2)C1)OCC 37434,CC(C)CC(CNC(=O)CCC1CCCCO1)NC(C1CC(O)CN1C(N)=O)=O 37435,C(CCCCCC(=O)NOCC1CC1)NC(c1c(C)nccc1)=O 37436,O=C1CC(C(N2CCC(OCCF)C2)=O)N(C(=O)C(=C2CCCCC2)F)C1 37437,N1(C(C(n2cc(CCCSC)nn2)C)=O)CC(C(C)=O)C(c2cnn(C)c2C)C1 37438,N1(C(c2ccc(C(N)=O)cn2)=O)CC2(CCN(C(=O)CN3CCCCC3)C2)C1 37439,c1(CN(C2CC2)CC2(C)CCCC2)cncc(C(F)(F)F)c1 37440,C1(NCC2CC(C)(C)CC(C)(C)C2)CCOC2(CCCCC2)C1 37441,c1(CNC(=O)NCC2(C)N=C(C)SC2)cc(C#N)ccc1C 37442,c1(SCC(N2C(C)C(NC(=O)C(O)CCN(C)C)CC2)=O)cc(F)cc(F)c1 37443,Cc1cc(F)cc(Br)c1C(=O)NCC1(c2ccccc2)CCN(C)C1 37444,C(=O)(C(CCOC)OC)NC(C1(CNC(CCOCC#C)=O)CC1)C 37445,N1(C(=O)Cc2cccc(Cl)c2)CC2(CCC(NCc3cnccc3Cl)C2)C1 37446,N1(C(c2cc3ccoc3s2)=O)CC2CN(C(N3CCOCC3)=O)CC2C1 37447,C12C3CC4CN(C1C4C3)C(=O)OCC2.CC1CCC(CO)(NC(C)(C)C)CC1 37448,c1(OC)ccc(CCNCC(O)C(C)c2ccccc2)c(F)c1F 37449,C(=O)(C1=CCCC1(C)C)N1CCCCC(NC(CC2CCN(OC)CC2)=O)C1 37450,C1(C(=O)NCC(C)(C)NC(c2cc(OCC)n[nH]2)=O)C(O)C(=O)N(C)C1C 37451,C1(C)(C(=O)NC(C(C)NC(c2csc(O)n2)=O)CO)Cc2ccccc2NC1=O 37452,c1(OC)ccc2c(c1)CC(C(N1CC3CS(=O)(=O)CC3(NC(C)=O)C1)=O)CO2 37453,c1(CC)ccc(F)c(C(=O)NCC2CCCC(NC(=O)CC3CCOCC3)C2)c1 37454,CC(C)CC(O)C(=O)NCCN(C(=O)CCc1nc(-c2ccco2)no1)C 37455,N1(C(CCCCSC)=O)CCCC(C2CCN(C(=O)C3CC3)CC2)CCC1 37456,Cc1nc(C(N2CC(NC(c3ccnc(O)c3)=O)CC(F)C2)=O)c(C)n1C 37457,N1(C(c2c(Cl)ccc(C)c2)=O)CCC(C2CC2)C1CNC(=O)C(N)=O 37458,C1(NC(C2CC(CNC(CC3(CC(=O)OC)CC3)=O)C2)=O)NC(=O)OC1(C)C 37459,N1(C(Cc2cc(C)on2)=O)CCC(C(=O)NCC2CC(C)CO2)C(C)(C)C1 37460,C1(CCC)(NC(=O)COCCSC)CCN(C(C2CC3CCC(C2)S3)=O)CC1 37461,C1(CC(=O)OC(C)C(=O)NC(c2ccc(Br)cc2)C)CCCCCC1 37462,C1(NC(c2cncc(-c3ccc(F)cc3)c2)=O)CCC(O)(c2ccccc2)CC1 37463,N(C1CCc2cc(Br)ccc21)(C(=O)CCc1ccc2c(c1)OCO2)CCO 37464,CCCCCCCN=c1nc(N2CCC(C(N)=O)(N(C)C)C2)c2c([nH]1)COC2 37465,C12(NC(=O)Nc3cc(CN4CCOCC4)cc(F)c3)CCC(O)(CC1)CC2 37466,N1(C(CN(C(COC)=O)C)=O)CC=CC(NC(C2CC3CCC2C3)=O)C1 37467,Cc1cc(C(N2CCC(CCNC(=O)CCS(C)=O)C2)=O)c(C)s1 37468,N1(C(c2cc(C)cc(N)c2)=O)C2CCC1CC(CNC(c1cn(C)nc1Cl)=O)C2 37469,N(C(=NCCCCl)N1CCC2(CNC(=O)C2)C1)CC(C)(O)c1cccs1 37470,c1(Cn2cc(COCC)nn2)cccc(C(=O)N(CC(C)(C)COC)C)c1 37471,C1(OC)CN(C(c2cn(C)nc2Cl)=O)CC1NC(c1ccccc1O)=O 37472,C1(CNC(C(c2cnn(C)c2)C)=O)CCC2CN(C(=O)CCC(C)(C)C)CC12 37473,CC1CN(C(=O)C(c2ccccc2F)O)CCN1C(=O)COc1ccon1 37474,Cc1ccc(C(C)NC(=O)C(=O)NCCC2COCC2(C)C)cc1C 37475,N1(C(C)=O)CCC(NCC2C(C(C3CCOCC3)O)CCC2)C(C)(C)C1 37476,Cc1ccc(O)c(C(N2CC=CC(NC(c3cc(=O)cc[nH]3)=O)C2)=O)n1 37477,N1(C(C(N2CCSCC2)C)=O)CCCOC(CNC(=O)C=Cc2cccs2)C1 37478,Cc1sc(C(=O)NC2CCCC(NC(=O)CC(C)NC(N)=O)C2)cc1[N+](=O)[O-] 37479,c1(OC)c(C(=O)NC(C2CCCN2C(c2ncccc2O)=O)C)c(C)nn1C 37480,c1(C(N2CC(CCNC(C3(OC)CC3)=O)(OC)C2)=O)cn2ccnc2s1 37481,Cc1cc(C(N2CC=C(CCNC(=O)CC(O)C3CC3)CC2)=O)c2n[nH]cc2c1 37482,C1(CCNC(C(C(=C)Cl)(C)C)=O)CCN(C(c2ccc(F)cc2O)=O)CC1(F)F 37483,C(CC(=O)NC1CN(C(c2cccnn2)=O)C(C)(C)C1)(C(C)C)OCC 37484,CCCCC(O)C(=O)N1CCCC(NC(c2ccc(C(=O)OC)cn2)=O)CC1 37485,N1(C(Cc2ccc(C)o2)=O)CCC(C)N(C(CCC(=O)OC(C)(C)C)=O)CC1 37486,C1(C(N(OC)C)=O)CCOCCN1C(=O)C(n1nccc1C)C 37487,C=CCC(CC)C(=O)N1CCC(n2cccn2)(C(=O)Nc2csc(C#N)c2)CC1 37488,CCC(C)C=CC(=O)NCC(C)=CC(=O)NCCN(C)C(=O)C1CC1 37489,c1(NC(C)=O)c[nH]c(C)c1C(=O)NC1CC(CCNC(=O)CC2CC(F)(F)C2)C1 37490,Cc1ccc2[nH]cc(CC(=O)NCC3C=CCN3C(=O)CC3(CO)CCC3)c2c1 37491,c1(OCC)ccc2ccccc2c1NC(=O)C(=O)NC1CCc2nc(C)nn2C1 37492,CCCCC(COC)(c1nnnn1C1COC1)NCc1cncc(C)c1 37493,N1(C(=O)OC(C)(C)C)CCCC1C(=O)NC1CCCC1NC(C1(C)CC=CC1)=O 37494,C1(NC(=O)C=CC=C(Cl)Cl)COCC1NC(c1n[nH]cc1Cl)=O 37495,N1(C(c2cncc(C)c2)=O)CC(NC(=O)Cn2ncn(C)c2=O)C(F)(F)C1 37496,c1(CCC(N2CCC(CO)(NC(C3CC(O)C3)=O)CC2)=O)cccc([N+](=O)[O-])c1 37497,C(=O)(CC(F)(F)C(F)F)NC1CCC(CNC(CC(C)(C)C)=O)C1 37498,C1(NC(C2CCN(C)C2=O)=O)CC(F)CN(C(c2ccc(OCCF)cc2)=O)C1 37499,N1(Cc2c(C)con2)CCCC(C)(CNC(c2cccnc2OC(F)F)=O)C1 37500,C(C(C(=O)NCCC1CC(=O)N(C)C1)C(C)(C)C)NC(c1cn(CC)nc1)=O 37501,CN1CCN(C(C2(F)CCCN(C(c3cc(N)cc(F)c3)=O)C2)=O)C(C2CC2)C1 37502,c1(-c2occ(CC(N3CC(CNC(C(C4CC4)OC)=O)C3)=O)n2)ccc(Cl)cc1 37503,C1(C(N(C2CCN(c3ncncc3C)C2)CCC)=O)CC(C)(C)CC(C)(C)C1 37504,C(=O)(CCCc1cncs1)NCC(CC)NC(=O)CSc1nc[nH]n1 37505,C1(C)(CNC(CC(C)O)=O)CN(C(=O)C(=O)C(C)(C)C)CCO1 37506,c1(C(=O)NCC2N(C(C(COC)C)=O)CC(O)C2O)cn2c(n1)COCC2 37507,C1(CNC(N)=O)CC(C(F)(F)F)CN1C(=O)CCOC(c1ccccc1)=O 37508,c1(-c2cc(C(N3CC(NC(C(CC)F)=O)C3)=O)on2)c(F)cccc1F 37509,Cc1nccc(=NCC2(CCNC(=O)C(C3CCC(=O)N3)C)CC2)[nH]1 37510,N1(C(C2CC(N(C)CC)C2)=O)CC(C)(C(=O)NCCC(O)C(F)(F)F)CC1(C)C 37511,Cc1noc(C)c1S(=O)(=O)NCC(=O)NC1COCCC1NC(=O)C(C)CF 37512,Cc1sc(C(F)(F)F)nc1C(=O)N(CC(C)(C)NC(=O)CC1C=NN(C)C1=O)C 37513,c1(C(N2CCN(CC(C)NC(c3cc(C)ncc3)=O)CC2)=O)cc(O)nc(C)n1 37514,c1(CNC(C(c2sc(Cl)cc2Cl)N(C(CC(=O)OC)C)C)=O)ccccc1Br 37515,CC(C(=O)N1C2CC(F)C(C2)C1C(N1CCCSCC1)=O)S(=O)c1ccccc1 37516,C(C(C(C)(C)C)NC(=O)C(O)C1CC1)NC(C=C(C)C(F)F)=O 37517,c1(C(C(=O)NCCC)N(C(C)C(F)(F)F)C2CC2)ccc(I)c(C)c1 37518,CCS(=O)(=O)CC(=O)NC(C)(CNC(=O)C(c1c(C)nn(C)c1C)C)C1CC1 37519,CC1(CC(=O)NC2(CNC(c3cc4sccc4[nH]3)=O)CC2)CCS(=O)(=O)N1 37520,O=C(C1CCc2nccn21)NCCC1CN(C(c2ncc3c(F)cccn23)=O)C1 37521,c1(OC)ccc(CN2CCN(C(N)=O)CC2)c(Br)c1O 37522,c1(COCC(=O)NCc2cccc(CNC(=O)C3=CCC3)c2)cc(F)cc(F)c1 37523,c1(N2CCC(CNC(C(c3cccnc3)C)=O)C2(C)C)ccc([N+](=O)[O-])cn1 37524,C(=O)(CCCCCS(N)(=O)=O)NCC1CCCCN(C(c2nc(C)c(C)[nH]2)=O)C1 37525,c1(NC(=O)OC(C(CC)C)C)cc(C#N)ccc1OC(C)(C)C 37526,CCCC(C(=O)NCC1(O)CCCN(C(=O)C2=NOCC2)CC1)S(N)(=O)=O 37527,C(C(C)(C(=O)N(C1(C(N2CCSC(C)C2)=O)CC1)C)OC)OC 37528,c1(CCNC(c2n(C(C)C)nnn2)c2csc(-c3ccsc3)n2)ncccc1F 37529,c1(CC(=O)NCC2C(NC(C(C)OCCC=C)=O)CCC2)cn2ccccc2n1 37530,c1(CCC(=O)NC2C(NC(C)=O)CCCC2)nc2c(O)nc(=O)n(C)c2[nH]1 37531,c1(C(N2CC(NC(c3coc(Cl)n3)=O)C(O)C2)=O)nc2ccccc2o1 37532,N1(C(C(CC)(C)F)=O)CCC2(CC1)CN(C(=O)C=Cc1cscn1)C2C(C)C 37533,N1(C(CC(C)SC)=O)CCOCC(CNC(=O)C(C)Nc2nc(C)cs2)C1 37534,N1(C(c2cc(OC)nn2C)=O)CCC(O)C(N(C(=O)CCC(C)C)C)C1 37535,N1(C(C(CC)(C)OC)=O)C2CCC1CC(NC(C13CCC(N=[N+]=[N-])C1C3)=O)C2 37536,c1(NC(C)C)nccc(=NC2CC2C(N2CCC(OC3CCCCC3)CC2)=O)[nH]1 37537,Cc1c(F)ccc(N)c1C(=O)NCC12CC(NC(=O)COC(F)(F)F)(C1)C(C)O2 37538,C=Cn1nccc1C(=O)NC1CC(C)(NC(C2CCCN(C(=O)OC)C2)=O)C1 37539,C(C(=O)N=S(C)(=O)c1cnn2c1CN(c1ncnc(C(C)(C)C)n1)CC2)=C(C)C 37540,c1(C(=O)NC)cc(C)[nH]c(=NCC2CCC(NC(=O)C(C)(C)CC(F)(F)F)C2)n1 37541,N1(C(c2c(C)ncnc2)=O)CCOCC(C)(CNC(=O)Cc2cnoc2)C1 37542,CN=S(C)(=O)c1ccc(C(=O)NCC2CCCCC2NC(c2cccs2)=O)cc1 37543,CC1CN(C(C2CSCN2C(C2(F)CCCCCC2)=O)=O)CC2(CCC2)O1 37544,Cc1cnc(F)cc1C(N1CC(NC(=O)C(O)CCn2cncn2)C(C)C1)=O 37545,N1(C(C(N2CC(C)C2)C)=O)CCC(C)(C)C(C(=O)NC2CC(C)(C)OC2=O)C1 37546,C1(NC(COCCCCC)=O)CC2C(CNC(=O)CCOC3CCCC3)C2C1 37547,CC1=NOC(C(=O)NCc2cn(CCNC(C34CC(C)C3C4)=O)nn2)C1 37548,c1(CC)c(C(=O)N(CC)CC2CCCN2C(=O)Cc2ccsc2)cnn1CC 37549,C1(NC(CC(C)(C)N(C)C(C2C=CCC2)=O)=O)CCCC(O)CC1 37550,N1(C(C(C=C)O)=O)CC2CCC1CN2C(c1[nH]c(CC)cc1C)=O 37551,N(C1CCCc2cc(F)c(F)cc21)C(=O)NC1(c2ccn(C)n2)CC1 37552,c1(-c2cn(CCCCCNC(c3c(C)cc(F)s3)=O)nn2)cccc(F)c1N 37553,C1(CNC(C(C)=C(C)C)=O)CCC(C)(C)CN1C(c1ccc(NC=O)cc1)=O 37554,C1(C(=O)NCC(=O)NC2N(S(C)(=O)=O)CCCC2)CCC2CCCCC2N1 37555,c1(C(N2C(CNC(C(C)CSc3ccccc3)=O)CC2)=O)ccc(C(C)C)cn1 37556,C1(C(N2CCC(CC)C2C(=O)NCC(F)(CC)CC)=O)OCC2CCCC12 37557,CCC(CCOC)C(=O)N(CCCOCCN(C(=O)C(C)(C)n1cccn1)C)C 37558,CC1(C)CCCC(N2CCCC(C(c3ccc(C#N)cc3)O)C2)C1 37559,CCC(CN(C)C)C(=O)NCC1(OC)CCN(C(=O)Cc2nc(C)sc2C)C1 37560,C1(NC(=O)C(C2CC2)C2CC2)CCC2CCN(C(=O)C(O)c3ccsc3)C1C2 37561,n1(CC(N2C(CN(C(=O)C#CC3CCC3)C)COCC2)=O)ncc(C#N)c1N 37562,N1(C(c2c(C)nc[nH]2)=O)CC(NC(c2cc[nH]c2)=O)CC12CCCCCC2 37563,CCC(C)(CN)C(=O)NCC1(Cc2cc(F)ccc2F)CC(O)C1 37564,c12ncccc1C(=O)Nc1nc(cs1)CC(=O)N2.N1(C(C)C)CCC(Br)C1 37565,C12(C(=O)NCC(CC)(CC)NC(c3cccc(OC)c3)=O)CCCC1C2(F)F 37566,CC1(C)CCCC(C(=O)NCCC2=CCN(C(c3ccc(C#N)[nH]3)=O)CC2)CC1 37567,c1(C(=O)NCC2(CCNC(C3CCCCO3)=O)CC2)cnc(O)c2ncccc12 37568,c1(CNC(=O)NCCC2CCC(C)O2)ncccc1Cl 37569,CCCC(CNC(c1scnc1C)=O)NC(=O)CSS(C)(=O)=O 37570,C(CS(=O)(=O)c1cccs1)NC(=NCC=C)NCCOC(=O)OC(C)(C)C 37571,c1(C(N2C3CC(NC(C(CCC)OC)=O)C3CC2)=O)cccc2c1nnn2C 37572,N1(CCC)CCC(N(C)CC2(COC)CCC2)C1 37573,C(C(C(F)(F)F)N1CCN(C(c2cn(CC)nn2)=O)CC1)NC(CC=CC=C)=O 37574,C=CCC(F)(F)C(=O)NC1CCCC(NC(=O)Cc2ccc(Cl)c(F)c2)CC1 37575,C(CCCCC(=O)N1CC2(NC(c3ccc(C)c(O)n3)=O)CCC1C2)OC 37576,C1(C(=O)OC)C(NC(=O)Cn2cc(Br)cn2)C2(C)CCC(C2)C1(C)C 37577,c1(C(N(C(C)C(=O)NCc2ccoc2)CCC)=O)cc(CC)on1.C1CO1 37578,c1(C(=O)NC2CCC23CN(C(c2cc(F)ccc2F)=O)C3)nccn2ccnc12 37579,CC1(c2cn(CCC(N3CC(F)(F)C3)=O)nn2)CCCO1 37580,c1(C(=O)NC(CNC(C2CC(OC)C2)=O)C)ccccc1C1(C#N)CC1 37581,C=CC1CCN(C(C2(CNC(=O)C(F)F)CC(=C)C2)=O)C1 37582,N1(CC(=O)N(C)CC2N(C(C3(CN(C)C)CC3)=O)CCC2)Cc2ccccc2C1 37583,C1(NC(c2[nH]cc(C)c2)=O)CN(C(c2cncc(Br)c2C)=O)CC12CCC2 37584,C1(OC)CC(CNC(c2cc(C)no2)=O)N(C(c2ccnn2C)=O)C1 37585,c1(NC(C)(C)C)ccc(C(=O)Nc2cccc(C(=O)OC3CCOC3)c2)c(Cl)c1 37586,c1(C(=O)Nc2cccc(CNC(C(C)N(C)C)=O)c2)cc2c(cc1N)CCCC2 37587,c1(CC(N2CCC(CC=C)(NC(=O)C(O)CF)C2)=O)cn2cc(F)ccc2n1 37588,c1(C(N(CCOC)CCNC(c2cn(C)nc2C)=O)=O)ccc(OC)cc1C 37589,C1(C(=O)NCC2OCCCN(C(C3CC(=O)OC3)=O)C2)Cc2cncn2C(=O)N1 37590,C#Cc1ccc(CC(N2CCC(C(N3CC4CCCC3C4)=O)C2CC)=O)cc1 37591,C(=O)(C(C)(CC)CC)N(CC(CNC(C(CCC)=CCC)=O)O)C 37592,C(=O)(C(F)C(F)(F)F)NCCCC(CO)NC(C=CCOCCOC)=O 37593,Fc1cc(Br)cc(NC2CCc3ccsc32)c1Cl 37594,CC1CN(C(c2cc(Br)ccn2)=O)CCN1C(=O)Cc1cnnn1C 37595,C1(F)(CNC(C(C)OCC)=O)CCC(NC(c2ccc(C3(C)CC3)cc2)=O)C1 37596,c1(C(C(=O)N(CC(C)N(C)C(C2(F)CCCCC2)=O)C)C)cncc(F)c1 37597,CC1OC2(CNC(=O)CC3CCCC(C)C3)CC1(NC(c1ccc[nH]1)=O)C2 37598,N1(C(C(C)SCC)=O)CCCC(CNC(C2CCCN2S(C)(=O)=O)=O)C1 37599,c1(OC)ccc(CC(C)(C)C(=O)NCc2ccc(Cl)cc2Cl)cc1OC 37600,CC(C)CC(CNC(c1csc(F)c1)=O)C(=O)NCC(N1CCOCC1)C 37601,N1(C(C(C)NC(=O)OC)=O)CC2(CCCN(C(=O)CC3COCCN3C)C2)C1 37602,C(=O)(CS(=O)(=O)C1CCCC1)NCCC1N(C(C(C)C2=CCCC2)=O)CCSC1 37603,Cc1cc(S(N)(=O)=O)oc1C(=O)NCCN(C(c1c(C)n[nH]c1C)=O)C1CC1 37604,N1(C(c2n(C)ncc2C#N)=O)CCC2(CC1)CCN(C(C1COCCO1)=O)C2 37605,c1(C(=O)NC2CN(C(C(C(=O)OCC)CC)=O)C2)cc(=O)n(C)c2ccccc12 37606,c1(CCC(N2CC(O)(CNC(c3ccc(F)nc3F)=O)C2)=O)c(Cl)cncc1Cl 37607,C1(C(=O)NCC#CCNC(c2cnoc2C2CCOCC2)=O)CC(Cl)(Cl)C1 37608,Cc1cc(C(=O)NCC(C2CC2)N(C)C(c2cnsc2)=O)cc(Cl)c1 37609,C1(CN(C(C=CCN(CC)CC)=O)C)CN(C(=O)Cc2cnc(C)s2)CC12CC2 37610,C(=O)(C1=CC2C=CC1C2)NC(C(=O)N(CC#C)CCOC)(C)CSC 37611,Cc1nccc(C(N2CCN(C(=O)CN(S(C)(=O)=O)C)C(C)C2)=O)c1Cl 37612,c1(OC)nccc(CNC(=O)CC2(NC(C3CC3(F)F)=O)CCCCC2)n1 37613,C1(C(N(C2CCN(C(c3nc(Cl)cs3)=O)C2)CCC)=O)CCC(C)(C)O1 37614,CCC(C(=O)N(C1CCCCN(C(c2c[nH]c(=N)cc2C)=O)C1)CC)C(C)C 37615,C1(C(=O)NCC2(CC)CCCC2)CN(C(C2(C(F)(F)F)CC2)=O)CC1(F)F 37616,c1(CC(=O)NCC(C2CCC2)NC(C(C)OCC=C)=O)ccc(Br)s1 37617,C1(CNC(C2N(CC#C)CCC2)=O)CN(C(C2CSC(C)=N2)=O)CCC12CCC2 37618,c1(CC(=O)NCC(CC=C)NC(c2n[nH]cc2Cl)=O)cnc2ccccc2c1 37619,c1(N2CCC(O)(C(C(=O)NC)(F)F)C2)cc(C)c(F)cc1[N+](=O)[O-] 37620,c1(C(NC(NCC(=C)C)=NCCC2CC2(Cl)Cl)C)ccc(C#N)cc1F 37621,Cc1nc(=N)[nH]c(C)c1C(=O)NCC(C1CC1)NC(C1OC(C)CC1C)=O 37622,C1(C)(C(=O)NCC2(CC(=O)NC3(C(=O)OCC)CC3)CC2)C(C)(C)C1(C)C 37623,CC1=C(C(=O)N2CCN(C)C(CNC(=O)COC3CCOC3)C2)S(=O)(=O)CCO1 37624,C(CN=c1[nH]c(=NC2CC3CCCC3C2)c2ncccc2[nH]1)c1cccc(Br)c1 37625,N1(C(C(CC=C)NC(=O)OC(C)(C)C)=O)CC2CCCC(C1)N2C(C1CC1C)=O 37626,c1(C(N(CC(C)O)CCNC(C(C)=CC)=O)=O)cc(C)sc1Br 37627,C=CC1(C(=O)Nc2ccc(N(C)C)cc2)CCN(C(C2CCN(C)C2)=O)C1 37628,c1(OCC)nccc(C(=O)NC2CCCCN(C(C3CC=C(C)CC3)=O)C2)c1F 37629,c1(CC)cc(OC)ccc1C(N1CCC(CNC(c2c[nH]c(=N)o2)=O)C(C)C1)=O 37630,C(=O)(CCCCCNC(N)=O)N1CC(NC(C2(CC#C)CCOC2)=O)(CO)C1 37631,c1(N(CC(C2CCC2)NC(=O)OC(C)(C)C)C(C2CC(F)C2)=O)ccc(Cl)cc1 37632,c1(C(=O)NCC2OCC(CNC(c3ccc(O)nc3)=O)C2)ccc2nn[nH]c2n1 37633,c1(CNC(C2CCN(C(Cc3cccc(C#C)c3)=O)C2)=O)ccc2ccoc2c1 37634,c1(OC)ccc(CC(=O)N(C2CCCC(NC(C3CC(F)(F)C3)=O)C2)C)c(C)c1 37635,c1(CN(N2CCC(C(CC)C)CC2)C)ccc(Br)c(OC)c1 37636,N1(C(C=CCC)=O)CC2CS(=O)(=O)CC2(NC(c2cc3c(cn2)OCCO3)=O)C1 37637,O=C(CCN=c1[nH]ccs1)NC1CCC(NC(c2cc(Cl)cc(Cl)c2)=O)CC1 37638,C(=O)(C1CCC(N)c2ccccc21)N1C(COC(C)(C)C)CCCC1 37639,C1(C(=O)NC2CC(C(=O)NCc3c(C)occ3)C2)CCC2(CCC2)C1 37640,N1(C(C=CCC)=O)CCN(C(=O)CC2C=NN(C)C2=O)CC1COC 37641,N1(Cc2ccc(NC(=O)C(F)F)s2)CCC12CCN(Cc1cncc(Br)c1)CC2 37642,N1(C(C(C)(O)C2CCC2)=O)CCC2(CCCN2C(c2coc(CO)c2)=O)C1 37643,C1(N(C(=O)CC2(CO)CC2)C)CN(C(C2CCN(CC(C)C)C2)=O)CC12CC2 37644,CC1(C)CCC(C(=O)NCC2=CCCOC2)(NC(=O)C=CCN2CCC2)C1 37645,c1(-c2cc(C(=O)NC(C)CN(C)C(c3ccns3)=O)no2)cccc(F)c1 37646,N1(C(C2(c3cccc(OC)n3)CC2)=O)CC2(CC(NC(=O)C(C)CCCOC)C2)C1 37647,c1(N2CCC(OCCNC(C3CCCOC3)=O)C2)nccc(-n2ccnc2)n1 37648,C(=O)(CS(=O)(=O)C(C)C)N1CCN(C2CCCN(C(C(CCCC)C)=O)C2)CC1 37649,CCCCC(O)C(=O)N1CCC(CC(=O)Nc2nc(F)ccc2Br)C1 37650,N1(C(Cc2ccc(C)nc2)=O)CC2CC(NC(C3CCCC3N(C)C)=O)CC2C1 37651,c1(N2CC(C(C)C)OCC2)[nH]c(=NCC2CC2C2CCOCC2)nc2scnc12 37652,N1(C(c2ccc(OC)nc2)=O)CCC2(COC(CNC(=O)CC(C)C3CC3)C2)C1 37653,C1(C)(C(c2nnnn2CSc2ccccc2)NC2C(C(C)C)C2)CCCC1 37654,N1(C(c2n(C=C)ncc2)=O)CCCC(NC(C2CC3CC3C2)=O)CC1 37655,C#CCCCCCCC(=O)N(CCCCCC(=O)NCc1cn(C)cn1)C 37656,c1(C(C)CC(=O)NCc2ccccc2O)ccc(F)cc1F 37657,c1(CC)cccc(F)c1C(=O)NCCC1CC(NC(=O)CC2(C)CCCC2)C1 37658,Cn1c(C(N2CCC(Cn3cc(C4CC4CO)nn3)C2)=O)cc2cc(Br)cnc12 37659,c1(NC(C(=O)NCC(CC(C)C)C)=O)ccccc1S(C)(=O)=O 37660,N1(C(c2ccc(SC)o2)=O)CCCC(C2CN(C(c3cc(O)cc(O)n3)=O)C2)C1 37661,c1(C(=O)Nc2c(C(=O)NCc3n(C)ccn3)n[nH]c2)ccc(I)c(O)c1 37662,C1(CNC(c2c(C)nccc2)=O)C2CCC1CN(C(=O)C(C)C(C)(F)F)C2 37663,C(CC(F)F)(C(=O)NOCCC(C)O)N(C(=O)CC(C)(C)C(F)F)C 37664,c1(C(=O)NCC2CC(SC)C2)cccc2occc12 37665,N1(C(CNC2C(C)(CO)CC2)=O)CC(O)C2CCCCC2C1 37666,c1(CCNC(CCNC(CN=[N+]=[N-])=O)=O)cc(C(F)(F)F)ccc1C(F)(F)F 37667,c1(C(=O)NCC2CCCC2NC(C2CCOC2)=O)c[nH]c2ccccc12 37668,C1(CNC(C2(CC#C)CCCO2)=O)CCCN(C(c2cc(O)cc(F)c2)=O)CC1 37669,c1(OC)ccc(C(N2CCOC(CCNC(=O)C=COCC=C)C2)=O)cc1OC 37670,c1(C(N(C(C)CNC(c2ccc(Cl)nc2O)=O)C)=O)cc(Cl)c(N)c([N+](=O)[O-])c1 37671,C(=O)(CCCN=c1nccc[nH]1)NCCCN(C(=O)C1=CCCOCC1)C 37672,Cc1cc(F)c(C(=O)NC2(C3CCCN3C(=O)C(O)C(C)(C)C)CC2)cc1F 37673,n1(C(=O)NCC(COC)C(C)C)c(C2CC2)nc2ccccc12 37674,N1(C(=O)Nc2nc(C(C)(C)C)cs2)CCN(C(c2ccc(CC)o2)=O)CC1 37675,O=C1OCc2cc(NC(C3CC34CCN(S(=O)(=O)C(F)(F)F)C4)=O)ccc21 37676,N1(C(c2c(OCC(=C)C)cccc2)=O)CCN(C(=O)CCCCC2CC2)C2CC12 37677,n1(CC)ccnc1C(=O)NCC1CCCC1NC(=O)CCC=C(C)C 37678,c1(C(=O)NC2CC(NC(C(C)C)=O)C2)ccc(NC(c2cnn(C)c2F)=O)cc1 37679,N1(C(C(C(CC)C)O)=O)CCC2(CC1)CN(C(=O)C(=O)NCC1CC1)CC2CO 37680,c1(C(N2CCC(NC(c3c(N)cn(C)n3)=O)CC2)=O)cccc2ccccc12 37681,CS(=O)(=O)c1cc(C(=O)N=c2nc[nH]n2C2CCN(C(=O)OC(C)(C)C)C2)cs1 37682,C1(C(=O)OC)CCC(C(=O)NC(C)(C)C(C)NC(=O)CCCN(C)C(C)=O)CC1 37683,Cc1ccc(C=CC(N2CC(C(C)NC(c3cnn(CC(F)F)c3)=O)C2)=O)cc1 37684,c1(CC)c(C(N2CCC(C)C2C(=O)NCc2cnn(CC)c2C)=O)ccn1C 37685,c1(N2CCC(F)(C(=O)Nc3cc(OC)cc(Br)c3)C2)ncc2ccccc2n1 37686,N(C1CCCn2ccnc21)C(C1(C)CCCN1C(=O)CC1(O)CCOCC1)=O 37687,c1(C(N2CCC(O)(CNC(C(CC)(C)CC)=O)C2)=O)noc(C)c1[N+](=O)[O-] 37688,C12CCC(C1)CNC2=O.c1(C(=O)NCC2CC(CC)C2)cc(C(=O)OC)on1 37689,C(=O)(CCCC(=O)c1ccc(C)cc1)N(CC(CC)O)C1CC1 37690,CCC(O)CC(=O)N1CC(CCNC(=O)C(c2cccc(F)c2)(C)C)C(C)C1 37691,O=C1NCCn2ncc(C(N3CC(CNC(C4CC(C(F)(F)F)C4)=O)C3)=O)c21 37692,C1(NC(C2N(C(c3c(OC)csc3)=O)CCC2C)=O)CC2(C1)CC(C)(C)C2 37693,S(=O)(=O)(c1ccc(N2CCN(C=O)CC2)c(F)c1)N1CCSC(C)C1C 37694,C12(C(=O)NCC3C(CNC(c4c(C)onc4CO)=O)C3)CCCN(CCC1)C2 37695,C1(C(=O)NCCOC2CN(C(c3cc(CC)sn3)=O)C2)(OC)CCC(C)C1 37696,c1(C(N2CC(C)C(CNC(=O)CC3CSC3)CC2)=O)c(Cl)ccc2ccoc12 37697,C(C(CC1CC1)C(=O)NCCC1COCC1O)NC(CSC)=O 37698,Nc1cc(F)cnc1C(=O)NCC(O)CC(=O)NC(CC1CC1)C1CC1 37699,C(CCF)(C(=O)NCCn1cc(CO)nn1)NC(CC=CC=C)=O 37700,c1(OC)cc2c(cc1C(N1CCC(NC(=O)CCc3cccn3C)C1)=O)OCO2 37701,C1(n2cc(C(=O)OC)nn2)CCC(NC(=O)NCCCOC(F)F)CC1 37702,CCC(C)(C)CCCC(=O)NC1CCC2CCN(C(=O)CCCC(C)O)C1C2 37703,c1(C(N2CCC(C)C(NC(=O)C=Cc3ccnn3C)C2)=O)ccc(N=[N+]=[N-])cc1 37704,C1(CC(=O)N(C2CCN(C(C3C(C)C3)=O)CC2)CCO)COC2(CCC2)CO1 37705,c1(C(N2CC(O)(CNC(c3cncc(CO)c3)=O)C2)=O)cnn2ccncc12 37706,c1(C(=O)NCC2(NC(c3cnn(C4CC4)c3)=O)CC2)cnc(S)n1C1CC1 37707,c1(C(=O)NC2C(C(=O)NC(C(=O)OC)CC(C)C)C2)cc(Cl)cc(Cl)c1[N+](=O)[O-] 37708,C(C(C(C)C)NC(C12CC(CO1)C2)=O)NC(C1C(C)C1C)=O 37709,c1(OC)cc(C)c(C(N2CCC3(C=CCO3)C2)=O)c(C)c1 37710,c1(CNC(C2CC(CC)C2)=O)nc(C(=O)N(CCCN=[N+]=[N-])C)c(C)o1 37711,c1(C(C)C)ccc2cc(C(N3CCC(O)(c4cnn[nH]4)C3)=O)ccc2c1 37712,CC(CN=C(NCc1ccnn1C)NCC1C(C)(C)C1(F)F)C(F)(F)F 37713,c1(C2(C(=O)NCCOCCNC(c3cn(CC)nn3)=O)CCC2)ccc(O)cc1 37714,C(=O)(CCC(C)(C)OC)NC(CC(=O)NCc1nnc(CC)o1)C 37715,c1(C(N2CCN(C(C3C(OC)(OC)CC3)=O)C(CF)C2)=O)ccc2occc2c1 37716,N1(C(=O)NCc2cccc(C#N)n2)CCC2(CC1)CC(=O)NC2=O 37717,Cc1cscc1C(=O)NCC1(C(N2CCCC2C)=O)CC=CC1 37718,N1(C(c2c(C)onc2)=O)CCC2C(CCCN2C(=O)CN2CCC(C)(C)C2)C1 37719,c1(N(CC(=O)NCCN(CCOC)C(c2nncn2C2CC2)=O)C)ccccc1 37720,c1(OC)nc(N2CC3CN(C(=O)CCCCCCBr)C3C2)nc2[nH]cnc12 37721,C1(C(N2CC(OCCF)C2)=O)COCCN(C(c2cccc(O)n2)=O)C1 37722,C1(C(=O)NC2C3CN(C(c4nn(C)c(O)c4)=O)CC32)CC2(CCCC2)C1 37723,c1(C(C)=O)ccc(Br)cc1NC(C1CN(C(C2(C)CC=CCC2)=O)C1)=O 37724,C1(NC(C=CCC)=O)CC12CCC(NC(c1ccc(C(F)F)o1)=O)CC2 37725,C1(NC(CN(CCC)C)=O)CCCC(NC(=O)C(C(C)CC)OCC)CC1 37726,C(C(C)(F)CNC(c1ccc(SC)o1)=O)NC(C(C1CC1)SC)=O 37727,C1(NC(=O)NCc2nc(C(C)(F)F)on2)CS(=O)(=O)CC1Cc1cccc(Br)c1 37728,c1(C(=O)NC(c2cnn(C)c2)C)conc1CNC(c1ccnn1CCF)=O 37729,c1(C(=O)NCC(C2CC2)NC(C2CC(C)(F)C2)=O)cc(F)cc2cc[nH]c12 37730,O=C(C#CC1CCCC1)NCCN(C1CCCC1)C(C12CCCC1CC(=O)C2)=O 37731,N1(C(C(C=C)(C)C)=O)CCC2(CC1)CC(CNC(c1cc(CO)[nH]n1)=O)C2 37732,C(C(O)C(C)(C)C)C1(NC(CCC2(O)CC(NC(=O)OC(C)(C)C)C2)=O)CC1 37733,n1(CC(=O)N)cc(C2CC2)nn1.C(C(=O)N(C)CC1(CO)CC1)SCC 37734,O=C(C1CSc2ccccc21)N1CCC(Cc2cccc3ncccc23)CC1 37735,N1(C(C(CC)N2CCCC2)=O)CCN(C(=O)C(C)n2cccn2)CCC1C 37736,C(=O)(C(C)C(C)(C)C)NC1C(CNC(c2cnn(C(C)C)c2C2CC2)=O)C1 37737,N1(C(C(C)CF)=O)CC2CCC1C1CN(C(c3c(Br)nnn3C)=O)CC21 37738,C1(C)(NC(C(C(C)C)NC(c2sccc2C#N)=O)=O)CCC(=O)NC1=O 37739,C1(C(=O)NCC(C2CC2)SC)C2CC2CN1C(c1cnccn1)=O 37740,C1(NC(=O)Nc2c(C)c(Br)ccc2F)CCN(Cc2ccccc2)CC12CCC2 37741,c1(C(N(CCCNC(c2cccc(OCC)c2)=O)C(C)C)=O)cc2[nH]ccc2s1 37742,C(C(=O)NCC1(CO)CNC1(C)C)(C(C(C)C)OC)OC 37743,C1(C(N(C)CC2N(C(Cn3c(C)ccn3)=O)CCCC2)=O)COC2COCC12 37744,C(=O)(CC(C)CC(C)(C)C)N1CC(c2cn(CC(=O)OC)nn2)CN(C)CC1 37745,c1(OC)cccc(C(=O)OC)c1-c1nc(CC(=O)OC)c(C)s1 37746,Cc1cccc2c1OC(C(=O)NCC(F)CNC(=O)CSCCC(F)(F)F)C2 37747,Cn1c(C(=O)NC2CCC2NC(=O)COc2cn[nH]c2)cccc1=O 37748,c1(C(=O)NC(C2(O)CN(C(CC(CC)C)=O)C2)C)cccc2nn(C)nc12 37749,C(=O)(CCCC(C)(C)C)NC(C)CNC(=O)C(C)(O)Cn1cc(Br)cn1 37750,C1(C(=O)NCC(CN(C(=O)C(C)CC(F)F)CC)(C)C)CCOC(=O)CC1 37751,N1(C(C(CCC)NC(C2CCOCC2NC)=O)=O)CCC(C)(C(C)C)CC1 37752,C1(C(N(C(CNC(=O)CC2CC2)C2CC2)C)=O)CCC(O)C1 37753,c1(C(=O)NCCCCCN(C(C(=Cc2ccco2)C)=O)C)nnc(S)n1C 37754,CC1(C)CC(C(=O)NC2CCC(CNC(c3cnn(C4CCOC4)n3)=O)C2)=NO1 37755,C1(C(=O)NCC2CN(CC)C(=O)O2)CC(NC(=O)CC2CC(C)=NO2)C12CCC2 37756,c1(C(N2CC(CCNC(C3(C(F)(F)F)CCO3)=O)C2)=O)cc(C(F)(F)F)ncn1 37757,CS(=O)(=O)c1ccc(F)c(C(=O)NCC2(NC(=O)CC3CC=CC3)CCOC2)c1 37758,CC(C)(CNC(C1C=CCN1C(C1CC(=C2CCC2)C1)=O)=O)CN=[N+]=[N-] 37759,C1(S(N)(=O)=O)(C(N2CC(CC)C(NC(c3[nH]c(O)nc3C)=O)CC2)=O)CCCC1 37760,C=CCC(CC(C)C)C(=O)NC12CC(CNC(=O)C3=CCCS3)(C1)C2 37761,c1(OC(C2C(C(=O)OCC)C2)=O)ccc(N2CCOCC2)cc1 37762,c1(C(N(CC(CNC(c2ccc(CC)cc2)=O)O)C)=O)c(Cl)cccc1[N+](=O)[O-] 37763,C(=O)(C1CSc2ccccc21)NCC(C)(O)CNC(=O)CC(C)(C)C(F)(F)F 37764,C(C)(N=c1[nH]c(=N)c2[nH]cc(Br)c2[nH]1)c1ccc(OCC=C)cc1 37765,N1(C(C(=O)N(C)CC)C)CCOCC(C(=O)NCC(n2nc(C)cc2C)C)C1 37766,c1(C(=O)NCC2CCN(C(c3c(OC)nsc3)=O)C2)ccc2nc(O)n(C)c2c1 37767,CN1CCN(Cc2cccc(N(C)C)c2)CC1c1cc(F)cc(F)c1 37768,C(=O)(C(O)CC[S+](C)C)NCCOC1CCN(C(C(C)(C)OCC)=O)C1 37769,CN=c1nc(C(N2CCCC(CNC(=O)CSc3ccccn3)C2)=O)cc(C)[nH]1 37770,C(=O)(C(C(=O)NCCCCC(=O)N(CC(O)CC)C)OC)OCC 37771,Cc1oc(C(N2CCOC(CNC(C3CC3C3CC3)=O)C2)=O)cc1Br 37772,C(C(CC(F)(F)F)NC(C1CCCN1N=O)=O)NC(Cc1n(C(C)C)cnn1)=O 37773,C1(NC(C(C)(CO)N(C)C)=O)C2CC3C1C3C2C(C1CCN(C)C1)=O.C1(CC)CCC1.C1CC1 37774,CC1CC(NC(=O)C=Cc2ccc(C(F)F)o2)CN1C(c1ccc(C#N)o1)=O 37775,c1(C(N2C(C3CCN(C(c4c(CC)csc4)=O)C3)CCC2)=O)ccc(S(C)=O)cc1 37776,C(=O)(CCC(CF)CF)N1C(C)CC1C(N1CC(c2ccon2)C1)=O 37777,C(c1ccc(F)cc1)=CC(N1CCCN(C(=O)CCC2CCCC2)CC1)=O 37778,c1(C(=O)NC(c2cccc(C)c2)CNC(C(CC#C)C)=O)ccc2c(c1)CC2 37779,C1(CNC(C(C)NC(C)=O)=O)CCN(C(C2CC2C(C)O)=O)CC1C 37780,C1(C(=O)Nc2cccc(CO)n2)CCCC12CCN(Cc1cc(Cl)cnc1Br)C2 37781,Cc1nc(O)[nH]c1C(=O)NC1CC2(C1)CC2NC(c1cc[nH]c1C1CC1)=O 37782,N1(C(CC=C)=O)CC(NC(c2ccc([N+](=O)[O-])cc2)=O)C(C2CC2)C1 37783,C1(COCC)CCN(C(C)C(=O)NCc2ncsc2C(F)(F)F)C1 37784,N1(C(CC2CC(C(C)C)OCC2)=O)CCC(CO)(NC(C2C3CCCC23)=O)CC1 37785,c1(C(C(=O)NCC(C2CC2)NC(Cc2cc(C(C)C)no2)=O)O)ccc(F)cc1 37786,C1(O)(c2cn(C(C)CNC(C3CCSC(C)(C)C3)=O)nn2)CCC(F)(F)CC1 37787,c1(CC(N2CC(NC(c3cccnn3)=O)C2)=O)c[nH]c2cc(Br)ccc12 37788,c1(OCC)nc(C(=O)NC2(C(=O)NC(CN(C)C)CCO)CC2(C)C)co1 37789,c1(C(N(CCCNC(C2CC2C)=O)CCC)=O)cc2n(n1)CCN(C)C2 37790,c1(N2CCC3C(COC)C3C2)nc(N2CCC(F)(CO)C2)c2c(ncn2C)n1 37791,c1(C(C(=O)Nc2ccccc2)N(CC(F)Br)C)cccc(Cl)c1Br 37792,N1(C(c2ccc(=N)[nH]c2)=O)C2CCC1(CNC(C1CCN(C3CC3)CC1)=O)CC2 37793,c1(CN2CC(NC(C3(F)CCCC=C3F)=O)C2)ccc2cc[nH]c2c1 37794,CCCC(C)CCCC(=O)NCCOCCNC(c1cn(CCO)nn1)=O 37795,Cc1ccc(C(N2CC(OCCCCOC(=O)C(C)CF)C2)=O)cc1Br 37796,c1(C(N2C(C3CCN(C(C4CCN(C)C4)=O)C3)CCC2)=O)cc2c(F)cccc2[nH]1 37797,N1(C(C(C)N2CCC2)=O)CCC(CCNC(=O)C(c2ncccc2F)(F)F)CC1 37798,c1(C(N(CC(CC)NC(=O)CCCNC(C)=O)C)=O)nccn2cnnc12 37799,N1(C(c2cc(C)on2)=O)CCCCC1CNC(c1cnc(C(C)(C)CF)o1)=O 37800,C1(NC(c2c(CNC(CCC(C)SC)=O)occ2)=O)CCC(C)(O)CC1 37801,C1(CC(=O)N(CCNC(C(C#C)(C)C)=O)CCOC)COC2(CCC2)CO1 37802,C1(C(N2CC(F)C(F)C2)=O)COC2(CCN(Cc3cncc(Cl)c3)CC2)C1 37803,Cn1nc(-c2ccsc2)cc1C(=O)NCCCN(C(=O)CC1(C)CCC1)C1CC1 37804,c1(SCC(=O)NC23CC(NC(CC4(COC)CCCC4)=O)(C2)C3)cccc(C)c1 37805,CCC(C)(C)CCCC(=O)N1CC(NC(=O)Cn2ccc(C)cc2=O)CC1CO 37806,c1(C(C(=O)NC(CC)C)N(C)C(C2(C)CC2)C)csnc1OC 37807,CC(C)CC(C(=O)N1CC2CC(NC(=O)CCC(C)(C)O)CC1C2)C(N)=O 37808,c1(SC)ncc(C(=O)NCC2(F)CN(C(C3C4COCC34)=O)C2)s1 37809,C(=O)(C1=C2CCCN=CN2NN1)N1C2C(NC(C3CC3C(F)F)=O)CC(C2)C1 37810,C1(S(N)(=O)=O)(C(=O)NCCC(C)N(C)C(c2cn(CCN(C)C)cn2)=O)CCC1 37811,C1(N(CC)CC2CCCN(C(C34CC(C3)C4)=O)C2)C(O)C(=O)N(C)C1C 37812,N1(C(C2CC(F)(F)C2)=O)CCC(CCNC(C2COCCO2)=O)CC1 37813,CCCCCC(CC)C(=O)NCCCOCCC(N1CCN(C(C)C)C(=O)C1)=O 37814,Cc1ccccc1C(C)C(=O)NC1CCC(NC(=O)CCC2CCCCN2C)C1 37815,C1(CNC(CC2C(CNC(C3ON=C(C)C3)=O)C2)=O)CCC=CCC1 37816,N1(C(C(CCC)O)=O)CCCC(O)(CCNC(=O)CSc2nc(C)cc(C)n2)C1 37817,c1(C(C(=O)NC2CC(CNC(c3cn(C)nn3)=O)C2)O)ccc(Cl)cc1 37818,C1(C(C(=O)NCC(C2CC2)OC)C)CCN(C(c2csc(C#N)c2)=O)CC1 37819,C(=O)(CC(C(C)(C)C)NC(=O)C(C)OCCOC(C)=O)NCCOC(C)C 37820,C=CCC(C)(CO)CN=c1[nH]c(N2CCC(C3CCC3)C2)nc2c1SCC2 37821,N1(C(COCCN(C)C)=O)CCC2(CCC(CNC(C3CCCO3)=O)CC2)CC1 37822,C1(O)(CN(C(C(C)OCC2CC2)=O)C)CCN(C(c2nnn3c2CCC3)=O)CC1 37823,C1(CNC(C(c2ccc(F)cc2)C)=O)C(C)CCN1C(c1nnn(C)c1N)=O 37824,C(=O)(CCCC(=O)NCC(C)CNC(c1cc(C)nn1C)=O)NC 37825,Cc1cc(C(=O)NC2CN(C(=O)Cn3nc(Cl)ccc3=O)CC2O)ccc1Cl 37826,c1(C(N2C(CC(=O)Nc3cnn(C)c3C#N)CCC2)=O)cc2ccoc2cn1 37827,CC(C)(CCCNC(=O)Cc1nc[nH]n1)NC(=O)CC1CC(C(F)F)C1 37828,c1(CC(=O)NCCN(C(C2CC2F)=O)C2CC2)c(F)cc(F)cc1F 37829,Cn1cncc(C(=O)NCCCN2CCN(C(=O)CCn3cccn3)CC2)c1=O 37830,CC1(OCCC(=O)NCCCOC2(CCCCO)CC2)CCC1 37831,c1(C(N2CCC(NC(c3cccn(C4CC4)c3=O)=O)C2)=O)ccn2ncccc12 37832,c1(C(C)NC(=O)C(=O)NCCCN(CCC(C)N2CCCC2)C)cnc(Cl)s1 37833,C(C(=O)NCCC1CN(C(C2(C(F)F)CC(F)(F)C2)=O)CCO1)(C(C)C)OC 37834,C1(NC(=O)Cc2nccs2)CCC2CN(C(c3cccc(Cl)c3)=O)CC2C1 37835,C12(CN3CC(C(=O)OCC)C3)CCCC1C2 37836,C(=O)(CC(C)C(F)F)NCCN(C(=O)C(O)(C1CC1)C1CC1)CC 37837,c1(-c2nc(-c3cc(Cl)ncc3)nn2CC2CCOC2)cc(F)cc(F)c1 37838,O=C1CN(C(=O)Cn2cnnn2)C(C(N2CCNC(=O)C2)=O)CN1 37839,N1(CN(C)CC2(C(C)C)CC2)CCN(Cc2cccs2)CC1 37840,C1(C(N2CCCC(N(C(=O)C=CBr)C)C2)=O)CC(F)(F)CCC1(C)C 37841,c1(C(=O)NC2CCCN(c3ccnc(Br)n3)C2)cnn2c1CCCC2 37842,C(=O)(CC(C)(C)c1ccc(F)cc1)NC1C(CNC(C2(CC=C)CC=CC2)=O)C1 37843,c1(OC)ccc(C(=O)NCC2CCN(C(=O)Cc3cc[nH]c3)CC2C)c(Cl)c1 37844,C12(C(N3CCN(C(c4cc(Br)c[nH]4)=O)CC3)=O)C3C4C1C1C2C3C41CO 37845,c1(C(=O)NC2(CNC(C(C)C3CC3)=O)CCC2)n[nH]c2c1COc1ccccc1-2 37846,C1(CC)(NC(=O)CC2CCCC2O)CN(C(C2CCC(C)O2)=O)C1 37847,CC(C)C(CCN(C(=O)C(C)C(F)F)C)NC(=O)C(c1ccc(Cl)cc1)=O 37848,c1(C(C(=O)NCCOC)N(C2CCC(F)(F)C2)C)ccc(F)c(Br)n1 37849,Cc1ccc(C(=O)NCC2CCN2C(C2CCCC2C)=O)c(N)c1C 37850,c12ccnn1C(C)(C)NC2=O.C1(CC2C(C(=O)OC)C2)CCCC1 37851,N1(C(=O)CCC2CCCO2)CC2CCC(C1)N2C(=O)CC1CC2CC2C1 37852,N1(C(c2ccsc2C(F)(F)F)=O)CC2(C1)CN(C(c1ccnc(Cl)c1)=O)CCO2 37853,C1(C(=O)NC(C2CN(C(=O)C=Cc3cnccn3)C2)C)C2CCC1(C)C2(C)C 37854,CC1C2C(CCN2C(=O)C=CC(C)(C)C)CN1C(C12CSCC1C2)=O 37855,C1(CNC(c2c(OC)nn(C)c2)=O)CN(C)CCN1C(c1cc(N)cc(N)c1)=O 37856,c1(C(=O)NC2C(CNC(C(CCCC)O)=O)CC2)cc([N+](=O)[O-])ccc1O 37857,C1(NC(c2cnn[nH]2)=O)CCCC12CCN(C(c1ocnc1C(F)(F)F)=O)CC2 37858,N1(C(CC2CC(=C)C2)=O)CCN(C(=O)C(N2CCOC2=O)C)C(CC(C)(C)C)C1 37859,c1(C(=O)NCC2C(NC(c3c(C)ncc(C)c3)=O)C2)cc(Cl)cc2c1OCC2 37860,CS(=O)(=O)c1ccc(C(N2CCC(NC(=O)CO)C(CO)C2)=O)cc1Br 37861,c1(N(C(c2ccnc(-c3ccc(OC(F)F)nc3)c2)=O)C2CC2)cnc(Br)nc1 37862,C1(C(N2CC(CC(=O)NCc3nccc(OC)c3)OCC2)=O)CC(=O)OC1(C)C 37863,c1(CC(=O)NC2CC3(C(NC(C(CC#C)O)=O)C3)C2)ccc(Cl)cc1F 37864,C(=O)(C(CNC(=O)CN1CC(C)(C)C1)C(C)(C)C)NCCc1c(C)ncs1 37865,CCCCCCn1nnnc1C(C(C)C1CCC1)NCCc1cccnc1 37866,CC1CN(C(=O)CC2NC(=O)NC2=O)CC(C)CN1c1nnc(-c2ccon2)s1 37867,Cc1c(C(=O)NC(C)C(C)NC(c2c(Cl)ccc(Cl)c2O)=O)sc2ccccc12 37868,C(CC(=O)NCc1cccc(NC(C2CN(C(N)=O)C2)=O)c1)(C(C)C)OC 37869,Cc1cc(C(=O)NC23CC(NC(=O)C(C)OCCC(C)C)(C2)C3)cc(C)c1N 37870,C1(CNC(CC(C)(C)SC)=O)CC12CCN(C(=O)Cc1cccnc1Cl)CC2 37871,c1(CC(=O)NC(CC)CNC(C2(Cc3ccoc3)CC2)=O)cccnc1Br 37872,C(=O)(C(F)(CC)C(=O)Oc1ccc(Cl)cc1)N(CC1N(C(C)=O)CCC1)CC 37873,c1(C(N2CCC(C)(NC(C3CCC(C)C3)=O)C2)=O)cc2c(s1)CN(C)CC2 37874,N1(C(CCCC(=C)C)=O)CCCC2(C1)CN(C(=O)CC1CCCCC1O)C2 37875,c1(C(=O)NC(CC=C)CNC(=O)C(CC)N2CCCC2=O)ccc(Cl)cc1F 37876,N1(C(C2CC(C#C)(O)C2)=O)CCN(C(C2(C(O)C(F)(F)F)CCC2)=O)CC1C 37877,c1(C(N2CC(O)(C(C(=O)Nc3ccc(CO)o3)F)C2)=O)ccc([N+](=O)[O-])[nH]1 37878,N1(C(CCC#C)=O)CCC(F)(F)C(C(=O)NC(C)(C)C#CCCC)C1 37879,c1(OC(C)C)ccc(Cl)cc1C(=O)NCCC(C)NC(=O)CC1CC(=O)C1 37880,C1(C(=O)NCc2c(C)nc(CC)o2)CN(C(C2CC(C)(O)C2)=O)CCC1(C)C 37881,N1(C(C2CC(C)OCC2)=O)CCCCC2(CCOCC2)C1 37882,C1(NC(C2(CC=C)CC=CC2)=O)CCC(NC(C2(COC)C=CCC2)=O)CC1 37883,c1(CNC2CCC(C(=O)NCc3ncc(CC)s3)OC2)cc(F)c(F)c(F)c1 37884,c1(C(N2CC(CNC(c3nc(C(C)=O)sc3)=O)C(C)C2)=O)c(C)nc(C)nc1C 37885,CC(CCC(=O)N1CC(n2cc(Cc3cccc(F)c3)nn2)C1)c1ccccc1 37886,C1(CNC(Cc2cc(C(C)C)no2)=O)(CNC(=O)CC2CC23CC3)CC12CCC2 37887,c1(C(=O)NC2CC(NC(C(CC)n3ccnc3)=O)C2)n[nH]c(C)c1Cl 37888,Cc1cc(C(=O)NC2CCCN(C(=O)CC(=O)NCC(F)(F)F)C2C)ccc1F 37889,C1(C(N(CCC)CCO)=O)CN(C(=O)CC(C)C(C)C)CCC1(C)C 37890,C#CCC(C)C(=O)NCC1(O)CC(NC(C2CCCN(C(=O)CC)C2)=O)C1 37891,N1(c2cc(CC(C)C)ncn2)C2CCC1C(C)C(NC(C1CCC1)=O)C2 37892,c1(C(N2CCCN(C(C(=O)NCC)=O)CC2CO)=O)[nH]c2ccc(F)cc2c1C 37893,N1(C(C)=O)CCCCC1CC(=O)N(CCNC(=O)Cc1ccccc1)CC1CC1 37894,N1(C(N(c2ccccc2)C)=O)CCN(C(c2ccc(Cl)nc2)C(=O)NC2CC2)CC1 37895,N1(CC(=O)NCCCC2(NC(C3CC3C(F)(F)F)=O)CC2)CCC(O)CC1 37896,N1(C(CCSCCCC)=O)CCC2(CCC2NC(=O)CNC(C2CCC2)=O)CC1 37897,C1(NC(C(C)C(C)(F)F)=O)CN(C(=O)Cn2ccc(=N)[nH]2)CC2(CCC2)C1 37898,c1(C(N2CCC(C(F)(F)F)C2(C)C)C(=O)NC(CC)C)cc(Cl)c(Cl)c(Cl)c1 37899,C(=O)(C(C)(C)C1CCCN1C(=O)CC1(C)CCOC1)NCCN(CCCF)C 37900,C1(C)(C(=O)NC2CCN(C(Cc3c(C(C)C)con3)=O)C2)CC(C(F)(F)F)=NO1 37901,c1(OC)cc(C(N2CCC(N(C)C(c3c[nH]c(=N)o3)=O)C2)=O)cc([N+](=O)[O-])c1Cl 37902,C1(C)(C(=O)NCC2(OC)CN(C(=O)CC3CSCCO3)C2)CCN(C)C1=O 37903,c1(CC)ccc(C=CC(=O)NCCC(C)N(C(=O)Cn2cncn2)CC)o1 37904,N1(C(c2c(C)cc(Br)cc2F)=O)CCC2CN(C(c3ccc(O)cn3)=O)CC2C1 37905,CCCS(=O)(=O)N=c1cc[nH]c(-c2ccc3nn(C)cc3c2)c1 37906,C1(NC(COCC(C)(C)C)=O)CN(C(C2CCOC(=O)CC2)=O)C(C)(C)C1 37907,c1(C(=O)NC2CC(NCc3c(C)nn(C)c3C)C2)cccc2ccccc12 37908,c1(C(=O)NC2CN(C(CCCCC)=O)CC2C)ccc2c(c1)C(C)CO2 37909,C1(C(N(CC(C)NC(=O)CC2(N(C)C)CCCCC2)C)=O)CC(F)C(=O)N1 37910,C1(C(=O)NC(c2cnn[nH]2)C)CCCN1NC(=O)c1c(Cl)cnn1C 37911,CCCC(C)(O)C(=O)NCC(CC1CC1)C(=O)NCC1CC=CC1 37912,C1(C(=O)NCCC(C)C)C2CCC(C2)C1NC(C1(O)CCCC1)=O 37913,C(CS(=O)(=O)C1CCOCC1)NC(C(N)Cc1ccccc1F)=O 37914,C(c1ccc([N+](=O)[O-])s1)=CC(=O)NCCCCN(C(C1CCC(C)CC1)=O)C 37915,N1(C(CC(C)C(F)F)=O)CCN(C(=O)C(C)(C)N(C)C)CCC1C 37916,c1(C(=O)NC2C3CN(C(c4ccnc(O)c4Br)=O)CC23)ccn2ncnc2c1 37917,C1(C(=O)NCC2C(NC(c3ccc(CCC)[nH]3)=O)C2)CC(=O)N(CC(F)(F)F)C1 37918,N1(C(C(=O)N(C)C)=O)CC2(CCC2NC(=O)CC2CCCC23CC3)C1 37919,C(C)(c1ccccc1)=CC(N1CCC(C)(CC(N2CC(C)(CC)C2)=O)C1)=O 37920,C(=O)(CC(F)(F)F)NC(C)C.C12CCC(C1)C(=O)NC(=O)N1CC(C1)C(=O)N2 37921,c1(CC(=O)N(CCCN(C(=O)Cc2cnsc2)C)C)cccc2c1OC(F)(F)O2 37922,C1(NC(c2ccc3ccnn3c2)=O)CCN(C(c2cccc(F)n2)=O)C12CCC2 37923,C1(C2CCC2)(CNC(C2C(C)OCC2)=O)CCN(C(c2cccc[n+]2[O-])=O)CC1 37924,CC1CC(CCNC(C2(C)CC2)=O)CCN1C(=O)Cn1ncnn1 37925,CCC(CC(=O)N1CCCC(CCNC(C2(C3CC3)CCCO2)=O)C1)C(C)C 37926,N1(C(C(C(C)C)CNC(=O)CNC=O)=O)CCOCC(C)(F)C1 37927,N1(C(c2occ(C)c2C)=O)CCOC(C)(CNC(=O)CSCCC(C)C)C1 37928,C=CCCCCCCCCNC1(c2nnnn2CC(F)F)CCCC1CCCC 37929,c1(CC(=O)N(CC(C)CNC(=O)C=Cc2ncco2)C)cn2cc(F)ccc2n1 37930,C(=O)(C(O)C(F)F)NCCC1CC(NC(COCC(=C)C)=O)C1 37931,c1(C(=O)NCC2CC(CNC(=O)CCc3cc(Cl)no3)C2)sc(F)cc1Cl 37932,C1(CN(C)CC)(CNCCCCOC)CCCC1 37933,c1(C(N(CCN(C(C2CCCC2OC)=O)CC)CC)=O)cccc(C#N)c1C 37934,C1(C(=O)NCC#CC2CC2)(COC)CN(C(=O)C(C2CCCCC2)C)C1 37935,c1(NC(N2CC(NC(c3cc(C)oc3C)=O)C(O)CC2)=O)ccc2c(c1)CCC2 37936,c1(NC)c(C(=O)NCC(CO)NC(=O)Cc2ccc(Cl)nc2)sc2nccnc12 37937,c1(C(=O)NC(C(=O)NCCCC=C)C2(O)CCC2)nccnc1N 37938,c1(NC2CCCC(C(N3CC(C(=O)N)C3)=O)C2)ncnc(C)c1C.CC 37939,CC(C)(C)CC(O)C(=O)NCC1CC(CNC(=O)CNc2nccs2)C1 37940,C(=O)(C1COc2ccccc21)NC(C)CC1CCN(C(=O)C(F)(F)C2CC2)CC1 37941,c1(C(=O)NCCNC(CC2(COC)CC2)=O)nnn(CCC2CCCCO2)c1C 37942,c1(C(N2CC(NC(C(CC)OC)=O)C2)=O)ccc(OC(C)(C)C)cn1 37943,Cc1ccc(C(N2CC=CC(NC(C3(C)CCCS3)=O)C2)=O)c(N)c1F 37944,CC1(CNC(=O)CCN2CCCCC2=O)CCCN(C(=O)Cn2cnnc2)C1 37945,C(C)(CN=c1[nH]nc(C(C)(C)C)o1)Oc1c(OC)c(OC)ncn1 37946,n1(CC)nc(C)c(-c2cscc2C(=O)NC(CO)C(C)C)c1C 37947,C(C)(CC(C)C(F)F)NC(CCN(CC#C)C(c1cnc(CC)o1)=O)=O 37948,c1(CC(=O)N(C2CCCCN(C(=O)C(O)C3CC3)C2)C)ccc2occc2c1 37949,c1(-c2c(C(=O)NCC3C(NC(CC(=O)OCC)=O)C3)c[nH]n2)ccccc1Cl 37950,Cc1nc2sccn2c1C(N1CCC(NC(=O)CC2CC2(Cl)Cl)C12CC2)=O 37951,C1(CCNC(C=CC(=O)OCC)=O)CSCCN1C(=O)CS(=O)(=O)NC 37952,c1(C(=O)NCC(C(C)C)NC(=O)C(C)Cc2cccc(F)c2)ncc[nH]c1=O 37953,c1(NCc2n(CC(=O)OC)ncc2)ccc2c(c1)CCC(C)C2 37954,Cc1cc(C(=O)NC2CC2NC(=O)Cn2cnc(=N)[nH]2)c2c(Br)cccc2n1 37955,C1(CN(C(COCC)=O)C)CCC(CNC(C2CCCN(C(C)=O)C2)=O)CC1.OCC 37956,c1cc2[nH]c(=NCC3CCCO3)[nH]c(=NCc3cncnc3)c2s1 37957,c1(NC(C2CN(C(c3cnc(O)nc3O)=O)CCS2)=O)ccc(I)c(Cl)n1 37958,c1(OC)ccc(CN2CCC(O)C(C(=O)Nc3nc(C4CC4)cs3)C2)c(Cl)c1 37959,N1(C(C(=C(C)C2CC2)F)=O)CCN(C2CCCC2NC(c2cscc2C)=O)CC1 37960,Cc1cc(C(N2CCOCC2C(N2CCOCC(O)C2)=O)=O)cnc1C 37961,c1(CC(C(=O)N(C)CC2(CNC(C3(OC)CC3)=O)CC2)C)c(C)nn(C)c1C 37962,c1(C(=O)NC(CNC(CCc2ccnc(C)n2)=O)C)cn(C2CC2)c(C)cc1=O 37963,CC(C)(C)C(C(=O)NC12CCN(C(=O)COC3CCCC3)CC1C2)NC=O 37964,CC(C)(C)CC(=O)NCC(c1ccc(Cl)cc1)N1CCOCC1 37965,C(C)(C(=O)N1CC(N(C(=O)CCc2cccs2)CCO)C2(CC2)C1)(C(C)C)OC 37966,C(=O)(CCC(C)(C)C)N1CC(NC(CCCCN(C(C)C)C)=O)C(C(F)(F)F)C1 37967,N1(C(C(C)OC)=O)CCC(CCC(=O)NCC(C)CCO)C1 37968,N1(C(CC(COC)C)=O)CC(C)(CNC(=O)CSS(C)(=O)=O)CC1(C)C 37969,CC(C)CCC(O)C(=O)N(CC(C)O)CCNC(=O)Cc1ccc(F)cn1 37970,S(=O)(=O)(c1ccc(NCc2ccncn2)c(Cl)c1)NCC(C)(C)CCCO 37971,c1(C(N(CC(C)(C)O)CC2C(C)OCC2)=O)ccc(=O)n(-c2cccnc2)n1 37972,Cc1ccc(C(=O)N(CCCCCNC(=O)CC2(CO)CCCCC2)C)cc1C 37973,c1(C(=O)NC2CCN(C(C(n3ccc(Br)n3)C)=O)C2)ccc2ccccc2n1 37974,CC(C)C(C)(C)C(=O)NC1CC(NC(c2c[nH]nc2[N+](=O)[O-])=O)C1 37975,c1(N(CCC2CC2)CC)nnc(-c2oc(CO)cc2C)n1CCc1ccccc1 37976,C(=O)(C(CC(C)C)NC(=O)CCCC1(OC)CCC1)N1C(CC(=O)OCC)CC1 37977,c1(C(=O)NCC(CCCC)NC(C2(CC#C)CC=CCC2)=O)cc(F)ccc1N 37978,c1(C(=O)NC2C3(CC(NC(C(CCSC)O)=O)C3)C2)cc(Cl)ccc1O 37979,Cc1cnc(N2CCOCC(C(=O)NC(C)CCO)C2)nc1N1CC(C)OC(C)C1 37980,C(=O)(CC(CN(C)C)CC)NCC(CC)NC(c1ccc(SC)o1)=O 37981,c1(C(C)OC)nc(N2CCC(CNC(C3CCC(N=[N+]=[N-])C3)=O)C2)cc(Cl)n1 37982,C(=O)(CN=c1cc[nH]cc1)N1CC(CC(N2Cc3c[nH]nc3C2)=O)OCC1 37983,N1(c2ncc(C(=O)OC)nc2)CCC2(CCCN(C(=O)CC3(O)CCOC3)C2)C1 37984,CCCCC(CNC(=O)COCCCOC)NC(C1CCS(=O)(=O)C1)=O 37985,CCC(CNC(C12COC(C1)C(NC(=O)C(c1cncnc1)C)C2)=O)CC(C)C 37986,c1(C(N2CCC(O)(CN(C)C(c3cc(F)n[nH]3)=O)C2)=O)[nH]c2ccccc2c1Cl 37987,C=CC1(CO)CCN(C(=O)C(C2(O)CN(C(=O)C(F)C(CC)CC)C2)F)CC1 37988,C12(C(=O)NCC3CN(C(c4cccc(N)c4)=O)C3)CC1Cc1c[nH]nc12 37989,CC1(C)CCOC(C(=O)NCc2ccsc2C(=O)NCC2CCCCC2(C)C)C1 37990,C1(CC)CN(C(c2cc(N)ccn2)=O)CC1NC(=O)CCCOC(C)C 37991,N(C(=NCC1CC1)NC1CCN(CC2CCCC2)C1)Cc1nnc(C)s1 37992,c1(C(N(C)CC)=O)cccc(C(=O)NCC2CN(C(=O)C(C)COC)CCO2)c1 37993,CCCCCC(C)NC(=O)CC1CCC(NC(=O)CCCC2CCCC2)CC1 37994,C(=O)(CC(F)(F)CS(C)(=O)=O)N1CC(CC(C(=O)Nc2n(CC)ccn2)F)C1 37995,c1(C(=O)NC2CCN(C(COCCCCC)=O)C2(C)C)cccc2nccnc12 37996,C(=O)(C1CC(=O)c2ccccc21)N1CCC(C)(NC(C=C(COC)C)=O)C1 37997,c1(C(=O)OC2C3CCCC23)cc2nccn2c(O)n1 37998,N1(C(C=CC)=O)CCN(C(=O)C(C(C)(C)C)N(C)C(=O)OC(C)(C)C)CC1C 37999,c1(SC(C(N2CCC(CN(C(=O)CCSC)CC)CC2)=O)C)ccc(F)cc1F 38000,C1(C(=O)NCCCCNC(Cc2ccc(C)o2)=O)CCn2nncc2C1 38001,c1(C(N2CC3(OCC(NC(CCC#C)=O)C3)C2)=O)cc(C)c2c(c1)CCC2 38002,CN1CCc2c(C(N3CCCC3C(=O)NC3CC3(F)F)=O)cccc21 38003,c1(C(=O)NC23COC(CNC(C4(CCO)CC4)=O)(C2)C3)cn2c(n1)CCC2 38004,N1(C(CSCCN(C)C)=O)CCC(N(C)C)(CNC(C2CCCSC2)=O)C1 38005,c1(CC)ccc(C(=O)NC(C)CNC(=O)CCC2CCOCC2)cc1S(C)(=O)=O 38006,c1(C(=O)NC(C2CCN(C(CSCC)=O)C2)C)cccc(Br)c1 38007,C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CC(C(=O)Nc2ccc(C=C)cc2)C(O)CC1 38008,c1(CC)cc(=NC(=O)C(CNC(C2(CC)CCC2)=O)CC(C)C)[nH]n1C 38009,C(=O)(C(=NOC)c1ccco1)NC1CCCCN(C(C2(CCC)CCC2)=O)C1 38010,N1(C(C(c2ccccc2Br)OC)=O)CCN(C(C2CCCO2)=O)CC12CC2 38011,N1(C(C2SCCS2)=O)CCC(c2cccc(F)c2)C(NC(C23CCCC2C3)=O)C1 38012,c1(CCN(C)CC2CCCN2C(C2(O)CC3CCC2C3)=O)c(F)cccc1F 38013,c1(C(=O)NC2CCCC(C(=O)N(C3CCOCC3)CC)C2)ccc2c(c1)CCCS2 38014,c1(CC(N2CCCCC(NC(C3CCCS3)=O)C2)=O)cnc2cccnn12 38015,c1(C(C)(C)C)nc(C(=O)NCC2CCC(NC)C2)n[nH]1.C(=O)(C(F)=C1CCCC1)N 38016,C1(CNC(N(C)CC2CC2)=O)(NC2CON(C)C2=O)CCCCC1 38017,c1(C(N2CC(NC(CCCC(C)=O)=O)CC2(C)C)=O)cc2ccc(F)cc2[nH]1 38018,N1(C(c2c(CC)nccn2)=O)CCC2CCC12CNC(c1cccc(Cl)c1O)=O 38019,N1(C(c2cccc(C)c2O)=O)CC(N=[N+]=[N-])CC1C(=O)NCC(O)C(N)=O 38020,c1(-c2ccc(-c3n(CC4(CC)CC5(C4)N=N5)ccn3)s2)nccc2ccc(Br)cc12 38021,Cc1cc(Cl)c(CN2CCOC(C(C)O)C2)c(Cl)c1 38022,C(=O)(C(C)(C)CO)NC(c1n(C)ccn1)c1ccccc1 38023,CC(C(=O)NCCC1CCN(C(c2ccc(C(F)F)cc2)=O)C1)C(F)F 38024,C12(NC(C3(CC)CC3)=O)CC1CN(C(C1(CN(C)C)CCCC1)=O)C2 38025,N1(C(CC2CC(OC)C2)=O)CCCC(F)(CNC(=O)C(C)(C)c2ccccc2)C1 38026,c1(CCNC(C2(SC)CCC(C)CC2)=O)cnc2c(Cl)cnn2c1 38027,N1(C(CCCOC)=O)CCC(C)(C)C(C(=O)NC(C)COC(C)C)C1 38028,Cc1cc(C(F)F)n(CC(N2CCCCC2C(C)NC(=O)C(C)(C)CO)=O)n1 38029,N1(C(C(C(=C)Cl)(C)C)=O)CCC2CC(C1)CN(C(=O)C#CC1CC1)C2 38030,c1(C(N2CCC(O)(CNC(c3cc(SC)c(C)o3)=O)C2)=O)ccc(N)c(Cl)c1O 38031,C(CC(C(=O)NC(C)Cn1cncn1)NC(c1ccc(OC)nn1)=O)OC 38032,c1(SCCn2cccn2)ncccc1NC(C(c1cn(C)nc1)=O)=O 38033,CCCCCCCC(=O)N1CC(CC(=O)NCCCCN(C)C)C2(CC2)C1 38034,C1(C(C)C)CCC(C(=O)NC(C2CN(C(c3ccc(C4CC4)o3)=O)C2)C)CC1 38035,c1(C(=O)NC2CCN(C(C3(N(C)C)CC3)=O)CC2O)c[nH]c2cc(C#N)ccc12 38036,C1(NC(C(C)C(F)(F)F)=O)CN(C(c2coc(C(F)F)n2)=O)C2(CCCC2)C1 38037,C1(C)(CC)CC(C(=O)NC(Cc2ccoc2)CO)CCO1 38038,C1(OC)CN(C(=O)Cn2nccn2)C(C)(CNC(c2ncc[nH]c2=O)=O)C1 38039,CC(C)(C)C(C(=O)NC1CCC(Oc2ccccc2)CC1)C1CCC1 38040,C12(C(=O)NCC3(O)CN(C(c4nc(C(C)C)oc4)=O)C3)CC(CO1)C2(C)C 38041,c1(C(=O)NCC2N(C(c3cccn(C)c3=O)=O)CCC2)cnn(C)c1S(C)(=O)=O 38042,N1(C(C(C)(C)OCC)=O)CC23CCCC2(C1)CN(C(c1ccncc1F)=O)C3 38043,c1(C(N2CCC(CCCNC(C3SC4C=CC3C4)=O)CC2)=O)cccnc1CO 38044,c1(CN2CCC(OCC)C(C(=O)O)C2)nc2cc(Br)ccc2n1C 38045,C(C1CC1)(C1CC1)=CC(=O)NCCCN(C(c1cc(SC)oc1C)=O)CC 38046,C1(CNC(C(N2CCSCC2)C)=O)CCCCC1NC(c1ccn(CC#N)n1)=O 38047,c1(C(N2CCC(COC)(NC(c3cnc(O)n3C)=O)C2)=O)c(C)nn(C)c1OC 38048,C=CC1CN(C(C2(N(C)C)CC2)=O)CC1NC(=O)CNC(=O)CCC 38049,N1(C(c2cc(C)no2)=O)CCC(NC(c2cnc(C(C)C)[nH]2)=O)C(C(C)C)C1 38050,C(=O)(CCCCC(F)(F)F)NC(CNC(C=C1CCC(C)C1)=O)C1CCC1 38051,N1(C(C2N(C(C3CC=C(C)CC3)=O)CCC2(C)C)=O)CCC(N=[N+]=[N-])CC1 38052,N1(C(=O)CSc2cn[nH]c2)CCC2CN(C(C3Cc4nccn4C3)=O)C2C1 38053,N1(C(C2CC(C)(CC)C2)=O)CC(F)(F)CC1CNC(c1cc(O)ccc1C)=O 38054,N1(C(CCSCCC)=O)CCC(NC(=O)CCc2cccc(OCC)c2)C2CC12 38055,c1(C(=O)NC2(C)CC(NC(c3cccnc3O)=O)C2)cc2c(s1)CCOC2 38056,N#CC1(CC(=O)NC2CCCCN(C(=O)CN3CCNC(=O)C3)C2)CCOCC1 38057,C12(C(=O)NC(C3CCN(C(C4CCC=CO4)=O)CC3)C)CCC(CC1=O)C2 38058,N1(C(CCCC2C(C)C2)=O)CCCN(C(c2cc(O)nn2C)=O)CC1C 38059,c1(C(=O)NC2CN(CC)C(=O)C2)ccc2c(c1)CCN(C(=O)C(O)CCSC)C2 38060,C12(NC(CCCOC)=O)CCCN(C(c3ccc(=N)[nH]n3)=O)CC1C2 38061,CC1CN(C(C2CCC(C)(C)CC2)=O)CC(C)N(C(=O)CCc2ccc(Cl)s2)C1 38062,c1(CNC2CCC(C(N3CCC(C#N)C3)=O)CC2)c(F)cc(Cl)cc1Cl 38063,c1(N2CCOCC(NC(c3cnn(CC)n3)=O)C2)ncc(Br)cc1C#N 38064,N1(C(C(CC=C)(F)F)=O)CC2CCC(NC(=O)C(C)CC3CCCC3)(C2)C1 38065,Cc1cc(Cl)cc(C(N2CCCCC2CNC(=O)CC2CCCOCC2)=O)c1N 38066,c1(C(=O)NCC(CNC(c2cn(-c3ccccc3)nn2)=O)OC)ncccc1Cl 38067,C1(COC(C2CCC(c3ccccc3)O2)=O)CCCCC1N1CCCC1=O 38068,CCC(C)C(C)CN=c1[nH]c(=NCCCc2nc(C)cs2)c2cc(Cl)ccc2[nH]1 38069,c1(C(=O)NC(C2(O)CCCCC2)C(=O)NCCCCN(C)C)cc([N+](=O)[O-])n[nH]1 38070,C1(Cn2cc(C(CCC)N(C)C)nn2)(Sc2ccc(C(=O)O)cc2)CCC(C)C1 38071,C1(C)(CNCc2nc(C)n(C)c2C)CCCC(C)(C)C1 38072,N1(C(=O)CC2CC3CC3C2)CCN(C(c2cnc(C3CCC3)o2)=O)C(CCO)C1 38073,c1(NC(=O)NC2(CNC(=O)OC(C)(C)C)C(C)CCCC2)cc(C#N)ccc1O 38074,CCCCCC(O)CC(=O)NC1CCC(NC(=O)CCCN(C)C(=O)OCC)C1 38075,CC(C)(C)C(C(=O)N1CC2(CCCO2)C1)NC(c1sccc1CO)=O 38076,C1(NC(C(CC=CC)CC)=O)Cc2ccccc2C1NC(=O)CCc1cn[nH]c1 38077,CCCN(OC)C(=O)CC(CNC(=O)C(CN(C)C)N(C)C)C1CC1 38078,n1(CCC(=O)NCC2C=CC(NC(C3C(C=C)C3)=O)C2)ccccc1=O 38079,C(=O)(C1=CCCC1(C)C)NC(C(C)(C)NC(CC1(C=C)CCC1)=O)C 38080,N1(C(C(F)=CC)=O)CCC2CCN(C(=O)CCC3CCCCN3C)C2C1 38081,N1(C(C2(C)CC2(F)Cl)=O)CC2CCC(C1)N2C(c1cnns1)=O 38082,N1(C(COC(C)(C)C)=O)CCC2(C1)CN(C(=O)CC(F)(F)Br)CCO2 38083,Cc1nc(-c2scnc2C)n(CCOc2ccc(-n3cnnn3)cc2)n1 38084,CCC(CC)(C(=O)NCC(C(C)(C)C)NC(c1ncccn1)=O)C(C)C 38085,C1(CC)CN(C(=O)CO)CCC1NC(=O)C(N1CCCCCC1)c1ccc(F)cc1 38086,c1(C(N(CCC#N)C)=O)cccc(Cc2cnc(C(F)(F)F)s2)c1 38087,c1(NC(C2CCN(C(c3cncc(C#C)c3)=O)C2)C)nc(CC)nc2sccc12 38088,C(=O)(C(O)C(C)(C)C)NC1CC(C)(NC(c2nc(CN3CCOCC3)cs2)=O)C1 38089,C#CCCCCCCCNC(=O)CC(CC)NC(c1cc(C)cc(C)c1)=O 38090,Cc1ccnc(F)c1NC(=O)NCCc1ccc(Br)cc1C(C)C 38091,C12(CN(C)C(c3cn(CCNC(c4ccoc4Cl)=O)nn3)=O)CCC(CC1)C2 38092,O=C(C(CO)c1nn[nH]n1)NCC1CC(Cl)(Cl)C1 38093,N1(C(c2cccc(Br)c2)C)C2CCCC1CN(C(C1(C)CC1)=O)C2 38094,N#Cc1c(C(N2CC(CNC(=O)CCC3CCC(C(N)=O)O3)C2)=O)cccc1F 38095,N1(C(=O)OC(C)(C)C)CCC(C2(O)CN(CCO)C2)CC1.c12ccc(c(Br)c1)NC2 38096,CCCCC(C)CCC(=O)N(CC(C)O)CCNC(c1cccc(C)c1N)=O 38097,c1(C(N2CCC(NC(C3(CC#C)CC3)=O)C(O)C2)=O)ccc2nc(C)[nH]c2c1 38098,Cc1c(C(=O)NC2(C)CCN(C(=O)C(C)O)CC2)sc2[nH]cnc(=O)c12 38099,C1(NC(C2C(OCC)C2C)=O)CCS(=O)(=O)C12CN(C(=O)Cn1cc(CO)nn1)C2 38100,C(C)(C(C(=O)NC1CC(O)C1O)NC(C1OCCC1(C)C)=O)OC 38101,C1(NC(C2(NC(=O)CC3CCOCC3)C(C)(C)C2)=O)CCn2nnnc2C1 38102,N1(C(C2=CC(C)(CC)C2)=O)CCCC2(NC(=O)C(F)=C(C)C3CC3)CCCC12 38103,Cc1nn(C)nc1C(=O)NCC1(CNC(c2cc(Cl)cs2)=O)CCCC1 38104,O=S(=O)(c1cnc(Cl)c(C(F)(F)F)c1)N1CCN(CC2CCOCC2)CC1 38105,c1(NC(C)=O)cccc(-c2cc(NC(=O)Cn3cc(Cl)cn3)ccn2)c1 38106,Cc1[nH]c(CN2CC3CC2C3C(=O)Nc2ccc(Br)c(Cl)c2C)c(C)c1[N+](=O)[O-] 38107,CCC(C)CC(C)C(=O)NCC1CC2CCC1N(C(c1cnnc(Cl)c1)=O)C2 38108,C1(C)(C(=O)NC(CCOC)C(N)=O)CCCN(C(c2ccco2)=O)C1 38109,N1(C(CC=CC=C)=O)CCC(NC(=O)CC(C)COC)C1C 38110,N1(C(c2cc(OC(C)C)ncc2)=O)CCC(C)N(C(=O)C(O)C(C)C)CC1 38111,C1(C(=O)NCCCC(C)NC(c2ccnn2CC2CCC2)=O)CC2CCC1CC2 38112,C(C)(C(=O)NC1CCCC1NC(C)=O)(C1CCOC1)NC(C)=O 38113,C1(CC)(NC(=O)C(C2CCCCC2)F)CN(C(=O)C(C)COC)C1 38114,c1(CC)c(C(N2CC(C(C#N)C#N)C2)=O)cnn1C(C)(C)C 38115,c1(OC)cnc(C(=O)NC2(C)CC(NC(c3n[nH]c(C4CC4)n3)=O)C2)c(F)c1 38116,C1(N(C(=O)Cc2cccs2)CC#C)CCN(C(=O)CC(C)C2CC2)C1 38117,C#Cc1ccc(C(=O)NCC2CCC(C)CN2C(=O)CSS(C)(=O)=O)nc1 38118,C(=O)(CCCCc1cn(C2CCC(C(=O)N(C(C)CO)C3CC3)C2)nn1)OC 38119,C1(C(=O)NC2CN(C(C34CC(C3)C4)=O)CCC2C(F)(F)F)CCc2nc[nH]c2C1 38120,c1(OCC)ncc(C(=O)NCCCNC(=O)Cc2ccc(C(F)F)cc2)cc1Cl 38121,c1(CC(N2C(C)(C(=O)NCC(C)OCC=C)CC2)=O)ccc(C)c(C)c1 38122,C(=O)(CCCC(C)(C)C#N)N1CCC(C(C)NC(C=CCN(C)CC)=O)CC1 38123,c1(C(=O)NC2(C)CC(C(N(CC(C)SC)C)=O)C2)cccc(F)c1F 38124,c1(C(=O)NCCN(C(C(C)C2CCCO2)=O)C2CC2)cnc2sccc2c1 38125,C1(CNC(C2(CC#C)CCCO2)=O)CC(C)CN(C(=O)C(OC)OC)C1 38126,c12cc(no1)CN(C1CCCCC1)C2=O.CC(C)(C)NCCN(CCO)CC#N 38127,C(CCC(CO)NC(=O)CCNC(C)=O)NC(c1c(CC)nc[nH]1)=O 38128,c1(C(N(C(CNC(c2ccc(C)nc2O)=O)C2CC2)C)=O)c(Cl)ccc(F)c1C 38129,C1(NC(c2cc(C)ncc2)=O)CC2CC1CN(C(c1ccnn1C)=O)C2 38130,C(=O)(C(O)CC(C)(C)C)NCCCC(CCC)NC(C1CS(=O)(=O)C1)=O 38131,C(N=c1cc2c(c[nH]1)CCCC2)C1C(CCCOC(=O)OC(C)(C)C)C1 38132,c1(C(=O)NC(C(C)(C)NC(C(CCSC)O)=O)C)ccc(C2=NOC(=O)C2)cc1 38133,CCCCC1N=C2C=CN(N2)C2NCCN(C1=O)CC2 38134,c1(C(N2CC3CN(Cc4c(OC)nccc4)C3C2)=O)cc(C)c(Cl)cc1Cl 38135,C(=O)(C1CCCc2n[nH]cc21)NCC1(NC(=O)Cn2cccc2)CC(OC)C1 38136,c1(C(N2CCCC(N(C)C(c3cncs3)=O)CC2)=O)cc2cccc(F)c2s1 38137,c1(OCC=CC)cccc(CC(=O)NC2CCCN(C(=O)CC34CC(C3)C4)C2)c1 38138,C1(NC(c2cc(-c3cccnc3)no2)=O)CC(F)CN(C(C2CCCSC2)=O)C1 38139,C=CCCCC(C)(C)C(=O)N1CC(CC(C)(C)CNC(=O)COC2CCCOC2)C1 38140,CS(=O)(=O)c1cccnc1C(=O)NCC1CCC2C(C1)C2(F)F 38141,N1(C(C)=O)CCC2CN(C(=O)C(C)(C)c3cscc3Cl)CCC2C1 38142,c1(NC(C2C3(CCN(C(CC#C)=O)C3)C2)=O)nc2ccc(Cl)cc2[nH]1 38143,N1(C(C2(C)N(C(C)=O)CCC2)=O)CCN(C(c2cc(C)ncn2)=O)C2(CCC2)C1 38144,c1(C(C)(C)C(=O)NCCNC(=O)CC2CC2C2CC2)ccc(Cl)nc1 38145,Cc1cnnc(C(=O)NCC2(O)CN(C(c3ccc(C(C)C)cn3)=O)C2)c1 38146,Cn1nc2c(c1NCCOc1cc(C#N)ccc1C(=O)O)CCC2 38147,C1(NC(NCCOC)=N)(CO)CC2(CC(F)C2)C1 38148,CCCCC(F)C(=O)N1CCC1C(N1CCC(OC)C(F)C1)=O 38149,Cc1ccnc2c(C(=O)NC(C)CCN(C)C(C34CC(C)(CCO3)C4)=O)cnn12 38150,c1(OC)ccc2cc(C(=O)NC3CCCN(C(=O)C(C)=C(C)C)C3)sc2c1F 38151,c1(C(N(C2CCN(C(C3COCCO3)=O)CC2)CC)=O)cccnc1N 38152,c1(N2CCC(NC)CC2)ncnc(NCCC2CC(O)C2)c1C 38153,c1(CNC(=O)NCC(c2cccc(C)n2)CC)c(C)cc(C(=O)O)cc1C 38154,C(=O)(C1=NN2CCC(C)N=C2N1)N(C(C)CNC(=O)CCC1CC1)CC 38155,C1(C(=O)NCCC(C)(C)NC(C2COC(=O)O2)=O)CC2(CCCC2)CO1 38156,C1(C(=O)NC(c2cc(OC)c(F)cc2)C)CC2OC(C)CC2N1 38157,C(CC(=O)N(CC)CC)(C(C)C)SC.n12nc(-c3ccc(F)cc3)nc1CCC2 38158,C1(NC(CNC2CC(C#N)C2)=O)CCn2nccc2C1 38159,N1(C(c2occ(C(=O)OC)c2)=O)CC2CC(NC(C3(OC)CC3)=O)C1C2 38160,N1(C(C2=NOC(CNC(c3ccc(C#N)cn3)=O)C2)=O)CCc2cncnc2C1 38161,C1(NC(C(C2CN(C(COCCN(C)C)=O)C2)O)=O)CCN(C)CC1(C)C 38162,Cc1nn(C)cc1CCNC(C1CN(C(=O)CC2(O)CCCC2)CC1C)=O 38163,N1(C(C(=Cc2ccc(C)cc2)C)=O)CC2(CC2)CC1CNC(=O)C1=CCCSC1 38164,C1(CCC)(NC(c2csnc2Cl)=O)CCN(C(c2cccc(O)n2)=O)CC1 38165,c1(-c2sc(C(N3CC(NC(C=C(C)C4CC4)=O)C3)=O)c(C)n2)c(C)nn(C)c1C 38166,c1(C(=O)NC)ccc(-c2nc(-c3cnn(C)c3)nn2-c2ccnc(O)c2)cc1 38167,C1(C(N(CC(C)O)CCNC(=O)C(C2CC2)C2CC2)=O)CCc2nn[nH]c2C1 38168,c1(C(=O)NCC(CNC(CCN(C(CCC)C)C)=O)F)cc(O)cc(Cl)c1 38169,C1(C(=O)NCCN(C(C2(NC(=O)NCC)CCCC2)=O)C)COCCN1C 38170,C1(OC)(OC)COC(C(=O)NOc2ncccc2Br)C1.C1CC1 38171,Cc1ccc(C(C)NC(C2CC=CCN2C(c2cnn(C)c2Cl)=O)=O)cc1 38172,c1(CN2C(CC)CN(C(c3c(Cl)ccnc3Cl)=O)CC2)ccc2nc(O)[nH]c2c1 38173,C1(C)(C(=O)NCC=CCNC(Cc2c(C)noc2Cl)=O)CCCCC1C 38174,C(C(=O)NCC1(F)CC1)(C1CN(C(=O)CSC(C)(C)C)C1)OC 38175,c1(C(=O)NC2CCCC(N(C(CCC(=O)NC)=O)C)C2)oc2ccccc2c1C 38176,c1(NC(=O)Nc2ccc(CC(=O)NC)cc2)c(Br)cc(F)c(F)c1F 38177,CC(N=c1[nH]c(=NCCOCC2CCOCC2)[nH]c2c1COC2)c1ccn(C)n1 38178,CC1=NS(=O)(=O)NC=C1C(=O)NC1CC(CCNC(C2(S(N)(=O)=O)CCC2)=O)C1 38179,C1(NC(c2c(C)noc2)=O)CC2CCC(C1C)N2c1ncccn1 38180,Cc1ccc2c(c1)CC(C(N1CC=CC(NC(=O)C(C)(Cl)Cl)C1)=O)S2(=O)=O 38181,C(=O)(CCCC(C)NC(=O)C(C1CCCCC1)F)NC(C(=O)OC)CO 38182,c1(C(=O)NCC2C3CN(C(C(C)n4cccc4)=O)C2C3)cc([N+](=O)[O-])ccc1Cl 38183,Cc1cncc(C)c1C(N1CC2(CO)CC1(C(=O)NC(CC(C)C)C(N)=O)C2)=O 38184,c1(C(=O)NCC2N(C(c3c(C)cncn3)=O)CC(O)C2)ccnc2ccccc12 38185,Cc1ccc(Br)c(CC(=O)NC2CCC23CN(C(=O)C=CCO)C3)c1 38186,N(C1CCc2sc(Br)cc21)C(=O)OC(C)(C)C.c12cccc(c1)CNC(=O)N2 38187,C1(CC)CCCCC1N(C)C(c1cncc(C(C)C)c1)=O.C12(CCC1)C(=O)NC2 38188,C1(CC(=O)NCCCCC2C(C)C2)CCCN(C(c2nonc2N)=O)C1 38189,C1(C(=O)NC(C)(C)CC(=O)NC2CCS(=O)(=O)C2)CC2(CCC2O)C1 38190,C1(O)(CNC(CC(=O)OC)=O)CCN(C(=O)C(C)Sc2ccccn2)C1 38191,C1(NC(C2(C#N)CCC2)=O)CN(C(C2CC(=O)CCO2)=O)CC(F)(F)C1 38192,C1(CNC(c2ccccc2)=O)CC2CN(C(C3(c4cccnc4)CC3)=O)CC12 38193,S(=O)(=O)(c1cnn2c1OCCC2)NC(Cc1cc(C)[nH]n1)=O 38194,CCC(CS(C)(=O)=O)NC(C1CC(NC(=O)OC(C)(C)C)C1)=O 38195,N1(C(C(c2ccc(Cl)cc2)C)=O)CC(C)(C)CC1CNC(C1CC1F)=O 38196,N1(C(Cc2cnc(C)o2)=O)CC2CCN(C(c3ccc4cnoc4c3)=O)CC2C1 38197,C1(C(N(C(C)CCNC(C23CC(C#N)(C2)C3)=O)C)=O)CC(=O)C12CCC2 38198,N1(C(C(C)Cc2ccncc2)=O)C(C(=O)N(C2COC2)C)CC2CCCCC12 38199,CC(C)(C)CCC(F)C(=O)N1CCCC(F)(CNC(=O)CCn2ccnc2)C1 38200,C1(CC(=O)NC(CCC)c2nn[nH]n2)CCCC1NC(C1(CO)CCOC1)=O 38201,C12(NC(C3N(C)CCOC3)=O)CCCC1CN(C(c1cc[nH]n1)=O)C2 38202,C1(NC(=O)NCCC(CC)C)CCCN(C(=O)OC(C)(C)C)C1c1cncn1C 38203,C1(C(N2CC3CC(C2)O3)=O)CC2CC2N1C(C1CCNC(=O)C1)=O 38204,C1(CN(C(c2c(CC)cc[nH]2)=O)C)CCC(NC(C2CC=CCC2C)=O)CC1 38205,N1(S(CCC)(=O)=O)CCCC(C(N2CCC(NC(=O)C(C)(CC)OC)CC2)=O)C1 38206,c1(C(=O)NC2CC(CNC(c3cc(F)c[nH]3)=O)C2)cnc2ccccn12 38207,c1(C(=O)NC2CC(CNC(CCc3cnn(C)n3)=O)C2)cccc(=O)o1 38208,c1(C(=O)OCC)nnn(C)c1C(=O)OCCn1cc(C(C2CCOC2)OC)nn1 38209,C1(C(=O)NC2(CF)CN(C(=O)CC3C=CCC3)C2)CC2CC(=O)C1C2 38210,C(=O)(C(CO)NC(=O)C=CC1CC1)NCC(C)(O)C1CC1 38211,c1(COC)cc(C(=O)NC(C(=O)NCC23CCCC2C3)c2cccs2)n[nH]1 38212,c1(C(=O)NCC(C)NC(=O)CC2CC=CCN2C)ccc2c(c1)CCC(C)(C)O2 38213,C1(C(N2CCC(CNC(c3c(CC)nns3)=O)CC2)=O)(OC)CCOCC1 38214,CCCCC(CC)CC(=O)N(CC(C)(C)C(=O)NCCS(=O)CC)C 38215,Cc1cn2c(n1)C(C(=O)NC13CCC1CN(C(c1cc(=O)n(C)o1)=O)C3)CCC2 38216,Cn1nc(C(=O)NC(C)(CNC(C2CC(CF)C2)=O)CO)cc1Cl 38217,c1(C(=O)NC2CC3(CN(C(CCC4C(C)C4)=O)C3)C2)ccc2c(n1)OCC(=O)N2 38218,N1(CC(CCC)OC)CCCC(c2nn[nH]n2)(C(C)C)C1 38219,c1(CC(N2CC(C)C(NC(=O)Cc3nc[nH]n3)CC2)=O)c(F)ccc(Br)c1F 38220,N1(C(c2snc(C)c2N)=O)CCCC(CC(=O)N(CC(C)(O)C2CC2)C)CC1 38221,C(=O)(CCCN=[N+]=[N-])N(CCOCCNC(C1(CC=C)COC1)=O)C 38222,C1(CNC(c2cc(C)oc2)=O)CN(C(=O)CSC(C)(C)C)CCC1C 38223,c1(CSC)cccc(C(=O)N(CC(O)CNC(C2CC(CF)C2)=O)C)c1 38224,c1(C(N(CCC2CCN(C(CC(C)F)=O)CC2)C)=O)ccn2cncc2c1 38225,C1(F)(CNC(CN(C)C(N)=O)=O)CCCN(C(=O)C(F)Cc2ccccc2)CC1 38226,CC(C)(C#N)CCC(=O)N1CCC(NC(=O)CSc2nc[nH]n2)C(F)C1 38227,CC1(C)CCCN(C(c2ccc(N)c(F)c2)=O)C1CNC(=O)C#CC1CCC1 38228,C1(NC(c2n(CC)ncc2Br)=O)CCCN(C(=O)CC2(OC)CCC2)CC1 38229,Cn1cc(C#CCNC(C2CC(C)(C)CCN2C(=O)CP(C)(C)=O)=O)cn1 38230,CC1CCCCC1C(=O)NCC1(O)CN(c2nccc(C(F)F)n2)C1 38231,c1(CNC(=O)COCCCF)ccc2c(c1)CN(C(c1cc(CO)ccn1)=O)C2 38232,C1(NC(C(CC=CC)C)=O)CCCOC12CCN(C(=O)Cc1cc(C)on1)CC2 38233,C1(C(=O)NCCCC2CCOC2)(COC)COc2ccccc2C1 38234,c1(CNc2c(C(=O)OC)cc(C)c(C)c2)ccc2c(c1)C(CCOC)C(=O)N2 38235,c1(N(CCCOCCNC(c2cnn(C(C)C)c2F)=O)C)ncccc1C#N 38236,CC1CN(C(=O)CCSc2ccccn2)CCC1CNC(=O)C=Cc1cc[nH]c1 38237,c1(-c2n(C(C)C3CC3)nc(Cn3cncn3)n2)cc2ccncc2s1 38238,c1(N(C(CN2CCCC(COC)C2)=O)CC2CC2)cc(S(N)(=O)=O)cnc1C 38239,C1(C(=O)NOCCO)(CC=C)CCCN1C(C1CCC(F)CC1)=O 38240,c1(C(N(CCC(C(C)C)NC(=O)CS(C)(=O)=O)C)=O)ccc2c(n1)CCO2 38241,CCC(CC)CC(F)C(=O)N1CCC2CCCC12C(=O)NC(C)C1CC1 38242,c1(C(=O)NCCCN(CCCNC(C=CCOC)=O)C)c(NC)ccnc1F 38243,N1(C(C(C=C)CC)=O)CCOC2(CCN(C(=O)Cc3ccnn3C(C)C)C2)C1 38244,C(=O)(C(F)(CNC(=O)C(CO)OC)C(C)C)NC(CCC)c1ccco1 38245,C(=O)(C(O)C(O)c1ccccc1)N(CCCCNC(C(=O)N(C)C)=O)C 38246,N1(C(C(c2ccc(F)cc2)C)=O)CCC(C(=O)NCc2occc2C(=O)O)CC1 38247,C1(C(N2CCC3CC23)=O)COCCC1NC(C12CCN(CC1)C2)=O 38248,CCC(O)C(C)C(=O)N1CCN(C(C2CCCC2C(=O)OC)=O)CC1C1CC1 38249,c1(C(N2C(C)(CNC(=O)C=CC3CC3)CCC2)=O)occ2c1CCOC2 38250,c1(NC(C2C(C(N3CC4C(C(=O)OC)(C4)C3)=O)C2)=O)cncc(F)c1I 38251,c1(CC)cccnc1C(=O)N(CC(C)NC(c1ccc(-c2cccs2)[nH]1)=O)C 38252,C=C(C)C1OCCC1CNC(=O)NC(c1cccc(Br)n1)C 38253,CCC(C(C)(C)O)NC(=O)CC1CCN(C(=O)C(c2ccnn2C)C)CC1 38254,c1(C(=O)NC2CN(C(C(c3cnccn3)C)=O)CC2O)nsc2ccccc12 38255,c1(SC)cc(C(N2CC3CC2CN3C(c2cn[nH]c2)=O)=O)cc(SC)c1 38256,C1(C(=O)NCc2n(CC)ncc2)CN(C(c2ccc(OC(C)C)o2)=O)CC1OC 38257,C1(C(=O)NC(C2CN(C(C(CC#C)(C)C)=O)C2)C)CC2(C1)CC1(CC1)C2 38258,c1(C(=O)NCC(CC(=O)NCCCC(=O)NCC(C)C)C)coc2ccccc12 38259,c1(CN2CCC(C)(C(=O)NCCC)C2)cc2ccccc2s1 38260,N1(C(C(c2ccccc2)C)=O)CC2CCC(C(=O)NC3CC3)(C2)C1 38261,c1(CNC(CCCNC(N)=O)=O)cncc(C(=O)NC2COC(C(F)F)C2)c1 38262,c1(C(C)=O)cccc(CC(=O)NCCC2CCN(C(=O)C=C3CCC(C)C3)C2)c1 38263,C(=O)(CCCNC(C)=O)NCC(COC)NC(=O)C(CC1CCC1)OC 38264,c1(NCC2(c3cn(C)nc3)CC2)nc(NC2CC3CC(CO)CC23)c2ccsc2n1 38265,C(=O)(CC(C)C(C)C(C)C)N(C)CC1(O)CN(C(c2cc(C)nc(C)c2)=O)C1 38266,C1(CNC(C(C)OC)=O)CN(C(c2cc(C)c(Cl)cc2F)=O)CCC1(C)C 38267,N1(C(=O)COCCF)CCC2CN(C(=O)CSCc3ccc(Cl)cc3)C2C1 38268,C12CCN(CC1)Nc1cnn2c1.C1(CN(C)C)CCCCC1C(=O)O 38269,N1(C(C2C(C(C)C)C2)=O)CCC(F)(F)C(CNC(=O)Cc2ccsc2)C1 38270,N1(C(C2CCCC(CF)C2)=O)CCOC2(CCC(NC(C34CC(C3)C4)=O)CC2)C1 38271,c1(C(=O)NCC2N(C(CC(=O)OC)=O)CCN(C)C2)ccccc1N=S(C)(C)=O 38272,C1(C(N(C2CCN(C(C3(C)CCC(C)CC3)=O)C2)CC)=O)CCc2nn[nH]c2C1 38273,CC(CC(=O)NCC1CCN1C(=O)CC1CCCC1)c1cnn(C)c1 38274,C1(CC)(CO)CCCN1C(C1C=CCN(C(=O)C(N2CCOC2=O)C)C1)=O 38275,c1(CC(=O)NCC2N(C)CCN(C(c3cn[nH]c3)=O)C2)ccn2cncc2c1 38276,c1(OCC)cc(NC(c2ccc(-c3cn[nH]c3)cc2)C)cc(Br)c1 38277,C12(NC(=O)C=C(Cl)Cl)CCC(CC1)N(C(C1C3C4CCC(C4)C13)=O)C2 38278,C1(C(=O)NCC2(COC)CCCN2C(=O)CN=S(C)(C)=O)COC2(CCC2)C1 38279,c1(C(N(CCNC(C(CC)CC(F)F)=O)C2CC2)=O)ccc2c(c1)CCCC2=O 38280,c1(CC)c(C(=O)NC2(COC)CN(C(=O)C(F)(F)c3nccn3C)C2)cnn1C 38281,N1(C(CC2CC(NC(C#CC)=O)C2)=O)CCC2(CCOC2)C1 38282,CC1CCN(C(c2cnc(O)o2)=O)CC1CC(=O)NCCC1CCCC12CC2 38283,C(=O)(C1CCc2cccc(=O)n21)NC1C(OC)CN(C(C2(C(=O)OC)CC2)=O)C1 38284,C(=O)(C(F)CC(C)(C)C)NCc1ccc(C(=O)NCC2(OC)CCCC2)nc1 38285,c1(C(=O)OC(C)(C)C)cccc(CN(C)C)n1.C12(C)CCN1C2=O 38286,C(=O)(C(C(C)(C)C)OC(C)(C)C)N(C)CC1CCN(C(C2(C(N)=O)CCC2)=O)C1 38287,N1(CC)C(=O)CCC1C(=O)NC(C1CCCC1)CNC(=O)C(=C1CCCCC1)F 38288,C(C1CCN(C(C2(C)CC(F)C2)=O)CC1)=CC(=O)NC1(CC=C)CC1 38289,N1(C(c2c(NC(N)=O)cccc2)=O)CC2(CCN(C(c3cc(CO)[nH]n3)=O)C2)C1 38290,c1(C(=O)NC(C)C(CO)NC(c2cc3n(n2)CC(F)C3)=O)cccn2nccc12 38291,C1(CNC(CCCc2ncc(C)o2)=O)CC(NC(=O)CNC=O)C12CCC2 38292,Cn1cc(C(=O)NCCCNC(=O)C(F)CC2CCCCC2)ncc1=O 38293,CCC(C)CCCCC(=O)NCC(C)N(C(c1ccc(OCCF)cn1)=O)CC 38294,C1(NCc2ncc(C(C)(C)C)s2)COC2CCCCC12 38295,Cc1cc(C(=O)NCC2(NC(=O)C=Cc3ccc(=N)[nH]c3)CC2)c2c(c1)CCC2 38296,Cc1cc(F)ccc1NC(N1CCC(C)(NC(=O)C(=O)NCC(F)F)CC1)=O 38297,Cc1ccnc(O)c1C(=O)NC(CNC(c1ccnn1CC(F)F)=O)C1CC1 38298,C(=O)(C(CC)(CC)CC)N1C(C)(CC(=O)NC(C(=O)OCC)CO)CC1 38299,C1(NC(=O)CN2C(=O)CNC2=O)CN(C(=O)CCc2nncs2)CC12CC2 38300,N1(C(C=CC)=O)CCN(C(=O)C(C)N(C)C(C)=O)C2(CC2)C1 38301,c1(C(N(CCN(C(C(COC)C)=O)C(C)C)C)=O)ccc2c(c1)NCCNC2=O 38302,C1(CNC(CCC(C)SC)=O)CN(C(=O)C(C)(C)n2ccnn2)CCCO1 38303,c1(N2CCC(N(C)C)CC2)nc(=NCC2CC2Cl)[nH]c2c1SCC2.C(=O)C(C)(C)C 38304,CCC(C(=O)NCC(C)CNC(=O)Cc1cccc(OC)c1F)C(F)(F)F 38305,C1(C(F)(F)F)(OC)CCCN(CC2CCC(C#N)CC2)C1 38306,CC1(C)CC(CNC(C2CC3(CCCO3)C2)=O)CN1C(c1ccc(C2CC2)o1)=O 38307,CC(CNC(C1CN2CCN1CC2)=O)C(F)C(=O)NCC(C)(C)N(C)C 38308,CCC(C(=O)NC(CO)C(=O)NCCCCO)n1ccnc1 38309,Cc1cc(O)c(C(N2CC(NC(=O)C=Cc3cnc[nH]3)C(C)(C)C2)=O)nn1 38310,c1(CC(CO)NC(Cn2c(C)c(Cl)cn2)=O)c[nH]c2ccccc12 38311,C1(NC(CC2CC(=C)C2)=O)CC(F)CN(C(=O)Cn2cccc(C)c2=O)C1 38312,C#CCC(C)(C(=O)NC(CCO)C1CCCC1)NC(c1ncnc(C)c1C)=O 38313,N1(C(C(C)(C)OC)=O)CC2(CCC2)CC1CNC(=O)C#CC1CCCO1 38314,C1(NC(CC2N(C)CC=CC2)=O)CCN(C(=O)CC2CN3CCC2CC3)CC1O 38315,c1(C(=O)NCCOC2CN(C(c3nn(CC)c(C)c3)=O)C2)sc(C)c(C)c1C 38316,c1(C(=O)NC2(C)CN(C(C3(C)CCCS3(=O)=O)=O)C2)ccc(F)c(C(F)F)c1 38317,C=CC1OCCC1C(N1CCC(CCN(C(=O)CC(O)CN(C)C)C)CC1)=O 38318,N1(C(C2(C#N)C(C)C2)=O)CCC(O)(CN(C)C(c2cn3ccsc3n2)=O)CC1 38319,C12(NC(C34CC(OC)C3C4)=O)CCCC1CN(C(=O)Cc1c(C)cccc1C)C2 38320,c1(C(=O)NCCC(C)(C)NC(=O)C(O)CCS(C)=O)nnc(O)c2ccccc12 38321,c1(C(=O)NC(C(=O)NC(CC)CCCO)c2ccoc2)c[nH]c(C)cc1=O 38322,Cc1cc(F)sc1C(=O)NC(C(=O)N(C)Cc1cccnc1O)C1(O)CCC1 38323,N1(C(C2(CC(C)C)CCC2)=O)CC2CC1CN2C(C1CC1(Cl)Cl)=O 38324,N1(C(C(OC)OC)=O)C2CCC1CC(NC(C1CCNC(=O)C1)=O)C2 38325,CC1CCN(C(=O)C2=CCCC2)CCN1C(c1noc2c1CCCC2)=O 38326,Cc1ccc(C(=O)NC2CCC(NC(c3cnn4cccnc34)=O)C2)c(C)c1Br 38327,c1(CC(=O)NC2C(CNC(=O)COc3ccsn3)C2)ccc(O)nc1 38328,Cc1oc2ccccc2c1C(N1CCN(C(=O)CC2COC(C)(C)C2)C(C)C1)=O 38329,C1(C(N2CCC(O)(Cn3cc(C4CCCC4O)nn3)C2)=O)CCCC2(CCC2)O1 38330,N1(C(C2(C3(C)CC3)CC2)=O)CCC2CCCN(C(c3cc4n(n3)CCC4)=O)C2C1 38331,N1(C(C23OC(C)C(CC2)C3)=O)CCOCC(C)(CNC(C2(C3CC3)CC2)=O)C1 38332,C(=O)(C(F)C(=O)N(C)CC1CCCCN1C(=O)C(C)(C)OCC(F)(F)F)OCC 38333,CCCC(C)(CCC)C(=O)NCCCNC(=O)C(C)OCC1CCCCO1 38334,C1(N=[N+]=[N-])(C(=O)NCC(CCC)(C)C)CCN(C(C2CCOC2(C)C)=O)C1 38335,c1(C(=O)NCC2CC(NC(C3(N(C)C)CCC3)=O)C2(C)C)ccc2c(c1)OCO2 38336,c1(CN(CC(N2CCC(Cc3c(C)noc3Cl)C2)=O)C)ccc2c(c1)OCCO2 38337,N1(C(c2cncc(N)c2)=O)CC2CCC1C1CN(C(c3cnc(O)o3)=O)CC21 38338,c1(C(CC)C(=O)N(CCCN2CCCC2)C)ccc2c(c1)OCO2 38339,Cc1conc1C(=O)NC(C1CN(C(c2cnn(C(C)C)n2)=O)C1)C 38340,C1(C(=O)NCC2(C(C)(C)O)CN(C(CSCC=C)=O)C2)CCCCCC1(F)F 38341,CC(C(C)(C)C(=O)NCCn1cccnc1=O)NC(c1cnc2n1CCC2)=O 38342,C1(C(=O)NCc2c(CC)cncc2)CCCN1NC(=O)C(F)C(F)(F)F 38343,C1(C)(C(=O)NC)CCCN1C(c1cn(CCNC(=O)CC2(C#N)CC2)cn1)=O 38344,C(C(F)(F)C(F)(F)F)O.C1(NC(CN(CCC)C(C)=O)=O)CCC1NC(=O)CC 38345,C=CC(C)(CC)C(=O)NCCC1(C(=O)NC2(c3ccccc3)CCC2)CC1 38346,n1(CCOC)ccc2cc(NC(c3cccc4c3COC4)=O)ccc12 38347,c1(CC)cccnc1C(=O)NC1CC(C)N(C(=O)CC(C)n2ccnc2)C1 38348,Cc1cc(NC(C2CC3CC3N2S(=O)(=O)c2cn[nH]c2)=O)c(C)cc1Br 38349,n1(C(C(=O)OCC)C)nnnc1C(C1CCCO1)(C)NCCc1nocc1CC 38350,C1(C(N(C(CN(C(C)=O)C)C)C)=O)CN(C(=O)C(c2cccn2C)=O)CC1(F)F 38351,c1(C(=O)NC(c2cccnn2)C)nc(Br)sc1Cl 38352,c1(C(=O)NCC(CC)NC(C2(C3CC3)CCCO2)=O)[nH]c2ccc(C)cc2c1C 38353,C#Cc1ccc(OCC(=O)NCC(CO)NC(c2ccc(Cl)cn2)=O)cc1 38354,C1(CC(=O)NCCN(C2CCCCCC2)C(=O)C=C2CCC2)CCS(=O)(=O)C1 38355,C1(OC)CN(C(=O)CN2CSCCSC2)CC1NC(=O)CCn1ccnc1C 38356,N1(C(c2c(C)csc2)=O)CCCCC1CNC(c1ccc(-c2ccco2)s1)=O 38357,N1(C(CC(C)C)=O)CC(NC(=O)C(CC(C)C)NC(N)=O)C(C)(C)C1 38358,Cc1n[nH]cc1C(C(=O)NC(C)C)N(C)CCC1CCCCC1 38359,C1(C(=O)OCC)(C(=O)NCCC2(C)CC2(Cl)Cl)CCCNC1 38360,C1(CNC(C(=O)N(C)Cc2ccn(CC)n2)=O)C2CCCCCC12 38361,N1(C(C(C)c2cncs2)=O)CC2CC(C1)CN(C(=O)C(CO)N(C)C)C2 38362,C1(NC(c2c(Cl)cn(CC)n2)=O)CC2CC(C1)CN(C(=O)CC1CC13CC3)C2 38363,N1(C(C(=O)N(C2C(C)OCC2)CCO)=O)CCN(S(=O)(=O)N2CCCC2)CC1 38364,C1(C(=O)NCC(CN(C)C(C2(C(F)F)CC2)=O)O)CCC=CCCC1 38365,C1(COC)C(O)C(O)CCN1C(C1CCCN(c2ccnn2C)C1)=O 38366,CC1(C)CC(C(=O)NCCCCCC(=O)NC2CCCSC2)CCO1 38367,c1(CC)ccc(F)cc1NC(C1CC(NC(=O)Cc2ccc(O)nc2)C1(C)C)=O 38368,Cc1cc(C)c(C(=O)NC2CCC(F)(CNC(c3cccn3C(C)C)=O)C2)cn1 38369,c1(C(=O)NCC(C=C)O)nc(CNC(=O)CN(C)C(C)=O)oc1C 38370,c1(C(N2CC3CC(NC(C(C)(C)OC)=O)CC3C2)=O)c(C)oc2nc(Cl)ccc12 38371,c1(C(=O)NCC2C(NC(CC(c3cccc(F)c3)C)=O)C2)ncnc2ccsc12 38372,n1(CC(N2CC(C(C)NC(c3n(C=C)nnc3)=O)C2)=O)nnc2ccccc12 38373,C(CCCCC(=O)N1CC=CC1C(=O)NCCN1CCCCCC1)=CC 38374,CCCC(C(=O)N1CCCC(N(C(=O)C(C)OCC(C)C)CC)C1)N(C)C 38375,CC1(C)CC(C(F)(F)F)(C(=O)NCC2CCC2NC(=O)CSc2ccccn2)C1 38376,N#Cc1n[nH]c(=NC2CCCC23CN(C(c2c[nH]cc(Cl)c2=O)=O)C3)s1 38377,CC1CC(C(C)(C)C)CCN1C(=O)Nc1ccnn1C 38378,C1(C(N2CCC(OC)C2C(C)C)=O)COC2(C1)CN(C(c1cccc(=O)o1)=O)C2 38379,C(=O)(C(C)CCCC(C)C)NC(CNC(C(=Cc1cn[nH]c1)C)=O)CO 38380,N1(C(C2COC(=O)O2)=O)CC23CCCC2(C1)CN(C(c1cnc(O)s1)=O)C3 38381,CC1CN(C(=O)C(c2ccc(F)cc2)F)C(C)CN1C(=O)C1=CCSC1 38382,N(C1COc2ccccc21)C(C(CC(F)F)NC(=O)Cc1cnns1)=O 38383,C12(NC(C3(C#N)CC(C)C3)=O)CCCC1N(C(=O)CCOCC(F)(F)F)CCC2 38384,c1(C(=O)Nc2cc(C)cc(O)c2)cn(C)c2ccc(-c3cccc(F)c3C)cc12 38385,CC1CN2CCN1CC2C(N1CC(NC(C2NC(=O)C3CCC23)=O)C(C)(C)C1)=O 38386,CC1(C)CCN(C(=O)C=C2CCC2)CC1C(=O)NCC1CC(O)C(O)C1 38387,C1(CCNC(CC2C(C)CCC2)=O)CCCN(C(=O)CC(C)(C)O)CC1 38388,C1(C(C)(C)O)(CNC(=O)CC2CCCC2)CN(C(=O)CN(C2CCCC2)C)C1 38389,N1(CC)C(=O)CCC1CC(=O)NCc1csc(CNC(C2COCC2(C)C)=O)n1 38390,C1(N(CC(=O)Nc2onc(C)n2)C)CCCN(c2ccccc2)C1=O 38391,N1(C(CC)C(F)F)CCS(=O)C(C)(C)CC1 38392,c1(NC(C2CN(C(C3CNC(=O)O3)=O)CC(F)C2)=O)nc(Cl)c(Cl)nc1CO 38393,C(C(C)C(F)C(=O)NCCC1C=CCC1)NC(c1noc(CC)c1C)=O 38394,C1(COC)(NC(=O)C(c2ccccc2)F)CCN(C(=O)CCOC(C)=O)CC1 38395,C(=O)(NNC(=O)C(CN)CC(C)C)c1c(C)nc(-c2nn[nH]n2)cc1 38396,N1(C(C(CC(C)(C)C)NC(c2cnn(CC)c2C)=O)=O)CC(C)C12CCOCC2 38397,Cc1nc(C(=O)NCC(C)NC(=O)CCCc2ccc(F)cc2)sc1C 38398,c1(CCNC(C(C2CCN(C(c3ccn(C)n3)=O)C2)(C)C)=O)ccc(F)cc1 38399,CC1CN(C)CC(C(N2CCCN(C(=O)CN3C(=O)CNC3=O)CC2)=O)O1 38400,C1(OC)CC(CNC(c2cccnc2)=O)N(C(=O)CC(F)(F)Cl)C1 38401,c1(C(N(CCN(C(CCc2cnc(C)s2)=O)C(C)C)C)=O)ccccc1N(C)C 38402,C1(NC(N(C2CN(C(=O)OC(C)(C)C)C2)C)=O)(SCC)CCSCC1.C1CC1 38403,c1(C(N2CC(O)(C(C)NC(C3CC3(C)C(F)F)=O)C2)=O)ccccc1C(C)(F)F 38404,C(=O)(C(C)C(O)CC)NCC1(C(=O)NC2(CC=C)CCCCC2)CCCC1 38405,c1(CCC(=O)N(CC(C)CNC(=O)Cc2ccon2)C)ccc(O)c(Cl)c1 38406,C(C1=CCN(C(c2ccsc2)=O)CC1)NC(c1cn(C2CCC2O)nn1)=O 38407,C1(C(N2CCN(C(c3n(C)nnc3)=O)CC2CCO)=O)CC2CCCCCC12 38408,C1(NC(c2cc(CCC)ncc2)=O)CCN(C(c2sccc2F)=O)CC1CO 38409,CC1(C)CC(=O)N(CC(=O)NC2C=CCN(C(c3cccc(F)n3)=O)C2)C1=O 38410,c1(C(=O)OC)cccc(NCc2ccncc2OCC(F)(F)F)c1OC 38411,C=CC1CN(C(c2cscc2C(N)=O)=O)CC1NC(=O)C(C(C)C)SC 38412,C1(C(=O)NCC(CC=C)(F)F)CC2CCC(C1)N2C(=O)C(C)(C)C(=O)OCC.O 38413,c1(C(=O)NCC(C)(C)NC(CC2CC(SC)C2)=O)ccc2c(c1)OC(C)(C)C2 38414,N12CC3CCC3(C1)C2=O.c1(NC(C2C(OCC=C)CC2)=O)cc(CC)cc(F)c1 38415,C(=O)(C(O)C(F)(F)F)NC1C(N2CCN(C(Cc3cc(C)sc3)=O)CC2)CCC1 38416,C1(NC(c2c(CC)cco2)=O)CCN(C(C2(C)CCCN2C)=O)CC1O 38417,Cc1c(NCC2CC2C)ncnc1N1CCN(c2ncccn2)CC1 38418,C1(C)(C(N(CCCNc2c(C(=O)OCC)cco2)C)=O)CCOC1C 38419,c1(C(=O)NC2CC(C(=O)NC3(CC)CCC3)C2(C)C)cc(C)c(C)nn1 38420,C1(NC(c2ccc(CCO)cc2)=O)CN(C(=O)C2=CCC2)C2(CCOCC2)C1 38421,C1(NC(C(CC=C)CNC(=O)C=C(C)C(F)F)=O)CC2CC1CC21CC1 38422,C1(C(N2CC(C)N(CCOC)C(C)C2)=O)CCc2n[nH]c(C)c2C1 38423,N1(C(CNC(=O)NC)=O)CCC(C)(NC(=O)COC2CC=CC2)C1 38424,c1(C(N2CCC(N(C(c3ncc[nH]c3=O)=O)CC)C2)=O)cc2c(ccn2C)[nH]1 38425,C1(NC(C(C)Oc2ccc(Cl)cc2)=O)CCN(CCF)C1(C)C 38426,c1(C(=O)NCCN(C(=O)Cc2cc(Cl)ccc2O)CC)cnc2ncccc2c1 38427,C1(C(=O)OC(c2onc(CC(C)C)n2)C)CCN(C(=O)NC(C)C)CC1 38428,N1(C(c2c(CC)nns2)=O)CCN(C(=O)Cc2ccc(C)c(C)c2)CC1C(C)C 38429,N1(C(C(CC)=CC)=O)CCC(CNC(=O)CCc2ccc(OC)c(Cl)c2)C(C)C1 38430,c1(C(N2CC(C)(C(=O)Nc3cncc(C(C)(C)C)c3)C2)=O)ccc(Br)nc1Br 38431,c1(C(N2CCCC(N(C)Cc3cc(C)no3)C2)=O)n[nH]c(C)c1[N+](=O)[O-] 38432,c1(C(=O)NC2C3(CC(NC(=O)Cn4cc(Cl)cn4)C3)C2)cccc2c1OCCO2 38433,N1(C(c2ncn(CC)c2)=O)C2CCC1CC(CNC(=O)C(=Cc1cscn1)F)C2 38434,CCCCCCCCC(C)CC(=O)NC1CC(CNC(=O)C(F)(F)C(F)(F)F)C1 38435,C1(CNC(C(F)=CCC)=O)CN(C(=O)CC2CC(C)(C)OC2=O)C2CCCC2O1 38436,N1(C(c2c(C)nc(N(C)C)s2)=O)CCCC12CCCN(C(=O)C(O)C1CC1)C2 38437,c1(OC)ccc(OC)c(C(N2CCC(C)(CNC(C3(C)CC(C)(C)C3)=O)C2)=O)n1 38438,Cc1ccc(C(N2CCOC(C(=O)NCCCN(C)C3CC3)C2)=O)cc1Br 38439,c1(C(=O)NCCC(C)N(C(=O)C(O)CC(N)=O)C)cccc(S(=O)(=O)C2CC2)c1 38440,O=C1Cc2c(C(N3CCC(CCn4cc(CCC5CC5)nn4)CC3)=O)cccc2N1 38441,C1(CNC(c2nc(CCC)sc2)=O)C(O)C(O)CN1C(C1CCCCS1(=O)=O)=O 38442,C1(NC(C(C)OCCN(C)C)=O)CCN(C(C2CCC(O)CC2)=O)CC1F 38443,c1(C(N2CCCC(=C)C2)C(=O)NCCCOC)cccc(F)c1I 38444,C1(c2cccs2)(C(=O)NC(C#C)(C)C)CCN(C)C1 38445,C(=O)(CC(C1CC1)C1CC1)NC(CN(C(C(=O)NCC)=O)C)CC 38446,CC1(CNC(c2coc(Cl)n2)=O)COCCN(C(c2ccnc(O)c2)=O)C1 38447,Cc1cccc(C)c1CC(=O)NC1CC2(C1)CC(NC(C1(F)C3CCCC13)=O)C2 38448,c1(C(=O)Nc2cc(O)n[nH]2)cnc2n[nH]c(-c3cccnc3C3CC3)c2c1 38449,N1(C(C(CC#C)C)=O)CC2CCC2(CNC(c2ccc(NS(C)(=O)=O)nc2)=O)C1 38450,c1(N2CC(C)S(=O)CC2)ncc(S(=O)(=O)NCCC2(CO)CCC2)cc1Cl 38451,Cc1c(C(=O)NCC2(C)CCN(C(=O)CCCNS(C)(=O)=O)CC2)cncc1Cl 38452,C=CCC(CC(=O)NCc1ncoc1C(C)C)NC(=O)C(CCC)N(C)C 38453,C1(N(C(c2cccc(Br)c2)=O)CC)CN(C(=O)CN2CCC2C)C(C)(C)C1 38454,c1(C(C)NC2(C)CCC(=O)NC2=O)cccc(S(=O)(=O)C(=O)N(C)C)c1 38455,c1(C(N2CCN(C(C(C(CC)C)O)=O)C(CO)C2)=O)cc(C)c2[nH]nnc2c1 38456,c1(C(N(CCN(C(C23CCC(OC)C2CC3)=O)C)C)=O)c(Cl)nc2sc(C)cn12 38457,C1(CCN(C(CC=C)=O)C)CCCCN1C(c1nc(CC(F)(F)F)sc1C)=O 38458,N1(C(CC2(C)CCCC2O)=O)CCn2cncc2C1.N12CC3C(C3C1)C2=O 38459,c1(C(=O)NC2CC3(CC(NC(CCC(CC)C)=O)C3)C2)ccc2c(c1)CCN2 38460,C1(NC(CC(C)N(C)C)=O)CC2CCC1CN2C(=O)CCCCC1CC1 38461,C1(CC(=O)NCC(O)CF)C2CCCC2N1C(=O)CC1CC2(CCC2)CO1 38462,C1(NC(CCCC=C)=O)CCC2(CC1)CC2NC(c1c(SC)cnn1C)=O 38463,n1(CC(=O)NC(C2CCN(C(C3CN(C4CCOC4)C3)=O)C2)C)cc(Cl)cn1 38464,C1(C(=O)NCC(C)NC(=O)CC(C)(C)O)CC(c2ccncc2)=NO1 38465,C=C(C)CCC(C(=O)Nc1ccc2c(c1)OCO2)N1C2CCC1CC(O)C2 38466,CC1COC(C(=O)NCc2csc(CNC(C3OCCO3)=O)n2)C1 38467,CCN=c1ccc(C(=O)NCC2(F)CCC(CNC(=O)CC3CC3)C2)c[nH]1 38468,c1(C(=O)NCCCn2cc(C(C)(C)C)nn2)ccc(CO)cc1F 38469,c1(C(N2CCC(CNC(C(C=C)O)=O)CC2C)=O)c[nH]c2c(F)cccc12 38470,O=S(=O)(CCCCC1CC1)NC1(c2ccc(F)cc2)CCCCC1 38471,N1(C(Cc2ncc(C)s2)=O)CC2CC(NC(c3cn(C)nc3C(F)(F)F)=O)C2C1 38472,CC1=C(C(=O)N2CCC(C)(NC(C3CC4CC4C3)=O)C2)CCCO1 38473,c1(C(=O)NCCC(=O)NC(C)C)ccc(CNC(=O)C(C)c2cc[nH]n2)cn1 38474,c1(CC)oc(C(=O)NCCC2(O)CN(C(=O)CCC(C)OC)C2)cc1C(=O)OC 38475,c1(C(=O)NCC(CNC(c2cnncc2C)=O)OC)c[nH]cc(C)c1=O 38476,Cc1cc(F)ccc1-n1cc(O)c(C(=O)OCC2C=CCC2)n1 38477,c1(OCC(=O)NC(CNC(C(C)=C(CC)C)=O)CO)ccc(Br)cc1Cl 38478,CC1CCC(C)(C(=O)NC2CCCC2NC(=O)CCC2OCCO2)C1(C)C 38479,c1(CNC2CCC3(CN(C(c4cnccc4Cl)=O)C3)C2)ccc2ncccc2c1 38480,c1(C(N2CCC(CNC(C3(C#N)CCCO3)=O)C2)=O)cn2cc(Cl)cnc2n1 38481,C1(CC(N2CC(CC(C)NC(=O)Cc3cnsc3)C2)=O)OCCC1(C)C 38482,C12(C(N(C3CCCN(C(C(CC#C)O)=O)C3)CCO)=O)CCOC(C)(C1)C2 38483,CN=c1[nH]cc(C(=O)NC2CCOCC2C(=O)NCc2cc(Cl)ccn2)s1 38484,C12(NC(COCCCC#C)=O)CCC(CC1)N(C(=O)CS(=O)(=O)C1CC1)C2 38485,N1(C(=O)NC(c2nc(C(=O)OCC)c(N)s2)C)CC(C2CCC2)CCC1C 38486,C(=O)(CC(O)(c1ccccc1)C1CC1)N(CC(C)NC(c1c[nH]c(Br)c1)=O)C 38487,c1(C(=O)NCC2CC3CCC2N3C(=O)CCSC(F)(F)F)coc2c1CCCC2 38488,C1(C(N2C(CNC(C3CC4(CCC4)C3)=O)CC3CC32)=O)CCc2nc(O)[nH]c2C1 38489,C1(CC(N2CCC(C(CNC(c3c(C)cns3)=O)C)CC2)=O)CCCCC12CC2 38490,c1(C(=O)NC2CC(CNC(C3CC4CC4C3)=O)C2)cccc2ccnn12 38491,N1(CC(=O)NC(C2(CNC(=O)C3CC3)CC2)C)C(=O)Cc2ccccc2C1=O 38492,N1(C(c2nn(C)c(=O)cc2)=O)CCC(NC(=O)CC2CC2C(F)(F)F)CC(C)(C)C1 38493,N1(C(Cc2n(C)cnc2)=O)CC2CC1CN2C(c1[nH]ncc1C#N)=O 38494,c1(C(=O)NC2(C)CCC(NC(=O)C(N)=O)CC2)coc(C#Cc2ccccc2)c1 38495,c1(OC(C)C)cnc(=NCCC(C)NC(C2CCc3nn[nH]c3C2)=O)[nH]c1 38496,O=C(CCCC(=O)Oc1cccc(Br)c1F)NC(COCc1ccccc1)CO 38497,N1(C(c2cc(OC)ncc2F)=O)CCCN(C(C2CC3CCC(C2)O3)=O)CC1C 38498,C1(Nc2c(C)oc(-c3ccccc3)n2)C2CC3C1C3C2C(=O)O 38499,N1(C(CCC(=C)Cl)=O)CCCCC(CNC(c2ccn(C(F)F)n2)=O)CC1 38500,C(C(C)CC(=O)N(C(C)CN(C(=O)Cn1nc(C(F)(F)F)cc1C)C)C)OC 38501,C1(N(C)C(c2ncoc2Br)=O)CCC(NC(=O)CN2CC=CC2)CC1 38502,C(=O)(CC(O)CNC(=O)CCc1ccsc1)N(C(C1CCCC1)CO)C 38503,C(CC(=O)NCC1(F)CCN(C)C1)(C(F)(F)F)NC(C1(OC)CCOC1)=O 38504,C1(NC(CNC(C(C)(C)C)=O)=O)CN(C(=O)Cn2nnc(=O)[nH]2)CC12CC2 38505,CCCC(C)(O)CC(=O)NCC1(C)CN(C(c2nc(C)c(C)s2)=O)CC1C 38506,N1(C(C2C(=C)CC2)=O)CCOC(CCCNC(c2cc(C(N)=O)co2)=O)C1 38507,C1(C(=O)NC2C(c3cn(C)nc3)C2)N(C(=O)CC2CCC=CCC2)CCC1(C)C 38508,C(=O)(C(CC(C)CCC=CC(C)C)N1CCC(C)(C=C)CC1)NCCSC 38509,Cc1ccc(CN2CCC(C(=O)NCc3cccnc3F)C(O)C2)cc1C#N 38510,CC(CN(C)C)N=c1[nH]c(N2CCC(C(C)(C)C)C2)nc2c(F)cccc12 38511,Cc1nc(O)ccc1C(N1CC2CC2C1C(=O)NCC1CC(C)(C)C1)=O 38512,C(CNC(c1cc(Br)no1)=O)(C(C)(C)C)NC(c1ccc(C(=O)OC)s1)=O 38513,N1(C(c2cnc(-c3ccccc3)o2)C(=O)NCC=C)CC(=O)N2CCCCC2C1 38514,C(=O)(CCCC(C)C)NC1C(SC)CN(C(=O)C(C)Cc2ccccc2)C1 38515,C(C(C)(CNC(C1COCC1NC(=O)CN(C)C(=O)OC)=O)CO)OC 38516,C1(CNC(c2n[nH]c(C)c2O)=O)(NC(=O)C(C)SC(F)(F)F)CCC(C)(C)CC1 38517,CC(=O)CCCC(=O)N1C2CCC(C2)C1C(=O)Nc1cn(C)nc1Cl 38518,c1(OC)ccc2oc(C(=O)NC3(C#N)CCN(Cc4ccccc4I)C3)cc2c1 38519,C1(N(C(C(CC)O)=O)C)C2CN(C(=O)CCCNC(=O)OC)CC12 38520,c1(OC)cc(C(=O)NC(C)C(C)NC(=O)Cc2cccc(C)c2Cl)ccc1F 38521,c1(C(=O)NC2C(CNC(CSCC(C)C)=O)CCC2)nnc(O)cc1O 38522,Cc1cc(=O)n(C)cc1NC(C1CC12CC(NC(=O)C(C)CN(C)C)C2)=O 38523,C(=O)(C(C)C(O)C(C)C)NCCCC(C(N1CCCC(C)(CC)C1)=O)O 38524,C1(NC(C2CCCN2C(c2cc(-c3ccccn3)[nH]n2)=O)=O)C2COCC12 38525,C1(C(=O)NC(c2cc(F)ccc2OC)CC)CC2(CCC(N)CC2)C1 38526,c1(OC)cc(C(N2CCC(O)(CN(C(=O)CCc3ccoc3)C)C2)=O)cc(F)n1 38527,S(=O)(=O)(c1ccc(N2CCC3CCCC3C2)cc1Cl)NCC1N(C)CC(O)C1 38528,c1(OC)ccc(C)cc1CNC(=O)Nc1cccc(N2CCCCC2=O)c1 38529,Cc1nnccc1C(N1CC=CC(C(=O)NCCc2ccc(O)cn2)C1)=O 38530,C12(CNC(C(C)NC(=O)NC)=O)CC1CN(C(=O)C=Cc1c[nH]nc1C)C2 38531,c1(C(=O)Nc2cccc(C(=O)NCCCS(N)(=O)=O)c2)cncc2[nH]ccc12 38532,N1(C(C(C)c2cccs2)=O)CCC(N(CCCC)C=O)CC1.C1(C=O)C(C)C1(F)F 38533,CC1(C2CCN(C(=O)C(CN=[N+]=[N-])NC(c3cnco3)=O)CC2)CC1 38534,C1(C(=O)NCC(CC)OC)C=CCN(C(C2(C)CC3CC3C2)=O)C1 38535,N1(C(C(=O)N2CC(C(CC)CC)C2)CCO)CCc2sccc2C1 38536,N1(CCCC(=O)NCC2N(C(C(CC)CC)=O)CCOC2)C(=O)CN(C)C1=O 38537,C1(C(=O)NC(c2ccnn2C)C(=O)N(CCCC)CCCO)CC(O)CN1C 38538,N1(CC(=O)NCC=CCNC(=O)CC2CCC2)CCCc2sccc2C1=O 38539,c1(C(N(C)CCc2cn(C(C)C(=O)O)nn2)=O)cc2c(=O)cc[nH]c2s1 38540,S(=O)(=O)(C1CC2C(C1)C2(F)F)N1CCC(N(C2CCCC2)C)C1 38541,c1(C(=O)NC(CNC(CC(CCC)C)=O)C(C)(C)C)ccc(C)c([N+](=O)[O-])c1 38542,C(CCCCNC(=O)C(C)NC(=O)C1CC1)NC(C(C1CCOCC1)OCC)=O 38543,C1(C(C)NC(=O)CSc2nncn2C2CC2)CCN(C(C2(C)CC2(F)Cl)=O)CC1 38544,N1(C(c2ccc(C(C)=O)o2)=O)CCC(O)(CCNC(C2CCNC2=O)=O)CC1 38545,C1(NC(C(C)SCC)=O)CCCN(C(C23CC(CC)(C2)C3)=O)C1 38546,N1(C(C2CCC(OC)C2)=O)C(C(=O)NC2(CCCCO)CC2)CCC1C1CC1 38547,CC1CN(C(=O)C(CO)NC(=O)Cc2ncccc2F)CC1(F)F 38548,c1(C(=O)NC)cn(CC(N2CCC(CNC(C3(Cl)CC3(F)F)=O)C2)=O)nn1 38549,N1(C(C2(C)C(C(=O)OC)C2)=O)CCOC(CCNC(=O)CCNS(C)(=O)=O)C1 38550,c1(C(=O)NCC(CN(C(CNC(CNC(C)=O)=O)=O)C)O)c(N)ccc(C)c1F 38551,C1(=CCNC(c2cc(CCC)on2)=O)CCN(C(=O)C(C)(COC)OC)CC1 38552,C=CC1CCCCN1C(=O)COC(C1CCN(C(=O)OCC(C)(C)C)CC1)=O 38553,N1(C(C2(CCNC(C(N3CCCCC3)C)=O)CCC2)=O)CCC(O)CC(C)C1 38554,C1C(C)(C)C(=O)NOCc2ccc(nc2)N1.c1(NC)ccc(C(=O)N(C)C)cc1 38555,N1(C(C(=O)N(CC(C)C)CCOC)=O)CCCC(C(C)C)CC1 38556,N1(C(c2c(CC)c(F)ccc2)=O)CCC2(CCN(C(C3CCC(C)O3)=O)CC2)C1 38557,N1(C(C(=O)NCCOC)=O)CCN(C(C2(SC)CCOCC2)=O)CCC1C 38558,CCC(CC(=O)N1CCOC(CC(=O)N(C)CC2CCCN2CC)C1)CC(C)C 38559,N1(C(C(CC2CC2)OC)=O)CCN(C(=O)Cc2cnn(C)c2C)CC(C)C1 38560,c1(C(=O)NC2CC(C)N(C(c3cncc(F)c3Cl)=O)C2)cccc2c[nH]nc12 38561,Cc1csc2c(C(=O)NC3(CNC(=O)C=Cc4ccoc4)CCC3)cccc12 38562,N1(C(COCCCC)=O)C2CCC1CC(O)(CNC(=O)C(F)Cc1cnc[nH]1)C2 38563,C1(CNC(CCc2c(C)ncs2)=O)CCC2CN(C(=O)CC3(C)CC3)CCC2C1 38564,C(C(=O)N1CC(NC(=O)C(C)OCCN(C2CCCCC2)C)C1)(C(C)C)OCC 38565,Cc1cc(C(C)(C)C)ccc1C(=O)NC1C=CCN(C(=O)C#CC2CC2)C1 38566,c1(CC(=O)NC2C3CCN(C(c4nc(C)oc4)=O)C32)c(C)cccc1C 38567,C1(C(=O)N(C2CCCC2C)C)(CC)CCN(C(=O)C#CC(C)(C)C)CC1 38568,C1(CCC)(CNC(c2[nH]ccc2COC)=O)CCN(C(C2CN3CCC2C3)=O)C1 38569,c1(C(=O)NCC2N(C(C34CC(C)C3C4)=O)CC2)cccc(Cn2cncn2)c1 38570,c1(C(=O)NC(CCNC(C2CCC(C(=O)OC)C2)=O)(C)C)nc(C)sc1Br 38571,S(=O)(=O)(c1ccsc1CNCc1cc(C(=O)O)cs1)N1CCCC(C)C1 38572,C1(C(N(C(C)CC(=O)NCC(O)(C2CC2)C2CC2)C)=O)CC12CCOC2 38573,CC(CCCCNC(C1(N(C)C)CCCOC1)=O)NC(=O)CC1COC2CC1C2 38574,C1(NC(c2nnnn2CCOC2CCOC2)(CC)C2CC2)CCC2(CC1)CSC2 38575,c1(C(=O)NC2C(NC(C(N(C)C)C3CC3)=O)CC2)ccc2cccc(Cl)c2n1 38576,c1(OC)ncccc1CNC(=O)CCC1CCN(C(=O)C(=O)NC2CC2)C1 38577,Cc1nc(C=CC(N2CC(NC(=O)CC3CCCCCO3)C(F)C2)=O)[nH]c1C 38578,C(=O)(CCCNC(=O)C1CC1)NCC(CNC(c1cnc(Cl)[nH]1)=O)OC 38579,CC(C(=O)N1CCOCC(CNC(=O)CN(C)C(=O)C2CC2)C1)S(C)(=O)=O 38580,C1(C(N2CC(OC)(CNC(C3(C)CC3(C)C)=O)C2)=O)CN2CCN1C(C)C2 38581,c1(N2CC(C)(C)N(CCO)CC2)nc(N2CC3(C)CCC3(C)C2)c2ncsc2n1 38582,CC1CCN(C(c2ccc(O)c(N)c2)=O)CC1NC(C1(C)CC(O)CN1C)=O 38583,c1(C(N2C(CNC(Cc3cn(CC)nn3)=O)CCCC2)=O)cc(Cl)c(F)c(Cl)c1 38584,c1(C(N2CCC(NC(c3ncc(CC)nc3)=O)CC2)=O)c(C)oc(C)c1C 38585,C1(CNC(C(C(C)C)N(C)C)=O)C2CCCC1N(C(=O)CSC(F)(F)F)C2 38586,c1(N(CCC)CCNC(=O)CCCN(C)C)ncnc2sc3c(c12)CCC(C)C3 38587,N1(C(C(C(C)(C)C)OC)=O)CCC(C2(NC(c3scc4c3OCCO4)=O)CC2)C1 38588,c1(CC)ncc(C(=O)NC2CC(N(C)C(c3c[nH]c(C(=O)OC)c3)=O)C2)[nH]1 38589,C1(c2n(CC)nnn2)(NCC2CCC3(CCCC3)C2)CC2(C1)CC(C)(C#N)C2 38590,Cc1cc(=NCC2(O)CCCN(C(C3(n4cncn4)CC3)=O)C2)[nH]c(C(C)C)n1 38591,CCC(CC(=O)N(CCNC(c1c(C)nnn1CC)=O)C1CC1)C(C)(C)C 38592,C1(CCCCNC(=O)CC2COCCO2)CCN(C(=O)CC2C=CCC2)CC1 38593,c1(NC(C(C)OCC)=O)c(C(=O)NC2CCN(C(C)C)C2)cnn1C 38594,N1(C(c2c(COC)n(-c3ccccc3)nn2)=O)CC=C(c2ccc(Cl)c(Cl)c2)CC1 38595,C1(NC(c2c(C)onc2CO)=O)CC2CC1N(C(=O)C(=CC1CCCCC1)F)C2 38596,C1(c2n(CCOCC)nnn2)(NCc2ccccc2C)CSC(C)C1 38597,c1(CNC(C(C)OCCOC)=O)cccc(CN(C)C(c2cscc2OC)=O)c1 38598,N1(C(=O)C(N2CCc3cccnc3C2)=O)Cc2cc(Br)ccc2C2CC1C2 38599,c1(CCC(=O)N(CCC)CCNC(C2CC3CC2C3)=O)ccc2c(c1)CCCO2 38600,c1(C(=O)OC(C(=O)NC(C)C2CC2)C)nc(C(F)(F)F)cs1 38601,CC1(C)Cc2cccc(CCNC(=NCCCCl)NCCC3CC=CCC3)c2O1 38602,N1(C(C(CC)(C)O)=O)CC2(CC2)CC1C(=O)Nc1ncc(Br)nc1C 38603,C#CCC(C(=O)N1CCC1c1cn(CC2(n3ccnc3C)CC2)nn1)SC.OC 38604,N1(C(c2cnc(C(C)C)[nH]2)=O)CC2C(N(C(=O)COc3ccc(Cl)cn3)C)C2C1 38605,C=CC(C)(CCOC)C(=O)NC1CN(C(=O)Cn2cc(Cl)cn2)CC1C(F)F 38606,C1(NC(COCCNC(COCCC=C)=O)=O)CCC(C(C)O)CC1 38607,C1(CNC(Cc2ccn(CC)n2)=O)CN(C(=O)C(c2nc(C)cs2)C)CCO1 38608,Cc1cccc(C(CNC(c2ncncc2C)=O)NC(c2cn[nH]c2)=O)c1 38609,C1(C(=O)NC(c2ccccn2)C)CCN(C(c2ccc(=O)n(C)c2)=O)C(C)(C)C1 38610,C(C(C)(CC(C)C)NC(=O)Cn1sc(=O)c2ccccc12)NC(CC=CCC)=O 38611,CCC(C)CCCC(=O)NCCCCC1CN(C(=O)CCC2OCCO2)C1 38612,c1(N2CCC(CN(C)C(C3CC3C(N)=O)=O)CC2)nc(Cl)ncc1C(N)=O 38613,N1(C(c2c(C)ccs2)=O)CCCCC1C(=O)Nc1cccnc1C(N)=O 38614,c1(C(N2CC(NC(CC3(C)CC3)=O)C2)=O)ccc(-n2cnnc2)cc1 38615,N1(C(CCC2CCCC(=O)N2)=O)CCCN(C(C23CSC(C2)C3)=O)CC1 38616,c1(C(=O)NCCN(CCOC)C(C2CC=CCC2)=O)csc(O)n1 38617,C1(C(=O)NC(CC#C)CC)CCCCN1C(=O)Cc1cc(C)on1 38618,Cc1csc2ncc(C(=O)NC34CCCC3N(C(=O)COCCC(C)C)CC4)n12 38619,C1(CN(C(C2CCCC(C(N)=O)C2)=O)CC)CCN(C(=O)CCF)CC1 38620,n1(CC)ccc(CC(=O)NC(Cn2ccnn2)C(=O)N2CCC2(C)CCO)n1 38621,Cc1ccc(C)c(N(C(c2nocc2C)C(=O)NC2CCOC2)CC(C)C)c1 38622,c1(CN2CC(C(N3CCC(F)(F)C3)=O)SCC2)c(O)cccc1O 38623,C1(NC(c2c(C)cno2)=O)CCC(CNC(=O)CN2CCOCC2=O)CC1 38624,C1(C)(C(=O)NCCCCN(C)C(C2CC2c2ccccc2)=O)CC(C2CC2)=NO1 38625,CC1CCN(C(=O)Cc2cnns2)CC1NC(=O)C(=CC1CCCCC1)F 38626,c1(C(=O)NCc2c(C(N3C(C(C)C)CC3)=O)occ2)ccc2nccn2c1 38627,Cc1c(Cl)cc(CNC(c2ccc(Br)cc2CO)c2nnnn2C(C)C)cc1I 38628,C(CC(C)(C)C)(C(=O)N1CCC(CO)(NC(=O)CSC(F)(F)F)C1)OC 38629,C1(CNC(CC=CC)=O)COCCN(C(C2(C)CC=C(C)CC2)=O)C1 38630,C1(C(N2CC(N(C)C(c3cnc(CC4CC4)s3)=O)C2)=O)CCc2nncn2CC1 38631,Cc1ccc(CC(N2CCC(C(C)NC(=O)C(C)CCO)C2)=O)cc1 38632,c1(N2CC(CC=C)(NC(=O)CC3C=CCC3)C2)ncnc2[nH]c3ccccc3c12 38633,c1(NC)cccc(OC)c1C(N1CC(CO)(NC(C2CCCC2C)=O)C1)=O 38634,C1(CN(C(=O)CCCc2ccncc2)CC)CCCN1C(=O)CCCC1CC1 38635,Cc1nn(C(C)(C)C)c(C)c1C(N1CC2CN(Cc3cc(O)ccc3F)C2C1)=O 38636,C12(C(N3CCN(C(C(C)=CC)=O)C(CC(F)F)C3)=O)CCC(N=[N+]=[N-])C1C2 38637,N1(C(c2cc(C)no2)=O)CC(CNC(=O)CCCc2cnn[nH]2)C(C(F)(F)F)C1 38638,c1(SC)cccnc1C(=O)NCCC1CN(C(c2ccn(CCF)n2)=O)C1 38639,Fc1cc(SCC2CC(CCC(=O)N)NC2)ccc1Br.c1(C)ccccc1 38640,CCCCC(O)C(=O)NCC(C(C)C)NC(c1cnn(CCOCC)c1)=O 38641,c1(OC)ccc(NC(C2CC2C2CN(C(=O)Cn3nccc3C)C2)=O)cc1C 38642,c1(OC)cc(C(=O)NCC2(NC(C3CCN(C)C3C)=O)CCOC2)ncn1 38643,C1(C)(NC(C(c2ccccc2)OC)=O)CCCN(C(c2cccnc2NC)=O)C1 38644,C(C(C)(O)CC(=O)NCC1CCC1NC(=O)CNC(c1ccoc1C)=O)OC 38645,C(=O)(C(CCC)C(=O)N(C(C)C)CC)NC(CCCC)C 38646,CCCC(C#N)C(=O)NCCN(C(=O)C(CSC)OC)C(C)C 38647,N1(C(c2c(C)c(N)cnc2)=O)CC2CCCC2(NC(=O)Cc2ccccc2Cl)C1 38648,N1(C(C(C)N(C(=O)OC(C)(C)C)C2CC2)=O)CCC(N2CCSCC2)CC12CC2 38649,C1(NC(CCC=CC(C)C)=O)CC(C(=O)NCCN2CCCNC2=O)C1(C)C 38650,c1(OC)ncnc(C)c1C(N1CC(C(C)NC(=O)CCCCC2CC2)C1)=O 38651,c1(C(Cc2nc(-c3cccc(C)c3)sc2)=O)cc(F)cc(-c2nn[nH]n2)c1C 38652,C=CCCCCCCC(=O)NCC(C)NC(c1c(N)cc(F)cc1F)=O 38653,c1(OC)ccc(C(N2CC3CC(NC(=O)C(C)n4cncn4)C3C2)=O)cc1N 38654,c1(OC)cc(Cl)cc([N+](=O)[O-])c1NC(C1CC1NCc1cc(F)c(F)c(F)c1)=O 38655,CC1CC2(CCN(C(=O)CC3CCCCO3)CC2)CN1C(c1nn[nH]c1Cl)=O 38656,c1(C(N2CC=CC(NC(c3cc(OC)ncn3)=O)C2)=O)cc2cccc(Cl)c2o1 38657,c1(C(N(CCC)CCNC(C2CCC2C)=O)=O)coc2ccc(OC)cc12 38658,C(C(=O)NN1CCSCC1)(C1CCCCC1)NC(=O)OC(C)(C)C 38659,c1(CC)c(OC)cccc1C(=O)NC(CNC(C1COCCC1(F)F)=O)C(C)C 38660,N1(CC(=O)N(CCC(=O)NCCC2CC2C)C(C)C)CC2CCC1C2 38661,N1(C(c2ccncc2)=O)CCC2(CCCN(C(c3ccc(Cl)nc3O)=O)C2)CC1 38662,N1(C(C(C2CCOC2)OCC)=O)CC2(CCCC2NC(=O)CC2CC2)C1 38663,N1(C(c2c(C)cc(N)cn2)=O)CC2COCC2(C(N2CCC(O)(C(N)=O)C2)=O)C1 38664,c1(OC)cc(OC)c(C(N2CCN(Cc3cccnc3Br)C3CC23)=O)cc1Br 38665,CCC(CC(F)F)C(=O)NC1CCCCN(C(C2CCCN(CC(C)C)C2)=O)C1 38666,CCCCC(C(=O)NCC1CC(OCC)C1)NC(c1ccoc1CC)=O 38667,Cc1ccc(Cl)c(O)c1C(=O)NCCCCC(C)NC(c1c[nH]nc1C)=O 38668,N1(C(=O)CC2=CCCC2)CCC2C(CCCN2C(c2cnc(C3CCC3)s2)=O)C1 38669,c1(C(=O)NCC(C)CN(C)C(C2CC(C(C)(C)C)=NO2)=O)ccc2n[nH]cc2n1 38670,C(c1cnc(C)nc1O)=CC(=O)N(CCNC(C=CCCC=C(C)C)=O)C1CC1 38671,c1(C(=O)NC2CCN(Cc3c(C)ccs3)CC2)cc(F)cc(Cl)c1 38672,c1(C(N2CCC(N(C(=O)CNC(C3CCC3)=O)C)C2)=O)ccnc(O)c1 38673,C12(OC)CCCCC(C(=O)N(CC(C)NC(=O)CCn3ccccc3=O)C)(C1)C2 38674,C1(C)(NC(CCSC)=O)CCN(C(=O)C(C(C)C)c2cnc(C)s2)CC1 38675,c1(NC(Cc2cccc(C(C)N)n2)=O)cc(Br)c(F)cc1F 38676,C12(C(=O)NC3CN(C(C4CCN(S(C)(=O)=O)C4)=O)C3)CCCC(=O)N1CCC2 38677,c1(C(N2C(C3CCN(C(C(CC=C)C)=O)C3)CCC2)=O)ccc(C)c2cccnc12 38678,N1(C(CC2C(C)(C)C2)=O)CCC(NC(c2cc(N)c(O)c(F)c2)=O)C(F)(F)CC1 38679,C1(F)(C(=O)NCc2nc(CNC(C(C)(F)F)=O)sc2)CCCOC1 38680,CN1CCC2CN(C(C3CCN(C(c4cc(Cl)ncn4)=O)CC3O)=O)CC2C1 38681,N1(C(CNC(C(CC)C)=O)=O)CC=C(C(=O)NCCC(=O)NC2CC2)C1 38682,Cc1nc(Cl)[nH]c(=NCC2CC(CNC(=O)CCc3ccn(C)n3)CO2)c1Cl 38683,C1(NC(C(c2n(C)cnc2)O)=O)CC2(CCC(NC(C3(C)CC3(F)F)=O)CC2)C1 38684,c1(C(=O)NC2CC(C)(NC(CCC(C)OC)=O)C2)csc2cc(C)ccc12 38685,C(CN=c1[nH]cnc2c(Cl)cc([N+](=O)[O-])cc12)C1(O)CCN(C(=O)OC(C)(C)C)C1 38686,c1(CC)cc(C(N2CCC(NC(c3cc(O)ncn3)=O)C2)=O)ccn1 38687,Cc1cc([N+](=O)[O-])c(Cl)cc1S(=O)(=O)CC(C)NC1(C(F)(F)F)CC2(C1)OCCO2 38688,n1(CCC)cc(Cl)c(C(=O)NC23CC2CN(C(=O)C(C)CC)C3)n1 38689,c1(COC)nccc(=NC2CCC3CN(C(c4n[nH]c(C)c4O)=O)CC23)[nH]1 38690,Cc1nnc2n1CC(C(=O)NCC1CCC1NC(=O)C=CCO)C2 38691,C(=O)(CCCC(C)(C)NC(c1n[nH]c(C)c1O)=O)N1CCC(OC)C(C)C1 38692,C(=O)(C(C)(C)S(C)(=O)=O)NC(CC1CN(C(Cn2c(=O)ccc(C)n2)=O)C1)C 38693,N(C1CCCn2cnnc21)C(CC(C)N(C(C(C1CCCCC1)C)=O)C)=O 38694,c1(C(N(C2CC(NC(C3CC=CCO3)=O)C2)C)=O)cc(Cl)cnc1O 38695,c1(OC)ccc(C(CCO)NCC2CCC3(CC3)C2)cc1 38696,N1(c2ccnc(NC(CC)COC)n2)CC2CCC(OC)C2C1 38697,C(=O)(C1Cc2ccccc21)NC(C1N(C(c2c(CC)ocn2)=O)CCC1)(C)C 38698,N1(C(CCSCC)=O)CCC(CNC(c2cnnc(C3CC3)c2)=O)C(F)(F)CC1 38699,C1(C)(COC)CCCN(C(=O)Cn2cc(CNC(C3(C#N)CC3C)=O)nn2)C1 38700,C1(CCNC(CCCOC(C)=O)=O)CCCN(C(=O)C(N2CCCC(O)C2)C)C1 38701,C(=O)(CCCCC(C)(C)C)N1CCC(NC(c2c(CC(C)C)onc2)=O)C1 38702,c1(OC)cc(COC(=O)C(C(C)C)c2ccc(F)cc2)c(-c2cnn(CCl)c2)cn1 38703,N1(C(COC2C(CC)CCCC2)=O)CCN(C(c2ccnnc2O)=O)CC1C 38704,C(CCCCCC(=O)Nc1cnn2c1OCCC2)NC(COCC#C)=O 38705,C(=O)(C1=C(C)S(=O)(=O)CC1)N1CC(NC(COC)=O)C(F)C1 38706,N1(C(C2C(=C)C2)=O)CCC2(CCCCN(C(C3CC4CCC(C3)C4(F)F)=O)C2)C1 38707,N1(C(C(C)=C(C)C)=O)CC(C(=O)NCC(N)=O)OC(C)C1 38708,N1(C(c2nc(C)n(C)n2)=O)CCC(C2CCCN(C(=O)C(C)(O)C3CC3)C2)C1 38709,N1(C(C(CC)C)=O)CC2(CC(NC(c3coc(Br)n3)=O)c3nccn32)C1 38710,C(=O)(C#CC(C)(C)C)N1CC(OC)C(NC(c2ccccc2SC(C)C)=O)C1 38711,c1(CC)nn(C)c(CC)c1C(=O)NC1CCC1CNC(=O)C=CC1CCCN1C 38712,N#Cc1c[nH]c(=NC(=O)NCc2nnc(-c3cccc(F)c3)s2)cc1Cl 38713,C(CCCCC(=O)N1CC(O)CC1(C)C(=O)N(C)Cc1ccncn1)OCC 38714,c1(C(N2CCN(CC(C)NC(C3C(=C)C3)=O)CC2)=O)nn(C)cc1[N+](=O)[O-] 38715,C1(C2CCCN(C(c3ccn4nccc4n3)=O)C2)(NC(CC(C)SC)=O)CC1 38716,C12(NC(C(CC)SC)=O)CCCC1N(C(c1c(OC)cccc1F)=O)CC2 38717,N1(C(C(CC)OCC)=O)CCCC(C2CN(C(c3cccc4[nH]ncc34)=O)C2)C1 38718,Cn1cc(C2CC2C(=O)NC2CCN(C(C3(O)CCOC3)=O)C2)cn1 38719,c1(C(C)C)conc1CC(N1CC(CC(C)NC(c2c[nH]nc2C2CC2)=O)C1)=O 38720,C1(C(=O)NCCNC(CC)=O)C=CCCN1C(=O)CC1(C)CC1 38721,N1(C(C=C(C)C)=O)CCC2(CCC2)C(NC(=O)CCOc2cccc(Cl)c2Cl)C1 38722,N1(C(CCc2nnc(C)n2C)=O)CCCC(NC(=O)CC2CC(C(F)F)C2)C1C 38723,c1(NCC)ccc2c(c1)OCO2.c12cccc(c1)N(C(C)=O)C2 38724,C(=O)(C1CC(=O)Nc2ncn(C)c21)NCC(C)CNC(C1C2(CC2)C12CC2)=O 38725,CCCC(CCC)CC(=O)NC(CCC1CC1)C(=O)N1CCC1CC(=O)NC 38726,N1(C(c2cc(C)c(F)cc2)=O)CCC2CCN(C(C3CCCC3(C)C)=O)C2C1 38727,c1(C(N(C2CC(C)(NC(=O)CC3CCC3)C2)C)=O)ccc(NC(=O)C2CC2)cc1 38728,N1(C(C(C(C)O)N(C)C)=O)CCOCC(C)(CNC(c2coc(CO)c2)=O)C1 38729,c1(C(CNC(c2ccc(OCCOC)nc2)=O)C)ccc2cc[nH]c2c1 38730,C(C)(CNC(C1(C(C)(C)C)CCCCC1)=O)(C(C)C)NC(Cc1nnc(C)o1)=O 38731,C(=O)(C(C)(C)CCCNC(=O)C(F)C1CCOC1)NC(C)Cn1cnnc1 38732,N1(C(C2CN(C(C(CC)(C)COC)=O)CC2SC)=O)CCOC2C(O)CC12 38733,CC(CO)CCCNC(C1CCCN(C(=O)Cc2cccc(O)c2)C1)=O 38734,C(=O)(CCCCC(C)C)N1CCC(OC)(CNC(C2COCCC2(F)F)=O)CC1 38735,C1(C(N(C(CNC(C2N(CC#C)CCC2)=O)C)C)=O)CCc2nncn2C1 38736,C(=O)(C1=NN(C)C(=O)CC1)NC1CCN(C(CC)=O)C(C2CC2)C1 38737,c1(C(N2CCC(OCC)C2)=O)cncc(-c2cccc(CC#N)c2)n1.OCC 38738,C(Cn1cncn1)(C(=O)N(C)CC1CCOCC1)NC(CSC)=O 38739,N1(C(=O)Nc2nccc(OCC)c2)CCCN(C2CC2)CC1 38740,C1(CC(=O)N(CC(C)C)CC(C)NC(=O)CC=CC(C)(C)C)OCCC1(C)C 38741,N1(CC(=O)NCc2cc(C(F)F)ncn2)CCC(C(F)(F)F)C(CO)C1 38742,c1(C(=O)NCC2(F)CCN(C(Cc3c(C)nsc3)=O)CC2)ccc(N)c(F)c1F 38743,C1(C)(C(=O)NC2CCC(C)N(C(C3C=CCCC3)=O)C2)Cc2ccccc2C1 38744,C1(C)(CNC(C(C2CC=CCC2)NC(CN(CCOC)C)=O)=O)CCCO1 38745,Cc1ccc(C(N2CC=CC(NC(=O)CC3CCN(C)C3)C2)=O)c(Cl)c1C 38746,C1(NC(C=CCCCCC)=O)C2CN(C(c3ccc(N4CCCCC4)s3)=O)CC12 38747,c1(C(=O)NC(CNC(c2ccc(C)cn2)=O)(C)C)cc(C2CCC2)n(C)c1C 38748,Cc1nnc(N2CCCC2c2csc(C)n2)n1CC1CCN(C(C)(C)C)CC1 38749,C(CCCC(=O)N1CCC(C(C)NC(=O)CC2(C)CCOCC2)C1)N(C(C)C)C 38750,O(NC(=O)CC1(NC(=O)Cc2ccns2)CCCC1)CC(=O)NC(C)C1CC1 38751,N1(C(C2C(C)(C)CCO2)=O)C2CCC(C(=O)NC3CCCCCC3F)C1CC2 38752,c1(C(=O)NC2C(C)CCN(Cc3c(OC)nsc3)C2)ccc(Br)c(F)c1F 38753,c1(CNC(N2CCC(C)C2CO)=O)ccc2c(c1)CN(C)C2 38754,C(CC(O)C(=O)NC1CCCC1NC(C1(C2CCCO2)CC1)=O)N(C)C 38755,c1(C(=O)Nc2ncc[nH]2)cc2ccc(-c3ccc4c(c3)CNC4=O)nc2[nH]1 38756,N1(C(COCCCC#C)=O)CCCCCC1CNC(C1CC12CC(F)(F)C2)=O 38757,c1(OC)cccc(C(CF)NC(=O)Nc2cnc(C3(C)OCCO3)s2)c1 38758,C1(C(N2CCC(CN(C)C(c3ncc(F)cc3N)=O)CC2)=O)CCCC(F)(F)C1 38759,CC1(C)CN(C(=O)CCCC(=O)C2CC2)CC1NC(c1c[nH]cc1Br)=O 38760,C(=O)(N=c1[nH][nH]c(C)c1Cl)C1C(C)(C)CCN(C(C(C)NC(C)=O)=O)C1 38761,c1(C(C)C)ccc(C(=O)NCC2CC(F)(CNC(C3(C)CC3(F)Cl)=O)C2)cc1 38762,C1(c2nnnn2CC2CC2)(NC(c2cccc(Br)c2)CC)CCCC(F)(F)CC1 38763,c1(CNC(c2c(C(C)(C)C)con2)=O)ccc(OC(F)F)nc1 38764,N1(C(Cc2ccc(C#C)cc2)=O)CC2CCC1CC2NC(c1c[nH]nc1CC)=O 38765,C1(CNC(C2(C)CCCC2)=O)CCCCCN1C(=O)C(F)CC1CCCC1 38766,c1(C(N(CC(N2CC(O)(COC)C2)=O)CCC)=O)ccnnc1O 38767,c1(N(CC)CC)ccc(C(=O)NC(C)COC2CCOCC2)cc1 38768,CC1CCN(C(C2CCCCC2O)=O)CC1CNC(C1(c2ccccc2)CC1)=O 38769,C1(NC(C(C)=CC)=O)CC2(CCCN(C(C3CC3CCC)=O)C2)C1 38770,C1(C(N2CC(C(CC)CC)C2)=O)(NC(c2ccn(CCF)n2)=O)CCSC1 38771,Cc1ccc2sc(NC(=O)NCc3cc4cccc(C)c4o3)nc2c1 38772,C1(C(=O)NCCCOCCNC(=O)C=CC2CCCO2)CC(C2CCCC2)C1 38773,C1(C(N(CCCNC(c2ncoc2C2CC2)=O)C2CC2)=O)CCCC(O)C1 38774,C(=O)(CCS(C)(=O)=O)N(CC(C)CNC(=O)CC1CCCC(C)C1)C 38775,N1(C(c2sccc2COC)=O)CCC2CN(C(c3cncc([N+](=O)[O-])c3)=O)C2C1 38776,N1(C(C=C(COC)C)=O)CCCOC(CNC(=O)CC2CC3CCC2C3)C1 38777,C1(C(N2C(C3CCN(C(C4CCCN4C4CC4)=O)C3)CCC2)=O)CC(=O)N(O)C1 38778,c1(CC(=O)Nc2cccc(CC)n2)n[nH]c2cc(-c3ccncc3OC)ccc12 38779,CC1(C)NC(=O)C2(CCN(C(=O)NCc3cc(C4CC4)no3)CC2)O1 38780,C(=O)(CCC(C)CN(C)C)N1CCC(CC(C)NC(C(CC=C)C)=O)CC1 38781,N1(C(C(N2CC(C)C2)C)=O)CCC(C)(C)CC1C(=O)NCC1CCC(C2CC2)O1 38782,CC1(c2nc(-c3cnn(CCO)c3)nn2-c2ccc(Cl)cc2)CCCC(F)(F)C1 38783,c1(COC(C2(C(N3CCN(CC)CC3)=O)CC2)=O)ccc(On2cccn2)cc1 38784,n1(CC)cc(NC(=O)CC(C)(C)N(C)C(c2cncc(C#N)c2)=O)ccc1=O 38785,Cn1ncc(C(=O)NC(CNC(c2csc(=N)[nH]2)=O)C2CC2)c1S(N)(=O)=O 38786,c1(OC(C)C(N)=O)cccc(NC(=O)C(O)Cc2cnc[nH]2)c1 38787,Cc1c(Cl)ccc(C(N2CCC23CN(C(=O)Cn2nc(Cl)ccc2=O)C3)=O)c1Cl 38788,C(=O)(CCC(C)(C)[N+](=O)[O-])NCC(C)CNC(=O)CSCc1ccccn1 38789,O=C1Nc2ccc(C(N3CC4CN(C(=O)CC5(O)CCC5)C4C3)=O)cc2C1=O 38790,N1(C(C(CC)N(C)C)=O)CCN(C(=O)C(N)=O)C(c2cn[nH]c2)C1 38791,C1(C2CCN(C(=O)CN3CCCC3C)CC2)(NC(CC(CC=C)(C)C)=O)CCC1 38792,C(CCCCC(=O)N1CCC(C)(C)C1C(=O)NC(C)C(=O)NC(C)C)SC 38793,CCC(O)C(F)(F)C(=O)N1CCC(C(C)NC(=O)CCCn2ccnc2C)CC1 38794,N1(C(CSCC)=O)CC(C)(C)OC2(C1)CN(C(c1cc(F)cc3ccoc13)=O)C2 38795,C1(NC(Cn2c(=N)[nH]nc2)=O)CCC2(CCOCC2)C1 38796,Cc1ncc2ccccc2c1C(=O)NC1CC1CNC(c1ccc([N+](=O)[O-])s1)=O 38797,C1(NC(c2nnn(CC)c2C)=O)COCCN(C(=O)COCC(=O)OC(C)(C)C)C1 38798,CCCC(C(=O)Nc1cnccc1OC)NC(=O)OC(C)(C)C 38799,N1(C(=O)Cn2ncccc2=O)CC2CCN(C(=O)CCc3ccncc3)C2C1 38800,C1(C(=O)NC(C#C)CC2CC(NC(=O)CCCOCCOC)C2)OCCC1(C)C 38801,n1(C(C)C)nncc1C(=O)NCC1CN(C(C2CNC(=O)N2)=O)C1 38802,c1(C2(C(=O)NCCC(C)(C)N(C)C(C3COCCO3)=O)CCC2)c(F)cccc1F 38803,CCC(CCCC(=O)NCC(C)CN(C)C)NC(=O)C(n1ccc(C)n1)C 38804,c1(CNC(c2ccc(CNC(c3cc(CC)[nH]n3)=O)cc2)=O)nnc2n1CCC2 38805,C1(COC)(NC(=O)CC(C)C2CCCO2)CN(C(C2(C(N)=O)CC2)=O)C1 38806,c1(C(=O)NCC2C(CNC(Cn3c(C)nnn3)=O)C2)ccc(NC=O)cc1 38807,C(=O)(CCCS(C)(=O)=O)N(CCCNC(c1ccc(F)c(C(F)F)c1)=O)C(C)C 38808,Cc1[nH]c2ccccc2c1C(=O)NCC1CN(C(C2C3CCC23)=O)CCN1C 38809,N1(C(Cn2nnc(C)n2)=O)CCC2(CCCCC2NC(C2CCC(=O)N2C)=O)C1 38810,O=C(NN1CCSCC1)C(=O)N1CCCCC1c1ncc[nH]1 38811,C1(OC)CC2(CCN(c3ccnc(-c4ccccn4)n3)C2)C1 38812,C(=O)(CC(C)CC(C)(C)C)NC1CC(CN(C2CCCC2)C(=O)COC)C1 38813,N1(CC(=O)NC2(F)CC(NC(COCc3onc(CC)n3)=O)C2)CC2C=CC1C2 38814,Cc1ccc(F)cc1C(F)(F)C(=O)N1CC(CNC(c2coc(C3CC3)n2)=O)C1 38815,c1(CC)ccc(C(N2CC(NC(c3ccc(CN(C)C)[nH]3)=O)CC2C)=O)cn1 38816,C1(CO)(NC(=O)Cn2nnc(-c3ccccc3)n2)CCN(C(=O)CCN2CC2)CC1 38817,c1(SCC)nc(C)c(CC(=O)NC(C)(C)CCCNC(C2(C)CC2(F)Cl)=O)s1 38818,c1(NC(C2CN(S(CCC(=O)OC)(=O)=O)CC(F)C2)=O)ccc2c(n1)NC(=O)CC2 38819,c1(CCC(N2CCC(C(C)NC(c3c(CC)occ3)=O)C2)=O)cccc(C#N)c1 38820,CCC(O)(CC(=O)NCc1ccc(N2CCCC2)cc1C)c1ccccc1 38821,C(CC(CNC(=O)COC1CC=CC1)NC(C1CCCN1C(C)C)=O)OC 38822,C(=O)(C(C)C(O)CC)NCc1cc(C(=O)NCCC(=O)NCC)n[nH]1 38823,C1(CNC(c2cc3cc[nH]c3cn2)=O)CC2CCC1N(C(=O)Cc1cnoc1)C2 38824,c1(C(N2CCC(NC(=O)C=CC3CCOC3)C2)=O)ccc(C(F)F)nc1O 38825,C(=O)(C(F)(F)C(C)(C)O)N1CC2C(NC(C3CN(C)C3)=O)(CC2)C1 38826,C1(C(=O)NCCOC2CCN(C(C3C(OCC)C3)=O)C2)CCC(C)CC1 38827,C1(C#N)(C(=O)NC(CC)CNC(C2CC(=O)N2)=O)CC12CCCC2 38828,N1(C(C(CC(C)C)F)=O)CC2C3CCC(C2C1)N(C(=O)CC1OCCC1(C)C)C3 38829,CC1CCC(NC(=O)Cc2ccsc2)CN1C(c1cc(-c2cccn2C)[nH]n1)=O 38830,c1(C(C(N2CCC(F)(CNC(C3CC=CC3)=O)C2)=O)O)cc(F)c(F)cc1F 38831,c1(C(N2CC3C(C(=O)NC(C)CS(C)(=O)=O)C3C2)=O)cn(C)c(=O)cn1 38832,n1(C(C(=O)NC(CC)CNC(c2cnccc2C)=O)C)cnc2ccccc12 38833,Cc1nc2cc(C(=O)NC(CNC(C3CCCC(=O)N3C)=O)C(C)C)cnc2[nH]1 38834,C1(C(N(CC(CCC)O)C)=O)CCC(C(C)C)N1C(C1CCCC(O)C1)=O 38835,CC1CC(C(=O)N(C)CCOCCNC(=O)C(C)(C)C2CCCCC2)C1(C)C 38836,Cc1ccc(C=CC(=O)NCC2(F)CC(NC(C3CCSC(C)C3)=O)C2)cc1C 38837,CCCC(C)CC(=O)N1CCC(C(C)C(=O)NC(c2nc[nH]n2)C2CC2)CC1 38838,c1(C2C(C(=O)NCC3(O)CN(C(C(c4ccsc4)=O)=O)C3)CC2)ccc(F)cc1 38839,C(=O)(CC(F)F)NCC1CC(NC(C=C(C)I)=O)C1 38840,N1(C(C(CC)C)=O)CC2(CC(NC(=O)COc3c(C)cccc3C)C2)C1 38841,c1(NC(CC(=O)NC)C)nc(N2CCN(C3CCSC3)CC2)cc(C)n1 38842,c1(C(N2CCN(C(CN3CC(C)C3)=O)CC2)=O)cc(Cl)cc([N+](=O)[O-])c1 38843,c1(C(N2CCCC(N(C(C(CSC)O)=O)CCO)C2)=O)cc(F)ccc1F 38844,C(=O)(C1=CCCCC1C)NCC1N(C)CCN(C(c2cc(C)on2)=O)C1 38845,C1(COC)CCN(C(c2nc[nH]n2)=O)C(C(=O)N(CC(C2CCC2)OC)C)C1 38846,C1(C(N2CC(C(=O)OC)C2)=O)COCCC1NC(=O)CSC(C)C 38847,C1(NC(c2n(CC=C)ccc2)=O)CCCCC1N(C(=O)Cn1nccc1C)C 38848,c1(-c2n(CN(CC(=C)C)CC)ccn2)ccc(Cl)cc1 38849,C(C(COC)CC(=O)Nn1nnc(CC2CN(C(=O)CC(C)(C)O)C2)n1)OC 38850,C(CC(F)F)(C(=O)NC1CC2C(C1)C2(F)F)NC(CC1(OCC)CCC1)=O 38851,c1(C(=O)NCC(CC)NC(=O)C=C(C)c2cnn(C)c2)cc(C)cc([N+](=O)[O-])c1 38852,Cc1cc(C(N2CCC(C)(CCNC(c3c[nH]nc3C(F)F)=O)C2)=O)cc(C)c1 38853,c1(OCCC(=O)NC(C(C)NC(c2ccncc2)=O)C)ccc(CC#N)cc1 38854,C1(C)(NC(CC2CC(CC)OCC2)=O)CCN(C(c2sncc2C)=O)CC1 38855,c1(CC)cc(C(=O)OC)ccc1NC(N1CC(O)CC1Cn1ccnn1)=O 38856,c1(C(N2C(C)CC(NC(c3cncc(COC)c3)=O)C2)=O)ccc(N)c(Cl)c1O 38857,c1(N2CC(C(C)NC(=O)CCC3CC3(Cl)Cl)OCC2)cc(-n2ccnc2)ncn1 38858,c1(C(=O)OC)ccc(C(F)(F)F)nc1N(CC(C)NC1CC(C)(F)C1)C 38859,c1(-c2cc(NCc3c(C)c4c(s3)cccc4)ncc2)ccc2c(c1)OC(C)(C)O2 38860,C1(CCCC)CN(C(=O)CNC(=O)C2CC2)CCN1C(C1CC12CCCCC2)=O 38861,C(C(F)(C(=O)NCc1coc(C)n1)C(C)C)NC(C(CC#C)O)=O 38862,c1(CC)cc(CC(=O)NC2CCN(C(=O)Cc3sccc3Br)C2)n(C)n1 38863,Cc1cccc(N(C2CCCSC2)CCOc2cncc(-c3cnn(C)c3)c2)c1 38864,C(C(=O)NCC1(CO)CC1)(C(C)O)NC(C)=O.C1(C=O)C2CCC1(c1cscn1)C2 38865,C(=O)(C(C(C)C)NC(N)=O)NC(c1cn(Cc2c(C)nn[nH]2)nn1)C(C)C 38866,c1(COC)conc1C(=O)NCC1CCC(NC(C2CCN(C3COC3)C2)=O)C1 38867,Cc1c(C(=O)NC2CC(C)N(C(=O)CSc3nnnn3C)C2)noc1C1CC1 38868,Cc1c(NC(=O)NC(c2cnn(C)c2)CO)cccc1Cl 38869,N1(C(C2(CC#C)CCCO2)=O)CCC(C)N(C(=O)CC2(CO)CCC2)CC1 38870,C1(N(C(=O)CC2CC2(Cl)Cl)CC)CCN(C(C2CCC2C(F)F)=O)CC1 38871,N1(C(=O)NC(C)CCn2cncn2)CC(F)(CF)C1 38872,C(=O)(C(CCC1CCC1)NC(c1cnsc1)=O)NC1(CC(C)(C)C)CC1 38873,CCCCC(CNC(=O)CN(C1CCC1)C)NC(=O)CC(C)C 38874,N1(C(C=C(CC)C)=O)CCC2CN(C(c3cc(CC4CCC4)c[nH]3)=O)CC2C1 38875,Cc1cc(CNC(C)COCc2ccccc2)ccc1[N+](=O)[O-] 38876,N1(C(C2CC(CN)C3CC23)=O)CCC(O)(C2(C(=O)O)CCC2)CC1 38877,C(C(C(=O)N(CC(=O)NCCC)C)C(C)C)NC(C1(CC=C)CCC1)=O 38878,Cc1ccc(C(N2CCN(C(=O)CC3=NNC(=O)C3)C3CC23)=O)c(F)c1F 38879,S(=O)(=O)(CCC(=O)NC1CCN(C(C2CCN(CC(C)C)C2)=O)CC1F)NC 38880,CC1CN(C(=O)CN2CCN(C(C3CC3c3ccco3)=O)CC2)CC(C)(C)O1 38881,Cc1cnc(C(N2CCC(c3nccs3)C2)C(=O)OC(=O)NC(C)(C)C)c(C)c1 38882,c1(C(=O)NCC2C(CNC(C(C3CC3)SC)=O)C2)cn(CCCF)nn1 38883,c1(CC(N2CC(CC(C)NC(c3ccc(C(N)=O)s3)=O)C2)=O)ccccc1O 38884,c1(C(C)NC(c2nnnn2C(C)C)c2ccns2)ccc(OCC#N)cc1 38885,c1(C(C)C)cnc2cc(C(N3CCC(CNC(=O)CO)C3)=O)[nH]c2c1 38886,c1(OCCC(C)C)ccc(C(=O)NCC(C)CNC(C2CCCN2C=O)=O)cc1 38887,c1(C(=O)NC2CC(C)N(C(=O)CC3(O)CCCC3)CC2)noc2cc(F)ccc12 38888,n1(CC)cc(N)c(-c2noc(CCC3CCN(C4CCCC4)CC3)n2)n1 38889,N1(C(C(COC(C)C)NC(Cc2c(C)nsc2)=O)=O)CCC2(CC2)C1 38890,C(=O)(CC(C)F)NCCC1(C(=O)NCCCC=C)CCC1 38891,C1(NC(C(F)=CCC)=O)CCCC12CCN(C(c1ccc(Cl)c(Cl)c1N)=O)C2 38892,c1(COC2CC(C(=O)OC)C2)cccc2c1CCC2 38893,c1(C(=O)NC2(CCOC)CCN(C(=O)C(C)=C(C)C)CC2)scc2c1CCCC2 38894,C1(C(N(CC(C)C#N)C)=O)OCCC1CNC(=O)C(=O)C1CCCC1 38895,c1(C(N2CCN(C(=O)CC(F)F)C3CC23)=O)cc2ncc(Br)cc2o1 38896,Cc1[nH]c(=N)[nH]c(=NCC2CCN(C3CCN(C)CC3)CC2)c1Cl 38897,N1(C(c2c(C)n(C)nn2)=O)C2CCC(C2)C1C(=O)NC1CC(C(F)(F)F)C1 38898,C(=O)(CCCCC(=O)OC)N1C(CNC(C(CC)C(C)O)=O)CCCC1 38899,C1(CCO)(CC)CN(C(=O)C(CO)NC(=O)CC2CC=CCC2)C1 38900,C(=O)(CCC(CF)CF)NC(C(=O)NC(C1C(C(=O)OC)C1)C)CC(C)C 38901,N(C(=NCC1COC1)NCC(F)F)CC1(CS(C)(=O)=O)CC1 38902,N1(C(Cc2c(F)ccc(C)c2)=O)CCCN(C(c2nc(C)ncc2Cl)=O)CC1C 38903,c1(C(=O)NCCCC(C)NC(C2CC3CCC2C3)=O)cc2sccc2s1 38904,N1(C(Cc2ccn(C)n2)=O)CCC2(CCC2)C(NC(c2cn(C)c(=O)n2C)=O)C1 38905,N1(C(C(CC)C(C)C)=O)CC(NC(c2ccc(C#N)c(C)c2)=O)CC12CCCC2 38906,CCCS(=O)(=O)C(C)C(=O)NC(C)(C)CN(C(=O)C=Cc1ncco1)C 38907,c1(SCCC(=O)NC2(CNC(C(CC)C)=O)CCOC2)c[nH]c2ccccc12 38908,CC(c1ccco1)=CC(=O)NC1(C)CC(NC(=O)CC#N)C1 38909,C=C(C)CC(C(=O)NCCn1ccccc1=O)NC(=O)CCC=CCC 38910,Cn1ncc(CNC(C2(O)CCOCC2)=O)c1C(=O)NC1CCCCC1F 38911,c1(C(C(=O)NC(Cc2c(OC)cccc2)C(C)C)OC)ccc(C#N)cc1 38912,C1(CCOC)(NC(c2ccc(Br)o2)=O)CCN(C(c2cccc(CC#N)c2)=O)C1 38913,c1(-c2cn(CC3N(C(C4CCC(C)O4)=O)CCC3)nn2)cc(=O)cc[nH]1 38914,Cc1ncc(Cl)cc1N(C(c1[nH]c(C)c(C(=O)NC2CCCCC2)c1C)=O)CCO 38915,c1(C(N2CCC(C(C)(C)F)C2)C(=O)NC)cccc(S(N)(=O)=O)c1 38916,C=CCCCCCC(=O)NC(C)(CC)CCNC(=O)CC1COCCN1CC 38917,N1(C(CCOCCOC(C)(C)C)=O)CC2(CCN(C(C3CCCC(C)C3)=O)C2)C1 38918,c1(OC)ccc(C(N2CCN(C(=O)Nc3ccc(F)cc3)CC2)C#N)cc1 38919,N1(C(c2c(OCC)c(Cl)sc2)=O)CCC(C2CCN(C(=O)C3=CCCOC3)C2)C1 38920,CS(=O)(=O)C1CCN(C(c2ccc(F)cc2)C(=O)NCC2CCOC2)C1 38921,c1(CNC(c2c(OC)csc2)=O)ccc(CCNC(=O)Cc2cc(C)cs2)cc1 38922,CSC1=C(C(=O)NC2CCN(C(=O)Cn3ccnn3)C(C)C2)CCCC1 38923,CC(C)(C)C(C)(O)CNC(C1CC1CNC(c1csnn1)=O)=O 38924,c1(CC)nonc1C(=O)NC(C)(CNC(c1ccncc1)=O)CO 38925,CC1(C(N2CCN(C(=O)Cc3cocn3)CC2)=O)C=CCCC1 38926,N1(C(c2ccc(CNC(CC(C)CN(C)C)=O)o2)=O)CC(CO)C(C)(C)C1 38927,c1(OC)c(F)ccc(F)c1C(=O)NC1CC(C)N(C(c2cn(C)cc2C)=O)C1 38928,C=CC1(C(N2CCC(C)(CC(=O)NCc3cncc(Cl)c3)C2)=O)CCCCC1 38929,C(=O)(CC1CCOc2ccccc21)NCC1N(C(C2CC(OC)C2)=O)CC(F)C1 38930,c1(C(=O)NC(CC(C)NC(=O)C=CC=C(Cl)Cl)C)cc2n(n1)CC1(CC1)C2 38931,Cc1cc(Cl)cc2cc(C(=O)N(c3cnn(-c4ccccc4)n3)C)[nH]c12 38932,C1(NC(C(CC)OC)=O)CN(C(c2cc(Cl)c(C)cn2)=O)C(C)(C)C1 38933,C1(C(=O)NCc2cc(CC)no2)CC(NC(=O)C(C)COC)C1(C)C 38934,c1(CCSCCC(N)C2CCC2)c(F)cccc1Cl 38935,CC1CC(NC(C2CC3CCC2O3)=O)CN(C(c2cccc(CC#N)c2)=O)C1 38936,c1(OC)cccc(C(N2CCC(N(CC(C)C)C(C3CC3(C)C)=O)CC2)=O)c1O 38937,C1(OC)CCCN(C(=O)C(CNC(=O)CCc2ncnn2C)OC)CC1 38938,CC1(C)C2CCC1(C(N1CCC(NC(=O)Cn3ncnn3)C(O)C1)=O)C2 38939,N1(C(C(C)(C)F)=O)CCC(NC(=O)Cc2cc[nH]n2)C(F)C1 38940,N1(C(C(n2cc(C)nc2)(C)C)=O)CC2CC(NC(C3CCS3(=O)=O)=O)C2C1 38941,c1(C(=O)OC)cc(=NCC(C)(C2CC2)NC(C2COC(C)C2)=O)[nH]c(Cl)n1 38942,c1(Sc2ncccn2)cccnc1NCC(F)(F)F.C(CC(=O)OC)N1C(=O)C1 38943,Cc1ccc(CCCN2CCCC2c2cnc[nH]2)o1 38944,c1(C(=O)NCC(CNC(=O)C(C)(C)C)OC)ncccc1N(C)C 38945,C(c1cncnc1O)=CC(=O)NC(C)C(C)NC(=O)Cc1nn(C)cc1Cl 38946,c1(OC)ccc(N)c(C(=O)NC2CC(CNC(=O)C(C)C3CCC3)C(O)C2)c1 38947,CCCC(CCC)=CC(=O)NCCOC1CN(C(c2c(C)cnn2C(C)C)=O)C1 38948,C(=O)(C#CC1CCCCC1)N1C(C)(C(=O)NC2CC(C(C)C)OC2)CCC1 38949,O=C1CCC2(CN(C(=O)Cc3cc(Cl)ccc3Cl)C2)N1 38950,N1(C(c2cc(=N)[nH]cc2)=O)CC2CC1CC2CNC(=O)CNC(C1CCCC1)=O 38951,CCC(C)CCC(=O)N1CCCOC(CNC(=O)C(C)(C)n2cccn2)C1 38952,CC(CC(N)=O)NC(C1C(CNC(c2nccs2)=O)C1(C)C)=O 38953,CN1CCC(NC(C2(CNC(C3CC3(F)Cl)=O)CC3(CC3)C2)=O)CC1 38954,c1(CC(=O)NCC(C)N(C(c2ccc(COC)[nH]2)=O)C)cncc(C#N)c1 38955,CCC(CC)C(=O)N(CCC(O)CNC(=O)CC1CCCC(C(F)(F)F)C1)CC 38956,C12(NC(CCC#C)=O)COC(C1)C(NC(=O)C(C)SCC)C2 38957,N1(C(CC(=C)C)=O)CCN(C(C2CCCCN2S(C)(=O)=O)=O)C(C(F)F)C1 38958,N#Cc1csc(CNC(=O)CN(C(=O)C(O)C2CC2)C2CCC2)n1 38959,C1(COC)(NC(c2ccc(O)nc2)=O)CCCN(C(=O)C(O)P(C)(C)=O)C1 38960,c1(NC(C2C(CC)CN(C(=O)Cn3cccc3)C2)=O)cc(CO)ccc1C 38961,C1(C(N2C(C=C)CCCC2)=O)CC2(CCN(C(=O)C(CC)N(C)C)C2)C1 38962,N1(C(c2c(SC)cn(C)n2)=O)CC(NC(C2CC(C)CCO2)=O)CC(O)C1 38963,C(=O)(C(F)(F)CCn1cccn1)NC1C(NC(c2c(N)nccc2)=O)CCC1 38964,c1(C(=O)NCCN(CCOC)C(C2CC(C)=NO2)=O)ccc(Br)c(C(F)(F)F)c1 38965,c1(CC)ncc(C(=O)NCCC2CN(C(c3scc(C)c3OC)=O)CCO2)cn1 38966,c1(CNC(c2n(CC(=C)C)nnn2)C2CC2)snc(OCC)c1Br 38967,N1(C(CC2CC(OC)C2)=O)CCCC2(C1)C(NC(c1nnsc1C)=O)CCN2C 38968,C1(F)(CNC(C2CCN(CC(C)C)C2)=O)CCC(NC(=O)Cc2c[nH]nc2O)C1 38969,Cc1nn2c(c1CNC(=O)CC1(C)CC1)CN(C(C1CC(O)CN1C)=O)CC2 38970,c1(C(=O)OC)cc(C(=O)NCCN(C(C2CCCC2O)=O)C(C)C)cs1 38971,CCC(C(=O)NCCC1(C)CCN(C(=O)COc2ccsn2)CC1)C(F)(F)F 38972,N1(C(C2CN(C(C(C=C)OC)=O)CC2F)=O)CCCOCC1C 38973,c1(N2CCC(CC)C2)cc(=NCc2nc(=N)n(C)[nH]2)[nH]c(C(C)C)n1 38974,C1(C(N2CCCC(C)(CNC(C3C(C)(C)C3)=O)C2)=O)CC(c2cccnc2)=NO1 38975,N1(C(CCSc2nc(C)[nH]n2)=O)CC2CN(C(=O)Cc3nccn3C)CC2C1 38976,Cc1cc(C(N2CCC(NC(C3(CO)CC3(F)F)=O)C2)=O)ccc1-n1ccnc1 38977,N1(C(c2c(Cl)cnc(CC)n2)=O)CCC(C2CCN(C(C3CC3CC)=O)CC2)C1 38978,N1(C(=O)NC(COC)C(C)C)CC2CS(=N)(=O)CC2C1 38979,C1(OC(C)C(=O)NCC(C)(C)NC(=O)CC2CC3(CC3)C2)CCCCC1 38980,C1(C(=O)NCCC2CC(NC(C=CCOC)=O)C2)Cc2nccn2C1 38981,c1(C(=O)NC(C(C)NC(=O)CC2(CO)CC2)C)ccc(Br)c(F)c1F 38982,CCC(C)CC(C)c1nc(-c2nc[nH]n2)nn1-c1cccnc1C 38983,N1(C(C2(C)C(C)C2)=O)CC2CCN(C(=O)CCc3ccc(C(C)(C)C)cc3)C2C1 38984,C1(NC(c2c(C)ccnc2C)=O)CC2CCC1C(NC(C1CCC(=O)N1C)=O)C2 38985,c1(OC)cc(C)c(NC(=O)C(C2CCN(C(C3CC34CC4)=O)CC2)C)cn1 38986,C1(O)(CNC(c2ccc(CNC(c3cnc(=N)[nH]c3)=O)cc2)=O)CCCCCC1 38987,C1(NC(c2c(NC)scn2)=O)CN(C(=O)C(CO)OC)C(C)(C)C1 38988,c1(C(=O)NC(C2(O)CCN(C(Cc3cnc(C)o3)=O)C2)C)c(F)ccnc1F 38989,C1(C(=O)OC2CN(C(CCc3ccc(OC)nc3)=O)C2)CCC(C)NC1=O 38990,CC1=CC(c2cn(CC3(F)CCCN(C(=O)CN(C)C)C3)nn2)=C(C)S1=O 38991,C1(C(=O)NC(CC=CC)C(=O)NCC2(CCC)CC2)CCC2CC1CO2 38992,C(=O)(N=c1ccn(-c2cc(C)c(F)cc2Cl)[nH]1)c1c(OC)csc1 38993,Cc1cc(C(N2CCN(C(C34CSC(C3)C4)=O)CC2)=O)c(N)c(F)c1 38994,C1(C(N2CCC(NC(c3c(C(C)C)nns3)=O)CC2C)=O)CCCCC12CCC2 38995,n1(CC(N2CCN(C(c3c(C)cno3)=O)CC2CCO)=O)ncc2ncccc12 38996,Cc1ncc2n1CCN(C(=O)NCCCCOc1ccc(Cl)cc1)C2 38997,C1(O)(CNC(CC(=C)C)=O)CCCN(C(C2CCC3CC3CC2)=O)C1 38998,N1(C(CCC(=O)OC)=O)CC2(CC(NC(C3CCSC(C)C3)=O)CO2)C1 38999,O=S(=O)(c1ccc(Br)cc1Cl)NC(c1ccc(F)cc1)CN1CCC1 39000,c1(C(N2CC(C)(C(C(C(n3ccc(C)n3)C)=O)=O)C2)=O)ccc(C)c(C)c1.CC 39001,N1(C(C=C(C)Cl)=O)CCC2(CC1)CN(C(=O)Cc1cnn(C)c1)CC2CO 39002,c1(C(=O)NC2C(NC(CC3(C=C)CC3)=O)CCC2)cnncc1C 39003,C1(NC(c2nn[nH]c2Cl)=O)CC2(CCN(C(=O)Cn3cccc3)C2)C1 39004,C(=O)(C1=CC2(CCOC2)C1)N(C1CCN(C(c2ccoc2Br)=O)C1)C 39005,CCCC(C)(O)C(=O)NCCC1COCCN1C(c1ncoc1C)=O 39006,N1(C(CC2ON=C(C)C2)=O)CCCCC1C(N1CCN(C(=O)C(C)C)CC1)=O 39007,C1(C)(C(=O)NCCN(CCC)C(c2ccc(C(C)(C)C)s2)=O)CC(C)OC(C)C1 39008,c1(C(N(CCCNC(C2(C)CCC(F)(F)C2)=O)C(C)C)=O)cnc2n1CCOC2 39009,c1(OCC(=O)NC2CCCCC2CNC(c2cnc(O)s2)=O)nc(O)nc(O)n1 39010,C#CCCC(O)CCNC(=O)C(CCCOC)NC(=O)CN1CCOC1=O 39011,N1(C(CCCC)=O)CCCC(O)(CCNC(=O)C(O)C(C)CC)C1 39012,C(C)(C(C)NC(c1ncoc1CNC(=O)C=Cc1cncs1)=O)(C1CC1)OC 39013,c1(C(=O)NC(C(=O)NCC(C#C)OC)CCC)nn(C)cc1C#C 39014,C1(CNC(=O)C(F)C2CC2)CC2(CO1)CN(C(c1ccc3c(c1)CCC3)=O)C2 39015,C1(C(=O)NCC2(CC)CCOC2)CN(C(=O)CN2CCNC2=O)C(C)(C)C1 39016,CCC(C#N)C(=O)NCCC1(NC(=O)CC2CCC(C)(C)C2)CCCC1 39017,Cc1ccc(C(=O)N(C(C)CCNC(=O)C(F)C(C)(C)O)C)c(N)c1Cl 39018,C1(C2CCN(C(=O)CN(C)C(=O)C3CC3)C2)(NC(CC(CCC)C)=O)CC1 39019,C1(C)(C(=O)NC2CC(NC(C3N(C(CCC)=O)CSC3)=O)C2)CCC(=O)NC1 39020,n1(CC)cc(C(=O)NC2CC(CNC(c3ccc(O)cc3)=O)C2)c(C)n1 39021,N1(C(C(C(C)C)(F)CNC(C2COCCO2)=O)=O)CCc2cccnc2C1 39022,c1(C(=O)NC(C2(O)CN(C(c3cc(F)cs3)=O)C2)C)ccc(-n2cncn2)nc1 39023,C1(C(N(C2CCCCN(C(=O)C=CSc3nc[nH]n3)C2)C)=O)CC2C(C1)C2(C)C 39024,N1(c2snc(C)n2)CC2CC(NC(C3(Br)CC3)=O)C2C1 39025,N1(C(Cc2n[nH]c(=N)s2)=O)CCC(C2(NC(c3ccn4nnnc4c3)=O)CC2)C1 39026,c1(C(=O)NCC(C)(CC)NC(C(CC)OC)=O)cccc2oncc12 39027,O=C1CCCc2cc(C(N3CC(NC(c4cc(F)cc(F)c4)=O)C3)=O)ccc21 39028,c1(C(=O)NC2C(C)CCN(C(=O)CO)C2)ccc(S(C)(=O)=O)cc1 39029,c1(C(N2CCN(CCNC(CCC=C(C)C)=O)CC2)=O)ccc2nn[nH]c2c1O 39030,C1(NC(c2nc(CC)oc2)=O)CC2CCC(C1)N2C(=O)Cc1cnc(Cl)cc1C 39031,S(=O)(=O)(c1cccnc1NCc1ccc(C)s1)NC(CC)C(O)C(C)C 39032,CCCC(CC(=O)NCC1CCC(C)CC1)NC(c1sc(C)nc1C)=O 39033,C1(C)(CNC(c2c(C)cns2)=O)CCCN(C(c2ccc(C(C)C)cc2F)=O)C1 39034,c1(C(N(CC(C)N(C(=O)CSS(C)(=O)=O)C)C)=O)cccc(C#CCO)c1 39035,C=C(C)C(C)(C)C(=O)NC(C1CCN(C(C2CSC3(C)CCC(=O)N23)=O)CC1)C 39036,C1(CC)CCN(C(=O)COC2CCCOC2)C(NC(=O)CC(C)(C)CN(C)C)C1 39037,Cc1ccc(-n2ncc(C(=O)NC(c3cccnc3)C3CC3)n2)cc1 39038,N1(C(C(CC2CCC2)NC(C)=O)=O)CCCCC1C1C(C(=O)O)C1 39039,N1(C2CCN(C)C2=O)CCC2(CC1)CC2C(N1CCCC1c1ccc(O)cc1)=O 39040,c1(C(N2CC(O)(CCNC(CNC(=O)NC)=O)C2)=O)c(C)[nH]cc([N+](=O)[O-])c1=O 39041,C1(NC(C(c2cc(C)sc2)(F)F)=O)CN(C(=O)C2CC2)C2CCCCC12 39042,C(=O)(CC(C)F)N(C1CC(NC(C(C2CCCCC2)OC)=O)C1)C 39043,C1(NC(c2ccc(C#C)nc2)=O)C2CCCN(C(=O)C=CC(C)C)C2C1(C)C 39044,C1(C(=O)NCC2C(NC(C(C3CCC3)OCC)=O)CC2)CCC(C)(C)CC1 39045,C(=O)(n1cnc(=NC(=O)N(CCN(C)C)Cc2cnn(C)c2)[nH]1)C(C)C 39046,C(=O)(CCCC(CC)CC)N1CCN(C(COCCCCOCC#C)=O)C(C)C1 39047,C(=O)(C1=CCN(C(=O)CC(C)(C)CN(C)C)CC1)NC1C=C(C)CCC1 39048,c1(C(N(CCC(C)(C)NC(C2CCCC(O)C2)=O)C)=O)nccc2[nH]ccc12 39049,C(C)(C(C(=O)NCc1ncc(F)cc1F)C(C)C)NC(C(F)=CCC)=O 39050,C(=O)(CC(C)(C)n1cccc1)N(CCCCNC(C(C)c1cccs1)=O)C 39051,N1(C(C2CC(C)(C(=O)OC)C2)=O)CC(NC(=O)C=CS(C)=O)C(F)C1 39052,CC1CCC(C(=O)NC2(CCNC(=O)Cc3cccnc3)CC2)O1 39053,c1(C(C)=O)ccc(C(=O)NCC(C)CN(c2ncnc(C)c2OC)C)c(F)c1 39054,N1(C(CCNC(=O)NC)=O)CC2C(CC(=O)NCc3cccc(CO)n3)C2C1 39055,c1(CNC(c2cccnc2-n2cc(CC(C)(C)CO)nn2)=O)ccc(Cl)cn1 39056,c1(NC(c2cn(CC3(CF)CC3)nn2)=O)onc2ccccc12 39057,N12Cc3cccn3CC(C1)C2=O.Cc1cc(C(=O)NC2C3COCC23)n(C(F)F)n1 39058,c1(OC(C)C)cc(C(N2CCCC(CNC(=O)CC3(C)OCCO3)C2)=O)ccn1 39059,CCC(F)(F)CC(=O)N1CCC(F)CC1C(N1CCC(C(C)(C)O)C1)=O 39060,C1(N(c2c(C(F)(F)F)cc(OC)nn2)C2CC2)CCN2CCCCC12 39061,N1(C(C2(Oc3cn(C)nc3)CC2)=O)CCCOC(CNC(=O)CCC2CCC2)C1 39062,C(C)(C)(CCCCC(=O)NCC1CN(C(C2CCO2)=O)C1)OC 39063,CC(C)(CN1CCOCC1)C(=O)NC1CC(CCNC(C2(C3CC3)CC2)=O)C1 39064,C(C(C)(C)C(=O)NCC1CCC(C)(CC)O1)NC(CCC#C)=O 39065,CC(C)(CCF)C(=O)NC1C=CCN(C(c2cc(CCO)on2)=O)C1 39066,C1(C(=O)NCC(CNC(c2ncoc2C2CC2)=O)OC)CCc2nc(C)nn2C1 39067,N1(C(C23C(C)(C)OCC2C3)=O)CCCC2(C1)CN(C(c1ncc(F)cc1F)=O)C2 39068,c1(CN(CCC)CCC)ccc(C(N2CC3CC2C3CN(C)C)=O)cc1 39069,c1(OCC(N2C(CCC(=O)NC3(C)CC=CCC3)CCC2)=O)ccccc1C#N 39070,c1(C(N2C(COC)(CNC(=O)C(C)C(C)O)CCC2)=O)cc2[nH]nc(C)c2cn1 39071,c1(OC)ccc2[nH]c(=NCCS(C)=O)[nH]c(=NCCc3ccc(Br)cc3F)c2c1 39072,c1(C(C)C(N2CCC(N(C)C(C3(C)CCCO3)=O)CC2)=O)ccc(Cl)c(Cl)c1 39073,c1(C(N2C(C)C(NC(=O)C(Cl)=CCl)CCC2)=O)cc(C#N)ccc1N 39074,Cc1ccc(CNC(=O)CN2CCC(CC(=O)N(C)Cc3ccccc3)C2)s1 39075,C#Cc1ccc(OCC(=O)NCCC2(NC(C3CCN(C)S3(=O)=O)=O)CC2)cc1 39076,c1(C(N2CC(NC(c3cccnc3)=O)C(C(F)F)C2)=O)cc(=O)n2nccc2[nH]1 39077,c1(C(=O)NC2C=CC(CNC(C(C)(C3CC3)OC)=O)C2)nc(Cl)oc1C 39078,N1(C(CC(CC)OC)=O)CCOCC(C)(CNC(c2ccc(C)cc2SC)=O)C1 39079,CCCC(CCC)=CC(=O)NC(C)CC(C)NC(=O)CCc1nccn1C 39080,c1(C(N(c2nnc(C(CC)(C)C)s2)C)=O)ccc2nc(O)n(C3CCCC3)c2c1 39081,c12cc(no1)NC2=O.C12(CSCCNC(C3(OCC)CC3)=O)CSC(C1)C2 39082,C1(NC(c2n[nH]cc2I)=O)CC12CCN(C(c1c(Cl)cc(F)cc1Cl)=O)CC2 39083,N#Cc1c(OCCNC(C2CCCN2C(C2CC2F)=O)=O)cccc1Br 39084,c12cc(c(C)o1)C(=O)NC2.c1(CC(=O)NC2CCC(SC)C2)cc(Cl)n(C)n1 39085,C(=O)(C(C(C)(C)C)OC)N(CC(=O)N(CC(N1CCCC1)C)C)CCOC 39086,C1(C)(CC(=O)NCCOCCCCC)CCN1C(=O)COCCCN=[N+]=[N-] 39087,Cc1cnc(Cl)c(CNc2ccsc2C(=O)NCC2(C)CC2)c1 39088,C1(OC)CCN(C(C2CCCCC2)C(=O)NCCCC2CC2)C1 39089,C(=O)(CS(C)(=O)=O)N1CC(C(C(=O)N(c2ccncc2)CC(C)C)OC)C1 39090,N1(C(C)C)CCCN(C(CCCNn2cccc(O)c2=O)c2ccccc2)CC1 39091,n1(CC(=O)NC2CC(CNC(c3ccc(C)cc3)=O)CC2O)nc(C)c(O)c1C 39092,c1(C(c2cccs2)NC(C2(C(F)F)CC2)C)nnnn1C1COC1 39093,c1(OCC)cccc(NC(=O)C(C)=CCNC(c2cc(C(C)=O)c(C)o2)=O)c1 39094,C(=O)(CCC(=O)N1CC(O)(CNC(C2C(Cl)(Cl)C23CC3)=O)C1)OC(C)(C)C 39095,C1(CN(C(=O)C2=CCC2)C)CCCCN1C(c1c[nH]c(-c2ccc(F)cc2)c1)=O 39096,c1(C(N2C(CNC(=O)COC3CCOC3)CC2)=O)ccnc(S)c1 39097,c1(C(=O)NC(CNC(c2nc(OCC)sn2)=O)(C)C)ccc(OC)c2ccsc12 39098,c1(C(C(=O)NCCC(C)CCNC(=O)C(C)C(F)(F)F)(C)C)cccc(C#N)c1 39099,C1(C(=O)OCCCOC)CCCCC1NCc1cccc(OCCC=C)c1 39100,N1(C(CCCC2C(C)C2)=O)CCC(C2CC2)C1C(N1CC(C#N)C1)=O 39101,c1(CNC(c2cccc(-n3c(C)c(C(=O)O)cn3)c2)=O)cn2cccc(C)c2n1 39102,N1(C(C2N(C(Cc3ccn(CC)n3)=O)CC2)=O)CC2CCC2(C)C1 39103,C(=O)(C(=O)N=c1cc(C)o[nH]1)NCC(CC)NC(c1ccc2c(O)n[nH]c2c1)=O 39104,C(C)(N=c1nc2c(ncn2C)c(NC(C)CS(N)(=O)=O)[nH]1)c1n(CC)ncc1 39105,c1(C(N(c2nc(OC)c(F)cn2)C2CCCNC2)=O)cc(O)ccc1[N+](=O)[O-] 39106,c1(C(=O)NCCN(C(c2c(C)nc(CCCC)s2)=O)CC)cc2n(n1)CCOC2 39107,C(CCC(C(=O)NCCC(=O)OC(C)C)NC(=O)CCc1nc(C)no1)OC 39108,c1(C(=O)NC2C(CNC(=O)CCC3CC3)CCC2)ccc(C(F)(F)F)nc1O 39109,c1(NC(C)=O)ccc(C)c(C(=O)NCC#CCNC(C2(C)CCCNC2=O)=O)c1 39110,C(=O)(C(C)(C)CCCO)NCC1CC2CN(C(c3cccc(OC)n3)=O)CC21 39111,C1(C(=O)NCc2c(C)occ2)CN(C(=O)CCC(=O)C2CC2)CC12CC2 39112,C(=O)(C1=CC2CCC=CCCC12)NCC1C(C)CCN(C(C2(O)COC2)=O)C1 39113,CCC(CC)C(=O)N1CCCCC1C(=O)N(CCN1CCCC1=O)CC 39114,C(C(C)NC(C1CCCC1)=O)(C(C)C)NC(c1ccn(C(C)C)n1)=O 39115,Cc1ccnc(C)c1NC(C12CCC1CN(C(=O)Cc1c(C)nn(C)c1C)C2)=O 39116,C1(C(=O)NCCc2cnn[nH]2)(NC(=O)C(c2ccccc2)F)CCOCC1 39117,CC1CN(C(c2cccnc2CO)=O)CCN1C(C1CCS(=O)(=O)CC1)=O 39118,c1(CC(=O)NC2C(CNC(=O)C=CC3CCC3)C2)nc([N+](=O)[O-])n[nH]1 39119,C(=O)(CCCCCCC=C)N1CC(CC#C)(C(=O)NC2CC(=O)N(CCC)C2)C1 39120,N1(C(c2ccc(CNC(N)=O)s2)=O)CC2CC1CCC2O 39121,CC(C)CN=C(NCc1ccccc1C(C)C)NCC1CCOC(C)C1 39122,Cc1cnc(-c2cn(CCN(C(=O)CC(C)(C)C#N)C(C)C)nn2)c(C)c1 39123,Cc1scc(C(N2CC(NC(C3(C4CCCO4)CCCC3)=O)C(O)C2)=O)c1N 39124,c1(NC(=O)NCCC)ccc(C2CC2)cc1.C12CC(C1)C(=O)NC2 39125,C1(CNC(C2CC(=C)C2)=O)CC(CNC(=O)Cc2cnn(CC(=O)NC)c2)CO1 39126,C1(C(N2CCCCC2)=O)CC2CCC1N2C(C1(OCC)CCCC1)=O.OCC 39127,CC(C)C1C(=O)N2CC3CC2C3C(=O)N1.C(=O)(C(N)=O)NCCSCOC(C)(C)C 39128,C1(NC(C(CCC)OC)=O)CC2CN(C(c3cn(C)c(=O)n3C)=O)CC2C1 39129,Cc1cnc(C#N)c(-c2c[nH]nc2C(=O)NCc2cc(F)c(F)cc2I)c1 39130,CC1C(NC(C2COCCN2C)=O)CCCN1C(c1[nH]ncc1C#N)=O 39131,N1(C(CC2(C#N)CC2)=O)CCN(C2CCCN(C(=O)Cc3c[nH]nc3O)C2)CC1 39132,CC1(C(=O)NCC2CN(C(=O)Cn3cc(C(F)(F)F)cn3)CC2O)CC=CCO1 39133,c1(CNC(=O)CC2CC=CCC2)ccc(C(N2CCC(c3cnn[nH]3)C2)=O)cc1 39134,C1(C)(COC(c2c(C)ccnc2C(C)C)=O)CC(C2CC2)=NO1 39135,c1(SC)ncccc1NC(=O)CCC1CCCN(C)C1 39136,C1(NC(=O)NC)CCN(C(=O)CCCN2CCOC2=O)C1 39137,c1(C(N2CCC(C)(CNC(C3CS(=O)(=O)C3)=O)C2)=O)c(F)ccc(Cl)c1N 39138,c1(C(N(CCCNC(C(C)SCC)=O)C2CC2)=O)cc(O)c2[nH]c(C)nc2c1 39139,C1(O)(CNC(CC2(CSC)CC2)=O)CCCN(C(c2csc(C#N)c2)=O)C1 39140,c1(C(C(N2CCC(CCOC)(C(=O)OC)C2)=O)C)ccccc1S(N)(=O)=O 39141,C1(NC(CCCC(=O)OC)=O)C2CC(CN(C(C3(CF)CC3(F)F)=O)C2)C1CO 39142,C1(NC(c2c(COC)scc2)=O)CCCCC1CNC(c1sc(C)cc1C)=O 39143,c1(CNC(c2cnc(SC)s2)=O)cc2n(n1)CCN(C(C1CC(C3CC3)C1)=O)C2 39144,N1(C(C2C=C(C)CS2)=O)C2CCC1CC(C(=O)NC(C)C(C)F)C2 39145,C1(CNC(C2ON=C(CC)C2)=O)CC2CCC1N2C(c1cc(C)ccc1C)=O 39146,N1(C(c2ncn(C(C)C)c2)=O)CCC2(CCN(C(C3CC3c3cccs3)=O)C2)C1 39147,C1(OC(C)C(=O)NCC(C)(C)CNC(=O)COC2CC2)CCCCCC1 39148,c1(C(N2CCC(NC(c3c(C)onc3C(F)(F)F)=O)C2C)=O)ccc([N+](=O)[O-])[nH]1 39149,C1(C(=O)NC(C)(C)CNC(c2c(C(F)(F)F)ncn2O)=O)CC(=O)OC1(C)C 39150,c1(C(CC)(C)C)cn(CC2CC(NC(=O)C(F)OC(F)(F)F)C2)nn1 39151,C1(C(N2CC(C)C(NC(c3ccncc3N)=O)C2)=O)Cc2nccnc2C1 39152,CC1=NNC(=O)C1CC(N1CCCCC1CNC(C1(c2ncco2)CC1)=O)=O 39153,CS(=O)(=O)C1CCN(C(C(=O)NCc2ccccc2)C2COC2)C1 39154,C(=O)(CC(CC(C)C)NC(=O)C(CCC)=CCC)NC1(CC=C)CC1 39155,CC1CCN(C(=O)C(=O)NCC2CCCN(C(=O)CC3CCCOC3)C2)CC1 39156,c1(C(=O)NC2C(C)CN(C(c3c[nH]nc3F)=O)C2)n[nH]c2c1CCCC2 39157,n1(CC(N2CC(NC(C(C)SCCCC)=O)C(C(F)F)C2)=O)ccc([N+](=O)[O-])n1 39158,c1(C(=O)NC)cccc(C(=O)NC(CO)C(C)NC(C2CCS(=O)(=O)N2)=O)c1 39159,C(=O)(CCS(=O)(=O)NC)NC(CNC(c1ccc(OCC)nc1)=O)(C)C1CC1 39160,C1(C(=O)NCCCC(C)NC(c2sccc2C(F)F)=O)CC2CC1CC2O 39161,C1(CNC(c2c(C)cc(C)[nH]2)=O)(NC(c2c(C)ccn2C)=O)CC2CCC1CC2 39162,Cn1cc2c(C(=O)NCCC3=CCN(C(=O)CSCC(N)=O)CC3)cccc2n1 39163,CC(C)CC(CC(C)C)NC(=O)CCCC(C)NC(=O)Cc1ccc[nH]1 39164,C12(CNC(c3ccc(C)nn3)=O)CC(NC(c3nc(Br)c[nH]3)=O)(C1)C(C)O2 39165,Cc1cc(C(N2CC(CC(F)C(=O)NC3COCC3CO)C2)=O)sn1 39166,c1(C(=O)NCCN(C(c2ccc(C(C)=O)cn2)=O)C)cc(=O)c2ccncc2o1 39167,c1(C(=O)NC)ccnc(CN(C(c2cocn2)=O)CC2C3CNC2C3)c1 39168,c1(CSCC(C(C)(C)C)OC)nc2ccccc2o1 39169,C1(C(=O)NC2(c3ccccc3)CN(C(CC3CC(=C)C3)=O)C2)CNC(=O)CC1(C)C 39170,N1(CCC(=O)NCC(CC)(C)NC(c2cnc(C(C)O)s2)=O)CCCCC1=O 39171,C12(C(=O)NC(CCCC)C)CCCC1CN(C(C1(COC)CC(=O)C1)=O)C2 39172,C1(C(C=CC(=O)OCC(COCC)O)=O)CCCN(C(C)=O)C1.C(=O)CC 39173,N1(C(C(Cn2ccnn2)NC(C2(CC)CC2)=O)=O)CCCN(C(C)=O)CC1 39174,Cc1cc(C(=O)NCC2CC2NC(=O)Cc2nc(C(C)C)c(C)s2)c(N)c(Cl)c1 39175,N1(C(CNC(=O)NC(c2nocc2N(C)C)C)C)CCN(C)CC1 39176,c1(C(N2C(CC=C)CCC2)=O)cn2c(n1)C(N)CCC2 39177,Cc1cccc(C(=O)N(C(CNC(c2ncccc2N)=O)C2CC2)C)c1Br 39178,Cc1nc(C)c(C(c2nnnn2CCCC2CC2)NC(C)CC(C)(C)C)s1 39179,c1(C(N(CCNC(C(C2CC2)OCC)=O)C)=O)nc(-c2ccccc2F)oc1C 39180,C1(C)(C(N2C(C)(CC(=O)NCCc3n(C)cnn3)CC2)=O)CCNC1=O 39181,S(=O)(=O)(c1cccc(Br)c1)NC1(C#N)CCN(Cc2c(F)ccc(Cl)c2F)C1 39182,CC1C(NC(=O)C=Cc2ccccc2)C(C)CCN1C(C1CCC=CO1)=O 39183,Cc1nc2ccc(-c3cncc(NS(C)(=O)=O)c3)cc2n1C 39184,N1(C(C2(COC)CC=CC2)=O)CC2CCC(C1)C2C(N1CCCC1CO)=O 39185,c1(C(N2CC(C(C)C)N(C(=O)CCN3CCCC3)CC2)=O)cc(O)cc(C#N)c1 39186,Cc1ccncc1C(=O)NC1(CCCC(=O)NCC2(C)CC(C)(C)C2)CCC1 39187,N1(C(CCOCC)=O)CC2C(CN(C)C(C3(CF)CC(F)(F)C3)=O)C2C1 39188,N1(C(c2nnc(O)nc2O)=O)CCC2CN(C(=O)C(O)CC(F)F)C2C1 39189,c1(C(=O)NCC2CN(C(CCCCSC)=O)CC2O)cc2cc(Cl)ccc2[nH]1 39190,C1(CNC(=O)C(=O)NC2CC2)CN(C(=O)CCC2OCCO2)CC12CCOCC2 39191,C(=O)(C(CC(F)F)N(C)C(C1CN2CCC1C2)=O)NCC1(F)CCN(C)C1 39192,O=C1NC(=O)C(CC(=O)NC23CC(C2)N(C(c2ccncc2O)=O)C3)N1 39193,N1(C(c2ccc(N)c(F)c2)=O)CC2ON=C(CNC(=O)CCc3nccs3)C2C1 39194,C(C(=O)N1CC(C)(NC(c2cscc2F)=O)C1)(C(C)C)NC(C(C)NC(C)=O)=O 39195,C12(C(=O)NCC3C(C)CCN(C(=O)COCCN(C)C)C3)CC(C)(C1)OC2(C)C 39196,C1(C2CCN(C(=O)Cc3cnsc3)C2)(NC(C2C3COCC23)=O)CC1 39197,Cc1scc(C(=O)NC(Cn2cccn2)C(=O)NCC2([Si](C)(C)C)CC2)c1C 39198,c1(C(=O)NC2C(NC(C3CCCC(C)(C)C3)=O)COC2)nc2cc(O)ccc2[nH]1 39199,CC1CCCc2ncc(C(=O)NC3CN(C(C4CC5CC4C5)=O)CC4(CC4)C3)n21 39200,N1(C(CC(CC)C2CCC2)=O)CCC(C(=O)N(CCCF)CC)C(C)(C)C1 39201,Cc1ccc(C=CC(N2CCCC(NC(=O)C=C3CCC(C)CC3)C2C)=O)nc1 39202,C1(NC(C2(NC(C(C)CC3CCCC3)=O)CC(O)C2)=O)CC1C1CC1C 39203,c1(NC(=O)OC(C)(C)C)sc(Br)cc1NC(C(C1CCOC1)N(C)C1CC1)=O 39204,C1(C(=O)OC)CC(NCc2cc(Br)co2)C12CCC2 39205,N1(C(C(CC)CC)=O)CCC2(CC1)CN(C(C1CCCC13CC3)=O)CC(C)O2 39206,C1(NC(C)C)CC(NC(C2COCCN2C)=O)C12CCC2 39207,C1(C(N2CC=CC(C(N(CCC)C)=O)C2)=O)CC(C)(C)CN1C 39208,c1(C(N(C)CC2CCCN2C(=O)C=CC2CCCO2)=O)cc(O)cc(C#N)c1 39209,C1(CNC(C=CC(=O)OCCCC)=O)CN(C(=O)CC)C2CCN1C2 39210,C1(CO)CCCC(N=c2[nH]c(=NC3CC(N4CCC4)C3)[nH]c3c2COC3)C1 39211,N1(C(=O)CC2CC(F)(F)C2)CCC2CCN(C(C3CC4CC3C4)=O)C2C1 39212,CC1CCC(NC(=O)CCC2(C#N)CCC2)CN1C(=O)CC1(N2CCCC2)CC1 39213,C1(C(N2CCC(CNC(CNC(CC)=O)=O)CC2)=O)CC1C1CC(F)(F)C1 39214,c1(C(=O)NCc2scc(CNC(CC3C(C)CCO3)=O)n2)cc(O)ncn1 39215,N1(C(c2ccc(C(C)C)c(Cl)c2)=O)CCN(C(c2cnncc2O)=O)C2(CC2)C1 39216,c1(OC)ccc(Cl)c(CC(=O)NC2CC(CCNC(=O)CCc3cc[nH]n3)C2)c1 39217,Cc1cc(=NCCCS(=O)(=O)C(F)F)[nH]c(N2CCSCC2)n1 39218,N1(C(CS(N)(=O)=O)=O)CCC2CCCN(C(=O)Cc3cccc4[nH]ncc34)C2C1 39219,C1(C(=O)NCCN(C(C(N2CCOCC2)C)=O)C2CCCC2)CC(F)(CF)C1 39220,C(=O)(C(C)S(=O)(=O)C1CCOCC1)NC1C2CN(C(C(C)NC(CC)=O)=O)C1C2 39221,C(=O)(CCCC(CC)NC(c1cnn(C(F)F)c1)=O)N1CC(N(CC=C)C)C1 39222,c1(OC)noc(C2CC2)c1C(=O)NCCC1CCCN1C(=O)CC1CC2CC2C1 39223,c1(CC)cc(C(=O)OC)ccc1NC(=O)NCC(C)(C)Cc1ccccn1 39224,CCC(C)CCCC(=O)NCC(CNC(=O)Cc1cc(O)nnc1O)OC 39225,N1(C(C2CCCN(C(C3(C)ON=C(C)C3)=O)C2)=O)CCC2(CC1)CSC2 39226,c1(C(N2CCC(C)(NC(CN(C(C)=O)C)=O)C2)=O)nn(C)c(C)c1N 39227,c1(C(=O)NCc2c(C(=O)NCCC(CC)CO)n[nH]c2)cccc2ccoc12 39228,C(=O)(CC1=Cc2ccccc2C1)NCC(CC)(C)NC(=O)CCCc1cc[nH]n1 39229,Cc1nc2cc(C(N3CCCC3CCCNC(=O)C(C)N(C)C)=O)ccc2s1 39230,C1(NCc2c(C)c(Br)ccn2)CCCC2CN(C(=O)OC(C)(C)C)CC12 39231,C1(CN(C(C(C)OC)=O)C)COCCN1C(=O)C(CO)OC 39232,C1(NC(C(n2cc(C3(C(N)=O)CC3)nn2)C)=O)C(C)(C)C(N(C)C)C1(C)C 39233,N1(C(C=CC(CC)=CC)=O)CCC2(CCCN2C(=O)CCc2ncc(F)cn2)C1 39234,c1(C(N2CCCC2CC)C(=O)NC(CC)C)cnc(C2CC2C)s1 39235,C1(C(=O)NC(C2CCN(C(C3C(C)CCO3)=O)C2)(C)C)CCCN(C)C1 39236,CC1(C)CC(NC(=O)CC2C=CS(=O)(=O)C2)CN1C(=O)CCCn1ccnc1 39237,N1(C(C=C)=O)CC2(C1)CN(C(C1COCCN1C1CCCC1)=O)C2 39238,c1(-c2cn(CCC(=O)NC(c3ccccc3)CC)nn2)cc[nH]c(=N)c1 39239,c1(C(=O)NCCC(C)NC(=O)CNC(c2ncccc2O)=O)nnc(O)cc1O 39240,C(=O)(CS(=O)(=O)c1ccccc1Cl)NC1CCC(F)(CNC(C(CC#C)O)=O)C1 39241,c1(C(N2CC(CCC)N(C(c3cncs3)=O)CC2)=O)ccc(Cl)c(F)c1O 39242,CC1(C)CN(C(=O)C=C2CCSCC2)CC1NC(=O)CSc1ccccc1Cl 39243,C1(C(N(CC(C)CNC(c2sc(Cl)cc2Cl)=O)C)=O)CCCC1C1CC1 39244,C1(CNC(C2(SC)CC2)=O)CCC(C)CN1C(c1ccc(C2CC2)o1)=O 39245,c1(C(=O)NCC(CO)NC(C2CCC(C(=O)OC)O2)=O)cnc(C2CC2)nc1O 39246,C(CCN=c1nc2scnc2c(NC(C2CC(F)(F)C2)C)[nH]1)N(C(C)C)C 39247,C(=O)(C(CC(C)C)NC(C1CCC1)=O)NCCNC(C1C(C(=O)OC)C1)=O 39248,N1(C(CCC=C)=O)CC2C(C(F)(F)F)CC2(NC(c2ccc(C)n2C)=O)C1 39249,N1(C(c2ccc(Cl)s2)C(=O)NCc2cccs2)CCCCCC1 39250,c1(OCC(=O)NCC(CO)NC(c2cnc(CC)[nH]2)=O)ccc(F)c(Br)c1 39251,N1(C(COCCN(C)C)=O)CC(C)(CNC(C2CCCCCCC2)=O)CC1(C)C 39252,c1(C(=O)NCC2CN(C(=O)CCC3CCCC(O)C3)C2)cc(Cl)c(F)cc1Cl 39253,Cc1nc(C(C)(C)C)nc(S)c1C(=O)NCC1CC2CC2N1C(=O)C(C)C(C)C 39254,N1(C(C2CCC(=O)N2)=O)CCC(C2CCN(C(C3CN4CCN3CC4)=O)CC2)C1 39255,C1(OCCNC(N(CCCOC)CCO)=O)CCC(F)(F)CC1 39256,C#CCC(C)(CC)C(=O)NCC1CN(C(c2ncsc2C2CC2)=O)CC1(C)C 39257,C1(N=c2[nH]n3cc(C)nc3s2)(CC)CCN(C(C2CCCC(F)C2)=O)CC1 39258,N1(C(C=NOC)=O)CCC2CC(NC(c3cnnn3C(C)C)=O)CCC2C1 39259,CCCCCCCCCCNC(C1CC(Nc2cc(SC)ncn2)C1)=O 39260,CC1CC(C(=O)NC(C)(C)CCCNC(=O)Cc2cnc[nH]2)CCS1(=O)=O 39261,CC1CC(NC(C2(CF)CCC2)=O)CN(C(=O)CC2CCCCO2)C1 39262,CC(CF)CC(=O)N1CCCC(CN(C(=O)Cc2cccn2C)C)C1 39263,N1(C(CCCCCCC)=O)CCC2CN(C(c3coc4c3COC4)=O)CCC2C1 39264,CCC(C)(CC)C(=O)NCC1(O)CN(C(c2cccc(C#N)c2)=O)C1 39265,c1(OC)ccnc(O)c1C(N1CC(CNC(=O)C=Cc2ccnn2C)C1)=O 39266,N1(C(c2cc(C(C)=O)[nH]c2)=O)CCN(CCNC(C2CC(=O)N(C)C2)=O)CC1 39267,c1(C(=O)NCC2(O)CN(C(C=CCCC=C(C)C)=O)C2)ccc(N)cc1F 39268,N1(C(c2c(C(C)C)cnn2C)=O)CCCC2(C1)CN(C(=O)CC1=CCCCC1)C2 39269,C1(CN(C)C)(CNCc2c(Br)ncn2C)CCN(C(=O)OC(C)(C)C)CC1 39270,C1(C(=O)NC(C(C)NC(C2CC3CC3C2)=O)CO)CC(C)(C)CO1 39271,C(c1cccc(C#N)c1)=CC=C.CN1CCN(C(=O)NOCCCO)CC1C[SH](=O)=O 39272,N#Cc1cccc(C(O)CNc2nccc(F)c2C)c1 39273,C1(NC(=O)CCOc2cccnc2)C=CCN(C(C2CCC=CCC2)=O)C1 39274,C1(C(C(=O)N(C2CSC2)CC#C)C)CCN(C(=O)COC2CCCC2)C1 39275,CC(C)(CCNC(=O)Cc1cocn1)NC(=O)CSC1CC1 39276,CC1CC(N(C)C(C2CC(O)CN2C(=O)C(F)CC2CCOC2)=O)CCO1 39277,C1(C(N2CC3C(CNC(CN4CCCC(CC)C4)=O)(C3)C2)=O)CC(C2CC2)=NO1 39278,c1(OC(C)(C)C)ccc2c(NC(N3CC(SCC(=O)O)C(O)C3)=O)cnn2c1 39279,C(C(C)(C)C(=O)NC1CCCN(C(=O)CC(=O)Nc2ccccc2C)C1)OC 39280,n1(CC=C)cccc1C(=O)NC(C1CCN(C(C2(F)CC2)=O)C1)C 39281,C1(C(=O)NCCCCCCOC)CC2(CCC2)CN1C(C12CC(F)(C1)C2)=O 39282,C(=O)(C1=COCCO1)NCC(CN(C(c1ccc(C2CCC2)cn1)=O)CC)(C)C 39283,c1(C(N2C(C(=O)NC3CC(=O)OC3)CC(F)C2)=O)nccc2ccccc12 39284,N1(C(C(C)OCCOC)=O)CCN(C)C(C(=O)NC2CC(CO)(CO)C2)C1 39285,C1(CC=C)(C(=O)NC(C=C)C2CCC2)CCCN1C(=O)C(C)CSC 39286,Nc1cncc(C(=O)NC2CC(NC(c3cc[n+]([O-])cc3)=O)C(O)C2)c1 39287,S(=O)(=O)(c1cccc(Cl)c1)N(CC(N1CCN(C(C(CC)OC)=O)C(C)C1)=O)C 39288,N1(C(C(C(C)C)OCC)=O)CC2(NC(=O)C(C)OC)CCC1CC2 39289,CC1CCCN1CC(=O)N(CC(=O)NC(c1cccnc1)CO)C1CCC1 39290,N1(C(c2ccc(OCC)nc2)=O)CCN(C(=O)CC2CC(N(C)C)C2)C(CC)C1 39291,C1(C(=O)NCC(CNC(c2ccnc(OC)n2)=O)O)CCOC(=O)CC1 39292,N1(C(C(CC)c2cccnc2)=O)CCCC(CC)(NC(c2cc(Cl)ccn2)=O)C1 39293,C1(NC(C=C(C)C(C)C)=O)CCC(CNC(=O)CCc2ncc(F)cn2)CC1 39294,C1(C)(OC)CCCN(c2cc(NCc3nc(C)c(C)o3)nc(C(F)(F)F)n2)C1 39295,CC1CCN(C(c2n[nH]cc2Cl)=O)CCN1C(=O)CCCS(N)(=O)=O 39296,c1(N2CCC3(C(NC(c4cnco4)=O)CC3)CC2)ncc2c(Br)cccc2n1 39297,c1(NC(=O)CC2CC(NC(=O)Nc3cn[nH]c3)C2)ccc(-c2ccccn2)cc1 39298,c1(Cc2nc(-c3ccc(C(=O)O)s3)on2)cccc(F)c1 39299,C(=O)(C(C(C)(C)C)n1ccnn1)N(CC(C)O)CCNC(=O)COC1CCOC1 39300,C(=O)(CS(=O)(=O)CCO)N1CCC(C)(CNC(C2C(CC(C)C)C2)=O)CC1 39301,N1(C(C=C(c2n(C)ncc2)F)=O)CCCC2(CCN(C(=O)CN3CC=CC3)C2)C1 39302,C(=O)(C1=CCCCO1)NC(CCOC)C(=O)N1CC(C)=C(C)C1 39303,C1(C(=O)NCC2N(C(CN3C(C)CCC3)=O)CCC2)CC(S(C)(=O)=O)C1 39304,CC1CN(C(=O)C2CC2)CC2(CCN(C(=O)C(C3COC(C)(C)O3)O)C2)O1 39305,CC(C)CC(O)CC(=O)NCC(C(N1CC(CO)CC(C)C1)=O)N(C)C 39306,N1(C(c2cncc(C(F)(F)F)c2)=O)CCN(C(=O)CCn2ccnc2)C(CF)C1 39307,C1(C)(C(=O)NCC=CCNC(C=C(CC)C)=O)CCCC1O 39308,N1(C(c2c(CC)[nH]cc2)=O)CCC(NC(C2CN(C3CCOC3)C2)=O)C(F)C1 39309,N1(c2nccc(C)c2)CCc2cc(C)ccc2C1C.C1CC2CC3C(C2)C13 39310,N1(C(c2ccccc2)C(=O)Nc2cccc(F)c2)CCc2cc(F)cc(Cl)c2C1 39311,N1(C(=O)Cc2sccc2Cl)CCCC(N(CCO)C(C2CC(F)C(=O)N2)=O)C1 39312,CN1CCCC(O)(CC(N2CC(C3(Nc4cc(O)nc(O)n4)CC3)C2)=O)C1 39313,N1(C(C(c2ccn(C)n2)C)=O)CC=CCC1C(=O)N(C)CC1(C)CC1 39314,CC(C)CCCC(C)C(=O)NC1(C2CCCN2C(c2cnc(C(C)C)o2)=O)CC1 39315,N1(C(C2C(=C)C2)=O)CC2CC(CNC(c3ccc(C(C)(C)C)[nH]3)=O)C2C1 39316,C1(N(C(C)=O)C(C2CCN(Cc3nc(C(=O)O)co3)C2)=O)CCS(=O)(=O)C1 39317,C(=O)(C(C)(C(C)C)NC(C)=O)N(CCNC(C1(C(=O)OCC)CCC1)=O)C 39318,N(C1CCCn2ccnc21)C(C1C(CNC(C(CO)N(C)C)=O)CC1)=O 39319,n1(C(C)C)ncc(C(N2CCC(CF)(NC(=O)CC3CCCC(=O)N3)C2)=O)c1Cl 39320,N=c1ccn(CC(N2CCCC2CNC(c2cc(C3CCOCC3)no2)=O)=O)[nH]1 39321,c1(C(N2CC(C)C(NC(c3c[nH]nc3-c3ccco3)=O)C2)=O)cc(=O)cc(Cl)[nH]1 39322,c1(C(=O)NCC(C)(C2CCC2)NC(c2cc(C3CC3)ncn2)=O)ccc(F)cc1 39323,N1(C(C2(OCC)CCCC2)=O)CCCN(C(=O)Cn2nnc(=O)[nH]2)CC1 39324,C1(CNC(CN(CC)CC)=O)CCCN(C(c2ccc(F)c(Cl)c2)=O)CC1 39325,c1(C(N2CC(C)(C)C2C2CCN(C(C3(CO)CC3)=O)CC2)=O)cnn2ccsc12 39326,N1(C(c2c(C)cnc(F)c2)=O)CC(C)OC2(CCN(C(=O)C(=O)C(F)(F)F)C2)C1 39327,N1(C(C(C2CCCC2)OC)=O)CCC(NC(c2cc(C(C)C)on2)=O)CC(O)C1 39328,C(=O)(NNc1c(C#N)cccc1Cl)NCCc1cc(C)ncc1 39329,CC1CCCC(N2CCN(C(c3ccoc3)=O)CC2)C1 39330,c1(CN2CCN(C(C3(CC(C)C)CC(=O)C3)=O)CC2)nc2ccccc2o1 39331,c1(C(=O)NCC2N(C(C(C)OCCC#C)=O)CCC2)ccc(OC(F)(F)F)cn1 39332,Cc1noc2ncnc(N3C4CCC3CC(NC(c3ncc(Cl)s3)=O)C4)c12 39333,c1(CN(C)C(C2(C)CC2)=O)cnn2c1CN(C(c1cc(F)ccc1F)=O)CC2 39334,C(=O)(C(O)C(F)(F)F)NC(C1CCN(C(C(COC)(C)OC)=O)CC1)CO 39335,C(=O)(C1=CCC(C)(C)CC1)N1C(CNC(c2cc(C(C)=O)sc2)=O)CCC(C)C1 39336,c1(C(N2CCC(O)(CNC(CCCC=C)=O)C2)=O)ccc2c(c1)SCCN2 39337,C1(C(=O)NCC(CC)NC(=O)C(c2ccc(F)cc2)(C)C)CCCCN1N=O 39338,C(=O)(C(Cn1ccnn1)NC(c1cc(C2CC2)[nH]n1)=O)NC(CCOCC)C 39339,c1(NC2CCN(C(=O)NCC(C(CC)O)C)CC2)csc2cc(C)ccc12 39340,c1(C(N2CC(CCNC(=O)C(c3ccn(C)c3)C)(OC)C2)=O)ccc([N+](=O)[O-])o1 39341,C1(O)(CNC(CC2C(NC(C(C=C)(C)C)=O)CC2O)=O)CCN(C)CC1 39342,C1(C(=O)NC(C(C)C)(C)CNC(=O)CC2CC3(CC3)CO2)CC2(C1)CC1(CCC1)C2 39343,C(c1ccc(N(C)C)cc1)=CC(=O)NC(C(C)C)CCNC(c1n[nH]cc1F)=O 39344,C(CCS(=O)(=O)c1ccccc1)NC1CC2(CC(NC(COC)=O)C2)C1 39345,N1(C(c2ccc(OC)cc2O)=O)CCC(C)C(NC(=O)CSC(C)C)C1C 39346,N1(C(CCCN(C(C2C(C(=O)OC)CC2)=O)C)=O)CCC12CCCCC2 39347,CCCCCCC(F)C(=O)N1CCC(CNC(c2ccc(O)c(N)n2)=O)C1 39348,c1(N(C(C(=O)COC(C2CCCCC2)=O)C2CC2)C)ccc(N(c2nnc(C)s2)C)cc1 39349,Cc1scc(C(=O)NC2CCC(N(C(=O)C(c3cccnc3)C)C)CC2)c1N 39350,n1(CCNC(C2CCC(NC(C3CCSCC3)=O)CO2)=O)ccc2ccccc12 39351,c1(CNC(CSCCNC(c2c(CC)nns2)=O)=O)c(C)cccc1C 39352,c1(NC(Cc2nc(C)oc2)=O)nc2c(s1)CC(O)CC2 39353,Cc1cccc2c1CN(C(C1CN(C(C3C(C)C3C)=O)CCC1(C)C)=O)C2 39354,c1(N2CC(C)C(F)(F)CC2)nc(N(C)CCN2CCCC2)c2cnn(C)c2n1 39355,C1(C(=O)NCC(C)N(C(C(C(=O)OCC)CC)=O)C)CC2(C1)CC(F)(F)C2 39356,C(C(=O)NOCC(=O)N(C)C)=CCN(C(C=CC=CCC)=O)C 39357,C(=O)(C(CC(C)(C)C)OC)N(CC(=O)NC1C(C)(CC)CCC1)CC(C)C 39358,C1(NC(c2c(OC)ccnc2)=O)CCCC2CN(C(C3(C)CCCC3C)=O)CC12 39359,n1(CCC(N2CCN(C(CSCCOC)=O)C(C)C2)=O)c(=O)oc2ccccc12 39360,c1(OC)nc(Br)ccc1NC(C1(F)CCN(C(=O)CC2(O)CCC2)C1)=O 39361,c1(C(c2n(CCC)nnn2)NCCCCOCC2CC2)cccc2nccn12 39362,Cc1cccc(OCCC(N2CC(NC(c3ncccn3)=O)CCC2C)=O)c1C 39363,C(=O)(CCN=c1[nH]ccs1)NCCNC(C1C2CC(C)(C2)OC1)=O 39364,n1(CC(=O)N(CCNC(C(N2C(=O)CCC2=O)CC)=O)C)cc(S(N)(=O)=O)cn1 39365,N1(C(c2ccc(C)cc2Br)=O)CC2COCCC2(NC(c2cncn2C)=O)C1 39366,C(C)(CO)(CS(C)(=O)=O)NC(=O)CCN(c1ccc(OC)cc1)C1CCCC1 39367,C(=O)(C(F)C(C)CNC(C1CC(=C2CCC2)C1)=O)NC(C(=O)NCC)(C)C 39368,C1(NC(C2(C#N)CCCC2)=O)CN(C(c2cnc(C3CC3)o2)=O)CCC1CO 39369,n1(CC)nc(C)c(NC(=O)C=Cc2ccsc2C(F)(F)F)c1C(=O)OC 39370,CC1(C)OCC2(CCN(C(c3coc(Cl)n3)C(=O)NC3CCC3)C2)CO1 39371,C(=O)(CC1=CCCC1)NCC(=C)CCNC(=O)C(F)(F)c1ccccn1 39372,CC(C)S(=O)(=O)c1ccc(C(N2CC(NC(=O)C3=NNC(=O)CC3)C2)=O)cc1 39373,CC(C)CC(CC(=O)NC1CCC(=O)NC1=O)NC(c1cncnc1)=O 39374,N1(C(CSCC(C)C)=O)CCC2CCN(C(C3CC4(C3)CC43CCC3)=O)CC12 39375,CCCC(CCC)CC(=O)N1CCCC1CNC(C1(CC)CC(C)(C)C1)=O 39376,c1(C(C)=O)ccc(C(=O)NC2CCC(CNC(c3ccc(Br)s3)=O)C2)o1 39377,C1(CNC(Cc2cc(C)[nH]n2)=O)COCCN(C(=O)Cc2ccccc2F)C1 39378,C1(NC(C(CC)OCC)=O)CN(C(c2cn(C(C)(C)C)nc2C)=O)CC12CC2 39379,C1(C(=O)Nc2cccc(CC(=O)OC)c2)Nc2cc(C)ccc2S(=O)(=O)N1 39380,c1(C(=O)NCCC(C(C)C)NC(=O)CCOC2CC2)cccc(N)c1O 39381,CC1CN(C(c2ccc(C(F)(F)F)[nH]2)=O)CC1CNC(C1(S(C)(=O)=O)CC1)=O 39382,N1(C(C2(C)CCNC2=O)=O)CC(CNC(c2ccc([N+](=O)[O-])s2)=O)C(C)(C)C1 39383,C1(=CC(=O)NC2(CNC(Cc3cn(CC)nc3)=O)CC2)CCCCCC1(F)F 39384,C1(CNC(c2c(CC)scn2)=O)CCC(C)CN1C(c1cc(C2CC2)n(C)n1)=O 39385,c1(CC)ccc(F)cc1C(N1CCC(NC(=O)CSC(F)F)C(CC)C1)=O 39386,n1(CC)nc(C)cc1C(=O)NCC(=C1CN(C(=O)CCC2CCC(O)CC2)C1)F 39387,N1(C(CCCSC)=O)CCC2(CCC(NC(c3ccc(C4CC4)cc3)=O)CC2)C1 39388,C1(NC(C=CCOCCOC)=O)C=CC(CNC(=O)C(N2CCOC2=O)C)C1 39389,C1(C(N(CCC(F)(F)F)C)=O)CCC(C)(C)N(C(c2csc(=N)[nH]2)=O)C1 39390,c1(C(N(CCC(C)NC(=O)CC(C)c2cccnc2)C)=O)ncncc1Cl 39391,CCCCS(=O)(=O)NCC(N1CCC(CCNC(C2CCCCC2C)=O)CC1)=O 39392,c1(OCC=C)ccc(Cl)nc1C(N1CCC(C(C)CNC(=O)CCOC)CC1)=O 39393,N1(CCCNC(CC2(C)CCCC2)=O)CCN(C(=O)CCC(F)F)CC1 39394,N1(C(C2(CC=C)CCC2)=O)CCC2(C1)CN(C(=O)C(C)NC(=O)OC)CCO2 39395,C1(CCC)CN(C(C2CSC2)=O)CC1NC(=O)C(C1CCOCC1)O 39396,C1(N(C)C)CC(N=c2[nH]c(=NCCP(C)(C)=O)[nH]c3c(F)cccc23)C1 39397,N1(C(c2ccc(CC)o2)=O)CC=C(CCNC(=O)C(C)COc2ccccc2)CC1 39398,C(=O)(C(CC)CC=C)NC1(CC=C)CN(C(C2(Cc3cnn[nH]3)CCC2)=O)C1 39399,n1(CC)ccc(C(N2CCC(CNC(=O)CCc3cncs3)C23CC3)=O)cc1=O 39400,CCCCC(C(=O)N=c1ccn(Cc2ccc(C(F)(F)F)cc2)[nH]1)C(C)C 39401,C1(C#N)(C(=O)NCC(CNC(c2ccc(N(C)C)cc2)=O)F)CCS(=O)(=O)CC1 39402,CCC(C)CC(C(=O)N(CC(N)=O)C)NC(=O)CCCC(F)(F)F 39403,C1(NC(C(CC)(C)CNC(=O)CCc2cscn2)=O)CC12CCCCCC2 39404,C1(CC(=O)NCC(C)(C)OCCNC(CC(=O)NCC)=O)CCCCC1C 39405,C=CCC(CC(C)C)C(=O)NC(C1CCCN1C(=O)C1=CCCS1)C 39406,c1(C(=O)NCC2(CNC(c3c(C)scn3)=O)CC2)cnn(C2CCOCC2)c1C 39407,C1(C(=O)NCCCCC#C)(OC)CCN(C(c2cc(C)cc(F)c2)=O)CC1 39408,C(CC(O)C(=O)NC1CCOCC1NC(c1cc(-n2cnnc2)ccn1)=O)SC 39409,N1(C(c2c(OCC)scc2)=O)CC2(CCN(C(=O)CCN(CC)CC)C2)C1 39410,C(=O)(CCCCC(C)C)NC(CCN(C(C=Cc1n(CC)ncc1)=O)C)C(C)C 39411,C1(C(=O)NCC(C)(C)NC(=O)CCc2ccc(C#N)cc2)CCS(=O)(=O)C1(C)C 39412,C1(C(=O)NC(c2nccs2)C)COC(CNC(=O)C(O)CC2CCCC2)C1 39413,c1(C(N2CCCC(CN(C)C)C2)=O)ccc(N=[N+]=[N-])cc1 39414,c1(C(=O)NCC2CCCN(C(C(CC(C)C)(C)O)=O)C2)ccnc2c1CC(=O)N2 39415,N1(C(CC(CC)NC(c2c(C#C)cnn2C)=O)=O)CCC2(C=CCO2)C1 39416,N1(C(CCSCCCC)=O)CCCCC1C(N(C)Cc1oc(C)nc1CC)=O 39417,c1(OC)cc(CN2CCCC(C(=O)NC3CCOC3)C2)ccc1O 39418,O=C(C#CC1CCCOC1)NCC1CN(C(=O)Cc2ccc(Cl)cn2)C1 39419,C1(CCNC(=O)C(C2CCCCC2)F)CCCN(C(=O)Cc2cccnc2)C1 39420,c1(OC)cccc2c1CC(C(=O)N(CCCN(C(=O)C=C(C)C(C)C)C)C)CO2 39421,CC1CCCCC1(C)NC(=O)C(c1cnn(C)c1)NC(=O)CC(=O)NC1CC1 39422,C(=O)(C(CCCO)c1ccccc1)N(CC=C)CCN(C(=O)COC)CC 39423,C12CCCC1CN(CCO)C2=O.C(=O)(CCCn1cc(C2(CO)CC2)nn1)OC 39424,C1(CN(C)C(C2CCC2F)=O)CCN(C(c2ccc(=N)[nH]c2)=O)CC1 39425,CCC(CC)CCC(=O)N1CCC2(C1)CN(C(C1CCCC(=O)O1)=O)C2 39426,CCC(CC(=O)N1CC2CCN(C(=O)Cc3cnccn3)C(C2)C1)CC(F)(F)F 39427,C(c1ccc(C)c(Cl)c1)=CC(=O)NCC1C(NC(C(n2ccc(C)n2)C)=O)CC1 39428,c1(CNC(C(C)N(C(CC)=O)CC)=O)cn(C2CCC(C(=O)NC)C2)nn1 39429,c1(C(c2nnnn2C2CC(F)(F)C2)NC2CC(CC)C2)cncn1C1CC1 39430,C(C(COC)C(=O)N1CSCC1C(=O)NCCn1cnnn1)OC 39431,N1(C(c2ccc(OC)nc2)C(=O)NCCCC2CC2)CCC(O)CC1C 39432,c1(C(N2C(COC)(CNC(C3CC(C)CO3)=O)CCC2)=O)ccc([N+](=O)[O-])n1C 39433,C(C(C)(C)CC(=O)NC(c1nn(C)cc1O)C)NC(Cc1c(C)scc1)=O 39434,CC(O)C(C)C(=O)N1CCN(C2CCN(C(C34CC3C4)=O)C2)CC1 39435,c1(OCC(=C)C)ccccc1C(=O)NCCC(C)CCNC(c1cc(Cl)ns1)=O 39436,N1(C(C=COCC)=O)CC(CNC(=O)CC2CC(C)OC2C)OC(C)(C)C1 39437,N1(c2c3ncn(C(CC)(C)CC(C)O)c3ncn2)CCCn2cc(Br)cc2C1 39438,c1(OCC=C)ccc(NC(=O)C(N)Cc2ccc(F)cc2)cc1C 39439,N1(C(=O)CN2CCN(C(c3cc(Cl)cs3)=O)CC2)CCC(C2CCOC2)C1 39440,N1(C(CCOCC#C)=O)CC(CNC(=O)C(CO)c2ccccc2)CC12CCC2 39441,c1(C(N2CCSCC2C2CCC2)C(=O)NCCCF)cc2c(Cl)nccc2s1 39442,C1(CCCNC(CCOC)=O)CCCCN1C(=O)C(N1CCC(C)CC1)=O 39443,C1(C(N2CCC(=CCNC(c3c(CC)nns3)=O)CC2)=O)CN(CP(C)(C)=O)C1 39444,C1(CNC(C2(C(C)C)CCC2)=O)CCN(C(c2cnn[nH]2)=O)C12CCC2 39445,N1(C(CCSC)=O)CCCC1C1CCCCN1C(=O)CN(C)CCO 39446,c1(N2CC3CC(NC(c4ccc(C)o4)=O)C3C2)c(Cl)cccc1[N+](=O)[O-] 39447,c1(CN(C)Cc2onc(C(C)OC)n2)cc(OC)c2c(c1)OCCO2 39448,CC(C)CCCCCC(=O)N(C)CC1(O)CCN(C(=O)CCC#N)CC1 39449,C1(C(N2C(CC(=O)NC(Cn3ncc(C)c3)C)CCC2)=O)CCC(CSC)CC1 39450,c1(C(N2CCC(NC(C(C)OCC=C)=O)CC2)=O)cc2n(n1)CCCC2 39451,c1(C(CC(=O)OC)NC(=O)CNC(N)=O)cccc(-c2cccnc2)c1 39452,CCC(C)CCC(=O)NCC(c1ccc(F)cc1)NC(=O)C=Cc1cc[nH]c1 39453,C1(NC(COCC#C)=O)CCOC(CNC(=O)CC2COCC2(C)C)C1 39454,C1(Cl)(C(=O)OC)CC1C(=O)NCCC(C)NC(C1(N(C)C)CC1)=O 39455,C12(NC(c3c(SC)ccs3)=O)COC(C1)C(NC(=O)C(c1ccnn1C)O)C2 39456,N#Cc1c[nH]c2ncnc(N3CC(F)CC3C(=O)NCCN3CCOCC3)c12 39457,C1(NC(C=CC(CC)C)=O)CCCCCN(C(=O)Cc2ccsc2)C1 39458,C(=O)(C(C)(C)C(C)(F)F)N1CC(OCCNC(C(CCC)c2ccc(Cl)cc2)=O)C1 39459,C(C(C)(C)C(c1ccccc1)NC(=O)N(c1ccccc1)Cc1cccs1)OC 39460,c1(CCC(=O)NC2C(NC(CCCNC(C)=O)=O)CCC2)cccc(F)c1F 39461,c1(OC)ccc(C(N2CCCC23CCN(C(=O)C(C)OC)C3)=O)n2nccc12 39462,CC(C(=O)N1CC(NC(=O)C(n2cc([N+](=O)[O-])cn2)(C)C)C1)C(C)(C)C 39463,Cc1ccc(F)cc1N(C(=O)C(C)NC(c1cc(Cl)cs1)=O)C 39464,Cc1cc(F)cnc1C(N1CC(NC(c2cccc(Cl)c2O)=O)CC(O)C1)=O 39465,c1(CCC(=O)N(CCCNC(C2N(C)CCOC2)=O)C2CC2)ccc(Cl)c(Cl)c1 39466,c1(C(N(CC(CNC(C2C(C)(CC)C2)=O)C)C)=O)cnn(CCO)c1 39467,c1(C(N2CCC(NC(c3nc(OC)c(C)s3)=O)C23CC3)=O)n[nH]c2c1CCSC2 39468,O=C(CCn1cc(C(c2ccccc2)=O)nn1)NNC(=O)NCC(F)(F)F 39469,N1(C(CCOC)=O)CCC(NC(CNCC(=O)N(C)C)=O)C1 39470,CCC(CCC(=O)N1CC=C(C)CC1)NC(=O)CCNC(=O)NC 39471,N(C(=NCCC(=O)N(C)C)NCC1CCN1C(C)(C)C)CC(CC)(C)C 39472,c12cn(nn1)CC2OC.C1(NC(c2sccc2-c2cccs2)=O)CCCC1OC 39473,CCC(C)(C(=O)NC(C1CCN(C(=O)C(C)(C)c2ccccn2)CC1)C)OC 39474,C1(C(=O)NC(C#CCC)(C)C)CCN(C(=O)C(=O)C2CCCC2)O1 39475,C1(OC)CC(NC(c2cc(C)oc2C(C)C)=O)CN(C(C2(C#N)CC2(C)C)=O)C1 39476,c1(OC)ccc(Cl)cc1C(N1CCC(CCNC(C2(C)CCN(C)CC2)=O)C1)=O 39477,C(=O)(C(C)CCCC(C)=O)N1CC(NC(=O)NC(C(CC)CC)C)C(CC)C1 39478,N1(c2nc(N3CCCC(CC(=O)NC)C3)nc(C)c2)CCc2nc(O)[nH]c2C1 39479,c1(SC)ncc(C(N2CCSC(C(=O)Nc3ccc(Br)nc3)C2)=O)c(Cl)n1 39480,C(c1ccsc1)=CC(=O)NC(C)CCN(C(=O)C(C)N1CCCC1)C 39481,Cc1noc(C(C)C)c1C(=O)NC(CNC(c1ccnc(C2CC2)c1)=O)C(C)C 39482,CC(C(C)NC(=O)CSc1nc[nH]n1)NC(c1csnn1)=O 39483,c1(CCN(C(=O)NC2CC2C(=O)OC(C)(C)C)C=O)ccc(Cl)c(C)c1.CN.O 39484,C1(C)(C(N2CCC(OC)CC2)=O)CCCN(c2cnc(C(N)=O)cn2)C1 39485,c1(NCC(CCCC)NC(=O)CC(C)OC)ncnc2sc(CC)cc12 39486,N#CC1CCCC(C(N2CCN(CC(=O)NCc3cnccn3)CC2)=O)C1 39487,C1(CCC)CCCN1C(C1CC1C(C)C)=O 39488,C(=O)(C(CC(C)(C)C)NC(=O)C(CN(C)C)N(C)C)NCCCOCCCC 39489,C1(C(C)NC(CCCOCC=C)=O)CCCCN1C(=O)CCc1nccn1C 39490,c1(C(=O)NC(C(C)NC(COC(CC)CC)=O)C)cc(C)c(F)cn1 39491,c1(N(CC#C)C(c2cccc(N3CCCC3=O)c2)=O)cccnc1OC(C)C 39492,c1(NS(=O)CCNc2ccc(C(F)F)o2)ccc2ncnn2c1.C12CCN(C1)C2 39493,C(=O)(CCCC)NC(C1CCN(C(=O)C(F)(F)c2ccccc2)C1)(C)C 39494,Cn1cc(C(N2CCCC2Cl)=O)c(C2CCC2)n1 39495,c1(SC)cc(=NC(=O)C2CC(C)(C)CCN2C(=O)C(c2cnn(C)c2)C)[nH]n1C 39496,C(=O)(C(CC)CC(F)F)NCCCN(C(c1n(C=C)ncc1)=O)CCO 39497,CN=c1[nH]cc(C(=O)NC2(COC)CN(C(C3CCCN3C)=O)C2)s1 39498,N1(C(C(CCOCC)NC(CCC#CC)=O)=O)CC(CC)CC(C)C1 39499,CCCCC(C(=O)N(C1(CC(N2CCCC(C)C2CO)=O)CC1)C)N(C)C 39500,C1(C(=O)NCCc2n(C)c(=O)on2)C2CC3C(C2NC(=O)CC2CCC(=O)C2)C13 39501,C1(CCNC(C(CC)N(C(=O)CCC2(C)CC2)C)=O)NC(=O)NC1=O 39502,c1(C(=O)NC(C2CCCN(C(=O)COC(F)(F)F)C2)C)ccnc2ccccc12 39503,C1(NC(c2cnc(CC)[nH]2)=O)CCN(C(c2nc(Br)cnc2N)=O)CC1C 39504,CC1(C)CCCC1NC(=O)C(N1CCCC(Cc2nc(C(F)(F)F)cs2)C1)=O 39505,c1(C(=O)NCCC2(NC(C3CC3(F)Cl)=O)CC2)c[nH]c2ccncc2c1=O 39506,N1(C(COCC)=O)CC(F)CC1CC(N1CCC(Cc2ccon2)C1)=O 39507,N1(Cc2ccc(C)cc2)CC2CN(C(=O)NNC(=O)C(C)C)CC2C1 39508,N1(C(c2c(C)c[nH]n2)=O)CCCC2CN(C(=O)Cc3ccc(C#N)cc3)CC12 39509,Cc1cc2ccccc2cc1C(=O)NCC(O)CNC(c1cc(Cl)ccc1N)=O 39510,Cc1nc(CNC(c2nnsc2N)=O)oc1C(=O)N(C)CCOCCCO 39511,C=CC(C)(O)C(=O)N(CC(C)C(=O)NCCn1cccnc1=O)C 39512,c1(C(=O)NC(C(C)=O)C2CC2)n[nH]c2cc([N+](=O)[O-])ccc12 39513,Cc1cccc2c1CCN(C(c1cc(Cl)ccn1)=O)C2.C1(N)C2CCC1CNC2 39514,Cc1ccc(C2=NOC(C(=O)NCC3CC(NC(C4CC4C4CC4)=O)C3)C2)cc1 39515,[SH](=O)(=O)c1ncc(F)cn1.CC(CS(C)(=O)=O)C(C)c1ccccc1 39516,c1(N(C)C)noc(CNC(c2cnn(C)n2)c2nnnn2C2CC2)n1 39517,C(C)(C)(C(C)NC(=O)CCCc1cc(C)no1)NC(CSCCC)=O 39518,C1(CNC(C2CC2c2nc(C(F)(F)F)no2)=O)CCC12CC(F)(F)C2 39519,c1(OC)c(C(N2CCC(O)(CNC(=O)C(C)OC)C2)=O)csc1C 39520,N1(C(C2CC(C#N)C2)=O)CCC(O)(CCNC(C2CC(=O)N(C(C)(C)C)C2)=O)C1 39521,c1(NC(C2(C)CN(c3ncncc3Br)C2)=O)cc(C#N)cn1C(C)(C)C 39522,Cc1ccc2nc(N3CC4CC3(CNC(=O)CC3C=CS(=O)(=O)C3)C4)sc2n1 39523,N1(C(=O)NCCn2c(C)cc(C(=O)OC)n2)CCCC2CNCC12 39524,Cc1cc(C(F)(F)F)c2cc(C(=O)NC(C)CCN(C)C)oc2n1 39525,CCC(CC)C(=O)N1CC(F)(CNC(C2CNC(=O)N2)=O)C1 39526,N1(C(C=CSC)=O)CC(N(C)C(c2cccc(-c3ccco3)c2)=O)C(C)(C)C1 39527,N1(C(c2cnc(C(C)C)s2)=O)CCC(C2CCCN(C(C3(C)CCC3)=O)C2)C1 39528,CON(C)C1CN(C(C2CCN(C(c3ccc(C)o3)=O)CC2C)=O)C1 39529,c1(N(CCCCO)C)nc(=NCc2cc(F)ccc2Cl)[nH]c2c1COCC2 39530,Cn1nnc(Cn2nnnc2C2(NCc3ccncn3)CC(OCC(=O)O)C2)n1 39531,C1(C(C)NC(=O)CCC2CCCOC2)CCCN(CC2CC3CCC2O3)C1 39532,C1(SC)CCC(N=c2nc(N(C)CC3CCCC3O)c3c([nH]2)CCOC3)CC1 39533,C(=O)(C(F)(F)C(O)C1CC1)N1CCC(NC(C(C(C)C)NC(N)=O)=O)C1C 39534,c1(C(OC)OC)ccc(C(N2CCC(NC(=O)Cc3nccn3C)C2)=O)o1 39535,c1(OCC)cc(C(=O)NCC(C(C)C)NC(c2cocc2C)=O)ccc1OC 39536,N1(C(=O)OC(C)(C)C)CCN(C(c2cccc3oncc23)=O)CCCC1C(=O)O 39537,CC1CC(=O)CCC1C(=O)NCC=CC(=O)N(CCN1CCCCC1)C1CC1 39538,N(C)(S(N)(=O)=O)CC(=O)N(C1CC(NC(=O)COCc2ccco2)C1)C 39539,C(=O)(C(O)CC(F)(F)F)NCc1c(C2CN(C(C(CC)OC)=O)C2)ocn1 39540,CC(CS(C)(=O)=O)C(=O)N1CC(O)(CN(C(=O)CCC(C)(F)F)C)C1 39541,C1(NC(COCC(=C)C)=O)(CO)CCN(C(c2ccc(CO)s2)=O)C1 39542,CC1(C(=O)NC2CCC(CNC(=O)CSc3nncs3)CC2)Cc2ccccc2N1 39543,c1(CCCCC)ccc(C(N2CC(O)(CN(C(=O)CC3CSC3)C)C2)=O)o1 39544,N1(C(CS(CCOC)(=O)=O)=O)CCOC2(C1)CN(C(c1ccc(N)c(F)c1)=O)C2 39545,c1(C(N2CCC3(C(C(=O)Nc4cnoc4)C3)CC2)=O)cc(F)c(Br)cc1[N+](=O)[O-] 39546,c1(C(N2CCC(NC(C(CC#C)(C)C)=O)C2)=O)cc2c(C)[nH]nc2s1 39547,c1(C(N2CC(CNC(CCSC)=O)C2)=O)ccncc1Cl 39548,C(=O)(C(O)CC(F)(F)F)NCCC1CCC(NC(C2CC3(CC(OC)C3)C2)=O)C1 39549,CCCC(C)(C)C(=O)NCC1CCC(C(N2CCC(CCN(C)C)C2)=O)CC1 39550,C1(C)(C(=O)NC)CCN(C(=O)C(=O)Nc2cnn(-c3nccs3)c2)CC1 39551,c1(CC)nc(=N)[nH]cc1C(=O)N(C)CC1CCCN1C(c1cncn(C)c1=O)=O 39552,C1(NC(c2c(C)nn[nH]2)=O)CC2(C(=O)NCC3=CCCCC3)COC1C2 39553,C12(C(=O)NC3C(C)CN(C(C4CCCC(C)(C)C4)=O)C3)CC=CCN1CCC2 39554,C1(C(=O)NC2CCN(C(c3nccc(SC)n3)=O)CC2F)Cc2ccccc2C1 39555,C1(C(=O)NCC23C(CN(C(CS(N)(=O)=O)=O)C2)CCO3)CCCCC12OCCO2 39556,Cc1ccn2nc(C(N3CC4CCC3C(NC(c3nsnc3O)=O)C4)=O)nc2n1 39557,c1(CC)cc(C(=O)NC2(CO)CN(C(C3CCCC3O)=O)C2)sc1C 39558,C(=O)(CC(C)CNC(C1CC(O)CN1C(=O)CP(C)(C)=O)=O)OC 39559,c1(CNC(=O)NC(c2ccc(OC)c(F)c2)C)c(C)cc(Cl)nc1Cl 39560,c1(OC)c(F)cc(C(=O)NCC2CCN(C(=O)CCCSC)CC2)cc1Cl 39561,N1(C(CCCOC)=O)CCC2CCCC12CNC(c1cc(Cl)ccc1F)=O 39562,C(=O)(N=c1nc[nH]n2cccc12)C1C2(CN(C(c3ccc(C#N)cc3Cl)=O)C2)C1 39563,C(=O)(C(F)C(C)(C)O)NC1CC(C(C)NC(c2cncc(CC)c2)=O)C1 39564,C(=O)(C1CCCc2n[nH]cc21)N1C2C(NC(=O)CCn3cnnn3)(CCC2)CC1 39565,C1(C(=O)Nc2cncc(NC(C)=O)c2)(C(=O)OC)CCC(O)CC1 39566,C1(CC(=O)NC2(C)CN(C(C(C)n3ccnc3)=O)C2)CCCC(C)(C)CC1 39567,c1(C(N(CC2N(C(C(CC#C)C3CC3)=O)CCC2)CC)=O)c(O)nnc2c1CCC2 39568,C(=O)(NNc1cc(C(F)(F)F)ccc1F)c1cnc2ccn(C)n2c1=O 39569,N1(C(c2ccc[nH]2)=O)CCC(N2CCN(c3ccc(F)cc3)CC2)CC1 39570,N12CC3CCCC1C3C2=O.C1(C)(CC(=O)NCC(OC(F)(F)F)C)CC1(F)Cl 39571,CC1=CC(C)CN(C(C2CCC(NC(=O)CCc3cccn3C)CC2)=O)C1 39572,C(C)(C(C(=O)N1CCC(F)CC1)C(C)C)NC(c1c(C)c(Cl)ccc1)=O 39573,Cc1ncc(Cl)cc1C(=O)NCC1(C(F)F)CCN(C(=O)C(C)N2CCC2)C1 39574,N1(C(C2CC23CCC3)C(=O)NCCCOC)CC(C)OCC(C)(C)C1 39575,C1(C2CCC2)(C(N2CC(CC)N(C(C3CC4(CCCC4)C3)=O)CC2)=O)CC1(F)F 39576,C1(NC(C2N(CC)CCC2)=O)CCCC12CCN(C(=O)COC(C)(C)CC)CC2 39577,N1(C(C(=O)N(CC(O)CN2CCCC2=O)C)=O)CCCCCC(S(C)(=O)=O)C1 39578,N1(C(C2C(C)(C)CC2)=O)CCC2C1CCCN2C(=O)Cc1ccco1 39579,c1(C(=O)NC(C(C)NC(c2cc(CC(C)C)on2)=O)C)cc2c(nn1)CCOC2 39580,c1(C2(CNC(CN(C)CC)=O)CCC2)cc(C(F)(F)F)ncn1 39581,C1(C(N(CCN(C(CCOC)=O)C(C)C)C)=O)CC2(C1)CC21CC1 39582,C1(NC(CCSC)=O)C2CN(C(=O)CCn3cccnc3=O)CC12 39583,C=CC(CCC)CC(=O)N(C)CC1CCCC(NC(c2sc(CO)nc2C)=O)C1 39584,C(=O)(CC(F)(F)CC(=O)NCC1CCN(C(C2(C)CCCO2)=O)C1)OC 39585,C1(C(=O)NCC(C)N(C(=O)C(C2CCOC2)OC)C)(CC)CCOCC1 39586,C1(CCCNC(C2C(Cl)(Cl)C23CC3)=O)CCCCN1C(=O)Cn1nccn1 39587,N1(C(C2C(C=C)CC2)=O)CCN(C(c2c[nH]nc2CC)=O)C(C2CC2)C1 39588,N1(C(CCN(C(C(CC(C)(C)C)OC)=O)C2CC2)=O)CCN2CC(F)CC2C1 39589,Cc1cc(C(F)(F)C(=O)NC2CC(CNC(c3cc[nH]c3C3CC3)=O)C2)cs1 39590,c1(C(C(=O)NCC(C)(CO)NC(=O)CNC=O)O)ccc(F)cc1Br 39591,CCC(CC)C(C(=O)N1CC(NC(=O)CC2CC2)C(CO)C1)OC 39592,CCC(O)C(F)(F)C(=O)N(C)CC1CCCCN1C(=O)CN(C)C(N)=O 39593,C1(CNC(C2(C=C)CCC2)=O)(NC(=O)C=Cc2cncn2C)CCCCCC1 39594,n1(CC)ccc(C(=O)NCC(CO)NC(c2c(C)coc2C(C)C)=O)c1C 39595,Cc1nc(O)[nH]c1NCC1CCN(C(c2nc(N)sc2-c2ccccc2)=O)CC1 39596,C1(SC)CN(C(=O)CCn2cc(Cl)cn2)CC1NC(C1CCNC1=O)=O 39597,C(C)(N=c1[nH]c(=NCc2ccc(N)cc2F)[nH]c2c1COC2)c1ccc(C)cn1 39598,c1(NC(C2CCCC(NC(C(C=C)(F)F)=O)C2)=O)cccc(F)c1C 39599,CC1CCOC(CCO)CN1S(=O)(=O)CCOCc1ccccc1 39600,c1(C(=O)NC(CN(C(c2c[nH]c3nccc-3c2)=O)CC)C)sc2cncn2c1C 39601,c1(C(=O)NCC2(NC(CCCOC)=O)CCCCC2C)cnc2c(c1)COCC2 39602,N1(C(=O)NC(c2c(CCC)nns2)C)CCC(CO)C(O)CC1 39603,c1(C(N2CCC(C(=O)NC3CC(C(COC)C)C3)CC2)=O)c(F)cncc1Cl 39604,N1(C(c2cc(OCC)n[nH]2)=O)CCC2CN(C(=O)C(C)(C)C)CCC2C1 39605,c1(NC(CNC(C2(CC#C)CC=CCC2)=O)C2CC2)ncn(C)c(=O)c1Br 39606,c1(-c2n(CC3C(CC)CC3)ccn2)cccc(-c2cc(OC(F)F)ncn2)c1 39607,C1(C(=O)NCC(COCC)C)CCN(C(=O)CCC2CCCC2)CCO1 39608,C1(CNC(c2n(C)cnc2)=O)CCCN(C(=O)Cc2ccn(CCF)n2)CC1 39609,C(CCCCC(=O)NCc1nc(C(=O)NCC2COC(C)(C)C2)co1)=CC 39610,C(=O)(CCCC(=O)N(C)C)NCC1(C(=O)NCC(C(=O)OC)(C)O)CC1 39611,O=C1NCCCCC1C(=O)NC1C2CN(C(=O)CCOC3COC3)CC12 39612,C1(C(=O)NCC2(C)CCCN(C(CC3(C)OCCO3)=O)C2)OCCOC12CCC2 39613,c1(N(CC)CC)ccc(C(N2CCN(C(=O)NC3CC(=O)C3(C)C)CC2)=O)cc1 39614,Cc1cc(C)c(C(N2CC(C(C)(C)O)(CNC(C3CC(=C4CCC4)C3)=O)C2)=O)o1 39615,c1(C(=O)NCC2CC(OC)CN2C(c2scc(C)c2C)=O)ccc(N)cc1F 39616,N(C1CC(C)(C)CCc2ccccc21)C(NNc1ccc(C)cc1Br)=O 39617,N1(C(C(CC)O)=O)CCN(C(=O)Cc2cncc(F)c2)C(CC(F)F)C1 39618,Cc1cc(C(=O)NCC2(C)CCN(C(=O)C(C)(C)O)CC2)ccc1I 39619,CCCC(C(=O)N1CCC(NC(=O)CCc2cnc(C3CCC3)o2)C1)C(C)C 39620,c1(C(N2CCCC(N(C(CC3N(C)CCC3)=O)C)CC2)=O)ccn2ccccc12 39621,N1(C(CC(c2ccc(C)cc2)(C)C)=O)CC(NC(c2cc[nH]n2)=O)CC(C)(C)C1 39622,C(C(C)CC(=O)NCc1ccc(CNn2cccn2)o1)NC(=O)OC(C)(C)C 39623,c1(NC(=O)C=Cc2cnccn2)ccc2c(c1)CN(C(=O)CC1CCC1)C2 39624,Cn1c(I)cc2c(N(C(c3cnnc(Cl)c3)=O)CC3(O)CCCNC3)ncnc12 39625,N1(C(c2cccc(N(C)C)n2)=O)CCCC12CCN(C(=O)CN1CC=CC1)CC2 39626,C1(OCC)CCN(C(=NCC2CC2)NCC(C2CC(F)(F)C2)OC)CC1C 39627,C12(C(N3C(CNC(COc4ccc(C)cc4)=O)COCC3)=O)COC(CCO1)C2 39628,c1(CC(=O)NC2(CO)CCN(C(C=Cc3cn(C)nc3)=O)C2)cc(F)cc(Cl)c1 39629,CC1CC(CCNC(c2cnn(C)n2)=O)CCN1C(=O)CCNC(=O)CO 39630,C(CCN(C(=O)CCCOc1cccc(Cl)c1)C)(C(C)C)NC(C1(OC)CC1)=O 39631,c1(OC)cc(C(=O)NC(C2CN(C(C3C4CC5C(C4)C35)=O)CCO2)C)ccn1 39632,N1(C(C(CC)O)=O)CC(C2CN(C(c3ccc(C)c(O)c3)=O)C2)C1 39633,C1(C(N)=O)(CNC(c2cnc(-c3ccccc3)[nH]2)=O)CN(C(C2OCCO2)=O)C1 39634,C(=O)(C(C)(O)CCc1ccccc1)N(CCC(C)NC(CCCOC)=O)C 39635,c1(CNC(c2c(C(=O)OC)ocn2)(C)C)ccc(Br)cc1Cl 39636,C1(NC(CCC#C)=O)CC(CNC(=O)CCc2nc(-c3ccoc3)no2)C(O)C1 39637,N1(C(CCOCCOC)=O)CCC(F)(F)C(CNC(c2scnc2COC)=O)C1 39638,N1(C(CC2CCC(C)(C)O2)=O)CCCC(CC(=O)NC2COCC(C)(C)C2)CC1 39639,C1(C(=O)NC2CCC(NC(C(CC)OCC)=O)CC2)CCC2CC2CC1 39640,c1(OC)ccc(C(=O)NCCCC(C)(C)NC(c2onc(OC)c2Br)=O)cc1 39641,C1(CNC(C2C(c3ccc(C)s3)C2)=O)CCCCN(C(C2CN(C)CCO2)=O)C1 39642,N1(C(C2C(C)(Br)C2)=O)Cc2ccccc2CC1CNC(C1CC(F)(F)C1)=O 39643,N1(C(C(C2CCN(C(C3(C4CC4)CC3)=O)C2)C)=O)CCC2CN(C)CC2C1 39644,c1(CC)ncc(Cl)c(C(=O)NCCCC2CCCN2C(c2nc(C)n(C)n2)=O)n1 39645,Cc1nc2ccccn2c1C(=O)NC1COCC1NC(=O)CCC(C)(F)F 39646,C1(NC(C2(C(C)(C)OC)CC2)=O)CC2CC1N(C(C1(C(F)F)CCCO1)=O)C2 39647,CC(C)(CCCCNC(C1CC=CC(O)C1)=O)NC(C1CC1(F)F)=O 39648,C(=O)(C(CCN(C)C)N(C)C)NCCOCCN(C(CC(C)N1CCCC1=O)=O)C 39649,c1(OC)ccc(-c2cn(CC3CCN(C(C4CCCCS4)=O)CC3)nn2)cc1F 39650,CC1(C(=O)NCC2CC(O)CN2C(C2COCCN2C=O)=O)CCCNC1=O 39651,N1(C(CCC(=O)OC)=O)CCC(C)C(NC(C2CN(C(=O)N(C)C)C2)=O)C1 39652,C1(CNC(c2nnn(CC)c2C)=O)CN(C(c2nnccc2C)=O)CCC1C 39653,C(C1CN(C(=O)C2=CCCCC2)CC1C(=O)NCC(C)(C)CC)=CC 39654,N1(C(Cc2cccc(C)c2)=O)CCC2CCC12CNC(=O)C=Cc1cncs1 39655,C1(NC(c2ncc(Cl)cc2Cl)=O)COC2(CCN(C(C3(O)CCSCC3)=O)C2)C1 39656,CC1CCCc2ncc(C(N3CCCC(C)(NC(c4cc(=O)cc[nH]4)=O)C3)=O)n21 39657,CCCCCCC(C(=O)NCC1CN(C(c2scnc2Cl)=O)CC1O)NC(C)=O 39658,c1(C(=O)OCC)cc(=NCCC2CC3(C2)CN(C(C2CC24CC4)=O)C3)[nH]cn1 39659,C(=O)(C(CC1CC1)OC)NC1CC(CNC(CCNC(COC)=O)=O)C1 39660,N1(C(CCC=CC)=O)CCc2ccccc2C1CNC(=O)CCC1(C)CC1 39661,C(=O)(C(CNC(C12CC(CO1)C2)C)CC(C)C)OC(c1c(CC)ncs1)=O 39662,C1(NC(c2cc(CCO)on2)=O)C2CCC(C2)C1C(=O)NC1CC2CC3C(C2)C13 39663,c1(OC)cc(C)ccc1CNC(=O)OC1CCNC1=O.C(C)(C)(C)OC 39664,CCC(C)(CCC(C)C)C(=O)N(CCCN(C)C(c1n[nH]c2c1CC1CC21)=O)C 39665,Cc1cn2cccc(C(N3CCSC4CCC34)C(=O)NCC3CC3)c2n1 39666,c1(C(=O)NCc2cccc(OC)c2OC)c(C)c(O)nc2ccccc12 39667,C1(C)(C(=O)OC)CN(C(C2CCC2)=O)C1.C12(CC1)C(=O)N2 39668,C(=O)(C(=O)CCC(C)C)NC1CC(C(=O)NC2C=C(C)CCC2)OCC1 39669,c1(C(N2CCC(O)(C(=O)Nc3c(OC)nccn3)C2)=O)cccc2c1CCC2 39670,N1(C(=O)CCCC2CCOCC2)CCC2(CCCN2C(=O)CCOC2CC2)C1 39671,c1(CC(=O)NCC2(O)CCN(C(C3CSCCS3)=O)CC2)cccc([N+](=O)[O-])c1 39672,C1(C)(CNC(C=NOC)=O)CC(F)(F)CN1C(c1ccc(C)nn1)=O 39673,C1(C2(O)CN(C(=O)CCC(F)(F)F)C2)(CNC(c2ccn3c2CCCC3)=O)CC1 39674,Cc1nc(=NN2CCC(C#N)CC2)n(-c2cccc(C(F)(F)F)c2)[nH]1 39675,c1(C(C(=O)NC2CCN(C(c3nncs3)=O)CC2F)O)ccc2ccccc2c1 39676,c1(C(N(C2CCC(CO)CC2)C)=O)n[nH]cc1[N+](=O)[O-].C12CC1CC(=O)NC2 39677,c1(OC)nn(C)cc1C(=O)NC1CC(CNC(CC2(OC)CC2)=O)C1 39678,c1(N(CC(=O)NCC2C(NC(c3c(C)scn3)=O)CC2)C)ccc(Cl)cc1 39679,C(=O)(C(C)(C)C(C)NC(=O)C(F)OC(F)(F)F)NC(CCC=C)(C)C 39680,c1(C(N2CC(CNC(C(CC)(F)F)=O)OC(C)(C)C2)=O)nccc2ccccc12 39681,C1(N(C)C(C2CNC(=O)C2)=O)CCCN(C(c2ccnc(O)c2)=O)CC1 39682,C1(C(C)C)(C(N2CCCCC2)=O)CCN(CC=CC2CCCC2)C1 39683,Cc1cc(Cl)ncc1NC(C1C=CC(NC(=O)Cc2cccs2)C1)=O 39684,C#CC1COCCN1C(c1ccc(OC)c(F)c1)C(=O)NCCOCC 39685,CCCCCCC(F)C(=O)NC1CC2CCC(C1)N2C(c1ccc(Cl)o1)=O 39686,NC(=O)CCCC(=O)NC1CCCCCC1NC(=O)CNC(=O)C(F)(F)F 39687,CN1CC2(CN(C(c3c[nH]nc3CNC(C3CC34CC4)=O)=O)C2)C1 39688,C1(C(=O)NC2C(NC(C(c3cccc(C)c3)F)=O)COCC2)CC2CCC1CC2 39689,C=Cn1nccc1C(=O)NC(CC1CCC1)C(=O)NC1(CC)CCOC1 39690,c1(OC)ccc(C(O)C(N2CCC(NC(c3nc(C(C)(F)F)cs3)=O)C2)=O)cc1 39691,C1(C(=O)NC2C(CNC(c3coc(-c4ccccn4)n3)=O)COC2)CCCCO1 39692,C1(C(=O)NCC(C(C)C)NC(C2CCN(CC(F)(F)F)CC2)=O)C2CCN1CC2 39693,Cc1cccc(-n2nc(Cn3nccn3)nc2-c2cnn3ccsc23)c1C 39694,C1(NC(C2(OC)CCCOC2)=O)CCCN(C(=O)C=Cc2ccn(C)c2)C1C 39695,C12(NC(C3CC4CCC3O4)=O)CCC1CN(C(=O)Cn1nc(O)ccc1=O)C2 39696,C1(C(N2CC(O)(CCC)C2)=O)(NC(=O)C(C)NC(C)=O)CCCC1C 39697,CC1(C)CCCC(NC(=O)CSCCNC(=O)CC2CC=CCC2)C1 39698,C(=O)(C(CN(C)C)C(C)C)N1CC(O)(C(CNC(C(C)C)=O)(C)C)C1 39699,c1(C(N2CC(COC)(NC(=O)CSc3ccccc3O)C2)=O)ccc(O)cc1 39700,N1(C(C23OCC(C)(C2)C3)=O)CCC(C2CC2)(CNC(=O)CCCC2CCC2)C1 39701,N1(C(C2(CC)CCCO2)=O)C2CCC(C2)C1C(=O)NC1C(C)C1(C)C 39702,c1(-c2nc(CCc3scc(C(N)=O)n3)on2)cc(F)cc(F)c1 39703,Cc1cncc(CC(=O)N(C(C)CN(C(=O)CC2CCCC(=O)C2)C)C)c1 39704,C1(CC(=O)N(CC(CNC(C(COCC)C)=O)C)C)CCCCC1(C)C 39705,c1(C(=O)OCC)ccc(NC(C2CCN2Cc2coc(C)n2)=O)cc1F 39706,C12(C(=O)NCCC3(O)CN(C(C(C)SC(C)C)=O)C3)CC(C)(C1)OC21COC1 39707,N1(C(Cc2c(C(=O)OC)nccc2)=O)CC2CC1CCN2C(C1(F)CCOC1)=O 39708,C1(NC(C(C2CCN(C(c3ccc(CC)nc3)=O)C2)(C)C)=O)CNC(=O)C1(C)C 39709,C1(CC)CCN(C(=O)NC2(CNC(=O)OC(C)(C)C)CCOCC2)CC1OC 39710,C1(F)(CNC(c2scnc2Cl)=O)COCCN(C(C2OCCCO2)=O)C1 39711,CCCC(C)(O)CC(=O)N1CC(NC(c2cnc(C(C)C)s2)=O)C(CC2CC2)C1 39712,c1(OCC)ccc(C(=O)NCCCCCCN(C(=O)CN2CCC2C)C)cn1 39713,c1(C(=O)NCC2CCCOC2)cn2cc(-c3ccncc3F)ccc2n1 39714,CC(O)C(F)(F)C(=O)NCCC(C)(C)CNC(=O)CCOCc1ccncc1 39715,N1(CCNC(c2cc(CNC(c3cnn(CCF)c3)=O)[nH]n2)=O)CCCOCC1 39716,C12(NC(c3c(CC)c[nH]c3)=O)CCN(C(C3(CC4CC4)CCC3)=O)CC1C2 39717,N#CC1(NC(c2csc(Br)c2)=O)CCN(Cc2cncs2)C1 39718,N1(C(Cc2cc(C(C)C)no2)=O)CCC(NC(=O)C(F)C(C)(C)O)C(CO)CC1 39719,C=CCC(F)(F)C(=O)NC1CC2CC1CC2C(=O)NCCc1nc[nH]n1 39720,C(=O)(C(F)CC(C)(C)NC(C1CC(=O)CC12CCC2)=O)NCC(=O)OCC=C 39721,C(=O)(C(F)CC(C)(C)NC(=O)CC1CCN(C)CC1)NCCC(C(C)C)C 39722,c1(C(C)=O)c[nH]c(C)cc1=NC1CCc2ncc(C(F)(F)F)cc2C1 39723,c1(OC)ccc(CNC(=O)C(N)Cc2cc(Cl)ccc2Cl)c(F)c1F 39724,CCC(CC(=O)N1CC2CC1CN(C(=O)C(C)(C)S(C)(=O)=O)C2)C(C)(C)C 39725,O=C(CCCCC(F)F)NCCC1CSCCN1C(=O)C(O)Cc1cnc[nH]1 39726,C1(COC(c2c(SCC)cccc2)=O)CCN(C(=O)CCc2ccc[nH]2)CC1F 39727,N1(C(c2cccc(CC)c2C)=O)CCC12CCN(C(c1cc(C(=O)O)c[nH]1)=O)CC2 39728,c1(CCC)cc(Cl)nc(NC(=O)C(N2CCCC(OC)C2C(=O)OCC)=O)n1 39729,C(CNC(=O)CC1(C)CCOC1)(CCNC(c1[nH]cnc1C)=O)OC 39730,C1(CNC(C=CCC)=O)CCC12CCN(C(=O)C=CS(F)(F)(F)(F)F)CC2 39731,N1(C2CCN(C(c3cc(COCC)[nH]n3)=O)C2)CCN(C(=O)CC(C)CF)CC1 39732,C(c1cncc(O)c1)=CC(=O)NCC1C(NC(C(C)(C)c2ccno2)=O)C1 39733,N#Cc1ccc(C(=O)NC2CCCC2CNC(=O)CC2CCC(O)C2)o1 39734,c1(CC)cc[nH]c1C(=O)NCCOCC(c1ccccc1)N1CCOCC1 39735,CCCC(O)(CCC)CC(=O)N1CCN(c2cc(CNC(=O)NC)ccn2)CC1 39736,CC1CCN(C(=O)CSCc2ccccn2)CC1CNC(=O)Cc1n[nH]c(=N)s1 39737,C1(NC(C(C)NC(=O)C2CC2)=O)C2CC3C(C2)C13C(=O)N(CCC[Si](C)(C)C)CC 39738,C1(CNC(C2CC(=C)C2)=O)CC2CN(C(c3cncc(COC)c3)=O)CC12 39739,N1(CC)CCC(NC(=O)C(c2ccoc2)NC(=O)C=CC(C)(C)C)C1 39740,CC(C(=O)NC(CNC(=O)C(=O)NCc1ncc[nH]1)CO)n1ccnc1 39741,N1(C(C(C=C)(C)C)=O)CC2(C1)C(NC(=O)C1Cc3ccc(F)cc31)CCS2(=O)=O 39742,Cn1nc2c(c1C(N1CCC1CNCC1(CO)CCCC1)=O)CS(=O)(=O)CC2 39743,C1(N(C(=O)C(C)COC)CC)CCCN(C(C23CC(OC(C)=O)(C2)C3)=O)C1 39744,C1(N(C(C(=O)NC)C)Cc2ccccc2)CCCN(C(c2ncn(C)n2)=O)C1 39745,c1(CNC(C(N2C(C(=O)NCC(C)N(C)C3CC3)CC2)C)=O)ccccc1 39746,c1(OC)cnnc(C(=O)NC(C)CCCNC(=O)C(C)OCC2CC2)c1 39747,C(C1=CCN(C(C2CCC(=O)NC2)=O)CC1)NC(=O)CCc1ccccc1F 39748,C(CCCCC(=O)N1CCC(C(=O)NCC2CC2(Cl)Cl)C1(C)C)OC 39749,Cc1ncc(C=CC(=O)NC2(CN(C)C(C3CC(C)(CO)C3)=O)CC2)s1 39750,c1(C(C(=O)NC2CC(CCNC(c3cnc(CC)s3)=O)C2)(F)F)ccccc1F 39751,C1(CNC(CCNC(N)=O)=O)CCCCC1NC(C12CC(CF)(CO1)C2)=O 39752,Cc1[nH]c2ccccc2c1C(N1CCCCC(CNC(c2cnns2)=O)C1)=O 39753,C1(C(=O)NCCC2CNC(=O)O2)CC1C1CCN(C(=O)C2=CCCOC2)CC1 39754,N1(C(CNC(C)=O)=O)CCC(NC(c2cnn3c2C(C)CCC3)=O)CC(C)(C)C1 39755,C1(CNC(CCC(=O)OC)=O)COC(C)(C)CN1C(C1CC2CCC(C1)N2C)=O 39756,N1(C(c2nnn(C)c2C(F)F)=O)CCC2CCN(C(c3cccc(Cl)c3)=O)CC12 39757,c1(C(=O)NCC2(CNC(C(C(C)C)O)=O)CC23CCC3)nc(O)nc(O)c1N 39758,N1(C(C(CC)=CC)=O)CCC2(CCCCN(C(C34CCC(F)(CC3)C4)=O)C2)C1 39759,N1(C(C2(C(C)C)CC2)=O)CC(C)(C)C(NC(=O)CC(C)(C)CN(C)C)C(C)(C)C1 39760,C12(CNC(C=CC(C)(C)C)=O)CN(C(=O)CCc3ccccn3)CC1(C(F)F)C2 39761,C1(CCC)CN(C(=O)CC2CCSC2)CC1NC(N1CCC(C(=O)OC)C1)=O 39762,c1(OC)cnccc1C(=O)NCCC1CCCCN1C(c1cc(C(C)=O)c[nH]1)=O 39763,c1(CN(CC)Cc2cc(C(F)(F)F)ncc2F)c2ccccc2cc2ccccc12 39764,C#Cc1cc(F)c(C(N2CC3CC3(NC(C3COC3)=O)C2)=O)cc1F 39765,O=C1COc2cc(C(N3C4CCC3CN(C(C3CCC5CC35)=O)C4)=O)ncc2N1 39766,N1(C(CCC2CCC(NC(C(C=C)(C)O)=O)C2)=O)CCC2(CCC2)C(O)C1 39767,C1(C(=O)NCC23CC(NC(c4ccn(C)n4)=O)(C2)C3)CCC(F)CC1 39768,c1(C(=O)NCC(CCC)C(=O)N(CCC(F)(F)F)C)ncn2ccccc12 39769,CC(C)CCCC(C)C(=O)N1CCC(CCNC(c2cc3occc3[nH]2)=O)C1 39770,C1(CNC(c2c(C)occ2C(F)(F)F)=O)CC(F)(F)CN1C(c1ccno1)=O 39771,c1(CC)nc(C(=O)NCC2(NC(=O)Cc3ccnc(C(N)=O)c3)CCC2)c(C)o1 39772,c1(C(=O)OC)occc1CNCCNC(=O)CNC=O 39773,C1(C)(NC(c2c(OC)c[nH]n2)=O)CCN(C(c2cccc(I)c2)=O)C1 39774,C1(C(N2C(CCNC(Cc3c(C)cnn3C)=O)CSCC2)=O)Cc2cscc2C1 39775,C1(N(CC(C)C)C(=O)COC2CCCC2)CCN(C(C2CC(F)C2)=O)C1 39776,C(c1cc(C)ccc1OC)=CC(=O)N(CCCCNC(CC(COC)C)=O)C 39777,N1(C(C(C(C)C)SC)=O)CCCCC(NC(=O)COc2cc(C)on2)C1 39778,Cc1ccc(C(N2CCCC2C(C)(C)CNC(C2OCC2(C)C)=O)=O)n1C 39779,c1(NC(CC2(C)CN(C(CN3CCN(C)CC3)=O)C2)=O)cc(F)cc2[nH]ncc12 39780,c1(NC(c2cc(C)sc2)=O)cnn(C)c1C(N1CCN(C(C)C)CC1)=O 39781,C(C)(CCCCNC(=O)CCc1nnc(C2CCCC2)o1)NC(C1C(C)C1C)=O 39782,Brc1c(-c2nc(C3CCCOCC3)no2)nc2n1CCC2 39783,N1(c2cc(C)nc(C3CCC3)n2)CCC(C)C(NC(=O)CC2CC=CCC2)C1C 39784,C1(O)(CNC(CCCC)=O)CCCN(C(=O)CC(O)C(C)C)C1 39785,c1(SC)cncc(NC(=O)CC2(C)CCN(C(=O)Cc3coc(C)n3)C2)c1 39786,CCCCCS(=O)(=O)CC(=O)NCC1(OC)CN(C(=O)C(O)c2cnc[nH]2)C1 39787,c1(CCC)c(NC(N2CCCC(CF)C2)=O)nnn1Cc1ccccc1Cl 39788,c1(C(=O)NCC(CO)NC(c2cn(C3CCOCC3)nn2)=O)ccc(Cl)nc1O 39789,c1(CCNC(C2N(C(CS(C)(=O)=O)=O)CCC(O)C2)=O)ccc(S(=O)(=O)F)cc1 39790,C(C1=CCN(C)CC1)NC(C1(NC(=O)CC2C(C)(C)C2(C)C)C(C)C1)=O 39791,N1(C(c2cnc(C(C)C)s2)=O)CCC(C)C(CNC(=O)C#CC(C)(C)C)C1 39792,N1(CC)CCN(C(C2N(C(=O)CC3CC4C=CC3C4)CCC2(C)C)=O)CC1=O 39793,c1(C(N(C2CCCC(NC(=O)CCF)C2)C)=O)ccc(P(C)(C)=O)s1 39794,c1(C(=O)OC)ccc2c(c1)OCCN(C(=O)CSCC(C)C#N)C2 39795,n1(C(C(=O)N(CCNC(=O)CN(CC(C)(C)C)C)CC)C)ccc(C)n1 39796,c1(OC)ccccc1N(C(c1cccnc1OC)C(=O)NCc1cccs1)C 39797,C(=O)(C1=C(C#N)CCC1)NCC1CC(C)(C)CN1C(C1COCC1(C)C)=O 39798,C1(C(N2CCC(n3cc(C(N4CCCC4)C)nn3)C2)=O)CCc2nncn2CC1 39799,Cc1ccncc1CCNC(=O)CC1CC(NC(C2C(C#N)C2(C)C)=O)C1 39800,C1(C(=O)NC(C=C)C)CC12CC(NC(c1c[nH]nc1C1CC1)=O)C2 39801,CC(C)CC(C(=O)NC1CC2C1CCN2C(=O)CC1CN2CCC1CC2)C(N)=O 39802,c1(OC)cccc(NC(=O)NCC2(CNc3cc(Cl)ccn3)CC2)c1 39803,C1(CNC(CSc2n(C)ccn2)=O)CCCCN1C(c1cn(C2CC2)cn1)=O 39804,N1(C(C2CCC(=O)N2)=O)C2CCC1(CNC(c1cn(CCO)nn1)=O)CC2 39805,c1(C(CCC)NCCc2ccncc2)nnnn1Cc1nnn(C)n1 39806,N1(C(=O)NC(c2cccc(Cl)c2)CC)CCC2(CSC2)C1 39807,Cc1ccc(F)c(O)c1C(=O)NC1CCCCN(C(=O)CCC2CC2)C1 39808,N1(C(CCCCOC)=O)CCC(C)(C)C(NC(=O)C(C(C)CC)NS(C)(=O)=O)C1 39809,C1(NC(CCC#C)=O)CCCC(N(C(=O)CCc2ccco2)C)C1 39810,C1(CNC(C2(C)CC2C(F)(F)F)=O)CCCN1C(=O)CC1CCOC1=O 39811,Cc1cc(C(C)NCC(C)CCCO)ccc1[N+](=O)[O-] 39812,c1(OCCC(=O)NC(C(C)NC(=O)C(C2CCCCC2)O)CO)cccc(F)c1 39813,C1(CC(N2CCC(CN(C(=O)CCC3CC3)C)C2)=O)CCCCCC1 39814,C1(CC(N2CCC(NC(C(C#C)(C)C)=O)C2C(C)(C)C)=O)NC(=O)CN(C)C1=O 39815,C1(CC(=O)NCC2(C(=O)NCC(CCNC(N)=O)O)CC2)CC2CCC1O2 39816,C(CCCCC(=O)NCC1CCCCC1NC(c1c(C)[nH]c(C)c1C)=O)=CC 39817,C(=O)(C(C)(C)CCC#N)NCCC(C)N(C)C(C1OCCN(C)C1=O)=O 39818,C(C)(CCCC(=O)N1CCOCC1C(C)(C)C)NC(COCCCC(C)C)=O 39819,Cc1cc(CNC(N2CC3CCC2C(C(=O)NC(C)(C)C)C3)=O)ccc1[N+](=O)[O-] 39820,c1(C(=O)NC2CN(C(C(CO)NC(N)=O)=O)C2)cc(Cl)c(Cl)cc1N 39821,C=CCCCCCC(=O)NC(C(=O)NC1CC(C)(C)OC1(C)C)C1CC1 39822,Cc1ccc2n[nH]cc2c1C(N1CCC2(CC1)CC2NC(=O)CCC1CCC1)=O 39823,N1(C(C2CCC2)=O)CCCC2C1CCN2C(c1sccc1F)=O 39824,N1(C(C(CC=C)NC(C)=O)=O)CCC(C(=O)NCc2nccs2)C1(C)C 39825,C1(F)(C(=O)NCCC2(CNC(C(C)C3CCOC3)=O)CC2)C(C)(C)C1(C)C 39826,CC1CCCC(OCC(=O)N(C)CC2CN(C(C3CCCC4CC34)=O)C2)C1 39827,c1(C(=O)NS(CCC(C)(C)C)(=O)=O)cc2cc(F)ccc2cn1 39828,C12(C(=O)NCCN(CCCC)C)CCC(CC1NC(c1cncc(O)c1)=O)C2 39829,CC1OC(C)C(C(=O)NC(C2CCN(C(C3CCCS(=O)(=O)C3)=O)CC2)C)C1C 39830,Cc1cc(=NC(C)CN(C(=O)Cn2nc(C)c(Cl)c2C)C)[nH]c(C)n1 39831,C(=O)(C(F)CC(C)(C)C)N1C(CC(=O)NC(C(=O)OC)C2CCC2)CCC1 39832,c1(C(N2CCC(CN(C(CCc3c(C)noc3)=O)C)C2)=O)cc(Cl)nn1C 39833,C(=O)(C1=NN(CC(C)C)C(=O)CC1)NC1C2N(C(C=NOC)=O)CC(CC2)C1 39834,c1(OC)c(C(=O)NC(C)CCc2cc(F)cc(F)c2)ccc([N+](=O)[O-])c1Br 39835,N1(C(c2c(OC)nsc2)=O)CCC(C=CC(=O)NCCC(O)C(F)(F)F)CC1 39836,Cc1cc(C2CC2)ncc1C(=O)NC(C1CN(C(c2ccncc2Cl)=O)C1)C 39837,Cc1cnc2ccc(C(=O)N(C)Cc3cccnn3)cn12 39838,O=C(NN1CCCC1C(=O)NCc1ncsn1)C1CC(CC2CC2)C1 39839,N1(C(CNC(C2C(C)C2)=O)=O)CCCCC1C(=O)NCC12CCN(CC1)C2 39840,c1(C(=O)OC)cc(C(N2CCN(C3CCOC3)CC2)C(=O)NCCCF)nn1C 39841,C#CC(CC1CCOC1)NC(=O)CCC 39842,c1(CC)cc(CC)nc(N(C)CC2(CNC(=O)C(F)=C(C)C)CC2)n1 39843,C1(C(=O)NCCCNC(C(C)c2ccon2)=O)CSc2ccccc2O1 39844,N1(C(C2(C)CC(=C)C2)=O)CC(N(C(=O)CCc2cc(C)cc(C)c2)C)C(C)(C)C1 39845,C(=O)(C(F)(F)C(F)F)N1CC(C(C(=O)NCC(C)Cc2cn[nH]c2)O)C1 39846,C(=O)(C(F)CC(C)(C)NC(c1ccc(F)cc1C)=O)NC(C#C)CC(C)C 39847,CN1CCN(C(=O)C(C2(O)CCCC2)F)C(CNC(=O)CCC2CCC2)C1 39848,c1(-c2cc(C)c(F)c(C)c2)cc(C(N2CCC(C)C(F)(F)C2)=O)cc2[nH]ccc12 39849,C(CCC(=O)NCC1CC(CNC(C2(C)CC2(F)F)=O)CO1)C1C(C)C1 39850,c1(C(N(c2cccc(C)n2)CCC)C2CC2)cc(C(C)(C)C)ccc1O 39851,c1(OC)cc(C=CC(=O)NC2CC(NC(=O)C(O)C3CCC3)C2)ccc1O 39852,C=C=CCCC(=O)NCC(=O)NC1CCCC1.c12noc-1n2 39853,c1(CC)[nH]nc(C(=O)NC2(C(=O)NCCCN(C)OC)CCCC2C)c1C 39854,N1(CC(=O)NCC2CCC3(CCC3)O2)CCC2(C=CCO2)CC1 39855,c1(CC(=O)OC(c2ccccc2)C)c(F)cccc1F 39856,c1(CCC(=O)NC(CCCNC(c2c(C)n[nH]c2C)=O)C)ccc(Cl)cc1Cl 39857,n1(CC(=O)NC2(C3CN(C(C4(C)CC=CCC4)=O)C3)CC2)ncc2ccccc12 39858,C1(N(C(C(C)NC(=O)NC)=O)CCO)CN(C(=O)CN2CCNC2=O)CC1(C)C 39859,N1(C(c2cc(C)n(C(C)C)n2)=O)CC(CNC(c2n[nH]cc2Br)=O)OC(C)(C)C1 39860,NS(=O)(=O)C1(C(=O)NCC2CC3CCC2N3C(=O)C2=CCCO2)CCCC1 39861,c1(CCOC)cc2oc(=O)n(-c3ccccc3)c2cc1OC 39862,Cc1cccc(C(=O)NCC2CCCC2NC(c2c(F)cccc2F)=O)c1C 39863,c1(C(=O)NCC(C)NC(CSc2c(C)n[nH]c2C)=O)cnc(N)c(N)c1 39864,C(=O)(C(C)(C)CS(C)(=O)=O)NCC(CNC(C1C(C(C)(F)F)C1)=O)C(F)(F)F 39865,n1(C(C(=O)N(CC(C)(C)NC(C=CCN(C)CC)=O)C)C)nccc1C 39866,Cc1ccn2c(C(=O)N(CC(C)(C)CNC(=O)CC(=O)NC3CC3)C)cnc2c1 39867,c1(C(=O)NCC2(O)CN(C(CNC(c3cn(CC)nc3)=O)=O)C2)cccc(F)c1 39868,c1(NCc2ccc(OCC(=O)NCC)c(OC)c2)cc2c(s1)CCOC2 39869,C1(C(=O)NCCc2cn(CC)nn2)C=CCCN1C(=O)CCCCOC 39870,C1(NC(C2(C#C)CCCC2)=O)CC2CC1N(C(=O)C(CC)=CC)C2 39871,C(CN=C(NCC)NC1CCCN(C(=O)OC(C)(C)C)C1)N(CCC)CC1CC1 39872,CC1N(C(C2CCC2NC(c2ncn(C)n2)=O)=O)CCCC12CCC2 39873,Cc1nc(O)ccc1C(=O)NCCc1cc(C(=O)N(C2CCC2C)C)no1 39874,Cc1cc(NC(=O)Nc2c[nH]nc2C2CC2)n2ncnc2n1 39875,N1(C(C23N(C(C(C=C)C)=O)CCC2C3)=O)CC2(CC(CO)CO2)C1 39876,N#Cc1ccc(-c2cn(C3CCCN(C(c4sccc4CO)=O)C3)nn2)s1 39877,C1(C(=O)NCC2(CCNC(C3(N(C)C)CCCCC3)=O)CC2)CCCCC(=O)C1 39878,c1(C(=O)NCC=CCNC(C2C(C)C2)=O)ccc(N2CCC(C)CC2)nc1 39879,c1(C(N2CC(N(C(=O)COCCOCC)CCC)C2)=O)ccncc1CC 39880,Cc1cccc(C)c1CC(=O)NC1CCC(NC(C2CCC(C)S2)=O)CC1 39881,C(N=c1nc(NC(N2CC3CC3C2)=O)cc(C)[nH]1)c1ccc(CSC)c(F)c1 39882,N1(C(C(C2CCC2)OC)=O)CC(NC(c2cc(Cl)c(F)cc2F)=O)C(N=[N+]=[N-])C1 39883,N1(C(CCCOC)=O)CCCC(CO)(CNC(c2ccon2)=O)C1 39884,c1(C(=O)NC2CC(CNC(C3CCN(C)CC3)=O)C2)cc(F)ccc1N 39885,N1(C(c2[nH]cc(CC)c2)=O)CCC(N(C(c2ccc(CN(C)C)s2)=O)CC)CC1 39886,C(=O)(CCC(C)(C)O)NC(C1CN(C(=O)C2=CCCCC2)C1)C 39887,c1(OCC#C)ccc(F)cc1CNC(=O)NCC1COCCC1c1ccccc1 39888,N1(C(c2cncc(N)c2)=O)CCN(C(c2cc3c[nH]nc3s2)=O)C2CC12 39889,C(=O)(C(=O)CC(C)CC)N1C(CNN(C(=O)CS(=O)CC)CC)CCCC1 39890,c1(C(=O)NC2CCC(NC(c3c(C(C)C)nns3)=O)CC2)cc2c[nH]cnc-2n1 39891,n1(CC)c(=O)c(C)nc2cc(C(N3CC(NC(C4CCC4CF)=O)C3)=O)ccc12 39892,Cc1cc(C(=O)CCC(=O)NCCCCCNC(C2CC2C)=O)c(C)s1 39893,CC1(C)CCC2CCN(C(=O)NC3CCOC3)c3cccc1c32 39894,C(=O)(C1OCCc2ccccc21)NC1(CC=C)CN(C(=O)C(C)(F)C(F)(F)F)C1 39895,S(=O)(=O)(c1[nH]c(=NC(C)Cn2ccnc2)ccc1Br)N(C)Cc1c(C)cccc1 39896,c1(-c2cnc(NC(C(C)(C)Br)=O)s2)cccc2cc[nH]c12 39897,CCC(C)(C#N)C(=O)NCc1nnc(C2CCN(C(=O)C3=CCC3)CC2)s1 39898,C(=O)(C(C(C)C)NC(=O)OC)NCCN(C(CCC=CC)=O)CC 39899,c1(C(C)=O)cc(C(=O)NCC(n2cc(-c3cccnc3F)nn2)C)c(C)o1 39900,C1(C2CCOCC2)(C(N2CCN(CC(C)NC(CCSC)=O)CC2)=O)CC1 39901,C1(C(=O)Nc2cccc(NC(C3(C)ON=C(C)C3)=O)c2)CCc2nnnn2C1 39902,C1(CC(=O)N(CCOCCN(C(C(C)N(C)C)=O)C)C)CCCSC1 39903,C(=O)(CC(C(=C)C)OCC)NC1CC2(C(NC(CC3(CC=C)CCCC3)=O)C2)C1 39904,c1(C(=O)NC(C2CCN(C(C(CC)OCC)=O)C2)(C)C)cc2n(n1)CCO2 39905,C1(NC(C2N(C(C)=O)CCC2)=O)CC2(C1)CN(C(=O)CC1C(=O)N(C)N=C1C)C2 39906,C(=O)(C(F)C(=O)NC1CC(CNC(=O)Cc2cc(=O)n(CC(C)C)[nH]2)C1)OCC 39907,Cc1ccc(CNC(C2(CNC(C3(c4cc[nH]n4)CC3)=O)CCC2)=O)cn1 39908,N1(C(c2ccnc(OC)n2)=O)CCC2(CNC(=O)C(C)=C3CCC3)CCCCC12 39909,C1(C(N(CCNC(C2CCCC(C)(C)C2)=O)CC)=O)CC12CCCCCC2 39910,C(=O)(CCCCC(F)F)N1CC2C(NC(c3ccc(N)cc3F)=O)C(C2)C1 39911,n1(CC)cc(Br)cc1C(=O)NCCOCCNC(C1(CF)CC(F)(F)C1)=O 39912,C1(CC=C)CCCCC1NC(c1ncnn1CCCC)c1nnnn1C1COC1 39913,C=C=CCCNC(=O)C(C)c1cccs1.C1(=O)C(C)O1 39914,Cc1cc(CNCc2cnc(N3CCOCC3)s2)c(O)c(Br)c1 39915,c1(C(=O)NC(CN(C(=O)CC2(N3CCCC3)CC2)CC)C)cccnc1C(F)F 39916,c1(NC(=O)NC2C(CCCC)CCC2)ccc2nc(OC(C)=O)[nH]c2c1 39917,C1(N(C(Cc2c(C)scc2)=O)C)CCCC(NC(=O)C=CBr)C1 39918,c1(C(=O)NCCC2CCN(C(CN3C(C)CCC3)=O)C2)cc(N)c(F)cn1 39919,C(=O)(CC(F)(F)F)N(CC(C(=O)NCC(=O)OC(C)C)C)C 39920,CC1=C(C(=O)NCC2CCCN2C(C2(C(F)(F)F)CCC2)=O)CCO1 39921,C1(C(N(CCn2c(C)ncc2)C)=O)CCCN(C(C2C=CCC2)=O)CC1 39922,N1(C(CC(=O)OC)=O)CCOC2CN(C(c3n[nH]c4cc(C)ccc34)=O)CC12 39923,c1(C(N2C(C)CCC(CNC(C(CC)N(C)C)=O)C2)=O)cccc2ccsc12 39924,N1(C(=O)Nc2ccc(Sc3ccccn3)c(Cl)c2)CCc2[nH]ccc2C1 39925,C(=O)(C(CC1CC1)NC(=O)CC=CC(C)(C)C)N1CC(CCC#C)C1 39926,c1(OC)ncc(C(N2CC(N(C(=O)CN(C)C3CC3)C)C(O)C2)=O)cc1F 39927,c1(Nc2c(C(=O)OC)cc(O)cc2)nc2ccccc2s1 39928,N1(C(c2c(C)nc(C)[nH]2)=O)CCN2CCOCC2(CNC(=O)CC(C)F)C1 39929,c1(C(=O)NCC(CC)(CC)NC(=O)C(F)CC(C)C)snc2ccccc12 39930,C1(SC)CN(C)CCN1c1cc(SC)ncn1.C1(N2CC2=O)CCCC(C#N)C1 39931,c1(C(=O)NC2C(NC(CC(COC)C)=O)C2)cccc(=O)n1C 39932,Cn1cnc2nc(=NCC3CCC(NC(=O)COC(F)F)C3)[nH]cc12 39933,N1(C(C2(C)C=CCN2C(=O)CN2CCSCC2)=O)CC2CC1CC2CF 39934,N1(c2nnn(C)n2)CCCC12CCN(C(c1cccc3c1CCOC3)=O)C2 39935,C1(C(N2CC(c3n(C)ccn3)C(NC(=O)C3=CCC3)C2)=O)Cc2cscc2C1 39936,N1(C(COCC(=O)OC)=O)Cc2ccccc2CC1CNC(=O)Cc1csnn1 39937,C(c1ccccc1F)=CCC(=O)NCCN(C(=O)CC1CCOC1)C 39938,C1(N(C(CN(C(=O)CC2CC=CCC2)CC)=O)C)CCN(C(C)C)C1 39939,CC1CCC(=CC(=O)NC(C)CNC(=O)C(C)N2CC(C)C2)CC1 39940,C1(C(N2CCOC(CCNC(c3cccc(Cl)c3)=O)C2)=O)(CSC)CCOCC1 39941,N1(C(C2C(C)(Br)C2)=O)CC2(C1)CN(C(c1nc[nH]c1C(F)(F)F)=O)C2 39942,C1(C(N(CCCCN(C)C(C2(CO)CC(C)(C)C2)=O)C)=O)CCC2(CCC2)OC1 39943,CCC(C)C(O)C(C)C(=O)NCC1(NC(=O)Cn2cc(C(=O)NC)nn2)CCC1 39944,C1(NC(c2ncn(C(C)C)c2)=O)CN(C(C2(O)CCOC2)=O)CC1C 39945,N1(C(C2C(CC)C2)=O)CC(NC(c2c(C)ncn2OC)=O)CC12CCCCC2 39946,CC(C)(C(=O)NCC1(CNC(=O)CC2CCCO2)CC1(F)F)c1ccccn1 39947,c1(OC)c(C(=O)NC2CN(C(c3c(N)cccc3Cl)=O)C2)oc2ccccc12 39948,C1(CC)C(C(=O)NCc2ccc(C)cc2)CCN1C(=O)C(C)O 39949,N1(C(CCC(=O)NC)=O)CCC(C2CC2)C1CNC(c1cnc(C)c(OC)c1)=O 39950,c1(OC)ccc(C#N)cc1NCc1nc(Nc2ccc(F)cc2)[nH]c(=N)n1 39951,N1(C(c2cccc(CNC(CCCCC#C)=O)n2)=O)CCC2C(CCN2C)C1 39952,c1(C(=O)NCCC2(NC(c3cncc(N(C)C)c3)=O)CC2)nc[nH]c2ncnc1-2 39953,c1(C(C)(C)NCCc2ccncc2)ccnc(Cl)c1F 39954,C(=O)(C1CCc2cccc(F)c21)N1CC(COC)OC(C)C1 39955,C(CC1=CCOCC1)NC(C(CC)N(C)C(c1cn(C)c(=O)cn1)=O)=O 39956,C1(NC(c2cc(Cl)no2)=O)CCC12CCN(C(=O)CCC1CC1)CC2 39957,N1(C(Cc2nc(C)sc2C)=O)CCCN(C(=O)CC(C)c2ccco2)C(CO)C1 39958,N(C(=NCCC)NC1CC(CC(N)=O)C1)C(C#C)CC 39959,C1(NC(N2CCC(NCC(C(C)C)(F)F)CC2)=O)CCC2(CCOCC2)C1 39960,Cc1ccc(CC(=O)NCC(C(C)(C)C)NC(=O)CC2(O)CCOCC2)c(C)c1 39961,N1(C(Cc2scc(C)c2)=O)CC(C)CN(C(=O)C(N2CCCCC2)C)C(C)C1 39962,C(C)(C)(CC(=O)NC(c1cn(C)nn1)C)NC(C=CCCC)=O 39963,c1(C(N2CC(CNC(CCC3(C)CCC(=O)N3)=O)C2)=O)cc2cc(Cl)ccc2o1 39964,C(=O)(CC(C)C(C)(C)NC(c1cnc(N(C)C)o1)=O)N1CCC(C)(CCC)C1 39965,c1(CC(=O)NC(CCNC(C2(OC)CC2)=O)C)csc2ccccc12 39966,c1(C(=O)NC(C2CCN(C(c3csc(C)c3N)=O)CC2)C)ccn2nnnc2c1 39967,c1(C(=O)NC2CCN(C(C(C)N(C3CCCCC3)C)=O)C2)cn2cnnc2cn1 39968,C1(NC(c2ccn(CC(C)C)n2)=O)CCN(C(=O)CC2CCC2)C1C1CC1 39969,CCC(C(=O)NC(CNC(=O)CC(C)N(C)C)CC(C)C)C(C)(C)CC 39970,C(=O)(CCC(C)(F)F)NCCN(CCC)C(c1c(Cl)cncc1Br)=O 39971,CC1Cc2ccccc2N1C(=O)CC1(NC(C2C(C(=O)O)C2(C)C)=O)CCC1 39972,CC(C)(CC(=O)NC1CCC(CNC(C2CCCC3CCCN23)=O)C1)C(F)F 39973,C1(C#N)(C(=O)NCC2CCC(NC(c3scc(C)c3Cl)=O)CC2)CC12CCCC2 39974,C1(C(N2CCC(OCC(N)=O)C2)=O)CCC(C)(C)N(C(C2CC2(Cl)Cl)=O)C1 39975,c1(CC(=O)N(C)CC2CCCN2C(C23CC(F)C2C3)=O)cc(Cl)sc1Cl 39976,CC(Cl)(Cl)C(=O)N1CCC(C2CCCN2C(c2csc(-c3ccco3)n2)=O)C1 39977,N1(C(C(CC#C)C)=O)CCN(C(C2(c3cccc(Cl)n3)CC2)=O)CC1C1CC1 39978,C1(OC)(CNC(C2C3CCCOC23)=O)CCN(C(=O)Cn2ncccc2=O)C1 39979,C#CCCC(C(=O)NCC(c1ccco1)O)NC(=O)C=C1CCC(C)CC1 39980,c1(C(N2CC(CNC(c3c(NC)snc3C)=O)C(C)C2)=O)cn2ccccc2n1 39981,c1(N(CC(=O)NC2CC2NC(=O)C(F)C2CCC2)C)ccc(C#N)c(Cl)c1 39982,C(=O)(C(F)C(F)(F)F)NCC1(F)CN(C(C(C)CO)=O)C1 39983,C1(C(=O)NC2(CNC(c3ccc(C#N)cn3)=O)CCOC2)C2(CCC2)C12CCC2 39984,N1(C(C(C(COC)C)C)=O)CCCC2(NC(C3CCCCC3C)=O)CCCC12 39985,O=C(C1=C(Cl)CCOC1)NC1CC(NC(c2cc(C(F)(F)F)nn2C2CC2)=O)C1 39986,c1(CC)ccccc1C(N1CCC(CCC(=O)NC2CCOCC2OC)C1)=O 39987,N1(C(C(C)NS(C)(=O)=O)=O)CCC(F)(CNC(=O)CNC(C2CCC2)=O)C1 39988,N1(C(Cc2c(C)scc2)=O)CC2CN(C(=O)C(=O)NC(C)C)CCC2(CO)C1 39989,C(=O)(C1=NOC(C)(C)C1)N1CC(NC(c2cnc(C(C)C)s2)=O)C(C)CC1 39990,C12(C(=O)NCC(C)(C)OC)CCC1CN(C(=O)CCN1CCN(C)CC1)C2 39991,C(=O)(C(C)S(N)(=O)=O)N1CCC(OCCNC(Cc2c(C)ocn2)=O)C1 39992,C1(C#CC(=O)NCC2CN(C(C34CC5CC3C4C5O)=O)CC2(C)C)(CC)CC1 39993,C(CC)(C(=O)NC1CCC1C(=O)N(C(C)CC1CC1)C)=CCCC 39994,O=C(CC1=CCCCC1)N1CCC2(CC2C(N2CCCC2CCO)=O)C1 39995,Cc1ccc(C(=O)C(=O)NC2CCC2CNC(C2CCCCC2)=O)cc1 39996,N1(C(c2c(CC)occ2C)=O)CC2CCCCC2(NC(=O)CC2CC23CC3)C1 39997,C1(O)(CNC(c2cc(-c3ccco3)no2)=O)CCCN(C(C2SCCS2)=O)CC1 39998,C(=O)(C(F)(CNC(=O)Cc1nocc1C)C(C)C)N1C(CC)CCC1 39999,N1(C(C2CC(C)OC2)=O)CC2CN(C(c3ccc4nccn4c3)=O)CC(C1)O2 40000,N1(C(Cc2nc(C(C)OC)sc2)=O)CC2CC1CN2C(c1sccc1F)=O 40001,C1(C(=O)Nc2cn(CC)nc2)CC12CCN(C(=O)COC(C)=O)CC2 40002,C1(CNC(C2(C)ON=C(C)C2)=O)Cc2ccccc2CN1C(=O)Cc1ccns1 40003,N1(C(C(C)(C)c2ccccn2)=O)CC2CN(C(=O)CC3CCCCC3(F)F)C2C1 40004,Cc1ccnc(O)c1C(=O)NCC1(CNC(C2C3COCC23)=O)CC(F)(F)C1 40005,c1(OCC)ccc(CCC(=O)NC(C)CC2CCN(C(=O)CSCC)CC2)cc1 40006,CC1CCCN(C(C)CNC(=O)NC2CN(Cc3ncccc3C(F)(F)F)C2)C1 40007,C12(C(=O)NC3C(NC(c4n(C)cc(C#N)c4)=O)CCC3)CC3CC(CC(C3)O1)C2 40008,c1(C(=O)NC(C(C)NC(CCN(CCC)C)=O)C)noc2c1CCCCC2 40009,C1(C)(C(N2CC(O)(CN(C(=O)CNC(c3cscn3)=O)C)C2)=O)C=CCCC1 40010,C(=O)(CCCNC(C1CCC1)=O)NC(CN(C(C1(C#C)CC1)=O)C)(C)C 40011,c1(C(N2CC(C3CN(C(C(C)(C)C#N)=O)C3)C2)=O)cc2ccsc2c(O)n1 40012,C1(NC(CCC(C)C)=O)CCCC12CN(C(C1(C)CCN(C)C1=O)=O)C2 40013,C1(C)(CNC(c2c(C)cno2)=O)CCCN1C(=O)CCSCC(N)=O 40014,Cc1noc(C)c1C(C1(CC2CCC2)CC1)Nc1cc(N2CCCC2)ncn1 40015,Cc1ccc(C(F)(F)F)c2c1N(C(N1CCCCC(N(C)C)C1)=O)CC(C)C2 40016,C(C)(CN=c1nc(C(=O)OC)[nH]cc1OC)NC(c1cc(OCC)ncc1)=O 40017,C1(C(=O)NC2(C(=O)NCC(O)CC3CCC3)CCN(C)C2)CCC2(CCC2)O1 40018,C1(C2C(C)C2)CC2CCC(C1)N2C(C1CCN(c2cc(F)cc(Br)c2)CC1)=O 40019,N1(C(C(C)N(C)C(=O)OC(C)(C)C)=O)CC(NC(=O)CCC(F)F)CC1C 40020,C(C(O)C(=O)N1CC(O)(C2CCCN2C(=O)CCc2nc(=N)[nH][nH]2)C1)SC 40021,N(C1CCCc2cn(C)nc21)C(C1CCCO1)CC 40022,N1(C(C(C)NC(CC)=O)=O)CC(CO)C2(C1)CN(C(=O)CC(C)(C)CCOC)C2 40023,N1(C(C2(CC=C)CN(C(c3cc(C)c(C)[nH]3)=O)C2)=O)CC(N(C)C)C(C)(C)C1 40024,N1(C(C(C2CCC2)OC)=O)CCC2CN(C(=O)Cc3cc[nH]n3)C(C)C12 40025,N1(C(CC(=C)Br)=O)CCC2(CCCN(C(=O)CCOC3CCCC3)C2)CC1 40026,C1(CNC(c2c(OC)ccs2)=O)CC(NC(c2ccc(C)nn2)=O)C12CCC2 40027,Cc1c(C(N2C3CCC(C3)C2C(c2nc3ccccc3s2)=O)=O)cc(Br)cc1F 40028,S(=O)(=O)(c1cccs1)NCCC(=O)NCC1(O)CN(C(C2(C)CC3(CC3)C2)=O)C1 40029,c1(CNC(c2c(CC)noc2)=O)ccc(CN(C(=O)CC2CC3CC3C2)C)cc1 40030,Cc1ccc(C(=O)NCC2(NC(c3ccn(C4CC4)c3C)=O)CC2)nc1O 40031,c1(C(CN(C2CC(C)(C)C2)Cc2ccccc2)O)ccc(F)cc1 40032,N1(C(C2CCN(C(C)=O)CC2)=O)CC2CCN(C(=O)Cc3cnccn3)C2C1.C(C=O)N 40033,N1(CC(=O)NCC2(CCCC)CCC2)C(=O)c2ccccc2C1=O 40034,N1(C(C2=C(C)CC2)=O)CC2CC(NC(c3nccc4n[nH]cc34)=O)C(C2)C1 40035,c1(C(=O)NC2C(CNC(C(CCC)OCC)=O)C2)cc(OCC)ccc1C 40036,c1(N2CCC(O)(C(C)NC(c3cn(CC=C)nn3)=O)C2)ncc([N+](=O)[O-])cc1Cl 40037,c1(OCCCC)ccc(C(=O)NC2CCCC2NC(c2n[nH]cc2Cl)=O)c(O)c1 40038,C1(C(N2CC(CC)(CO)C2)=O)CCN(C(c2cnn(C3CC3)c2)=O)C(C)(C)C1 40039,c1(C(=O)OC)sc(C(N2CCC(NC(C3(CC(F)F)CCC3)=O)CC2)=O)cc1N 40040,O=C1NCC2CN(C(c3ccccc3OC(F)(F)F)=O)CC12 40041,c1(NC(CC2C(CNC(CCSC)=O)C2)=O)cnc2[nH]cnc2c1 40042,Cc1ccc([N+](=O)[O-])c(C)c1C(N1CCC1CNC(c1cnc(C2CC2)s1)=O)=O 40043,N1(C(c2noc(CC)c2C)=O)CC(NC(c2ccc(C#N)[nH]2)=O)CC(O)C1 40044,C12(C(=O)OC)CCOCC1CN(C(=O)Cc1ccccc1OC(F)F)C2 40045,c1(NC(C2CC(O)CN2C(c2ccc(S)cc2)=O)=O)cccc(C(F)(F)F)c1 40046,C1(C(=O)NCC2(C)CCCC2O)C2CCC(C2)C1NC(C1(C)COCCO1)=O 40047,c1(OCCC)ccc(C=CC(N2CCN(CC3CC3)C(C)C2)=O)cc1 40048,Cc1ccccc1N1CCC(NC(=NCc2cc(C(F)F)nn2C)NCCF)CC1 40049,c1(CNC(C2C(OC)CCC2)=O)ccc(CNC(c2c[nH]c(C)c2)=O)cc1 40050,C1(NC(CSc2c(C)cccc2)=O)CN(C(=O)CCCC(C)N(C)C)CC1(C)C 40051,CC(CC(=O)N1CC(F)(C(N2CCCC(NC(N)=O)C2)=O)C1)C(F)(F)F 40052,c1(C(=O)NC2CC(CNC(CC(COC)C)=O)C2)ccc(Br)cc1O 40053,c1(C(=O)NC(C)CCCNC(c2csc(=N)[nH]2)=O)nccn2nccc12 40054,N1(C(c2cc(C)on2)=O)CC(C)(C)OC2(C1)CN(C(C1C3(CC3)C13CC3)=O)C2 40055,CC1=NS(=O)(=O)NC=C1C(=O)N1CC(NC(c2c[nH]cc2C)=O)CCC1C 40056,C1(N(C(CSCC#C)=O)C)CN(C(C2CCCCN2S(C)(=O)=O)=O)CC1(C)C 40057,O=C1CCCCC(C(N2CCC(NC(C3CC(O)C3)=O)C(O)C2)=O)N1 40058,CCCC(CC(C)C)C(=O)N1CC(COC)(NC(=O)CCC(=O)NCCC)C1 40059,C(=O)(CCC(C)(F)F)NC1C(OC)CN(C(=O)CC2CCCCC2)C1 40060,N1(C(C(C2CCCCC2)C)=O)CCCC2(NC(c3nc(=O)n(C)[nH]3)=O)CCCC12 40061,CCCCCC(C)(CC)C(=O)N1CC2CCC(C1)N2c1ccncn1 40062,c1(C(=O)Nc2scc(C(C)NC(C3CC3C(N)=O)=O)n2)ccc(F)c(Cl)c1 40063,N1(C(c2c(CCC)nns2)=O)CC2CC2(CNC(=O)CCSCC(=O)OC)C1 40064,c1(C(=O)NCCCN(C(C(CC)=CC)=O)Cc2ccccc2)cncc(OC)c1 40065,N1(C(CCNC(c2ccncc2)=O)=O)CCCC2CCN(C(C3(O)CC3)=O)CC12 40066,N1(C(C2CC3(CC(C)C3)C2)=O)CC2CCN(C(=O)CC3CCCCN3C)C(C2)C1 40067,c1(C(=O)NCC2(F)CCC(NC(C(CCOC)C)=O)C2)cc(OC)c(O)c(N)c1 40068,N1(C(C2C(C(C)(C)C)CC2)=O)CCC2CN(C(C3C=CCS3)=O)C2C1 40069,S(=O)(=O)(c1ccc(NCC2(CCO)CCOC2)c(Cl)c1)N1C(C)CC2(CCC2)C1 40070,C1(CNC(c2cn(CCC)nn2)=O)C(C)CCCN1C(C1CCC(CO)CC1)=O 40071,CCC(C)CCC(=O)N1CCOCC1CCNC(c1cc[nH]n1)=O 40072,c1(C(=O)NC2CC3(C(=O)NC(CO)CCCO)COC2C3)c[nH]c2ccncc12 40073,C1(NC(c2cc(COC)oc2C)=O)(CO)CCN(C(=O)C(C)CC(F)F)CC1 40074,c1(CCC(=O)N(C2CCCN(C(C3CN(C(=O)N(C)C)C3)=O)C2)C)cccnc1F 40075,N1(C(CC(=O)NCC)=O)C(C(=O)N(C2CCCC2(F)F)C)C2CC(O)C1C2 40076,N1(C(N2CC(OCCOCCOC)C2)=O)CCC(CC(F)F)C1 40077,C(C)(C1CCCc2ccccc21)NC(=NCC)NCCc1ccc(Cl)cc1F 40078,N1(C(=O)CN2CCCC2)CCC2(CC1)CC2C(N1CCC2(C=CCO2)C1)=O 40079,C1(C(=O)NCC(CNC(C2CC3(CCCC3)CO2)=O)O)C2Cc3ccccc3C12 40080,CCCCC(CNC(=O)CCOCC)NC(C1C=C(C)CS1)=O 40081,c1(CC(=O)NC(CN(C(CN(CCOC)C)=O)C)C)ccc(Br)c(F)c1 40082,c1(C(C(N2CCCC(N(C(CC(=C)C)=O)CCO)C2)=O)C)c[nH]c2ccccc12 40083,C(CC(C)C)(C(=O)N1CCCC(CNC(c2c(C)noc2C)=O)C1)OC 40084,n1(C(C)C)cccc(C(=O)NCC2CC2CNC(=O)C(O)CN2CCCC2)c1=O 40085,C=C(C)C(O)CC(=O)NCCC1CN(C(c2cnn(CC3CCOC3)c2)=O)C1 40086,C12(CC(=O)NCc3cccc(C)n3)CCC1CN(C(C1CCCCNC1=O)=O)C2 40087,CC(C)C(O)C(C)(C)C(=O)N1CC(C(=O)NCCC(C)C(F)(F)F)C(F)C1 40088,C(C(C)C)(C(O)C(=O)N1CCCCCC1C(=O)N(C(C)CC1CC1)C)OC 40089,C(=O)(C#CC1CCCOC1)NCCCNC(c1cc(C(=O)OCC)no1)=O 40090,C1(C(=O)NC2C(NC(=O)Cn3cnnn3)CCCC2)CC2C=CC1CC2 40091,C1(NC(c2ccc(C)nc2)=O)CN(C(c2ccc(SC(F)(F)F)s2)=O)CCC1C 40092,C=CCC(C)(C(F)F)NC(=O)CN(C(=O)CC(C)COC)CCOC 40093,Cc1nc(C)c(CC(=O)NCCCC2(NC(=O)CN(C)CCO)CC2)c(O)n1 40094,CCCC(C(=O)NCCCCCN1CCN(C(C2COC(=O)C2)=O)CC1)N(C)C 40095,C1(CNC(c2cc(C)on2)=O)(CO)CCN(C(=O)CC2CCCC2C)CC1 40096,C1(C(=O)NCC(C)(C)NC(c2ncoc2Br)=O)CCOCC1(C)C 40097,C(=O)(C(F)CC(C)(C)C)N1C(C(=O)NC(c2c(C)nccn2)C)COCC1 40098,c1(C(=O)NCCCN(C(C(C)C2CCCC2)=O)C)cc(F)cc(S(N)(=O)=O)c1 40099,C(CCC(C)CC(=O)N1CC(O)(CCNC(C2CCCOC2)=O)C1)=C(C)C 40100,N1(C(c2cc(C)[nH]c2)=O)C2CCC(C(=O)NCc3cncs3)C1CC2 40101,C1(CCNC(c2cc(C(=O)OC)sn2)=O)CCCN(C(=O)C(C)C2CCC2)C1 40102,c1(C(N(CC(C)NC(c2c(OC)cccn2)=O)C)=O)cc(Br)cnc1C 40103,N1(C(c2c(C(C)C)occ2)=O)CCCCC12CN(C(C1SC3C=CC1C3)=O)C2 40104,C1CCC(=O)N1.c1(CC(CN(C(C)C)C=O)O)ccccc1 40105,C1(c2n(CCC)nnn2)(OC)CCN(CC)C(C)(C)C1.C12CC(C13CCC3)NC2 40106,C1(CNC(c2c(OC)n[nH]c2)=O)CN(C(=O)Cc2c(C)cccc2Cl)C(C)(C)C1 40107,CS(=O)(=O)c1cc(C(N2CCC3CN(S(=O)(=O)CC4CC4)CCC23)=O)ccc1F 40108,C1(NC(C(c2n(C)ncc2)O)=O)(COC)CCN(C(=O)CSc2nncn2C)C1 40109,Cc1cc(Cl)c(C(N2CC(C)(C)C2Cn2cc(C3CCCCO3)nn2)=O)s1 40110,C1(N(CC(N2CCCCC2)=O)C(=O)NC2CC(CC)C2)CCS(=O)(=O)C1 40111,C(=O)(C1=NOC(C)C1)NCCN(C(C1C(C=C)OCC1)=O)C 40112,C1(NC(CC(=O)OC)=O)CC(O)CN(C(=O)Cc2ccc(OC(F)(F)F)cc2)C1 40113,C(CCCCC(=O)N1CC2CC1(CNC(=O)Cc1cc(C)cs1)C2)OCC 40114,c1(C(=O)NC2CCCN(C(C3C4COCC34)=O)C2)cc2oc(Br)cc2s1 40115,c1(CC(=O)NC2(COC)CN(C(c3cc(C#N)cs3)=O)C2)cnccc1Cl 40116,C(=O)(C(CCN(C)C)N(C)C)N1CC(C)(CCC(=O)N(CCOCC=C)C)C1 40117,C1(CC)CCCN(C(=O)CC2CC(F)C2)C1C(=O)NCC(C)(C)n1ccnc1 40118,c1(C(NNC(=O)OC2CC(OCC)C2(SC2CC2)CC)=O)csc2ccccc12 40119,O=S(=O)(c1cccnc1NCCC1CCC2CC12)NCc1cc(C(F)F)on1 40120,c1(C(=O)NC2C(C)N(C(=O)CCc3cnoc3)CC2)nccc2[nH]ccc12 40121,Cc1c(C(N2CCN(C(=O)C(C)(C)CO)CC2CS(C)(=O)=O)=O)cccc1C#N 40122,C(C(CC(C)C)C(=O)NC1CC(CCNC(=O)C(C2CCCC2)OC)C1)OC 40123,C(C(C)(F)F)N(C(C=CC(C)NC(C1(C(N)=O)CC1)=O)=O)C 40124,N1(C(C2CCSCC2)=O)CC2CCC(C(N3CCC(N4CCCC4)C3)=O)(C2)C1 40125,c1(C(C(=O)NCCOCC)N(C2(CCO)CC2)C)ccc(C2CCC2)cc1 40126,N1(CC(N2CCCN(C(CCC#CC)=O)C(C)C2)=O)CCSC2CCCCC12 40127,C1(NC(c2c(C)nn(C3CCOC3)c2)=O)C2CCCC1CC2 40128,N1(C(c2cccc(CC)c2)=O)CCC2(CC1)CC2NC(C1(C)CCSCC1)=O 40129,N1(C(COc2ccn(C)n2)=O)CCC2CN(C(c3cc(N)cc(O)n3)=O)CC12 40130,CC1OC2(CO)CC1(C(N1CC3(C1)CN(C(=O)C(O)(C1CC1)C1CC1)C3)=O)C2 40131,C1(C(F)F)(CNC(CC(=O)NCC)=O)CCN(C(c2cnn(C)c2OC)=O)C1 40132,c1(CC)nc[nH]c1C(N1CCCC1CN(C(=O)CC1CCSCC1)C)=O 40133,C1(C)(C(=O)NCCC(C)N(C(=O)CCCCN2CCOCC2)C)CCC12CCC2 40134,c1(C(=O)NCCOCCN(C(CC2CCCC(OC)C2)=O)C)cc(Cl)ccc1N 40135,C1(C(N2CC(OCC(=O)NCc3ccc[nH]3)C2)=O)Cc2nccn2C1 40136,N1(C(CC2OCC(C)(C)C2)=O)CC2CC(C1)N(C(c1ccc(F)cc1)=O)C2 40137,C1(NC(Cc2cnc(C)s2)=O)CC(N=c2[nH]c3cccc(F)c3s2)C1 40138,C1(N(C(C(C)OCC(F)(F)F)=O)C)CN(C(=O)CCc2nccs2)CC1(C)C 40139,c1(C2C(C(=O)NCCN(C(=O)Cc3cnn(C(F)F)c3)CC)C2)ccccc1Cl 40140,C1(NC(C(C)CNC(c2ccccc2)=O)=O)CN2CCC1(F)CC2 40141,c1(C(N2C(CNC(C3C(C=C)CC3)=O)CC(C)(C)C2)=O)ccc(Cl)c(N)c1Cl 40142,N1(C(c2c(C)nsc2C)=O)CC(NC(=O)CC(O)CN(C)C)CC2(CC2)C1 40143,C(C)(CCN=c1cc(C2CCCCC2)nc[nH]1)NC(c1ccn(CC(C)C)n1)=O 40144,c1(-n2cc(C3(F)CN(C(C4(CSC)CC4)=O)C3)nn2)ccc(C)cc1C 40145,C1(C(=O)NC(COCC)C)CN(C(C2(CC)CCCC2O)=O)CC1(F)F 40146,c1(C(N(C(CNC(CC(C)OC)=O)C2CC2)C)=O)cnc2ncnn2c1C(C)C 40147,C1(CNC(CCC=CCC=C)=O)CC(NC(c2coc(Br)n2)=O)C12CCC2 40148,C1(CC#C)(C(=O)NCC(C)(CNC(=O)C=CCN(C)C)OC)CCOC1 40149,c1(C(=O)NCC(C)(C)OCCNC(C(CC=C)C)=O)c(C)cc(C)nc1O 40150,CCC(C(=O)NCCc1cnc(C)s1)N(C(=O)CNC(=O)CNC(C)=O)C 40151,N1(C(C(C(C)(C)C)NC(=O)C(F)OC(F)(F)F)=O)CC2C3CCC(O3)C2C1 40152,C(C(C(=O)N1CCN(C(C)C)C(=O)C1)C(C)(C)C)NC(CCC=C)=O 40153,CN(CP(C)(C)=O)Cc1cnn(C2CC2)c1 40154,c1(C(N)=O)cc(C(=O)NCC2OCCC2C(=O)NCC2(F)CC(O)C2)n[nH]1 40155,Cc1cc(C(=O)NC2CC(O)(c3cccnc3)C2)c2c(c1)CCC2 40156,c1(C(=O)NCCNC(Cc2c(C)scc2)=O)cccnc1SC(F)F 40157,C=C(C)CC(C(=O)NCCC1CC(F)(F)CN1C(C1CCCOC1C)=O)OC 40158,N1(C(c2n(CC)nnc2)=O)CCC(NC(=O)C(C)(C2CC2)OC)C1C 40159,c12nnnn1n1cc2nn1.C1(C)(CC)CN1.C(=O)(CC(C)SCCCC)OC 40160,Cn1cncc1C(c1nnnn1Cc1cccs1)NCCC(=O)NO 40161,c1(C(N2C(CNC(C3C(C#N)C3)=O)CCCCC2)=O)noc2cc(F)ccc12 40162,O=C(N=c1[nH]c(Cl)ncc1O)C1CN(S(=O)(=O)C2CC2)CCC1O 40163,C1(N=[N+]=[N-])(C(=O)NC(C(C(=O)OC)C)C)CCN(C(C2CCCC2C(C)C)=O)C1 40164,N1(C(CC(C)N2CCCC2=O)=O)CCC(CO)(CNC(C2(Cl)CCC2)=O)C1 40165,c1(C(=O)NCC2CCN2OC)cccn2nncc12.c12csc(c1)C(=O)NC2 40166,C#CC1CCN(C(=O)C(CCC=C)NC(C2CCS2(=O)=O)=O)CC1 40167,c1(C(=O)NCC2CN(C(CC(C)(C)C)=O)CC2O)c(N)c(F)cc(F)c1F 40168,CCC(Cc1ccccc1Br)C(=O)NCC(c1cnn(CC)c1)N1CCCC1 40169,S(=O)(=O)(c1cc(C(=O)O)c(Cl)cc1Cl)N(C1CC(C(N)=O)C1)C 40170,Cc1cc(-n2cccn2)ccc1NC(C)C(C)S(C)(=O)=O 40171,C=C(C)C(C)(C)C(=O)NCC1(CNC(c2ccnc(C3CC3)n2)=O)CCOCC1 40172,c1(C(N2CCC(O)(C(C)NC(=O)C(O)C3CCCC3)C2)=O)ncc2ccccn12 40173,C(=O)(NN1CCCC1C(N1CC(O)(C(F)(F)F)C1)=O)C1(CC(C)=O)CC1 40174,N1(C(C)=O)CCC(NC(=O)CC2(OC)CN(C(C3SCC=C3C)=O)C2)C1 40175,c1(C(=O)NCCC2CN(C(C=C(COC)C)=O)C2)cc(C)c(C)c2ncccc12 40176,N1(CCC(=O)NC)CCCOC(CNc2ccc(-c3cc(CO)on3)cc2)C1 40177,N1(C(C2CC(SC)C2)=O)CCC(C(C)NC(=O)Cc2cnnn2C)C1 40178,S(=O)(=O)(c1cnc(NCCc2cccc(Cl)c2C)c(Cl)c1)NC(COC)C1CC1 40179,n1(CC)nc(C)c(C(=O)N(C)CC2CCN(C(=O)CC(C)OC)C2)c1Cl 40180,C12(Cl)CC13CCN(CC3)C2.c1(C2(OC)CCC2)cnn(Cc2ccccc2)c1 40181,CCC(O)C(C)C(=O)NC1CN(C(=O)Cc2ccc(-n3cnnc3)cc2)C1 40182,C(=O)(C(O)CCCNC(=O)CCC(=O)NC)NCC(CC)(C)CO 40183,C(C(CNC(=O)CCc1cnoc1)NC(=O)CC1CC(C(C)(C)C)C1)OC 40184,CC1(C)C(NC(c2cc(C3CC3)no2)=O)CCN1C(=O)Cc1cnoc1 40185,C=CC(C)C(C)C(=O)N(CC(CO)(CO)NC(c1cc(C(F)F)no1)=O)C 40186,N1(C(C2CC(=C)C2)=O)CC2CCC1C1CN(C(c3ccsc3S(N)(=O)=O)=O)CC21 40187,C(=O)(CCN(OC)C(=O)C(C)(O)C(F)(F)F)NCC(C#C)CC 40188,C1(S(C)(=O)=O)(C(N2CCCC(NC(C=CCOC)=O)(CO)C2)=O)CC(O)C1 40189,C1(NC(C2Cc3n(cc(C)n3)C2)=O)CC2CCC(C1F)N2C(C1(C)CC1(C)C)=O 40190,N1(C(CCN(C(c2ncn(C)n2)=O)C2CC2)=O)CCOCC(CO)C1 40191,C(=O)(C(O)CC(N)=O)N1C(C(N(CC)Cc2ccoc2)=O)CC=CC1 40192,c1(CC(N2CC3C(CNC(=O)NCC)(C3)C2)=O)cccc(OC)c1O 40193,N1(C(C=NOC)=O)Cc2ccccc2CC1CNC(C1CCC2CC2CC1)=O 40194,N1(C(CCOc2ccc(C)cc2)=O)CCN(C(C2CCCCN2C)=O)CC1C 40195,c1(C(=O)NCC2CCCC(C)C2)cccc(S(C)=O)c1 40196,c1(CN2CC3C(C(=O)Nc4c(OC)nccn4)(C3)C2)ccc2c(c1)OCCO2 40197,c1(C(N2CCCC(CCNC(C(F)OC)=O)C2)=O)cc2cccc(Cl)c2o1 40198,CC1CN(C(C)C(=O)N(CC(=O)NC(C(N)=O)C2CCCC2)C2CC2)C1 40199,C1(NC(c2csc(-c3ccco3)n2)=O)CC(O)CN(C(C2CC(O)C2)=O)C1 40200,C(=O)(CCC(=O)NN(C)C)NC(CNC(C(C)(C)NC(=O)NCC)=O)(C)C 40201,c1(CC(=O)NC2CCC(NC(C3C(C(N)=O)C3)=O)CC2)cc(Br)ccc1Cl 40202,c1(SC)cc(C(N2CCC(C3CCCN3C(c3ccc(O)nn3)=O)C2)=O)c(C)o1 40203,C1(CC)CN(C(=O)C=C(C)c2cccs2)CC1NC(C1(C(C)(F)F)CC1)=O 40204,c1(OC)cc(N)c(Cl)cc1C(=O)NCC1(NC(C2CC23CC(O)C3)=O)CCOC1 40205,CC1(O)CCN(C(=O)C(c2cn(C)nn2)NC(C2(F)CCCCC2)=O)CC1 40206,N1(C(c2c(C)c(F)ccc2)=O)CCC2CCCN(C(c3cnco3)=O)C2C1 40207,C1(C(=O)NC(C)CN=[N+]=[N-])CN(C(C2CC(=C3CCC3)C2)=O)CCC1(C)C 40208,c1(C(c2n(CC)nnn2)NCC2(n3cccn3)CC2)cc(Cl)cc(C)c1OC 40209,c1(CN(C(Cc2cc(C)no2)=O)C)cccc(CNC(C2CCCC(O)C2)=O)c1 40210,C1(C(N(CCN(CC)CC)C)=O)CC12CCN(C(c1cncc(NC)c1)=O)C2 40211,N1(C(c2c(C(N)=O)cccc2)=O)CCC(F)C(NC(C2CCC(F)CC2)=O)C1 40212,c1(NC(C2CC23CN(C(c2ccc(Cl)c(I)c2)=O)C3)=O)cc([N+](=O)[O-])ccc1I 40213,CC1OCCC1(F)C(=O)NC1CC(C(=O)N(C)CCC2CCCCC2)C1 40214,C12(CNC(C(C)=C(C)C)=O)CCC(C1)N(C(=O)CN(CC(C)(C)C)C)C2 40215,c1(C(=O)NC2C(CNC(c3ccc(C4CC4)o3)=O)C2)cc2c(s1)CCCC2 40216,C(=O)(C(CCC(N)=O)n1cc(C2C3COCC23)nn1)NC(CCC)C 40217,n1(C(=O)N)nccc1C(F)(F)F.C(=O)(C(C)(C)CC)N(C)CCOCCOCCOC 40218,C1(C2CCCN(C(=O)Cc3ccc4n[nH]cc4c3)C2)(NC(C=CSC)=O)CC1 40219,C1(NC(CNC(=O)CN2CCOCC(O)C2)=O)CC2(CCC2)CO1 40220,C1(NC(C(C(C)C)C)=O)CC2(COC(C)C2)C1 40221,N1(C(c2c(CC)occ2C)=O)CCN(C(C2(C)CCOCC2)=O)C2(CC2)C1 40222,c1(CC(=O)NC(CCNC(CCCOCC)=O)C)cccc(Br)c1 40223,c1(C(=O)NC2CCC(N(C(=O)OC)C)CC2)ccc(C(C)=O)nc1O 40224,C(=O)(C(O)CC[S+](C)C)NCC1(F)CCN(C(C2(COC)CC2)=O)C1 40225,c1(OC)nccc(C(=O)NC2CCN(C(=O)C(C)(C)Br)CC2F)c1Cl 40226,[N-]=[N+]=NCCC(=O)NCCC(O)C(=O)N1CCOC(C2CCC2)C1 40227,C(=O)(C(F)C(CC)CC)N1C(C(=O)NC(CN(CCCC)C)C)CC(OC)C1 40228,N1(C(=O)CCCc2cncs2)CC2(CCCCN2C(=O)CCN2CCOCC2)C1 40229,Cc1ncc([N+](=O)[O-])cc1-c1ccc(NC(c2ccnc(F)c2)=O)c(F)c1 40230,C(CN=c1ccnc(NC2CC(C(C)(C)C)C2)[nH]1)N1CCCC(C)C1 40231,c1(C(=O)NC(CCNC(Cc2ccn(CC)n2)=O)C)cc(C)cc(O)c1 40232,c1(C(=O)NC2CC(C)(C)CN(C(=O)C#CC3CC3)C2)c[nH]c2ccncc2c1=O 40233,C1(NC(CCNC(CC(C)C)=O)=O)CN(C(=O)C(C)(C)C(F)F)CCC1O 40234,CC(C)C(C)CC(=O)NCC(C(=O)N1CCCC1C(C)(C)C)N(C)C 40235,c1(-n2cc(CCN(C(c3c(C)cccc3)=O)C)nn2)c[nH]c2cc(C#N)ccc12 40236,N1(C(C(C)(C)C#N)=O)CC=C(CCNC(C2(CO)CC2(F)F)=O)CC1 40237,c1(C(N2C3CC(NC(COCC(=C)C)=O)C2CC3)=O)ccc([N+](=O)[O-])cn1 40238,C1(C(N(C(CCNC(c2c(C)ncnc2)=O)C)C)=O)COc2ccc(F)cc2C1 40239,c1(NC2CC(C)N(C(=O)CCCc3ccsc3)C2)ncc([N+](=O)[O-])cc1Cl 40240,O=C1CN(CC(=O)Nc2ccc(Cl)nn2)C(=O)N1.C12C3CN(CC13)CC(=O)N2 40241,c1(C(=O)NCC2C=CC(NC(C(CC)SC)=O)C2)c(Cl)ccc2c1OCO2 40242,c1(C(N2C(CC(=O)NCC3CC(C)(F)C3)CCCC2)=O)cccn2cncc12 40243,C12(C(=O)NCc3ccnc(C)n3)CCC1CN(C(C1CCCC1F)=O)C2 40244,C(=O)(CC(C(C)OC)NC(=O)C(F)C(C)C)N(CCC#C)C1CC1 40245,C(C(=O)NCC=CCSC)(C1(C)CC1)NC(C=CC)=O 40246,c1(C(N(C(C)CCNC(=O)CC2CCC(F)(F)C2)C)=O)cccc2c1CCC2=O 40247,C(C(CO)C(F)(F)F)NC(C(C)CNC(C1CC1(F)Cl)=O)=O 40248,C#Cc1c[nH]nc1C(N1C(C(N2CC(C(CC)CC)C2)=O)CC1C)=O 40249,C1(NC(C2(COC)CCCC2)=O)COCCN(C(=O)Cn2cc(Cl)cn2)C1 40250,C(=O)(C1=CCCCO1)NC(CCOC)C(=O)NCC1CC(=O)NC(C)C1 40251,C1(NC(c2cnc(CC)s2)=O)(CF)CCN(C(=O)C(c2cscn2)N(C)C)C1 40252,c1(C(=O)NC2CC(NC(C=NOC)=O)C2)cnc(O)c2c1NCCC2 40253,c1(OC)ccc(Cl)cc1CC(=O)NCC(C)(C1CC1)NC(=O)CCc1ccsc1 40254,N1(C(c2nc(CNC(C(C)C3CCCC3)=O)oc2)=O)CC(C2CCCCC2)C1 40255,C12(CNC(c3ccn(C(CC)CC)n3)=O)CCC(CC1)N(C(=O)CCC(N)=O)C2 40256,C12(NC(C(=O)NC(c3ccc(F)cc3Cl)(C)C)=O)CCC(CO)(C1)OC2 40257,C(CCC)(C(=O)NCCC1(NC(=O)COc2ccsc2)CCCC1)=CCC 40258,C1(C(=O)NC2CC(NC(CC(C=C)(C)C)=O)C2)COc2ccc(OC)cc2C1 40259,Cc1nc(=N)[nH]cc1C(N1CCN(C(=O)Cn2ccnn2)CC1C1CC1)=O 40260,C1(C(=O)NCCC(C)NC(=O)C(c2ccc(F)cc2)(F)F)CCCCN1C 40261,C1(C(=O)NC(CC)C(=O)NC)CNC(=O)CN1C(=O)C1=COCCC1 40262,C#Cc1cc(=NCC(c2ccncc2)OC)cc[nH]1 40263,Cc1nn(C)cc1C(=O)NCCOC1CCN(C(c2ccccc2Cl)=O)C1 40264,c1(C(=O)Nc2ccnc(N3CCOC(C(F)(F)F)C3)c2)cc2c(cc1O)CCCC2 40265,CC(C)CC(O)C(=O)NC(C)CNC(c1cc(C(F)(F)F)cc(N)c1)=O 40266,C(=O)(C1CCCn2ccnc21)NCC(C)(C)NC(C1N(CCCC)CCOC1)=O 40267,N1(C(C=CCNC(C2CC(C)(O)C2)=O)=O)CCc2ncccc2C1 40268,C1(C(=O)NC(CCOCC)C)(C(=O)NC)C=CCN1C(=O)CNC=O 40269,C(C(CNC(C1(Cl)CC1)=O)S(C)(=O)=O)NC(C(C(C)C)n1cnnn1)=O 40270,c1(NC(CNC(=O)Nc2nn(CCOC)c(C)c2)=O)ccc2ncsc2c1Br 40271,N#Cc1cncnc1N1CCCC(NC(=O)Cc2ccccc2O)C1 40272,N1(C(c2nc(CC)sc2)=O)CC(NC(=O)C(c2ccccc2OC)(C)C)CC1C 40273,C12(CC)CC1CN(C(C1CCC=CC1NC(=O)C(C1CCOCC1)F)=O)C2 40274,c1(C(=O)NC(C2CN(C(C(=O)NCC)=O)C2)C)ccc2nnc(O)n2c1 40275,c1(C(=O)NC(CCOCC)C(=O)N2CC(c3nn[nH]n3)C2)cccc(=O)n1C 40276,c1(CC(N2CC(C)N(C(C3CCN3C(C)(C)C)=O)CC2)=O)cccc([N+](=O)[O-])c1 40277,Cc1ccc(C(C)C)cc1C(=O)NC1CCN(C(=O)C(O)P(C)(C)=O)CC1O 40278,O=C(C(O)Cn1cncn1)NC1CN(C(C2CC2(Cl)Cl)=O)C1 40279,Cc1nc(CC2CC2)sc1C(=O)NC1CN(C(c2ccccc2C(C)C)=O)C1 40280,c1(C(=O)NCc2ccccc2)ncccc1C(=O)C1CC1.C12(CCCC1)NC(=O)N2 40281,C1(C(=O)NCC2C(CNC(CC=CC)=O)C2)CCc2ncsc2C1 40282,c1(C(=O)NC(C(=O)NCC(c2ccc(Cl)cc2)(F)F)=O)cnc2[nH]ccc2n1 40283,Cn1nc(C2CC2)nc1CNC(=O)C(=O)NC1CN(C2CCCCC2)C1 40284,N1(C(Cc2ncc(C)s2)=O)CCC(NCc2cc(=O)n(C)o2)CC1C 40285,C1(NC(c2c(C)nc(Cc3ccccc3)o2)=O)CC12CCOc1ccccc12 40286,c1(CNC2CCC(C(=O)Nc3cc(OCC)c(O)cc3)C2)ccc2n[nH]cc2c1 40287,c1(C(=O)NCCCN(C(CC(C)n2ccnc2)=O)C)cccc(P(C)(C)=O)c1 40288,c1(CNC(=O)OC(C)(C)C)ccc(S(=O)(=O)NCCC2(O)CCCC2)cc1 40289,Cc1ccsc1-c1cn(C(C)C(=O)N(C2CC2)C2CC2)nn1 40290,CCCC(CC(C)C)C(=O)NCC1(F)CC(CNC(c2cc(N)ccn2)=O)C1 40291,NS(=O)(=O)C1CN(C(=O)Cn2nnc(-c3ccc(Cl)cc3)n2)C2(CCC2)C1 40292,c1(CC(=O)NCc2c(CCNC(C(C)(C)C3CC3)=O)ocn2)ccc2c(c1)CC2 40293,c1(C(N2CC3C(CNC(C(CCC)N(C)C)=O)C3C2)=O)cn(C)c(C)cc1=O 40294,CC1(C)C(C(=O)NC(CCO)C2CC2)CCN1C(=O)CCCn1cccn1 40295,Cc1nc(C2CC2)ncc1C(=O)N(CCCNC(c1ccco1)=O)C(C)C 40296,CC(CNC(C1COCCC1C)=O)C(F)C(=O)NC1(CC2CCC2)CC1 40297,n1(CC=C)c(SCC2NCCC2C)nc2sc3c(c2c1=O)CCC3 40298,C=CCC(F)(F)C(=O)NCC1(C)CCC(NC(=O)CCSCC)C1 40299,N1(C(C=C(C)Cl)=O)CCCN(C(=O)CCOC2CCC2)C(c2ccccc2)C1 40300,CC(C)C(O)C(F)(F)C(=O)NCC1C(C)CCCN1C(=O)CCc1cnc[nH]1 40301,c1(C(=O)NC(CNC(C2C(=C)CC2)=O)CCOC)c(C)cc(C)oc1=O 40302,C1(C(N2C(CNC(C3(CCCC)CC3)=O)C=CC2)=O)CC2(C1)CC(C)(C)C2 40303,C12CCN(CC1)C2.c1(CN(C(CNC(CC)=O)=O)C)cc(C)c(C)s1 40304,CCCCCC(C)CC(=O)NCCC(O)CNC(c1ncoc1C1CC1)=O 40305,CC(C)CC(C(=O)N(C)CC1(CO)CC1)NC(C1CCC(=O)N(C)C1)=O 40306,C(CCSC)(C(=O)NCc1cn(CCNC(=O)CCc2ccccn2)nn1)OC 40307,C1(C(N(CCC)CC)=O)CCC(O)CN1C(=O)CC(Cl)Cl 40308,C1(C(=O)NC)CC2OCCC2N(C(C2CCc3ccoc3C2)=O)C1 40309,c1(C(=O)NC2C(NC(=O)C=Cc3cocn3)C2)cc2c(s1)CCCC2 40310,Cc1nn(CO)cc1C(N1CC(CNC(=O)CCC(=O)C2CCCO2)C(O)C1)=O 40311,CCCC(CCC)C(=O)Nc1cccc(C(N2CCCC2C(N)=O)=O)c1 40312,Cc1nc(N2CCOC(C(=O)Nc3nc4c(s3)CCC4)C2)c2c(n1)CCC2 40313,Cc1cc2sc(C(=O)N(CCC(C(C)(C)C)NC(c3ccccc3)=O)C)cc2s1 40314,C(=O)(C(C)(C)C(C)(F)F)NC(C1CC(NC(C2CC2C2(O)CCC2)=O)C1)C 40315,c12ncccc1C(=O)NC2.CC1CC(CCC(=O)N2CC(CF)C2)C1 40316,N1(C(C(CCCNC(C2(OC)CCCOC2)=O)O)=O)CC2(CNC(=O)OC2)C1 40317,C1(CNC(C(CC)COC)=O)(OC)CCCN(C(C2(c3cc[nH]n3)CC2)=O)C1 40318,c1(C(=O)NCCC2CC(NC(C3CC3Cl)=O)C2)cc2c[nH]cnc-2n1 40319,Cc1ccc(F)c(C(N2CCCC(C)(CNC(c3c[nH]c(C#N)c3)=O)C2)=O)c1F 40320,O=C1CCC2(C(=O)NCC3COCCN(C(c4ccoc4Cl)=O)C3)CCCC2C1 40321,C1(C(=O)NCCCC(C)C)CN(C(=O)C(C)C(C)C)CC1(C)C 40322,N1(C(c2cc(C)n(C(C)(C)C)n2)=O)CC(NC(=O)CN2CCC(C)C2)CC(F)C1 40323,c1(C(N(C2CCCN(C(c3csnc3Cl)=O)C2)CCO)=O)ccc2[nH]ccc2c1 40324,c1(C(C(=O)O)N(C)C(c2nnn(C3CC3)c2C(F)(F)F)=O)c(F)cccc1F 40325,n1(CC)ncc(C(N2CCN(C(=O)CNC(=O)C(C)OC)CC2)=O)c1C(F)(F)F 40326,N1(C(CCNC(=O)NC)=O)CCCC(O)(CNC(c2cc(CO)ccc2Cl)=O)C1 40327,N1(C(C(C)=CC2CC2)=O)CCC2CC2(C(=O)Nc2cccc(CO)c2)CC1 40328,CC(CCNC(=O)C=Cc1ccco1)CCNC(C1COCCN1C)=O 40329,c1(C(N2CC(C(C)NC(c3c(C)scc3)=O)C2)=O)cnc2ccccn12 40330,C1(OC2(CC(=O)N(CC(=O)OC(C)(C)C)C)CCC2)CCCCCC1 40331,c1(C(N2C3C(CNC(CC=CC=C)=O)C(CCC3)C2)=O)nc2n(c1Cl)CCCC2 40332,N1(C(C(CC)(C)OC)=O)CCc2nc(CNC(=O)CCCn3cncn3)sc2C1 40333,C=C(C)CCCC(=O)NCC(CCOC)NC(c1nc(OC)cc(OC)n1)=O 40334,c1(C(C)C)ccc(C2CCCN(C(=O)C(C)n3cnnn3)C2)cc1 40335,C12(CC(=O)Nc3ccc(CO)cc3)CCC1CN(C(c1ccncc1O)=O)C2 40336,C(=O)(C(C#N)CC)N(CCC)CCNC(=O)CCN1CCOCC1 40337,C1(CC=C)(NC(c2ncc(OC)nc2OC)=O)CC2CCC(C1)N2C(=O)COC 40338,c1(-c2c(CCC(C)OC)cccc2)cc(F)ccc1F 40339,CC(C)(C)CC(C)(C)C(=O)N1CCC(C)(CC(=O)NCCCOCC(F)F)C1 40340,C1(O)(C(=O)N)CC(C)(C)C1.C1(NC(CN(C)C(N)=O)=O)COCCC1Nc1cn[nH]c1 40341,N1(C(CC2CN(C)C2)=O)CC(NC(=O)CCNC(c2ccoc2)=O)CC(F)C1 40342,c1(C(C(N)=O)NC(=O)NC(c2cc(C)n(C)n2)CO)ccc2ccccc2c1 40343,c1(N(CCC)C)ccc(C(=O)NC23CC2CN(C(=O)C(C)n2cccc2)C3)cc1 40344,CCC(C)C(O)CC(=O)NCC(C)(C)OCCNC(c1cnc2ccccn12)=O 40345,C1(NC(=O)COC2CC=CC2)CN(C(=O)C(F)=C2CCCC2)CC(F)(F)C1 40346,c1(C2CCN(C(c3c(COC)noc3)C(=O)NCC(C)C)C2)ccc(Cl)c(Cl)c1 40347,N1(C(CCN(CCC)C)=O)CCC(C(=O)N(C)Cc2scnc2C)C1 40348,c1(C(=O)NC(CNC(CC=C(C)C)=O)C2CC2)csc(C2CC2)n1 40349,Cn1ccc2cccc(C(N3CCC(C)(NC(C4CCCS4(=O)=O)=O)C3)=O)c12 40350,N1(C(C2C(C)=C2)=O)CC2CCC(C1)N2C1CCN(C(=O)C(C)(C)C(F)F)CC1 40351,c1(C(C(=O)NC2CCCC2)N(CCC)CC)cnc2n1CCC2 40352,N1(C(CCSC)=O)CC2=C(C1)CN(C(c1cnc(C(F)F)c(C)c1)=O)C2 40353,c1(C(N(C2CN(C(C(CC)(F)F)=O)CC2O)C)=O)cc(F)c(C(C)C)cc1F 40354,c1(CNCC2N(C(CN(C(C)C)C)=O)CCOC2)ccc2nccn2c1 40355,c1(C(=O)NCC(C)N(C(=O)Cc2cc(Cl)ccc2O)C)cccc2c[nH]nc12 40356,C(=O)(C1=CCC(C)(C)CC1)NCC1(F)CCCN(C(CSCC=C)=O)C1 40357,c1(NC(C2(C(C)NC(=O)C(C)CF)CC2)=O)cc(C(F)(F)F)c(C)c([N+](=O)[O-])c1 40358,C(CC(C)C(=O)NCCOCCNC(=O)C(C)(C)Cc1cccc(Cl)c1)=CC 40359,CC(C)C(C)C(=O)N(C)CC1(O)CCN(C(c2ccc(CC#N)cc2)=O)C1 40360,C(=O)(CN1C(=O)CCc2ccccc21)NCC1C(NC(CC2CN(C)C2)=O)CC1 40361,c1(NC(C=CCN2CCC(NC(CC(CC)C)=O)CC2)=O)ccc(Br)cc1F 40362,CC1(C)COCCC1C(=O)NC1C2CCN(C(c3ccc(F)cn3)=O)C12 40363,C1(CNC(=O)NCCN(CCC)C)CCC1C(=O)OCC 40364,N1(C(Cc2c(C)cnn2C)=O)CCN(C(=O)COc2ccsn2)CC(O)C1 40365,C(=O)(C(C)C(O)CCCC)NCCC1(O)CN(C(CC(=C)C)=O)C1 40366,c1(C(=O)NCC2(C(C)(C)O)CN(C(C3C(C)CC3C)=O)C2)ccnc2ncnn12 40367,N1(C(C(C)(C)F)=O)CCC2(CCN(C(c3coc(-c4ccc(F)cc4)n3)=O)C2)C1 40368,N1(C(C2N(C(CC(C)(C)C(F)F)=O)CCCCC2)=O)CCC2(CCCCO2)C1 40369,c1(C(=O)NC2CC(CS(N)(=O)=O)C2)cccc(C(=O)O)c1 40370,Cc1ncc(C(=O)NCC2(C(=O)NC(C)(CO)C(F)(F)F)CC2)c(C)n1 40371,C1(NC(c2c(C(C)C)onc2)=O)CC(C)N(C(c2cn(C)cn2)=O)C1 40372,N1(C(COCCOC)=O)CCN(C)C(CNC(C2CN(C)CCO2)=O)C1 40373,C1(NC(C2(C)CCC2)=O)CCC2(CC1)CCN(C(=O)CC1CCCC1(F)F)CC2 40374,C1(NC(=O)C(CC(F)F)N2CCOCC2)CCN(C(=O)C(Cl)=CCl)CCC1(F)F 40375,Cc1csc2ncnc(NC(C)CC(C)NC(c3ccc4nccnc4c3)=O)c12 40376,c1(CN2CCN(C(c3ncc(-c4ccccc4)s3)C)CC2C)ccc2c(c1)C(=O)NC2 40377,c1(CC)nc(N2CCCC(NC(c3sc(C(C)C)nc3C)=O)C2)c(CC)c(Cl)n1 40378,O=C1Cc2cc(C(=O)NC3CN(C(C4CS(=O)(=O)C4)=O)CC3O)ccc2N1 40379,c1(N2CCCC(NC(=O)C=Cc3ccc(Br)s3)CC2)cc2ncnn2cn1 40380,c1(C(=O)NCCCN(C(C2C(C=C)C2)=O)CCO)ccc2c(c1)OCC2 40381,Cc1no[nH]c1=NC(=O)C1(C)CCN(c2ncncc2I)C1 40382,c1(C(N2CC(C(=O)OC)CC(CC)C2)=O)ccc2c(Br)cnn2c1 40383,N1(C(C(C=C)OC)=O)CC(CC(=O)NCC(C)(O)CCC)C2(CC2)C1 40384,CN1CCN(C(C2CC3CC3N2Cc2cccnc2C(F)(F)F)=O)CC1=O 40385,C1(C(N(CCN(C(c2ccc(C(C)C)cc2)=O)C)C)=O)CCC(N=[N+]=[N-])CC1 40386,c1(NC(CC)=O)ccc(F)c(NC(=O)CCC(=O)c2cccc(OC)c2)c1 40387,c1(C2CN(C(C=C(C)C(C)C)=O)C2)ccc(F)c(F)c1 40388,CCCCC(COC)NC(=O)CCN(C(=O)CC(OC)OC)CC1CC1 40389,N1(C(C2(C(=O)NC)CC2)=O)CCN(C(c2cn(C)nn2)=O)CC(CO)C1 40390,CC1CCC(Cl)=C(C(=O)NC2CC(NC(C3(n4cncn4)CC3)=O)C2)C1 40391,c1(OC(C(=O)NCC(CNC(C(C)(C)OC(C)C)=O)C)C)ccc(Cl)cc1 40392,C1(CCC)CN(C(c2cc(Cl)ccc2F)=O)CCN1C(=O)CC(O)C1CCCC1 40393,Cc1[nH]c2ccccc2c1CNC1(c2nnnn2C2COC2)CCN(C(C)C)C1 40394,C=CC1CN(C(=O)C(CN(C)C)NC(=O)CCSCC)CCO1 40395,c1(C(N2C(C)CC(NC(C3CCC(=O)NC3)=O)C2)=O)cc(F)cnc1Cl 40396,C(=O)(CCCCC(C)CC)NC1C(CC)CN(C(=O)C(N2CCN(C)CC2)C)C1 40397,C1(CNC(c2cn(C)nc2C(C)(C)C)=O)CC2COCC2N1C(=O)C(C)(C)CO 40398,C(=O)(N=c1nn[nH]n1CCC(C)C)NC(c1ccc(Cl)cc1)CCC 40399,C(=O)(C(C)(C)C(=O)N(C)C)N1CCC(CC(C)NC(C(CC)F)=O)CC1 40400,C12(COC)COC(C(N3CCCC(C(C)NC(=O)C(Br)=C(C)C)C3)=O)(C1)C2 40401,c1(COC)cc(NC2CCCN(C(=O)Cc3cccnc3)C2)ncn1 40402,C(C(=O)N1CCCC1C1CCCC(C)(C)C1)(C(C)(C)C)n1cc(C(=O)OC)nn1 40403,c1(C(=O)NCCOC2CN(C(Cc3cn(CC)nc3)=O)C2)csc(Cl)c1Cl 40404,c1(C(C2(c3cn(C4CCC4O)nn3)CCC2)=O)ccc(Br)c(NC(C)=O)c1F 40405,c1(C(=O)NCC2N(C(C(CCSC)O)=O)CC=C2)cn(C)c(=O)n(C)c1=O 40406,c1(C(N(CC(CNC(Cc2c(C)noc2)=O)O)C)=O)cncc(-n2cccn2)n1 40407,N1(C(c2nccc(OC)c2F)=O)CCC2CCCN(C(c3ccncn3)=O)C2C1 40408,C1(C2CCN(C(C3C(C(C)O)C3)=O)C2)CCCCN1C(=O)C(c1ccncc1)C 40409,C(CCCCCCC(=O)NC(CNC(=O)CC(C)C(C)C)C1CC1)SC 40410,c1(OC)ncc(C(=O)N(C2C3CN(C(c4cnc(OC)cn4)=O)CC23)C)nc1C 40411,CC(O)(CCNC(N1CC2(CCC2)C1CO)=O)C(F)(F)F 40412,c1(C(N2CCCC(CN(C(=O)C#CC3CC3)C)C2)=O)ccc(N)c(N)c1 40413,N1(C(CCOC(C)=O)=O)CC(C2CC2C(=O)N(C2CCOCC2C)C)C1 40414,N1(C(C(C)=O)=O)CCN(C(c2cnc(CC(C)C)s2)=O)CC1C 40415,C1(NC(Cn2c(C)c(Cl)cn2)=O)CC2CCC1N2C(c1cnn(C)c1N)=O 40416,CC1=C(C(=O)NC2CCC(NC(c3cn(C)nc3Cl)=O)C2)C=C2CCCN=C2N1 40417,CCCCCCOC(C)C(=O)NCC(CC)NC(c1ccnn1C1CCCC1)=O 40418,C1(C)(C(=O)NCC2CCN(C(COCC)=O)C2)CNC(=O)C1 40419,N1(C(C2(OC)CC2)=O)CCC(O)(CNC(=O)CC2CCN(C)C2=O)CC1 40420,N1(C(C2(CC=C)CCN(C(=O)C=CCN3CCC3)C2)=O)CCCCC(OC)C1 40421,C1(C2CCN(C(C3CCC34CCC4)=O)CC2)(NC(C(CCCC)O)=O)CCC1 40422,C(c1ccc(C(F)(F)F)cc1C)=CC(N1CCCC(CC)(NC(=O)CC#N)C1)=O 40423,C1(COCCO)CC=CCN1c1nnnn1CC1CC2CCCC12 40424,C1(CNC(C(CC#C)C2CC2)=O)(NC(c2nccnc2C)=O)CC2CCC1CC2 40425,C1(C2(NC(=O)CSc3cscn3)CC2)CCCCN1C(C1CC12CCC2)=O 40426,n1(C(C)C)cccc1C(=O)NCC1CC(F)(CNC(C2(c3ncco3)CC2)=O)C1 40427,C(C(C)C(=O)NCC(C1CC1)NC(c1ccn(CC#N)n1)=O)SC 40428,N1(C(C(Cn2cccn2)NC(c2c(COC)cc[nH]2)=O)=O)CC(CO)C1(C)C 40429,C1(C#N)(C(=O)NCC2(F)CC(CNC(CCC=C(C)C)=O)C2)CC2CC2C1 40430,Cc1[nH][nH]c(=N)c1C(=O)NCCCCCCN(C)C(c1coc(C(F)(F)F)c1)=O 40431,C1(CC(=O)N(CC)CC2CCCN2C(C2CC=CC2)=O)CCC(C)(C)O1 40432,CC1CN(C(=O)CN(C(=O)C2=CCOCC2)C)CCC1N(C)C 40433,C=CCCCC(C(=O)Nc1cccc(NC=O)c1)NC(=O)CCC(=O)CC 40434,n1(CC(=O)NC2C(NC(C(F)=CCC)=O)CC2)cc(Cl)c(C)n1 40435,N1(C(c2ccc(C)c(F)c2)=O)CCN(C(c2cncc(F)c2)=O)CC2(CC2)C1 40436,C(c1cnn(C)c1)=CC(=O)NC(CC=CC(=O)N(C1C(C)CCC1)C)(C)C 40437,C1(NC(CCC(C)OC)=O)CCCC12CN(C(=O)Cc1nc(C)sc1C)C2 40438,C1(C(N(C(CC)C)CCO)=O)COCCN(C(C2(C#N)CC2)=O)C1 40439,C(CCCCC(=O)NC1CC2CCC1O2)n1cc(CC(=O)O)nn1 40440,CC1(C)CCC(CS(=O)(=O)NC2CC(CSC3CCSCC3)C2)OC1 40441,C#CC1(C(=O)N(CCC(N2CC(O)(C(N3CCCC3)=O)C2)=O)C)CC(=O)C1 40442,CCCC(C(=O)NCC1C2CN(C(c3cc(Br)ccn3)=O)CC12)OCC 40443,N1(C(C=C(C)C2CC2)=O)CC(C(=O)NCCn2ncnn2)C(C)(C)C1 40444,C(=O)(CC(c1ccccc1)NC(N)=O)NC(C(C)NC(C=C(CC)CC)=O)C 40445,N1(C(C2(CC=C)CC=CC2)=O)CC2(CCC2NC(=O)CSS(C)(=O)=O)C1 40446,C1(CN2C(C(=O)OC)CC2C)CN(C(=O)OC(C)(C)C)CC1C 40447,C1(CNC(C(N2C(=O)CCC2=O)CC)=O)CC(C)(C)CN1C(=O)CCOC1CC1 40448,C1(NC(COCC=C)=O)CC(C)CN(C(c2c(C)coc2C2CC2)=O)C1 40449,C(CCCC(=O)NCC(c1ccco1)O)NC(c1cc(OC)n[nH]1)=O 40450,C(C(C)(C)CNC(c1ncn(C)n1)=O)N(C(C1(CCC=C)CC1)=O)C 40451,Cc1nc(C(C)C)ccc1C(=O)NCC1CCCC(NC(=O)CNS(N)(=O)=O)C1 40452,N1(C(COCCCC)=O)CCC(C)(C)C(NC(=O)CCOCC(F)(F)F)C1 40453,C1(C(=O)NCC2(Cn3cc(CC4CC(CF)C4)nn3)CC2)COC2(COC2)C1 40454,C1(CNC(c2ncn(CC)c2)=O)CC(C)N(C(C2CCC(=O)N2C)=O)C1 40455,Cc1ccccc1C(=O)NCC(C)CNC(=O)CCCc1cncs1 40456,C(C(CNC(=O)OC(C)(C)C)CO)NC(C1N(C(C2(OCC)CC2)=O)CC1)=O 40457,c1(SCCN(CC(C)O)C(=O)CC(C2(c3cc[nH]n3)CCC2)=O)cccnc1Cl 40458,c1(OC)ccc2cc(C(=O)NC3CCN(C(C4(C)CCN(C)C4)=O)CC3)[nH]c2c1 40459,C1(NC(CCc2nc(=N)[nH][nH]2)=O)CCC2CCN(C(c3csc(Cl)c3)=O)C12 40460,c1(OCCC)cccnc1NC(N1CCC(CC)(CC)C1)=O 40461,N1(C(Cc2c(C)con2)=O)CCC(C)(C)C(CNC(c2cc[nH]c2C(C)C)=O)C1 40462,C1(C2CCOCC2)(C(N2CCC(CNC(C(C(=O)OCC)C3CC3)=O)C2)=O)CC1 40463,c1(C(N(C(c2ccccc2)CNC(C2CCNC2=O)=O)C)=O)cc(Cl)ncc1N 40464,C1(NC(=O)Cc2cccnc2O)C2CC3CN(C(C4CCCS4)=O)C1C3C2 40465,N1(C(C2C=C(C)CS2)=O)CCC2(CNC(C3Cc4cccnc4C3)=O)CCCC12 40466,C1(CN(C)C)CCN(C(C2CC(F)CN2CC(N)=O)=O)CC1 40467,c1(C(=O)NC(CCOC)CNC(=O)CC(C)CF)ccc(S(N)(=O)=O)c(F)c1 40468,C(=O)(C1=CCCSC1)NC1(CNC(=O)COCCCF)CCOCC1 40469,N1(C(c2cc(CC)no2)=O)CC(NC(C2CC2c2ccccc2)=O)CC(F)(F)C1 40470,C12(C(N3CCN(C(c4ccc(C)c(C)c4)=O)C(C)C3)=O)CCCC1CC(=O)C2 40471,CC1(C)CCC(CNC(=O)C(C2CCCCC2)O)N(C(=O)CN2CCSCC2)C1 40472,c1(C(N2CC(C)C(NC(c3cc[nH]n3)=O)C2)=O)cccc(C(C)(C)C)c1N 40473,N1(C(COCCCC#C)=O)CC2CCN(C(c3nnccc3C)=O)CC2C1 40474,N1(C(c2n[nH]c(C)c2O)=O)CCC(C(=O)NC(c2nncn2C)C)C12CC2 40475,C1(C(N2C(CN(C(c3scc(OC)c3)=O)C)CCC2)=O)(OC)CS(=O)(=O)C1 40476,C1(C(=O)NCC2CCC(CNC(CNC(C)=O)=O)CC2)CCCCC1(F)F 40477,c1(CN(c2snc(C(=O)OC)n2)C)cc(C#N)ccc1F.C12CCN(C1)C2=O 40478,C1(C(=O)NCCC(C)(C)F)C2CCN(C(c3cccc(O)n3)=O)CC12 40479,CCC(C)(CCC(C)C)C(=O)NC1CCC(C(N2CCC(O)C(O)C2)=O)CC1 40480,c1(-c2cc(C)[nH]c2C)csc(=Nc2cccc(F)n2)n1CCC1CCSC1 40481,C=CCCC(C)NC(c1cc(C2CCC2)[nH]n1)c1nnnn1CCCF 40482,C=CC1CN(C(C2CC23CCSCC3)=O)CC1NC(c1cnccc1Cl)=O 40483,C=CCC(C(=O)NC(CNC(c1cnc2[nH]ncc2c1)=O)C1CC1)C(C)C 40484,c1(NC2(c3nnnn3C3CC(F)(F)C3)CC(COC)C2)nc2cc(Cl)cnc2[nH]1 40485,C(=O)(C(C)(C)C1=CCN(C(=O)CC2CCCC2C)C1)NC1CC(SC)C1 40486,N1(C(C2(OC)CCOC2)=O)CCCC2(CCN(C(C3(N(C)C)CC3)=O)C2)C1 40487,c1(OC)ncc(C(=O)NCC2(O)CCN(C(c3n[nH]cc3C)=O)C2)c(C)n1 40488,c1(NC2CCN(C(C3CC34CC(O)C4)=O)C2)ncc2ccsc2n1 40489,C12(C(N(C(C3CCCC3)C)C)=O)COCC1CN(C(=O)CCc1csnn1)C2 40490,C(=O)(CC(C)CC(C)C)N1CCC(C(C)NC(C(CCC)CC)=O)C1 40491,c1(CN(C)C(C2(N(C)C)CC2)=O)ccc(CNC(C2CCCS2(=O)=O)=O)cc1 40492,c1(CC(=O)N(c2ccc(F)cc2)CCOCC)ccc(F)c(C(F)(F)F)c1 40493,CC1CN(C(C(=O)NC2CCCC2)c2ncco2)CCS(=O)(=O)C1 40494,Cc1cn2cc(CC(=O)NCC(C)CNC(=O)CC(C)CF)nc2s1 40495,c1(C(=O)NCC(C2CC2)NC(CCC(=O)NCC)=O)nccc(Cl)c1Cl 40496,n1(C(CNC(C(C)n2cncn2)=O)C)cc(CCCNC(=O)C(F)(F)F)nn1 40497,C1(NC(c2ocnc2C2CC2)=O)CCCC1CNC(c1snnc1C1CC1)=O 40498,c1(C(=O)NC(c2ncc[nH]2)CC)ccc(CNC(=O)COc2ccsc2)s1 40499,CC1=C(C(=O)N2CCC(O)(C(C)NC(=O)C(C)NC=O)C2)CCO1 40500,Cc1ccc([N+](=O)[O-])cc1C(N1CCC(F)(F)C(NCc2cnn(C)c2C)C1)=O 40501,N1(C(C(C)=NOCC#N)=O)CCC2(C=C(C(=O)N(C3CCOC(C)C3)C)C2)C1 40502,C1(C(=O)NCC2CCCC(CNC(c3c(C)nsc3)=O)C2)C2CCC(F)(F)C12 40503,c1(CC)sc(C(=O)NC(C)(C)CNC(c2cc(CC(C)C)[nH]n2)=O)cc1C 40504,C(CCCC(=O)N1CC(C(=O)NC2CCS(=O)(=O)C2)OC(C)C1)(OC)OC 40505,CCCCC(CC)C(=O)N1CC(C(=O)NCCN2CCC2)CC1(C)C 40506,C1(C(=O)NCC(CNC(c2ccn(CCCC)n2)=O)(C)C)C2CCC(=O)C12 40507,c1(C(=O)NCc2c(CNC(CCCC#CC)=O)cccc2)cnc2[nH]nnc2c1 40508,N1(C(c2ncn(CC)c2)=O)CCC2(NC(c3cc(C)ccc3F)=O)CCCC12 40509,c1(C(N2CCN(C(C3C(C)=CCC=C3)=O)CC2)=O)ccc(C(C)C)c(Br)c1 40510,CC1(NC(c2ccc(F)cn2)=O)CCN(C(=O)C=CBr)C1 40511,Cc1occc1C(=O)NC(C1CCCN1C(c1cc(CCO)on1)=O)(C)C 40512,C#Cc1cncc(C(=O)NCC(CNC(=O)Cc2ccc(Br)cc2)OC)c1 40513,c1(C(N2CC(SC)C2)=O)[nH]c(C)c(CNC(=O)COC2CCOC2)c1C 40514,C(=O)(C(Cc1ccco1)NC(=O)CC1CNC(=O)O1)N(CCCC)CC 40515,Cc1c(C(=O)NCC(c2ccccc2)NC(=O)CN(C)C2CC2)nc2sccn12 40516,C1(C(=O)NCC(CNC(Cc2c(C)ncnc2C)=O)C)OCC2CCCCC12 40517,CCC(CC(=O)NC1CCC(C)(NC(c2cnn(C)c(=O)c2)=O)CC1)CC(C)C 40518,c1(C2(C(N3CC(C(C)NC(c4c(C)cco4)=O)C3)=O)CC2)ccc(F)c(Cl)c1 40519,CCCCC(CC)C(=O)NC1CC(C)(C(=O)N(C)Cc2ncc[nH]2)C1 40520,C(=O)(C1=CC2(CN(C(=O)C(O)CN3CCCC3)C2)OC1)NCC(COC)(C)CO 40521,c1(C(N2CC(C)NC(=O)C2)=O)ccc2c(n1)CCN(C(=O)Cc1ccccc1)C2 40522,CCCCCC(C(=O)NC1CCC(NC(=O)Cc2cn(C)nc2Cl)CC1)C(C)C 40523,c1(C(N(CC(CNC(COC)=O)C)C2CC2)=O)oc2ccccc2c1CS(C)=O 40524,c1(CNC(C2(NC(CCC=CC(C)C)=O)CCC2)=O)ccc(F)c(F)c1 40525,C1(C(=O)NCCCN(CC)CC)CCCCC1(C)NC(c1cc(C)sc1C)=O 40526,N1(C(CC2CC(OC)C2)=O)CCCC1(C)CNC(=O)CC1CCC=CCC1 40527,C1(C(N2CC(CNC(c3cncc(C)n3)=O)OCC2)=O)CCCCC1(C)C 40528,C(C(F)(F)C(N)=O)NC(C1(CCC=C)CN(C(=O)CN2CCC(C)C2)C1)=O 40529,Nc1cc2c(cc1C(=O)NC1CCC(NC(C3CC3(Cl)Cl)=O)CC1)CCC2 40530,C(=O)(CCCC(F)(F)CO)N1CC(CNC(=O)CC23CCC(CC2)CC3)C1 40531,C1(F)(CNC(C(SC)SC)=O)CCN(C(=O)C=Cc2cn(C)cn2)CC1 40532,c1(C(=O)NCc2c[nH]c(=NC)s2)ccc(OC)cc1S(C)(=O)=O 40533,Cc1nc(C=CC(=O)N(C2CCC(NC(=O)Cc3ccco3)C2)C)cs1 40534,c1(SC)ccc(NC(=O)NCCOc2cccc(F)n2)cc1C#N 40535,N1(C(c2ccn(CCC)n2)=O)CCC(C)(C)C1CNC(=O)C(C)(CC)CO 40536,c1(C2(COC(CN(C(CC)(C)C)C3CC3)=O)CCC2)ccc(Cl)c(Cl)c1 40537,c1(C(N2CC(C(=O)Nc3ccc(O)nc3)SCC2)=O)cn2ccc(Cl)cc2n1 40538,c1(OC)cc([N+](=O)[O-])c2cc1NC(=O)N2.C(C(=O)CCC(C)C)OC 40539,C1(O)(C(=O)NC(C2CN(c3cc(CC(C)C)ncn3)C2)C)CC2CCC1C2 40540,N1(C(CCC)=O)CCCN(C(c2cc(C)n(C3CCCCC3)c2C)=O)CC1CO 40541,C(=O)(CCCCc1ccc(C)cc1)NCC(C)N(C(c1cc(C)no1)=O)C 40542,C(C)(C)(CCCCC(=O)NCC(C1CC1)N(C(=O)C1=CCC1)C)OC 40543,C1(NC(Cn2ncc(NCC)c2)=O)CCN(C(=O)OC(C)(C)C)CC1C 40544,Cc1cc(N2Cc3ncsc3C2)nc(=NCCCc2nncn2C)[nH]1 40545,N1(C(c2c(C)nco2)=O)CCC2(CC(NC(=O)C(F)(F)c3ccnn3C)CO2)C1 40546,c1(C2CN(C(=O)OC(C)(C)C)C2)nnc(S)n1C.N12CCC1(C)C2=O 40547,C#CCCCCC(=O)N1CCCC(C)(CNC(=O)C(CCC)OC)C1 40548,C1(C(N2C(C#C)CCCC2)=O)CN(C(=O)Cc2cnnn2C)CCC1(C)C 40549,N1(C(C2CCCC(OC)C2)=O)CC2CC(NC(C3CC(=O)NC(=O)C3)=O)CC1C2 40550,c1(C(=O)NCC2=CCN(C(CCOCC#C)=O)CC2)cc(=O)c2ccccc2o1 40551,Cc1cc(F)c(C(N2CCC(C)(CNC(=O)C=Cc3cncs3)C2)=O)c(F)c1 40552,Cc1cc(C(N2CC(C)(CCC(=O)NCCOCCCF)C2)=O)cnc1C 40553,CC1CN(C(c2ccncc2F)=O)CC1CCNC(=O)CC1CCC(F)(F)C1 40554,CC1CC(C(=O)NCCC2(NC(=O)Cc3ccc(O)nc3)CC2)CC(C)C1 40555,N1(C(C(c2cnn(C)c2)C)=O)CCC(C2(NC(=O)Cc3cc(Cl)n(C)n3)CC2)C1 40556,C1(NC(C(C)OC)=O)CCC(NC(=O)Cc2cnn(C)c2C)CC1 40557,c1(C(=O)NC2C(CNC(c3ccc(CC)nc3)=O)CCC2)cccc(Cl)c1C 40558,N(C)(S(=O)(=O)N(C)C)CC(=O)NC(C)CNC(c1cn(C2CCCC2)nn1)=O 40559,C1(NC(C=CC=CC)=O)CCC(C)(CNC(=O)CC2(OC)CCOCC2)C1 40560,C=C(C)CC1C(=O)N(C)CC=CC(=O)N1.C(C)(CCSC)SC 40561,C1(C#N)(C(N2CCN(c3n(C)cc(C#N)n3)CC2)=O)C(C#N)C1(C)C 40562,N1(C(CC2N(C(C(CC(C)C)O)=O)CCC2(C)C)=O)CCOC(C)(C)C1C 40563,c1(OC(C(=O)N(CC(CNC(C2N(C(C)=O)CSC2)=O)O)C)C)ccc(C)cc1 40564,N1(C(c2c(CC)n(CC)nc2)=O)CCCN(C(=O)CC2(OC)CC2)C(C)C1 40565,c1(C(=O)NC2C(NC(C3(COC)CCCC3)=O)C2)cc(F)c(N)c(F)c1 40566,c1(OC)cc(NC(C2CCCN2C(c2ccc(C)nc2O)=O)=O)ccc1O 40567,N1(C(c2c(CC)cccn2)=O)CCCC12CCN(C(C1CC=CCC1)=O)C2 40568,c1(CC(=O)NCC2N(C(C(C(C)C)OC)=O)CCCC2)cc(F)ccc1Cl 40569,c1(C(=O)NCC(CC)NC(=O)C(C)(C)C(N)=O)ccc([N+](=O)[O-])cc1 40570,N1(C(c2c(COC)cc[nH]2)=O)CC(CNC(=O)C=C2CCN(C)C2)CC1(C)C 40571,Cc1nc(C(=O)NC2(CN(C)C(C3(C)CC=CCO3)=O)CC2)ccc1C#N 40572,Cc1occ(-c2ccccc2)c1C(=O)NC1C=CCN(C(=O)C#CC(C)C)C1 40573,CCCC(C(=O)N1CCC1Cn1cc(-c2cnn(C(C)C)c2)nn1)OC 40574,C1(NC(=O)NCCC(C)(C)c2ccccc2)CCOC(c2cccc(F)c2)C1 40575,C(=O)(C=CCNC(=O)COC(C)=O)N(CC=C)CCO 40576,N1(CC2(O)CCN(c3c(OC)cccn3)CC2)CCC2(CCCC2)C1 40577,C1(CNC(C2CC(OC)C(OC)C2)=O)CCCN(C(=O)Cc2coc(C)n2)CC1 40578,c1(CC(=O)NC(CC)CNC(C23CCC2C3)=O)nnn(-c2cccc(Cl)c2)c1C 40579,C1(C(=O)NC2CCCCN(C(CC3OCC(C)(C)C3)=O)C2)CNC(=O)CC1(C)C 40580,N1(C(c2c(C)cns2)=O)CCOCCC1C(=O)NCCc1cncs1 40581,C1(NC(CC2CC(C)C2)=O)CC2(C1)CC2NC(c1ccc(SC(F)(F)F)o1)=O 40582,C(=O)(C(C)(C)CCF)N1CC(CN2CCN(C(C3C(CCC)CCC3)=O)CC2)C1 40583,c1(C(=O)NC(C(C(C)C)C)CNC(c2cccnc2O)=O)noc2c1CCCC2 40584,CC1(C)CCC(C(N2CC=CC2(C)C(=O)NCCN2C(=O)CNC2=O)=O)C1 40585,N1(C(c2ccccn2)=O)CCC(NC(C2(CC)CC2)=O)C1Cc1ccccc1 40586,C1(NC(c2cc(CCC)on2)=O)CCCN(C(=O)C=C(CC)CC)C1C 40587,C1(O)(CCNC(C2CC3CC3C2)=O)CCN(C(c2ccc(O)nc2)=O)CC1 40588,c1(C(N2CC(CNC(CCC3CC(C)C3)=O)OCC2)=O)ccc(F)c(Cl)c1N 40589,Cc1c(Br)csc1C(N1CC(CC(C)NC(=O)C(C)C2CCC2)C1)=O 40590,C(C(=O)N1CC(O)C(O)CO1)C1N(C(c2ncc(CC)cn2)=O)CCC1(C)C 40591,C1(C(=O)NC2C(OC)CN(C(C3(C4CCC4)CC3)=O)C2)CCC(C)(O)CC1 40592,C1(CNC(C2CCCC(NC(CC(C)F)=O)C2)=O)CC12CCOCC2 40593,C1(C)(CCC(=O)NC(CC)CN(C(=O)COC2CCC2)C)CCC(=O)N1 40594,C(=O)(C(C)CC(C)(C)C)N1CCC(N(C(Cn2ncc(CC)c2)=O)C)C1 40595,c1(N(CC(O)CF)C)ncc(S(=O)(=O)NCC2CC(=O)N(C(C)(C)C)C2)cc1Cl 40596,CCCCCCC(C)C(=O)N1CCCC1CN(C)C(C1CCCCN1N=O)=O 40597,N1(CC(=O)NCC=CCNC(C(c2ccnn2C)C)=O)CCCCCCC1=O 40598,C(=O)(C1=CCOCC1)N1CCN(CC(=O)Nc2c(C(C)C)n(C)nc2)CC1 40599,Cc1cc(NC(=O)C(=O)NCCc2ccc(Br)s2)ncn1 40600,C(c1ccncn1)=CC(=O)NC(C(=O)NCC(=O)N(C)C1CC1)C1(O)CCC1 40601,Cc1cccc([N+](=O)[O-])c1C(N1CC(N(C(=O)CC2OCCC2C)C)C1)=O 40602,c1(C(=O)NCC(CNC(C2CCN(C)C2)=O)(C)O)c[nH]c2cccc(Cl)c12 40603,C(=O)(CS(=O)C(F)(F)F)NC1C(CO)CCN(C(C(C)OC(C)=O)=O)C1 40604,CC1CCc2ncc(C(N3CCC(NC(c4cnc(C(C)(F)F)s4)=O)C3)=O)n2C1 40605,N1(CC(=O)NC(C)CN(C(=O)C(C)C2CCC2)C)CCCNS1(=O)=O 40606,N1(C(C2CC(N(C)C)C2)=O)CCC(C)(CNC(C2CC3C=CC2C3)=O)CC1 40607,C12(NC(c3oc(C)c(CO)c3)=O)CCCC1CN(C(c1ccoc1C1CC1)=O)C2 40608,N1(C(C2(COC)CCC2)=O)CC(C(N2CC3CC2CC3CF)=O)OC(C)C1 40609,N1(C(c2c(N)nccc2)=O)CCC=C(CNC(=O)CCN2CCCC2)C1 40610,CCCCC(C)C(=O)N1CC(C(=O)N(CC)CC2CCOC2)C(F)C1 40611,c1(C(N2CC(C#N)OCC2)=O)cc(-c2cccc(OC(F)F)c2)c2[nH]ccc2c1 40612,C[S+](C)CCC(O)C(=O)N1CC(O)(CCNC(=O)COC2CCOC2)C1 40613,c1(C(=O)NCC2N(C(C=CC(C)(C)SC)=O)CC(O)C2)cc(C2CC2)nc(O)c1 40614,c1(C(C(=O)NC)N(C2CCC(F)(F)CC2)C)ccc2c(c1F)CCC2 40615,c1(C(=O)NCC(CNC(C(CC)(C)OC)=O)CO)ccnc2ncccc12 40616,c1(C(N2C3CN(C(c4c(OC)ccnc4O)=O)CC32)=O)ccc2c(C)noc2c1 40617,N1(C(c2c(CC)ncs2)=O)CC2CN(C(c3cnc(C(C)(C)C)o3)=O)CC(C1)O2 40618,c1(N2CCN(CC)CC2)cc(C)c(S(=O)(=O)NC)cn1.C(C)(C(C)SC)NC(=O)OC 40619,C12(C(=O)Nc3c(CC)cccc3C)CCN(C(=O)CC(O)C(C)C)CCC1C2 40620,Cc1ccc(CN2CCCC2CCC(=O)Nc2ccnc(OC(C)C)c2)cn1 40621,c1(C(N2CCC3CCN(C(CC=C)=O)C3C2)=O)cnc2c(c1)OCC(=O)N2 40622,N1(C(Cc2c(C)occ2)=O)C(C)C2CC1C2NC(c1cccnc1O)=O 40623,N1(C(COCC#C)=O)CCC(NC(=O)CCc2cccs2)C1C1CC1 40624,c1(OC)cc(N)ccc1C(=O)NCC1CCC1NC(=O)CCN1CCNC(=O)C1 40625,C1(C(=O)OC)(Nc2c(CS(=O)(=O)N(CCCC)C)cccc2)CCC(C)(C)C1 40626,C(N=c1ccc(CC(F)F)c[nH]1)N(C(C)C)CCN 40627,c1(NC(N2CCC(NC(CN3C(C)CC3)=O)(CO)C2)=O)cccc2c1CCCC2 40628,c1(NC(c2c(OC)cc(OC(F)(F)F)cc2)=O)cc(F)c(C)c(F)c1 40629,c1(C(=O)NCC(CN(C(c2c(COC)ccs2)=O)C)C)cc(S(N)(=O)=O)ccn1 40630,N#Cc1cc(C(=O)NCC2CC2NC(c2c(Cl)ccc(F)c2F)=O)c(N)nc1O 40631,C12(CCOCC1)C(=O)NCCCCN(CC)C2=O.c1(C(C)CO)ccccc1 40632,c1(NC(c2cc(-c3ccc(C)o3)[nH]n2)=O)nccnc1C(=O)Nc1ccccc1 40633,CC1CCCCC1(CNC(c1ccc(O)c(O)c1)=O)NC(c1c[nH]ccc1=O)=O 40634,Cc1cccc(S(C)=O)c1NC(=O)C(N1CCCC(C)C1C)=O 40635,C1(CNC(c2scc(C)c2)=O)CC(NC(c2coc(N(C)C)n2)=O)C12CCC2 40636,C(=O)(C(O)CCNC(C1COCCN1C)=O)NC(c1cc(C)no1)(C)C 40637,C1(CNC(c2c(CC)cncc2)=O)N(C(=O)CCNS(C)(=O)=O)CCCC1(C)C 40638,C(=O)(CCCNC(=O)C(C)Cn1ccnc1)N(CCC(=O)OC)CC=C 40639,c1(CC)nc(C)[nH]c1C(=O)NC1CC(CCNC(=O)Cc2[nH]cnc2C)C1 40640,CC1(NC(=O)COC2CCOC2)CCCN(C(c2c(Cl)nsc2Cl)=O)C1 40641,c1(CC(C)NC(=O)COC2CN(C(=O)C(C)C3CCCC3)C2)ccc(Cl)s1 40642,C1(C(C)C)N(C(c2cncn2C)=O)CC12CCN(C(C1CC1F)=O)CC2 40643,N1(C(C(=O)NCCC2(OCC)CCOCC2)=O)CCCCNC(=O)C2CCCC12 40644,CC(C)(C)C(CC(=O)NCC1CCN(C(=O)CN2CSCCSC2)C1)C(F)F 40645,c1(C(=O)NC2(COC)CN(C(C3CC3c3ccccc3)=O)C2)ccc(SC)cc1 40646,CN1CCOCC1C(=O)NCC1(C(N2CC=CC2CF)=O)CC1 40647,Cc1c(C(=O)NC(C)CNC(=O)CCc2ccon2)ccn1C 40648,c1(C(N2CC=CC(C(=O)OCC)C2)=O)cc(S(=O)(=O)NC)cn1C 40649,C(=O)(C1=NOC2(CCN(S(=O)(=O)CC3CCCO3)C2)C1)Nc1cccc(C#N)n1 40650,N1(C(COCCOC)=O)CCC2(CCCCN(C(c3coc(COC)n3)=O)C2)C1 40651,C12(CNC(C(C3CC3)OC)=O)CCCC(CN(C(=O)C(C)(C)c3ccno3)C1)C2 40652,Cc1cc(OCC(N2CC(C)C2c2ccccc2)=O)no1 40653,c1(N2CC(NC(C3C(C)(Br)C3)=O)(CO)C2)ncncc1Br 40654,N1(C(C2C(C)(C)CC2)=O)CCCCC1C1CCN(C(c2cc(Br)no2)=O)CC1 40655,N1(C(c2c(CC)n(CC(C)C)nc2)=O)CCCC(CNC(C2CC(=O)N2)=O)CC1 40656,N1(C(C(C2CCN(C(=O)C(N3CCOCC3)C)C2)C)=O)CCC(O)C(C)C1 40657,C1(C(N2CCC(C(=O)OC)C2C)=O)CC2C=CC1N(C(=O)C(C)n1ccnn1)C2 40658,Cc1sc(C)c(C(N2CC3(CC(NC(=O)C(C)CC(N)=O)CO3)C2)=O)c1C#N 40659,C1(C(=O)OCC)CCC(C)(C(=O)NCCN(C(=O)Cn2nccn2)C)C1 40660,CC(c1ccccc1)=CC(=O)NCC1CCC1NC(C1(N(C)C)CC1)=O 40661,N1(C(C(C)CC(F)(F)F)=O)CCCC2(NC(=O)CN3CCC3)CCCC12 40662,C1(CC(=O)NCC(C(C)C)(C)C)C2CCC(C2)N1C(=O)CCCn1cncn1 40663,c1(C(N2C(CNC(COC3(C)CCC3)=O)CC2)=O)ccc(Cl)cc1Br 40664,N1(C(CN(C2CC2)CC)=O)CCN(C)CC1C(=O)NCCCc1n[nH]c(C)n1 40665,c1(C(N(CCCNC(=O)Cn2cc(C3CCOC3)cn2)CC)=O)ccc(O)nn1 40666,N1(C(C=C(C)C)=O)CCC2(NC(=O)COc3cccc(C)c3)CCCC12 40667,Cc1ccsc1C(=O)N(CCC(=O)NC(CCO)C1CCCC1)C1CC1 40668,C(=O)(CCCS(=O)(=O)N1CCCC1)NC(CN(C(COCCC#C)=O)C)C 40669,c1(OC)cccc(Cl)c1CC(=O)NC1CCN(C(=O)CC2OCCO2)C(C)C1 40670,c1(COCC(=O)NCC(CN(C(CN(C)CC)=O)C)C)ccnc(O)c1 40671,N1(C(CC(C)C)=O)CC2CCCC1CN(C(=O)Cc1ccc3nc(O)[nH]c3c1)C2 40672,C(=O)(CCCC(C)(C)C)NCc1cn(CC(=O)NC(CC(C)C)C(N)=O)nn1 40673,N1(C(C(C)S(N)(=O)=O)=O)CCC2(CCCC2NC(c2cc(Cl)cn2C)=O)CC1 40674,C(CCCC(=O)NCC1(O)CN(C(c2cn(C(C)(C)C)nc2C)=O)C1)NC(C)=O 40675,N1(C(c2ncc(NC)nc2)=O)CCC(C(=O)N(C)CC2CCN(C)C2)=C(F)C1 40676,O=C(C1=CC2CCCC12)NCC1CC(NC(c2ncnc(O)c2Br)=O)C1 40677,CCC(C)C(O)C(=O)NCC(CO)NC(c1ccc(F)c(C(F)(F)F)c1)=O 40678,CCC(C(=O)NC1C=CC(CNC(=O)CCc2ccn(C)c2)C1)C(C)(C)CC 40679,C#CC1(C(=O)NCCN2CCOC(C)C2)CCN(C(=O)CC2CSC2)CC1 40680,c1(C(c2nnnn2C2(CO)CC2)NCC2C(C(C)(C)C)C2)ccc(F)c(Cl)c1.OC 40681,c1(C(N2CC(CNC(c3ccco3)=O)C(C(F)(F)F)C2)=O)cnc(F)c(F)c1 40682,Cc1[nH][nH]c(=N)c1C(=O)NCC1(O)CCN(C(=O)CCC2CNC(=O)N2)C1 40683,C1(CNC(=O)CNC(C2(CCF)CC2)=O)CCN(C(c2cccs2)=O)CC1(F)F 40684,c1(C(N(CCCCC2C(C)C2)C)=O)ncnc2c1ncn2C1CC1 40685,c1(C(N(C2CCCN(C(CC(C)F)=O)C2)C)=O)ccc2oc(S)nc2c1 40686,C1(NC(C(C)SC(C)C)=O)CCCN(C(=O)COCc2ccc(Cl)cc2)C1 40687,N1(C(C2(NC(c3n(CC)nnc3)=O)CC(CO)C2)=O)CCC(O)CC1 40688,N1(C(C(C)N(S(CCC)(=O)=O)CCC)=O)CCC2(CCOCC2)C(NC(c2ccccc2)=O)C1 40689,N1(C(CC=C=C)=O)CCC(NC(c2ccn(-c3ccccc3)n2)=O)C1C(C)C 40690,c1(C(N2CC(C(=O)Nc3cc(C(CC)C)no3)C2)=O)cc(NC(C)=O)ccc1F 40691,c1(CC)cc(NC(=O)NCC(C)CN(C(=O)COCC2CC2)C)oc1CC 40692,c1(C(=O)NCC(CC)NC(c2cnn(CCO)c2C)=O)cccc(F)c1OC 40693,C(=O)(C1=CC2CCC(C1)C2)NC1CC(NC(CSCC)=O)CC1O 40694,C1(NC(=O)CS(=O)(=O)NC2CC2)CN(C(=O)C=CBr)CC2(CC2)C1 40695,N1(C(c2cc(CNC(c3c(C)ocn3)=O)nn2C)=O)CC2(CC2)CC1CO 40696,C=C(F)C1(CC(=O)N(CCC(=O)NCC(c2ncn(C)n2)C)CCCO)CCC1 40697,c1(C(C(=O)NCC(C)C)N(C2CCCC2)C(C)C)c2c(nn1C)CCSC2 40698,O=C(N=c1[nH]ccc2cc(Cl)ccc12)C1CCN1C(c1c(Cl)cc(F)cc1Cl)=O 40699,C(=O)(C1=C(C)CCOC1)N1CCCC(=O)N2C(CCC2)C1.C(C)(C)(C)SC 40700,C1(NC(=O)NCC(c2ccsc2)C)CCC=CC1O 40701,N1(C(c2ccc(OC)o2)=O)CCN(C(=O)CC(=O)N(C)C)C2CCCCC2C1 40702,c1(C(N2CCCC(N(C(C3CC=C(C)CC3)=O)CCF)C2)=O)cc2n(n1)CCC2 40703,c1(OCc2cn(CC(CNC(c3ccc(CC)o3)=O)OC)nn2)cccc(F)c1 40704,C12(CNC(CCCC#C)=O)CCC(C1)N(C(=O)C(C)NCC1CCC(=O)N1C)C2 40705,C1(OC)CN(C(=O)CCN(CC(F)(F)F)C)CC1NC(=O)Cc1cccn1C 40706,Cc1ncc(Br)c(Nc2nc(C)c(C(N3CCCC(CO)C3)=O)s2)n1 40707,CC1CCN(C(C2CC(=O)NC(=O)C2)=O)CCN1C(=O)C=CC=C(Cl)Cl 40708,C1(C)(CC)CCN(C(=O)CC2(NC(=O)COC)CCC2)CC1 40709,C1(C(N2C(CCNC(=O)Cc3ncc(Cl)s3)COCC2)=O)CC2CCC(C1)C2 40710,C1(CNC(c2c(C)c[nH]n2)=O)CN(C(c2ccc(F)cn2)=O)CC1C(F)(F)F 40711,Cc1nnc(NCC(C)N(C)C(c2ncccc2Cl)=O)c(C#N)c1C 40712,C#CC1CC2(CC2)CN1C(C1CCN(C(C2CCCCC2OC)=O)CC1(C)C)=O 40713,c1(CC(=O)NCCC(=C)CNC(=O)CCCc2ccsc2)nn(C)cc1Br 40714,C(=O)(C(CC1CCC1)NC(=O)COC1CC=CC1)NCC(C)SC 40715,c1(OC)cccc2c1OCCC2NC(c1c(Br)ccc(C(F)(F)F)c1F)=O 40716,N1(C(c2c(C)cncn2)=O)CCC(O)C(C(=O)NCC(C)(C)CN(C)C)C1 40717,N1(C(c2nc(OC)oc2)=O)CC2=C(C1)CN(C(=O)CC1COCC3(CCC3)O1)C2 40718,C(=O)(C1CC(C)(C)Oc2ccccc21)N(CCCCNC(C1CC1(C)C(F)F)=O)C 40719,C1(N(C(C(CC)O)=O)CC2CC2)CCN(C(=O)C=Cc2sccc2C)CC1 40720,c1(C(=O)NCC2N(C(C(C)S(N)(=O)=O)=O)CC3(CC3)C2)coc2ccc(O)cc12 40721,N1(C(c2cc[nH]n2)=O)CCCC(C2CCCN2C(=O)Cc2ccccc2Cl)C1 40722,N1(C(c2c(C(C)C)nn(CC(F)F)c2)=O)CC(C)CCC(C)C1 40723,CN1CC2(CCN(C(NC3CCCc4ccoc43)=O)CC2)c2ccccc21 40724,N1(C(C2C(C(=O)OC)C=C2)=O)C(C(=O)NCc2cnn(C)c2OC)CC2CC12 40725,c1(OCC(=O)Nc2c(C(=O)OCC)cncn2)cc(C)ccc1C(C)C 40726,c1(NC2(CNC(C3(C)CC(C)OCC3)=O)CCCC2)ncc2c(ncn2C)n1 40727,C1(CC(=O)NC)SC(=Nc2ccccc2CO)N(Cc2cc(Br)ccc2Cl)C1=O 40728,N1(C(c2cn(C(C)C)nc2)=O)CCC(C)(CNC(c2[nH]nnc2C2CC2)=O)CC1 40729,CC1(OCC(=O)NC2COCC2NC(=O)C=CCOCC(F)(F)F)CCOCC1 40730,c1(C(N(CCCCCCNC(C(C)=C(C)C)=O)C)=O)cc(=O)n(C)cc1Br 40731,CCC(CC(=O)N(C(C)C(=O)NC1(CCO)CCCCC1)CC)OC 40732,C1(C(N2CCCC(NC(=O)CCC(F)(F)F)CC2)=O)CCc2nc[nH]c2C1 40733,C1(CC(=O)NCC(CNC(CCOCC#C)=O)(C)C)CCC(=O)N1CC 40734,C(C)(C)(C(=O)N1CCCCO1)C1CCN(C(c2ccn(CCC)n2)=O)C1 40735,Cc1ccsc1C(N1CCC(NC(C2(CC3CC3)CCCO2)=O)C1)=O 40736,C=CCC(C)(C)CC(=O)NCC(O)CCNC(C1(CC)CC1)=O 40737,C1(CNC(C(C)Sc2nncn2C)=O)CCCCN1C(=O)Nc1ccccc1F 40738,N1(C(C2C3COCC23)=O)CCC2(CCCN2C(=O)C2=CCCC2)C1 40739,c1(-c2[nH]c(=NCc3c(OC)c(F)ccc3)sc2)cc(F)c(C#N)cc1F 40740,N1(CCCc2cccc(C)c2)CC2CCC1CN2C(c1nnn(C(C)(C)C)n1)=O 40741,C1(C(N2C(CCNC(C(C)(Cl)Cl)=O)CCCC2)=O)CCC2CCC1O2 40742,CCC(O)C(C)(C)C(=O)N1CC2CCCC2(NC(c2ccoc2C2CC2)=O)C1 40743,C(=O)CCC(F)(F)Cn1cc(C(C)(C)O)nn1.C1(NC(C)C2CC2)(C)CCCCC1 40744,N1(C(c2c(OC)cncc2)=O)CCC(C)(C)C1C(=O)NCCCSCCO 40745,c1(OC)cc(Cl)c(C(N2CCCN(C(C)=O)CC2)C(=O)NC2COC2)cc1OC 40746,c1(NC(c2n(CCOCC)nnn2)CCOc2ccccc2)ccc(Cl)cc1 40747,C1(N(C(c2ncn(CCNC(C(C3CC3)OC)=O)c2)=O)C)CCC(C)(C)C1 40748,C(=O)(C=C1SCC(=O)N1C)N1C2CC(NC(C(COC)(F)F)=O)CC1CC2 40749,CCC(C)(C)C(=O)NCc1nc(C(=O)Nc2ccc(C(N)=O)cc2)c(C)o1 40750,c1(OC)ccc(CC(=O)NC2C3CN(C(=O)C(F)=CC4CC4)CC23)cc1 40751,C1(CNC(CC2CCN(C)C2)=O)CC12CCN(C(=O)Cn1nnc(=O)[nH]1)CC2 40752,Cn1nnc(CNC(=O)Cc2csc(-c3ccco3)n2)n1 40753,C1(C(=O)NCC2CN(C(CC(=C)C)=O)CC2C(F)(F)F)Cc2nccn2C1 40754,n1(CC)c(C(=O)NC(CC(N)=O)c2cn(C3(C)CCCC3O)nn2)cnc1O 40755,c1(C(N(CC(CNC(CCC(=C)C)=O)O)C)=O)cnc2c(cnn2CC)c1 40756,N1(C(C(CC=C)CNC(=O)CNC(C)=O)=O)CC(C)CCCC1C 40757,c1(NC(C2C(C(N(c3ccc(Br)c(Cl)c3Cl)C)=O)C2)=O)cccc2cn(C)nc12 40758,C1(CC=C)(NC(=O)C(c2ccccc2)F)CCN(C(=O)C(C)(C)COC(C)C)C1 40759,S(=O)(=O)(c1ccc(=NCc2cnn(C(C)(C)C)c2)[nH]c1)N(C1C(C)CCCC1)C 40760,c1(C(N2CCC(CNC(CCCSC)=O)C2)=O)ccc(Sc2ccsc2)cc1 40761,CC1(NC(=O)NC2CCOC2)CN(CCO)C1 40762,C(C1CCCN1C(=O)CN1CCCC1C)=CC(=O)N(C)CC1CC(=C)C1 40763,c1(OC)ccc(F)cc1C(=O)C(=O)NCC1COCC1NC(C12CC(F)(C1)C2)=O 40764,C#Cc1cncc(C(=O)NC2CCCCC2CNC(=O)C(F)C(C)(F)F)c1 40765,C1(C(N2C(COC)CCCC2)=O)CN(C(=O)C(C)c2cc[nH]n2)CC1(C)C 40766,c1(C(N2C(C(=O)NCCNC(=O)NC)COCC2)=O)cc(C)c(F)cn1 40767,CN1CCN(C(=O)Cc2ccsn2)C(C(=O)NC2CCN(C)C2)C1 40768,N1(C(CC(CC)C)=O)CCCCCC(NC(C2OCCC2(C)C)=O)C1 40769,c1(C(=O)NC2CCN(C(c3c(C)nn[nH]3)=O)CC2C)cc2c(s1)CCSC2 40770,Cc1cc(F)c(Cl)cc1C(=O)NCC(C(C)(C)C)NC(=O)CC(O)C(C)C 40771,C1(NC(COC(CC)CC)=O)C2CCC1CN(C(c1cc(O)n(C)n1)=O)C2 40772,C(=O)(CC1=CCCCC1)NCC1CCCN(C(CCCOC(C)=O)=O)C1 40773,c1(C(C(=O)NCCCCNC(c2n(COC)ncc2)=O)C)ccc(Cl)c(Cl)c1 40774,CCC(C(C)O)NC(c1c[nH]nc1CNC(c1cc(C2CC2)on1)=O)=O 40775,C1(CC(=O)NCCN(CC(C)O)C(=O)C=Cc2ccsc2)CCC(F)(F)CO1 40776,c1(C(C)C)cc(C(=O)N(C(C)C(=O)N(CC(O)CO)CCO)C2CC2)n[nH]1 40777,C=CCC(CC(=O)N1CCCC(N(C)C)CC1)NC(c1ccc(C)c(C)c1)=O 40778,C(CCN(C)C(C1CCC(O)CN1C)=O)(C(C)(C)C)NC(C1ON=C(C)C1)=O 40779,c1(C(N2CC(NC(c3ccc(C)cn3)=O)C3C2C3)=O)cnc(C2CC2)nc1C 40780,CC(C)CC(C)(C)C(=O)NC1CCOCC1NC(C1CN(CC(F)(F)F)C1)=O 40781,Cc1nn(C)c(C)c1CNC(=O)C(C(C)O)NC(=O)OC(C)(C)C 40782,C(=O)(C1=Cc2ccccc2OC1)NCC(CN(C)C(C1CCCC1(C)C)=O)(C)C 40783,c1(C(C(=O)O)NC(C2(C)COC(=O)C2)=O)cccc(Cl)c1Cl 40784,C(C)(C)(C(C)NC(C1(N(C(=O)CC2CCC2)C2CC2)CCC1)=O)OC 40785,C(=O)(C(C)C(O)C(C)C)N1CCC(C(C)NC(C(Br)=C(C)C)=O)CC1 40786,C1(C(=O)NCC(C)N(C)C(c2csc(C3CCCCC3)n2)=O)CC=CCC1 40787,C1(C)(CC(=O)N(CCN(C)C)CCO)CCN(C(C2(O)CCCC2)=O)C1 40788,c1(C(N(CCCCCNC(CC(CCC)C)=O)C)=O)ccc(=O)n2c1COCC2 40789,c1(C(=O)NCC2CCN(C(=O)Cc3ccnc(Br)c3)C2)cc2n(n1)CCO2 40790,CCC(CCC(=O)NCC(C)(C)OCC(=O)NCC(F)(F)C(F)F)OC 40791,C(=O)(C(C)(F)C(C)(C)F)NCCCC1(NC(CCc2cccc(OC)c2)=O)CC1 40792,C1(NC(C(CSC)C)=O)CC2CCC1N2C(=O)Cn1nc(O)ccc1=O 40793,c1(C(=O)NCC(COC)(C)OC)cc2c(cc1O)CCCC2 40794,C(CC1CC1)(C(=O)NCc1ncsn1)NC(C(OCC)OCC)=O 40795,N1(C(Cc2ccc(CC)cc2)=O)CCC(C(C)C)CC1CNC(=O)C(CC)OC 40796,C1(NC(c2ccc(-c3cccc(F)c3)o2)=O)CC(O)CN(C(=O)CSC(F)F)C1 40797,C1(CNC(c2cc(C(C)C)n(C)n2)=O)C2CCCC1N(C(=O)C(C)S(N)(=O)=O)C2 40798,CC1=C(C)CC(C(=O)NC2CCC2C(N2CCCC2C2CCOC2)=O)CC1 40799,c1(CC(=O)N(C2CCN(C(C3(C)CCCC3C)=O)C2)CC)ccccc1O 40800,C1(NC(c2ccc(OC)nc2C)=O)CCN(C(=O)CC(C)N(C)C)CC1(C)C 40801,C=CC(C)(CCOC)C(=O)NC1CCC(C)N(CC(=O)NC2CCCCC2C)C1 40802,C1(C(N2CC(C)N(C(c3nnc(Cl)cc3N)=O)CC2)=O)COc2ccccc2O1 40803,CC1(C(=O)NCC2CC2NC(c2ncoc2C2CC2)=O)CC2(CCC2)C1 40804,C1(C(N(C)CC2(CNC(c3cnns3)=O)CC2)=O)C2Cc3c(Cl)cccc3C12 40805,c1(N2C(CO)CC(C(=O)O)CC2)nc2ccc(CO)cc2s1 40806,C1(CNC(CCOCCCNC(c2cc(C)sn2)=O)=O)CC2(C1)CC(O)C2 40807,c1(C(N2CCC(N(C(C(C(C)C)F)=O)C)C2)=O)cccn2nccc12 40808,c1(C(C)(C)C)ccc(NC(=O)CC2COCCN2Cc2ccnc(F)c2)cc1 40809,c1(C(N2CCCN(C(C3CCC(C(N)=O)O3)=O)CC2)=O)cccc2c1CCO2 40810,N1(C(C2C(NC(=O)COc3ccc(F)cc3)CCC2)=O)CCN2CCC1CC2 40811,C(=O)(C(C)(O)C(C)C)NCC#CCNC(c1c(C)[nH]nc1C(F)(F)F)=O 40812,N1(C(C(CCC#C)NC(=O)Cc2ccn(CC)n2)=O)Cc2cncnc2C1 40813,C1(C(N2CC(CNC(C(C)N(C)Cc3ccccc3)=O)C2)=O)CCS1(=O)=O 40814,C12(CNC(c3cc(OCC)ncc3)=O)CCC(CC1)N2C(C1(F)C2CCCCC12)=O 40815,C1(C2CCC(=O)NC2)(C(=O)NC(C2CCCN2C(=O)C2=CCOCC2)C)CCC1 40816,C1(N(C(c2cc(C)sc2)=O)C)CN(C(c2n[nH]c(C)c2Cl)=O)CC1F 40817,C1(CC)(NC(C2CC2F)=O)CCN(C(c2cc(Cc3ccccc3)[nH]n2)=O)CC1 40818,c1(C(N2CC(CC=C)(NC(C3CC3F)=O)C2)=O)ccc2[nH]c(=N)[nH]c2c1 40819,Cc1ncc(C(=O)NC(C(=O)N(CCC#N)C)c2ncco2)s1 40820,C1(C(N2CC=CC(NC(C3CCC(C)(CC)O3)=O)C2)=O)CCC(F)(F)C1O 40821,c1(C(N(C(CNC(CC2(C(=O)OC)CC2)=O)C2CC2)C)=O)nc(C)ncc1Cl 40822,CC#CCCC(=O)N1CCC(N2CCN(C(c3cnn(C)c3N)=O)CC2)CC1 40823,N1(C(C(C)C2(O)CCC2)=O)CCC2CCC(C1)N2C(c1cc(Br)cs1)=O 40824,c1(C(=O)NCC23N(C(CC45CC(C)(OC4)C5)=O)CC(C2)C3)cc(O)cc(=O)o1 40825,C1(C)(C(=O)NCC(CC=C)NC(=O)COc2cc(C)on2)CCCCNC1=O 40826,C(C)(N=c1[nH]c(=N)[nH]c(=NCc2ncnn2C(C)C)[nH]1)c1nnc(C)o1 40827,N1(C(c2cnn(C3CC3C(=O)OC)c2)C(=O)NCCCSC)CC2CCC1C(O)C2 40828,CC(CC(F)(F)F)C(=O)N1CC(CC(=O)NCCP(C)(C)=O)CC1(C)C 40829,c1(C(=O)NCC(CNC(CCOCCC)=O)OC)c(Br)ccc2n[nH]cc12 40830,C(=O)(CC(C)NC(N)=O)NCC1CC(NC(C2C(COC)(CC)C2)=O)C1 40831,C1(C(N2CCC(CCNC(CSc3c(C)noc3C)=O)C2)=O)CC(C(C)C)=NO1 40832,O=C(C1=C2CCCN=C2NN1)Nc1ccc2c(c1)CN(C1CCC(=O)NC1=O)C2=O 40833,C1(NC(c2cc(C)sn2)=O)CCC2(CC1)CCN(C(=O)CCc1cnn[nH]1)CC2 40834,C(=O)(CCC(=O)NC1CCC(CNC(c2ccn(C(C)C)n2)=O)C1)NC 40835,C1(C(=O)NC2CN(C(=O)Cn3ccc(C(F)F)n3)C2)(NC(CC)=O)CCCC1 40836,c1(NC)snc(C)c1C(N1CC(C(C)(C)O)(CNC(C2(C)CCCS2)=O)C1)=O 40837,C1(NC(Cc2cccc(C(C)C)c2)=O)CN(C(=O)C(C)n2cncn2)CC1(C)C 40838,CC1CN(C(C2CCN(C)CC2)=O)CC(C)N1C(c1cnn2ccncc12)=O 40839,C1(NC2CCCC(C(N(C(C)C)C(C3CCC(=O)O3)=O)=O)C2)CCCCCC1C 40840,c1(C(C(=O)NCC=C)N(C)CCc2cccs2)cc2n(n1)CC(C)(C)CO2 40841,C1(CNC(c2n(C3CC(F)(F)C3)nnn2)CCCCl)C(F)(F)C12CC2 40842,C1(CN=c2nc(CC)[nH]s2)CC(C)(C)CCC1NC(c1cc(C(C)C)nn1C)=O 40843,C1(Nc2nc(C)cc(C)n2)CCC2CN(C(=O)CC3CCCOCC3)CC2C1 40844,c1(C(=O)NCCC(C)NC(c2cc(C)nnc2O)=O)c2c(nn1C)CCC2 40845,C=C(F)C1(CC(=O)NCC=CCC(=O)NCC2CC(CC)=NO2)CCC1 40846,CC1(C)COCC(NC(=O)C(C2(C)CC2)NC(=O)Cc2cnns2)C1 40847,C1(CCC)(OC)CCN(C(=O)C(CO)NC(C2CCC(=O)N2)=O)CC1 40848,c1(C(c2n(CC)nnn2)NC2CN(c3nncs3)C2)cc(C)nnc1C 40849,C1(N(C(c2ccc(NC(=O)NC)cc2)=O)C)CCCN(C(=O)C(F)C(C)C)CC1 40850,N1(C(C(CC=CCC)C)=O)CC2CC(NC(=O)C3=C(C)CCC3)C1C2 40851,C1(C(=O)NCC(CNC(CCN2CCN(CC)CC2)=O)CO)CCC2CC2CC1 40852,c1(C(=O)NCC(CC)NC(c2cccnc2NC(C)C)=O)c(SC)cccc1F 40853,C#Cc1cn(C)nc1C(=O)NCC1CC(NC(=O)C2=COCCO2)CC1O 40854,Cc1nc(CN=C(NC(C)C)NC2CCCN(S(C)(=O)=O)C2)c(C)o1 40855,CC(C)C(CCN(C(=O)CC1(CO)CCCCC1)C)NC(=O)CC1CCOC1C 40856,N1(C(C(CCC)OCC)=O)CC(CNC(c2cn(C)nc2O)=O)OC2(CCC2)C1 40857,CC(C)(C)C1=CCN(C(=O)COC2CCN(C(c3ccc(C(N)=O)[nH]3)=O)C2)CC1 40858,c1(C(=O)NC2CC(NC(=O)C(F)(F)C3CC3)C(O)C2)n[nH]c2c1CCCC2 40859,N1(C(C(C(C)C)O)=O)CCN(C(=O)CCCCCC#N)CC(CO)C1 40860,C1(NC(C(CNC(C2(COC)CC(=O)C2)=O)C)=O)C(O)C2CCOC12 40861,C(=O)(C1=COCCO1)N1C(CNC(C2OCCO2)=O)CCC1 40862,c1(OC)ccc(C(N2CCC(N(C)C(c3cc(F)ccc3N)=O)C2)=O)c(F)c1Cl 40863,c1(CC)c(C(=O)NC(C)C=CC(=O)NCC(C)OCCO)ccn1C 40864,C1(CCNC(CNC(C(CC)C)=O)=O)CCN(C(c2cc(F)c[nH]2)=O)CC1 40865,c1(CCNC(C=C(C)CNC(=O)C(C)CN(C)C)=O)ccc(C)s1 40866,N1(C(C2CN(C(C)=O)C2)=O)CCCC2(NC(C3COCCN3C)=O)CCCC12 40867,c1(C(=O)OC)cc(F)c(F)cc1NC(C1CC(O)CCN1C(c1nc[nH]n1)=O)=O 40868,C(C)(C)(CN=c1nc(N2CCN(CC(C)F)CC2)c2c(ncn2C)[nH]1)OC 40869,CC(CC1CCCCO1)C(=O)NNC(=O)c1cnn(-c2ccccc2)n1 40870,c1(CCCC(=O)N)ccc(C#N)cc1.C(=O)(C(C)=CC(C)(C)C)N(CCC#N)C 40871,C(=O)(CCCC(C)(C)C#N)NCC1CCCN(C(c2c(Cl)ccc(OC)n2)=O)C1 40872,N1(C(c2cc(N)c(Cl)cc2)=O)C2CCC1CN(C(c1cn(C3CCC3)nn1)=O)C2 40873,n1(CCC(=O)NCC(C)NC(C2CCCCO2)=O)c(=O)oc2ccccc12 40874,N1(C(C2CC(C)=C(C)CC2)=O)CC2CN(C(C3(CCF)CC3)=O)CC2(C)C1 40875,c1(CC)ncc(C(=O)NC2(CCCNC(c3ccc(CC)s3)=O)CC2)[nH]1 40876,c1(C(=O)NC(C2(O)CN(C(C3CC34CCC4)=O)C2)C)ccc(Cl)c2c1OCCO2 40877,c1(COC(C(C)OCC)=O)ccc(OCC(F)(F)F)c(Br)c1 40878,N1(C(c2c(C)nc[nH]2)=O)CCSCC1CCNC(C1NC(=O)OC1C)=O 40879,CC1CC(NC(C2CC3(C2)CC(C(N)=O)C3)=O)CCN1C(C1CCCCC1)=O 40880,C1(CNC(=O)C=CC2CC2)CC2COCC2N1C(=O)Cn1ccc([N+](=O)[O-])n1 40881,N1(C(c2csc(Cl)n2)C(=O)NCCC)CCC(C2(C)CC2)CC1 40882,CCCCCCC(C)(c1nnnn1CCC)NC1CCn2cncc2C1 40883,C(CN(C(=O)CC1CSCCS1)C)(CO)(CO)NC(COCC#C)=O 40884,c1(C(N2CCC(NC(C(C)OC)=O)C(F)C2)=O)noc2c1COCC2 40885,C#Cc1cccc(CC(N2CCC3(NC(c4nn(C)cc4C)=O)CC3C2)=O)c1 40886,C1(C)(C(=O)NC(C2CN(C(c3cc(O)ncn3)=O)CCO2)C)COC(=O)N1 40887,C1(NC(c2occ(C)c2C)=O)CCC(C)N(Cc2ccc(F)cc2Cl)C1 40888,C=C(C)C1CCC(C)CC1NC1CC2CC1CC2(OC)OC 40889,N1(C(C(=O)NCC)=O)CCOC2CCN(C(C3CC3(COC)CC)=O)CC12 40890,c1(C(=O)NC(CN(C(=O)COC2CC=CC2)CC)C)cc(C(C)(C)C)no1 40891,n1(C(C)C(=O)N(C)Cc2cncs2)cc(C2CC2CO)nn1 40892,C1(C(=O)NCC2(CC)CCC(=O)N2)CCCCCCN1C(C1CC=CC1)=O 40893,C1(NC(c2cnc(C)nc2O)=O)COC2(C1)CN(C(=O)CCC(C)CN(C)C)C2 40894,c1(CC(=O)NCC(=O)NC(c2nc[nH]n2)CC)ccncc1Br 40895,C(=O)(C1=COCC1)NCCCN(c1ccn(C)n1)CC(c1ccnn1C)C 40896,c1(C(N(C(C)CN(C)C(c2csc(Cl)c2)=O)C)=O)ccc(F)c(Br)c1 40897,N1(C(CC(C)(F)F)=O)CCC(NC(c2cnn[nH]2)=O)C(CO)C1 40898,C(CNC(=O)C(C)N1CC(C)C1)(C(C)C)NC(C1CN(C(=O)NC)C1)=O 40899,N1(C(C2C(C(C)NC(c3cccc(C)n3)=O)C2)=O)C2CCC1CN(C)C2 40900,C1(C(=O)NC2(c3cn(CCCC)nn3)CCC2)CCc2ncc(C)n2C1 40901,CN1CCC(C)(C(=O)NCCN(C(=O)COC2CC(F)(F)C2)C2CC2)C1 40902,C(C(CN=c1cc(NC(c2ccc(Br)cc2)CF)nc[nH]1)OC)OC 40903,C1(C(=O)NC(C)C(CO)NC(=O)C(C)n2ccnc2)CC2COCC(C1)C2(F)F 40904,C1(CNC(Cc2ccn(C(C)C)n2)=O)CC(C)(C)CN1C(C1CC(C)C1)=O 40905,C1(NC(c2ccc(C)s2)=O)CN(C(=O)CC2CC=CCN2C)CC1C 40906,N1(C(C(c2cn(C)nc2)=O)=O)CCCC(CC(=O)NCC(=O)NC2CC2)CC1 40907,Cc1cc(C(=O)NC2CCCC(NC(=O)C3=NOCC3)C2)cc2c1NCCC2 40908,c1(C(N2CC3C(NC(=O)CCC=CBr)(C3)C2)=O)cc([N+](=O)[O-])n[nH]1 40909,c1(C(=O)NC2C(N(C)C(C3CC3(Cl)Cl)=O)CCCC2)n[nH]c2c1CCOC2 40910,c1(NC(=O)NC2CC(CCNC(=O)OC)C2)ccnnc1O 40911,CC1CCOC(C(=O)NCCc2n[nH]cc2C(N2CC=CC2)=O)C1 40912,CCC(C(=O)NC(C1(O)CCN(C(C2CCC3(C2)N=N3)=O)C1)C)C(C)C 40913,N1(C(N2CCN(C(COC)C)CC2)=O)CCCc2cc(C)cc(F)c21 40914,c1(CC(=O)NCCCN(C(CCC2CCN(C)C2)=O)C2CC2)cccc(Cl)c1 40915,C1(c2nnnn2-c2ccccc2)(NC(CCSC)CCO)CCC(C)(C)C1 40916,C(=O)(CCCC(=O)N(CCF)CCNC(=O)COCCOCCO)NC 40917,c1(CCOC)nn(C)cc1C(=O)Nc1onc(OC(C)C)c1Br 40918,C(=O)(C1=NN(C(C)C)C(=O)CC1)NCC1N(C(c2cc(CC)on2)=O)CCCC1 40919,c1(C(C2CC2)NC(c2nc(C)c(C)o2)c2n(CCOCC)nnn2)ccccc1C 40920,C1(NC(CN(C(c2cccc(CC=C)c2)=O)C(C)C)=O)CCC12CCCC2 40921,N1(C(CS(C)(=O)=O)=O)CCCC(O)(CNC(C2OCCC2C(F)(F)F)=O)C1 40922,c1(NC(N2CC(C(C#C)C)C2)=O)cc(C(=O)OCC)cc([N+](=O)[O-])c1 40923,Cc1ccc(C)c(C(=O)NCC2C(C)CCN2C(=O)CNc2ccccn2)c1C 40924,N1(C(c2cnn(C)c2C#N)=O)CCC2(CC1)CC(NC(=O)C(F)C1CCOC1)C2 40925,C1(C(=O)NC(C2CCCN(C(=O)CCC3CC3)C2)C)(NC(C)=O)CCCCC1 40926,C(=O)(C1=CCCSC1)NCC(c1ccc(C)cc1)NC(c1cc(=O)c(C)c[nH]1)=O 40927,Cc1ccc2cc(C(N3CCC(C(C)NC(C4CCCC4F)=O)CC3)=O)cn2c1 40928,c1(C(N2CCCN(C)CC2)C(=O)Nc2ccccc2C#N)cnc2n1CCOC2 40929,C1(C(=O)NCc2ncc[nH]2)(COC)CCCN1C(=O)CC(O)CN(C)C 40930,C(C(CC(F)(F)F)NC(=O)CC(C)CF)NC(c1ccc(C(N(C)CC)=O)cc1)=O 40931,c1(C(N2C(CNC(c3ncn(CC)c3)=O)CCC2)=O)cc2scnc2[nH]1 40932,CN1CCN(C(C2CS(=O)(=O)C2)=O)C(C(=O)NC2CN(C)CC2O)C1 40933,c1(C(=O)NC(CCC)C2CCC2)oc(CNC(C2(Cl)CCCCC2)=O)nc1C 40934,N1(C(C2CC3(CC(=C)C3)C2)=O)CC2(CCN(C(=O)C=Cc3ccc(C)o3)CC2)C1 40935,N1(c2c(CC)c(Cl)ncn2)CCC2(CCN(C(=O)CNCC(=O)N)C2)C1.C(C)=O 40936,C#CC1(C(=O)NC(COC)C(C)C)CN(C(c2cnnn2C=C)=O)C1 40937,N1(C(CN(C)Cc2ccccc2)=O)CCOC(c2cccc(C(F)(F)F)c2)C1 40938,c1(C(=O)NCCNC(=O)CCC2CCC2)cccc(F)c1 40939,N1(C(C(C)=C(CC)C)=O)CC2CC(C1)C2NC(=O)CC1CC(OC)C1 40940,CC1CC2CC(C(=O)NCCC3CCCN(C(=O)C4=COCCO4)C3)(C2)O1 40941,c1(C(C)NCC2(NC(=O)OC(C)(C)C)CCCCC2)ccc(Cl)c(F)c1 40942,N1(C(C2C(C(=O)OC)CC2)=O)CCC(C(=O)NC(c2nc(C)no2)C)C12CC2 40943,C1(NC(C2(C(=O)OC(C)(C)C)CCC2)=O)CCOC(c2ccc(F)cc2)C1 40944,n1(CC(=O)NC2CN(C(CC3(OC)CCCCC3)=O)CC2O)cc(F)ccc1=O 40945,CC1OC2(C(=O)NCCCOCCNC(=O)CC(C)C3CC3)CCC1CC2 40946,N1(C(c2cn(C)c(=O)cc2)=O)CC2CN(C(c3cc(Br)c[nH]3)=O)CC2C1 40947,CCCC(CCC)CC(=O)N1CCN(C(=O)COCCSC)C(CS(C)(=O)=O)C1 40948,C1(C(=O)NCCNC(C(C(C)C)NC(=O)C(C)(C)C)=O)CCC(F)(F)CO1 40949,C(=O)(C(C)(C#N)CC)NCc1c(CNC(c2c(CC)nn(C)c2)=O)cccc1 40950,N1(C(c2cc(C)c(Cl)cn2)=O)CCCC(C2CCN(C(=O)CCCC#N)C2)C1 40951,C(c1cncnc1O)=CC(=O)NCC1(NC(Cc2nn(C)c(Cl)c2)=O)CCOC1 40952,CC(C1CCCCC1)=CC(=O)NCC(C)NC(=O)Cc1cc(C)n(C)n1 40953,NC(=O)CCCCC(=O)NCC1CCCN1C(c1ccc(F)cc1O)=O 40954,CCC(C(=O)NCCC1CCN(C(=O)C(N2CCC(C)CC2)=O)CC1)C(C)O 40955,c1(C(N2CCC(NC(C(C(C)C)OCC)=O)C2)=O)cnc(C)nc1C1CC1 40956,N1(C(CC(C)F)=O)CCC(CNC(=O)CN(S(C)(=O)=O)C)C(F)(F)CC1 40957,N1(C(c2cnc(COCC)s2)C(=O)NCCC)CCCC(C(=O)OCC)(C(F)F)C1 40958,CC(C)(C)CCCCC(=O)NCCC1CCN(C(c2cc(F)c(F)cc2O)=O)C1 40959,C(C)(C)(C(=O)N(CCCNC(C1(C)CCCC1)=O)CC1CCC1)N(C)C 40960,N1(C(COC(CC)C)=O)CCCC(C(=O)N(C)CCC2CCCC2)CC1 40961,CCCC(C)(C)C(=O)N1CC(NC(=O)CSc2nnc(S)s2)CC(C)C1 40962,O=C(C1CNc2ccccc21)N1CCN(Cc2ccc(Cl)cc2)C(=O)C1 40963,C=CCC(CC=C)C(=O)NCCNC(C1N(CCCC)CCC1)=O 40964,CS(=O)(=O)c1coc(C(=O)NCC2CCCCN2C(C2CC3CCC(C2)O3)=O)c1 40965,Cc1c(C(=O)NCCCOCCCNC(C2CCC(O)C2)=O)ncn1C 40966,Cc1nc(Cl)[nH]c(=NC(C)CC(C)NC(=O)CC2CCCC2)c1[N+](=O)[O-] 40967,CCCCC(CNC(=O)C1=CCCC1)NC(=O)CCc1cnc(C2(C)CC2)o1 40968,C1(C(N2CCC(C(CC)CC)C2)=O)C2CC3C(C2NC(=O)C(C)(O)CCOC)C13 40969,N1(C(C(C)=C2CCC2)=O)CCN(C(=O)CC(F)(F)Cl)C(C(C)C)C1 40970,c1(C(N(CC(C)NC(c2n[nH]cc2Br)=O)C)=O)cc2c(cc1O)CCC2 40971,C1(CNC(CC2(CNC(CCCOC)=O)CC2)=O)CCOC(C)(C)C1 40972,c1(C(N2CCC(C)(NC(COCCCOC)=O)CC2)=O)ccc2occc2n1 40973,CN1CC(C(C(n2cc(CN)nn2)=O)=O)C(=O)N1.n1(CC(=O)N)cc(Cl)cn1 40974,c1(NC(C2C3(CCN(Cc4ccn(C)n4)C3)C2)=O)ccc2nc[nH]c2c1 40975,c1(CNC(CC)C(N)CO)cc(C(F)(F)F)ccc1F 40976,c1(C(=O)NCC(CO)NC(c2c(COC)nn[nH]2)=O)cn2c(n1)CCCC2 40977,c1(C(C2CC3CC3C2)NCCOC2(C)CCC2)nnnn1CCC1CC1 40978,c1(CC)ccc2occ(C(N3CCC(C)(CNC(c4cc[nH]c4C)=O)C3)=O)c2c1 40979,c1(C(=O)NC(CNC(C=NOC)=O)CO)cc(Br)c([N+](=O)[O-])[nH]1 40980,C1(NC(C2(N(C)C)CC2)=O)CCCC(N=c2[nH]c(Cl)nc3ncn(C)c23)C1 40981,C(C1c2ccccc2CN1C(c1ncoc1C)=O)NC(CCC(CC)C)=O 40982,c1(C(C)C)ncc(NC(=O)C(C)NC(=O)CC2CC2C2CC2)cn1 40983,CC(C)(C)C(C)(O)C(=O)NC1CC(SCc2cccs2)C12CCC2 40984,N1(C(CSCC(=O)OC)=O)CC(NC(=O)C(C2CCC2)OC)CC2(CCC2)C1 40985,c1(C(N2CCCC(CCNC(CC(=O)N(C)C)=O)C2)=O)cc(Cl)ncc1N 40986,CC1(C)CCC(C(=O)NC2(CNC(C3CCOC3)=O)CCOC2)C1 40987,C1(NC(COCCOC)=O)CC(C)CN(C(=O)C(c2c(OC)cccc2Cl)=O)C1 40988,CCN=C(NCC1CCCC1C(=O)NC(C)(C)C)NC(C1CCOC1)C 40989,C1(CC(=O)NCCCCN(CCCNC(C(CCC)C)=O)C)COC(C)(C)CO1 40990,C(=O)(CC1OCCc2ccccc21)NC1CC(NC(C2(C)CCC(O)CC2)=O)C1 40991,C12(CNC(c3cc(C)[nH]n3)=O)CCC(N=c3nc(C(C)C)[nH]s3)(CO1)C2 40992,C12(C(N3C(CNC(c4c(C)onc4C4CC4)=O)CCC3)=O)CCC(CC1)C(C)O2 40993,C1(CN(C(=O)Cc2ccnn2C2CCC2)CC)CCCN1C(C1CC(C)=NO1)=O 40994,CCC(C)CC(C(=O)NCc1c(C)coc1C)NC(C1CN(C)C(=O)N1)=O 40995,N1(CCOCCN)CCCN(Cc2ccc(NC(c3cscn3)=O)cc2)CC1 40996,C1(F)(CNC(CC2(COC)CC2)=O)CC(NC(=O)C(C)(C)C2CCCCO2)C1 40997,c1(C(N2CC(C(C)NC(Cc3c(C)noc3)=O)OCC2)=O)ccn2nnnc2c1 40998,N1(CS(C)(=O)=O)CCN(C2CCCN(C(=O)CSc3ccccn3)C2)C(=O)C1 40999,c1(C(N2CC3(C(NC(c4ccc(F)s4)=O)CC3)C2)=O)coc2ccccc12 41000,c1(C(N2CCC(C)(CCNC(CN3C(C)CC3)=O)C2)=O)cnc2[nH]cnc2c1 41001,CC(CN(C)C(=O)NC(CCCC(=O)OC(C)(C)C)c1ccccc1)S(C)(=O)=O 41002,c1(C(=O)NCCOCCNC(CC(COC)(C)C)=O)cc(N)c2ncccc2c1 41003,c1(C2CC2SCCC(=O)NCCNC(C(C)(C)F)=O)ccc(F)cc1F 41004,C(C(CC(C)C)NC(=O)C(O)C(F)F)NC(CCCN(C(=O)OC)C)=O 41005,N1(C(CCSC)=O)CCC2C(C1)NC(=O)N2C1CCN(C(=O)CC(C)(C)C)CC1 41006,C=CCCC(C1CC1)NC(=O)C(CNC(=O)C(C)CC1CCCC1)N(C)C 41007,C1(NC(C2C(C)C2)=O)CCOCC1C(=O)NCC(=O)NC1CC1 41008,CC(C)CC(O)C(=O)NCC1OCCC1C(=O)NC1(CO)CC(F)(F)C1 41009,c1(C(=O)NC(C(CO)NC(COc2cccc(OC)c2)=O)C)ccc(C)nc1O 41010,C(=O)(C1=NN(C)C(=O)CC1)N1C(C)CCC(NC(=O)Cc2csc(NC=O)n2)C1 41011,N1(C(c2c(-c3cn(C)nc3)onc2)=O)CC(C2(NC(c3ccncc3N)=O)CC2)C1 41012,CC1CN(C(=O)CSc2n[nH]c(O)n2)CCC1NC(=O)C(C)n1ccnc1 41013,c1(C(N2CCOC(CCNC(C3(CF)CC3)=O)C2)=O)ccc2cnsc2c1 41014,CC(C)C(O)C(F)(F)C(=O)NC1CN(C(c2onc3ccccc23)=O)CC1C 41015,c1(C(=O)OCC2Cc3ccccc3CO2)n[nH]c2c1CCCCC2 41016,CC#CC1CN(C(C2CCN(Cc3cn[nH]c3)CC2)=O)C1 41017,N12CCC(C=C)(CC1)C2=O.c1(CNC(COCCC#C)=O)noc(C)n1 41018,Cc1cc(C)n(CCCNCc2ccccc2-c2ccc(F)cc2)n1 41019,C(c1cc(Cl)c2c(c1)OCO2)=CC(N1CC(NC(C(C)(O)C(F)(F)F)=O)C1)=O 41020,C1(C(N2CCC(CCNC(C(CSC)O)=O)CC2)=O)CCc2ccccc2C1 41021,N1(C(C2(O)CCN(CC3CCOC3)CC2)=O)CCc2cccc(O)c21 41022,CCCC(CNC(=O)CSC(F)F)NC(=O)CCOCC 41023,c1(C(=O)NC2(CF)CCN(C(Cc3c(C)nc(C)s3)=O)C2)cc(C)c(F)cc1F 41024,C1(NC(c2cc(OC)c(F)cc2)=O)CCN(C(C2CC2(Cl)Cl)=O)CCC1CO 41025,Cc1c(C(=O)NCC(C2CCCCN2C(c2cnc[nH]2)=O)(C)C)cnn1C(C)C 41026,N(C1c2ccccc2CC12CCNCC2)C(C1N(C(N)=O)CCC1)=O 41027,N1(C(COC(C)C)=O)CC(NC(=O)CC2(C)CC2)C2CC12 41028,N1(C(CC2CN(C)C2)=O)Cc2ccccc2CC1CNC(C1CC2C=CC1C2)=O 41029,N1(C(Cc2cnc(C)[nH]2)=O)CCOCC(C)(CNC(=O)C(C)NC(=O)C2CC2)C1 41030,CC1(C)C=C(C(=O)N2CCN(C(c3cn(C4CC4)nn3)=O)C(C3CCC3)C2)C1 41031,N1(C(c2ccc(OC)nc2)=O)CC2CC(C1)N2C(=O)CN1CCN(C)C(=O)C1 41032,N1(C(C(CC#C)C2CC2)=O)CCC2CN(C(c3cc4sc(C)cc4s3)=O)CC12 41033,c1(C(N2CC(N(C(CCSC)=O)C)C(F)C2)=O)cc(Cl)cc(Cl)c1[N+](=O)[O-] 41034,CC(C)(CS(N)(=O)=O)C(=O)NCC1CN(C(C2(O)CCC2)=O)CC12CC2 41035,CN1CCC(C(=O)NC2(C)CCN(C(C3CCSCC3)=O)C2)S1(=O)=O 41036,C1(C(=O)NCC2CCC(C(=O)NCc3cnc(CC)s3)O2)CC2CCC1O2 41037,CC(c1cccnc1)=CC(N1CC(NC(c2nccc(C)c2N)=O)C2(CC2)C1)=O 41038,Cc1cc(NC(=O)C(=O)NCC2COCCC2C)cc(C(F)(F)F)c1 41039,CCC(CC(=O)N1CCN(CC2CN(C(=O)CCSC(F)(F)F)C2)CC1)SC 41040,Cc1nc(F)ccc1OC(c1ccc(OCCC(C)C)cc1Cl)=O 41041,c1(CC(=O)NC(c2cn(-c3ccc(C)cn3)nn2)C)ccc2occc2c1 41042,c1(C(=O)NCCN(C(=O)C2=CSCCO2)CC)c[nH]c2c(OC)nccc12 41043,C(=O)(CC(C)CC(C)C)NC(CC=CC)C(=O)NCCc1cccnc1F 41044,c1(C(=O)NC2CC(NC(C(C3CCCCC3)OC)=O)C2)cccc(C(F)(F)F)n1 41045,C#CC#CC(C)(C)NC(C1(F)CN(C(=O)CC2CC3CCC2C3)C1)=O 41046,O=C(C1=Cc2cc(F)ccc2OC1)NCC1CC(NC(c2ccno2)=O)C1 41047,c1(OC)cc(NC(=O)CC2CCCN(C(C3CCC3)=O)C2)ccc1Cl 41048,C12(CNC(c3nccc(C)c3)=O)CCCOC1CCN(C(c1csnn1)=O)C2 41049,c1(C2C(C(=O)OC)C2)cccnc1-c1ccccc1N 41050,CC1CCCC(C)C1NC(=O)CCOCCCNC(c1ccc(CC#N)cc1)=O 41051,c1(CN(c2ccncc2)CC=C)[nH]cnc1C 41052,C=CC(CC)C(=O)NC1(CC(=O)N(C(C)COC)CC)CC1 41053,N1(C(c2c(NCC)scn2)=O)CC2C(CC(=O)NCc3ncoc3C(C)C)C2C1 41054,C(CC(C)C(=O)NCCOCCNC(=O)CC(O)(c1ccccc1)C1CC1)OC 41055,c1(C(=O)NCCCCC(C)NC(=O)C(F)(F)C(F)F)cnc2c[nH]nc2c1 41056,C1(CC(=O)N(C(C)CCNC(=O)C2=COCCC2)C)COc2ccccc2O1 41057,N1(C(C2=C(C#N)CCC2)=O)CCC2(CCC2)C(CNC(c2ccoc2Cl)=O)C1 41058,C1(CNC(c2cc(C(C)=O)sc2)=O)CN(C(c2ccc(O)nn2)=O)CC1C 41059,Cc1nc(C(=O)NC2CN(C(C3CCCN3C=O)=O)CC2C)c2ccccn12 41060,N1(C(CN(CC#C)C(c2cn(C)nc2CC)=O)=O)CCCC(CN(C)C)CC1 41061,N1(C(C2(CNC(=O)C(O)C3CCCC3)CCCCC2)=O)CCC2(CC1)CC(O)C2 41062,C=Cn1nncc1C(=O)NCCCCCNC(c1c(Br)n[nH]c1C)=O 41063,C(=O)(CC(CC(C)C)NC(c1ncccc1CC)=O)N(C(C=C)C)C 41064,C(C)(CC(=O)N(C1CCN(C(C2(N(C)C)CC2)=O)C1)C)=C(C)C 41065,C(=O)(C(CCN(NC(c1cc(C)oc1CC)=O)CC)C(COC)CCC)OCC 41066,c1(C(=O)NC2C(NC(CCN(CC(F)(F)F)C)=O)CC2)cccc(N)c1 41067,c1(CC(=O)N(CCCCCNC(C2(C#C)CCC2)=O)C)cccc(F)c1F 41068,C12(C(N3CCC(N(C(c4ccc(Cl)cc4)=O)CC)C3)=O)C3C4C1C1C2C3C41CO 41069,N1(C(Cn2cc(C(=O)OC)nn2)=O)CC2CC3CC2C1C3NC(=O)CSC(C)C 41070,Cc1cc(C#N)c[nH]c1=NCC12CC(NC(=O)CCc3cscn3)(C1)C(C)(C)O2 41071,c1(C(N2CC3CC(CNC(CC(CCC)C)=O)C3C2)=O)cc(N)c(Br)c(F)c1 41072,c1(C(=O)NC(C2CN(C(=O)CC3CCC(=O)N3C)C2)C)ccc2nc(O)[nH]c2n1 41073,Cc1[nH]nc2ccc(CN3CC4(C)CN(C(=O)CNS(C)(=O)=O)CC4(C)C3)cc12 41074,S(=O)(=O)(c1cccnc1NC(C)CC=C)NC1(CC=C)CCOC1 41075,C1(COC)(NC(c2nocc2Br)=O)CCN(C(=O)OC(C)(C)C)CC1 41076,C1(C)(CNC(CC)=O)CN(C2CCN(C(c3ccsn3)=O)CC2)C1=O 41077,c1(C(C(=O)NC(C(CO)NC(C(CC)C)=O)C)(C)C)cccc(F)c1 41078,c1(C(N2CCC(N(C(C(C=C)c3ccccc3)=O)CC)C2)=O)nccnc1SC 41079,C1(CC)CN(C(c2cnn(C)c2CC(C)C)=O)CCN1C(=O)CS(=O)(=O)N(C)C 41080,c1(CC)oc(C)cc1C(=O)NCCC(C)N(C(=O)Cc1cc(C)cs1)C 41081,CC(C)CC(O)C(=O)NC1CCCN(C(c2cccc(C3(F)COC3)c2)=O)C1 41082,N1(C(c2ccc(C)cc2O)=O)CCC2CN(C(C3(C)C=CCC3)=O)CC2CC1 41083,C1(N(C(C(C)CC2CC2)=O)C)CCCN(C(=O)Cc2cncc(Br)c2)C1 41084,N1(C(C2C(NC(=O)CC3CSCCO3)COC2)=O)CCC2(CC1)CC(O)C2 41085,c1(NC)ccccc1C(=O)NC(CCC1CC1)C(=O)N1CC2CC2(CO)C1 41086,c1(C(N2CC(N(C)C3CC3)C2)=O)cc(CNC(c2c[nH]c(=N)o2)=O)on1 41087,C1(NC(c2cnn(CCC)c2C)=O)CC2(CCN(C(C3(C(N)=O)CC3)=O)C2)C1 41088,C(=O)(C1=C=CCCCC1)NCC(CNC(C1CCC(=O)NC1)=O)F 41089,c1(C(N2C(CCC=C)CCC2)=O)ccc(CNC(=O)C(C)=C(C)C)nc1 41090,Cc1ccc(OC(C)C(N2CC(NC(=O)C(C)N(C)C)C(C)C2)=O)cc1 41091,N1(c2ncc(C)c(O)n2)CC(CNC(C2(C)CCCCO2)=O)OC(C)(C)C1 41092,c1(OC)nccc(CN(C(=O)CC2(OC)CN(C(C3CCOC3C)=O)C2)C)n1 41093,N1(CC(C#C)C2CCC2)CCCC1(C)C 41094,c1(CNC(C2C(C(C)C)CC2)=O)nnn(C)c1C(N1CCC(OC2CCC2)C1)=O 41095,Cc1cc(F)c(C(N2CCC(NC(c3ncccn3)=O)C(C)C2)=O)cc1F 41096,C1(C#N)(C(=O)NCCCCCCNC(CC2C(C)CCO2)=O)CCCCCC1 41097,CCC(C)CCCCC(=O)N(C)CC1C2CN(C(=O)C=C(C)C(F)F)CC12 41098,c1(C(=O)NC2CC(C)(NC(C3CC3c3cccs3)=O)C2)cccc2nc(O)oc12 41099,C1(C(=O)NC(C#C)(C)C2CCC2)CN(C(=O)CC2CCC(=O)C2)CC12CC2 41100,c1(CCCC)ncc(C(N2CC(C(N)=O)(CNC(=O)CC3CN(C)C3)C2)=O)s1 41101,c1(C(=O)NCC2CCCN(C(c3n(CC#N)ncc3)=O)C2)cc2n(n1)CC(F)C2 41102,c1(C(=O)NC2C(NC(c3cc(C4CCC4)on3)=O)CCC2)ccn2ccsc12 41103,c1(C(N(CCC(=O)N(C)C)C(C)C)=O)cnc(O)c2cncn12 41104,c1(C(N(CC(CNC(C2(SC)CCC2)=O)(C)C)C)=O)ccnnc1C 41105,C=C(CNC(=O)C(CCC1CCC1)NC(C1CC(=O)C1)=O)C(F)(F)F 41106,Cc1ccccc1C1(C(=O)NCC2CC(NC(c3n[nH]cc3Cl)=O)C2)CC1 41107,C1(CNC(COCCCC)=O)CN(C)CCN1C(c1cc(C2CC2)nc(O)c1)=O 41108,N1(C(C2(F)CN(C(c3cc(C)no3)=O)C2)=O)CC2CCC2(C)C1 41109,c1(C(=O)NCC2C3CN(C(CC(=O)NC4CC4)=O)CC32)ccc2scnc2c1 41110,N#Cc1ccc(S(=O)(=O)N2Cc3ccc(O)nc3C2)nc1 41111,c1(C(=O)NCC2(F)CC(CNC(=O)CC3CCC4CC34)C2)cccn2nncc12 41112,Cc1[nH]c(C#N)cc1C(N1CCC(C)(CC(=O)NCCN2CCNC(=O)C2)C1)=O 41113,C1(C(N2CCC(N(C(c3cc(C)co3)=O)CC)C2)=O)C(C)OC(C)C1C 41114,C(C(C(C)C(C)C)NC(=O)C(C)(C)O)NC(c1c(OC(C)C)cccc1)=O 41115,c1(C(N(CC(CN(C(CCOC(C)C)=O)C)O)C)=O)cn(C)cc1C(F)(F)F 41116,c1(Nc2ccccc2)cccc2c1OCCC2.O=C1CCC(F)C(=O)N1 41117,c1(C(=O)NCCC2(C(=O)NCc3c(C)occ3)CCC2)cn(C)c(C)n1 41118,c1(C(=O)NCCCCNC(C(C)(C)OC(C)=O)=O)snc(Cl)c1Cl 41119,C1(NC(c2cncc(SC)c2)=O)CCCN(C(c2ccc(=N)[nH]c2)=O)CC1 41120,C(=O)(N=c1[nH]nc(-c2ccc(OC)cc2)s1)N1C(CC(C(=O)OC)F)CC1 41121,C1(O)(C(NCc2c(COC)ccs2)C2CC2)CCCC1C 41122,O=C(CCCn1cncn1)NCCCc1cn(C2CCCC2O)nn1 41123,C(CC1=CCCCCC1)NC(CC(CC#C)NC(c1ccc(C2CC2)cc1)=O)=O 41124,C1(NC(C2(CC)CC2(F)F)=O)CCN(c2ccc(Sc3ccccc3)cc2)C1=O 41125,Cc1nc(C(=O)NCC2(C)CCC(NC(=O)Cc3cnsc3)CC2)c(C)n1C 41126,C1(O)(CNC(C2CC(CCC)C2)=O)CCCN(C(=O)COC(=O)CO)CC1 41127,CC1(C(=O)NC2CCC(C(=O)NC3CCOCC3F)C2)CC2C=CC1C2 41128,C#CCC(CC#C)C(=O)N1CC(CNC(c2cncc(C)n2)=O)C2CC12 41129,C1(CCOC)(NC(c2c(CCC)[nH]cc2)=O)CCN(C(=O)C(C)(C)CN(C)C)C1 41130,C1(NC(=O)C#CCNC(=O)CC2CCC(=O)C2)CCN2CCCCC12 41131,C(CCC(C)NC(c1cscc1OCC)=O)NC(CN(S(CC)(=O)=O)C)=O 41132,N1(C(C(N2CCC(CC)CC2)=O)=O)CCC2(CC1)CC2C#N 41133,N1(C(COC)=O)CCN(C(=O)CNC(c2cccs2)=O)C(C)CC1C 41134,c1(NC(=O)N(C)C2CC2)cc(Cl)ccc1CNC1OCCC(CSC)C1 41135,c1(C(=O)NCC(C)C(=O)Nc2cncc(CO)c2)c[nH]c2ncccc12 41136,c1(NC(CCC2N(Cc3nc(C)oc3)CCC2)=O)ccc(C(=O)C(F)(F)F)cn1 41137,C1(NC(c2c(C)oc(C(C)C)c2)=O)CCCN(C(c2[nH]nnc2C2CC2)=O)C1C 41138,CC(C)(C)C(CC(=O)NC12CCOC(CNC(=O)CN3CC=CC3)(C1)C2)C(F)F 41139,Cc1cc(C)cc(C=CC(=O)NCC(CNC(C2C(C#N)C2(C)C)=O)CO)c1 41140,C(=O)(C1=NN(CCO)C(=O)CC1)N1CC(C)(C)C(NC(=O)C#CC2CCCO2)C1 41141,c1(C(N2CCC(NC(CN(C)C)=O)C2(C)C)=O)cnc2ncc(Br)cc2c1 41142,N1(C(C2CN(C(C)C)C(=O)C2)=O)CC(NC(=O)CCOC2CC2)CCC1C 41143,CC(C)(C)C(CO)C(=O)NCc1cccc(NC(C2CCn3ncnc3C2)=O)c1 41144,N1(C(c2c(C)ccn2C)=O)CCC2(CC1)CN(C(=O)C1=CCCCC1C)C2 41145,C1(CN2C(=O)NC(c3cc(F)cc(F)c3)C2=O)CC2(C1)CC(F)(F)C2 41146,c1(OC)cc(Cl)ccc1C(N1CC2(NC(=O)C(C3CCCC3)OC)CCC1C2)=O 41147,c1(C(=O)NC2C(NC(=O)C=CC3CC3)C2)cc(C2CCCC2)no1 41148,CCC(C)CC(=O)C(=O)NCC(C(=O)N(C1CCC1)CCN(C)C)C(C)C 41149,C(c1cccc(Cl)c1)=C(C)C(N1CCN(CCNC(C2COC(=O)O2)=O)CC1)=O 41150,N1(C(CCOc2c(C(C)C)cccc2)=O)CC(NC(C2CC2F)=O)CCC1C 41151,c1(C(N2C(CNC(c3cc(C(=O)OC)on3)=O)CC(O)C2)=O)ccc([N+](=O)[O-])[nH]1 41152,C1(n2cc(N(C(c3c(OCC=C)cccc3)=O)CC)nn2)CCCC1S(C)(=O)=O 41153,c1(Cn2ncc(C(N(C)CCN(C)C(C3CC3Cl)=O)=O)c2)ccccc1Cl 41154,CC1CCN(C(C2CCCN(C(N)=O)C2)=O)CC1NC(=O)C(F)n1cccn1 41155,N1(C(C2(COC)CC2)=O)CCC(NC(c2cc(O)no2)=O)C(C)C1 41156,c1(NCCC(N2CC3C(NC(C=CC=CC)=O)(C3)C2)=O)oc(C)nc1C#N 41157,C1(NC(=O)OC(C)(C)C)CCOC(C(=O)NCc2cccn2CCO)C1 41158,N1(C(CC(c2cccc(OC)c2)C)=O)CCCC(N=c2nc[nH]s2)C1 41159,c1(C(=O)NCC2(C)CCN(C(CCCOC)=O)C2)cc2scc(C)c2[nH]1 41160,CC(CC1CCCC1)C(=O)N(C)CC1CCN(C(=O)C=CCn2cncn2)C1 41161,CC(C(=O)NCC1(CNC(C2(c3cccc(Cl)n3)CC2)=O)CC1)C(F)(F)C(F)F 41162,C(=O)(C1CS(=O)(=O)c2ccccc21)NC1C(C)N(C(c2cncn2C)=O)CC1 41163,c1(C(C(=O)N(CC(C)C#N)C)NC(=O)C(F)C2CCC2)cn(C)nn1 41164,C1(C(N2CC(COC)(NC(=O)CC#N)C2)=O)CC2CCC1CC2(F)F 41165,N1(C(CN2N(C)C(=O)C2)=O)CC(O)(C2(CNC(=O)CNc3ccccn3)CC2)C1 41166,C1(C(=O)OCC)CCC2(CN(C(=O)Nc3csc(-c4ccccc4)n3)C2)O1 41167,c1(C(=O)NCC(C)(C)NC(C2C(C)C2C)=O)cc(C(F)(F)F)ccc1N 41168,Cc1ccc2c(c1)CCC2C(=O)NCC(O)CCNC(=O)CCOCC(C)C 41169,C(CC(C)C)(C(=O)N(C1CN(C(c2ccc(CCO)cc2)=O)CC1O)C)OC 41170,c1(C(=O)NC2C(CNC(Cc3ccc(C)s3)=O)CC2)ccc2nccn2c1 41171,C1(COC)(CNC(=O)C(c2ccccc2)C)CCCN1C(=O)CC1CSCCS1 41172,c1(CC)nc(C)n(C)c1C(=O)NCC1CN(C(=O)C=CSc2nc[nH]n2)CCO1 41173,c1(-c2ccc(OCC)c(CN3CC(O)CO3)c2)cc(OC)c(CSC)cc1OC 41174,n1(CC)ncc(CNC(C2(OC)CCN(C(=O)Cc3cncnc3)C2)=O)c1C 41175,C=CC1(C(=O)NC(c2cccc(O)c2)C)CCN(C(c2[nH]ccc(=O)c2C)=O)C1 41176,c1(OC)nc(C)ncc1C(=O)NCC(C)NC(C1CCC2CC2CC1)=O 41177,C1(CNC(=O)C=Cc2ncc[nH]2)C2CCC1CN(C(C1CCCN1C=O)=O)C2 41178,C1(CC)CCCCC1CNC(=O)C(C1CCN(C(c2cncnc2CC)=O)C1)F 41179,N1(C(c2cncc(OC)c2)=O)CC2CCC1C2NC(=O)CS(=O)(=O)N(C)C 41180,Cc1cc(F)cc(NC(C2CC2NC(=O)CCCn2ccnc2)=O)c1Br 41181,C1(NC(c2c(CC)scc2)=O)CN(C(c2ccc(C)cc2)=O)CC1N=[N+]=[N-].C1CC1 41182,C(=O)(CC(C)CC(C)C)N1C(CNC(c2n(C(CC)CC)ncc2)=O)CC1 41183,C1(NC(C23C(C)(C)OCC2C3)=O)CCCC12CN(C(c1coc(C(F)F)n1)=O)C2 41184,c1(N(C)C)ccc(F)c(C(=O)NC2CN(C(=O)CCC3CC3(C)C)C(C)(C)C2)c1 41185,CCCC(CC1CCCC1)C(=O)NC(CNC(=O)CN(C1CCC1)C)C(C)C 41186,Cc1ocnc1C(=O)N(CC(C)N(C)C(C1CC(CF)C1)=O)C 41187,C1(NC(CC(C=C)CC)=O)CCSC12CN(C(=O)C(CC(C)C)N(C)C)C2 41188,C1(C(C(=O)N(CCOC(C)=O)C)C)CCN(C(c2c(C)noc2C(C)C)=O)CC1 41189,CC1C(NC(C2CC3(CC3)CO2)=O)CCCN1C(=O)CCNS(C)(=O)=O 41190,C#Cc1cnc(NC(c2[nH]c(C)c(C(=O)Nc3cc(OC)n[nH]3)c2C)=O)cn1 41191,C1(C(N2CC(OC3CCN(C(C(C4CC4)OC)=O)C3)C2)=O)COC(C)(C)O1 41192,Cn1ncc2nc(Cl)nc(NCC3CCCN(C(=O)CC4C=CCC4)C3)c12 41193,C1(C(N)=O)CCN(C(c2cccnc2CNC(=O)COc2cccnc2)=O)CC1 41194,C(CN=c1[nH]c2c(c(=NC3CCCc4occc43)[nH]1)SCC2)CNC(=O)NC 41195,C(CC(C)(C)C(=O)NCCC(C)CCNC(c1cncc(N(C)C)c1)=O)SC 41196,Cc1[nH]nc(C(=O)NC(C)CNC(c2ccc(-n3cncn3)cn2)=O)c1C 41197,Cc1ncnc(C(=O)NCc2ccc(CNC(=O)C(C)C(C)(C)C)c(F)c2)c1C 41198,c1(CCC(=O)NC23CN(C(C4CCN(C)C4)=O)C(C2)C3)ccc(Cl)cc1Cl 41199,N1(C(=O)Cc2cccs2)CCCC(C2CCCCN2C(=O)CSCC(F)(F)F)C1 41200,N1(C(CC(=O)OC)=O)CCCC(F)(C(N2CCC2(C)C(C)C)=O)C1 41201,N1(C(C2CCCS2)=O)CCOC2(CCC(N=c3[nH]c4ccc(F)cc4s3)CC2)C1 41202,C1(C(=O)NC(C2(O)CCN(C(C(C)(C)OC(C)C)=O)C2)C)CCCCC12CCC2 41203,N1(C(C(c2ccc(Cl)s2)C)=O)CCN(C(=O)COCC(C)(C)C)C(CC2CC2)C1 41204,C1(C(=O)NC(CC)(C)CNC(c2cc([N+](=O)[O-])n[nH]2)=O)CC2CC1CC2(F)F 41205,C1(C(=O)NC(C2N(C(CCC(C)SC)=O)CCC2)(C)C)CCc2ccccc2C1 41206,C(CN=c1[nH]c(=NCCOC(F)F)[nH]c2c1COC2)(c1ccccc1Cl)N(C)C 41207,CC1CNC(=O)CN1C(C1(NC(c2coc(C(N)=O)c2)=O)CC(F)(F)C1)=O 41208,C1(CN(C)C(C2CCC3CC23)=O)CCN(C(=O)CCCc2cncs2)C1 41209,C1(C(=O)NC2CCN(C(CCOC)=O)C2C(C)(C)C)CN(C)C(=O)CCO1 41210,C1(CCC)CN(C(c2ccn(C)n2)=O)CC1NC(c1ccnc(S)c1)=O 41211,CCC(CC)(CCNC(=O)C(F)C(C)C)NC(c1cc(C(=O)OC)co1)=O 41212,Cc1ccnc(O)c1C(=O)NCCCC1CN(C(C2CCNC(=O)C2)=O)CCO1 41213,C1(C(=O)NCC(n2cc(C(c3ccccc3)O)nn2)C)CCCN1CC1CC1 41214,c1(CC)ccc(C(=O)NC23CC(C(=O)NC4(C)CCSC4)(C2)C3)s1 41215,Cc1coc(C)c1C=CC(=O)N(CCNC(C1CC=CCO1)=O)CC1CC1 41216,C1(N(C(C2CC(CC)C2)=O)C)CCCN(C(=O)CCC2CCC(=O)NC2)CC1 41217,Cn1nccc1CN1CSCC1C(=O)NOCC(=O)NC1CCCC1 41218,c1(C(N2CC(NC(C(C)NC(C)=O)=O)(CO)C2)=O)cc(N)c(C)cc1C 41219,CCC(C)C(C(=O)NC1CCCC1CNC(=O)CCCOC)N(C)C 41220,CN1CCC(C(N2CCN(C(=O)C=Cc3cnccn3)C(C3CC3)C2)=O)CC1=O 41221,c1(C(N2C3CN(Cc4c(OC)c(F)ccc4F)CC32)=O)cnc2ccc(Br)cc2c1 41222,Cc1c(NC(C2CC(CCNC(=O)C(c3cccs3)SC)C2)=O)cnn1C 41223,CCCC(C)(C)CC(=O)NCC1CCN(C(C2C3CCCOC23)=O)CC1O 41224,c1(C(=O)NCC2CC(NC(c3c(SCC)nccn3)=O)C2)c(O)nnc(C)c1C 41225,CC1(C)CCC(C(N2CC(C(N)=O)(CNC(=O)CCC3CCCCO3)C2)=O)OC1 41226,c1(C(=O)NCC(N(C(C(CC)(C)O)=O)C)C2CC2)cc(Br)ccc1C1CC1 41227,C(=O)(CC1=CCCCC1)N1C(C(C)NC(=O)C2=CSCS2)CCCC1 41228,c1(C(=O)NC(C2CCCC2)CNC(c2nnc(C)s2)=O)cc(Cl)cc(F)c1F 41229,CC1C(NC(=O)Cc2csc(Cl)c2)CCN1C(=O)CCc1cccs1 41230,c1(CC)ncc(C(N2CCC(CN(c3ncccn3)CC)CC2)=O)c(C)n1 41231,C1(CNC(C2CC2c2cccs2)=O)CC2(CCN(C(=O)C=C(Cl)Cl)CC2)CO1 41232,C(=O)(C(C(C)C)n1cnnn1)NCC(CCNC(C1CCN(C2COC2)C1)=O)OC 41233,N1(C(CN(C2CC2)CC)=O)CCC(C)(NC(c2nc(Cl)oc2C)=O)C1 41234,c1(OCC)ccc(Br)cc1S(=O)(=O)NCc1ccc(C2COC2)cc1 41235,c1(N(C)CC2CCCO2)nnc(-c2ccccc2F)n1CCN1CCCS1(=O)=O 41236,C1(C)(CNC(C(C)NC(=O)C(C)(C)NCC(C)=O)=O)CCN(C(=O)OC)C1.C(C)(C)(C)O 41237,C1(=O)CCCC(=O)NCCC(C)CCN1.C(C)(C)(C)OC(=O)NCCN(C)C 41238,C(=O)(C1=C(Cl)CC1)NC1(C)CN(C(C(C)CC2CC2)=O)C1 41239,C1(C(=O)NCCC(C)(C)NC(=O)C(F)=CC2CC2)CC(C(C)(C)C)=NO1 41240,c1(N2CC(C=C)OCC2)nc(=NCCc2nc(=N)[nH][nH]2)[nH]c2c1CCC2 41241,C1(COC)N(C(c2ccncc2-n2cccn2)=O)CC12CCC2 41242,CC1CC(=O)NC1C(=O)NCCCNC(=O)CCOc1cccc(Cl)c1 41243,c1(C(=O)NCC2CCN(C(C3(C)ON=C(C)C3)=O)CC2O)cc(F)c(F)cc1O 41244,c1(OC)cc(C(=O)NCC2(OC)CN(C(c3cnccc3OC)=O)C2)cc(C)n1 41245,C12(C(=O)NCC(CNC(CCCOC(C)C)=O)F)CC3CC(F)(C1)CC(F)(C3)C2 41246,C(=O)(C1=C(C)OCC1)NC(C(N1C(CC)CCC1)=O)CN(C)C 41247,CC1CCCC(C(=O)NCCNC(N2CCN(CCN3CCCC3=O)CC2)=O)C1 41248,N1(C(C(C2CC2)OC)=O)CC(O)(CNC(C2(CO)CCC2)=O)C1 41249,c1(C(=O)NCC(CC=C)NC(=O)CCC2CCCC2)n[nH]c(CCC)c1[N+](=O)[O-] 41250,Cn1ncc([N+](=O)[O-])c1NC1CC2CCC1N(C(c1cnsc1)=O)C2 41251,C1(C(=O)NCCN(C(=O)CN(c2ccc(Br)cn2)C)CC)COCC(C)(C)O1 41252,C1(C(=O)N)CCCC(F)C1.c1(CCSC)cn(C2COCC2C)nn1 41253,N1(C(c2cc(C)c(F)cc2F)=O)CCC2C(CCN2C(C2COCCO2)=O)C1 41254,C1(NC(C(C)SC)=O)CC(C(=O)NOCC(F)F)C1(C)C 41255,c1(CS(N)(=O)=O)ccc(CNC(N)=O)cc1.c12cncn1C2 41256,N1(C(c2c(C)con2)=O)CC2COCC2(C(=O)NC(C)CC2CCC2)C1 41257,C(=O)(CCCCCS(N)(=O)=O)N1C(C(C)(C)NC(C(C)O)=O)CCC1 41258,c1(C(=O)NC2CC(CNC(C(CC)SC)=O)C2)oc2c(C)ccc(C)c2c1C 41259,C(CC(O)C(=O)Nc1cccc(NC(C2CCC(=O)N2C(C)C)=O)c1)SC 41260,CC(C)CC(C)(CNC(c1nccn1C)=O)NC(C1CCC(=O)N(C2CC2)C1)=O 41261,C1(C(N2C(C)(C(=O)NC3CCCC(COC)C3)CCC2)=O)CC2(CC(=O)C2)C1 41262,c1(OC)ccc(CCC(=O)NC2CCC2NC(=O)COc2ccc(F)cc2)cn1 41263,N1(C(c2nn(CC)c(=O)cc2)=O)CCOC2CCN(C(C3(O)CC3(C)C)=O)CC12 41264,N1(C(C2(C)CCCCC2)=O)CC2(CNC(C3CC(F)(F)C3)=O)CC1CO2 41265,CC1C(=O)CCC1CC(=O)NC1(CCNC(c2coc(C3CC3)n2)=O)CCC1 41266,N1(C(C=CCN(CC(F)(F)F)C)=O)CC(F)(c2ccncc2)C1 41267,C1(CNCC2(CC(=O)OC)CCCC2)CC(F)CN1C(=O)CCc1ncnn1C 41268,C1(C(N2CCCC(C)(NC(c3cc[nH]n3)=O)C2)=O)CC2(C1)CC21CCC1 41269,C1(NC(c2ccc(C(F)(F)F)cn2)=O)CC(CNC(C2CC(O)C2)=O)C(O)C1 41270,c1(C(=O)NCC2CC(OC)CN2C(C2C(C)C2C)=O)c[nH]c2c(C#N)cccc12 41271,c1(-c2nc(C(C)CC(F)F)n(C3CCC(C(F)(F)F)C3)n2)ccc(Cl)cc1O 41272,Cc1cc(=NC(=O)c2cc(CNC(=O)C(C3CCCCC3)O)no2)[nH]n1C 41273,N1(C(C2C(CC)OCCC2)=O)CCN(C(=O)CSc2ccccc2)C(CO)C1 41274,c1(C(N(CC(CN(C(=O)C2=COCCO2)C)O)C)=O)cc(F)ccc1C(F)F 41275,Nc1cc(C(=O)NCC(CO)NC(=O)CC2CC3CC3C2)cc(C(F)(F)F)c1 41276,CCC1=C(C(=O)N2CCCCC2C(C)NC(=O)CCCOC(C)=O)CCCO1 41277,C(C(CC1CC1)C(=O)Nc1cscc1C1CC1)NC(C(C)Cn1ccnc1)=O 41278,CCC(CC)C(C)C(=O)NCCOC1CCN(C(c2csc(C(=O)OC)c2)=O)C1 41279,N1(C(C(C)=C(CC)C)=O)CC2(NC(=O)CCc3cccc(Cl)c3)CC1C2 41280,Cn1ccc2ccc(C(N3CCC4(CCCC4NC(=O)C=C4CCC4)C3)=O)cc12 41281,c1(NC(CC2N(C(c3c(C)ncnc3)=O)CCC2)=O)cnc(Cl)c(Br)c1C 41282,C1(NC(C2CCOCC2)=O)CCC2CN(C(C3(O)CCCC3)=O)CC2C1 41283,N1(C(C(C(C)C)S)=O)CCCC2(C1)CN(c1ccnc(Br)n1)CCO2 41284,C(=O)(C(C)S(=O)(=O)CCC)NC1C2CN(C(c3cn(CC=C)nc3)=O)C(C2)CC1 41285,CC(=O)CCCCCCC(=O)NC1CCCC(NC(=O)C(C)CO)C1 41286,c1(C(=O)NC2(CO)CN(C(c3n(C)cnn3)=O)C2)cccc(CN2CCCC2)c1 41287,CC1(C)C(NC(=O)C2=C(Cl)CCC2)CCN1C(=O)CCC1CCCO1 41288,N=c1[nH]c2c(s1)CN(C(=O)Oc1ccc(Br)c(C(F)(F)F)c1)CC2 41289,c1(-c2cc(C(=O)OCC)n[nH]2)ccc(NC(c2cc(CN(C)C)no2)=O)nc1 41290,C1(NC(C(C)NC(=O)OC)=O)CC=C(C(=O)Nc2cnc(C(C)C)nc2)C1 41291,C1(C(N(CC(CC)NC(C2(CCCC)CC2)=O)C)=O)CCCC2(CCC2)C1 41292,C#Cc1ccccc1C(c1nnnn1CCOC)NCC(C)CC(F)(F)F 41293,CC1CN(C(c2cn(CCNC(C3CNC(=O)N3)=O)cn2)=O)CCO1 41294,C1(CC(C)NCc2cn(C)nc2Br)CCCN(C(=O)OC(C)(C)C)C1 41295,c1(C(N2CCCC(O)(CNC(C3CCCSC3)=O)C2)=O)cc2n(n1)CCOC2 41296,CCC(C)CCC(=O)N1CCCC1C(=O)NCC(c1cnc[nH]1)C 41297,n1(C(C)F)cc(-c2noc(C3CCCN3C(=O)OC(C)(C)C)n2)cn1 41298,C(=O)(C(C)S(=O)(=O)c1ccc(F)cc1)N1CC=C(CCNC(=O)OC(C)C)CC1 41299,c1(C(=O)NCCC2(CNC(=O)CC3CCOC3=O)CC2)cnc2ncnn2c1O 41300,N1(C(C(N2CC(C(C)NC(=O)CCc3nc(=N)[nH][nH]3)C2)=O)C)CCN(C)CC1 41301,C1(C)(C(=O)NCCCCN(C(=O)C(O)C2CC2)C)CCCO1 41302,N1(c2c(OC)c(Cl)ncn2)CCC(C2CC2)(CNC(c2cnoc2C(C)C)=O)C1 41303,C1(OC)CCC2(C(=O)NC(C)(C)C(=O)NC(Cc3ccco3)CO)CC12 41304,N1(C(c2ccc(C)o2)=O)CCN(C(c2c(Cl)cccc2I)=O)C(C#N)C1 41305,N1(C(C2CC(C)(C)O2)=O)CC2(CCC(CNC(c3cccc[n+]3[O-])=O)O2)C1 41306,N1(C(c2c(C)c(N)cnc2)=O)CC2CC(NC(=O)CC3(N(C)C)CCC3)C(C2)C1 41307,c1(NC(C(C2CC2)NC(c2ccc(OC)cc2)=O)=O)cc(C)ccc1C 41308,c1(C(N(C)CC2(O)CN(C(C(C(C)C)OC)=O)C2)=O)cncc2c(O)nccc12 41309,C1(N(C(=O)CSCC2CCCCO2)CC)CCCN(C(=O)C(C)(C)O)CC1 41310,N1(C(CS(N)(=O)=O)=O)CCC(CN2C(=O)CNC2=O)CC12CC2 41311,C1(O)(CN(C(C(CCC)O)=O)C)CCN(C(c2cc(C)c(CC)s2)=O)CC1 41312,c1(C(N(C2CC(NC(c3c[nH]ccc3=N)=O)C2)C)=O)ccc2c(c1)CCO2 41313,N(C(=NCCN1CCCC1)NCC1CCCC1C)Cc1c(OCF)ccc(Cl)c1 41314,c1(C(=O)NCCC2(OC)CN(C(=O)Cc3ncc(Cl)s3)C2)cccc2c1NCC2 41315,C1(CNC(C(=O)N(C)Cc2ccc(CO)cc2)=O)CCC(C)(C)CC1 41316,CC1CCN(C(c2sccc2C2CC2)=O)C(CNC(c2cc(=O)cc(Cl)[nH]2)=O)C1 41317,C(CCC(=O)NCc1nocc1C(=O)NC1CCCSC1)OC(C)=O 41318,c1(C(=O)NCC2N(C(CCCCOC(C)C)=O)CCCC2)nc2c(s1)COCC2 41319,c1(CCC=C)ccc(C(N2CC(COC)(NC(C3CNC(=O)C3)=O)C2)=O)cc1 41320,C(=O)(C1=CC2CCCCCC12)N(CCNC(CS(C(C)(C)C)(=O)=O)=O)C1CC1 41321,c12sc(c(C#N)c1C)[nH]c2=O.C12(CC)CC(NC(=O)CNS(=O)(=O)C3CC3)(C1)C2 41322,Cc1cc(C(=O)NC2CCC(N3CCOCC3)C2)nc(C)c1 41323,N1(C(c2cnn(-c3cccc(C)c3)c2C)=O)CCN(C(C23CC2C3)=O)CC(O)C1 41324,c1(NC(C2C(C(=O)NC(C)C(F)(F)F)C2)=O)ncc(I)nc1Cl 41325,C1(C(=O)NC2CC(NC(CN3CCC(C)CC3)=O)CC2O)SC2C=CC1CC2 41326,N1(c2n(Cc3cc(C)on3)c(CS(N)(=O)=O)nn2)CCOC(C)(C(C)C)C1 41327,C(=O)(N=c1[nH][nH]c2cc(C#N)ccc12)c1n(C)cc(NCc2ccnc(Cl)c2Cl)n1 41328,c1(NC(C2CN(Cc3c(Cl)cccc3Br)CCS2)=O)cc(Br)cnc1Br 41329,C12(NC(C(CSC)C)=O)CC1CN(C(=O)Cc1ccnn1C)C2 41330,N1(C(c2ccc(CC)nc2)=O)CCN(C(=O)C(C)=C(C)C)CC1c1ccnn1C 41331,c1(C(=O)NC2C(CNC(=O)CCC3CCCC(=O)N3)C2)cccc2[nH]nc(O)c12 41332,C(CCC(=O)N1CCCC1CCCNC(C1(C)C=CCC1)=O)N(C(=O)OCC)C 41333,CCC(CCC(=O)N(C1C2CN(C(c3cncn(C)c3=O)=O)CC12)C)NC(C)=O 41334,C(c1cc2ccccc2o1)=CC(N1CC(CNC(C(C=C)(C)C)=O)C(O)C1)=O 41335,C(CCCC(CO)NC(C1(N2CCCC2)CC1)=O)NC(CC(CC)SC)=O 41336,CCCCCC(F)C(=O)N(CCC(C)(C)NC(c1ccsc1)=O)C 41337,C=CCC(C)(C)C(=O)N1CCCOC(CNC(C2CC2C(C)O)=O)C1 41338,C1(C(N(CCC(=O)NC(C)CCN(C)C)CC)=O)CCCSC1 41339,c1(CC)sc(C(=O)NC(C)CCNC(c2nnsc2C)=O)cc1Br 41340,C1(C(=O)NCC(C23CCC(CC2)C3)NC(C(C(C)C)F)=O)CN2CCN1CC2C 41341,CC1(CNC(=O)Cc2ccoc2)CC(NC(=O)Cc2cc(Br)cs2)C1 41342,N1(C(C(C)CC(N)=O)=O)CC2CC(NC(=O)C=Cc3cccs3)CC1C2 41343,C(CSC)(C(=O)NCc1cc(C(=O)NCC(C(C)C)OC)no1)OC 41344,C1(C(N(CCCCNC(c2cc(C)c(O)nn2)=O)C)=O)CCc2ncsc2C1 41345,C(=O)(CS(=O)CCC(F)(F)F)NCC(C1CC1)NC(CCC(N)=O)=O 41346,C=CCCCCC(C(=O)NCc1cccc(Br)c1)N1CCC(O)C(C)(O)C1 41347,O1NC(=O)CC(CC=C)NC(=O)COC1C#C.C1(OC2CCC2)CCOCC1 41348,c1(C(c2ccc(C)o2)NC(C(C)(C2CC2)OC)C)ccc(S(N)(=O)=O)cc1 41349,CC1CN(C(=O)CCOc2ccc(F)cc2)CCCN1C(=O)C(N)=O 41350,c1(C(=O)NC(CC)CNC(c2ccc(O)c(C)c2)=O)cnn2ccc(O)nc12 41351,C1(CC(=O)OCC)NC(=O)N(CC(C)OC(F)F)C1=O 41352,C12(CNC(C3N(C)CCCC3)=O)CCC(CC1)CN2C(c1cc(Cl)cnn1)=O 41353,C(=O)(C1=C(Cl)CCOC1)NC1C(CNC(c2nc(CCOCC)oc2)=O)CCC1 41354,CC(C)C(C(=O)NCC1CN(C(C23CCC(C2)OC3)=O)C1)n1cccc1 41355,C1(CNC(C=C(CCC)C)=O)OCCC1C(N1CC(N2CC(F)C2)C1)=O 41356,C1(C(=O)NCCn2c(C)cnn2)CCN(C(=O)CCc2cccn2C)C1C 41357,N1(C(=O)OC(C)(C)C)CC2CCC1C2C(N1CC(CNC(=O)C(N)=O)C(C)C1)=O 41358,C1(C(=O)NCC(c2cccc(F)c2)C)CC2CC1CN(C(=O)Cn1cnnc1)C2 41359,C=CCCC(C(=O)NCc1ccnc(OC)n1)NC(c1cnc(OC)nc1)=O 41360,C1(CNC(CN(C)C)=O)CN(C(c2ncc3ccccn23)=O)CCC12CCOC2 41361,CC1(C)CC(NC(=O)C(N)=O)CCN(C(c2ccnc(F)c2O)=O)C1 41362,C1(C(=O)NC(CC=C)CNC(C2CC(=O)OC2(C)C)=O)CC2(CCCC2)CO1 41363,C(=O)(C1CCCc2c[nH]nc21)NC(C)CNC(=O)CNC(=O)C(F)(F)F 41364,N1(C(C2N(C(C)=O)CCCC2)=O)CC(Nc2ncnc3ccsc23)CC(C)(C)C1 41365,CC1(CCC(=O)NCC2CCC2NC(=O)CCCc2csc(=N)[nH]2)CCC(=O)N1 41366,CC1(OC(F)F)CCN(C(=O)CN(C2(C)CCCOC2)C(C2CCC2)=O)CC1 41367,c1(C(N2CCCC(n3cc(C(C)OC)nn3)C2)=O)cc(O)nc(Cl)c1 41368,C=CCC(CNC(C1CCSCC1)=O)NC(=O)C(C1CC1)N(C)C 41369,C1(NC(CN(C2CC2)CC)=O)CN(C(c2ccnc(C(F)F)c2)=O)CC1C 41370,C(=O)(N1CC(n2cc(C3(C)CCCCO3)nn2)CO1)c1n(CC=C)ccn1 41371,c1(C(=O)NC2CCN(C(c3ccc(COC)o3)=O)C2)cccc(CSC)c1C 41372,N1(CC(=O)N(C2CCC(CNC(=O)CSC3CCCC3O)C2)C)CCC(C)(C)C1 41373,CC1(C)Cc2cccc(S(=O)(=O)NCCn3ccc(O)nc3=O)c2O1 41374,C1(O)(C(C)NC(=O)CCSc2nccn2C)CCN(C(=O)CCN(C)CCO)C1 41375,CN=c1[nH]c(C(=O)NCC2CN(C(=O)CC3CC(SC)C3)CC2C)cs1 41376,c1(C(C(=O)NC(C)C(CO)NC(=O)C=CCN2CCCC2)O)ccccc1F 41377,N1(Cc2c3ccc(OC)cc3ccc2)CCC(N=c2[nH]cnc3cc(I)sc23)C1 41378,c1(CN(C(=O)C=CC(=O)NC2CCCC2)C(C)C2CC2)ccccn1 41379,C(=O)(C1=CC2(CCOC2)C1)N1CC(CC(=O)NC(CC=C)C2CC2)OCC1 41380,c1(C(C)C(N2CC(F)(c3cn(CCn4cccn4)nn3)C2)=O)ncccc1F 41381,C1(CC(=O)NCCN(C(CN(C)CC)=O)C2CC2)COCCN1CC(F)(F)F 41382,c1(CC)cc(Cl)ccc1C(=O)NCC1(CNC(=O)C(C(C)C)NC)CCCC1 41383,C(c1ccc(OC)cc1OC)=CC(=O)NCCNC(CCCOCCOC)=O 41384,C(=O)(C(CC(C)C)N(C)C(c1cc(CO)on1)=O)N1CCC(C(CC)CC)C1 41385,Cc1cc(C(=O)NC2CN(C(=O)CC3CCCN3C)CC2F)c(O)nn1 41386,N1(C(C(C)OCC=C)=O)CC2CC(O)C1C2NC(c1cc(C)sn1)=O 41387,C1(OC)CCC(COCC(=O)NC(CNC(c2csc(C3CC3)n2)=O)CC)CC1 41388,C12(CNC(CCOCC)=O)CCC(C1)N(C(c1ccc(C(F)F)nc1O)=O)C2 41389,N1(C(c2ccc(OC)c(O)c2)=O)CC2OCCN(C(=O)COC(C)C)C2C1 41390,c1(C(=O)NCC2C3CN(C(c4c(C)nn(C)c4C)=O)CC32)ccc2c(c1)CCO2 41391,c1(CCCCCC)ccc(C(N2CC3CC2C3C(=O)Nc2cncnc2)=O)cc1 41392,C1(C)(NC(C2C(NC(CCCNC(C)=O)=O)COC2)=O)C=CCCC1 41393,N1(C(CC(=O)NCC)=O)CCC=C(CNC(=O)C(C)CC2CCC2)C1 41394,N1(C(c2c(C)n[nH]c2)=O)CC2CCCCN2CC1CNC(c1cc(O)ncn1)=O 41395,C1(CC(=O)NCc2nc(C(N3CC(n4cnnn4)C3)=O)co2)COCCOC1 41396,C1(CNC(CN(C(C)=O)C)=O)CCC(C)(C)CN1C(C1CCOC1)=O 41397,C(C)(C(=O)NC1COCCN(C(c2cc(F)ccc2Cl)=O)C1)(C(C)C)OC 41398,N1(C(c2cc(C)ncc2)=O)CCN(C(=O)C(C2CCCCC2)O)C(CC2CC2)C1 41399,c1(N2CC(C(=O)Nc3c(C(=O)OCC)nc[nH]3)C2)ncc2cc(Br)cnc2n1.CCO 41400,c1(C(N2CC(CC(C)NC(=O)C=Cc3cn[nH]c3)C2)=O)c(F)cccc1F 41401,c1(C(N(C(C(=O)OC)(C)C)C)C)ccc(S(C)(=O)=O)cc1 41402,N1(C(C(C)C(C)NC(c2ccc(CO)s2)=O)=O)CC2(C1)CC(C)(C)C2 41403,CC(CCC(=O)NCC(c1cccnc1)O)NC(C1(C)CCC1)=O 41404,N1(C(CN(C(=O)OCC)C)=O)CC(OC)CC(NC(=O)CC2CCC(C)CC2)C1 41405,c1(C(=O)NC2C(NC(C3(C(C)=O)CC3)=O)CCCC2)ccc(F)c(C#N)c1 41406,Cc1cc(NCC2CCCCN2C(c2sccc2Cl)=O)ccc1[N+](=O)[O-] 41407,CC(C(C)C(=O)N1CCCC(NC(C23CCC(CC2)CO3)=O)C1)S(C)(=O)=O 41408,O=C1Nc2ccc(C(N3CCCC3(C)CNC(=O)CC3CC=CC3)=O)cc2CO1 41409,C(CCN=c1[nH]c(N2CCOCC3(CC3)C2)nc2ccccc12)SC 41410,CN1CCN(C(C2CC2CF)=O)CC1NC(=O)CC1CCN(C2CC2)CC1 41411,c1(C(=O)NC2C(NC(c3n(OC)cnc3C)=O)COC2)cnc(O)n(C)c1=O 41412,c1(CCCC)cc(F)c(CSCCC2(N)CC(NC(C)=O)C2)cc1Br 41413,C1(CC=C)(C(=O)NCC2(F)CC(NC(c3coc(C(F)F)n3)=O)C2)CC=CC1 41414,c1(C(N2CC3C(CNC(c4cn(CCCC)nn4)=O)(C3)C2)=O)ncc(F)cc1F 41415,N1(C(c2cnn(C)c2Cl)=O)CC2=C(C1)CN(C(=O)CP(C)(C)=O)C2 41416,C1(NC(c2c(C)nc(C)o2)=O)CCN(C(=O)Cc2cc[nH]n2)C12CCC2 41417,C1(CNC(C2OCCN(CC)C2)=O)CC(C(C)(C)C)CN(C(=O)C(C)(C)SC)C1 41418,C1(NC(COCCCC)=O)CC2CCCC(C1)N2C(C1CC12CCCC2)=O 41419,N1(C(C=CC)=O)CCN(C(c2cc(C)c(CO)cn2)=O)CC(CO)C1 41420,Cc1cc(CC(=O)NC(C)(C)CNC(C2CCCC(C)(C)O2)=O)ccc1O 41421,c1(OC)cc(F)ccc1CC(=O)N(CC(C)NC(c1nccnc1C(N)=O)=O)C 41422,c1(C(N2CCC(NC(C(C)c3ccsn3)=O)C2)=O)c(N)cc(F)cc1Cl 41423,C1(CC(=O)NCCOCCN(C(Cc2cn(CC)nn2)=O)C)CCCCC1F 41424,c1(C(N2CC(CC)C(OC)CC2)=O)ccc2cnn(CCOC)c2c1 41425,C(=O)(C1CC(=O)Nc2ncccc21)NCCCN(C(C1CC(C)(CC)C1)=O)C 41426,N1(C(Cc2c(C)cccn2)=O)CCOC(C)(CNC(C2CCC(F)(F)CC2)=O)C1 41427,N1(C(C(CC)n2nccc2C)=O)CCN(C(=O)C(C(C)(C)C)N(C)C)C2(CC2)C1 41428,c1(OC)cccc(Br)c1C(=O)NC12CC1CN(C(=O)C(=O)NCC(F)F)C2 41429,CC1C(=O)CCC(C(=O)N(C2CC2)Cc2ccc(F)c(Cl)c2)C1(C)C 41430,C=C1CC(CC(=O)NCC(C)(C2CC2)NC(=O)Cc2ccsn2)C1 41431,CC1=CCC(C(=O)NCCCN(C(=O)CN(c2ccccc2)C)C2CC2)CC1 41432,C#CCCC(C(=O)N(CC(O)CCC=C)C)NC(c1sccc1CO)=O 41433,c1(C(=O)NC2C3CC(NC(C(=O)NCC)=O)CC32)ccc2c(c1)C(=O)CCN2 41434,c1(-n2cc(CN3CCC(OCC(C)C)C3)nn2)ccccc1I 41435,CCC(C)C(O)C(=O)N1CCCC1C1CCN(C(c2c[nH]c(=NC)s2)=O)CC1 41436,c1(CNC(=O)NC(C)CC#N)ccccc1OCc1cccnc1 41437,c1(C(N2CCC(CNC(C(C)SCC)=O)C2)=O)[nH]c2c(c1C)C(=O)CC(C)(C)C2 41438,CC(C)CC(C(=O)NCc1ccc(C(=O)NCC(=O)N(C)C)cc1)C(N)=O 41439,CCCC(C(=O)NCC1(NC(=O)C(C)NC(N)=O)CCCC1)OCC 41440,Cc1c(Cl)ccc(C(N2CCOCC2CC2CCCN2C)=O)c1N 41441,N1(C(c2cccc(NC)n2)=O)CCC2CCN(C(=O)Cc3sccc3Cl)C2C1 41442,CCCC(CO)NC(=O)NCC(n1ccnn1)C 41443,C(=O)(CC(F)(F)C(F)F)NC(CCN(C(C(CC#C)O)=O)C)(C)C 41444,C123CC(C1)(C2)OC3=O.C1(O)(C(C)NC(=O)C=CC(=O)N(C)C)CCOC1 41445,C1(NC(CCSCCC)=O)CC2CC1CN(C(c1ccnn(C)c1=O)=O)C2 41446,C1(CNC(c2c(C)n[nH]c2C)C)CC2(CCC2)C(=O)O1 41447,c1(C(=O)NC2CN(C(C3(O)C(C)(C)C3)=O)CC(F)C2)cc(F)c(F)cc1F 41448,C1(NC(=O)COc2cccc(C(F)(F)F)c2)CC2CCC1N(C(C1CC(O)C1)=O)C2 41449,C12(C(N3CC(=CC)C3)=O)CC(CN(C(C3CCC(C)=C(C)C3)=O)C1)C2 41450,CC(C)CC(C(=O)NC(c1cccnc1O)C)NC(C1CC(=O)NC(=O)C1)=O 41451,C(=O)(CC(O)CNC(=O)C(CC)OC)N1CC(N(CCC=C)CC)C1 41452,CC1CC(C(N2CCC(C(=O)N(CCC(=O)N(C)C)C)CC2)=O)CCO1 41453,C1(C(N(CCCNC(C(CC=CC)C)=O)Cc2cccnc2)=O)CCC(C)=C(C)C1 41454,C12(CC(N3C(C)CC(NC(c4c(C)nn(C5CC5)c4)=O)C3)=O)CCC(CC1)CC2 41455,N1(C(C(C)=CC)=O)CCN(C(C2CC3CCC2O3)=O)C(c2ccc(F)c(F)c2)C1 41456,C=C=CC(C)C(=O)NC1CC1CNC(=O)Cc1cc(Cl)sc1Cl 41457,C1(NC(CSCC#C)=O)CCC(N(C)C(c2cnc(-c3cnn(C)c3)s2)=O)C1 41458,c1(CN(C(C)C(=O)N(C)CC2(NC(C3CS(=O)C3)=O)CC2)C)ccccc1 41459,S(=O)(=O)(c1ccc(NC2CCN2C2CCCCCC2)c(F)c1)N(C)CCC1CC1 41460,C(=O)(C1=NOC2(CCCN(C(=O)C(O)Cc3cccc(Cl)c3)C2)C1)NCCOC 41461,Cc1cccc(NC(C2OCCC2NC(c2cnsc2C)=O)=O)c1C 41462,C(=O)(C1CCc2ccc(Cl)nc21)NC1(CO)CN(C(C(CCC)C)=O)C1 41463,c1(C(N2CC3C(NC(C4C(C)(C)CO4)=O)C3C2)=O)ccc2c(c1)CCCC2 41464,c1(OC)cc(Br)ccc1C(=O)N(CC(C)NC(c1cc(F)ccc1C)=O)C 41465,CCCCC(CNC(c1c(C2CC2)noc1C)=O)NC(=O)C(C1CC1)OCC 41466,Cc1cc(=NCCCc2nnc3ccccn23)[nH]c(=NCC2CCSC2)[nH]1 41467,c1(OC)cc(CC(=O)NCC2CN(C(C3CC3C(N)=O)=O)CC2C)ccc1C 41468,CCC(CC(=O)NC1CC(CCC(=O)N(C)CCOC2CCCC2)C1)C1CCC1 41469,C#Cc1ccc(F)c(C(=O)NCC2CC(OC)CN2C(c2cnn(C)c2N)=O)c1 41470,CCC(CCOC)C(=O)NC1C=CCN(C(=O)CC(C)(F)F)C1 41471,C1(C(N2CCC(NC(CCc3nc(C)sc3)=O)C2C)=O)CCc2nc[nH]c2C1 41472,c1(CCN(CCCNC(=O)OC(C)(C)C)C(N)=O)ccccc1.C1(=O)C(=O)NN1 41473,N1(C(c2cc(C)c(F)nc2)=O)CCc2ccccc2C1CNC(=O)C1=COCC1 41474,C(=O)(C#CC1(C)CCCO1)N1CC2(CC(CC(=O)NC(C)CCC(C)(C)C)C2)C1 41475,CC1(C)CCN(C(C2CCC(F)C2)=O)CC1CNC(c1cc(C2CC2)on1)=O 41476,c1(C(N(CC(CC)CC)CCC)=O)c(CNC(=O)C(C)OCC(C)C)nnn1C 41477,c1(C(=O)NCC(CC)(C)NC(=O)COCC2CCOC2)ccc(C(F)F)c(Cl)c1 41478,N1(C(C(C)(c2ccccc2)OC)=O)CCC2(CCC(=O)NC2)C1 41479,Cc1ccc(F)c(C(=O)OC(C)(C)C)c1.C1(N2CC2)CC(C)(C)C1CC(C)C 41480,C(=O)(C1OCCc2c(O)cccc21)N1CCOCC(CNC(C=CC=CC)=O)C1 41481,C1(C(C)NC(c2ccc(CO)o2)=O)CCN(C(=O)C(CC)NC2CCCC2)CC1 41482,C#CC1(NC2CCn3nccc3C2)CC2(CCCC2)C1 41483,c1(NC(CCSCCCC)=O)cccc(NC(c2cc(Br)sn2)=O)c1 41484,Cc1ncc2n1CCN(C(C1CCCC1CNC(C1(C3CC3)CC(=O)C1)=O)=O)C2 41485,C(=O)(CC(C)(C)CC(F)F)NC12CCC(NC(CN(CC)CC)=O)(CC1)C2 41486,C1(C(=O)NCC2N(C(c3c(C)nc(C4CCC4)o3)=O)CCC2)CCN(C)S1(=O)=O 41487,N1(C(C2(CC)CCC2)=O)CCCC(C2CC2NC(c2ccccc2O)=O)C1 41488,CN1CC=C(CC(=O)N2CCC(O)(CNC(C3Cc4ccncc4C3)=O)C2)CC1 41489,C12(C(N3CCC(C)CC3)=O)CCC(NC(C3CC=CCC3C)=O)(CC1)C2 41490,N1(C(c2cnn(C(CC)C)c2C2CC2)=O)CCN(C(C2CC23CCC3)=O)CC1C 41491,C(CCCCC(C)C)NC(C1CCCCN1Cc1cnc(C(=O)OCC)s1)=O 41492,Cc1cc(C)c(C(=O)NCC2(C(C)NC(c3cocc3C)=O)CC2)c(O)n1 41493,C1(NC(CC)=O)CC2CCC(C1C)N2C(c1cnn(C)c1C(F)F)=O 41494,C1(NC(c2cc(CNC(CC3C(C)(C)C3)=O)on2)=O)CCC(C#N)CC1 41495,Cc1ccc(F)c(CC(N2CC(CNC(c3nnsc3C)=O)C3(CC3)C2)=O)c1 41496,N1(C(=O)OC(C)(C)C)CCC(n2cc(CCNC(C(N)=O)c3ccc[nH]3)nn2)C1 41497,C1(CNC(=NC)NCCCCOC)CC2(CCOCC2)O1 41498,CC(N=[N+]=[N-])C(=O)NC(CNC(=O)CC1COCCOC1)C1CC1 41499,CCCCCCC(CC)(CC)C(=O)NC1CC(NC(C2CC3(CCCO3)C2)=O)C1 41500,C1(C(N(CC(C)CNC(c2csc(S)n2)=O)C)=O)COC(C)(C)C1 41501,CCC(CNC(c1ccncc1Br)=O)(CC)NC(=O)COCc1nc[nH]n1 41502,N1(C(C(CC)c2ccccc2)=O)CCCC2(CCCCN2CC2CCOC2C)C1 41503,Cc1ncc(C(=O)NOC(CC(C)C)C(=O)NCCN(C2CCCC2)C)c(=N)[nH]1 41504,C12(CNC(C=CC(=O)N(C)C)=O)CC1CN(C(=O)CCCCc1cnn[nH]1)C2 41505,c1(C(CC)C(N2CCC=C(CNC(C)=O)C2)=O)cccc2cc[nH]c12 41506,C1(CNC(CC2(C=C)CC2)=O)CC(OC)CN1C(C1CCC(=O)N1)=O 41507,c1(NC(c2c(CCC)occ2)=O)cccc(NC(=O)C(C(=O)OC)OC)c1 41508,N1(C(C(CC#C)(C)C)=O)CC2CCC(CNC(=O)Cc3nc(C4CC4)cs3)(C2)C1 41509,C1(NC(CC(CN(C)C)O)=O)CN(C(=O)COCc2ccccn2)CC12CCC2 41510,CC1C(C(=O)N2CCC(C)(C)C2C(=O)NC2CC(C(C)(C)C)C2)=NOC1C 41511,C1(C(=O)NCC(CC)(CC)NC(C2C3COCC23)=O)CC12CCCCCC2 41512,CCC(CC)C(=O)NCC1CC1NC(=O)CCOc1ccccc1COC(C)=O 41513,c1(CNC(C(=O)N(CCCN)CC)=O)cccc(NS(C)(=O)=O)c1 41514,Cc1cc(N)c(C(=O)NCC2(CNC(c3cnc(N(C)C)o3)=O)CC2)cc1C 41515,C(=O)(CC(CCCC(C)C)NC(C1(NC)CC2(C1)CC1(CC(F)(F)C1)C2)=O)OCC 41516,CC1(NC(=O)CCCNC(C2(C(F)(F)F)CC2)=O)CCCOC1 41517,N1(C(C=CC)=O)CCC(NC(c2cccn(C)c2=O)=O)C(c2ccccc2)CC1 41518,c1(CCC)nc(C)c(C(=O)NCC2CC(NC(C3CCOC3(C)C)=O)C2)o1 41519,CCCCC(C)C(=O)N1CCC(C2CCCN2C(c2ccc(Cl)cc2O)=O)C1 41520,N1(CC)CCN(C(C23CC(CO)(CN2C(C2(C)CC(C)=NO2)=O)C3)=O)C(C)C1 41521,N1(C(C=CCC)=O)CC(C)N(C(c2cc(CC(C)C)c[nH]2)=O)CC1C 41522,C1(CC(=O)OC)CN(C(=O)NC2COCCN2CC(F)F)C2(CCC2)CO1 41523,N1(C(CCc2cccc(C)n2)=O)CCC2COC(CC(=O)N(C)CCN(C)C)C2C1 41524,N1(C(COC(CC)C)=O)CCCC1C(=O)NCC(C)CO 41525,N1(C(c2cnc(OC)s2)=O)CCC2(CC1)CC2CNC(c1cccc(F)c1O)=O 41526,N1(C(c2ccc(C(C)=O)s2)=O)CC2CC(NC(c3oncc3C)=O)CC1C2 41527,c1(CC)ccc(C(=O)NC2CCN(C(=O)C#CC3CC3)C23CC3)cc1OC 41528,C(=O)(C(C)(O)Cn1ccccc1=O)NC1C(NC(c2ccc(OC)s2)=O)C1 41529,C=C(Br)CC(C)(C)C(=O)N(C)CCN(C(c1noc(C2CC2)c1C)=O)C(C)C 41530,C1(O)(CNC(=O)C(c2cccc(Cl)c2)O)CCN(C(c2cc(F)cs2)=O)CC1 41531,C1(NC(C(C)NC(CC)(C)C)=O)C=CCN(C(=O)CCC2CC2(F)F)C1 41532,C(=O)(C(C)NC(C1CC(=O)C1)=O)NCCN(CCC)CCC 41533,n1(C2CCC(C(C)C3CC3)C2)cnc2c(N3CCC(S(N)(=O)=O)CC3)ncnc12 41534,Cn1cc(NC(=O)C=CC2CCCCC2)c(C#N)n1 41535,c1(C(=O)NCC2COCCN2C(=O)C(O)C2CC2)nc[nH]c2nccc1-2 41536,C1(CC(=O)OC(c2ccccc2Cl)c2nc(C)on2)COCCN1C 41537,C1(S)CC2CC(=O)C1C2.C12CC(C(=O)O)N(C1)CC2.CO 41538,C1(C(=O)NCc2snnc2C2CC2)CSCCN1C(=O)CCCCC1CC1 41539,CC1CC(NC(=O)COc2ccccc2)CN1C(c1ccsc1Cl)=O 41540,c1(C(=O)NCC(CN(C(c2cnc(C)n2C)=O)C)(C)C)cnc2ccc(F)cn12 41541,c1(NC(c2c(Br)cc(C)s2)c2nnnn2C(C)(C)C)cc(Cl)cc(Cl)c1[N+](=O)[O-] 41542,C(=O)(CCCCC1CC1)NC1(CCCCNC(CCOCC#C)=O)CC1 41543,CC1=CCC(C(=O)NC2CC(C)(NC(=O)CC(C)(C)O)C2)CC1 41544,c1(OCCC(N2CCC(O)(OCC(C)(C)[N+](=O)[O-])C2)=O)c(Br)cncc1Br 41545,c12ccnc(c1)C(=O)NC2.C1(CNC(C2(OC)CCOC2)=O)CCOC(C)C1 41546,C(C)(CN=c1ccnc(NCc2nnc(O)n2C)[nH]1)(C1CC1)OC 41547,Cn1ccc(=NC(=O)C2CC(O)CN2C(c2ccn(C(C)(C)C)n2)=O)[nH]1 41548,C1(C(=O)NC(C(=O)NCC(CSC)(C)O)CCF)C2CCC(C2)C1C 41549,c1(OC)ccc(F)c(F)c1CN1CCN(Cc2cc(C(F)(F)F)nn2C)CC1C 41550,C(=O)(CCCCC(N)=O)NCC(C)NC(c1cnc(OCC(F)F)c(Cl)c1)=O 41551,C#CCCCCCCCC(=O)N1CCC(O)(C(C)NC(c2cc(C)[nH]n2)=O)C1 41552,c1(C(=O)NCC(CO)NC(C2CC23CCC3)=O)nnc2c(F)cccc2c1O 41553,C(=O)(C(C)(O)COC)N(C)CC1N(C(CC(=O)NC)=O)CCC1 41554,CCCCC(O)CCC(=O)NCC(C)(C1CC1)NC(C1CCCCN1N=O)=O 41555,C1(C)(C(=O)NC(C)CCN(C(=O)Cc2nccn2C)C)CC2CCC(C1)S2 41556,Cc1cc(CN(CC(C)(O)C2CCCC2)C=O)cc(F)c1 41557,C(=O)(CC1=CCN(C)CC1)N1C(CNC(C2(C(=O)OCC)CCC2)=O)COCC1 41558,C1(CNC(C(C)OCC(C)C)=O)(CO)CCN(C(c2ccn(C(C)C)n2)=O)C1 41559,c1(NC(N2CCOC(c3cn(CC(F)(F)C(F)F)nn3)C2)=O)ncc(Br)cc1F 41560,C12(CNC(COCCOC)=O)CC(CO1)N(C(c1cnn(C)c1SC)=O)C2 41561,C1(CC(=O)NCC2OCCN(C(c3c(C)cn(C)c3)=O)C2)COCC(C)(C)O1 41562,CCCC(CCC)C(=O)N(CCC(=O)NC1CC=C(C)CC1)C(C)C 41563,N1(C(CNC(C)=O)=O)CC2CS(=O)(=O)CC2(CNC(c2cc(Cl)cs2)=O)C1 41564,C1(NC(COCC)=O)CCCN(C(=O)CC(CC#N)c2ccccc2)CC1 41565,CCC(CC(=O)OC)NC(C1(N(C)C)CCCSC1)=O 41566,C1(COC)(CNC(C2CCCC23CC3)=O)CCN(C(c2cc(C)cc(C)n2)=O)CC1 41567,c1(OC)ccc(-c2csc(CN3CCC(CO)CC3)n2)cc1 41568,c1(SC)ccsc1C(=O)NC(C)(C)CNC(=O)CC1CC(c2ccccc2)C1 41569,c1(OCC(=O)NCCN(C(=O)C(C(C)C)N(C)C)CCC)cccc(F)c1F 41570,C=CC1CCCCN1C(C12CC1CN(C(=O)CC(C)(C)Cc1ccccc1)C2)=O 41571,c1(CNC2(C(=O)NCC)CCCC2)ccc(-n2cccn2)cc1.C12(CC1)C(=O)N2 41572,c1(C(N2CCC(n3cc(CCCC)nn3)C(C)(C)C2)=O)cccc2c1CC(=O)N2 41573,C12(NC(C3CC(F)C3)=O)CCCC1N(C(c1cnc(Cl)s1)=O)CCC2 41574,c1(C(=O)NC2C(NC(Cc3c(C)ccs3)=O)CC2)cnn(C(C)C(C)C)c1C 41575,n1(CCOC)cc(C(=O)NCC2COC(CNC(c3nn[nH]c3Cl)=O)C2)c(C)n1 41576,S(=O)(=O)(c1c(Cl)ccc(C)c1F)NC(C(=O)OCC)(C)Cc1ccccc1F 41577,CC1(F)CCN(C(=O)CC2CCCN(C(=O)Cc3cncnc3)C2)C1 41578,C1(C(=O)NCC(CN(C(=O)CCc2ccccn2)C)O)CC(=O)CCO1 41579,CCC(CC(=O)NCC(CC)(CC)NC(c1ccc(CC(N)=O)cc1)=O)C1CC1 41580,CC1CC(C(=O)N(C)CCNC(C2(CF)CC(F)(F)C2)=O)CCO1 41581,C#CCC(C)C(=O)NCC(C)(C)CN(C)C(c1cc(Br)n[nH]1)=O 41582,C1(CC(=O)NCC2ON=C(C)C2)CCC(NC(C2CS(=O)(=O)C2)=O)CC1 41583,CC(CCCc1cn(C(C)CO)nn1)C(=O)NC1CN(C2CCN(C)C2)C1 41584,CCC(C(=O)NC1CCN(C(c2oc(C)cc2C)=O)CC1O)C(F)(F)F 41585,CC1(C)CCN(CCNC(=O)C(C)(C)C2CCCN2C(=O)C=CCF)C1 41586,c1(C(C)NC(N2CC(C(O)CO)C2)=O)cc2c(s1)CCC(C)(C)C2 41587,c1(C(=O)NCCCC(C)NC(c2cncc(SCC)n2)=O)ccc(N)c(C)c1 41588,Cc1ccc(F)c(N)c1C(=O)NCC1(F)CC(NC(=O)C(=O)NC(C)C)C1 41589,N1(CCC(=O)Nc2c(C)nc(CC)s2)CC(CN)C(C2CC2)C1 41590,c1(CC)nnc2c(C(N3CCC(NC(C4(O)CC4)=O)CC3C)=O)cccn12 41591,C(=O)(C(C)(C)C(C)O)NCCC1(OC)CN(C(=O)Cc2c(Cl)c(CO)nn2C)C1 41592,c1(N(C)C)ncnc(N2CCOC(C3CN(C(=O)CC(F)(F)F)C3)C2)c1[N+](=O)[O-] 41593,C1(CC)(NC(=O)CN2CCOCC2=O)CCCN(C(=O)C(CC)n2ccnc2)C1 41594,N1(c2n(C)c(Cc3ccc(F)c(C#N)n3)nn2)Cc2ccccc2OC2(CCOC2)C1 41595,C(=O)(CCCCC1CC1)NCC(C=C)O.C12(CC1)C(=O)N2 41596,c1(C(=O)NC2C3(C)CN(C(C(=O)N(C)C)=O)C2C3)cn2cccc(F)c2n1 41597,C12(CNC(=O)C=CCN3CCCC3)CCC(NC(=O)CN3CCCC3=O)(CO1)C2 41598,n1(C(C)C)cc(C(=O)NC2CC(O)CN(C(c3cn(C)[nH]c3=N)=O)C2)ccc1=O 41599,N1(C(COC2CCCC(C)C2)=O)CC2CC(C1)C2NC(c1ccnc(O)c1)=O 41600,c1(NCC)ccc(C)cc1C(=O)NCCCNC(c1cccc(C(=O)NC)c1)=O 41601,CCC(C)C(=O)C(=O)NC1(C(=O)N(C(C)CC(C)C)C)CC(CO)C1 41602,N1(C(C2(C)C=CCC2)=O)CCCCCC(NC(=O)C(c2ccc(O)cc2)=O)C1 41603,N1(C(C(C)CBr)=O)CCC2(CCN(C(c3cc(C4CC4)nn3C)=O)C2)C1 41604,c1(CNC(=O)Nc2ccc(=O)n(CCc3ccccc3)c2)c(CO)cccc1F 41605,CC12CC(NC(C3CC4CC4C3)=O)(C1)C1(CCN(C(c3sccc3Cl)=O)CC1)O2 41606,N1(C(c2c(Cl)ccc(OC)c2)=O)CC2CCC1C(CNC(C1CCOCC1)=O)C2 41607,c1(C(=O)NC2(C3N(C(C(CC)O)=O)CCC3)CC2)cc(F)c(Cl)c([N+](=O)[O-])c1 41608,c1(-c2cc(C(=O)NCC(C)N(C(C(C)=C(CC)C)=O)CC)no2)ccc(Cl)cc1 41609,CC1(CNC(C2CCOC(=O)N2)=O)CCCN(C(c2cn(CCO)nn2)=O)C1 41610,c1(CC(N2C(C(N3CCCOCC3)=O)CC(=C)C2)=O)cccc(Cl)c1F 41611,CC1(CNC(c2cccc(Cl)c2)=O)CN(C(c2ncn3c2CCC3)=O)CCO1 41612,C1CCCC(N=c2[nH]c(=NCC3CCSC3)c3ccccc3[nH]2)C1 41613,c1(CC)ccc(C(=O)NCC2(Nc3cc(Cl)nc(C)n3)CCCCCC2)c(F)c1 41614,N1(C(C=C(C)c2cccs2)=O)CCCC1C1CCCN1C(=O)C1=NOCC1 41615,c1(C(C(=O)NCCCSC)N(CCOCC=C)C)csc(Cl)c1 41616,N1(C(C)CNC(=O)CCn2cccc2)CCN(C(=O)CCc2csnn2)CC1 41617,C(c1ccc(C(=O)NC(C)CNC(=O)CC(C)C2CC2)cc1)=CC(=O)OC 41618,C1(C(N(C(c2ccsc2)=O)CC)=O)CCN(C(=O)CCOC)O1.C(C(F)F)O 41619,Cc1[nH]c(C)c(C(=O)NC2CC(C)(NC(c3ccnn3CCF)=O)C2)c1C 41620,CN1CC(NC(c2occc2CNC(C2C3CCCC23)=O)=O)C(F)(F)C1 41621,C12(C(N3CC(C)C(NC(C4(F)CCCCC4)=O)CC3)=O)C3CC(CC13)C2(F)F 41622,N(C(=NCCOc1ccc(Cl)cn1)NCC1CCC(F)CC1)CC(COC)C 41623,N1(C(C2C3CN(C(C(CSC)O)=O)C2C3)=O)CC2C(C1)C2(F)F 41624,C1(CN(C(CC(=O)OC(C)(C)C)=O)C2CC2)CN(C(c2cc[nH]n2)=O)CCO1 41625,c1(C(=O)NC2CCC(CCC(=O)NCCOCC=C)C2)nc(C)ccc1C 41626,C1(NC(=O)COc2cccnc2)CN(C(=O)Cc2ccc(Cl)cc2)CC1F 41627,C1(C(=O)N)(OC)CCN(C(c2cncc(SCC34CC(CO)(CO3)C4)c2)=O)C1 41628,C1(C#N)(C(=O)NCC2(C)N(C(C3CCN(C)C3=O)=O)CCC2)CCOCC1 41629,c1(C(N(C(=O)CN(C)Cc2cccn2C)CCOC)=O)cc(Cl)ccn1 41630,c1(C(N)=O)cc(CC(=O)NCC2(O)CN(C(C3(n4nccn4)CC3)=O)C2)on1 41631,c1(CC)c(C(=O)NCC2CCC(C)N(C(c3cc(C)oc3C)=O)C2)cccc1C 41632,CCCC(C)CC(=O)NCC1CCCN(C(c2cc(CC)ccc2C)=O)C1 41633,CCCC(C)CN=c1cccc(S(=O)(=O)NC(C)Cn2ccnc2CC)[nH]1 41634,c1(OC)ccc(C)c(OC)c1C(=O)N(CC(C)CNC(=O)CCOC)C 41635,C12(C(=O)OC)CCN(N3C(C(F)F)CNCC3CCC3(C)CCCC3)CC1C2 41636,C1(C(N(CC(=O)NCCC2CC=CCC2)CC)=O)C(C(C)=O)C1(C)C 41637,c1(CC)[nH]nc(C(=O)N(CCCN(C)C)CCNC(=O)C(O)CC2CC2)c1Cl 41638,C=CCC(C)C(=O)N1CCC(n2cc(CNC(C3CC(C(=O)OC)C3)=O)nn2)C1 41639,N1(C(C(CC)N(C)C)=O)CCC2(C=C(C(=O)N3CCCN(C)CC3)C2)C1 41640,c1(C(N2C(CNC(c3ccc(Br)nc3Br)=O)COCC2)=O)cc2cccnn2n1 41641,C(=O)(C(CC(C)C)NC1(C(C)C)CC1)N(CC(COC)O)C 41642,C1(O)(CNC(C2(C)C(C)(C)C2)=O)CCCN(C(c2cc(Cl)ccn2)=O)C1 41643,N1(C(COCC#C)=O)CC2CCC1CN2C(C1CCS(=O)(=O)CC1)=O 41644,c1(C(=O)NC2CC(F)(CNC(C3CC(C)OC3)=O)C2)ccc(-n2cncn2)c(N)c1 41645,N1(C(C(CC)=CC)=O)CCCC12CCN(C(C1CCN(C3CC3)C1=O)=O)C2 41646,CN1N=C(CC(=O)N2C3CCCC2CC(NC(=O)C(C)(C)CO)C3)CC1=O 41647,N1(C(Cn2cc(C(C)=O)nn2)=O)CCC(CF)(NC(C2CCC(=O)NC2)=O)C1 41648,N1(C2CC2)CCN(C(c2ccnc(CC)c2)=O)CC1=O 41649,CCCCCCC(F)C(=O)NC1CC2(C1)CC2NC(=O)C.c1(O)c(C)cccc1C 41650,C(CN=C(NCCSc1ccco1)N(C)Cn1ncc(O)nc1=O)c1cnc(C)s1 41651,c1(NC(C(N2CCCC(CC)C2)=O)=O)c(-c2ccc(OC)cc2)c(C)nn1C 41652,c1(NC(C)C(=O)OCC(C)CNCCCC)c([N+](=O)[O-])c(C)nn1CC 41653,CC1(C)CCCC(CC(N2CC(CNC(c3cncc(N)c3)=O)C2)=O)O1 41654,CC1CC(N(C(=O)COC2CCN(C(C3(C)CCCCCC3)=O)C2)C)CC(C)C1 41655,C(CO)(CC(C)(C)C)NC(C(CC=C)NC(c1cc(CO)on1)=O)=O 41656,CC1CN(C(c2c[nH]c(=N)o2)=O)CC1CNC(c1cnn(C)c1C(F)(F)F)=O 41657,c1(C2N(CC)CC2)nc(-c2ccc(OC(C)(C)C)cc2)nn1CCCN(C)C 41658,Cn1c(C(=O)NC2CCN(C(C3(F)CC=CC3)=O)CCC2CO)cc2sccc12 41659,N1(C(C(C)CC2CCC2)=O)CCOCC(C(=O)NC2CN(C)CC2(F)F)C1 41660,C1(NC(c2cnc(OC)nc2)=O)(CNC(=O)CN2CSCC2=O)CCCCC1C 41661,CC(C)CC(O)C(C)C(=O)N1CSCC1C(N1CCCC(C)C1CO)=O 41662,C1(C(N2CCN(CCCNC(=O)CCOCC(F)F)CC2)=O)C2CCCCCC12 41663,N1(C(Cc2nn(C)c(Cl)c2)=O)CCC2CN(C(=O)C(O)CC3CC3)CC12 41664,Cn1ncnc1C(N1CCCC1C(=O)NCc1ccccc1)C(=O)NC1CCC1 41665,CC#CCC(C(=O)NCC(C)C(C)(C)C)NC(C1CN2CCC1C2)=O 41666,N1(C(CCCCC)=O)CC2(C1)SCCC2NC(c1ccccc1OC)=O 41667,c1(SC)nc(Oc2ccc(N3CCCCC3=O)cc2)nc(N)n1 41668,c1(C(=O)NC(c2c(C(N3CC(=CC)C3)=O)con2)C)cc(CC)oc1C 41669,N1(C(COCc2cc(C)no2)=O)CC(NC(c2ccc(=O)oc2)=O)C(O)C1 41670,C1(O)(CNC(=O)CCn2cccc2)CCCN(C(c2nc(Cl)cs2)=O)C1 41671,C1(NC(C=COCC)=O)CS(=O)(=O)CC1NC(c1cc(Br)sn1)=O 41672,C1(NC(CCN(C)CC)=O)CCN(C(=O)CC2CC23CC3)C1C 41673,C(CN=c1nc(CC2CC2)[nH]s1)CCC1CCCN(C(c2cnc(OC)s2)=O)C1 41674,C1(N(C(=O)COc2cn[nH]c2)C)CCCCN(C(=O)C=Cc2cccc(O)c2)C1 41675,c1(C(=O)NC(CC#C)(C)C)cccc(CNC(=O)CN2CCC(C)CC2)n1 41676,N1(C(c2c(CC)ccs2)=O)CCC2CN(C(C3(C)CCCS3(=O)=O)=O)CC12 41677,CCC(C)(CNC(=O)CCc1ccccc1F)C(N)=O 41678,c1(C(=O)NC2CC(C)N(C(c3ccc(Cl)o3)=O)C2)cncc2sccc12 41679,C1(C(=O)NCC2C(CNC(=O)CCCn3cccn3)C2(F)F)CC2C=CC1O2 41680,C(=O)(C(C(F)(F)F)C(F)(F)F)N(C(CN(C(C(C(CC)C)O)=O)C)C)C 41681,C(=O)(CC(C)C(C)(C)CC)NCCCOCCN(C(CCC=CC)=O)C 41682,Cn1c(C(N2C3CN(C(=O)Cc4cccnc4Cl)CC23)=O)cc2ccccc12 41683,Cc1ccc2oc(C(=O)NC3C4CCN(C(C5(C)CCCOCC5)=O)C34)cc2n1 41684,c1(C(=O)NC2CC(C)(NC(c3ccc(C)cc3N)=O)C2)ccn2nncc2c1 41685,c1(CC(=O)NCC(CN(C(C(C)SC)=O)C)C)cncc(C)c1 41686,c1(C(N2CC(C(C)NC(C3CCCCC3C)=O)C2)=O)cn(C)c2ccccc12 41687,C1(F)(CNC(C2N(CCC)CCC2)=O)CCN(C(c2nc(O)c(C)s2)=O)C1 41688,CC(=O)CCCC(=O)NC1C2CN(C(c3cc(C)c(C)s3)=O)CC12 41689,C(=O)(C(F)(F)CCC=C)N(CCCNC(=O)C(C)OC(CCCC(C)C)=O)CC#C 41690,CC(C(=O)NCc1ccc(C(F)(F)F)cn1)N1C(=O)COc2ccccc21 41691,Cc1cccc(NC(=O)C(C)N(C(=O)CCCC2CCCO2)C(C)C)c1 41692,CC(C)(C)CC(O)C(=O)NC(Cc1cc[nH]n1)C(N1CCCCCC1)=O 41693,c1(C(=O)NCC(CN(C(C(C)OC)=O)C)C)cn(-c2ccccc2Cl)nc1C 41694,CCC(CC(=O)N(CCC(C)NC(=O)COC1(C(F)(F)F)COC1)C)OC 41695,c1(CNC(C2N(C(Cc3cn(CC)nn3)=O)CCCC2)=O)n[nH]c2ccccc12 41696,C1(C)(C(N(CCNC(=O)C=C(C)C)CC)=O)CCC(=O)NC1 41697,N1(C(C(C)OCC#C)=O)CC(NC(c2sccc2OCC)=O)C2CCCCC12 41698,C1(CCOC)(NC(=O)C=CC2CCCN2C)CCN(C(=O)C(C)(C)C2CCC2)C1 41699,C(=O)(CC(C)(F)F)N(CC(C)O)CCNC(C1C(C)C1C)=O 41700,C=CCCCC(C(=O)N1CCC(n2ccnn2)C1)NC(c1cn(C)cn1)=O 41701,N1(C(C(c2[nH]c(=N)sc2)(F)F)=O)CCC2(NC(c3ncccc3Cl)=O)CCCC12 41702,c1(NC(C(CC=CC)NC(=O)CCc2nc(=N)[nH][nH]2)=O)cc(C)ccc1CC 41703,c1(CNC(C(C)NC(=O)NC)=O)cccc2c1CN(C(=O)C(C#N)C(C)(C)C)C2 41704,CCC(C)CCNC(=O)OC(C)(C)C.C1(SC)CC(OC)C1 41705,N1(C(C(CC)Cl)=O)CC(NC(C2CCCC2C)=O)C2(COC2)C1 41706,n1(CC(=O)NC2CCCC(NC(Cc3c(C)nc[nH]3)=O)C2)cc2ccccc2n1 41707,C(=O)(C(CC)CC(C)C)NCCCC(C)NC(c1c(CC)c(F)ccc1)=O 41708,C1(C(=O)Nc2ccccc2)CCCN(CC(F)F)C1.C1C(C)CNC(=O)CN1CC 41709,N1(C(c2c(C)c(Br)no2)=O)C2CCC1CN(C(=O)CC1CC3C=CC1C3)C2 41710,Cc1nn(C)c(Cl)c1C(N1CCOCC(C(=O)N(CCC#N)C2CC2)C1)=O 41711,CCC(C(=O)N1CCC(N(CCO)C(c2csc(C(C)=O)c2)=O)C1)C(C)(C)CC 41712,c1(C(=O)NC(CC)CNC(c2ncccc2Cl)=O)cc(Cl)sc1S(N)(=O)=O 41713,c1(C(=O)NC(CCN(C(C(C)NC(CC)(C)C)=O)C)C)nccc2nn[nH]c12 41714,Cc1nc(CNC(C2CCN(c3cc(-n4cncn4)ncn3)CC2)=O)sc1C 41715,CCN=C(NCc1cc(COC)no1)NCc1ccc(-n2ccnn2)cc1 41716,CC(O)(C(=O)NCC1CC(NC(C23CC(CC(F)F)(C2)C3)=O)C1)c1cccs1 41717,C1(NC(Cc2c(OC)cccc2)=O)CCSC12CN(C(C1CCCOC1)=O)C2 41718,c1(C(=O)NCC(C)N(C(=O)CO)C)cc[nH]c1C1CCCC1 41719,CC(C)CC(CNC(=O)CCN1CCCCC1)NC(C1COC(=O)N1C)=O 41720,C12(CNC(c3c(OC)nsc3)=O)CCC1CN(C(C1CC(O)CN1C)=O)C2 41721,CS(=O)(=O)C1CCCN(C(=O)CC2CCN(C(=O)CCc3ccco3)C2)C1 41722,N1(C(COCCCC#C)=O)CCCC(O)(CNC(c2c(Cl)csc2Cl)=O)C1 41723,Cc1c[nH]c2ncnc(N3CCSC(C(=O)Nc4cnc(C(F)(F)F)nc4)C3)c12 41724,c1(NC(C(c2c(C)nccc2)C)=O)ncc2c(n1)COCC2 41725,C(=O)(C(C)(C)C(N)=O)NCC(C)(C)NC(=O)C(C(C)(C)C)N1C(=O)CCC1=O 41726,N1(C(C=C(CC)CC)=O)CCC(O)(CN(C(=O)Cc2cnn(C)c2)C)C1 41727,O=C1CC(CC(=O)NCCC2CCCN2C(c2cc(Cl)ns2)=O)CCCN1 41728,c1(C(=O)NC2CCN(C(C3COCC4(CCC4)O3)=O)C2)cc2cc(F)ccc2s1 41729,CC1(C(=O)NCCc2nn[nH]n2)CCCN1C(c1nc(Cl)cs1)=O 41730,CC1CCCC=C1C(=O)NCC1CC1NC(c1cc2n(n1)CCCC2)=O 41731,C(=O)(CCCC(C)(F)F)NCCC1OCCN(C(c2c(C)csc2)=O)C1 41732,C1(NC(c2nocc2C2CC2)=O)CC2CC(NC(=O)CC3CC=CC3)CC2C1 41733,N1(C(CN(C(C)C)C)=O)CCOC2CN(C(c3ccsc3C(F)(F)F)=O)CC12 41734,C1(CC(=O)NCc2cc(C)on2)COCCN1C(C1CC1C(N)=O)=O 41735,Cc1ncc2n1CC(C(=O)NCCN(C)C(C1CC3(CCCC3)CO1)=O)CC2 41736,N1(C(C(C)OCC=C)=O)CC(C)(C)CC1CNC(=O)C(C)(C)C1CCCCC1 41737,N1(c2c(C)c(C(=O)OC(C)C)ncc2)CCC2(CC1)CC(C)NC2=O 41738,N1(C(CC=CC=C)=O)CC(O)(CN(C)C(C2CC3CCC23)=O)C1 41739,N12CCCC(C1)CNC2=O.N1(CCCc2cn(C)nn2)CCCCCC1 41740,N1(C(C(CC)N(C)C)=O)C2CCC1CN(C(=O)C(C)Oc1ccccn1)C2 41741,CC(C)CCC(C)C(=O)NCC1(CC(=O)OC(C)(C)C)CC1(F)F 41742,C1(CC(=O)Nc2ccc(OCC)cc2)CN(C(=O)CC2(C)N=N2)CCC1C 41743,C1(CNC(CC2(CS(N)(=O)=O)CC2)=O)CCN(C(=O)C=Cc2cccs2)C12CC2 41744,C(=O)(C(C)(CC(C)C)NC(=O)Cc1cc(C(F)(F)F)c(O)nn1)OC 41745,N1(C(C(C)C)C(N)=O)CCC(C2CCCN(C(c3nccc4ccsc34)=O)C2)C1 41746,c1(CCNC(C2C=CCN2C(c2ccnnc2)=O)=O)ccc(F)cc1 41747,c1(C(N2CC3C(CNC(c4cnc(CCC)s4)=O)C3C2)=O)cc2nc[nH]c2cn1 41748,C1(C(=O)OC)OC(c2nc(Cc3ccoc3)no2)CC1C 41749,C1(CC)CN(C(C2COCCOC2)=O)CCN1C(C12CCCC1(C(N)=O)C2)=O 41750,c1(C(=O)NCC(CNC(C(CCCC)N(C)C)=O)F)oc2ccccc2c1CO 41751,c1(CC(=O)NCCC(=C)CNC(=O)C(O)C(C)CC)ccc(Cl)c(OC)c1 41752,C1(C(=O)NC2CC(C)(NC(Cc3ccc(C)nc3)=O)C2)CCCCNC1=O 41753,c1(C(=O)NC2(CNC(C(CC)CC3CCCC3)=O)CCC2)cc2cccnn2n1 41754,N1(C(C2(CC=C)CC2)=O)CCN(C(c2cnc(-c3ccc(Cl)cc3)s2)=O)CC1C 41755,N1(C(CC(C)F)=O)CC2CCOC2(CNC(c2cc(=O)cc(Cl)[nH]2)=O)C1 41756,C1(NC(=O)C2=CCSC2)CC2CN(C(c3c[nH]cc3Br)=O)CC2C1 41757,c1(-c2c(C(CC(N3CCCC3)=O)=O)c[nH]c2)ccc(-c2ccncn2)cc1 41758,CN1CCC(F)(C(=O)NCCCCCCNC(c2cccc(O)n2)=O)CC1 41759,CCC(C)(CNC(C1(F)CCN(C(c2ccc(CO)cn2)=O)C1)=O)C(N)=O 41760,C(=O)(C(C)C(CC)CC)N1CCCC(n2cc(C(C3CCCOC3)OC)nn2)C1 41761,c1(C(C)(C)C(N)=O)ccc(NC(C2CC2c2cncc(Br)c2)=O)cc1 41762,C(=O)(C1=CC(O)C(O)C(O)C1)N1C(C(N2CCC(N(C)C)C2)=O)C=CC1 41763,C(=O)(CC(F)(F)CS(C)(=O)=O)NCC1N(C(c2c(C)nccn2)=O)CCC1 41764,C(CCC(=O)NCc1nocc1C(=O)N(C1CCOC1)CCO)N(C(C)C)C 41765,c1(OC)ccnc(C(C(=O)NC2CCOC2)N(C2CCCCC2C)C)c1C 41766,N1(C(C2N(CC)CCC2)=O)CCC(C(=O)NC(CC2CC2)C(=O)NC)C1(C)C 41767,c1(OC)cc(SC)ccc1C(N1CC(O)(C(C)NC(c2nccnc2C)=O)C1)=O 41768,C1(C(N(C2CCCN(C(c3sc(C)nc3C)=O)C2)CC)=O)CC2(CCC2)CO1 41769,Cc1cccc(CN(C(=O)C(c2cccs2)NC(=O)C(C)n2ccnn2)C)c1 41770,c1(C(N2CC(CC(C)NC(C(C)NS(C)(=O)=O)=O)C2)=O)ccn(CCO)c(=O)c1 41771,c1(C(N2CCN(C(C(C(=O)OC)C)=O)CC2)=O)nc2ccc(F)cn2n1 41772,C1(C(N2CC(N(C(=O)CCSc3nnnn3C)C)C2)=O)CCn2nccc2C1 41773,C1(C(=O)NC(CC2CCC2)CO)CCN1C(=O)C=C1CCC1 41774,C1(CNC(c2nc(COC)sc2)=O)CCCC(CNC(=O)C=CC=C(C)C)C1 41775,C(=O)(CCCC(=O)NC1(C(=O)N(C2CCN(CC)C2)CC)CCC1)OCC 41776,C1(NC(C2(CC#C)CCC2)=O)CCCC(NC(c2cc(C)n(C)c2)=O)C1 41777,Cc1nc2cc(C(=O)NCCCNC(=O)C(C)c3cccs3)ccc2n1C 41778,c1(C(C(=O)NCCCF)N(CC#N)CC)ccc(F)c(F)c1F 41779,C1(CC)CCC(C(=O)NC23CC(C(=O)NCC(F)(F)CO)(C2)C3)CC1 41780,C1(C(=O)NCCCOC=C)CN(Cc2cc(Br)c(Br)s2)CCS1 41781,c1(OCC)ccc([N+](=O)[O-])c(C(=O)NCC2CC2NC(=O)C2=C(C)CCCC2)c1 41782,Cc1nn(CC(=O)NCC2CCCC2NC(=O)Cn2nccn2)c(=O)cc1Br 41783,C1(N(C(C(C(C)C)NC(Cc2cn(CC)nc2)=O)=O)C)CCOC(C)(C)C1 41784,C1(C(N2CC3C(CNC(c4c(CC)[nH]cc4)=O)(C3)C2)=O)CC(C2CC2)=NO1 41785,C(C(=O)NC12CC(NC(c3csc(Cl)c3)=O)(C1)C2)(C(C)(C)C)NC(C)=O 41786,c1(C(=O)NCC2C(C)CCN2C(=O)C(F)=CCCF)cnn2c1OCC2 41787,CCC(CC)C(CNC(=NCCOCC)NC(c1csc(Br)c1)C)N(C)C 41788,N1(C(C(CC)C)=O)CCCC(C(N2CCCC2Cc2ccccc2)=O)C1 41789,N1(C(CCc2n(C)ccn2)=O)Cc2n[nH]cc2C1C(=O)NC1CNC(=O)C1 41790,C=CCCCCCC(=O)N(C(C)C(=O)NC1CCCC(CC)C1)C 41791,C1(C(=O)NCCC(C)N(CCC)C)COCCN(C(=O)OC(C)(C)C)C1 41792,N1(C(C=C(C)C2CC2)=O)CC2C(NC(c3ccc(-n4cnnn4)cn3)=O)C2C1 41793,CCCCCC(F)C(=O)NC1CCCCC1C(N1c2ncccc2NCC1)=O 41794,n1(CC)ncc(=NC(=O)C(CC2CC2)CC2CC2)[nH]1 41795,c1(NCC)cccc(C(=O)NC2CCCCC2CNC(C2CCCCN2C)=O)c1 41796,CC1(C)Cc2occc2CN(C(=O)CC(C)(C2CCC2)N(C)C)C1 41797,c1(CNC2CN(C(C3(C(=O)OC)CC3)=O)CCC2(F)F)ccc(S(N)(=O)=O)cc1 41798,C1(CCNC(C(C)(C2CN(C(=O)OC(C)(C)C)C2)OC)=O)CC2(C1)CC21CCC1 41799,c1(CCC(=O)NC(C2(O)CCN(C(CCOC(C)=O)=O)C2)C)c(F)cccc1F 41800,C1(OCCn2cc(COCC)nn2)CCCC(C(=O)OC(C)(C)C)CC1 41801,C(CC(=O)NNC(=O)CN1CC(C(F)(F)F)CCC1=O)CC(C)=O 41802,C(=O)(C(C)N(OC)C(=O)C=CC(C)NC(=O)C(C)NC(=O)C1CC1)OC 41803,N1(C(CCn2c(C)cc(C)n2)=O)CC(C)(C)CC1CNC(c1cc(Cl)sc1Cl)=O 41804,N1(C(C2(CC)CN(C(C(C=CC)O)=O)C2)=O)CCC(O)(COC)C1 41805,c1(C(=O)NCC(C)NC(CC)=O)cc(-c2ccccc2)n[nH]1 41806,C(=O)(CS(=O)(=O)CCC(F)(F)F)N1C(C(C)NC(c2cscn2)=O)CCCC1 41807,Cc1nc(C)c(C(N2CSCC2C(=O)NC(C2CCC2)C)=O)o1 41808,C1(CC(=O)NC2CN(C(c3nn[nH]c3Cl)=O)C2)(NC(C)=O)CCOCC1 41809,Cc1ncncc1C(N1CCC(=CC(=O)Nc2ccc(F)nc2)CC1)=O 41810,C1(CC(=O)NOCC2CCOCC2)CCCN(C(c2cn[nH]c2)=O)C1 41811,C#Cc1ccc(OC)c(C(=O)NCC2(C)CC2C)c1 41812,C1(=O)C(CCNC(c2ccoc2)=O)OC2CC(C2)N1C.CCS 41813,N1(C(C2(NC(C=Cc3ccc(C)o3)=O)CC(F)C2)=O)CC(C)OC2(CCC2)C1 41814,N1(C(C2C(CNC(C=C3CCC(C)CC3)=O)CCO2)=O)CC(C)C(F)(F)C1 41815,CC1(CNC(=O)Cn2cnnn2)CCN(C(c2ncncc2F)=O)CC1 41816,CC1CC(CO)CN(C(=O)C(C)NC(c2ncccc2Cl)=O)C1 41817,C(=O)(C(C)CC(N)=O)NCC(CCNC(C(CCC)NC(N)=O)=O)OC 41818,CCN=c1ccc(C(=O)NC2CCC2NC(c2cccc(F)c2F)=O)c[nH]1 41819,c1(N2CCN(C(CCNC(C)CC(C)(C)O)=O)CC2)ccc2cnccc2c1 41820,CC1CN(C)CC(C(N2CCOCC(C(=O)NC(C)C(O)C(F)F)C2)=O)O1 41821,c12coc(c1)CNC2=O.C(=O)(C(O)CSC)NCC1CN(C(=O)OC)C1 41822,Cc1nn(C)c2ccc(C(=O)NCC3CN(C(=O)Cc4ccco4)CC3O)cc12 41823,c1(C(N(CCCCNC(C(CC)O)=O)C)=O)c(C)sc(C)c1C#N 41824,c1(C(=O)NCCN(C(C(c2cccnc2)OC)=O)C(C)C)cnn2ccccc12 41825,c1(C(N(CCCCNC(c2ccc(C(N)=O)cc2)=O)C)=O)cccc2c1NCC2 41826,N1(C(c2ccc(CCC)cc2)=O)CC(C)(C)OC2(C1)CN(C(C1(O)CCC1)=O)C2 41827,Cc1cncc(CC(=O)NC(C2CCCN2C(C2COCCO2)=O)C)c1 41828,N1(C(C(CC)OC2CCCCC2)=O)CC2(NC(c3ncncc3C)=O)CC1C2 41829,CC(C)CC(CNC(C1Cc2nccn2C1)=O)C(=O)NCCC(C)C(F)F 41830,C(=O)(C(CNC(c1cnsc1)=O)(CC)CC)N(c1ccccc1)CC=C 41831,CCC(C)C(C)CNC(C1CCC(NC(c2cc(C)nn2CC)=O)CC1)=O 41832,C(=O)(C#CC1CC1)NCC#CCNC(c1nc(CS(C)(=O)=O)sc1)=O 41833,C1(NC(CCc2ccn(C)n2)=O)CC12CC(NC(c1[nH]nnc1C(F)F)=O)C2 41834,N1(C(C=C(C)C(C)C)=O)CCC(C)C1CNC(c1cn(CC(F)(F)F)nn1)=O 41835,C1(NC(C2(C3(C)CC3)CC2)=O)CCC2CN(C(c3cccc(=S)n3O)=O)CC12 41836,C1(NC(C(COC)N(C)C)=O)CC(OC)CN(C(=O)CSC(F)(F)F)C1 41837,c1(OC)cccc2c(CC(=O)NCC(O)CCNC(=O)CO)c[nH]c12 41838,c1(CC(=O)NC2(CN(C(=O)C=CC3CC3)C)CC2)cc2cc(c1)CO2.O(C)OC 41839,C1(NC(c2cccc(F)c2F)=O)CN(C(=O)Cc2csc(Cl)c2)CCC1CO 41840,N1(C(c2nnn(C(C)(C)C)n2)=O)CC2(CCC2C(C(=O)C(C)(C)CNC)(O)O)C1 41841,C(=O)(C(F)(F)C(F)F)N1C(C(C)NC(C(c2ccc(C)cc2)(F)F)=O)CCCC1 41842,c1(C(C(C)NC(=O)Cc2cc[nH]n2)NC(=O)C(F)F)ccccc1 41843,c1(C(=O)NCCCC(C)NC(=O)C2=NNC(=O)C2)cc2cc(Cl)cnc2o1 41844,N1(C(c2c[nH]c(C)c(Cl)c2=O)=O)CCC2(CC1)CCN(C(=O)C(=O)NC(C)C)C2 41845,C1(C(N(C2CCN(C(c3nn[nH]n3)=O)CC2)CC(C)C)=O)(CN)CC2C=CC1C2 41846,CC1OC2(CNC(C3CC3F)=O)CC1(NC(c1nccc(F)c1Cl)=O)C2 41847,N1(C(C=COCC)=O)CC2CN(Cc3ccc(NC(C)=O)c(I)c3)CC2C1 41848,N1(C(C(CC)NC(N)=O)=O)CC(CNC(C2CC(F)(F)C2)=O)C2CCCCC12 41849,C1(NC(c2coc(O)n2)=O)CCC2CN(C(=O)Cn3cc(Cl)cn3)CC2C1 41850,CC1=NOC(CONC(C2(NC(c3coc(C(N)=O)c3)=O)CC(O)C2)=O)C1 41851,Cc1csc(C(N2CCCC2CCNC(c2ocnc2C(F)F)=O)=O)c1 41852,c1(C(N2CC3CC2CS3=O)C(=O)NCCCOC)noc2c(Cl)cccc12 41853,C(CN=c1[nH]c(=NCc2cccc(Cl)c2Br)[nH]c2c1COCC2)N(C)C 41854,C(=O)(C(C#N)(CC)CC)N(CCNC(C1CC(C(C)C)=NO1)=O)CC 41855,C1(OC)CC(NC(C2CC(F)(F)C2)=O)CN(C(C2CCN(C3CC3)C2=O)=O)C1 41856,CC1CCCC(C)N(C(C2CC3CCC(C2)N3C(c2ccncc2Cl)=O)=O)C1 41857,C(=O)(C#CC1CCOC1)N1CC(CNC(CCc2cc(C)cc(C)c2)=O)C1 41858,C1(CC(=O)N(CC(F)Cl)C)CC(F)CN1C(=O)C=CC1CCCC1 41859,Cc1ccc2occ(C(=O)N(C)CC3(O)CN(C(C4CC4C)=O)C3)c2c1 41860,Cc1nc(C)c(CC(=O)N(C2CCN(Cc3cn(-c4ccccc4)nn3)C2)C)s1 41861,C(=O)(C(C(C)(C)C)C1CCC1)NCC(C)NC(=O)C(C)S(C)(=O)=O 41862,N1(C(C(c2cnn(C)c2)OC)=O)CCCC(O)(CCNC(=O)CC(F)(F)Cl)C1 41863,O=C(N=c1[nH]oc2cc(Cl)ccc12)C1CCN(Cc2cnc(Cl)c(Cl)c2)CC1O 41864,Cc1c(Cl)ccnc1C(N1CCCCC1CNC(C1(N=[N+]=[N-])CC1)=O)=O 41865,N1(C(c2cc(CC)no2)=O)CCCC(N(C(=O)Cc2ccnc(O)c2)C)C1 41866,C1(N(CCCCC)CCC(=O)NC)CCN(C(=O)C(F)C(C)C)CC1 41867,Cc1cccnc1CC(=O)NCC1(F)CN(C(C2CCCCC2C)=O)C1 41868,C1(NC(Cc2cccc(C(N)=O)c2)=O)CS(=O)(=O)C2CN(C(=O)CC3CC3)CC12 41869,c1(C(=O)NCCC(C)NC(=O)CCC2(C)CC2)cc2ncc(Br)cn2n1 41870,CCC(C)C(O)C(=O)NNC(=O)c1ccc(NC(c2ccccc2)=O)nc1 41871,C(=O)(CCCCC(=O)c1ccccc1)NC(C1OCCN(C(C(C)OC)=O)C1)C 41872,C#CC1CCCCN1C(C1CN(C(=O)CCC(=O)NCCC)CC1CCC)=O 41873,c1(CNC2CC(C(N3CCCC(CO)C3)=O)C2)cc(Br)ccc1Cl 41874,CCCCCCCC(=O)NC(CCCOC)C(=O)NCc1cn(C(C)C)nn1 41875,CCCCC(C)CCC(=O)N1C(C(=O)NCCOC2CC2)CCC1C(C)C 41876,c1(C(C(=O)NCC2(CNC(=O)COCCCF)CCC2)OC)cnn(C)c1 41877,N1(C(C(CC=C)(C)C)=O)CC2CC(NC(=O)CCc3cnc(C)nc3O)CC1C2 41878,C1(C(N(CCN(C(CC(C)F)=O)C(C)C)C)=O)CCC2(CC1)NC(=O)N(C)C2=O 41879,c1(SCC)ccc(CC(=O)NC(CCNC(c2ccsc2SC)=O)C(C)C)cc1 41880,c1(C(N2CCCC(C(CNC(CC=C)=O)(F)F)C2)=O)ccc(F)c(C(F)(F)F)c1 41881,C(c1ccc(Cl)s1)=[SH]CC(N1CCC(C(N2CCC(CC3CC3)CC2)=O)CC1)=O 41882,N1(CC(=O)N(C)Cc2ccnn2-c2cccnc2)CC2CC(O)C(O)CC2C1 41883,N1(C(CC(C)n2ccnc2)=O)CCC(C)(NC(C2CCC=CO2)=O)CC1 41884,CC(F)(F)C(C)(C)C(=O)N1CC(NC(c2cc(Cl)sc2Cl)=O)C(O)C1 41885,c1(C2(C)CC2)ccc(C(N2CC(O)(CNC(C3CC(C)(C)CO3)=O)C2)=O)cc1 41886,N1(C(C(C)Cc2ccc(O)cc2)=O)CCC2(CC1)CN(C(C1(C)CCCO1)=O)C2 41887,C(=O)C(C)C(C)C.CCC(C)(C)OCC(=O)NCCCN(C)C(C)C 41888,N1(C2CCN(C(C(C)=O)C)CC2)CCN(S(N)(=O)=O)CC1 41889,N1(C(CC2(N(C(Cn3nnc(C)n3)=O)C)CC2)=O)CCOC(C)C1 41890,C1(C(N2CC(N3CCCC3)C2)=O)CCCCCCN1C(C1CCCOC1)=O 41891,c1(C(=O)NCC(C)(C2CC2)NC(CCCCOC)=O)ncnc(O)c1Cl 41892,C#CCC(CC(F)F)NC(C1CC12CCN(C(C1(C)CC=CCC1)=O)C2)=O 41893,C1(C(N)=O)CCC(C(=O)NC(CC2CCC2)C(=O)N2CCC(N3CCC3)C2)O1 41894,N1(C(C(CSC)OC)=O)CC(CNC(=O)C=Cc2cccnc2)OC2(CCC2)C1 41895,c1(C(=O)NC(c2nc(C)[nH]n2)C(C)C)nsc2cc(Br)ccc12 41896,C12(NC(=O)CSc3cn[nH]c3)CCC1CN(C(=O)CC1CCNC(=O)C1)C2 41897,Cc1cccc(C(C)C(=O)N2CC(C)C2)c1.C(C(F)(F)F)NC.C1(=O)C=CCN1C 41898,c1(C(N2C(CNC(CCCCOCCC=C)=O)CC2)=O)ccnc(C)c1O 41899,N1(C(COCCC#C)=O)CC2CC(NC(c3nc(C(F)(F)F)oc3C)=O)C1C2 41900,c1(C(N2CCCN(CCNC(C(CC)F)=O)CC2)=O)cccc2c1CCCN2 41901,CC1CN(C(C2CNC(=O)N2)=O)CC1(C)C(=O)NC1CCNC(=O)CC1 41902,Cc1scc(C(=O)NCC(O)CNC(c2csc(CC(F)F)n2)=O)c1C 41903,C1(C(=O)NCCN(C(=O)Cc2csnc2C)CCC)CC12CCC(C)(C)CC2 41904,CC1(NC(C2CC3(CCC3)CO2)=O)CCN(C(=O)COc2ccon2)CC1 41905,N1(C(C(COCC)C)=O)CCC(CNC(=O)Cc2n[nH]c(=N)s2)(COC)CC1 41906,C(=O)(CCCCC(N)=O)NC1CCC(C)(CNC(C2(CF)CC(F)(F)C2)=O)CC1 41907,CCCC(CC(C)C)C(=O)NCCOCCCNC(=O)Cc1cc(C)ccc1C 41908,N1(C(C(CC)=CCCC)=O)CCC2(C=C(C(=O)NC(C)C(=O)N3CCCC3)C2)C1 41909,C#CC1(C(=O)NCC2(C)CCCN(C(C3(O)CCC3)=O)C2)CCOCC1 41910,N1(C(c2cc(F)c(F)c(F)c2)C(=O)NCC2CC2)CC2C3C=CC(C3)C2C1 41911,C1(C(=O)NCC2(C(=O)OCC)CCC2)(NC(=O)CSCC)CC(O)C1 41912,N1(C(C(CC)N(C)C)=O)CC2CN(C(=O)C(C)CSC)CC2C1 41913,Cc1cc(C(N2CCCC(NC(=O)C(C)(C)OC(C)C)CC2)=O)c(F)cc1F 41914,CCC(C)CC(C)C(=O)NCC1(CCNC(=O)CC(C)(C)C#N)CC1 41915,N1(C(C=C(C)C(C)(C)C)=O)CCOC(C)(CNC(c2cc3sccc3s2)=O)C1 41916,C(CCCC(C)(C)C(=O)NNC(=O)C1CCCS1(=O)=O)NC(C(CC#C)O)=O 41917,Cc1cnnc(O)c1C(=O)NCc1nc(C(N2CCCC2CC2CC2)=O)co1 41918,Nc1cc(C(=O)NCC(F)CNC(c2cccc3c2CCC3)=O)c(F)c(O)c1 41919,C1(NC(c2c(Cl)cn(CCC)n2)=O)CCN(CC=C(Cl)Cl)CC1C 41920,c1(C(C)(C)C(=O)NC2CCCC2CNC(=O)Cc2cnco2)ccc(O)cc1 41921,Cc1cc(NC(=O)CC2CC(NC(c3cc(O)ncc3Br)=O)C2)cc(Br)n1 41922,c1(C(C(=O)NC(CNC(c2c(CC)con2)=O)C)(C)C)ccc(F)cc1F 41923,c1(CN2C(C(N3C(C)CCC3CO)=O)CC3CC32)cc(F)c(Cl)c(F)c1 41924,CC(C)CC(O)CNC(C1(C)CCCN1C(=O)C1CC1)=O 41925,C1(NC(COC2(C)CCC2)=O)CCCN(C(c2ccc([N+](=O)[O-])o2)=O)CC1 41926,C1(C(=O)NC(C)(CO)C2CCC2)CCN(C(C2CCCCS2)=O)C1 41927,N1(C(CCOCCOC(C)=O)=O)CCC2CN(C(c3ccc(C)nn3)=O)CC2C1 41928,C(=O)(C(F)C(C)CNC(c1cccn1C(C)C)=O)NCc1cnc(C(C)C)[nH]1 41929,C12(COC)CCC(C(=O)NCC3C4CN(C(=O)C=C(C)Cl)CC34)(CC1)CO2 41930,c1(C(=O)OCC)c[nH]c(=NC2CN(C(C3CC(C(C)(C)C)=NO3)=O)CC2C)cn1 41931,c1(C(C(=O)N(CCN(C(=O)CC2CC=CCN2C)C)C)O)ccc(Br)cc1 41932,N1(C(CC(=O)OC)=O)CC2CC(C(N3CC(C)(N(C)C)C3)=O)CC2C1 41933,N1(C(C2CC=CC(NC(C3C(C)(C)OCC3)=O)C2)=O)CCC2(CC1)CC2 41934,N1(C(C2C(C)C2C)=O)CC2CCCC(NC(c3ccc(C(N)=O)c(Cl)c3)=O)C2C1 41935,CC(C)C#CC(=O)NC(C)(CO)C(=O)NCCCc1ccccc1 41936,C1(C(=O)NC(CNC(C2CC(SC)C2)=O)CO)CCCC12CCC2 41937,C1(NC(C2N(CC)CC2)=O)CCC(O)CN(C(c2cn(C)nc2OC)=O)C1 41938,N1(C(c2cnc(SC)s2)=O)CCCC2CCN(C(=O)Cc3ccn(C)n3)CC12 41939,C1(C)(CNC(CN(C(=O)C(O)C2CCC2)CC)=O)CCCCO1 41940,N1(C(c2c(-n3cccc3)sc(C)c2C)=O)CCCN(C(=O)CCC(N)=O)C(C)C1 41941,C1(C(=O)NC(C(=O)NCC)C)CC(C)CCN1C(C1CC2(CCC2O)C1)=O 41942,N1(C(c2cn(C)nn2)=O)CC2C(C(=O)N(C3CCCC3)Cc3ccccc3)C2C1 41943,c1(C(=O)NCC2(OC)CN(C(=O)COc3ccccc3)C2)cc2scnc2[nH]1 41944,C(=O)(C1CCc2cccnc21)NCC1(C)CCN(C(=O)COC2CCOCC2)C1 41945,CC(C)CC(F)C(=O)NC1COCC1CNC(c1coc(C(C)(C)C)n1)=O 41946,N1(C(CC(C)NC(=O)C(N)=O)=O)CC(Nc2ccccc2C(N)=O)CC2(CC2)C1 41947,CC(C)CCCC(=O)N1CCN(C(=O)C=CCO)CC1CO 41948,C1(CNC(C(C)(C)OCC)=O)CC(C)N(C(c2cccc(-n3cccc3)n2)=O)C1 41949,c1(OC(CNC(C)=O)=O)ccc(OCC(=O)SC2CCCN2C)c2ccccc12 41950,N1(C(C2N(C(C)C)CCCC2)=O)CC2(CCN(C(=O)CC3(CO)CCC3)CC2)C1 41951,C1(C(=O)NCC(Cc2ccccc2)NC(c2cc[nH]n2)=O)CCC=CCC1 41952,C1(CNC(c2cc(C)n(CCO)n2)=O)CC2(CC2)CN1C(C1CCS(=O)(=O)C1)=O 41953,N1(C(=O)Nc2cnc(CCC)s2)CCC(C(C)(C)C)C(O)C1 41954,C(C(=O)NC(C(=O)NCCNS(N)(=O)=O)C1(C)CC1)(C(C)C)OCC 41955,c1(C(N(C2CCN(C(=O)C=Cc3ncc[nH]3)C2)C)=O)ccc2cnnc(O)c2c1 41956,c1(C(=O)NCC2N(C(C(C(C)(C)O)F)=O)CCC2)cc2c(O)cccc2[nH]1 41957,C#CC(C)(C)C(=O)N1CC(=O)CC1C(N1CCC(C(N)=O)C1)=O 41958,c1(C(=O)NCCC(C)(C)NC(CSC)=O)ccc(S(=O)(=O)N2CCCCC2)o1 41959,n1(CC=C)cc(C(=O)N(C2CCCC2)CCNC(=O)CSCCC(F)(F)F)nn1 41960,c1(C(N(CC(C)NC(c2c(SCC)cccn2)=O)C)=O)cn2c(n1)CCC(C)C2 41961,c1(CC(C(=O)NCC2CN(C(CCC=CC)=O)C2)O)cccc(C(F)(F)F)c1 41962,C1(NC(C=COCC)=O)CCC2CCN(C(=O)CC(C)n3cccn3)C1C2 41963,N1(C(C=Cc2cnc(C)s2)=O)CC(NC(c2cc(C(N)=O)ccn2)=O)CC(O)C1 41964,c1(C(=O)NC(CNC(CCc2n(C)ccc2)=O)C2CC2)coc2ccccc12 41965,N1(C(Cc2nc(C)sc2C)=O)CC2CCCC(NC(=O)CC3(O)CCCC3)C2C1 41966,C12(C(N3CC=CC(NC(C4C(C(=O)OC)C4)=O)C3)=O)CC(C)(C1)OC2(C)C 41967,c1(OC)ccc(OCCC(=O)NC2CC2NC(c2ccco2)=O)cc1 41968,N1(C(C(CC2CC2)OC)=O)CCC(N(C)C(c2cc(N)c(C(=O)OC)s2)=O)CC1 41969,c1(C(N2CC(F)CC(NC(=O)CC3CC=CC3)C2)=O)cc2cc(Cl)ccc2o1 41970,C(=O)(C(CC(C)C)NC(=O)OC)N(CCNC(c1sc(O)nc1O)=O)CC 41971,N1(C(c2cc(C)nc(C)c2)=O)CCOC2(C1)CN(C(=O)C(C)OC1CCOC1)C2 41972,N1(C(CC(CCC)C)=O)CCC2(C1)CN(C(C1CCCN1c1cnccn1)=O)C2 41973,C1(C(N(CC(C(C)C)C)C)=O)C(C)OCCN1C(c1c[nH]c(=O)cn1)=O 41974,C1(NC(CC2C(C)CCO2)=O)(CNC(C2CC(N(C)C)C2)=O)CCCCC1 41975,c1(CC)nccnc1C(=O)NCC(N1CCN(C(=O)C(O)C(C)SC)CC1)=O 41976,C1(CC)CN(C(C)=O)CCC1NC(=O)C(=O)NCC1(c2ccccc2Cl)CC1 41977,c1(C(=O)NC(c2ccccc2)CNC(C2(CF)COC2)=O)cccc2nc[nH]c12 41978,C(=O)(CC(C)CC(=O)N1CCCN(C(=O)Cc2ncc(Cl)s2)CC1C)OC 41979,c1(CC(=O)NCC2CCCC2NC(=O)CNC(c2cccs2)=O)cncc(F)c1 41980,c1(OC)c(C(=O)N(CC(C)CNC(c2nocc2C(C)C)=O)C)cc(Cl)cc1Cl 41981,N1(C(C2CC(NC(c3c(CC)ncs3)=O)C(O)C2)=O)CCS(=O)C(C)C1 41982,C1(NC(C2C(C=C)OCC2)=O)CC(F)CN(C(c2ccc(Cl)cc2OCC)=O)C1 41983,C1(NC(Cc2c(C)ocn2)=O)CN(C(C2CC3CCCCCC23)=O)CCC1(C)C 41984,N1(C(CC2OCCN(C(c3c(C)ccnn3)=O)C2)=O)CC(O)CC(C)(C)C1 41985,C1(NC(=O)Nc2cc(C)c(-n3cccn3)cc2)C2Cc3ccc(Br)cc3C12 41986,c1(OC)ncc(Br)cc1CN1CCOCC1CC(=O)Nc1ccc(C)cc1OC 41987,c1(C(N2C(CCNC(CSC(C)(C)C)=O)CCC2)=O)coc2c1C(=O)NCCC2 41988,N1(C(=O)C=CC2CCC2)CCC(NC(c2sccc2-n2ccnn2)=O)C(CO)C1 41989,c1(CC(=O)NCC(CC)NC(c2cccc(CO)c2)=O)ccc(Br)c(OC)c1 41990,C1(CC(N2CC(CNC(C(COCC)C)=O)OCC2)=O)CN2CCC1CC2 41991,N(C1CN(C(=O)Cn2cncn2)CCc2ccccc21)C(C1=CC(C)(C)C1)=O 41992,Cc1nc(=NCC2CCCCN2C(c2ccc(C3CC3)cc2)=O)[nH]cc1[N+](=O)[O-] 41993,CC(CC(=O)NCc1ccnc(C(N2CCCC2(C)CO)=O)c1)CC(C)(C)C 41994,CCCC(CC)CCC(=O)NCc1cn(CCNC(=O)CCN2CCCC2)nn1 41995,N1(C(C2N(C(CC)=O)CCCC2)=O)CC(NC(=O)CC(C)(C)O)C2CCCCC12 41996,c1(C(=O)NCC2(C)CCCN(C(CCC(C)(C)F)=O)C2)ccc2nc(O)oc2c1 41997,C(C)(CNC(=O)COc1ccc(C2CC2)cc1)(C(C)C)NC(C=C(CC)C)=O 41998,NS(=O)(=O)c1ccc(C(N2CC(CC(N3CCN(CCCO)CC3)=O)C2)=O)o1 41999,CC(C)CC(C)CN=c1[nH]c(N2CCC(C3CCN(C)C3)CC2)nc2c1CSC2 42000,C(=O)(CCC(C)(C)[N+](=O)[O-])N(CCC(C)C(F)F)C.C1(=O)C(C)(C)CN1 42001,CC1COC(CC(F)(F)F)N1C(=O)Nc1ccccc1-c1cccnc1 42002,N1(C(c2cn(C3C=CCCC3)nn2)=O)CCN(CC(F)(F)F)CC1.CC(C)(C)O 42003,N1(C(c2c(OC)n[nH]c2)=O)CCN(C)C(C(=O)NC2CCNC(=O)C2)C1 42004,C1(NC(C2C(C)(C)C2)=O)CCCN(C(c2cc(Cl)nnc2Cl)=O)CC1 42005,Cc1ccc2c(c1)CC(C(=O)NC(CNC(=O)CCc1cnoc1)C1CCC1)O2 42006,Cc1c(C(=O)NCC(C)(C)CN(C(=O)C(C)N(C)C)C)ccc(Br)c1F 42007,C1(N(C(=O)CSC(F)F)C)CCCCN(C(=O)C(C)(C)C2CCCC2)C1 42008,N1(C(CCNC(C2C(C)C2)=O)=O)C2CCC1CC(CNC(=O)CC1CC13CC3)C2 42009,N1(C(C(C(C)C)N(C)C)=O)CC2(CCN(C(C3CC3(C)C)=O)CC2)C1 42010,c1(C(=O)NC)cccc(C(=O)NCc2nc(CNC(C3COC(C)C3)=O)cs2)c1 42011,C1(C(N2CC(CCNC(c3c(C)nc(CC)s3)=O)OCC2)=O)CS(=O)(=O)CCO1 42012,N1(C(CCC(C)(C)C)=O)CC2CCN(C(=O)Cc3cccc4c3CCC4)CC2C1 42013,c1(CC(N2CCC(CN(C)C(C3(C4CC4)CC3)=O)C2)=O)cnc2c(=O)[nH]ccn12 42014,C=CCC(CC)C(=O)NCC1(NC(=O)Cc2sc(O)nc2O)CC1 42015,Cc1ccc(C(N2CC(C)CC2C(=O)NC2CC(C)(C)C23CC3)=O)c(O)c1 42016,c1(C(=O)NC2CCC(CC(=O)NC(C(C)O)C)C2)ccc(N(C)C)cc1 42017,c1(CN(c2cc3ccccc3[nH]2)C)ccc2nccn2c1 42018,N1(C(CC(=O)NCC#C)=O)CCN(C(=O)CC2(CO)CC2)C(CCC)C1 42019,N1(CC)OCC(N(C(=O)CC2CCN2C(c2cocc2C(N)=O)=O)CC)C1=O 42020,N1(C(COCC(=O)NC)=O)CC(C)(C)OCC1CNC(C1CCCC(F)(F)C1)=O 42021,N1(C(C(C)CN(C)C)=O)CCN(C(C2(n3cncn3)CC2)=O)CC1CCN(C)C 42022,C1(C(=O)NCC2CC2CNC(c2coc(C)n2)=O)(OC)CCCOC1 42023,Cc1cn2c(=O)c(C(=O)NCCNC(C3C(C)C3C)=O)cnc2s1 42024,O=C(CS(=O)(=O)CCO)NCC1CCCC1NC(C1CNC(=O)N1)=O 42025,N1(C(C2C(NC(c3ccnc(SC)n3)=O)C2)=O)CC(F)(F)C(F)(F)C1 42026,c1(OC)ncc(C(=O)NC2CC(NC(=O)CC3CCOC(C(C)C)C3)C2)c(C)n1 42027,CC(C)CC(C)CC(=O)N1CCC=C(CNC(c2cn(C(C)C)cn2)=O)C1 42028,N1(C(C2N(C)C(=O)CC2)=O)CC2(C1)CN(c1ccnc(C#N)n1)C2 42029,N1(C(CC2CCCC(C)C2)=O)CC2(CC(NC(=O)CC=CC(C)(C)C)C2)C1 42030,c1(OC)cc(N2CCC3CCC(C2)N3C(C2CCCO2)=O)ccc1[N+](=O)[O-] 42031,C(=O)(C1=CCC(F)(F)CC1)NC1CCC(NC(C(CCC)(C)O)=O)CC1 42032,N1(C(c2cnc(C(C)(C)C)nc2)C(=O)NCC)CCn2c(cnc2C(F)F)C1 42033,c1(C(=O)NCC2N(C(C(CC)F)=O)CCC2)ncc(C)cc1C 42034,c1(CCC(=O)NCC2C(NC(c3nnc(C)s3)=O)COC2)ccccc1Cl 42035,C=CC(C)(CC)C(=O)NCC1(C)CCN(C(C2(Sc3ccccc3)CC2)=O)C1 42036,N1(C(C(CC)Oc2ccccc2)=O)CCC(NC(=O)C(C)(C)n2cnnn2)CC1 42037,C1(C#N)(C(N2CC(CNC(C3(C(=O)NC)CC3)=O)C2)=O)CC1C(F)(F)F 42038,C(=O)(C1=C(C)CCOC1)NC(C(=O)NCC(C)OCC#C)C1CC1 42039,c1(C(=O)NCC(C)(C)NC(=O)CCc2ccsc2)cc(F)c2ccccc2c1 42040,CC1(C)CC(N=c2cc(C(F)(F)F)nc(Cl)[nH]2)CN(C(=O)CCC2CC2(F)F)C1 42041,c1(N2CCC(CNC(C3C(CC)OCC3)=O)C2)nc(Cl)c(C#N)s1 42042,N1(C(COC(c2nccn2C)C)=O)CCC(C(C)NC(c2ccns2)=O)CC1 42043,C1(CNC(C2CCN(CC)C2)=O)CC2CCC1N2C(=O)CCCCOC 42044,c1(C(CF)NC(=O)C(=O)Nc2ccccc2)ccc(Cl)cc1.C1(N)CC1CO 42045,CC(C)(CCCNC(=O)C(CO)C(F)(F)F)C(=O)NCC12CCC(CC1)OC2 42046,c1(C(N2C(C)(CC(=O)NC3(C#C)CC3)CC2)=O)cc(C#N)[nH]c1C 42047,c1(N2CCCC(NC(N)=O)C2)nc2c(c(=NCc3ccc(Br)s3)[nH]1)COC2 42048,C1(O)(CNC(C#CCNC(C2C(C(C)(C)C)C2)=O)=O)CCCOC1 42049,c1(CN(C(=O)C(=O)NCC2CC2)CCOC)c(C)nn(C)c1C 42050,N1(C(C(CC)N(C)C)=O)CCCC2CN(C(=O)COC3CCOC3)CCC12 42051,c1(C(C)(C)C)cccc(C(N2CC(NC(c3cnsc3)=O)C2)=O)c1.C1C=CCO1 42052,c1(NC(C2CCC3(CCCNC3)C2)=O)ccnc2c(Br)cc(F)cc12 42053,c1(C(=O)NC2CC(C3C(=O)NC(=O)N3)C2)ccc(S(F)(F)(F)(F)F)cc1 42054,CC1(C)CC(NC(=O)C=Cc2ccc(F)cc2)CN(C(c2ccsc2C#N)=O)C1 42055,N1(C(C(c2ccccc2)=O)=O)CC2CC(NC(C3(C4CCCO4)CC3)=O)CC1C2 42056,C(=O)(C(C)(C)C(=O)N(C)CC1CCN(C(c2ccccn2)=O)C1)NC 42057,c12nnnn1CC(=O)NCC1CCN1C(=O)C21CC1.C1(C)(N)CC1(C)C.CCC 42058,C#CCC(CC#C)C(=O)N(C1CN(C(c2ccc(S(C)(=O)=O)o2)=O)CC1(C)C)C 42059,C1(NC(c2c(F)cncc2Br)=O)CC2(C1)CN(C(=O)C(O)C(F)F)C2 42060,n1(CC(=O)NCC2(CN(C(=O)CC(C)(C)C)C)CC2)cccc(N)c1=O 42061,CC1(C)CN(C(c2ccoc2)=O)C1C1CCN(C(C2(O)CCSC2)=O)CC1 42062,N1(C(C2CCCN(C(N)=O)C2)=O)C2CCC1CC(CNC(C1CC=CCC1)=O)C2 42063,c1(OC)ncc(Cl)cc1C(N1CC(CNC(C2CCC(C)(O)CC2)=O)C(C)C1)=O 42064,O=C(O)CC(C1CCCC1)NC(C1C(c2ccccc2)C1(F)F)=O 42065,c1(C(=O)NC2CCN(Cc3n(CCC)ncn3)C2)cc(OC)ccn1 42066,CC1CN(C(c2ccnc(O)c2F)=O)CCC1N(C(=O)C=C(Cl)Cl)C 42067,c1(C(=O)NCC(CN(C)C(C2(F)CC2c2ccccc2)=O)O)nnc(C(C)(C)C)s1 42068,c1(CC(N2CCOCC(NC(C(C(C)C)O)=O)C2)=O)ccc(C#N)cc1F 42069,c1(C(=O)NC(C(C)NC(=O)CC2CCCOCC2)CO)cnc2sccn12 42070,C1(C(N2CCC(NC(c3ncccc3Br)=O)C2)=O)CCC=CCCC1 42071,CCC(C)(CNC(=O)CCc1cnoc1)NC(=O)CC1CC=CCC1 42072,c1(C(=O)NC(C(=O)N(CCCC)CC)CO)cnncc1OC 42073,c1(C(=O)NCC(CC)NC(c2ccc(N)cc2Cl)=O)cc(P(C)(C)=O)ccn1 42074,Nc1ccc(C(=O)NC2(C3CN(C(C4CCN4S(C)(=O)=O)=O)C3)CC2)cc1F 42075,Cc1n[nH]cc1CC(=O)NC1CC(C)(CNC(=O)C(C)OCOC)C1 42076,CC(C)(CN=c1nc(N2CCC(C(N)=O)C2)c2sccc2[nH]1)C(F)(F)F 42077,C1(C(=O)NC2C(NC(C3CN(S(C)(=O)=O)C3)=O)C2)CS(=O)(=O)CC12CC2 42078,C1(OC)CCn2cc(C(=O)NC3CCCC(CNC(c4cscn4)=O)C3)nc2C1 42079,C1(C(N(CCNC(C2CC(C(F)(F)F)(OC)C2)=O)C(C)C)=O)CCOCC1C 42080,C(=O)(CC(C(F)F)n1ccnc1)NC(C(=O)OCC)Cc1ccccc1Br 42081,CCCS(=O)(=O)CC(=O)NCC1CN(C(c2sc(C)c(C)c2C)=O)CC1O 42082,Cc1cccc(C)c1C(=O)NCC1C(CNC(=O)C(C)NCC(F)(F)F)C1(F)F 42083,C1(CNC(=O)CC2CC23CC3)CN(C(=O)Cc2ccc(O)c(Cl)c2)CCCO1 42084,N1(C(C(C(C)C)O)=O)CC(C)OC2(CCN(C(c3ccc(F)cc3O)=O)C2)C1 42085,c1(C(N2CCC(NC(=O)C(F)(F)C(F)F)C2)=O)ccc2c(c1)CNC2=O 42086,c1(CC(=O)NCCC2CC(NC(CN(C)C3CC3)=O)C2)cnn2ccccc12 42087,CC(C(C(=O)NC)N1CCCC(CS(C)(=O)=O)C1)=Cc1ccc(Br)s1 42088,N1(C(C2(c3ccc(C)cc3)CC2)=O)CCC(NC(=O)CCCCBr)C(F)C1 42089,c1(C(=O)NC(C)(C)CCNC(c2sccc2CO)=O)ccc2c(c1)CCN2 42090,C12(C(=O)NCC3(C#C)CCCC3)C(NC(c3cccc(C)c3F)=O)C3CC1C2C3 42091,C1(CC(=O)NCc2c(C(=O)NCC#C)con2)CCCC12CC2 42092,c1(OC)nccc(C(N2CC(NC(C3(OC)CCC3)=O)C(O)C2)=O)c1Br 42093,CC1C(NC(=O)C#CC2CCCC2)C(C)CCN1C(=O)CNC(N1CCCC1)=O 42094,N1(CC(=O)NCC(CNC(c2ccc(OC)o2)=O)CO)CCC(F)CC1 42095,C1(O)(CCNC(c2c(C)cns2)=O)CCN(C(C2CCCC(O)C2)=O)C1 42096,C1(C2CCN(C(C3C(C(C)C)(CC)C3)=O)C2)CCCCN1CC1CCCC1(C)C 42097,C1(C(N2CCC(O)(CN(C(C(C)=CC)=O)C)C2)=O)Cc2cncn2C(=O)N1 42098,C(=O)(C#CC1(CC)COC1)NC(CC=C)C(=O)NCC(C)(C)n1cccn1 42099,C(C)(CCN=c1[nH]c(Cl)nc(C)c1F)NC(c1c(C)nsc1C)=O 42100,C1(NC(C2C(OC)CC2)=O)CCN(C(c2cnc(S)n2C2CC2)=O)CCC1(F)F 42101,c1(C(=O)NC(CC)CNC(=O)C=Cc2ncc[nH]2)cnc(O)n1CC 42102,C1(C)(C(N2CC3(CN(C(=O)Nc4c(C)cccc4C)C3)C2)=O)CC(C(C)C)=NO1 42103,CC1(C)CCC(C)(C)c2cc(C(N3CC4CCS(=O)(=O)CC4C3)=O)c(Br)cc21 42104,N1(C(c2ccc(NC(C)=O)s2)=O)CCC(CNC(=O)CCN2CCC2)CC1 42105,C1(C(N(C)CC2CCN(C(=O)CC#N)C2)=O)C2CCC1(c1cncs1)C2 42106,C1(n2cc(C3N(C)CCC3)nn2)CCCC(NC(=O)CC2CC=CCC2)C1 42107,CCC(CC(=O)NCCc1cnc(C)cn1)N(C(=O)CCCCSC)C 42108,C(C)(C(C)N=c1cc[nH]cc1S(=O)(=O)N(C1CC2(CC2)C1)C)n1ncc(C)c1 42109,c1(C2(C(N3CCCN(C4CCOCC4)CC3)=O)CC2)ccc(F)c(OC(F)F)c1 42110,C1(F)(CNC(c2nc(OCC)sn2)=O)CCCN(C(C2CNC(=O)C2)=O)C1 42111,c1(CNC(=O)Nc2c(C#N)cc(CC)s2)ccc2ccccc2n1 42112,C12(C(=O)NC3CC(CC(C)(C)C)C3)CC(NC(=O)CSCC(N)=O)(C1)C2 42113,C1(CC(=O)NCCCCCNC(c2nc(C)n(C)n2)=O)(NC(C)=O)CCCCC1 42114,c1(CNC(C2(NC(C(C)O)=O)CC(O)C2)=O)cncc(O)c1 42115,N1(C(C=CCOC)=O)CC(NC(=O)COc2cc(C)on2)CC(C)C1 42116,c1(C(=O)NC2(CC=C)CCC2)c(CNC(=O)C(C#N)CC)cnn1C 42117,C12(CNC(=O)C=Cc3nccs3)CC(CN1C(=O)COc1ccccc1)C2 42118,CC1(C)CCC(CC(N2CCCCC2C2(NC(C3COCCN3C)=O)CC2)=O)C1 42119,C1(CNC(C(C)=CC2CC2)=O)C(C)CCCN1C(c1cccnc1)=O 42120,C=C(C)C1OCCC1CNC(=O)C(O)C1CN(C(C2(C)CC3C=CC2C3)=O)C1 42121,N1(C(CCOCCC)=O)CCC(C(C)NC(=O)C(c2cncn2C)=O)C1 42122,C1(F)(C(N(C2CCN(C(c3cnc(C(N)=O)s3)=O)CC2)CCC)=O)CCOCC1 42123,C1(C(C)C)(C(=O)NC2(c3ncco3)CC2)CCN(C(=O)CCn2cncn2)C1 42124,c1(CNC(CCC2CC(OCC)C2)=O)nn(C)cc1C#C.C12CC1CC(=O)NC2 42125,C(c1cc(F)cc(F)c1)=CC(=O)NCC1CCCN1Cc1cc(Cl)ncc1Cl 42126,Cn1cncc1CC(=O)NC1CCCC1C(N1CC(N2CCNC2=O)C1)=O 42127,C1(C(=O)NCc2scc(C)c2)C=CCCN1C(C1CCSC1)=O 42128,c1(CNC(c2c(CNC(C(CC3CC3)OC)=O)noc2)=O)ccnc(F)c1F 42129,c1(CC)c(C(=O)NC2CCCCC2CNC(C2(C)CC2)=O)ccn1C 42130,N1(C(C(C)CC2CCC2)=O)CCC(F)(F)C(CNC(=O)C2=CCS(=O)(=O)C2)C1 42131,Cc1c(F)cc(CN2CCCC(CNC(c3cnn4ccccc34)=O)C2)cc1Br 42132,c1(C(N2CCCC(N(C(=O)C#CC3(C)CC3)CC)C2)=O)nn2c(c1C)CCCC2 42133,CCC(C)(C(=O)Nc1cccc(NC(=O)CC2C=CCCC2)c1)OC 42134,C1(CCC2N(C(C(=O)N(C)C)=O)CCC2)CCCCN1C(=O)C=Cc1cocn1 42135,C(=O)(C(C)(C)CF)NCC(CCOC)NC(C1(N2CCCC2)CCC1)=O 42136,Cn1ncnc1C(c1nnnn1C1COC1)NCC1(c2ccccc2)CCCO1 42137,C(=O)(CC(C)C(F)(F)F)N(CCC)CCNC(C1C2CCC1(c1cnco1)C2)=O 42138,Cc1ccoc1C(=O)NC1CCC(C(=O)NCCC2CC=CCC2)C1 42139,c1(CCC(=O)N(C2CC(NC(CC=CC)=O)C2)C)cnn(C)c1C 42140,CC1(C)CN(C(=O)Nc2cnn(C(C)(C)C)c2C(F)(F)F)CCS1(=O)=O 42141,c1(OC)ccc2cc(C(=O)NCC3CC4CC3CO4)[nH]c2n1 42142,CC(C)C(C(C)NC(=O)C=CCF)NC(c1cc(C2(C)CC2)on1)=O 42143,C1(CNC(CSCCOC)=O)CC2CCC1N2C(c1cc2n(n1)CCO2)=O 42144,O=C1CC(C(=O)NCC2(C3CC3)CCCO2)N(C(C2CCCCC2)=O)C1 42145,c1(C(N(C(CNC(C2(CN(C)C)CC=CC2)=O)C2CC2)C)=O)ccc(CF)cc1 42146,C1(C(N2CC(NS(C)(=O)=O)C2)=O)CC(n2cc(-c3ncccc3F)nn2)C(O)C1 42147,C1(NC(CC2(COC)CCCC2)=O)CN(C(=O)CN2CCOCC2)C2(CCC2)C1 42148,O=S(=O)(c1cccc(=NC2C=CCCC2)[nH]1)NCC1C2C3CCC(C3)C12 42149,c1(CCC(=O)N(CC(C)O)CCNC(=O)CP(C)(C)=O)ccc(Cl)cc1F 42150,c1(CC(=O)NCC(C2CCOC2)NC(CCC)=O)coc2cc(Cl)ccc12 42151,C=CC(C)CC(=O)N(C1(C(=O)NCc2ccc(Cl)cn2)CCC1)C1CC1 42152,C12(CNC(CC(CN(C)C)O)=O)CCCC(CN(C(=O)C=CC(C)(C)C)C1)C2 42153,C(C(CC(C)C)C(=O)N1CC2(CC(C)CO2)C1)NC(C1C(OCC)CC1)=O 42154,N1(C(CSCC#C)=O)CC(C2CC2C(N2CC(N3CC(O)C3)C2)=O)C1 42155,c1(CC(=O)N(C2CCN(C(C(CCC)OC)=O)C2)C)c[nH]c2ncccc12 42156,c1(C(=O)NC(CNC(CC(C=C)c2ccccc2)=O)C)cc([N+](=O)[O-])oc1C 42157,C1(N(C(C2CC2(C)C(C)C)=O)CC)CCN(C(c2snnc2C)=O)CC1 42158,c1(C(N(C)CC2CCN(C(CC3(COC)CC3)=O)C2)=O)cncc(OC)c1C 42159,C1(NC(C(C)NS(CCC)(=O)=O)=O)CC(NC(=O)CCNC(C)=O)CC1O 42160,C1(CC=C)(NC(c2cc(Cl)cnc2O)=O)CCCN(C(=O)CN(S(C)(=O)=O)C)C1 42161,c1(CC(=O)NCCC2N(C(C=C(C)C)=O)CCC2)ccc2c(c1)CCCC2 42162,N1(C(C(n2cc(C3(O)CCCC3)nn2)C)=O)CCC(CO)C1CC1CCCC1 42163,C(=O)(C(O)CC(C)(C)C)NC(C(=O)NCC1CC(C)OC(C)C1)Cc1cn[nH]c1 42164,C1(C(=O)NCCCN(C(C#CC(C)(C)O)=O)C2CC2)CC2(CCOCC2)CO1 42165,N1(C(C(CC)OC)=O)CC(N(C)C(c2sc(C)nc2C)=O)C2(CC2)C1 42166,c1(C(=O)NCC2CN(C(c3c(OC)n[nH]c3)=O)C(C)C2)nccc2[nH]ccc12 42167,c1(C(=O)NCC2C(NC(c3c(CC)scn3)=O)CC2)c(C)nn2cccnc12 42168,c1(CC(=O)NC(C)(CO)C2CC2)cnnn1C.C1(C(=O)NC)(CCNC=O)CCC1 42169,c1(CC)ccccc1C(=O)NC(CCF)C(=O)N(CCC1CC1)CC 42170,C1(CC(=O)NC2C(CNC(=O)CNC(=O)Cn3cncn3)C2)CN2CCN1CC2 42171,C1(CNC(C=CC=CCC)=O)CCCCCN1C(=O)CC(C)(C)CNC(C)=O 42172,C(=O)(CCCCCCCCCCC(=O)O)NCCSCCOC 42173,C=CC1(CC(=O)NCC(c2ccccc2)NC(=O)CC2(O)CC2)CCCCC1 42174,CCCCC(O)C(=O)NC1COCCN(C(C2CCCCN2C)=O)C1 42175,C1(NC(=O)CCCn2c(O)nnc2O)COCCN(C(c2ccsc2CO)=O)C1 42176,c1(CNC2(c3n(CCCOC)nnn3)CN3CCC2C3)ccc2cccnc2n1 42177,N1(c2nc(OCC)c(Cl)cn2)CCC2(NC(c3ncccn3)=O)CCCCCC12 42178,Cc1ccc(C(=O)N(CCCCCC(=O)NCC2CCC(F)C2)C)nc1C 42179,N1(C(C=C(CC)C)=O)CCN(C(C2(C(C)(C)O)CC2)=O)CC12CC2 42180,O=C1NCc2ccc(NS(=O)(=O)CC3CCCC(C(F)(F)F)O3)cc21 42181,c1(C(=O)NCC2N(C(C3CC(N(C)C)C3)=O)C3CCC2C3)ccc2ncnn2c1 42182,N1(C(c2cn(CC)nc2)=O)CCC2CCCC12C(=O)NC(C)Cc1nncn1C 42183,C(=O)(C1=CCCCC1C)N1CC(N(C(CSc2cccc(OC)c2)=O)C)C(F)C1 42184,c1(C(N2C(CNC(Cc3cc(C)[nH]n3)=O)CC(F)C2)=O)c(F)c(F)cc(F)c1F 42185,C(C(CC=C)C(=O)NCc1ncsn1)NC(C(C)=CC=C)=O 42186,c1(C(c2nn[nH]n2)CNC(=O)COCC2CCNC2)ccccc1 42187,C1(NC(CC2C(CNC(=O)COc3cccc(O)c3)C2)=O)CCC2(CC1)N=N2 42188,c1(CC(=O)NC2CCN(C(c3cocc3C(=O)O)=O)CC2)ccccc1Cl 42189,CC1CCCCC1C(=O)NC(C1CN(C(C2(C)CC(F)C2)=O)C1)C 42190,Cc1nc(C(=O)NCC(C)NC(c2cnc(C(C)O)s2)=O)cc(O)n1 42191,c1(CC(=O)OC)ncccc1C(=O)NC1CC(C)(NC(=O)C(C)SC(C)C)C1 42192,N1(C(=O)NCCc2cccc(C)n2)CCC(F)(F)C2(CC1)NC(=O)NC2=O 42193,c1(C(N(C2CCC(NC(=O)CCc3ccco3)C2)C)=O)ccnnc1O 42194,c1(C(=O)NCCN(C(c2n(C=C)nnc2)=O)C(C)C)cc(Cl)cc(C)c1C 42195,c1(CC)ccc2occ(-c3nc(CN4CCOCC4)nn3C3CCOC3C)c2c1 42196,N1(C(c2c(C)csn2)=O)CC(NC(=O)C(C2CCOCC2)C)CCC(O)C1 42197,CC1(C(N2CCN(C3CN(C(=O)C(O)C4CC4)C3)CC2)=O)CC=CCC1 42198,Cc1c(CC(=O)NC2CC(NC(=O)CC(C)F)C2)c(=O)oc2cc(O)ccc12 42199,C1(N(C)C)CN(C(C2CC23CC(NC(=O)CCCC2CCCO2)C3)=O)CC12CC2 42200,N1(C(c2c(CC)nn[nH]2)=O)CC(CNC(=O)Cc2c[nH]nc2O)CCC1C 42201,N1(C(C2OCC(C)(C)C2)=O)CC2(CC2)CC1CNC(c1cc2n(n1)CCC2)=O 42202,C1(NC(C(C(=O)NC)(C)C)=O)CCN(C(C2CC3C=CC2C32CC2)=O)CC(O)C1 42203,c1(C(N2C(CNC(C(C(C)(C)C)O)=O)C3CCC2C3)=O)sc2ncccc2c1N 42204,CC1(C)CNc2ccc(C(=O)NCCCCCCCO)cc21 42205,C1(OC)CCCC(NCC(=O)Nc2cccc(I)c2)C1 42206,C1(NC(Cc2cc(C)on2)=O)CCOC(C(=O)NCc2ccc(Cl)cn2)C1 42207,CC(C)C(C(=O)NCC(C)CN(C)C(C1CN(C)C1)=O)n1ccnc1 42208,C1(NC(Cc2c(C)nccc2)=O)CS(=O)(=O)CC1NC(C1(CF)CC1)=O 42209,c1(C(=O)NC(CNC(C2(CC)CCNC2=O)=O)C(C)(C)C)cncc(C)c1Cl 42210,C(=O)(CC(C)(C)CC(F)F)NC1CCC(CNC(CCN(C)CCO)=O)C1 42211,N1(C(c2cc(C)nc(O)c2)=O)CC2CCC(C1CO)N2C(c1ccnc(O)c1)=O 42212,C(CC)(CCC(=O)NCC1(O)CCSC1)NC(CCC#C)=O 42213,C1(NC(C2(CO)CCN(C(CN(C)C(N)=O)=O)C2)=O)CCCCC1C#N 42214,C(N=c1[nH]c(=NCC(C)C#N)[nH]c2c1SCC2)c1cc(C)c(C)s1 42215,c1(OC)c(NC(C2CNCCN2Cc2c(Cl)ccnc2OC)=O)cccc1C#N 42216,C1(C)(C(=O)NCCCC(C)NC(c2ocnc2C2CC2)=O)CC(C(C)(C)C)=NO1 42217,C(c1ccccc1F)=CCC(=O)NC1CN(C(C2(CCCC)CCC2)=O)CC1O 42218,CCC(C)(C)C(c1ccccc1)NCCCCC(=O)OC 42219,c1(C(=O)NCC(c2cc(OC)c(C)cc2)=O)cnc2onc(C(C)C)c2c1 42220,c1(C(N2CC(O)(CN(C(CC=CC)=O)C)C2)=O)ccc2c(c1)CCCS2(=O)=O 42221,C1(NC(=O)OC)CCC(C(=O)C2CC2)CC1.C12CCN(CC1)C2=O.C12(CC1)NC2 42222,N1(C(C2(C(=O)OC)CCCC2)=O)CC(C2(NC(C3(F)CCOC3)=O)CC2)C1 42223,CON1CCC(N(C(=O)C(c2cn(C)nn2)NC(c2ccc(Cl)cn2)=O)C)CC1 42224,C1(CSC)(CNCC(=O)NC(C2CNC(=O)O2)=O)CCOCC1 42225,C1(NC(c2cc(CC)oc2C)=O)CCN(C(=O)CCOC(C)C)CC1F 42226,Cc1c(C(=O)NCCC2CC(NC(=O)C(C)c3cccs3)C2)cnn1CC(F)F 42227,N1(C(N2C(c3n(CC)cnc3)CCCC2)=O)CCCc2ccc(F)cc21 42228,C1(C(NOC)=O)CC(C)N1C(c1cncn1C)=O 42229,N1(C(c2nc(CC)sc2)=O)CCC(C2CCCN(C(C3(O)CC3(C)C)=O)C2)CC1 42230,C(=O)(C(C)C(C)(C)C)N(C(C)CN(C)C(c1cn(C)nc1C(C)(F)F)=O)C 42231,N1(CCC(=O)N(C(C)CNC(c2ccn(C(F)(F)F)n2)=O)CC)CCCCC1=O 42232,Cc1cn2c(=O)c(C(=O)N(CC(O)CNC(C3CCCS3(=O)=O)=O)C)cnc2s1 42233,c1(C(N2CCN(c3nc(COC)nc(Cl)c3)CC2)=O)cc2cc(C)ccc2cn1 42234,c1(NC(C(C)N(C(C2(C#N)CC23CCC3)=O)C2CC2)=O)cnc2ncnn2c1 42235,C1(CC(=O)O)CC(C(=O)Nc2cnn(-c3ccccc3Br)c2)CCO1 42236,N1(Cc2ccc(N3CCCC(C(=O)O)C3)o2)CCCc2ccccc21 42237,Cc1cc(CNC(C2CC(NC(C3(N(C)C)CCOCC3)=O)CCO2)=O)ncn1 42238,C1(CC)(CC)CNC(=O)C1NC(c1cc(OC)c(Br)s1)=O 42239,c1(OC)ccc(C(C)NCC2CC(F)(F)C2(C)C)c(OC)c1 42240,C(c1cc(C)cc(C)c1)=CC(=O)NCC(CCOC)NC(C1(CO)CCCO1)=O 42241,c1(C(=O)NC(c2cccc(Cl)c2)CNC(CN(C2CC2)CC)=O)nc(C)nn1C 42242,N1(C(c2cccc(CC)c2)=O)CCC(F)C(NC(C2CCCCC2CC)=O)C1 42243,CCCC(O)CC(=O)NC(CNC(C1CCCS1)=O)(CC)CC 42244,c1(-c2ccc(=NC)[nH]c2)ccc(C(N2CCC(CO)C(O)C2)=O)c(C)c1F 42245,CC(C)CCCCC(=O)NC1(CNC(=O)C(C)C2CC2)CCCC1 42246,Nc1c(Cl)cc(C(=O)NCC2(F)CC(NC(C3CC3[N+](=O)[O-])=O)C2)cc1[N+](=O)[O-] 42247,N1(C(CC2(OC)CC2)=O)CCC(C(C)NC(=O)C(c2ccc(F)cc2)(C)C)CC1 42248,Cc1nc(C)c(F)c(=NCC(C(C)(C)C)NC(C23CCC(N=[N+]=[N-])(CC2)C3)=O)[nH]1 42249,c1(C(N(CC(C)NC(=O)Cn2cc(C(N)=O)nn2)C)=O)csc(C(F)F)n1 42250,C1(NC(C2(COC)CCCC2)=O)CC(NC(=O)C(C)(C)Cn2cccn2)C12CCC2 42251,n1(CC(N2CCC(C(C)NC(CS(CC)(=O)=O)=O)C2)=O)cc([N+](=O)[O-])c(C)n1 42252,CN1CCOC(C(=O)NCc2cc(C(=O)N(C3C4CCCC34)C)ccn2)C1 42253,N1(C(CN(C)C(N)=O)=O)CC2CCC(NC(c3c(Cl)ccnc3F)=O)CC2C1 42254,c1(CNC(CC2(N(C(CNC(C)=O)=O)C)CC2)=O)cnn(C)c1 42255,C12(NC(CCOCCCOC)=O)CCCN(C(C3(C)COC3)=O)CC1C2 42256,C(CN=c1[nH]c(=NC(C)c2ccoc2)c2sccc2[nH]1)c1c(C)nc[nH]1 42257,n1(CC)cc(Cl)c(C(=O)Nc2cccc(NC(=O)CCC3CC3CC3CC3)c2)n1 42258,C1(O)(CCC)CCN(C(=O)C(C(C)CC)N(C(=O)CCCC#N)C)CC1 42259,C(CCCCCCCO)=CC(=O)NC1C(CNC(C(COC)(C)O)=O)CC1 42260,CC1C(NC(C2CCCC2)=O)CC2CCC1N2C(c1ccc(C(F)F)o1)=O 42261,c1(C(=O)NCC(CCC)NC(C2CCCC2F)=O)cc(C)c(C)o1 42262,c1(OC)cc(F)c(F)cc1S(=O)(=O)N1CC(C)(C)CC1C 42263,C(CC(C)C)(C(=O)NCC1CCN1C(=O)Cc1cccc(N(C)C)n1)NC(C)=O 42264,N1(C(C2C(CNC(CC(C=C)CCC)=O)CCO2)=O)CCc2cc(C)ccc21 42265,c1(CN(C2CC2)CC)cccc(OC)n1.C12CCC(CC1)CC(=O)N2CCO 42266,C1(NC(c2c(C)nsc2C)=O)CC12CCN(C(c1cnn3ccn(C)c13)=O)CC2 42267,N1(C(C(C2CCCN(C(C(CC)(C)COC)=O)C2)C)=O)CC(C)N(C)C(C)C1 42268,C(C(C)(C(=O)N(CC(C)(C)CO)C)NC(c1cc(=N)[nH][nH]1)=O)SC 42269,C1(C(=O)NC(C)(CO)CCF)CCCC(NC(=O)C=Cc2ccco2)CC1 42270,N1(C(C(C)NC(CC)=O)=O)CC2CC(NC(c3coc(C(C)C)n3)=O)CC1C2 42271,c1(C(N=c2[nH]nc(-c3n(C)cnc3)s2)=O)cc2c(cc1Cl)NC(=O)C2 42272,N1(C(C2CC(C)(C#N)C2)=O)CC2CCCC2(CNC(c2ccccc2CO)=O)C1 42273,CCC(O)C(F)(F)C(=O)N1CC(CNC(=O)C(CC)C2CCOCC2)(OC)C1 42274,c1(C(=O)NCC(C)N(C(=O)CCCn2cncn2)CC)c(C)cccc1C 42275,C1(O)(CNC(C(CC)(C)F)=O)CCCN(C(=O)CN2CCCCC2=O)CC1 42276,N1(C(CC2(C)CC2)=O)C2CCC1CC(CNC(=O)CCCC1CCCC(=O)N1)C2 42277,C(CNC(C1(Cl)CC1(F)F)=O)(CC(=O)NCCc1cnn(C)c1C)OC 42278,C1(CC)(NC(c2cc(OC)cs2)=O)CCN(C(C2CCCC23CC3)=O)CC1 42279,CCCC(C)(C)CC(=O)N1CCC(N(C(=O)CCOCC2CCC2)C)C(C)C1 42280,CCCCC(CC)CC(=O)N(C1CC(NC(c2csnn2)=O)C1)C 42281,CC1C(C)N(C(=O)C=Cc2ccco2)CCN1C(=O)C=Cc1ccc(C2CC2C)o1 42282,N1(C(c2c(C)cnnc2)=O)CC(NC(=O)CCC2NC(=O)NC2=O)C(C)(C)C1 42283,C1(CC(=O)NC(C(C)NC(CC2C(CC)C2)=O)CO)(CO)CCCCC1 42284,Nc1ccc(C(=O)NC(CNC(=O)C(O)C2CC2)CC(F)(F)F)c(Br)c1 42285,c1(N(C)C)ccc(Br)c(C(N2CCC(NC(c3cnn(C)c3)=O)C2)=O)n1 42286,CCC(CC)C(=O)N(CCC(N1CCCC(O)C1)=O)CCCO 42287,C12(CCNC(c3cncc(C)c3)=O)CCC1CN(C(C1CCCN1C(N)=O)=O)C2 42288,C12(C(N3CC(C(=O)OC)C3)=O)CC1CCN2C(c1ccc(C(C)=O)o1)=O 42289,c1(C(=O)NC2C(NC(c3c(C4(C)CC4)cccc3)=O)C2)ccc2cc[nH]c2c1 42290,C(c1sc(Cl)nc1Cl)=CC(=O)NC1(COC)CCN(C(C23CCCC2C3)=O)C1 42291,N1(C(C2C(C)OCC2)=O)CCC(NC(c2c[nH]cc(Br)c2=N)=O)C(C)(C)C1 42292,c1(C(=O)NCC(C)N(C(c2ncn(C(C)C)c2)=O)C)ccc2c(c1)COC2(C)C 42293,CC(C)C(CCNC(C1(c2ccccc2)CC1(F)F)=O)NC(c1cncc(O)c1)=O 42294,Cc1cc(C(=O)NCC=CCNC(c2ccc(CCC3CC3)cc2)=O)nc(O)n1 42295,C1(c2n(-c3ccc(NCC4CC(C)C4)cc3)nnn2)(OC)CCCN(C2CC2)C1 42296,c1(NC(C2C(C(=O)NCCc3ccccc3O)C2)=O)cc2ccccc2cc1O 42297,c1(CNC(C2(N(C)C)CCC2)=O)ncccc1CNC(=O)CCc1ccsc1Cl 42298,C1(N(C(C=Cc2n(CC)ncc2)=O)C)CCCN(C(=O)CC2CC2C2CC2)CC1 42299,CC(CC(=O)N(C1CC(NC(c2sc(Br)cc2Cl)=O)C1)C)C(F)F 42300,C1(C(C(=O)N(CC(C)NC(=O)CSC(F)F)C)OC)CCOCC1 42301,C(C(=O)C(C)=O)OC1CCN(C2CCN(C(CC)=O)C2)C1 42302,N1(C(c2c(COC)con2)=O)CCC2CN(C(C3(C(=O)OC)CC3)=O)CC2CC1 42303,C(CN=c1[nH]c(=NCC2CCOCC2)[nH]c2c1CSC2)c1c(F)ccc(Cl)c1 42304,c1(C(=O)NCC2CC(NC(c3ccc(COC)o3)=O)C2)cnc(O)c(Cl)c1 42305,c1(OC)cnnc(C(=O)N(C)CCOC2(CN)CC2)c1 42306,N1(C(c2cc(C)[nH]c2C)=O)CCN(C(C2(F)CCS(=O)(=O)C2)=O)CC1C1CC1 42307,c1(C(N2CCCC(CC)C2)C(=O)NCc2nnn(C)n2)cc(Br)c(Cl)cc1OC 42308,Cc1ccnc(C)c1C(=O)OCCCOCC1CC1c1cnn(C2CC2)c1 42309,c1(C(=O)NC2C=CCN(C(C(C)OCCC=C)=O)C2)nc2c(s1)COCC2 42310,c1(C(C(=O)N(C(C)C)C)NC(COC(=O)OC(C)(C)C)C)cnc(O)nc1O 42311,C(=O)(NNC(=O)CNC(c1cccc(F)c1)=O)NCC1(O)CCC(C)C1 42312,N1(C(CCCn2cc(CCN(C)C)nn2)=O)CCCC(n2ccnn2)CC1 42313,c1(CNC(C2CC(CCC)C2)=O)cn(C2CCN(C(c3cnc(Cl)s3)=O)C2)nn1 42314,C(=O)(C(C)S(C)(=O)=O)NCC(C)(C1CCC1)NC(Cc1cc(C)n(C)n1)=O 42315,C1(C(N2CC(NC(C3C(C)(C)C3)=O)C(F)C2)=O)CC2(CCCO2)C1 42316,c1(C(=O)NCC2=CCCN(C(C3OCCN(C)C3)=O)C2)n[nH]c2ccccc12 42317,c1(NC(C)=O)cnc(O)c(C(=O)NCC2CCC2NC(C2(C)CC3CC3C2)=O)c1 42318,C1(NC(c2cc(CC)on2)=O)CC2(C1)CC2NC(=O)C(O)C(C)C 42319,CCC(C)C(C(=O)N(CCN1CCCC1)CC)NC(=O)NC1CCCO1 42320,Cn1cc(OCC(N2CC(C)(NC(=O)CCc3cscn3)C2)=O)cn1 42321,CS(=O)(=O)C1CN(C(=O)C=Cc2cnccn2)CC1NC(=O)C(=O)NC1CC1 42322,c1(CN(C)C)ccc(C(N2CCCC(CNC(=O)C=CBr)C2)=O)cc1 42323,c1(OC)cnc(C(N2CC3C(CNC(=O)C=Cc4ccc(Cl)s4)C3C2)=O)c(F)c1 42324,c1(C(N2CC(C)(C(=O)NC(CCC)CO)C2)=O)cc2cnccc2nc1C 42325,c1(C(N2C(CNC(c3c(OC)ccs3)=O)CC2)=O)cc(C(F)(F)F)cc(O)c1 42326,C(C1CN(C(=O)CN2CC3CC3C2)CC1C(=O)NC1C2CCCCCC12)=CC 42327,c1(C(=O)NCC2CC(COC)CN2C(=O)Cc2cncnc2)cccn(C)c1=O 42328,CCCCCCCCCCS(=O)(=O)N1CCCC(C(=O)Nc2ccsc2CC)CC1 42329,N1(C(CCC(=C)Cl)=O)CC(NC(c2n[nH]c3c2CC2CC32)=O)CC12CCCCC2 42330,C1(=CC(=O)NC2(CCCNC(CC3C(CC)C3)=O)CC2)CCOCC1 42331,N1(C(c2cc(COC)[nH]n2)=O)CCCC1(C)CNC(=O)C#CC1CC1 42332,C1(C2CCCCC2)(C(=O)NC(CC(C)NC(c2cc(OC)no2)=O)C)CC1 42333,N1(C2CCN(C(C(C)(C)OCC)=O)C2)CCC(NC(=O)C=Cc2cocn2)CC1 42334,C1(C(C)NC(C2CCC(C(=O)OC)O2)=O)CCN(C(c2cncnc2C)=O)CC1 42335,c1(C(c2nnnn2CC(F)F)NCC(C)(C)SC)cnn(C)c1C 42336,C1(OCC(=O)NC(C2CCCN2C(=O)C=Cc2c[nH]cn2)C)CC(F)(F)C1 42337,N1(C(c2cc(C)c(Cl)cc2)=O)CC2CCC(C1)N(C(=O)CCC(F)(F)C(F)F)C2 42338,c1(CC(=O)NCC(CNC(=O)C(=CC2CCCC2)C)OC)ccccc1SC 42339,Cc1c(-c2cn(CCCC(=O)N(CC(N)=O)C)nn2)c(=O)oc2ccc(O)cc12 42340,C(=O)(CCCCCCN=[N+]=[N-])NC1C(C)CN(C(=O)Cc2csnn2)CC1 42341,N1(C(C(CSC)O)=O)CCC2(CCCCC2NC(c2ncc(F)cc2F)=O)CC1 42342,c1(CCNC(C(=O)N(C(c2c(C)cccc2)C)C)=O)ccc2c(c1)CC(C)O2 42343,c1(C(=O)NCc2cccc(NC(C3CC(=O)NCC3)=O)c2)ncnc2[nH]cnc12 42344,N(C(=NCCN1CCOCC1)NCC1CCC(F)C1)CC1(CS(C)(=O)=O)CCC1 42345,C#CC1(NC(=O)C(O)CCNC(c2cc(C)no2)=O)CCOC1 42346,N1(C(C(CCC)OCC)=O)CCN(C(c2sccc2CC)=O)CC(C)(C)C1 42347,C1(CNC(c2scc(C(N)=O)c2)=O)CCCN(C(=O)C(=O)NCC(F)F)C1 42348,C1(C)(C(=O)NCC(CN(C(=O)COC2(C)CCC2)C)(C)C)CCC(=O)NC1 42349,c1(C(N2CCCN(C(C(C(C)C)F)=O)CC2)=O)coc2cc(F)ccc12 42350,C(=O)(C1=CC2CC=CCC12)NCC1CN(C(CCc2n(C)ncc2N)=O)C1 42351,CCC(O)C(=O)N1CCC(N(C)C(c2cc(-c3ccc(Cl)s3)on2)=O)C1 42352,Cc1ccc(F)cc1C(N1CC2(CNC(c3cc(Cl)c(Cl)n3C)=O)CCC1C2)=O 42353,C1(NC(C2C(CNC(C(CC)(C)C)=O)CCC2)=O)CCCOC12CCC2 42354,C1(NC(C2CCc3ccnn3C2)=O)CC1C1CCCN(C(=O)C2=CCCCC2)C1 42355,c1(NC(c2nnc3ccccn23)CCC)nccc(=NCCCNC(C)(C)C)[nH]1 42356,C1(C(N(C2CCN(C(c3ncc(F)cn3)=O)CC2)CC#C)=O)CN(C)CC(C)O1 42357,CN1CC(O)CC1(C)C(=O)NC1CCCCC1CO 42358,C1(C2(O)CCN(Cc3ccccc3)CC2)(NCC2Cn3c(C)nnc3CC2)CC1 42359,C1(c2ncc(C)s2)CCCCN1CC#CC(C)(C)C 42360,C1(NC(c2cocn2)=O)Cc2ccccc2N(C(c2cocn2)=O)C1 42361,c1(C(=O)NCC2(O)CCCN(C(CC(C)F)=O)C2)cc(O)cc(F)c1F 42362,N1(C(C(C)OCOC)=O)CCC(C(=O)NCCc2cnnn2C)C(C)(C)C1 42363,N1(C(c2cc(F)c(F)cc2F)C(=O)NCC(F)F)CCc2cccc(Br)c2C1 42364,C1(C(=O)NCC2CCN2C(C2CCCC23OCCO3)=O)CCCC12CCOCC2 42365,C1(N(c2ccncn2)C)CCCN(C(C2CCCC(N(C)C)C2)=O)C1 42366,c1(C(N2CCC(NC(CC3C(C)C3)=O)C(C)(C)C2)=O)n[nH]c2ccc(F)cc12 42367,c1(NC(C(=O)NC2CCCC(CC(C)C)C2)=O)ccc(Br)c(Cl)c1 42368,c1(CC)nn(C)cc1C(=O)NC(C)(C)CC(=O)NCC(O)C(F)(F)F 42369,CCC(C)(CCC(C)C)C(=O)N1CCC(CN(C)CC2CCNC(=O)C2)C1 42370,c1(C(=O)NC2CC(CNC(C3C(CC)OCC3)=O)C2)cc(C)cc2c[nH]nc12 42371,C1(NC(c2n(C(C)C)ncc2)=O)C2CCC1CN(C(c1ccc(F)cc1Br)=O)C2 42372,c1(C(=O)NCCCC(C)(C)NC(C=CCC)=O)ccc2c(c1)C(=O)NC2=O 42373,Cc1cc(C(N2CCCC2CCNC(=O)CS(=O)(=O)N(C)C)=O)nc(O)n1 42374,CC(CC(=O)N(CCCNC(=O)CC1(C(F)(F)F)CC1)CCO)C1CCCO1 42375,O=C(CC1CC2CC1C2)NNc1ccc(Br)c(F)c1F 42376,Cc1ccc(OCC(N2CCC(CNC(C34CC(CF)(CO3)C4)=O)C2)=O)c(C)c1 42377,Cc1cc2[nH]c(C(N3CCC4(NC(c5nccc(Cl)c5O)=O)CC4C3)=O)cc2s1 42378,c1(N2CC(NC(C=C(C)Cl)=O)CC3(C2)CC3)nc2cc(F)ccc2o1 42379,c1(CN(CCC)C)ccc(C(=O)OCC2(O)CCCSC2)cc1 42380,CCCC(CC)C(=O)NCC1(C)CCN(C(C2(CC3CC3)CCOCC2)=O)CC1 42381,C(=O)(C(F)C(F)(F)F)NC(CC)CNC(=O)COCc1ccncc1 42382,CC1(C)CC(NC(=O)C(C)(F)C(C)(C)F)CCN(C(c2c(O)cccc2F)=O)C1 42383,Cc1nc(C(=O)NCC2(C)CCN(C(=O)Cc3cnc(C)s3)C2)c2ccnc-2[nH]1 42384,c1(N2CCN(C(=O)Nc3cccc(F)c3)C3C2C3)ncnc2sccc12 42385,C1(NC(C(COC)OC)=O)CN(C(c2ccccc2OC(F)(F)F)=O)CCC1O 42386,C12(CC(=O)NCC3(F)CC(CNC(c4ncccn4)=O)C3)CCC(CC1)OC2 42387,c1(C(=O)NC2CC(CNC(C(CCC)C)=O)C2)ccc2nc(O)cn2c1 42388,c1(C(N(C)CC2N(C(C(C)(CO)OC)=O)CCC2)=O)cc2c(cn1)COCC2 42389,c12cc(OC)c(c(Cc3cnc[nH]3)c1)CN1CC3CC(C1)N23.CO 42390,C1(C(N(CCCNC(c2cn(C)nc2C(C)(C)C)=O)C)=O)CCOC(=O)CC1 42391,CC(C(=O)NCC1(F)CN(C(c2ccc(SC(F)(F)F)s2)=O)C1)S(N)(=O)=O 42392,c1(C(N2CC(COC)(NC(=O)CC(C)SC)C2)=O)cccc2c1COC2 42393,N1(C(CC2CC(=O)C2)=O)C2CCCC1CC(NC(C13CSC(C1)C3)=O)C2 42394,c1(C(=O)NCCN(C(=O)CN2CCC(C)C2)CCOC)nccc(Br)c1C 42395,C1(NC(CNC(C(c2ccccc2)C)=O)=O)CC(C)(C)C12CC2 42396,CCCCC(O)CC(=O)NC1CCCC(NC(=O)COc2c(F)cccc2F)C1 42397,C1(CCNC(CCC#C)=O)CC(F)(F)CN1C(=O)C=Cc1scnc1C 42398,Cn1oc(C(N2C(CNC(C34CC(CN3C3CC3)C4)=O)CC3CC23)=O)cc1=O 42399,N1(C(=O)NC2CN(C(CCCCC)=O)C2)CC(C)NCC1C 42400,C(=O)(C#CC1CCCCC1)NC1CC(C(=O)NC(CC=C)CC(F)F)C12CCC2 42401,C1(NC(C(C=CC)O)=O)CCC12CN(C(C1(C(N3CCCC3)=O)CC1)=O)C2 42402,C1(C(=O)NCc2c(C(=O)NCCCn3cccn3)nco2)(CC)CCCC1O 42403,n1(CCC)ccc(C(=O)NC2CCC2CNC(C2CNC(=O)N2)=O)n1 42404,Cc1ccc(C(=O)NC2(C(=O)NCc3ccc(CO)o3)CCCC2)c(O)n1 42405,C1(NC(=O)C(=CC2CCCCC2)F)CCN(C(=O)C(N2CCCC2)C2CC2)C12CC2 42406,NS(=O)(=O)C1CN(C(=O)NCNC2COCCC2(F)F)C2(CCC2)C1 42407,CC1CC2CN(C(c3cnc4[nH]cncc3-4)=O)CC2N1C(=O)Cc1cn[nH]c1 42408,C1(C)(C(c2n(CC(=C)C)nnn2)NCCc2cnoc2)CCCC(F)(F)C1 42409,c1(C(=O)NS(=O)(=O)CCC2CCCOC2)cccc(C(F)(F)F)c1 42410,c1(CC(=O)NC2CCN(Cc3cn(CC(CC)O)nn3)C2)c(F)cc(Br)cc1F 42411,c1(C(=O)NC(C2CCN(C(C(CC#C)(C)C)=O)C2)(C)C)ccc2c(O)n[nH]c2c1 42412,C(CC(=O)N1CCOC(CC(C)C)C1)(C(F)(F)F)NC(C(CCCC)N(C)C)=O 42413,c1(OC)cccc(OC)c1S(=O)(=O)NC1C2CN(C(c3csc(Cl)n3)=O)CC12 42414,C1(N(CC)CC2CC2)CCN(C(=O)C(=O)NC)CC1.c1(C2C(=O)N2)ccnn1C 42415,C(=O)(CCCC(F)(F)CO)N(C)CC1(O)CN(C(C2C(C)OC(=O)N2)=O)C1 42416,CCC(CNC(=O)C(C)N(C)C)(CC)NC(=O)CC1(OC)CCC1 42417,c1(CC)cc(C(=O)NC2CC23CCN(C(=O)CCC2CC(OC)C2)C3)ccc1F 42418,Cc1ccc(C2(CC(N3CCN(CC4CCCS4(=O)=O)CC3)=O)CC2)cc1 42419,c1(OC)ccc(CN2CCN(C(C3CC3C)=O)C(C)C2)nc1Cl 42420,c1(C(N2C(C)CC(NC(C3CC34CCC4)=O)C2)=O)cccc2cc(O)ccc12 42421,C1(CC(=O)NC2CC=C(C)CC2)N(C(c2csc(F)c2)=O)CCC1(C)C 42422,N1(C(c2c(C)n[nH]c2)=O)Cc2cccc(CNC(c3cc(F)ccc3Cl)=O)c2C1 42423,Cc1c(CN2CCC(SC(C)(C)C)C2)occc1=O 42424,C(=O)(C(c1cccs1)NC(=O)C(C)N1CC(C)C1)NCC(=O)OCC 42425,N1(CC(C)C)CCCC(C(=O)NCC(F)CNC(=O)Cc2cccc(C(C)C)c2)C1 42426,C1(NC(C2C(C)CCN2C(C2C3CCCC23)=O)=O)CC2(C1)CC(C)(C)C2 42427,C(C(F)(C(=O)NC(COCC1CC1)CC)C(C)C)NC(c1c(CC)nco1)=O 42428,c1(C(=O)NCC(C2CCC2)NC(c2c(C(C)(C)C)ncs2)=O)cc[n+]([O-])cc1 42429,N1(C(c2cnn(CC)c2Br)=O)CCC(NC(=O)Cn2ccc(C)n2)CC1C 42430,C12(C(=O)NC3(SCC)CC3)COCC1CN(C(=O)C(C1CC1)OCC)C2 42431,C(CCCCCN(C)C)NC(C(C1CCCO1)NC(c1c(C)occ1)=O)=O 42432,c1(C(=O)NCC(C2CCOC2)NC(c2ccon2)=O)snnc1-c1ccccc1 42433,C(=O)(C(C)(C)C(C)C)NC(c1sc(C(=O)NCC(CSC)OC)c(C)n1)C 42434,c1(C(N(C2CCN(C(C(Br)=C(C)C)=O)C2)CCO)=O)cnn2c(N)ccnc12 42435,C1(C(=O)NC2CCN(C(=O)NC)C2)CC1C1CCN1C(=O)CSc1nc[nH]n1 42436,C(=O)(C(O)CCCNC(c1cnnn1CC)=O)N(CCO)CC 42437,N1(C(c2c(CCC)nco2)=O)CC(C)C(NC(=O)C2=CCCCCC2)C(C)C1 42438,N1(C(c2n(C)nc(C3CC3)c2)=O)CCCC(CNC(c2c[nH]c(Br)c2)=O)CC1 42439,c1(-c2nnc(N(CCC)C)n2CC(=O)N(C)C)cc(Cl)ccc1OCC 42440,Cc1c(C(N2CC3CC(C2)N(C(=O)C(C)C#N)C3)=O)cc(Br)cc1Cl 42441,N1(C(C(CCC#C)O)=O)CCCN(C(=O)CCCc2cccs2)CC1CO 42442,C(=O)(C1=CC2(CCOC2)C1)N1CC(NC(c2c(C)nc(O)[nH]2)=O)C(C)C1 42443,C(=O)(C1=CCCOCC1)N1CCCC(CC=C)(NC(=O)Cc2cnn(C)c2C)C1 42444,c1(C(C)Nc2cnccc2-c2ncsc2C2CCC(=O)NC2)cc(C)cc(F)c1 42445,C=CC1(CC(=O)N(CCO)CC2CC2)CN(C(=O)C(C)(C)n2cncn2)C1 42446,C1(CC)CN(C(c2ccc(C)n2C)=O)CCN1C(c1cc(Cl)cnc1C)=O 42447,Cn1nc(C2CC2)cc1C(=O)Nc1cccc(NC(c2cc(C3CC3)no2)=O)c1 42448,CC(CC1CC1)C(=O)N(CCCOCCNC(C1(C2CCCO2)CCC1)=O)C 42449,N1(C(C(N(C(=O)CCCc2ncco2)C)C2CC2)=O)CCC12CCCC2 42450,N1(C(c2n(C)nc(O)c2)=O)CCC2(CCC2CNC(=O)COC2CCCC2)CC1 42451,C1(C(=O)NCC2NCCC(C)C2)Cc2ccccc2C1C 42452,Cc1cc(C)c2cc(C(N3CC(F)CC3CN(C(=O)C(C)N(C)C)C)=O)sc2n1 42453,C=CC(C)(CCOC)C(=O)NC(CNC(=O)C(C)C(=O)OCC)CO 42454,c1(OC)cc(F)c(C(=O)NCC2CC(C)N(C(C3CC(=C(C)C)C3)=O)C2)cc1N 42455,C1(C)(C(N2CCCC(C(C)NC(=O)CN(C)CCO)C2)=O)CCC(C)C1(C)C 42456,c1(C(=O)NC(CCC)CNC(=O)C(F)Cc2ccccc2)nccc(C)c1N 42457,C1(CC)CC(C)CN(C(=O)CC2CC(NC(=O)CCC(C)CC)C2)C1 42458,O=C1CC2CC(C(N3CC4(C3)CN(C(=O)CCCn3ccnn3)C4)=O)C1C2 42459,Cc1nc(O)nc(O)c1CCC(N1CCN(c2ccc(C#N)nn2)CC(O)C1)=O 42460,c1(CC)cc(C)c(C(=O)N(C2CN(C(=O)Cn3cc(CO)nn3)C2)C)o1 42461,Cc1nocc1CC(=O)N(CCCNC(C1CCCN1C(=O)NC1CC1)=O)C(C)C 42462,C1(NC(CCOCCOC)=O)CC2CCC1N2C(=O)CC1CCCCC1(C)C 42463,C(=O)(C(C(C)(C)C)n1ccnn1)NC1CCC(NC(c2nn(CC)nc2C)=O)C1 42464,C1(NC(C(C)=C(C)C)=O)CCN(C(=O)CCOCC2CC2)CC12CCC2 42465,S(=O)(=O)(c1cccnc1NCC1SCCc2ccccc21)NCCC(C)O 42466,c1(CC)ccc(F)c(C(=O)NCC2CN(C(=O)CC3CCCC3)CCCO2)c1F 42467,C=CCC(CC(=O)N(C)CCOCC)NC(C1CCCCS1)=O 42468,C(CC1=CCN(C(C23CCC(O)(CC2)CC3)=O)CC1)NC(C1(C)CC1(F)Cl)=O 42469,C(=O)(C(C)C(C)NC(=O)C(N)=O)N(CC=C)C(C)C 42470,C1(C)(NC(CCN(C(CN(CC)CC)=O)CCCO)=O)CCC(=O)NC1=O 42471,c1(C(N(CCN(C(c2nnn(C)n2)=O)CC)CC)=O)cc([N+](=O)[O-])n[nH]1 42472,C1(C(=O)NCC2CC(OC)CN2C(=O)COC2CCC2)C2CCC1(C)C2(C)C 42473,c1(C(N2CC(SC)C(NC(=O)C(F)n3ccnc3)C2)=O)cc(C)cc(C)c1 42474,N1(C(COCCC)=O)CC2CC(NC(C3(C(C)C)COC3)=O)C(C2)C1 42475,N1(C(C=CCOCCOC)=O)CCOCC1CN(C)C(c1c(C)ncn1O)=O 42476,CCC(CC(=O)N1CCN(C)C(C(=O)NCCC2CCOCC2)C1)C(C)(C)C 42477,c1(C(N2CCCC(Cn3cc(C(CC)(C)O)nn3)C2)=O)c(C)[nH]c2ncccc12 42478,C1(NC(C(C=C)(F)F)=O)CC2CC1CN(C(=O)C(CO)OC)C2 42479,CC1CN(C(c2csc(F)c2)=O)C(C)CN1C(c1ccnn1CCF)=O 42480,CCCC(CNC(=O)C=CC1CCOCC1)C(=O)N1CCC(c2cnn[nH]2)C1 42481,C1(CNC(c2c(OC)cnnc2)=O)CC(C)CN(C(=O)Cn2nc(C)cc2C)C1 42482,N1(CC(=O)NC(C(=O)NCCC(=O)OC)(C)C)CCC(F)CC1 42483,CCC(C)(CC)C(=O)NCC1(C)CCC(NC(=O)COCC(C)(C)C)C1 42484,CN1CCCC(CCC(=O)NC2(CNC(C3CSCCS3)=O)CC2)C1 42485,C(=O)(CCCCCCCSC)NC1C(NC(c2cccc(CC)n2)=O)CCC1 42486,N1(C(C2(OC(C)=O)CC2)=O)CCC2(CC1)CC(C)N(C(=O)CCC1CCCO1)C2 42487,c1(COCC(=O)NC2CC(C)(NC(C3CCCCO3)=O)C2)cccc(C(F)F)c1 42488,N1(C(c2c(=O)ccn(C)c2)=O)CC2CCC(C1)C2CNC(c1ccn(C)c1)=O 42489,c1(NC(=O)Nc2ncn(C)n2)cc(F)ccc1C(N1CCC(CO)C1)=O 42490,CC1(C)C(C(N2CC3CC(NC(=O)CC4CC=CC4)C2C3)=O)CCS1(=O)=O 42491,c1(C(=O)NC(C(C)NC(CCc2c(C)ncs2)=O)CO)ccn2ccccc12 42492,C1(C2(O)CN(C(C3CC3CC(C)(C)C)=O)C2)(CNC(C2CN(C)C(=O)C2)=O)CC1 42493,C#Cc1cccc(CC(=O)NC2CN(C(C3COCC3C(N)=O)=O)CC2OC)c1 42494,N1(C(c2c(C)nc(O)cc2)=O)CC2(C(=O)NC(C)C(F)F)CC1CCO2 42495,C1(C(N(C2CCN(CC)C2)C)=O)CC2CC2N1C(c1cc(O)n(CC)n1)=O 42496,N1(CC)CCC(N(C(=O)C(Cc2ccoc2)NC(=O)COCCN(C)C)C)C1 42497,CC#CCCC(=O)NC(c1ccccc1)CNC(c1[nH]cnc1C)=O 42498,C(=O)(C(C)C(O)CCCC)N(C1CC(C(=O)NCCC(CCC#C)O)C1)C 42499,n1(CC)nc(C)cc1C(N1CC2C(C1)N2C(=O)Cc1csc(C)n1)=O 42500,Cc1ccc(CC(=O)NCC(O)CCNC(C2(N3CCOCC3=O)CC2)=O)cc1 42501,C1(C(C)NC(c2c(C)nc[nH]2)=O)CCCN(C(c2ccc(C3CC3)nn2)=O)C1 42502,C1(C(=O)OC)C(F)(F)C12CC(C(=O)NC(C)(CNC(c1cc[nH]n1)=O)CO)C2 42503,c1(C(N(CC(CC)NC(c2n[nH]c(C)c2Cl)=O)CC)=O)ccc2nncn2c1 42504,c1(NC(C(N2C(CC)C(C)CC2)c2occc2Br)=O)c(C)cc(C)cc1C 42505,C1(N(C(c2cscc2OC)=O)CC)CCCN(C(=O)C(C)=CC(C)(C)C)C1 42506,S(=O)(=O)(c1ccc(C#N)cc1Cl)Nc1c(F)ccc(OC)c1 42507,C(=O)(C(CC)C(C)O)N(C1CCC(NC(c2c(CC)nco2)=O)CC1)C 42508,c1(CNC(=NCCOCC)NCc2ccoc2)nn(C)c(C)c1S(N)(=O)=O 42509,C1(C(=O)NCC2C(C)(C)COC2)CCC2(CC2)N1C(c1cc(C2CC2)no1)=O 42510,N1(C(C2N(S(C)(=O)=O)CC2)=O)CCC2(CCN(C(c3cc(Cl)c[nH]3)=O)C2)C1 42511,n1(CC)c(C(N2CC(C)C2C(=O)N(C2CN(C(C)C)C2)C)=O)cnc1O 42512,C1(C(=O)NCc2c(C(=O)NCC(C(C)O)C)con2)CC1C1CCC1 42513,c1(NCc2cnc(CC)[nH]c2=N)cc(=NC2CCCN(C)C2)[nH]c(CC)n1 42514,N1(C(c2c(C)nccc2)=O)CCC(C)C(NC(=O)CC2CCCC(F)(F)C2)C1 42515,n1(CC(=O)NC2C(NC(C(C)OCCOC)=O)CCC2)ncccc1=O 42516,C(=O)(C#CC1CCCO1)N1CC(CNC(Cc2[nH]c(=N)sc2)=O)C(C(F)(F)F)C1 42517,Cc1ncn(C)c(=O)c1C(=O)NCCN(C(=O)CNC(C1CCC1)=O)C 42518,C(=O)(C(CC(C)(C)C)OC)N1C(C(=O)Nc2c(CC)n(C)nc2)CCC1 42519,N1(C(C(C)C(C)(C)C)=O)CC(NC(=O)CN2CCCNC2=O)C(S(C)(=O)=O)C1 42520,Cc1nn(C)cc1C1CCCN1C(=O)CCCn1cc(-c2cccc(CO)n2)nn1 42521,c1(C(=O)NCCC2(OC)CN(C(C3C(C=C)C3)=O)C2)cc(OC)nc(Cl)c1 42522,c1(CNC(C(CNC(C2CCCN2C)=O)OC)=O)cnccc1Cl 42523,CCC(C)C(C)C(=O)N1CCCC(CNC(c2c(Cl)n[nH]c2C2CC2)=O)C1 42524,C(=O)(C(CN(C)C)NC(C1CCCN1C1CC1)=O)N(CCNC(C)=O)C 42525,C1(C(N2C3C(NC(CC4CCN(C)C4)=O)C(CC3)C2)=O)CC(C)(C)CC(C)(C)C1 42526,Cc1cnccc1C(C)C(=O)NCC(C)(O)CNC(=O)CCc1cccnc1 42527,CCN=C(NCc1nccn1CCc1ccco1)N1CCOC(C(F)(F)F)C1 42528,C1(NC(COc2cn(C)nc2)=O)CCN(C(=O)C(C)(C)C2CCC2)CC1F 42529,C(=O)(C(CCSC)OC)N1CC(CC(=O)NC2C(CC)OCC2)(OC)C1 42530,c1(-c2c(F)ccc(CN(C)C)c2)cccc2c(NC3CC3)cccc12 42531,N1(C(CSS(C)(=O)=O)=O)CCC2CN(C(=O)COCC3CCCO3)CC12 42532,c1(CC)nc(=N)[nH]c(=NC(C)C2CN(C(C3CC(n4ccnc4)C3)=O)CCO2)[nH]1 42533,C#Cc1cnn(CC(N2CCCCC2CCCNC(=O)C(C)C(C)O)=O)c1 42534,C=C(F)CN=c1[nH]c(N(C)CCOc2ccccc2)nc2c1CCC2 42535,c1(N(C)C)cccc(-c2cnc(NC(=O)N(CCO)Cc3nccn3C)[nH]2)c1 42536,C1(CC)(CNC(=O)C(C2CCC2)NC(c2csnc2C)=O)CCOCC1 42537,c1(C(=O)NCC2(CNC(c3c(OC)c(=O)cco3)=O)CC2)nc[nH]c2ncnc1-2 42538,CC(=O)CCCCCCC(=O)N1CCN(C(C2CC3CC3C2)=O)CCC1C 42539,CC12CSCC1CN(C(=O)C(c1ccccc1)NC(c1cnc(O)o1)=O)C2 42540,N1(CN(C(CC(C)NC(c2ccccc2)=O)=O)C)C(=O)c2ccccc2C1=O 42541,C1(C(C)C)CN(C(c2ccnnc2O)=O)CCN1C(c1cc2[nH]ccc2s1)=O 42542,C1(NC(CCC=CC(C)C)=O)CC2C1CCN2C(=O)CC(C1CCC1)C1CCC1 42543,N1(C(C(CC)N(C)C)=O)CC2(CCN(C(=O)Cn3ncnn3)CC2)C2COCC12 42544,C1(C)(C(=O)NC(C(=O)NCc2snc(CC)n2)CC2CC2)CCC(O)CC1 42545,C1(C(N(CCCC)C2CC2)=O)CN(C(C2CC23CCCC3)=O)CC1C1CC1 42546,Cc1nsc(C)c1C(=O)NCc1cc(C(N2CCCC2CC2CCC2)=O)n[nH]1 42547,C(c1cc(F)cc(F)c1)=CC(N1CCN(C(C2CC2F)=O)C(CC2CC2)C1)=O 42548,CN1CC(C(=O)N(CCCOCCNC(c2ccc(CCF)cc2)=O)C)CC1=O 42549,C1(C)(CC)C=C(C(=O)NCC2(C)CCN(C(c3c[nH]nc3F)=O)CC2)C1 42550,c1(C(=O)NCC(C)(C2CCC2)NC(CN(C(=O)OC)C)=O)cc2ccnn2cn1 42551,c1(OC)cc(C(C(=O)NC2CCCO2)N(C)C)cc(F)c1ONCC1CCC1 42552,N1(C(C2(C=C)CCC2)=O)CCCCC1C(C)NC(=O)CCCCNC(N)=O 42553,N1(C(c2n(CC)nnc2)=O)CCC2(CCC2NC(c2cccc(F)c2C)=O)CC1 42554,C1(C(N(C(CCNC(C2(NC(C)=O)CCCC2)=O)C)C)=O)CCS(=O)(=O)C1 42555,C=C=CC(C)C(=O)NCCOCCOCCNC(C1(C#N)CC(C)C1)=O 42556,N1(C(C(=O)NC(CC)CN(C(=O)Cc2nc[nH]n2)CC)C)CCCCCC1=O 42557,c1(C2(C)CC(OC(C(c3ccccc3F)OC)=O)C2)cccc(Cl)c1 42558,c1(C2C(CN=C(NCc3nnn(C)n3)NCc3ccccc3)C2)c(F)cccc1F 42559,C1(CC)CCCCC1OCC(=O)NC(C1CCN(C(=O)C(=O)NC)C1)C 42560,C12(NC(CCc3n(C)ccn3)=O)CCC1CN(C(=O)CSC1CCOC1=O)C2 42561,c1(SCC(N2C(C)C(NC(C3CN(C)C3)=O)CC2)=O)ccc(C#N)cc1 42562,C1(C(N2CC(C(C(=O)NC3CCOCC3)OC)C2)=O)Cc2nccn2C1 42563,n1(CC(=O)Nc2c(C)cc(C(F)(F)F)cc2)nc(CN)c2c1CCC2 42564,c1(C(=O)NCC2CCN2C(C23CC(CO2)C3)=O)nc(Br)c2ccccn12 42565,C1(NC(c2cccc(C#C)c2)=O)CN(C(=O)C(C)SC(F)(F)F)CC12CCC2 42566,c1(C(=O)NC(C(C)NC(c2nc(OC)nc(O)c2)=O)CO)c(F)cc(N)cc1F 42567,N1(C(C2(NC(C(COC)C)=O)CC2(C)C)=O)CC(O)(C2CCC2)C1 42568,N1(C(C(C2CCCCC2)C)=O)CCC(CNC(=O)C(O)C2CCC2)C1(C)C 42569,C=C1c2ccccc2C(=O)N1CC(N1CC2(C1)CN(C(C1NC(=O)OC1C)=O)C2)=O 42570,Cc1cccc2c(CC(N3CC4CC4(NC(c4c(Cl)cnn4C)=O)C3)=O)c[nH]c12 42571,N1(C(Cc2c(C)cnn2C)=O)CC2(CC(CC(=O)NCC(C)(O)CO)C2)C1 42572,c1(OCC(=O)N(C)CC2CCN(C(CC(=C=C)C)=O)CC2)cc(C)ccc1F 42573,c1(C(N2C(CNC(C(CC)(C)CO)=O)CCCCC2)=O)onc2ccccc12 42574,N1(C(CC(=O)OC)=O)CCC(CC(=O)NCc2nccn2C(C)C)CC1 42575,C1(OC)CCCC(CC(=O)NC2CC(C)(NC(C3CCCN3C(C)=O)=O)C2)C1 42576,CCCC(CC1CCCC1)C(=O)N1CCC(O)(CNC(c2[nH]nnc2C)=O)CC1 42577,CC12CCN(CC1)CC2C(=O)NC1CN(C(=O)CCc2ccsc2)CC12CCC2 42578,C1(S(C)(=O)=O)(C(=O)NCC(CO)NC(Cc2c(C)ccc(C)c2)=O)CC(O)C1 42579,N1(CC(=O)NCCN(CCOC)Cc2cncc(OC)n2)CCCCS1(=O)=O 42580,N1(C(c2nc(Oc3ccc(Cl)cc3)ccc2Cl)=O)CCC2CC2(CO)CC1 42581,c1(NC(C)=O)cccc(C(N2CCC(Cc3ccc(C(C)C)cc3)CC2)=O)c1 42582,N1(C(COCCC=C)=O)CCC(C)(CCNC(c2ccc(OCCF)cc2)=O)C1 42583,C1(NC(CSCCC)=O)CCCN(C(=O)C(c2ccc(OCC)cc2)C)CC1 42584,C(=O)(CC(C(F)F)c1ccccc1)N(CCCN(C(C=CC=CC)=O)C)C 42585,c1(COC)nc(N2CCCC(N(C(=O)CC3(O)CCC3)C)CC2)cc(Cl)n1 42586,N1(C(C(F)=CCC)=O)CC(C)CCC1CNC(=O)COC1(C)CCC1 42587,c1(C(=O)NC(CC=C)CNC(c2c(Cl)sc(Cl)c2C)=O)cccc2nonc12 42588,c1(CNC(N(C(C2(OC)CCSC2)=O)C2CC2)=O)ccc(C)c2cccnc12 42589,c1(CC)cccc(F)c1C(=O)NC1(COC)CN(C(C2CCN2C)=O)C1 42590,c1(C(N(CCN(C(=O)C(F)C(C)C)CC)CC)=O)ccc2c(c1)COCCN2 42591,C=CC1(C(N2CC(CCNC(C3(CCF)CC3)=O)C2)=O)CCCCC1 42592,COn1cnc(C)c1C(=O)NCCCN(C)C(c1sc(Br)cc1C)=O 42593,C1(CC(=O)N(CC(=O)NC(C)CN(C)C)C)(NC(C)=O)CC1 42594,c1(C(=O)NC(CC)(CNC(C2(CO)CC2(F)F)=O)CC)cnc2c[nH]nc2c1 42595,Cc1nc(C(C)C)sc1C(=O)N(CCN(C(=O)COc1ccsc1)C)C(C)C 42596,c1(C(=O)NCCCOCCN(C(=O)C(O)C2CC2)C)csc(C2CC2)n1 42597,N1(C(C2(C(N(C)C)=O)CC2)=O)C2CCC1CC(NC(C1CC13CC3)=O)C2 42598,C1(C(N(CCO)CC)=O)CCOC1CNC(C1C=C(C)CS1)=O 42599,Cc1ncc(C(N2CCC(CCNC(=O)C(F)C(F)(F)F)CC2)=O)cc1N 42600,Cc1cc(C(=O)NC2CC(O)CN(C(=O)COc3cccnc3)C2)c(F)cc1N 42601,c1(C(=O)NC2C(CC)N(C(C3CCOCC3)=O)CCC2)cc(F)c(C)cc1N 42602,C12(CNC(c3ccc(CC)nc3)=O)CCCC1CN(C(C1CC(C3CC3)C1)=O)C2 42603,n1(CC(=O)NCC2N(C(CCCC=C)=O)CC(F)C2)nc2n(c1=O)CCCCC2 42604,C(C(=O)NCCNC(=O)C(c1ccc(F)cc1)(C)C)(C(C)C)NC(C)=O 42605,C(=O)(C(C)(C)CC(C)C)NCCOCCNC(C(CC)(O)c1ccccc1)=O 42606,N1(C(C=COCC)=O)CCC(n2cccn2)(CNC(C2CC2C(F)F)=O)CC1 42607,CC1(NC(C2CCC(P(C)(C)=O)C2)=O)CCCc2ccccc21 42608,c1(CC)ccc(C(=O)NC2CCCCC2CNC(=O)C(C)CSC(F)(F)F)cc1 42609,Cc1cc(O)cc(=O)n1CC(=O)NCC1CC(NC(=O)CCC2CCC(=O)N2)C1 42610,C(CC(=O)N(C)CC1CCOC1C)(CC(C)C)NC(C1C(CCC)C1)=O 42611,CCC(CC(=O)NCCCC(C)(C)NC(=O)C(CO)C(C)(C)C)C(C)(C)C 42612,C1(OC)(OC)CC(C)(CNC(c2cnn(CCO)c2C2CC2)=O)C1 42613,N1(C(CN2CCN(C)CC2)=O)CCC2CN(C(=O)C(C)(C)C3CCCCC3)CC12 42614,c1(C(N2C(C)(CNC(C(C=C)(C)C)=O)CCC2)=O)cccc2oc(C)nc12 42615,Cc1ccccc1COCC(=O)NC1C2CC1N(C(C1(C)CC(C)C1)=O)C2 42616,N1(C(C2(OC)CCC2)=O)CCC2C(CCN2C(c2cc(C)ncc2Cl)=O)C1 42617,Cc1cc(C(N2CC(C(=O)NCCSC(F)F)CCC2C)=O)nnc1C 42618,Cc1c(CNC(N2C(Cc3cccc(C4CC4)c3)CC3CC23)=O)cccc1F 42619,c1(SC)cc(N2CCC(C)(CNC(=O)Cc3ccoc3)CC2)nc(SC)n1 42620,N1(C(c2cc(CC)n(C)n2)=O)CCCC(N(C(=O)Cc2ccc(Cl)cn2)C)CC1 42621,C(=O)(C(C)CC(F)F)N(CCCNC(C(CC)(C)OC)=O)CCO 42622,c1(CN2CC3C(CNC(c4cc(C(F)(F)F)no4)=O)C3C2)ccc2ncnn2c1 42623,CCCCC(CNC(=O)C(CC)OC1CCCC1)NC(C1CC(F)C(=O)N1)=O 42624,c1(C(N2CC(O)(C(C)NC(C(CSC)C)=O)C2)=O)ccn2cccc2c1 42625,N(C1CN(C(=O)C(O)CC2CC2)Cc2ccccc21)C(c1c(C)nc[nH]1)=O 42626,C1(NC(C2CC(CCC)C2)=O)CCCC(C(N2CCSCC2)=O)CC1 42627,N1(C(CCC(=C)Cl)=O)CCC2(CC1)CC2CNC(c1sc(C)cc1OC(F)F)=O 42628,C1(N(C(=O)C(F)F)CC#C)CCN(C(C2(C(C)(F)F)CC2)=O)CC1 42629,N(C1CN(C(C2(C)CC=CC2)=O)Cc2ccccc21)C(c1cc(C)[nH]n1)=O 42630,C1(c2cn(CCNC(c3ccncc3F)=O)nn2)CC2CCC1O2 42631,c1(C(=O)NC(C(C)NC(CCC(=O)NCCC)=O)C)cc(C)c(C)nc1C 42632,c1(C(=O)NC2CC(CNC(CCOCCSC)=O)C2)c(NC(N)=O)cccc1F 42633,CC1CN(C(c2cn[nH]c2)=O)CC1CNC(C1CCNC(=O)C1)=O 42634,C1(N(C(C=CC(CC)=CC)=O)CC)CCCN(C(c2ccncc2CC)=O)C1 42635,CC1CC(C)(C(N2CC(CC(C)NC(c3csc(Cl)c3Cl)=O)C2)=O)CC(C)O1 42636,CC(C)(C(=O)NCCC1CN(C(=O)COc2ccsc2Cl)C1)C(F)F 42637,c1(C(=O)NCC(=O)NCC(=O)NCc2nc(C)sc2)ccnnc1O 42638,c1(OC)ccc(C(N2CCC(CNC(=O)CC(C)OC)(OC)C2)=O)cc1F 42639,c1(NC(C(C)OCC)=O)cccc(NC(c2snnc2C(C)C)=O)c1 42640,N1(C(CC(C)(C)OC)=O)C2CCC1CN(C(c1cnoc1C)=O)CC2 42641,C1(CNC(C=CC(C)C)=O)CC(NC(c2coc(C3CCOCC3)n2)=O)C1(C)C 42642,C(=O)(C(C)CC(N)=O)N1CCCC(NC(c2c(C)c(C3CC3)[nH]n2)=O)C1 42643,N1(C(C(C)n2cccc2)=O)CC2CC1CC2CNC(=O)C(C)(C)c1cnn(C)c1 42644,c1(C(=O)NC(C(C)NC(CCOc2ccc(C)cc2)=O)C)cc(F)cnc1O 42645,N1(C(CCCC(C)=O)=O)CC2CCOC2(CNC(=O)C(C)C#N)C1 42646,c1(OC)cc(C)nc(N(C)CC2CCN(C(=O)CC(C)SC)CC2)n1 42647,C1(CC)C(C(=O)NCc2nc(CO)n[nH]2)CCN1C(=O)C(c1cncnc1)C 42648,C1(c2n(CC(=C)C)nnn2)(NCc2cc(Br)no2)CCC2(CCOCC2)C1 42649,Cc1cccc2cc(C(=O)NC3(CNC(C45CC(F)(C4)C5)=O)CCOC3)nn12 42650,c1(C(N2CC(O)(C(C)NC(c3nn(C)cc3Cl)=O)C2)=O)n[nH]c2c1CCCCC2 42651,c1(NC)ccccc1C(N1CCC(C)(CNC(=O)CCc2ccnc(Cl)c2)C1)=O 42652,CC(F)(F)CC(=O)N1CCN(C(=O)CCc2cnccn2)CC1 42653,c1(OC)nc(C(=O)N(C(C)CN(C(=O)C(C2CCCC2)OC)C)C)cc(O)n1 42654,CCC(C)C(C)CN=c1[nH]c(C)cc(=NCc2ccc3nn[nH]c3c2)[nH]1 42655,C1(N(C2CC3CC2CN3)C(=O)COCCOC)CCNCCC1C 42656,S(=O)(=O)(c1ccc(N2CC(C)C(O)C(C)C2)nc1)NCC(=C)CC 42657,N1(C(C2(C)CCN(C)C2)=O)CC2CCC(C1)N2C(c1cnn2ccccc12)=O 42658,C1(C)(N(C(=O)COc2ccn(C)n2)C)CCN(C(=O)CCc2cccs2)C1 42659,c1(C(N2CCCC(C)(NC(CN(C)C)=O)C2)=O)ccc2c(Br)nn(C)c2c1 42660,C#CC1(C(N2CCC2CC)=O)CCN(C(c2cccc(C)c2F)=O)CC1 42661,C1(CC(=O)NCCc2cc(C)ncc2)N(C(=O)C=Cc2ccco2)CCC1(C)C 42662,C1(NC(c2n(C)nnn2)c2ncc(-c3ccccc3)s2)C(=O)OC2CCCC12 42663,C(C)(C)(CC(=O)NCC1(F)CCC(NC(c2cc(OC)cnn2)=O)C1)OC 42664,c1(OCC)n[nH]c(C(=O)NC2CCCC2c2nc[nH]n2)c1Cl.c12c(cnn1C)SC2 42665,CCC1=C(C(=O)N2CC=CC2CNC(c2c(Br)noc2C2CC2)=O)CCCO1 42666,c1(-n2cc(C(N(CCCC)C(C3CCCC3)C)=O)nn2)ccc(C(=O)O)cc1 42667,N1(C(C(CCOC)C)=O)CCC2(C=C(C(=O)Nc3ccc(C)cc3OC)C2)C1 42668,C(C(=O)NOCCN1CCCC1=O)(C1CN(C(=O)Cc2cccc(O)c2)C1)OC 42669,Cc1cnn(CC(N2CCC2CNC(=O)CC2CCC(C3CC3)O2)=O)c1 42670,C#Cc1cncc(C(N2CCN(C(=O)C(C)(C=C)CC)CC2CC(=O)NC)=O)c1 42671,N1(C(Cc2nc(CC)sc2)=O)CCCC(C(C)NC(=O)C=Cc2ccsc2)C1 42672,c1(C(N2C(C)CN(C(=O)Cc3cnns3)CC2)=O)cc2c(nc1N)CCC2 42673,c1(-c2n(CC(C)(C)C)nc(CCC(F)(F)F)n2)ccc2c(c1)C(C)(C)CO2 42674,Cc1ccc2oc(C(=O)NCC3(F)CC(CNC(=O)C(C)(O)C4CC4)C3)cc2n1 42675,C1(NC(c2cn(C)nn2)=O)CCOC12CCN(C(C1CC(F)C1)=O)CC2 42676,C1(NC(Cc2n(C)ncc2)=O)CCC12CCN(C(c1ncc(F)cc1F)=O)CC2 42677,CC(CO)CCCN=c1[nH]c(=NCC2CC3OC2C2CC32)c2sccc2[nH]1 42678,C(=O)(CC(C)CCC=C(C)C)NCC1CC(NC(c2cncc(OC)n2)=O)C1 42679,N1(C(c2ncc(OC)cn2)=O)CCC(C2CC2)C1CNC(=O)C=C1CCCC1 42680,N1(C(c2occc2Br)=O)CC(C2CCCCN(C(=O)C(F)OC(F)(F)F)C2)C1 42681,c1(NC(=O)CC2(O)CN(C(c3cc[nH]n3)=O)C2)ccc(Cl)c(Br)c1 42682,Cc1cccnc1CC(=O)NCCC1COCCN1C(=O)CO 42683,c1(C(=O)NCC2C(C(=O)NCC(COCC)C)C2)cccc2nccn12 42684,C1(NC(c2c(C)cccc2Cl)=O)COC2C(NC(C3CC(F)(CO)C3)=O)COC12 42685,c1(SC2COCCN2C)ccc(F)cc1.C12CCCN1C(=O)C1(CC1)CN(C)C2 42686,C(=O)(CC(C)CCCCC)N1C(C2CCN(C(COCC=C)=O)CC2)CCCC1 42687,CN1CC2(CC2)CC1C(=O)NCC1CN(C(=O)CNc2nccs2)C(C)(C)C1 42688,N1(CC(N2CCC(C(=O)NCCC(=O)OCC)C2)=O)CCCCC1C 42689,c1(NC2C(C)COCC2)nc(N(CCCS(C)(=O)=O)C)nc2c1cnn2C 42690,C1(NC(C(=CC2CCCC2)C)=O)CC1C1CCN(C(C2(C)CC2C)=O)CC1 42691,CCC(CC(=O)N1CCC2C(NC(=O)Cc3ccc(SC)cc3)C12)C(C)C 42692,C1(C(=O)NCC(C)(C(C)C)NC(Cc2c(C)noc2C)=O)C(O)C(=O)N(C)C1C 42693,c1(C(N2CC(NC(C3C(C)(C(F)F)C3)=O)C2)=O)c(C2CC2)nc2sccn12 42694,N1(C(c2c(CC)ccs2)=O)CC2=C(C1)CN(C(=O)C(c1ccccc1OC)O)C2 42695,Cc1ccc2[nH]cc(C#N)c(=NCc3c(F)cccc3Br)c2c1 42696,Cc1c(F)cc(C(N2CC3CN(Cc4ccc(O)c(I)c4)C3C2)=O)cc1Br 42697,c1(NC(CCNC)C)ncnc2sc3c(c12)CCCCC3 42698,Cc1n[nH]c(C)c1C(C)CC(=O)NCC(F)CNC(=O)CCC(F)F 42699,S(=O)(=O)(CCC(=O)NC)CNC(COC)=O.C1C(O)CN(C)C(=O)COCCN1 42700,C(c1ccccc1C)=CC(N1C(C)(CNC(CCSCCC)=O)CCC1)=O 42701,C12(C(=O)NCCC(=O)OCc3ccsc3)CC(CO1)N(c1ncccn1)C2 42702,CC(CN(C)C)CCC(=O)NCC(C1CCC1)NC(C1(CCN(C)C)CC1)=O 42703,CC1(C)CN(C(c2ccsc2Cl)=O)CCC1NC(=O)CCCC1CC1 42704,C1(C)(CNC(Cc2c(CC)con2)=O)CCCN(C(c2cc(OC)cs2)=O)C1 42705,CCCCC#CC(C)(C)NC(c1c(CNC(=O)CC2CC(C)C2)cnn1C)=O 42706,c1(CC(=O)NC2CCC(CCNC(CC=C(C)C)=O)C2)ccc2nn[nH]c2c1 42707,C1(C(N2CC3C(C(N4CC(CC)C4)=O)C3C2)=O)CCc2ccccc2C1 42708,N1(C(=O)NCC(C2COC(C)(C)O2)O)CCC(=C(Br)Br)CC1 42709,Cc1cccc2[nH]c(C(N3CCC(NC(=O)CCCc4cccs4)C3C)=O)cc12 42710,C(=O)(C(C)(F)C(F)(F)F)N1CCC(CN(C(C2(C)CN(C)C(=O)C2)=O)C)CC1 42711,N1(C(CSC)=O)CCCC(N(C(=O)CCc2nnc(C3CCCC3)o2)C)CC1 42712,C(c1nc2ccccc2s1)=C(C)COc1ccc(C)c(OC(F)(F)F)c1 42713,CC1(F)CC(C(=O)NC(C(=O)NCc2nn[nH]c2C2CC2)c2ccoc2)C1 42714,N1(C(CS(=O)(=O)N(CC)CC)=O)CC(OC)CC(NC(c2cn[nH]c2)=O)C1 42715,c1(NCCCCCCSC)[nH]c(=NC2CCC(C(F)(F)F)CC2)nc2sccc12 42716,N1(C(C(F)=CCC)=O)CCN(C(=O)CN2CC(C)(C)C2)CC1COCC 42717,C(=O)(C(C(C)C)C(C)C)NC1C2(CN(C(c3ccc(NC(=O)OC)cc3)=O)C2)C1 42718,C1(COC)CCN(C(c2csc(CNC(c3ccc(Cl)s3)=O)c2)=O)CC1 42719,c1(OC)ccc(C(=O)NC(C)CCNC(C2CCN(C)C2=O)=O)c(F)c1F 42720,C(CC1=CCCCCC1)NC(=O)CC1CCN(C(C2COC(=O)N2)=O)C1 42721,O=S(=O)(c1ccc2[nH]ccc2c1)NC1CCCNCC1F 42722,c1(C(=O)NCC(C2CC2)NC(C(CC=C)C(C)C)=O)ccn2cnc(C)c2c1 42723,C(=O)(CCCCCn1cc(-c2cnn(C(C)C)c2)nn1)N(C(C)(C)C)CCC 42724,C(=O)(C1=CCN(C(c2csc(CO)n2)=O)CC1)NC1(CC)CCCC1 42725,N1(CCC)CCCCC1C(=O)NC1CCC1NC(c1ccn(CCN(C)C)n1)=O 42726,C1(C(=O)NC2CC(NC(=O)Cc3ccon3)C2)COc2cc(Cl)ccc2C1 42727,N1(C(C(C=C)(C)CC)=O)CCC2(CCCN2C(C2CC(F)(F)C2)=O)C1 42728,c1(C(=O)NC(CNC(CN(C)CC)=O)CC(C)C)cnc2n1CCS2 42729,c1(CC(=O)NC2CC(C)(NC(C(C(C)(C)C)=O)=O)C2)ccc2ccccc2c1 42730,C1(c2cn(CC3N(C(=O)CCOC4CCC4)CCC3)nn2)CC2CCC1CC2 42731,C12(C(N3CC(CNC(C=C(C)C)=O)C(C(F)(F)F)C3)=O)CCN(CC1)S(=O)(=O)C2 42732,CC(C)(CC1CCOCC1)C(=O)NC1CN(C(=O)CCc2cocn2)C1 42733,n1(CC)cnnc1C(=O)NC1CC1CNC(=O)C(C)OCCOC 42734,c1(C(N2C(CNC(CCC#C)=O)C(C)(C)CC2)=O)ccc2c(c1)OCCC2 42735,N1(C(C2N(CC)CCC2)=O)CCC=C(C(=O)NCCN2CCNC2=O)C1 42736,c1(C(=O)NC2(CC)CCN(c3nnc(C(N)=O)s3)CC2)cccc2c1nnn2C 42737,C(=O)(C1CCc2ccc(OC)cc21)N1CCC(NC(C(CC)C(C)O)=O)C(C)C1 42738,c1(N2CCCC(=O)CC2)nc(NC2CCC3(C2)CC3(F)F)c2ccsc2n1 42739,C1(C(=O)NCCC(C)NC(C2CCC3CC2C3(C)C)=O)CCC2CCCCC2C1 42740,c1(OC)ccc(C(N2CCN(C(=O)C=Cc3cc(Br)cs3)CC2C)=O)c(OC)c1 42741,S(=O)(=O)(CCC(=O)NC1CN(C(c2ccc(CO)cc2F)=O)C1)NC(C)(C)C 42742,C1(OC)CC(NC(c2cc(C)ns2)=O)C12CCN(C(=O)Cc1cnc[nH]1)CC2 42743,C(=O)(CC(C)(C)CNC(=O)C(C)C)NCCn1c(C)cc(C)n1 42744,C1(C(=O)NC2CN(C(C(=O)NCCOCCCC)=O)C(C)C2)CCCC(=O)N1C 42745,C1(NC(C2CC2C2CCC2)=O)CC2CC1CC2C(N1CCC1C1CCCCC1)=O 42746,CC(C)C(C(=O)NCC(C)CNC(C1CC(C(N2CCOCC2)=O)C1)=O)NC=O 42747,N1(C(=O)CC2CCCOC2)CCC(S(=O)(=O)N2CCCC2)CC1 42748,N1(C(c2c(C)ccc(C)n2)=O)CC(C(N2CC(C(C)(C)C)C2)=O)C2(CCC2)C1 42749,c1(C(=O)NCCN(CCC)C(c2cnc(C(C)C)o2)=O)c(C)coc1C1CC1 42750,c1(COCC(=O)NC(CNC(CSCCCC)=O)C2CCC2)cnn(C)c1 42751,c1(NC(C(CN(C)C)NC(=O)CC2CC3C=CC2C3)=O)ccc(Cl)cc1O 42752,N1(C(c2nnn3c2CSCC3)=O)CC2(CCN(C(C3CC(=C4CC4)C3)=O)CC2)C1 42753,C1(CCC)(NC(C2CC(=O)NC(=O)N2)=O)CCCN(C(c2ccnc(C)n2)=O)C1 42754,Cc1nncc(C(=O)NC(CCN(C)C)C(=O)NCC(O)C2CCC2)c1C 42755,N1(C(C2ON=C(CC)C2)=O)CCN(C(=O)Cc2ccc3c(c2)CC3)C(C2CC2)C1 42756,C1(NC(COC)=O)COC2(CCN(C(c3ccc4c(C(=O)OC)n[nH]c4c3)=O)C2)C1 42757,c1(CCC(=O)NC(C)CN2CCC(F)(F)C2)ccc(Br)c(Cl)c1 42758,C1(C(=O)NC(C)CNC(=O)CC2(C#N)CCCCC2)CCc2n[nH]cc2C1 42759,C1(C)(COC)CC(NC(c2c(C)cnn2C)=O)CN1C(c1scnc1Cl)=O 42760,c1(CC(=O)NCC2(F)CCN(C(C3(O)CCSC3)=O)C2)cnn2ccccc12 42761,CCCCCCCC(=O)N(C)CC1CN(C(=O)CC2CC(C(F)F)C2)CCO1 42762,Cc1cocc1C(c1nnnn1CCCO)NCC1(C(N)=O)CCCC1.N(C)C 42763,c1(OC)ccc(C=CC(=O)NCCCCCCN(C(=O)CC(C)CF)C)cc1O 42764,N1(C(C(=O)NCCOC)C2CC2(Br)Br)CC2CCCC2(C(N)=O)C1 42765,C1(CCC(=O)NC(CNC(=O)Cn2ncc(Br)n2)CO)CC2CCC1C2 42766,c1(CCC(=O)NC(C)CNC(C23CCCC2C3)=O)ccc2ccccc2n1 42767,C(C(C)CN(C(=O)CCN(C(=O)C=CCl)C1CC1)C)NC(C1C(C(=O)OC)C1)=O 42768,C12CCCCC1N2.c1(NC(=O)CSc2cnco2)ncccn1 42769,c1(NC(c2c(COC)n(C)nc2)=O)nccc2[nH]ccc12.C(C(C)(C)CC1CC1)N 42770,c1(-n2c(C3CC3(c3ccccc3)F)nc(COCC)n2)cc(C)ccc1C 42771,C1(C(N(C2CCCC2)CC=C)=O)CCC(C)(C)N(C(C2CC2(F)Cl)=O)C1 42772,C(=O)(C(C(C)(C)NC(C)=O)c1ccccc1)N1CCN(CCCOCC)CC1 42773,c1(NC(N(C(CC(=O)OCC)Cc2ccccc2)C)=O)ccc(F)cc1F 42774,CCCC(C)CN=c1cc[nH]cc1S(=O)(=O)NC(c1nc(C)cs1)(CC)C1CC1 42775,c1(C(N(C(C2CN(c3cccc(OC)c3)C(=O)C2)=O)C)=O)cccc2nn[nH]c12 42776,N1(C(C2(NC(=O)CCC3OCCO3)CCCC2)=O)CCC2C(C1)C2(F)F 42777,c1(C(=O)OC)cc(C(=O)NCC2(NC(c3cscc3F)=O)CC2)n2c1COCC2 42778,C(C1=CCN(C(=O)CC2(C(F)(F)F)CC2)CC1)NC(c1cccs1)=O 42779,c1(C(CC)(C)O)cn(CCCNC(c2coc(C(C)C)n2)=O)nn1 42780,CC1(C)CC(O)CN(C(c2c[nH]nc2CCNC(C2CN(CCF)C2)=O)=O)C1 42781,CCC(C)(C)C(O)C(=O)N1CCCCC(C(=O)NC2CN(C(=O)C3CC3)C2)C1 42782,c1(N2CCC(CCNC(C(C(C)C)(C)O)=O)CC2)ncc([N+](=O)[O-])cc1C(N)=O 42783,c1(C(=O)NC(C)C(C)NC(=O)C(C)(C)CS(N)(=O)=O)cc2c(cc1Cl)NC(=O)C2 42784,c1(CC)cc(=NC(=O)C2CCN(C(=O)CN3CCC(C)CC3)CC2O)[nH]n1C 42785,c1(NC(C)=O)ccc(C(N2CCCCC2C(N2CC3CC3C2)=O)=O)cc1 42786,Cc1n[nH]c(C)c1CC(N1CC2C(CNC(=O)C(C)(C)C)C2C1)=O 42787,C1(C(=O)NC2CC(NC(CCc3onc(C(C)C)n3)=O)C2)CC(F)(F)C12CCC2 42788,N1(C(c2c(C)c(F)ccc2)=O)CCC2(CNC(c3cscc3F)=O)CCCCC12 42789,CC1CCC(CNC(C2CCCCC2)=O)CN1C(=O)COC1(C)CCCC1 42790,c1(C(C(=O)O)NC(=O)NC(c2nc(C(F)(F)F)cs2)C)cccc(Cl)c1 42791,c1(SCC)ncc(Cl)cc1C(=O)OCC(C(C)C)OCC1CC1 42792,C1(NC(C(CC)OCC)=O)CCN(C(=O)Cn2nnc(C3CC3)n2)CC(C)(C)C1 42793,C12(NC(C(CC#C)CC#C)=O)CCCC1(F)CN(C(=O)C(C)COCC)C2 42794,Cc1nnc2c(C(=O)NC(C)C(C)NC(c3ccncc3N)=O)cccn12 42795,c1(C(N(CCCN(c2nnnn2C2(C)CC2)C)CC)=O)cccc(C(F)(F)F)c1 42796,n12cc(nn1)C2.C(=O)(CCCn1cc(C)cn1)CN(C(CC1(CSC)CC1)=O)C 42797,C1(C(=O)NC(c2cccc(C)c2)CNC(C(C)=C2CCC2)=O)COCC1(C)C 42798,C(=O)(C1=CC2CC(C1)CC2O)NCC(CNC(Cc1c(F)ccc(C)c1)=O)CO 42799,S(=O)(=O)(c1ccc(F)cc1Cl)NCC(N1CCOCC2(COC2)C1)=O 42800,C1(C2CC2)(CNC(=O)CCN2CCCCC2=O)CCN(C(=O)C(O)C2CCC2)C1 42801,c1(OCC)ccc(C(C)NC(=O)CCC2(C)CC2)cc1F 42802,CC(CC(F)(F)F)C(=O)NC1CCN(C(=O)C=C2CCSCC2)CC1O 42803,c1(C(=O)NC(C)CN2CCCCC2C)cnc(Br)c(Cl)c1 42804,CCCC(C)(CCC)C(=O)N1CCC(CNC(=O)CN(C)C)(OC)C1 42805,c1(NCC#CC)cc(=NCC(C(C)C)c2ccnn2C)[nH]cn1 42806,C1(C(=O)NC(C2(C(N(CC)Cc3cccnc3)=O)CC2)C)CCN(C)CC1 42807,c1(-c2cn(C(C)C(N3CCC(C(C)(C)C)C3)=O)nn2)ccc2[nH]ccc2c1 42808,CCC(CC1CC1)C(=O)N1CC(NC(=O)CCN(C)CCO)C(F)C1 42809,Cc1nc(CCCC(=O)NC2CC(NC(c3cscc3C(F)F)=O)C2)cs1 42810,C1(CC)C(C(NC[Si](C)(C)C)=O)CCCN1C(c1ccccc1F)=O 42811,N1(C(c2cnns2)=O)CCC2(CCCN2C(c2cc(Cl)n[nH]2)=O)CC1 42812,C1(CNC(C(=O)NCc2ccc(-n3c(C)cc(C)n3)cc2)=O)CC2CCCC2C1 42813,N1(C(c2n(C)cnc2)=O)CCc2sc(CNC(=O)CCc3cnc(O)[nH]3)nc2C1 42814,c1(C(N2CCC(NC(C(OC)OC)=O)(CO)C2)=O)cc2occc2n1C 42815,C1(CN(C(C2CC(C)C2)=O)C)CCCC1NC(=O)C(CN(C)C)c1ccccc1 42816,CC1CN(C(C2CC(CCO)C2)=O)CC(CCNC(c2nnn(C(C)(C)C)n2)=O)O1 42817,C1(CC)CC(C)CN(C(=O)CC(C)(C)NC(=O)CCCN=[N+]=[N-])C1 42818,c1(C(=O)NC(CC(=O)N(C23CC(C2)C3)CC)C)cnn2c1OCC2 42819,C1(NC(c2c(C)cn(C)c2)=O)(CO)CCCN(C(=O)CC(O)c2cnc(Cl)s2)C1 42820,N1(C(C(C)NC=O)=O)CC(NC(c2cc(-c3ccccc3)on2)=O)C(F)C1 42821,c1(C(=O)NC2C(NC(c3ccc(OC4CC4(F)F)cc3)=O)C2)ccc[n+]([O-])c1 42822,C1(C(N)=O)CN(C(=O)C(=O)NCc2cc(N3CCCC3)n[nH]2)c2ccccc2O1 42823,c1(C(N(CCCN(C(CCNC(C2C(C)C2)=O)=O)C)C)=O)scc2c1CCCC2 42824,C(=O)(CC(CC(C)C)NC(=O)CC1CCSCC1)NC1(CO)CC(OC)C1 42825,Cc1cnn(C)c1CC(N1CC(N(C)C(C2C3COCC23)=O)C1)=O 42826,C1(CC)C(NC(=O)C(C)NC(=O)CC(C)(C)C)CCN1C(=O)CC1CCSCC1 42827,C1(CC(N2CC(OCCC(C)C)C2)=O)CC(C)(C)CN1C(c1cc[n+]([O-])cc1)=O 42828,c1(OC)c[nH]c(C(N2CC(N(C(=O)C(C)SC)C)C(O)C2)=O)cc1=O 42829,CCC(C)C(O)C(C)C(=O)N1CC(NC(=O)CCCCCC(C)C)C(O)C1 42830,N1(C(c2n(COC)ncc2)=O)CC(NC(=O)C=CCCC(C)C)CC(C)C1 42831,CC12CC1CN(C(=O)C(N1CCC(c3cccc(Br)c3)CC1)=O)C2 42832,c1(C(=O)NC2CC(CNC(C(CC)O)=O)C2)ccc(C(C)C)cc1 42833,N1(C(C(CC)OCC)=O)CCC(CC(=O)N(CC(C)(F)F)C)C1(C)C 42834,C1(C)(C(N2C(CCCN(C)C)CCCC2)=O)CCCN(Cc2ccccc2F)C1 42835,O=C(CCCc1ccsc1)NCc1nccn1C(F)F 42836,C=C=CCCC(=O)NCCCOCC(c1ccccc1)NC(=O)CCC1CC1(C)C 42837,C(C(C(=O)N(C)CCN(C)C1CC1)C(C)C)NC(c1c(C)n(C)cn1)=O 42838,c1(C(=O)NC(C(=O)NCCc2n(CC)cnn2)C2CCOC2)nnc(S)n1C 42839,S(=O)(=O)(CCC(=O)NC1CN(C(C2CCSC2)=O)CC1CC1CC1)NC 42840,C(C(O)CS(C)(=O)=O)NC(N(C(c1onc(C)n1)C)C)=O 42841,C(=O)(CC(C)(C)CCC)NCC(CC=C)C(=O)NC1COCC1O 42842,C(=O)(CCCC(C)=O)N1CC(NC(C(C)=CC)=O)C(c2nccn2C)C1 42843,C1(C(N(C(C)C)CCN(C)C(c2cc(O)n(C)n2)=O)=O)OCCOC12CCC2 42844,N1(C(=O)OC(C)(C)C)CCC(C(C)(O)CNC(c2cc(CC3CC3)ns2)=O)CC1 42845,C1(C(=O)NC(CC)CNC(C2CC(F)(CO)C2)=O)COCCN1CC 42846,C=CC(C)CC(=O)NC1CC(C(=O)NCc2ccccc2CC)CC1O 42847,O=C(C1=CCN(C(=O)COC(F)(F)F)CC1)NC1CC1C1CCCC1 42848,C(=O)(C(F)(F)C1=CCOCC1)N(C)CC1(O)CN(C(=O)C(F)(F)C(O)C2CC2)C1 42849,c1(CC)sc(C(=O)NC23CC(NC(C4CCN(C(=O)OC)CC4)=O)(C2)C3)cc1C 42850,C1(C(=O)NC2C(C)CCN(C(C=C(C)C)=O)C2C)CCc2nc(O)[nH]c2C1 42851,c1(C(=O)NC2CC(CNC(=O)CC3CCCCC3O)C2)ncc(F)cc1F 42852,C1(NC2(CC(=O)NCc3ccccc3)CC2)CCCCC1CO.c1(N)cc(Cl)ncn1 42853,C(=O)(C(F)(F)C(F)(F)OC(F)(F)F)N1CCN(C(C)=O)C(c2nccn2C)C1 42854,C1(CC(N2CCC(C(=O)NCC)C2)=O)CCN(S(=O)(=O)Cc2ccccc2)C1 42855,c1(C(=O)NC2C3CN(c4c(C#N)nccn4)CC32)cc2cc(Cl)cnc2[nH]1 42856,C(CCCC(=O)NCC1CCCCN1C(c1cccc(F)c1SC)=O)(OC)OC 42857,N1(C(C(CCSC)OC)=O)CC2CC3CC2C1C3NC(=O)Cc1ccc(Cl)s1 42858,c1(CC(=O)N(C2CN(C(c3ncoc3C(F)(F)F)=O)C2)C)c(O)ncnc1O 42859,N1(C(CSCC#C)=O)CCN(C(=O)Cc2ccc(F)cc2)C(c2nccn2C)C1 42860,c1(-c2ccc(-c3n(CC(CC)CO)ccn3)s2)cc(-c2ccccc2)n(CC)n1 42861,Cc1cc(C(N2CC3CC3(CNC(=O)OC(C)(C)C)C2)=O)cnc1C 42862,Cc1ccc(C(=O)NCC2COC(CNC(=O)Cc3csc(Cl)c3)C2)cc1CO 42863,C(C(C(=O)N1CCC(C)(NC(c2cccnc2)=O)C1)C(C)(C)C)OCC=C 42864,c1(C(=O)NCC(CNC(=O)C(CO)N(C)C)OC)ccc2c(c1)NC(=O)CC2 42865,C1(C)(CC(=O)N(C)CC2(O)CN(C(CC3CCCN(C)C3)=O)C2)CCS(=O)(=O)N1 42866,C(=O)(C(C)(C)C(=O)N(C(C1CC1)C1CC1)CCO)N1C(C)CC1C(=O)N(C)C 42867,Cn1ncc2cc(C(N3CC(NC(C4C=CCC4)=O)CC(F)C3)=O)sc12 42868,CCCC(CCC)CCCC(=O)N(C)CCNC(c1cc2c(cn1)CCCC2)=O 42869,CC(C1CC1)=C(F)C(=O)NC(C)C(C)NC(C1(CN(C)C)CC1)=O 42870,c1(OCC)ccc(C(N2CCCC(N(C(=O)C=C(C)C)CCF)C2)=O)cc1Cl 42871,CCS(=O)CC(=O)NC1CCN(C(C)C(N)=O)C1 42872,C1(CCNC(C(n2ncc(C)c2)C)=O)CCCN(C(c2ccc(F)nc2)=O)C1 42873,C(CC(=O)NCC(C)NC(=O)CCC1CC1(Cl)Cl)N(C)C(=O)OC(C)(C)C 42874,c1(CS(N2CCC(Oc3ccc(C)cc3)CC2)(=O)=O)nc2ccccc2[nH]1 42875,N1(CC)CCC(CNC(=O)CC(C)CNC(=O)C(C2CCCCC2)O)CC1 42876,N1(C(c2cc(OCC)ncc2)=O)CCCC(NC(c2ccncc2)=O)C(F)C1 42877,C1(C(N2C(CCC)CN(C(=O)CC(C)(C)C)CC2)=O)Cc2cncn2C(=O)N1 42878,C#Cc1c[nH]nc1C(=O)NC1CN(C(c2csnc2C2CC2)=O)CC1O 42879,c1(C(=O)NCC2C(NC(c3ccc(CN(C)C)nc3)=O)CC2)cc2ccsc2s1 42880,N1(C(C2C(C3(C)COC3)C2)=O)CC2CC(C(=O)NCC3CCCCCC3)C(C2)C1 42881,C1(C(N(CC(CC)(C)OC)C)=O)CC(C2CCCCC2)CN1C 42882,C(=O)(CC(=O)NC1COCC1C(=O)NCC(C)(C)CC1CC1)NCC#C 42883,C(=O)(CCCC(C)(C)C)NC1(CC=CC)CCN(C(=O)C(=O)NC(C)C)CC1 42884,c1(C(N(C2CCN(C(=O)CCc3nncs3)C2)C)=O)ccnc2ccc(O)cc12 42885,C1(C(=O)NCC2(CCOC)CCC2)CCN(C(c2cc(C)[nH]n2)=O)C1C 42886,C1(C(N2CC3C(CO)C3C2)=O)CC(F)(F)CN1C(c1cc(C(F)(F)F)ccn1)=O 42887,c1(C(C(=O)NC(CNC(C(CC#C)(C)CC)=O)(C)C)C)ccc2ccccc2c1 42888,c1(N2CCC(C)C(NC(C3(C)CCCCO3)=O)C2)ncnc2c1c(Br)nn2C 42889,C#CCCC(C(=O)NC1CCCC(O)C1O)NC(C1COCC(C)O1)=O 42890,C(C(=O)N1CC(NC(=O)C2=CCSC2)C(C(F)F)C1)(C(C)C)SCC 42891,CCC(C(=O)N1CC(NC(C2(n3cccc3)CCCC2)=O)C1)NC(N)=O 42892,C=CC(C)(CC)C(=O)NCC1CCN1CCc1ccc(-n2cccn2)c(C)c1 42893,c1(C(=O)NC(C2N(C(C(COC)OC)=O)CCC2)C)n[nH]c2ccc(OC)nc12 42894,C1(CC=C)(NC(c2ccnn2C)=O)CN(C(c2cc(C(C)(C)C)c[nH]2)=O)C1 42895,N1(C(C=C2CCC(C)CC2)=O)CC2=C(C1)CN(C(C1CC1(C)C(F)F)=O)C2 42896,c1(C(=O)NCC2(O)CC(NC(CCS(C)=O)=O)C2)c(F)cccc1Cl 42897,c1(CC)ccc(N)c(C(=O)N(CC(O)CN(C)C(c2cscc2C2CC2)=O)C)c1 42898,C(=O)(C(C)C(O)C(C)CC)N1CCC(C(=O)NCC(C#C)OC)C12CC2 42899,n1(CC(=O)NCC2CC(F)(CNC(C3CC(=C)C3)=O)C2)cc(C#N)cn1 42900,C1(O)(CNC(C(C=CC)O)=O)CCN(C(=O)Cc2ccccc2C)C1 42901,N1(C(C2CCC(C)(CC)O2)=O)CC2CCCC(C1)N2C(c1cc(C(F)F)cs1)=O 42902,c1(C(N(CC(C)SC)C)=O)ccn(CCNC(=O)CN(C)C(C)C)c1 42903,N1(C(C(C)NC(=O)NC)=O)CC(CNC(=O)CCn2cc(Cl)cn2)C(C)C1 42904,N1(C(Cc2c(C)nsc2)=O)CCN(C(c2ccn3nnnc3c2)=O)C2CCC12 42905,CC(C)S(=O)(=O)CC(=O)N(CCCNC(=O)CP(C)(C)=O)C 42906,N1(C(c2c(C)nsc2)=O)CCN(C(C2CC(C(F)(F)F)C2)=O)CC(CO)C1 42907,CC(C)C(C)CC(=O)N1CC(N(C(=O)CCc2cc(Br)ccc2F)C)C1 42908,N1(C(CC2C(C)(C)OCCO2)=O)CCC2CN(C(=O)C=CC=C(Cl)Cl)CC2C1 42909,Cc1cc(C(=O)NCC(CC(C)C)NC(C2CCC(F)CC2)=O)cnn1 42910,c1(NC(C)=O)ccc(NC2CCN(C(=O)N(C3CCN(C)CC3)C)CC2)cc1Cl 42911,c1(C(=O)NC(c2cccc(CO)c2)C(=O)NC(CCC)CCC)nn(C)c(C)c1Cl 42912,N1(C(c2cnn(C(C)C)c2F)C(=O)NCC)CC(C(C)C)c2ccccc21 42913,C1(C(=O)NCC(CC(C)C)NC(C2C=CCS2)=O)CC(C2CCCC2)C1 42914,C1(C)(C(=O)NC2CCC(C(=O)NCCn3c(C(C)C)nnc3)C2)CC(F)(F)C1 42915,C1(CC(=O)NC(C)C(N2CCOCC2)=O)CCCCC1NC(=O)C(CO)N(C)C 42916,C1(CC(=O)NCC2C(C)(C)CCCN2)CCc2ccccc2N1 42917,N1(C(c2scc(C)n2)=O)CCC(O)C(C(N2CCC(c3ccncc3)C2)=O)C1 42918,N1(C(C(COC)OC)=O)CCC(C)C(NC(c2cc(-c3cn(C)nn3)on2)=O)C1 42919,c1(C(C)NC(C23CC(NC(c4c(CC)c[nH]n4)=O)(C2)C3)=O)ccc(Cl)cc1 42920,CCCCCCC(CC)(CC)C(=O)NCC(CNC(=O)CNC(=O)C(C)C)CO 42921,C1(CN(CC(=O)NC2CC(C(C)(C)C)C2)CC(=O)O)CCC(F)(F)CC1 42922,C(C)(C(C)S(C)(=O)=O)N(C(C(=O)NC1CN(C(C)C)C(=O)C1)=O)C 42923,N1(CC(C)OC)CCCC1CCCNC(c1cnc(N(C)C)o1)=O 42924,c1(CNC(CCC=C)=O)n[nH]c2c1CN(C(=O)C(C)S(N)(=O)=O)CC2 42925,c1(C(N2CC3CCCC(C2)N3C(C23CC(C2)C3)=O)=O)ccc2ncccc2c1 42926,C1(O)(NC(C2(COC)CN(C(=O)CCCC(C)(C)C)C2)=O)CCCC(C)CC1 42927,c1(CCC(=O)NC2(C)CC(NC(=O)Cc3cnoc3)C2)cncc(F)c1 42928,c1(C(=O)NC2CC(F)(CNC(C3(C)CCN(C)C3)=O)C2)cccc2nc(O)[nH]c12 42929,c1(OC)cc(C)[nH]c(=NCC2CC3CCC2N(C(c2csc(C(C)C)n2)=O)C3)n1 42930,N1(C(c2ccc(SC)nc2)=O)CCCC(O)(CNC(c2cc(C3CC3)on2)=O)C1 42931,c1(C(=O)NC(C(=O)NCCc2ccc(C)s2)C2CC2)cnc(C)c(C)c1 42932,c1(CNC2CCC(C(=O)NCc3c(F)cccc3Cl)CC2)ccc(O)c(F)c1F 42933,c1(C(N(C(C)C)CCNC(=O)C(F)F)=O)ccc(N2CCCCCC2)nc1 42934,N1(C(C2CN(C)C2)=O)Cc2ccnn2CC(NC(C2CCCCCS2(=O)=O)=O)C1 42935,C(C(C)C(=O)NC1COCC1NC(c1cc(C(N)=O)c[nH]1)=O)OCC 42936,C1(C(C(=O)NCCN(C)C(C2(C)CCCN2C)=O)(C)C)CCC(O)CC1 42937,c1(C(CC)C(=O)N(CC(O)CN(C)C(C2(OC)CC2)=O)C)ccc(F)cc1 42938,C12(CNC(c3nc(CC)cs3)=O)CCCC1N(C(=O)C(CCOC)OC)CCC2 42939,Cc1cc(C(=O)NC(C)CCNC(=O)Cc2ccncc2Cl)c(Cl)cc1Cl 42940,c1(C(C)=O)cccnc1NC(C1CCC(NC(c2ccccn2)=O)C1)=O 42941,c1(C(C)(C)NC(CC(CC)(C)C)=O)ccc2c(c1)OCCO2 42942,c1(C(N(CCNC(c2c(C)nn(CCC)c2C)=O)C)=O)ccc2nc(S)oc2c1 42943,N1(C(c2cn(CC)nc2)=O)CCC2(CCC(CNC(c3csnn3)=O)OC2)CC1 42944,Nc1c(CNC(=O)NC2CCCC2c2cccc(Br)c2)cccc1F 42945,c1(CCC)ccc2c(N)c(C(N3CCNC(C)CC3)=O)sc2n1 42946,c1(C(=O)NCCCC(C)NC(COCCC)=O)cc(Cl)c(F)cc1F 42947,C1(NC(C2CC(=C3CCC3)C2)=O)CCOC(C(N2CC(O)(c3cc[nH]n3)C2)=O)C1 42948,C(C(=O)NCC12CCC(CC1)N2C(C1(C#N)CCCO1)=O)(C(C)(C)C)SC 42949,c1(CCCC)nc(CN(C)Cc2cn(C3C(NC)CCCC3)nn2)c(Cl)[nH]1 42950,c1(SC)cc(C(=O)NCC2C(C)CCCN2C(=O)CC(=O)NC2CC2)ccc1F 42951,CC(C)(CC1CCOC1)C(=O)N(C1CCN(C(=O)CCc2cnoc2)CC1)CCO 42952,CCC(C(=O)N1CC2C(NC(=O)Cc3scnc3-c3cccs3)C2C1)C(C)(F)F 42953,C(CCC(F)(F)F)N(C(CC1N(C(Cc2c(C)con2)=O)CC1)=O)C 42954,c1(C(N(CCCCCC)CCNC(=O)C(C)C#N)=O)ccc2nonc2c1 42955,CC(C)CC(C)(CNC(=O)C(C)(C)c1ccno1)NC(c1cc(C(C)C)on1)=O 42956,c1(C(=O)NC2(CO)CCCN(C(c3cn[nH]c3)=O)C2)cnc2cccnc2c1 42957,Cc1ccc2oc(C(=O)NC(C)(C)CCCNC(C3(CO)CCC3)=O)cc2c1 42958,CC(C(=O)NCCOCC(=O)NCCCN(C)C(C)C)=CC1CC1 42959,c1(CC(=O)NC23CC(CNC(C4CCCSC4)=O)(C2)C3)ccccc1F 42960,C1(N(C(C(CNC(c2nc(C(C)C)oc2)=O)O)=O)C)CCCC1(C)O 42961,Cc1cc(Cl)cc(C(=O)NCCCNC(c2n[nH]c3c2CSCC3)=O)c1C 42962,CCC(CC)CCCNC(=O)CCNC(=O)OC 42963,c1(OCC)cccnc1C(N1CCCC1CNC(c1[nH]c(C2CC2)nc1C)=O)=O 42964,N1(C(C2C(C)(Br)C2)=O)CCCC(C2CC2NC(c2cnn(CC3CC3)c2)=O)C1 42965,c1(OC)cccc(C(N2CCC(=CCNC(=O)COC3CCOC3)CC2)=O)n1 42966,Cn1nc2c(c1CNC(=O)CCCOc1ccc(I)cc1F)CCCC2 42967,C(=O)(C(C)CC(F)(F)F)N(CC(C)NC(=O)Cc1coc(C(F)F)n1)CC 42968,C(=O)(CCn1ccnc1)NCC1CCC1.CC(O)CN1C(=O)CC2(CC2)C1 42969,c1(SC(C)C(N)=O)ccc(C(=O)NC2(C)CN(C(c3ccncc3)=O)C2)cc1 42970,c1(C(=O)NC2(CC=C)CC3CCC(C2)N3)sc2cccc(F)c2c1C 42971,c1(C(N2CC(NC(=O)C(F)(F)CO)CC(C)C2)=O)nc2cccnc2s1 42972,CCCCC(CNC(C1CCCN1C)=O)NC(c1snc(Cl)c1Cl)=O 42973,N1(C(C(C2CC2)OC)=O)CCC(Cn2cc(CCc3ccccc3)nn2)CC1 42974,CC1CC(NCCc2ccc3ccccc3c2)c2c(O)ccc(F)c21 42975,N1(C(C2CC2)=O)CCCCCC1.C(=O)(CCn1cnnn1)N.n1(CC2CC2)cnnn1 42976,C(=O)(CC(COC)COC)NC(CC=C)CNC(C1CCNC(=O)C1)=O 42977,N1(C(CC(=C)Br)=O)CC2CCN(C(=O)C#CC3(C)CC3)CC12 42978,c1(OCC(N)=O)ccc(C(=O)NCC(C)NC(=O)C=CSc2ccccc2)cc1 42979,c1(C(N(C2(C(=O)NCc3ncccc3F)CC2)C)=O)ccc(O)cn1 42980,C1(NC(c2c(CC)c[nH]n2)=O)CCN(C(=O)CSc2cccc(F)c2)CC1(C)C 42981,C(=O)(C1COc2ccccc21)N1C(C)(C)C(NC(C2(F)C(C)(C)C2(C)C)=O)CC1 42982,c1(-c2cn(CCC(=O)N(C3CCC(=O)NC3)CC)nn2)nc(C)cc(C)n1 42983,N1(C(C2N(Cc3c(N(C)C)cccc3)C(C)CC2)=O)Cc2ccc(Cl)cc2C1 42984,Cn1cc(C(=O)NC2CC2CNC(c2ccc(-n3cncn3)cn2)=O)n(C)c1=O 42985,N1(C(c2cncc(SCC)n2)=O)CCN(C(=O)CC=C(C)C)C(C)C1C 42986,c1(C(N2CCC(N(C(CC(CCCC)O)=O)C)C2)=O)ccc(S(N)(=O)=O)cc1Cl 42987,c1(C(=O)NCC(CN(C(C(CC#C)C)=O)C)C)cncc(C)c1Cl 42988,N1(C(C(CNC(C=CC(=O)NC(C)C)=O)N(C)C)=O)CCCC(N(C)C)CC1 42989,c1(C(N)=O)nc(Br)cnc1NC(C1CC(NC(c2ncc(Cl)cc2C)=O)C1)=O 42990,Cc1c(NC(=O)Cc2ccccc2NC(=O)Cc2ccsc2)ccnc1Cl 42991,C1(C)(C(=O)NCCC(C)CCNC(=O)CCCc2ccccn2)CC2CCC1C2 42992,C1(C(=O)NCC2C(CNC(C(CCC)=CCC)=O)C2)COC2COCC2O1 42993,c1(C(N2CCC(C)(NC(c3nc(C)c(C)[nH]3)=O)C2)=O)ccc2[nH]c(=N)[nH]c2c1 42994,CCCN=C(NCC(O)C1(C)CC1)NCC(C)(C)C.C1C(=O)N1 42995,c1(CNC(C(C2CCOCC2)C)=O)cc(C(=O)NCC2CC(CO)CO2)on1 42996,C(=O)(C(C#N)C(C)(C)C)N1C(C(N(C(C)C2CC2)CC)=O)C2CCC1C2 42997,C(=O)(C1=C(Cl)CCCC1)N1CC(CC(N2CC(CCO)C2)=O)OCC1 42998,N1(C(c2cc(C)sc2)=O)CC(NC(C2(Cc3cnn[nH]3)CCC2)=O)C(C)C1 42999,c1(-c2c(C(=O)OC)cccc2)ccc(Br)cc1C(N1CCC(O)CC1C(=O)O)=O 43000,C(C)(C(=O)NC1CC(NC(=O)CCc2nc[nH]n2)C1)=CC 43001,N1(C(C2C(C)(Br)C2)=O)C(CNC(=O)Cn2cnnn2)CC2COCC12 43002,C1(NC(CC2(COC)CCCC2)=O)CCC(C)(C)CC1CNC(=O)C=CBr 43003,c1(OC)cc(C=CC(=O)NCCc2ccc(CNC(c3cnn[nH]3)=O)cc2)sn1 43004,Cc1ccncc1C(=O)NCCC1CCC(NC(c2c(C)coc2C2CC2)=O)C1 43005,c1(C(N2CC3CCN(C(c4c(SC)ccs4)=O)C3C2)=O)ccc(C)cc1[N+](=O)[O-] 43006,C(C(=O)NCC(C)(CO)NC(C1CN(C2CCC2)C1)=O)(C(C)C)OC(C)C 43007,N1(C(C(CC=C)C)=O)CCCCC(NC(c2cc(-c3ccc(F)cc3)cs2)=O)C1 43008,c1(C(=O)NCC2C(C)CCN2C(C2(C(=O)N(C)C)CC2)=O)cc2ncccc2o1 43009,c1(C(CN2CC(CC(=O)OC)(N(C)C)C2)O)cccc(OC)c1 43010,c1(C(N2C(CNC(C(CC#C)O)=O)CC(F)C2)=O)cnn2c1NCCC2 43011,c1(N2CCC(N(C(c3c(CC)c[nH]c3)=O)C)C2)cc(C)ncn1 43012,c1(CNC(=O)NCC2CCN(C(=O)OC)CC2)ccc2cccnc2c1 43013,CC1CC(CNC(c2cccnc2)=O)CN1C(=O)CCCC1CCCC1 43014,CC1Cn2nc(C(=O)NC3COC3)cc2CN1C(=O)OC(C)(C)C 43015,C#CC1CN(C(=O)C(C(C)OC)NC(=O)C(C2CC2)SC)CCO1 43016,N1(C(C(C)CO)=O)CC(NC(c2cncc(F)c2)=O)CC12CCCC2 43017,C1(NC(c2ccc(C)nc2)=O)CC2(CCC(NC(C3C(C)CC3C)=O)CC2)C1 43018,N1(C(CC(C)OC)=O)CCCC(C)(NC(=O)Cc2ccc(O)cc2C(F)(F)F)C1 43019,N1(C(CN=[N+]=[N-])=O)CCc2occc2C1C(=O)N=c1cc(Cc2ccccc2)[nH][nH]1 43020,Cc1ccc(O)c(CNC(=O)CC=CCNC(c2cn(C)cn2)=O)n1 43021,Cc1ccc([N+](=O)[O-])cc1C(=O)NCC(CO)NC(=O)CCCC1CCOCC1 43022,N1(C(CC2CN(C(C(C)NC(C)=O)=O)C(C)(C)C2)=O)CC2(C1)CC(C)(C)C2 43023,CC1(C(=O)NCCCCNC(=O)Cc2ccc(O)cc2Cl)CCC12CCC2 43024,Cc1ccc(CC(N2CC(CNC(C3CC(=O)CO3)=O)C2)=O)c(Cl)n1 43025,C=CCC(CC=C)C(=O)N1CC(O)CC1(C)C(=O)NCCCCC 43026,Cc1cnc(CNC(=O)C(c2cccnc2)NC(=O)CN2CCC(C)C2)cn1 43027,c1(OCC)nc(C)ccc1C(=O)NCC(C)(C)CNC(c1ccnc(C)c1O)=O 43028,c1(C(=O)NC(C)CN(C(=O)CO)C)ncccc1Br 43029,C1(C(=O)NC2C(NC(c3ccncc3C(F)(F)F)=O)C2)CCCC(F)(F)C1 43030,c1(CCC(=O)NCC2CCCN(C(c3cccnc3S)=O)C2)ccc(F)cc1 43031,c1(C(=O)NC(C(C)NC(CC2(CSC)CC2)=O)C)cnccc1C(C)(C)C 43032,CCCCC(O)C(=O)N1CC(N(C(=O)CCCC(=O)C2CC2)C)C1 43033,C1(OC)CC(NC(=O)C(C)CC(C)C)CN(C(c2ccc(Cl)c(N)c2)=O)C1 43034,C1(C(=O)Cc2ccccc2)CN(C(=O)C(O)C(F)(F)F)CCN1C(=O)C(F)=CF 43035,c1(C(C)C)cnc(O)c(C(=O)NC2CCN(C(C3CC(C)(C)CO3)=O)C2)c1 43036,C1(C(N)=O)CC(F)CN(C(=O)CC2CCN(C(=O)Cc3ccc(O)cn3)C2)C1 43037,N1(C(C(CCC)N(C)C)=O)CCCC2(NC(c3ccoc3Cl)=O)CC2C1 43038,c1(NC(CCC2(C)CN(C(N3CC4CC4C3)=O)C2)=O)cccc(N2CCCC2)c1 43039,C(C(=O)N=S(C)(=O)N(C)C)CN(C(CC)C(=O)Nc1ccccc1)C 43040,c1(OCC)cc(N2CCOCC2)ccc1NC(=O)C=CC(=O)O.S1(=O)(=O)CCN1 43041,C1(C(C)C(=O)NCCNS(N)(=O)=O)CCN(C(C2CCN(C)CC2)=O)CC1 43042,N1(C(CCCCSC)=O)CC(C)C(C)(CNC(=O)C(C2CC(F)(F)C2)OC)C1 43043,C#CC1CC2(CC2)CN1C(=O)CCC(C)NC(C1(C#N)CC1)=O 43044,c1(OC)ccc(CC(N)C(=O)NCC(=O)Nc2cccc(OC)c2)c(OC)c1 43045,N1(C(C2CCN(C(C(=O)NCC)=O)C(C)C2)=O)CC(C#N)C2(CCC2)C1 43046,N1(C(C(CC)(C)CO)=O)CCCN(C(=O)Cn2cc([N+](=O)[O-])c(C)n2)C(CO)C1 43047,c1(OC)ccc(F)c(C(=O)NCCCN(C(=O)COCCF)C(C)C)c1 43048,C1(C(=O)NC(C=CC(=O)NC(C(C)F)C)C)OCC2CCCC12 43049,C1(C(=O)OC(C)(C)C)(NC(C(=O)N(C)Cc2c(CC)noc2)=O)CCC(C)CC1 43050,N1(C(C(C)(C)OC)=O)C2CCC1C(CNC(c1nccnc1C(N)=O)=O)C2 43051,CC1=C(C(=O)NC2CCCC2C(=O)Nc2ccc(Br)nc2)CCO1 43052,c1(CNc2c(C)nc(-c3c(OC)cccc3)s2)c(C)nn(C)c1C 43053,c1(NC(C2N(Cc3ccc(SC)s3)CC(F)C2)=O)nc(Br)c(Br)cc1Br 43054,C1(CNC(Cn2c(C)c(Cl)cn2)=O)CN(C(=O)C=C2CCC2)C(C)(C)C1 43055,C(=O)(CC(C=C)CC)NCC(C(=O)N(CC#C)CC#C)CC1CC1 43056,c1(CC(=O)NCCCN(C(C2(O)CCCCCC2)=O)C2CC2)c(O)ncnc1O 43057,C1(OC)CC2CC(C(=O)NCCCC(CO)NC(C3(F)CC3)=O)CC12 43058,C1(NC(=O)CCC=CBr)C2CCC1N(C(c1ccc(CF)cc1)=O)C2 43059,c1(C(N(C)CC2CCN(C(c3ccc(F)cc3N)=O)C2)=O)cnc2[nH]ccc2n1 43060,C1(CC(N2CC(O)(CCNC(C(COC)OC)=O)C2)=O)COCC2(CCC2)O1 43061,CCCCC(O)C(=O)NCCC(C)NC(=O)CC(F)(F)c1ccccc1 43062,N1(C(C2C(CC)C2)=O)CC(O)(CNC(C2(c3ccccc3)CC(F)C2)=O)C1 43063,c1(CCC(c2n(CC)nnn2)NC(C)Cc2nccn2C)cc(Br)cc(Cl)c1F 43064,C(=O)(C1=CCCCCC1)N1CCC(C)(NC(c2nc(C)n(C(F)F)c2)=O)C1 43065,N1(C(C(C)=O)=O)CCOCC(NC(C2(C(F)F)CCCO2)=O)C1 43066,C1(NC(c2cc(Cl)ccn2)=O)COC2(C1)CN(C(=O)CC1CCC(C3CC3)O1)C2 43067,c1(C(=O)NCC2CC(NC(C(C)C3CCCO3)=O)C2)cc(F)c(N)c(F)c1 43068,N(C1CS(=O)(=O)Cc2ccccc21)C(=O)C(c1ccc(O)cc1)O.C(C(O)CO)N 43069,C1(C(=O)NCC2OCC3(CN(C(C=CC=CC)=O)C3)C2)CCC(C2CCCO2)O1 43070,C1(P(C)(C)=O)(C(=O)OCc2cnc(C)s2)CC1 43071,C1(CNC(C2(OC)CCCC2)=O)CC2(CC2)CN1C(c1cc[nH]c1)=O 43072,C(C)(CN=c1nc2c(ncn2C)c(NCC2CCN(C)CC2)[nH]1)N(CC)CC 43073,C(C(O)C(=O)NCCc1noc(C)n1)NC(C1C(C(=O)OC)C=C1)=O 43074,C1(NC(CCSC)=O)CCN(C(C2COCCN2C)=O)C1(C)C 43075,CC(C)CC(C(=O)N1CCCC(NC(=O)CNC(c2ccccc2)=O)C1)N(C)C 43076,C1(NC(CN(C(COC)=O)C)=O)CC2CC(C1)N(C(C1CC3CCC1CC3)=O)C2 43077,C1(C(C)NC(=O)CN(C)CCO)CCCN(C(=O)CCCn2cccn2)C1 43078,C12(CC=CCC1)c1nnc(n1CC1CCCO1)N(C)C2.n1(CC)nc(C)cc1Cl 43079,Cc1ncc(C(=O)NC2CC(OCC(=O)N(CC(C)(C)C)C(C)C)C2)c(=N)[nH]1 43080,Cc1noc(C)c1CSCCC(=O)NC1CCCN(C(c2cc(O)nn2C)=O)C1 43081,c1ccc(C2CC(NCc3cnc(C4CCC4)o3)CN2)cc1 43082,CC1CC(C(N2CC(O)(CNC(=O)CSCC(F)F)C2)=O)CN1C 43083,c1(NC(C)=O)ncc(S(=O)(=O)N2CCCC(c3ccc(CO)cc3)C2)s1 43084,Cc1ccc(C(C)C(=O)NCC2(F)CCC(CNC(c3cnc(O)o3)=O)C2)cc1 43085,c1(C(=O)NCCC2CC(C(=O)NCCC3CCC4CC34)C2)ccccc1Cl 43086,C1(NC(c2n(C)cc(Br)n2)c2nnnn2Cc2cccs2)CC2(CCCC2)C1 43087,C(C(CC(C)C)C(=O)NC12CC1CN(C(c1ccnc(C3CCC3)c1)=O)C2)OC 43088,CC1=C(C)CC(C(=O)NC(C)C=CC(N2CCCC2C2(C)CC2)=O)CC1 43089,C1(C(=O)NC2CC3CCC(C2)N3C(=O)C(O)C2CCC2)(OC)CCC(F)(F)CC1 43090,C(C(CC(C)C)NC(=O)Cc1ccc(F)cn1)NC(C1CC(C)(CC)C1)=O 43091,C(C)(CC(C)NC(c1sccc1C1CC1)=O)NC(CCN(CC)CC)=O 43092,N1(C(CC(CC(=O)OC)C)=O)CCN(C(C2CC(=O)N2)=O)CC(C)(F)C1 43093,CC1CCN(c2nnc(C(F)(F)F)s2)C(C)C1NC(C1CSC1)=O 43094,C1(C(N(C2CCN(C(c3ocnc3C)=O)CC2)CC)=O)C2C(=O)OCC12Br 43095,c1(C(=O)NCC(CC(C)C)NC(=O)C=CS(C)(=O)=O)cc2cc(F)ccc2o1 43096,c1(C(N2CC(NC(c3nccc(C)n3)=O)C3C2C3)=O)cc2cccnc2s1 43097,C(=O)(C(=O)C(C)(C)CC)N1CCC(CCC(N2CC(C)(CC)C2)=O)C1 43098,C#Cc1cc(C(=O)NCCC(C)NC(C2(C)CCCS2(=O)=O)=O)ccc1C 43099,c1(C(=O)NCC23C(CN(C(C(C)=O)=O)C2)C3)cc(Cl)cc(Cl)c1O 43100,CCCC(CC)CC(=O)NCc1cccc(NC(c2c(N)cc(F)cc2F)=O)c1 43101,C1(NC(c2c(C)ccnn2)=O)COC2C(NC(=O)CCCC(F)F)COC12 43102,c1(C(C(=O)NCC=C)N(C)C(C2CCOCC2)C)c(Cl)nc2sccn12 43103,c1(Nc2nnc(CCSC)s2)nc(Cl)cc2cc(Br)ccc12 43104,Cc1cc(S(N)(=O)=O)sc1C(N1C(CNC(C2C=CC=CC=C2)=O)CC2CC12)=O 43105,N1(C(C2CC(=C)C2)=O)CCC(CC)(NC(c2ccccn2)=O)CC1 43106,Cc1nc(C(N2CC3(NC(c4ncoc4C)=O)CC2C3)=O)n(C)n1 43107,N1(C(c2ccc(C(=O)OC)cn2)=O)CCC2(CC1)CC2NC(=O)CN(C)S(N)(=O)=O 43108,C12(NC(CNC(CCC(C)C)=O)=O)CCOCC1CN(C(=O)CC1CCCC1)C2 43109,C1(CNC2CC(C)SCC2)CCc2n[nH]cc2C1 43110,c1(CCC(=O)NCC2C(NC(C(CC)F)=O)COC2)ccc(Cl)cc1Cl 43111,O=c1c2c(ncn1C(F)(F)CC(F)(F)F)[nH]c1ccncc21 43112,Cc1ccc2c(c1)CN=C2NCC1CC2C=CC1C2 43113,C(=O)(C1=CCCOCC1)N(CCNC(=O)C(C(C)(C)C)C1CCC1)CC 43114,c1(C(=O)NC(C2CCN(C(C3CC4CC3CC4O)=O)C2)C)ccc(C#N)cc1F 43115,c1(C(=O)OC)cc(NC(=O)NCCCC(c2ccccc2)C2CC2)c(Br)cc1C 43116,C12(CNC(C3C(C)CCO3)=O)CCC(CN(C(=O)C=C3CCN(C)CC3)C1)C2 43117,N1(C(c2n(CCC)ncc2)=O)CCC(C(=O)NCC(C)C)C1(C)C 43118,N1(C(C(CCC#C)O)=O)C(CNC(c2cccc(C(C)C)c2)=O)CC2CCCC12 43119,CCCCC(CNC(c1conc1C(C)(C)NC(=O)COC(C)(C)CC)=O)OC 43120,CCCC(C(O)C(=O)NCC(F)(CC)CC)NC(=O)C(O)C(C)(C)C 43121,c1(C(N2CCN(C(CCP(C)(C)=O)=O)C(CO)C2)=O)ccc(N)c(Cl)c1O 43122,CC(N=c1[nH]c(=NC2CCN(c3ccncc3)C2)[nH]c2c1COCC2)C1CC1 43123,C1(C(N2CCCC(OC)C2)=O)COCCN(C(C2CC2(C)C(F)F)=O)C1 43124,Cc1nc(N2CCCC2)nc(O)c1CCC(N1CCN(C(=O)CO)CC1C1CC1)=O 43125,N1(C(CCCC(=C)C)=O)CC2COCCC2(NC(C2CCOCC2(C)C)=O)C1 43126,Cc1cc(N)c(C(=O)NCC2(CN(C(=O)CC3CC4(CC4)CO3)C)CC2)nc1C 43127,C1(NC(C(c2cccnc2)NC(C2C(=C)C2)=O)=O)CCC(C)(C)CC1 43128,CC(C)CC(C(=O)NC(C)CNC(c1ccncc1Cl)=O)N1CCCCC1=O 43129,c1(C(N2CC3C(NC(=O)COCC(F)(F)F)(C3)C2)=O)cnc(O)c2cnccc12 43130,c1(N(C(C2CC(OCC)C2)C(=O)Nc2ncn(C)n2)CCOC)ccc(F)cc1 43131,C1(N(C(=O)CCc2ncco2)CC)CCCN(C(=O)CCC2CCCO2)CC1 43132,c1(CC)n[nH]c(CC)c1CC(N1CC(C)(NC(C2CC2C)=O)C1)=O 43133,Cc1ccc(CC(N2CCN(C3CCN(C(c4csnn4)=O)CC3)CC2)=O)cn1 43134,CC(C)C(CC(=O)N1CCN(C(c2cc(Cl)cs2)=O)CC1CO)c1ccccc1 43135,C(=O)(C(C#N)C(C)(C)C)NC(CCC)C(=O)N1CC(CCO)C1 43136,CCC(CNC(=O)Cc1ccc(CO)cc1)(CC)NC(=O)C=Cc1scnc1C 43137,c1(C(=O)NC2C(CNC(c3cc(OC)ncc3)=O)CCC2)noc2c1COCC2 43138,N1(C(CC(C)C)=O)CCC(N(C)C(c2cc(-c3cccnc3)[nH]n2)=O)C(C)C1 43139,N1(C(C=C(CC)C)=O)CCC2(NC(=O)Cc3c(F)cccc3Br)CC2C1 43140,C12CCC3(CN(C3)C1=O)O2.Cc1cc(C(=O)NCCOCc2cccnc2)c[nH]1 43141,C1(CC(=O)NC2CC(F)(F)CC2NC(C2SCCCS2)=O)CN2CCC1CC2 43142,N1(C(Cc2c(C)con2)=O)CC2(CCN(C(=O)C(C)(c3cccs3)N(C)C)C2)C1 43143,c1(C(N2C(CNC(C3(C(C)(F)F)CC3)=O)CCC(C)C2)=O)cnn2c1OCCC2 43144,c1(C(=O)NC(C2CCCC2)CNC(C2(C#C)CC2)=O)cnn2c1CC(F)(F)C2 43145,Cc1cccc(CN(C(N)=O)CC2CCN(C(C3CCCCO3)=O)CC2)c1 43146,N1(C(C(C)(C)OC)=O)CCN(C2CCCN(C(c3cnsn3)=O)C2)C(=O)C1 43147,N1(C(c2c(C)scn2)=O)CCC(OCCNC(=O)CC2CCS(=O)(=O)C2)CC1 43148,CC1=CCC(C(=O)NCCCN(C(=O)CC(C)NC(=O)OC(C)(C)C)C)CC1 43149,CCCC(O)C(CO)NC(C1(CSC)CCC1)=O.C12(CC1)N(C)C2=O 43150,N1(C(c2n(C)ncc2)=O)CC(C(N2CCCC3C(O)CC23)=O)CCC1(C)C 43151,C1(C(=O)NC(c2ccoc2)C)(CNC(C2CCCCC2)=O)CC(C)(C)C1 43152,N1(C(C(C)N(C)C)=O)CCC(CNC(C2NC(=O)C3CCC23)=O)C(F)(F)CC1 43153,C(=O)(CC(O)CCCC)N(CCCCC(N1C(CC=CC)CCCC1)=O)C 43154,Cc1cc(CCC(=O)NCCC(O)CNC(C2(C)CCN(C)C2=O)=O)cc(C)c1 43155,C#Cc1cncc(C(=O)NCCC2CC(F)(F)CN2C(c2nocc2Cl)=O)c1 43156,CC1CN(C(c2cc(OCC3CC3)ncc2Cl)=O)CCN1C1CCCCC1 43157,C(CC(C)CC)(C(=O)N1C2COCC1C2)NC(CC=C=C)=O 43158,n1(CC(N2CCC(CNC(C(COC)C)=O)CC2C)=O)cc([N+](=O)[O-])nc1C 43159,N(C1CC(C)n2ncnc21)C(C1CCC(NC(C2(CCC=C)CC2)=O)CC1)=O 43160,N1(C(c2c(N)nc(Br)cc2)=O)CCC2(C1)CN(C(C1CCC(O)CC1)=O)C2 43161,N1(C(CC2(COC)CCCC2)=O)CCC(C)(C)C(NC(=O)C(C)OC)C1 43162,c1(CNC(C(C(C)C)F)=O)nnc2n1CCN(C(C1(C)CCOC1)=O)C2 43163,C1(NC(C2(CCCC)CCC2)=O)CN(C(C2CN(C)C2)=O)C2(CCOC2)C1 43164,C1(C(=O)NC(C)CCCCNC(c2cnc(C(C)(C)C)[nH]2)=O)CC2(CC2)CN1C 43165,CCC(C)(C)CCCC(=O)NCCC(C)NC(c1nc(C)ncc1Br)=O 43166,CC(C)(CC(=O)N1CCC(O)(CNC(=O)CCCC(F)(F)CO)C1)CC(F)(F)F 43167,c1(C(=O)NCC#CCNC(=O)CCc2cnccn2)cc(Cl)c2c(c1)OCO2 43168,C(=O)(C(F)(CNC(=O)C(O)C1CCC1)C(C)C)N(CC)CC1CCCOC1 43169,c1(C(N2CC(C)C(C)C2)=O)cc(Br)cc(F)c1N 43170,N1(C(Cc2cc(C)[nH]n2)=O)CC(C)(C(=O)N(CC2=CCSC2)C)CC1(C)C 43171,C(=O)(CC(C)(C)C(F)F)N(CC(C)(C)CNC(=O)Cc1ccon1)C 43172,C1(CC=C)(NC(C2CCSC(C)C2)=O)CCCN(C(c2csc(C(C)=O)n2)=O)C1 43173,c1(NC(C2CN(C(c3c(C)nc[nH]3)=O)C2)=O)cnn2ccccc12 43174,C1(CC(=O)N(CC)CC2CCCN2C(c2ccoc2CC)=O)COCC(C)(C)O1 43175,N1(C(c2cc(C)c(O)cc2)=O)CCC(F)(F)C(NCc2ccc(Cl)nc2Cl)C1 43176,N1(C(c2ccc(C(C)=O)[nH]2)=O)CC(C)(C)CC1CC(N1CCOC(CCO)C1)=O 43177,O(NC(=O)C(CNC(C1CC2CCC(C1)O2)=O)CC(C)C)CC(CC)C 43178,N1(C(C(C2CC2)SC)=O)CCC(C)(NC(=O)CC2(O)CCCCC2)CC1 43179,C1(NC(CCCCOC)=O)CCC2(CC1)CC2NC(=O)C(=O)N(C)C 43180,CC1CCN(C(c2cnc(N)c(Br)c2)=O)CC1NC(=O)C(C)(C)C1CC1 43181,N1(C(c2c[nH]c(=N)s2)=O)CCC(NC(C2CC(OC3CC3)C2)=O)C12CCC2 43182,C1(CNC(C2C(C(=O)OC)CC2)=O)CC(C2CC2)C1.C12(CC=CC1)C(=O)NC2 43183,C(=O)(C(CCNC(=O)CCn1cncn1)OC)N1CCC(C(CC)CC)C1 43184,c1(C(=O)NCC(Cc2ccccc2)N(C(C2CC(=C)C2)=O)C)ccn(O)c(=O)c1 43185,CC1CN(C(=O)CC2CC3CCC2O3)CCC1CNC(C1(O)CCCCCC1)=O 43186,c1(C(C(=O)NC2(C)CC2)N(C(c2ccccc2)C(=O)OC)C)c(SC)cccc1F 43187,C12(NC(CCC=CC(C)C)=O)CCC1CN(C(C1(N(C)C)CC1)=O)C2 43188,c1(C(N2CCC3CN(C(C4ON=C(C)C4)=O)C3C2)=O)cnc2sc(C)cn2c1=O 43189,c1(C(=O)NC2CN(Cc3cnc(Cl)cn3)CC2F)cc(F)c(F)cc1F 43190,C1(C(=O)NCCc2noc(C3CCCCC3)n2)CC2OC(=O)OC2C1 43191,C1(NC(C2C(C(N)=O)C2)=O)CCC(NC(c2c[nH]nc2C(F)(F)F)=O)C1 43192,c1(CNCC2CCC(C)(C)O2)ccc(Br)nc1F 43193,C1(C(=O)OCC)Cc2c([nH]c3ccccc23)CN1CC(=O)Nn1cc(C#N)cn1 43194,c1(SC)cc(F)ccc1OC(C)C(=O)Nc1ccc(OC(=O)C(C)(C)C)cc1 43195,c1(SCC(=O)NC2COCCN(C(CC(=O)OC)=O)C2)ccc2c(c1)CCC2 43196,N1(C(c2c(C)ncc(C)c2)=O)CCN(C(=O)CC(O)C(C)C)C2(CCC2)C1 43197,N1(C(C)=O)CCCN(C(=O)C(=O)NC(CC)CC(=O)NC2CCC2)CC1 43198,C1(C(=O)NCC(C)NC(c2cccc(-c3nnco3)c2)=O)CN(C)CCO1 43199,N1(C(C=CCCC)=O)CC(CNC(=O)Cc2cc(-c3ccccc3)on2)C2CC12 43200,C#Cc1ccc(OCC(C)Nc2conc2C2CN(C(=O)OC)C2)cc1.C(=O)O 43201,c1(C(N(CCN(C(C2C(C(=O)OC)C2)=O)C)C)=O)nnn2c1CSCC2 43202,C(CCCCC(=O)NC(C)CCC(=O)N(C)C(c1ccccc1)C)=CC 43203,C(C)(CCCN=c1nc(CO)cc[nH]1)NC(C(C)CC1CCCCC1)=O 43204,C=CC(C)C(C)C(=O)NCC1CN(C(C2(N(C)C)CCCC2)=O)C1 43205,c1(C(N2CC(CC)C2)=O)cc(Br)cc2c1cnn2CC.c12cncc(c1)NC2=O 43206,CC1CN(C(C2CC2c2cccc(Cl)c2)=O)CC1NC(=O)C(C)(Cl)Cl 43207,c1(CN2CCN(C(C(=O)N(C(C)C)C)C)CC2)nccc2ccccc12 43208,C#Cc1cc(C(=O)NC2C3CC(NC(C4CCC(OC)C4)=O)CC23)cc(N)c1 43209,c1(C(N2CCC(NC(C3(CC)CCC3)=O)C2)=O)ccccc1OCc1ccoc1 43210,C(=O)(N=c1cc[nH]c(C)c1F)C1C(NC(c2c(C)nc3cccc(Cl)c3c2)=O)C1 43211,c1(OC)cnc(N2CCN(C(=O)NC(C)CCN3CCOCC3)CC2)nc1 43212,N1(C(c2n(CC#C)ccc2)=O)CC(NC(=O)C(C)c2cc[nH]n2)CCC1C 43213,C(c1csc(C)n1)=CC(=O)NCC(CC)NC(C1CSCC(=O)N1)=O 43214,c1(C(N2C3C(NC(CCC(C)O)=O)(CCC3)CC2)=O)nn(C)c2c1CCCC2 43215,Cc1oc(C(=O)NC2CN(C(C3C(C)C3(F)F)=O)CC2O)cc1S(N)(=O)=O 43216,CC(C)C(C)C(C)CC(=O)NCC12CC(NC(c3cnn(CC(F)F)c3)=O)(C1)C2 43217,c1(N2CC(C)S(=O)CC2)ccc(S(=O)(=O)NCCc2cnoc2)cc1Cl 43218,CC(C)CC(O)C(C)C(=O)N(C)Cc1ccc2ccccc2c1 43219,N1(C(C2C(CC)OCC2)=O)CCC(CCNC(C2(OC(C)=O)CCCC2)=O)CC1 43220,c1(CC)cccnc1C(=O)NCCC1(O)CCN(C(=O)C(C)OCCC(C)C)C1 43221,c1(C(N2CCN(C(c3c(C)ccnc3O)=O)CC2C)=O)cccc(C#N)c1Br 43222,O=C1CCCCC(C(N2CCC(C(C)(C)NC(c3ccc(F)cc3F)=O)C2)=O)N1 43223,c1(C(N2C(C(N3CCC3c3ccccc3)=O)CCC2)=O)nnc(O)nc1O 43224,c1(OC)cc(C(N2CC(NC(C3(C)CCC(=O)N3)=O)C2)=O)sc1S(N)(=O)=O 43225,C(CNC(=O)C(C)CN(C)C)(CC(F)(F)F)NC(C=Cc1nnc(C(C)C)o1)=O 43226,c1(C(=O)NC23CC(C(=O)NC4CCCN(C(C)C)C4)(C2)C3)c(F)cc(Br)cc1F 43227,CCC(C)C(O)CC(=O)N1CC(F)CC1C(N1CCC(OCC(N)=O)C1)=O 43228,c1(C(N(C2CCN(C(C3=C(C)CCC3)=O)C2)CCO)=O)c(C)nn2c1CCCC2 43229,c1(OC)ccc(C(=O)NCCN(C)C(C2CC3CC23)=O)c(C(F)(F)F)c1 43230,CCCN(OC)C(=O)CC1CCN(C(C23CCC(C2)C3(C)C)=O)CC1 43231,C1(OC(CC)C)CN(C(=O)Cc2ccc(C(C)=O)cc2)CC1OCC 43232,N12CCc3cc(ccc3C1)C2=O.c1(OC)ccccc1CO.C12CC1C(=O)N2 43233,C1(C(=O)NC(C2CCN(C(=O)CCc3cccnc3)CC2)C)CCCCC(=O)C1 43234,c1(C(=O)NCC(CNC(C=CC(=O)NC2CC2)=O)F)ncoc1C1CCCO1 43235,C1(C(=O)NC(c2ccccc2)CC)CCC(n2cc(C3CCC3)nn2)C1 43236,CCCC(C)CC(=O)NCCOCCCNC(=O)CC=C(Cl)Cl 43237,CC1CC(NC(=O)CC2(C)CCN2C(=O)C=Cc2ccncc2)c2nccn21 43238,N1(C(=O)OC(C)(C)C)CCC2CCCC12COC(=O)Cc1cncnc1O 43239,CC(C)C(C(C)NC(C12CCN(CC1)C2)=O)NC(c1cc(C(F)(F)F)n[nH]1)=O 43240,C12(CNC(C3C(C)(C)C3)=O)CCC1CN(C(=O)Cn1nnnc1C1CC1)C2 43241,C(=O)(C(F)C(C)C(F)(F)F)NC1C(CC)CN(C(=O)C=Cc2cn(C)nn2)CC1 43242,Cc1cncc(C(=O)NCCN(CC(C)O)C(c2cn(C3CCOC3)cn2)=O)c1 43243,c1(C(N2CCCC(NC(c3ccccc3Br)=O)C2)=O)cc(Br)cc(Br)c1 43244,c1(C(=O)NC(CN(C)C)C(=O)NCC#CC(F)(F)F)ccc(C#N)n1C 43245,C1(NC(CSC)=O)C=CCN(C(c2cc(C)sc2Br)=O)C1 43246,Cc1ncc(C(=O)NCC(C)CNC(=O)Cn2c(C)c(C)sc2=O)c(C(C)C)n1 43247,c1(C(=O)NCC2N(C(C(CCOC)OC)=O)CC(OC)C2)scc2c1CCCC2 43248,C(C(C)(C)CNC(c1cc(CSC)on1)=O)N(C(=O)C(C)NC(=O)OC)CC 43249,C1(C(=O)NCC#CCCO)(CC)CCN(C(=O)C(C2(O)CCCC2)F)CC1 43250,C1(NC(c2c(CC)ncnc2)=O)CN(C(=O)Cc2cccc(F)c2)C2CCCC12 43251,C1(c2n(CCCSC)nnn2)(NCC2(F)CCCC2)CCOCCC1C 43252,N=c1[nH]c(=NC(CCO)c2ccc(F)cc2F)[nH]c(=NC2CCC(=O)NC2)[nH]1 43253,c1(C(=O)NC(C(C)NC(Cn2c(C)cnc2)=O)C)ccc(C(N)=O)c(Cl)c1 43254,C1(CN(C2CC(C)CCO2)CC)CCCN(C(=O)CCCc2cnccn2)C1 43255,CC1CC(O)CCN(C(=O)CC(C2CC2)NC(c2cnn[nH]2)=O)C1 43256,C(CCCC(CO)NC(=O)C(F)C1CCC1)NC(c1ncn(C(C)C)n1)=O 43257,C1(C(=O)NC2(C(COC)O)CC2)CC(C)(C)CN1C(=O)C(n1ccc(C)n1)C 43258,c1(C(=O)NCC=CCNC(c2cscn2)=O)cc(C2CC2)[nH]n1 43259,C1(C(CCC)C)CCCCN1N1CCC(CCO)(C(=O)OCOC)CC1 43260,N1(C(c2c(CNC(C3C(C)C3)=O)n[nH]c2)=O)CCC12CC(C)(CO)C2 43261,c1(C(=O)NCC(=C)C)ccc2cccc(-c3cc(C)ccc3C)c2n1 43262,C1(C(=O)NCCC2C=CCC2)(N(C(C(C)N2CCCC2)=O)C2CC2)CCN(C)C1 43263,N(C(=NCCOc1ccc(Br)cc1)NC1CCOCC1)C1CCC(SCC)C1 43264,c1(C(N2C(CCNC(c3ccc(C)s3)=O)CC(OC)C2)=O)cccn2cnnc12 43265,c1(C(N2CC(C(=O)NCC=CCNC(CC)=O)(CC)C2)=O)ccc(=O)n(CC)n1 43266,C(=O)(CC(C)C(F)(F)F)NCCCC(C)NC(C(C(C)C)C)=O 43267,C1(NC(C(C)OCC)=O)CS(=O)(=O)C12CCN(C(c1cc(Cl)nc(=N)[nH]1)=O)CC2 43268,FCCCN=C(NCC1CCCO1)NCC1(c2ccc(F)cc2)CCCC1 43269,C(=O)(CCC(=O)N1CC=CC1CNC(=O)C(O)CC1CCOCC1)OC 43270,C1(C(=O)NCCN(C(=O)C(C)n2cnnn2)CCOC)(OCC)CCOC1 43271,N1(C(CC(C)c2ccccc2)=O)CCN(C(=O)COCCOCCO)C2CCC12 43272,c1(C(N2CCC2Cn2cc(CC3CCOCC3)nn2)=O)cc2n(c1)CCCC2 43273,c1(N2CCC(N(C34CCCCC3C4)CC)CC2)nc2ccc(C)nc2s1 43274,C1(C(N(C(C)CNC(c2ccccc2SC)=O)CC)=O)NC(=O)OC1C 43275,N1(C(c2cc(C)sn2)=O)CCC2(CC1)C(NC(C1CC3CCC1O3)=O)CS2(=O)=O 43276,Cc1cc(C(=O)NC2CC2NC(=O)C(C2CCCCC2)C)cnc1C 43277,c1(SCCN(C(C2CCCN2C)=O)CC2N(C(CC)CC)CC=C2)ccc(F)c(F)c1 43278,Cc1cc(C)c(C(=O)N(CCCNC(=O)C=C2CCSCC2)C)c(=O)o1 43279,c1(CNC(C2N(S(C)(=O)=O)CC2)=O)cnn2c1CN(C(C1(C(N)=O)CC1)=O)CC2 43280,c1(-c2ncc(C(=O)NCC(c3ccncc3)O)s2)cccc(Cl)c1 43281,N1(C(CSCC(C)=O)=O)CCOCC1c1cn(CCn2nc(C)cc2C)nn1 43282,c1(C(N2CC(NC(C(C)=C(CC)C)=O)C(C3CC3)C2)=O)cccc([N+](=O)[O-])c1Cl 43283,N1(CC2C(CC(F)(F)F)CCCC2)CCc2cnccc21 43284,c1(N2CCN(c3cc(NC(CC=C)C(=O)O)ncn3)CC2)c(F)ccc(Cl)c1F 43285,C(CS(=O)(=O)CC(=O)N1CC2(CC(NC(=O)CCCCC(C)C)C2)C1)OC 43286,c1(C(=O)NCC2CCCN2C(C2CCS(=O)(=O)CC2)=O)ccc2ocnc2c1 43287,N1(C(CC=C)=O)Cc2[nH]nc(C(=O)NCC(COC)C(C)C)c2C1 43288,N1(C(c2c(C)n[nH]c2C)=O)CCCC1C1CCCN1C(=O)C=CCO 43289,Cc1c(NC(=O)CN(c2ccc(C#N)cn2)C)cc(F)cc1[N+](=O)[O-] 43290,N1(C(c2c(CC)csc2)=O)CCC2(CCN(C(=O)COC)C2)C1 43291,C(=O)(C(C)(C)CC(C)(C)C)NC1CC(C)N(C(C2CCSC(C)C2)=O)C1 43292,Cc1cc(C(=O)NC2C3CC2CN(C(=O)C(C)C(C)C)C3)c(N)c(C)c1 43293,c1(C(N2CC(CC)N(C(=O)C(O)CC(C)C)CC2)=O)ccc2ocnc2n1 43294,CC(C)CC(C)(O)C(=O)N(C)CC1CCCN(C(c2cc(C(F)(F)F)c[nH]2)=O)C1 43295,C1(C(N(CCNC(C2(C(F)(F)F)CCN(C)C2)=O)CC)=O)CNC(=O)CC1(C)C 43296,c1(NC(C(CCOC)NC(=O)C(=O)C2CCCC2)=O)ccc2nccn2c1 43297,C1(CC)CN(C(=O)Cc2ccc(C(F)F)cc2)CCN1C(c1ncc(F)cn1)=O 43298,C1(NC(C2(F)CC3(CCC3)C2)=O)CCOC2(CCCCC2)C1 43299,C(CCC(C)(C)C(=O)NCc1nonc1C)NC(C(=Cc1ccco1)C)=O 43300,C=CCC(CC(=O)Nc1cnc(Cl)cc1C)NC(=O)CCC1OCCO1 43301,c1(C(N2C(CN(C(=O)CC#N)C)CCC2)=O)cnn2c1CCC2 43302,N1(C(C2C(OC)CCC2)=O)CCCC2CN(c3ncc(O)cn3)CC12 43303,C1(C(N2CC3C(C(=O)NC(CC(=O)NC)C)C3C2)=O)CC(=O)NC(C)C1 43304,C#CCC(CC(=O)NC(C(C)C)C1CCC1)NC(=O)CCCNC(C)=O 43305,c1(OC)cncc(C=CC(=O)NCCCCNC(c2c(C3CC3)cnn2C)=O)c1 43306,C(C(C)C(C)C(=O)NC1CC(CCNC(=O)COCc2ccnc(O)c2)C1)OC 43307,c1(CC(=O)NC2CCC2NC(c2ccc(O)nc2Cl)=O)n[nH]c2ccccc12 43308,N1(C(COC2(C)CN(N(c3ccc(C=O)o3)C)C2)=O)CCCC1(C)C1CC1 43309,C(=O)(NN1CCCC1C(=O)NCC(C)(CO)OC)c1cc(CC)nn1C 43310,Cc1sc(Cl)nc1C(N1CC(NC(c2cc(C(N)=O)c[nH]2)=O)CC1C)=O 43311,C1(C(N(CC(=O)NCCC)C)=O)N(C(=O)C(C)SC(C)C)CCC1(C)C 43312,Cc1ncnc(C)c1NC(C1CCCCN(C(C23CC(F)(C2)C3)=O)C1)=O 43313,N1(C(C(C)CS(C)=O)=O)CCN(C(=O)CNC(=O)Cn2cncn2)C2(CCC2)C1 43314,N1(C(C=C(CC)CC)=O)CCC(O)(CCNC(c2csc(Cl)n2)=O)CC1 43315,c1(C(N2CCCC2CCCNC(C2COCCO2)=O)=O)ccc(C(F)(F)F)cn1 43316,c1(N(C(=O)C(C)(c2cccnc2)Nn2cc(CO)nn2)CC)ccc(OC)cc1 43317,CCCC(CCCS(C)(=O)=O)C(=O)NCCCC(C)NC(=O)CC1(C)CCCC1 43318,c1(C(N2CCC(NC(C3(C)CCC(C)CC3)=O)C(O)C2)=O)c(F)cc(Cl)cc1F 43319,c1(C(=O)NC2CN(C(c3c(OCCC)cccc3)=O)CC2O)cc(Cl)ccc1Cl 43320,c1(C(N(C(CCNC(C2(CC(C)C)COC2)=O)C)C)=O)cc(C(N)=O)cs1 43321,C1(C(N2C(CC#C)CCCC2)=O)CN(C(=O)CCc2cnn[nH]2)CCN1C 43322,c1(C(=O)NC2CCN(C(c3scnc3Cl)=O)CC2)cnc2c(c1)C(=O)CCC2 43323,C1(O)(CCNC(c2cc(C)n(C)c2)=O)CCCN(C(=O)C2=CCC2)C1 43324,N1(C(C(C(C)C)SCC)=O)CCN(C(=O)Cc2sc(C)nc2C)CC(C)(C)C1 43325,C(=O)(CCC(C)(F)F)NCC(C)C(=O)NCCN1CC(C)(O)C1 43326,N1(C(C(C=C)(C)CC)=O)CC(C2CN(C(c3[nH]c(=N)ccc3C)=O)C2)C1 43327,c1(N2C3C(NC(=O)CC4CCOC4)(CCC3)CC2)ncnc2[nH]ccc12 43328,N1(C(Cn2ncc(C)c2)=O)CCCCC1c1cn(Cc2ccoc2C(=O)O)nn1 43329,C(CC)(CCCC(=O)NCc1cc(C#N)cs1)NC(C1(CC#C)CC1)=O 43330,C(CCC(N)=O)(C(=O)NCCCCCNC(C1CCC1(F)F)=O)N(C)C 43331,CCCCC(CC)C(=O)NC(C)(C)C(C)NC(c1ccc(COC)cc1)=O 43332,C1(C)(CNC(CCN(C(C)C)C(c2cc(N)cc(F)c2)=O)=O)CCCCC1O 43333,C(CCC(C)C(=O)NCC1(C)CCN(C(C2(C)CC3CCC2C3)=O)CC1)OC 43334,C(=O)(C1Cc2ccccc21)N1CCCC(CN(C(CCc2ncc(C)[nH]2)=O)C)C1 43335,c1(C(=O)NC2(C)CCN(C(C3C(Cl)(Cl)C34CC4)=O)C2)cnc2cccnn12 43336,c1(CC(c2c(C(=O)O)c(-c3ccccc3)cs2)=O)csc2ccc(Cl)cc12 43337,Cc1nc(N2CCC(C)C2CNC(C2CN(C(N)=O)CCO2)=O)[nH]c(=N)n1 43338,c1(C(=O)NCC=CCNC(C(C2CC2)SC)=O)cccc(CS(C)(=O)=O)c1 43339,C1(C(N2CCC(C)(CNC(c3c[nH]c(=NC)s3)=O)C2)=O)CCN(C2CC2)S1(=O)=O 43340,c1(C(N2CCC(C)C(NC(C3(C)CC(C#N)C3)=O)C2)=O)ccc(Cl)c2occc12 43341,n1(CC)cc(Cl)c(C(N2CCCC2C(C)(C)NC(=O)C(COC)N(C)C)=O)n1 43342,c1(C(N(C(CNC(CCOC(C)C)=O)C)C)=O)ccc(F)cc1 43343,C1(C(=O)NCCC(N2CCOCC2)=O)CCN(C(=O)Nc2cc(O)ncn2)CC1 43344,c1(OCC)cccc(C(=O)O)c1COC(c1ccc(NC2CCOCC2)nc1)=O 43345,N1(C(C2(COC)CCCO2)=O)CCCC(N(C(=O)CCn2ccnn2)C)C1 43346,C(=O)(C(C)C(C)C(C)(C)C)NCCC1(CNC(c2c(C)cc(CC)o2)=O)CC1 43347,C(C)(C)(CC(=O)NCC(O)CC(=O)Nc1cnn(CCF)c1)OC 43348,N1(C(c2c(CC)occ2)=O)CC(C(N2CCC3C(OC)CC23)=O)C(F)(F)C1 43349,C(C(C)(C)C(=O)NCCC1CN(C(=O)C(C)Cn2ccnc2)C1)OC 43350,c1(NC(C(N2CCN(C3COC3)CC2)C)=O)ccc(C2CCC(=O)NC2)cc1 43351,C1(CNC(c2cc(-c3ccc(C)s3)[nH]n2)=O)CCC(C)CN1C(=O)C(C)C 43352,Cc1cc(O)cc(C)c1CC(=O)NCC1(O)CC(NC(c2coc(CO)c2)=O)C1 43353,c1(C(N2CC(NC(C(COC)C)=O)C2)=O)ccc(N2CCOC2=O)cc1 43354,Cc1ccc(C(N2CCCCC2CNC(=O)C(C)(C)C(N)=O)=O)c(O)n1 43355,c1(C(N2CCC(C(=O)NCC=C3CCSCC3)(OC)C2)=O)cc(C#N)oc1C 43356,C1(C(=O)NCCOCCN(C)C(c2cccs2)=O)CCCC1S(C)(=O)=O 43357,C1(CNC(c2ccc(NS(C)(=O)=O)cc2)=O)CC(F)(F)CN1C(C1CCCS1)=O 43358,N1(C(CCOC2CN(C(CC3CCC(C)CC3)=O)C2)=O)CCCNC(=O)C1C 43359,C1(C(=O)NC2C3CN(C(C(COC)N(C)C)=O)C2C3)CCn2cnnc2C1 43360,C=CCC(C)C(=O)N1CCC(OCCNC(C2C(C(=O)OC)C2(C)C)=O)C1 43361,c1(COCC(=O)NCC2CCCN(C(c3cccc(F)c3)=O)C2)ccnc(O)c1 43362,N1(C(c2c(C(=O)OCC)con2)=O)CC(C2CCCN(C(=O)C(C)C(C)O)C2)C1 43363,C1(C)(CNC(Cn2c(C)c(Cl)cn2)=O)CN(C(c2cncnc2)=O)CCO1 43364,Cc1cccnc1C=CC(N1CCN(C(=O)CC(C)C(F)F)C(CO)C1)=O 43365,c1(C(N2CCCC(CCC)(NC(=O)C(O)C3CCC3)C2)=O)ccc2nncn2c1 43366,C1(F)(C(=O)NC(C(=O)NC(C)CCC2CC2)CSC2CC2)CCCCC1 43367,C12(CNC(C(CC)c3ccccc3)=O)CC(NC(c3cc(C)[nH]n3)=O)(CCO1)C2 43368,c1(C(C)(C)C)ccc(C(=O)NC2CC(NC(C3CC3(F)F)=O)C2)o1 43369,C1(NC(CCC=CC)=O)CN(C(=O)CN2CCN(S(C)(=O)=O)CC2)CCC1F 43370,c1(C(N(CCCCNC(CC2CCN(C)C2)=O)C)=O)cncc2nc[nH]c12 43371,c1(C(N2CC(NC(C(n3ncc(C)c3)C)=O)C(F)C2)=O)c(F)cccc1Br 43372,c1(N2CCCC(C(C)C)C2)nc(N2CCS(=O)C3(CCC3)C2)nc2cccnc12 43373,C1(NC(c2c(C)cc(C)s2)=O)CN(C(C2CC3(C2)CC3F)=O)CC2(CCC2)C1 43374,c1(N(c2ccccc2)C(C2CCN(C(C)=O)C2)=O)nc(C)cc(O)n1 43375,C1(CNC(C(CCC)O)=O)C2CCC1CN(C(c1cnc3[nH]ncc3c1)=O)C2 43376,c1(CC)cc(N)ccc1C(=O)NCC1CCN1C(C12CC(CO)(C1)OC2C)=O 43377,c1(C(N2CCOCC(NC(CC(C)(C)OC)=O)C2)=O)cc2cc(F)cc(F)c2[nH]1 43378,c1(C(N(C2CN(C(c3nc(C)sc3)=O)C2)C)=O)cc(Br)cn2ccnc12 43379,n1(C(CC)CC)nc(C)cc1C(=O)NCC(C(C)C)NC(C1CCN(C)C1C)=O 43380,C1(CNC(C(CC)(F)F)=O)CC2CCC1N(C(=O)C(COC)NC(C)=O)C2 43381,CC(C)(CNC(C1(C)CCCN1C(=O)CCN1CCOC1=O)=O)C(N)=O 43382,C(=O)(C1=C(C)CCCC1)NC1C(SC)CN(C(=O)C(=Cc2ccc(F)cc2)C)C1 43383,N1(C(C(C)C2(O)CCC2)=O)CC2(C=C(C(=O)NC3CCCN(C)C3=O)CO2)C1 43384,c1(OC)c(C(=O)NCC#CCNC(C2CNC(=O)CC2C)=O)oc2ccccc12 43385,c1(CC)cc(C(=O)NC(CC(=O)N(CC(=O)OC)C)C2CC2)n[nH]1 43386,c1(CC(C)NC(=O)C2=C(Cl)CC2)ccc(CNC(=O)CSc2nncn2C)cc1 43387,n1(CC)nc(C(=O)NC(C)(CSC)C(=O)NCC(=O)OC(C)C)c(C)n1 43388,c1(OC)ccccc1CCCNC(=O)C(=O)NC1CCCNCC1 43389,c1(C(=O)NC2CC2C)ccc(C(=O)O)cc1.C12(CC1)C(C)NC2 43390,N1(C(C=CC(C)(C)C)=O)CCN(C(=O)CCc2ccc(Br)cc2)CC12CC2 43391,N(C(=NCCCN(S(CC)(=O)=O)C)NC(C1(O)CCOCC1)C)CCCOC 43392,CCC(O)(C(=O)N(CC(O)CNC(=O)CN(C)C1CC1)C)c1ccccc1 43393,C1(COC)CC(CNC(C2(C)CCNC2=O)=O)N(C(=O)CCSCC(C)C)C1 43394,C1(CNC(C(C)OCCC(C)C)=O)CCC(NC(=O)COCCCF)C1 43395,CC(C)(CC(F)F)C(=O)NC1CC2CC1N(C(=O)CCc1ccc[nH]1)C2 43396,c1(OC)c(C(=O)NCc2ccc(I)cc2)cccc1Br.c12ccc(nc1)[nH]c2=O 43397,C1(CS(=O)(=O)Nc2ccc(C(=O)OCCOC)cn2)(OC)CCOCC1 43398,N1(C(c2ccn(CC)c(=O)c2)=O)CCCC2CN(C(C3(CC4CC4)CC3)=O)CC12 43399,c1(N(C(=O)CCCn2cccn2)Cc2ccc(Cl)cc2)cccc2c(I)n[nH]c12 43400,Cc1cccnc1C(=O)NCCOCCN(C(=O)Cc1cncn1C1CC1)C 43401,C1(C(=O)NC(CCN(C(c2c(C)onc2)=O)C)C(C)C)CCC(=O)C(C)C1 43402,C12(C(=O)NC(CN(C(C=C(C)C(C)(C)C)=O)C)(CO)CO)CC3CC1C2C3(F)F 43403,Cc1cc(C(F)(F)F)nn1CC(N1CC2CC2(CNC(C2C3COCC23)=O)C1)=O 43404,N1(C(c2ccccc2Cl)C(=O)NC2COC2)CC23CCCC2(COC3)C1 43405,c1(C(=O)NC2C3(NC(c4ccncc4O)=O)CCC(C2)C3)nnn2c1CCCC2 43406,Cc1cc(NC(C2CC(F)CN(C(c3cc(Cl)cnc3Br)=O)C2)=O)cnc1C#N 43407,Cc1c(NC(c2csc(C3CC3)n2)C)ncnc1N1CCOC(C2CC2)C1 43408,Cc1c(-c2nnc(CC3CCCC(C)C3)o2)ccn1C 43409,Cc1c(NCC2CC23CCC3)ncnc1N1CCOC(C(C)(C)C)CC1 43410,C12(NC(CCC(=C)Br)=O)CCC(C1)N(C(C1CC(C3CC3)=NO1)=O)C2 43411,N1(C(C(Cc2ncn(C)c2)O)=O)CCCC2C1CCCN2C(=O)CCOC1CC1 43412,c1(OC(CC)C)ccccc1C(=O)NC1CCN(C(=O)C(F)CC)CC1 43413,CC(C)CC(O)C(C)C(=O)N1CCC(CNC(c2coc(CO)c2)=O)CC1 43414,C1(C(=O)NC(CNC(COC2(C#C)COC2)=O)C)CN2CCCC2CO1 43415,CC(N=c1[nH]c(=NCC(CO)C(F)(F)F)c2[nH]ccc2[nH]1)c1c(F)cccc1Cl 43416,c1(OC)cc(CC(N2CC3CC(N(C(=O)C(C)C)C)C2C3)=O)cc(OC)c1O 43417,C1(CNC(=O)COc2ccccc2)CCN(C(=O)C=C2CC2)C12CC2 43418,c1(NC(C(N2C(C)CC(NC(C3(SCC)CC3)=O)C2)=O)=O)ccc(C)c(C)c1 43419,CCCC(C(=O)N1CC(C(=O)NCC2CCC2C)C1)OC 43420,Cc1cc(C(=O)NCCN2CCC(NC(=O)CC3CCC(=O)N3C)CC2)nn1C 43421,C1(C(N(CCC(=O)NCc2c(CC)c[nH]n2)CC)=O)CNC(=O)CC1C 43422,c1(OC)ccccc1C1CC1C(=O)N(CC(C)(C)NC(c1nn(C)cc1C)=O)C 43423,N1(C(CC2CCN(C(C)=O)CC2)=O)CCOC2CN(c3nccc(C)n3)CC12 43424,n1(C2C(C)CCC2)nc(CO)nc1-c1ocnc1CN(C)C(=O)OC(C)(C)C 43425,c1(C(=O)OC)ccc(F)c(C(=O)NC2CCN(C(=O)C=CCN(C)C)CC2O)c1 43426,C1(C(N2CC(C)(NC(c3cc(OC)n[nH]3)=O)C2)=O)(C(=O)OC)CC1S(C)(=O)=O 43427,c1(OC)cc2[nH]ncc2cc1C(N1CCC1C(=O)Nc1[nH]nc2cnccc12)=O 43428,C1(CNC(Cc2cc(OC)no2)=O)CC2CCC1N2C(C1CN(C)C(=O)N1)=O 43429,C1(C(N2CC3C(NC(Cc4c(C)cc(F)cc4)=O)(C3)C2)=O)CN(CP(C)(C)=O)C1 43430,n1(CCOC)cc(C(N2CC(NC(=O)Cc3cncs3)CC(C)C2)=O)ccc1=O 43431,C1(N(C(C(CCC)OCC)=O)C)CC2CCC(C1)N2C(=O)C(C)c1ccsc1 43432,C1(CNC(C(C)OCCCC)=O)CC2(CC(NC(=O)CS(=O)(=O)N(C)C)C2)C1 43433,c1(ONC(C2CC3(CC(NC(CCCN=[N+]=[N-])=O)C3)C2)=O)ccc2c(c1)COC2 43434,N1(C(C2CCN(CC(C)C)CC2)=O)CC(NC(=O)Cc2cnns2)CC12CCC2 43435,Cc1cc(C(=O)NC2CC3CC2N(C(C2(CF)CC(F)(F)C2)=O)C3)cnc1O 43436,c1(C(=O)NCC2N(C(C(C)C#N)=O)CC2)cnccc1C(F)(F)F 43437,c1(CCC(N2CCCC(NC(C(C)OCOC)=O)C2)=O)cccc(F)c1F 43438,C12(CC(=O)NCCCCNC(c3nccc(N(C)C)c3)=O)CCCCC1C2(F)F 43439,C1(CNC(COc2cccc(C(C)C)c2)=O)Cc2ccccc2CO1 43440,N1(C(C(C=C=C)C)=O)CCCC(C2CCN(C(=O)CCC(=O)OC)CC2)CC1 43441,c1(OC)cccc(C(=O)NC2CC(NC(C3CCC(C(F)(F)F)C3)=O)C(O)C2)c1 43442,Cc1cn(C)nc1C(N1CCCCC1CC(N1CCCC1(C)CO)=O)=O 43443,c1(OC)ccc(Cl)c(C(=O)NC2CCC(NC(c3cnc(Cl)n3C)=O)CC2)n1 43444,C(=O)(C(C)(C)CNC(=O)CCc1ccc[nH]1)NC1CC(CCOC)C1 43445,Cn1cnc2sc(C(=O)NCC(C3CC3)NC(C3CSCC(=O)N3)=O)cc12 43446,N1(C(C(C)OCC)=O)CCN(C)C(CNC(C2(c3ccccc3)CC(O)C2)=O)C1 43447,c1(C(=O)NCC(CN(C(Cc2c(C)cccc2)=O)C)O)ccc2c[nH]nc2c1 43448,C1(NC(C=CCCC(C)C)=O)CCCN(C(c2cnn(C3CC3)c2)=O)CC1 43449,c1(NC(c2c(OCC#C)nccc2)=O)cc2c(C)cc(=O)[nH]c2cc1C 43450,c1(CCC(=O)NCC(CNC(C(C)CN2CCCCC2)=O)O)ccc(O)cc1 43451,CC(C)(CN=c1[nH]cnc2ccc(O)cc12)c1nc[nH]n1 43452,N1(C(c2c(C)cn(C)n2)=O)CC(NC(C2COCC(C)O2)=O)C2(CCCC2)C1 43453,Cc1cc2c(C(=O)NC3COCC3NC(c3cc(CO)[nH]n3)=O)nccn2n1 43454,C1(C(N(CCC(C)NC(c2cc(O)nn2C)=O)C)=O)CCC2(CCCCC2)C1 43455,CCCCC(C)CCC(=O)NCC1COCCN1C(c1ccc2nccn2n1)=O 43456,N1(C(C(C)C(F)F)=O)CC(CNC(C2(c3cccc(C#N)c3)CC2)=O)CC1(C)C 43457,N1(C(C=CC2COC(C)(C)O2)=O)CC(NC(=O)CC2CC2)CC2(CCC2)C1 43458,c1(C(N2CCCC(C(C)NC(c3ccc(Cl)cn3)=O)C2)=O)cc2n(c1)CCOC2 43459,c1(-c2cnc(CNc3cnc(N(CC)CC)s3)s2)ccc(F)c(C)c1 43460,C(=O)(C1=C(F)CN(C(=O)Cc2csc(C)c2)CC1)N1C(CF)CC(OC)C1 43461,C1(C(=O)OCC)CC2(CCN(C(c3c(C(F)(F)F)cccc3F)=O)CC2)C1 43462,n1(C(C)C)cc(C(N2CCC3(CC3NC(=O)C(C)n3cncn3)C2)=O)ccc1=O 43463,c1(C(N(C2CCCC(NC(C3(C)C=CCCC3)=O)C2)C)=O)cnc2[nH]ccc2n1 43464,Cc1cnc(S(C)(=O)=O)nc1N1CCC2(C(N3CC(CO)C(O)C3)=O)CC2C1 43465,N1(CCC)CCC(C(=O)NC2CN(C(=O)OC(C)(C)C)C2)C(O)C1 43466,CC1Cn2nc(C(=O)NCCCCCNC(=O)C(F)OC(F)(F)F)cc2C(=O)N1 43467,c1(CCC(=O)NCCC(C)NC(=O)CC2COCCN2)ccc(F)cc1Cl 43468,C(=O)(C(CCC(C)C)NC(=O)CCC1CCCCC1)Nc1ccc(OC)c(C)c1 43469,c1(N(C)C)ncnc(NC(C2COCCN2C(=O)OC(C)(C)C)=O)n1 43470,c1(N2CC(NC(C(C3CCOCC3)C)=O)C(C)(C)C2)ncc(Br)cc1C#N 43471,C(N=c1[nH]c(=NCCc2nccc(O)n2)c2[nH]ccc2[nH]1)c1c(C#N)cccc1 43472,O=C(CC1(C(=O)O)CCc2ccccc21)NC(c1cc(Br)ccc1F)C1CCCO1 43473,CC(C)CC(O)CC(=O)NCc1occc1C(=O)NCCn1cccnc1=O 43474,c1(C(CNC(C2(C(C)C)CCC2)=O)NC(c2cc(CC)on2)=O)cccc(C)c1 43475,c1(OC)cc(NC(c2cnc(CNC(=O)CC3CCC(C)O3)nc2)=O)ccc1O 43476,c1(OC)ccccc1NC(=O)C(C1CN(C(C2(SC)CCC2)=O)C1)OC 43477,C1(c2nnnn2C2CC2)(NCCC(=O)NC2CCCCC2)CCC(=O)NC1 43478,N1(C(c2nc(C)oc2C)=O)CCOC2CCN(C(C3CCC(F)CC3)=O)CC12 43479,N1(C(C(C)SCC)=O)C2CCC1CN(C(=O)Cc1ccccc1SC)C2 43480,C1(C(=O)Nc2c(C)cc(Sc3nccn3C)cc2)CCc2ccnn2C1 43481,C1(C(N(CC(=O)NC)CC)=O)CC12CCN(C(=O)Cc1ccc(C)nc1)CC2 43482,C1(C(=O)NCC(CN(C(=O)CNC(=O)C2CC2)CC)(C)C)CCCC2CCCN12 43483,C(=O)(CCCC(F)F)NC(c1nc(C(N2CCN(CCCC#C)CC2)=O)cs1)=O 43484,N1(C(CC=CCC)=O)CC2ON=C(CNC(C3CC(S(C)(=O)=O)C3)=O)C2C1 43485,N(C(=NCC)NCC(=O)NC1CCCCC1)C(C1CCOCC1)C#C 43486,Cn1ncc2c(C(=O)NC3CN(C(=O)Cn4cc(Cl)cn4)CCC3F)ccnc12 43487,CC1(C)CC(C(N2CCCCC2CCNC(=O)CC2COC(=O)C2)=O)CO1 43488,CC12CN(C(=O)C3=COCC3)C(C(=O)NC(c3cscn3)CO)(C1)C2 43489,N1(C(c2c(C)n(C3CC3)cc2)=O)CCOCCC1C(C)C 43490,C1(C(=O)NC(C)(CC(=O)O)c2cccc(F)c2)CCn2nncc2C1 43491,C12(NC(CCCSC)=O)CCN(C(c3cc(O)nn3C)=O)CCC1C2 43492,Cc1cccc(C(O)C(=O)NCCC(C)NC(c2c(C)[nH][nH]c2=N)=O)c1 43493,C(C(S(C)(=O)=O)C1CC1)NC(c1ncccc1F)c1n(CCCOC)nnn1 43494,C1(C)(C(=O)NCC2C(C)CN(C(c3ccc(F)cn3)=O)CC2)CCC(C)(C)CC1 43495,CCC(C)CC(C)C(=O)N1CCC(C)(NC(c2cc(=O)c(OC)cn2C)=O)C1 43496,N1(C(C(C)=C(C)C)=O)CCCC1C1(NC(=O)COC2CC=CC2)CC1 43497,N1(C(c2c(OCC#C)nccc2)=O)CCCC(C2CCN(CCO)C2)C1 43498,N1(C(C(C)SC)=O)CCC(NC(=O)COc2ccc(F)cc2F)C(F)(F)CC1 43499,C1(NC(c2n[nH]c(CC)c2Cl)=O)CCN(C(=O)CSCC(=O)OC)CC1C 43500,Cc1ccccc1CN1CCCC1CN(C(=O)CCCOCCN(C)C)C 43501,N1(C(c2cc(CNC(c3c(CC)nn(C)c3)=O)sc2)=O)CCN(C)C(C(C)C)C1 43502,N1(C(CSc2c(C)n[nH]c2C)=O)CCC(NC(=O)CN2C(=O)CCC2=O)CC1C 43503,N1(c2nnc(C)s2)CCC(CNC(c2ncnc3c(C)csc23)=O)C(F)(F)CC1 43504,N1(c2n(CC(C)C)c(-c3cnc(O)nc3)nn2)CCC2CCCC12C(F)(F)F 43505,C1(O)(CC(N2C(CN(C(=O)C=CSc3nc[nH]n3)C3CC3)CCC2)=O)CCCCC1 43506,CC1(CCCO)CCCN1C(=O)Cn1cc(I)nn1 43507,c1(CC(N2CC(NC(c3cc(C)sn3)=O)C(F)C2)=O)cc(F)c(C)cc1F 43508,C(C(CC(C)C)C(=O)N(C)Cc1ccoc1)NC(C=CC(=O)NCCOC)=O 43509,c1(C(=O)NCC(CO)NC(C(COC)(C)OC)=O)c(C)cc(Cl)cc1N 43510,C(=O)(C(C)(F)C(F)(F)F)NCC1CCN(C(C=Cc2ccc(C)cc2)=O)C1(C)C 43511,C1(C)(CNC(c2c(C)nn(C)c2)=O)CN(C(=O)C=Cc2ccc(Cl)s2)CCO1 43512,C1(N(C)C)CCOC(C(N2CCN(C(C3COCCO3)=O)CC2)=O)C1 43513,C(=O)(CC(O)CC(C)C)NCCC(CC)(C)NC(=O)C(C)CC(F)F 43514,C12(C(=O)NCC3(C(F)(F)F)CCN(C(C(N)=O)=O)C3)CC(CO)(C1)OC2(C)C 43515,CCCCCC(C(=O)N1CCC(C)(NC(c2onc(C)c2C)=O)CC1)C(C)C 43516,C(=O)(C(CCC(N)=O)n1cc(CN2CCCC2CO)nn1)NCc1nnc(C)o1 43517,c1(C(=O)NC(C)CCCNC(=O)C(c2cnccn2)C)nc(Cl)sc1Cl 43518,CC1(C)CCCC(CNC(C2CCC(CNC(C3SCCS3)=O)O2)=O)O1 43519,CC(C(C)(C)C(=O)NCCC(=O)NC(C)(C)C)NC(c1cc(Cl)ns1)=O 43520,C12(NC(C(CC=CC)CC)=O)CCC(CN(C(c3ccc(OCC)nc3)=O)C1)C2 43521,Cc1cccc(C)c1CNC(C1(NC(=O)C(CO)NC(=O)CC#N)CCC1)=O 43522,C1(NC(C2(CC)COC2)=O)CC(NC(=O)C(C)OCC(C)C)CC1O 43523,C1(C(C)NC(C(C)CO)=O)CCN(C(c2cn(-c3ccccc3Cl)nn2)=O)CC1 43524,Cc1nc(C)c(CNC(C2CC2C(C)NC(c2ccc[nH]2)=O)=O)[nH]1 43525,CC1CC(C(c2ccccc2)=O)CCN1C(C1CCCN1C(N)=O)=O 43526,C=C(COC(C)C)CCNC(CCNC(C1(C)CC1)=O)=O.c1(C=O)cccs1 43527,c1(C(=O)NC2CCCC(NC(c3c(C)sc(Cl)n3)=O)C2)cn(C)c2ccccc12 43528,C1(NC(C(C)C2CCC2)=O)C(C)CCN(C(c2ncc(C(F)(F)F)n2C)=O)C1C 43529,C1(C)(C(=O)NC(C2CCOC2)(C)C)CCCN(C(c2cccc[n+]2[O-])=O)C1 43530,C(CN(C)C)(CN=c1nc(N(C)Cc2nc(=N)[nH][nH]2)cc(C)[nH]1)OCC 43531,c1(C(=O)NC2C(C)CCN(C(c3cc(Cl)cnn3)=O)C2)ccc2cncn2c1 43532,C1(C(=O)NCCc2cc(C(=O)O)no2)(OC)CCS(=O)(=O)C1 43533,C1(C(N2CCCC(F)(C(=O)NCc3snc(C)n3)C2)=O)CC(=O)CC12CCC2 43534,N1(C(c2cn(CCCOC)nc2)=O)CC(O)CC1C(F)(F)F 43535,c1(OCCOC)ncccc1C(=O)NCCC(C)NC(=O)CC1CCC(C)(C)C1 43536,N1(C(C(C)OCC=C)=O)CC2CC1C2CNC(=O)C(C)COC 43537,c1(OCCC(N2CCC(C(C)NC(CCC#C)=O)CC2)=O)cc(C)cc(C)c1 43538,C(=O)(CC(C)(C)C1CC1)N(C1CC1)CC1N(C(C(c2ccc(Cl)s2)C)=O)CCC1 43539,C1(CNC(C(C)SC)=O)CN(C(c2ccc(C(F)(F)F)cc2N)=O)CC1(F)F 43540,C1(CCNC(C(c2cscn2)OCC)=O)CCCN1C(=O)CC1CC(CF)C1 43541,c1(C(=O)NCC2C3N(C(c4c(C)cc[nH]4)=O)C(CC3)C2)cc2ncccc2o1 43542,C1(C(=O)NCC(C2CCCCC2)NC(C(C)n2ccnn2)=O)CCCC(C)(C)O1 43543,C(=O)(C(CO)C(F)(F)F)N(C)CC=CC(=O)NCC1CC(F)C1 43544,N1(C(Cc2c(C)ncnc2O)=O)CC(C)CN(C(=O)C(F)=C2CCCC2)CC1C 43545,c1(N(CCCSC)C)nc(=NCc2ccns2)[nH]c2c1CC(C)CC2 43546,C1(C(N2CCN(C(C3CN(C(C(C)(C)O)=O)C3)=O)CC2)=O)CC2(C1)CC(C#N)C2 43547,N1(CC(N2CCC(COC)C2)=O)CCN(C(=O)Cc2ccccc2I)CC1=O 43548,C1(NC(c2c(C)nc(CCC)o2)=O)COCCN(C(c2ccc(C#N)s2)=O)C1 43549,O=C(N=c1ccn(CCCC2CCCO2)[nH]1)C1=C2CCCN=C2NC=C1 43550,C1(CC)CN(C(C2C=CCC2)=O)CCC1NC(c1ccc(=O)n(C)c1)=O 43551,C1(C(=O)NC(CC)(C)C2CC2)CN(C(c2ccc(OCC)s2)=O)CC1C1CC1 43552,c1(OC(C)C)ccc(COC(C2CC2(Cl)C(=O)O)=O)nn1 43553,C12(C(N(C)CC3(OC)CCC3)=O)CC(C)(CN1C(=O)Cn1cc(C#N)cn1)C2 43554,C(C(CCC)C(=O)NC1(C)CCCCCC1)NC(C=CCCC)=O 43555,c1(C(N2CCC3CCCC23CNC(C2(CO)COC2)=O)=O)cn2cccnc2n1 43556,C12(NC(CCCC#C)=O)CCCCC1CN(C(C1CCCC1(C)C)=O)C2 43557,Cc1cccnc1CC(=O)NC1(CCC(=O)NOCC2(C)CCC2)CCCC1 43558,C1(C(N(CCCNC(=O)CCc2cccc(O)n2)C)=O)CCC2CCCCN12 43559,C(=O)(C(C)(C)CC1CCOC1)NC1C(NC(=O)NC)CCC1 43560,N1(C(CN(C)C)=O)CCC2CN(C(c3cc(C4CCOCC4)[nH]n3)=O)CCC12 43561,N1(C(C2(CC#C)CCCO2)=O)CCC(NC(=O)C(CCO)N(C)C)CC1 43562,CC(C)(CC(F)F)C(=O)N1C2CCC1CC(NC(c1ccc3cc[nH]c3n1)=O)C2 43563,CCC(CCCC(=O)NCC1(CF)CCC1)NC(c1cc(OC)n(C)n1)=O 43564,c1(CC(=O)NC2C(CNC(c3c(OC)scc3)=O)CC2)nn(C)c2ccccc12 43565,C1(NC(C=C(C)C)=O)CCN(C(c2ccc(Br)cc2C)=O)C2CC12 43566,N1(C(C(CC)N(C)C)=O)CCC(NC(C2CN3CCC2CC3)=O)C12CCCC2 43567,N1(C(COCC)=O)CCC(NC(c2cc3n(n2)CCO3)=O)C(C(C)C)C1 43568,O=C1CCC(CNC(c2ccc(CNC(=O)CC3CCCO3)s2)=O)O1 43569,C1(NC(=O)CN2C(=O)C=CC2=O)CN(C(c2cccc(CO)c2F)=O)CC1(F)F 43570,N1(C2(C(=O)OC(C)C)CC2)CC(C)(CNC(C2(CF)CCC2)=O)CC1(C)C.C(F)(F)F 43571,c1(NC(C2(C)N(C(CC(OCC)OCC)=O)CC2)=O)c(Cl)nc(C)nc1Cl 43572,C1(C(N(C2CCCOC2)CC)=O)CC12CCN(C(C1CC3CC(=O)C1C3)=O)CC2 43573,N1(C(C(C)=C2CC2)=O)CC(C)CN(C(c2nc[nH]c3nccc2-3)=O)C(C)C1 43574,c1(Oc2ccc(C(=O)OC)nc2I)c([N+](=O)[O-])cc(C(F)(F)F)cc1[N+](=O)[O-] 43575,n1(C(C)C)cc(C(=O)NC23CC(NC(=O)C(F)F)(C2)C3)cn1 43576,C(CCCC(F)(F)F)OC.N1(c2n3c(nn2)CCC3)CC2CCC2(OC)C1 43577,C1(CC)(CC)CCN1C(c1n[nH]c(C)n1)C(=O)NC1(C)CC1 43578,CCCC(O)C(=O)NC1(C)CN(C(=O)COCC(=O)OC)C1 43579,C(CN=c1[nH]c2ccc(Br)cc2s1)NC(=O)CCNC(N)=O 43580,CC(C)(C)CCCNC(=O)NCCN1CCCC(N(C)C)C1 43581,C1(N(C(C(=O)NC(C)C)c2cnsc2)C2CC2)CCS(=O)(=O)C1 43582,C(CCC(=O)N1CCN(CCO)C(C)C1)(C(C)C)NC(c1c(C)coc1)=O 43583,C12(NC(C(CC=C)NC(=O)C=Cc3ccccc3C)=O)CCC(C1)C(O)C2O 43584,C(=O)(CC(C)(C)CNC(=O)CC1CCCCC1O)N(C)CC 43585,Cc1ccccc1C(=O)N(C1CN(C(c2cnn(CC(F)F)n2)=O)CC1F)C 43586,N1(C(C=CC=CC)=O)CC(CNC(=O)Cc2cc(C(F)(F)F)co2)OC2CCCC12 43587,C1(C)(CNC(C2C=CC(NC(C(C)n3cccc3)=O)C2)=O)NC(=O)NC1=O 43588,c1(-n2c(-c3cn(C4COCC4F)nn3)nc(COC)n2)ccnc2c1cnn2C 43589,N1(C(c2c(C)occ2)=O)CCC(NC(c2cnc(N(C)C)cn2)=O)C(O)C1 43590,CC(C)C(O)CC(=O)NCC1CC(F)CN1C(=O)C=Cc1cc[nH]c1 43591,C1(C(=O)NCc2cnco2)(NC(=O)Cc2ccsc2)CCCCC1 43592,CC(C(=O)NC1CN(C(c2ncccc2N)=O)CCC1CO)C(C)(C)C 43593,C(=O)(C(F)C(F)(F)F)N(CCC)CCNC(C1CCC1C(C)(C)C)=O 43594,C(=O)(C1CCc2cccnc21)NCC1(F)CN(C(C(C)NC(=O)OC(C)(C)C)=O)C1 43595,N1(C(CCSCCCC)=O)CC(CNC(c2cc(OC)cnn2)=O)CC1C 43596,c1(OCC(=O)N(CC(CNC(C(C)O)=O)O)C)cccc(Cl)c1 43597,c1(NC(c2cccc(NC(c3cnc(Cl)nc3)=O)c2)=O)cc(Br)cnc1O 43598,C1(C(N2C(C(C)(C)NC(c3[nH]cc(CC)c3)=O)CCC2)=O)CCCN(C)C1 43599,Cn1c(C(N2CCC(C)(CNC(=O)C(O)C(F)F)CC2)=O)c(Cl)c2ccccc12 43600,CCC(CC)C(=O)N1C(CNC(c2cc(CC(C)C)nn2C)=O)CC2CC12 43601,c1(C(=O)NCC2CC(NC(CC(=C=C)C)=O)C2)cc(C)ccc1OCC 43602,Nc1cc2ccccc2cc1C(N1CC(CNC(C2CC3CC3C2)=O)C1)=O 43603,C1(NC(C2=C(C)OCCC2)=O)C2CC(CN(C(=O)C(F)=CCCF)C2)C1CO 43604,C1(C(N(C2CCN(C(=O)CCCc3cnn[nH]3)C2)CC#C)=O)CCN(CC)C1 43605,C(=O)(C1=NNC(=O)C1)NCC(C)(C)NC(C1CN(C2CCOC2)C1)=O 43606,C1(C(=O)NCC(CNC(CCCOCC)=O)C)CCCC12OCCO2 43607,N1(C(CC2(OC)CC2)=O)CC(C)CN(C(=O)COc2ccc(C)c(C)c2)C(C)C1 43608,c1(CNC2C(C(N(CCC(F)(F)F)CC)=O)CCC2)ccc(F)c(F)c1Br 43609,C1(C(N(CC(C)(C)CO)C)=O)C(C2CC2)CCN1C(c1ncccc1Cl)=O 43610,Cc1nc(C)c(C(N2CCC(OCCNC(c3cccc(F)n3)=O)C2)=O)[nH]1 43611,C1(NC(C(CC=CC)CC)=O)CCCCCN(C(c2ncsc2CC)=O)C1 43612,Cc1nn(CC(=O)NCCCN(C)C(C2CCC(C3CC3)C2)=O)c(=O)n1C 43613,c1(C(CC)NC(=O)CSCCNC(=O)C(F)n2ccnc2)ncnn1C 43614,C1(CCNC(C(C)SCCCC)=O)(OC)CN(C(C2(c3ccnn3C)CC2)=O)C1 43615,c1(NCCCc2n(C)ncn2)[nH]c(=NCCc2ncc[nH]2)nc2c1cnn2C 43616,Cc1c(C(=O)NC(CNC(=O)CCc2cccn2C)CO)noc1C1CC1 43617,c1cc(NCC2CCC2C2CC2)cc(-n2cnnn2)c1 43618,c12cc(N(C)CCn3cccn3)nc(n1)CN2C.CCC(C)OC 43619,Cc1oc(C(C)(C)C)cc1C(=O)NCCC(C)NC(=O)C(C)(F)c1ccccc1 43620,c1(CC(=O)N(CCOCCSCC)C)ccnn1C.C(CC(=O)NC)S 43621,Cc1cc(C(=O)NC(C)(C(=O)NCCc2cc(C)ns2)C2CCC2)ccc1C#N 43622,c1(CN2C(C(=O)NC(c3cc(C)cc(C)c3)C)CC(O)C2)cccc(C=O)c1Br 43623,C1(C(N2CC(NC(C(C)Cn3cccn3)=O)C2)=O)C2C3CCC(C3)C12 43624,C1(CNC(C(C=C)(C)CC)=O)CN(C(C2OCCO2)=O)CCC1(F)F 43625,c1(C(=O)NCC(CNC(=O)OC(C)CF)OC)ccc(=NC(=O)OC(C)(C)C)[nH]n1 43626,C1(NC(=O)Cc2ccc(O)cn2)CN(C(=O)C2=CCCSC2)C2(CCCOC2)C1 43627,N1(CC#C)CCN(C(C2CCN(C(C3CCCCO3)=O)C23CC3)=O)CC1=O 43628,c1(-c2ccc(NC(C3N(C)CCC3)=O)cc2)cc(O)nc(O)n1 43629,Cc1ccnc(CC(=O)N(C)CC2CCCN2C(=O)CCc2ncc(F)cn2)n1 43630,c1(SC)ncc(-c2cccc(NC(COC)=O)c2)cc1O.N12CCC1C2=O 43631,CC(C(=O)N1CCN(CCNC(C2CCCN(C(=O)C(N)=O)C2)=O)CC1)C(F)F 43632,N1(C(C=C(C)C(F)F)=O)CC(NC(c2ccncc2C(F)F)=O)CC(O)C1 43633,C1(C)(C(=O)NCC2N(C(c3c(CC)nc(C)o3)=O)CCOC2)CCC12CCC2 43634,N1(C(=O)NC)CCC(C(=O)NC(CNC(c2cccn2C)=O)CO)CC1 43635,c1(NC)cnc(C(N2CC(CNC(c3n[nH]cc3Br)=O)C(C(F)(F)F)C2)=O)cn1 43636,Cn1c(C(=O)N(CCCN2CCc3ccccc32)C(C)(C)C)cc2ccsc12 43637,C=CC(C)(C)CCCNC(C1(NC(C2CC(=O)OC2(C)C)=O)CSC1)=O 43638,CCCC(C)CCCC(=O)N1CC(O)(CN(C)C(c2cc(Cl)ns2)=O)C1 43639,c1(C(C)=O)cc(C(N2CC(CCCCNC(c3csc(CO)n3)=O)C2)=O)no1 43640,CC1(CC(N2CC(O)C(O)C2)=O)CCN(C(=O)C=CC2CCOC2)C1 43641,Cc1ccccc1C1(C(=O)NC2C3CC2N(C(=O)COCCN(C)C)C3)CC1 43642,C12(C(=O)OC)CCC(C(N3CCC(C)C(NC(=O)C(C)SC)C3C)=O)(CC1)CC2 43643,N1(C(CCSCCCC)=O)CCC2CCCC12C(=O)NC1CC2(C1)CC(C#N)C2 43644,C1(C(N(CC(CNC(c2c(C)nc(O)[nH]2)=O)(C)C)C)=O)CC2CCCCC2O1 43645,C1(C(C)C)C(=O)NCCN1C(C1C2CCC(C2)N1C(c1cc(C#N)cs1)=O)=O 43646,n1(CC(N)=O)cc(C(=O)NCC(C2CC2)NC(c2n[nH]cc2Br)=O)nn1 43647,N1(C(C=CCCC(C)C)=O)CCCC(NC(c2ccc(CC(C)(C)C)cc2)=O)C1 43648,c1(C(N2CCC(NC(=O)C(O)Cn3cncn3)C2)=O)cc2sc(Cl)cc2s1 43649,N1(CCC)CC(C(=O)NC2(CNC(=O)CCCC3CCCC3)CCCC2)CC1=O 43650,N1(c2snc(C(C)C)n2)CCN(C(=O)NC(C)C(C)n2cccn2)CC1 43651,C1(C(=O)NCCc2nc(CC)[nH]n2)CCN(C(=O)c2cccnn2)O1 43652,c1(CCCC)cc(=NC(=O)Cc2csc(NC(=O)N(C(C)(C)C)CC)n2)[nH]n1C 43653,CN1CC(C)(C)CC1C(N1CC(NC(=O)C2=C(Cl)CC2)C(O)C1)=O 43654,C1(C(=O)NCC(CC(=O)NC(C)C(C)C)OC)CC2(CCC2O)C1 43655,c1(CC)nc(CC(=O)NCC(C2CCOC2)NC(=O)COCc2cccs2)cs1 43656,N1(C(CC=C)=O)CC(NC(C2(C(=O)OCC)CCCO2)=O)C(c2cnn(C)c2)C1 43657,C1(NC(c2ccc(C(F)(F)F)nc2)=O)CCOCC1NCC=CC=C(Cl)Cl 43658,N1(C(C2C(C)C2)=O)Cc2ccccc2C(NC(c2cccc(C(C)(C)C)n2)=O)C1 43659,CS(=O)(=O)CCC(=O)NCC12CCC(CC1)N2C(c1cncc(OC2CC2)c1)=O 43660,C1(CNC(c2c(Cl)nsc2Cl)=O)CC(F)(F)CN1C(C1CCCC12CC2)=O 43661,c1(C(=O)NC2CN(C(C=CSC)=O)CC2C(F)F)cccc2[nH]ccc12 43662,N1(C(C(C)c2ccsc2)=O)CCOC2(CCN(C(c3ccc(F)o3)=O)CC2)C1 43663,CCCC(C)(O)CC(=O)N1CCCCC(CNC(=O)CCNC(C2CCC2)=O)C1 43664,c1(OC)cccc(C(=O)NC2CC(CCNC(C3CCC(=O)NC3)=O)C2)n1 43665,Cc1nc(CC(=O)N(C)CCN(C(=O)C2=CCCC2)C)c(Cl)s1 43666,c1(OC)ccc(Cl)c(F)c1C(=O)NC(C1CCOC1)CNC(c1occc1C)=O 43667,c1(OC)cc(C(=O)N(C2CCN(C(c3onc(C)c3C)=O)C2)C)cc(N)c1O 43668,c1(CC)nc(C(=O)N(C)CC2(NC(=O)CC3(CO)CC3)CC2)cs1 43669,Cc1occc1S(C)(=O)=NC(=O)CC1(C)CC1 43670,C(c1ccc([N+](=O)[O-])s1)=CC(=O)NC1CN(C(C(C)(C(C)C)OC)=O)CC1O 43671,C(=O)(CC(C(F)(F)F)NC(c1ccc2ccoc2c1)=O)NC(CCC)C1CCC1 43672,N1(C(COC2(C)CCC2)=O)CCC2(CCN(C(C3CCC3C(F)F)=O)C2)C1 43673,C1(CNc2cncc(C)c2)CCC(C)N(C(=O)CCc2cncnc2O)C1 43674,C1(CC(=O)N(C2CSC2)CCN(C)CCO)CCCCC1NC(=O)CC1CC1 43675,N1(C(CC2CC(=C)C2)=O)CCC(N2CC(O)C2)C1(C)C.N12CCC(C1)C2=O 43676,CN1CCC(C(=O)NCC2CCC(NC(=O)CN3CCC(O)CC3)C2)CC1 43677,Cc1cc2sc(C(N3CC(F)(CNC(=O)C(C)n4ccnc4)C3)=O)cc2s1 43678,N1(C(C2(C#C)CN(C(=O)C(O)CN3CCCC3)C2)=O)CCC(C2CCC2)C1 43679,c1(C(N(CC(C)NC(c2cnc(Cl)c(N)c2)=O)C)=O)cnc2ncc(Cl)cn12 43680,c1(CC)cccc(C(=O)N(CC(C)CNC(=O)C=CC2CCCN2C)C)c1F 43681,c1(C(=O)NCCCCCN(C(CC2(CC)CC2)=O)C)c(C(C)C)cccc1C 43682,c1(NCC(=O)N(C2CCCC2c2ccccc2)c2cn(CC)nc2)cccc(=O)n1C 43683,CS(=O)(=O)C(CNC(=O)CC1CCCOCC1)CNC(C1CC(F)(F)CS1)=O 43684,C1(NC(C2CCCN(CCC)C2)=O)C2CC1CN(C(=O)CCN1CCCC1=O)C2 43685,C(=O)(CC(C(C)(C)C)NC(=O)Cc1cncs1)NCC(CN(C)C)O 43686,Cc1cncc(C(=O)NCC2CCN(C(=O)Cn3ccc(=N)[nH]3)C2)c1 43687,C1(C(=O)OC)CCc2cc(OC)ccc2N1C(C1(C)CC1(F)Cl)=O 43688,c1(C(=O)NC2(CC=C)CCN(C(=O)C(C#N)C(C)C)C2)c(F)cccc1Cl 43689,N12CCN(C(C(=O)OC(C)(C)C)C1)C2=O.c1(CC(C)C)nc(-c2ccccc2)no1 43690,C(=O)(C(CNC(c1n[nH]c2c1COC2)=O)CC(C)C)Nc1c(C)ncnc1 43691,C(=O)(C(C)(C)C(C)NC(c1c[nH]c(C)cc1=O)=O)Nc1c(OC)cccc1 43692,c1(C(N(CCNC(C2(CC=C)CC2)=O)C)=O)cccc2ncnc(O)c12 43693,N1(C(CC2CCCC(NC(CCCCC=CC)=O)C2)=O)CC(C)CCCC1C 43694,C1(NC(c2c(C)noc2)=O)CCN(C(c2cn(C3CCOC3)cn2)=O)CC1(C)C 43695,CS(C)(=O)=NC(=O)C(=O)NC1CN(C(C2CCCN2C(C2CCCC2)=O)=O)C1 43696,c1(C(=O)NCCC(C)NC(C(C)=C2CCC2)=O)ccc(-n2cccc2)cc1 43697,N1(c2cc(NCCOCCOC)nc(C)n2)C2CCC1CC(N(C)C)C2 43698,CC1CC2(CCN(C(=O)CCN3CCCC3=O)CC2)CN1C(C1CCC1(C)C)=O 43699,c1(OC)ccc(O)cc1C(=O)NCC1(NC(c2nnn(C)c2C)=O)CCOC1 43700,N1(C(COC(C)=O)=O)CCCC12CCN(C(=O)Cn1cc3ccccc3n1)C2 43701,C1(CC)CN(C(c2ncc(F)cn2)=O)CC1NC(=O)C(C1CC1)SC 43702,C1(CNC(C(CC)CC)=O)CCC(C)(C)CN1C(c1cccc(C2CC2)c1)=O 43703,CC(C)C(F)C(=O)NC1CCCN(C(c2cc(C3CCC3)[nH]n2)=O)C1 43704,C1(C(=O)NCCC2N(C(C(F)=C(C)C)=O)CC(F)(F)C2)CCc2nc[nH]c2C1 43705,C=C(C)C(C)(O)C(=O)NC(C)CN(C(c1cc(Br)ccn1)=O)CC 43706,C12(C(=O)OC(C(=O)NCC)C)CCC(CC1)C2(C)C 43707,C1(CC)OCCC1NC(c1ncc(I)s1)C 43708,c1(C(=O)NCC2CCN(C(C(C)O)=O)C2(C)C)ccc2cc(Cl)ccc2n1 43709,c1(C(=O)NC(C2CCCN(C(C3CS(=O)(=O)C3)=O)C2)C)cnc2sccn12 43710,c1(CC)cnc(Cl)[nH]c1=NC(CNC(c1ccc(C)c(Cl)c1)=O)c1ccccc1 43711,C1(CNC(C(CC)NC(N)=O)=O)CCCN(C(C2(CO)CCC2)=O)CC1 43712,N1(C(c2c(N)c(Cl)ccc2)=O)CCN(C(c2ccc3[nH]ccc3c2)=O)CC(O)C1 43713,CC1C(C(=O)N(C(C)(C)CC(N2CC3C=CC2CC3)=O)C)=NOC1C 43714,c1(C(N(C2CCN(C(c3cnnc(O)c3)=O)C2)CC)=O)cnn2ccn(C)c12 43715,C#CCCC(O)CCNC(=O)CC1CC1CNC(=O)C(CC)(CC)OC 43716,N1(C(c2nccc(CC)c2)=O)CC2CCC2(NC(c2cnc(C3CC3)s2)=O)C1 43717,N1(C(C2CC(OC)CN2C(=O)Cc2cccc(O)c2)=O)CC(F)(F)CC1CO 43718,C1(CC(=O)N(CCCCN(C(c2cc(C)sc2)=O)C)C)CCOC(C(C)C)C1 43719,c1(CNC(c2c(CCC(=O)O)occ2)=O)cccc(F)n1 43720,C(=O)(C(O)CC(C)C)N1CC(NC(C(=C(C)C2CC2)F)=O)C(C)C1 43721,CCCC(CC)C(=O)N1CCN(C(=O)CCCOc2ccc(F)c(F)c2)C(C)C1 43722,C(N=c1[nH]c2c(c(=NC3CCc4cccc(Cl)c43)[nH]1)SCC2)C1CNC(=O)O1 43723,C(CC(CC)C(=O)N1CC(NC(=O)C=Cc2cncc(F)c2)C2(CC2)C1)=CC 43724,Cc1ncc(C(N2CC(C)(NC(=O)CCC3CC(C)C3)C2)=O)cc1C#N 43725,c1(CN2CCN(C(=O)CC3CCC(C(F)(F)F)O3)CC2)ccc2c(c1)COCC2 43726,c1(CC)csc(C(F)(F)C(=O)NCCCN(C(c2cc(CO)on2)=O)CC)n1 43727,c1(CNCC(c2ccccc2)F)cc(Cl)cc(Br)c1 43728,c1(C(=O)OC)ccc(NC(C2(NC(C)=O)CCCC2)=O)nc1C(F)(F)F 43729,C1(NC(c2cc(OC)ncc2)=O)CCN(c2ccnc(C(F)(F)F)n2)CC1C 43730,C(C(C)C)(C(O)C(=O)N(C)CC1CN(C(=O)COC(C)C)CCO1)OC 43731,C1(C(N(CCCCCNC(CC(C)C)=O)C(C)C)=O)CC(C)(C)CO1 43732,C(C(C(C)(C)C)SCC(=O)Nc1ccc(Cl)[nH]1)OC(Cn1cc(C(C)=O)nn1)=O 43733,N1(C(CCC(=O)NC)=O)CCC2(CC1)CC2(C)C(=O)NC(C)C(C)(C)C 43734,Cc1cc(C(=O)NCC2CC(NC(=O)CC3CCC(C)CC3)C2)cc(N)c1 43735,C1(NC(=O)CCCCC2CC2)CC12CCN(C(=O)C=Cc1cncs1)C2 43736,C1(CC)CCN(C(c2c[nH]ccc2=O)=O)C(C(N2CC=CC2CF)=O)C1 43737,N1(C(c2cccc(C)c2C)=O)CC(C2CN(C(=O)CC3CCC4CC34)C2)C1 43738,c1(CC)c(C(=O)Nc2cccc(-n3cc(CCC(C)O)nn3)c2)cnn1C 43739,CC1CCN(C(c2ccc(Cl)c(N)c2)=O)CC1NC(c1c(Cl)nsc1Cl)=O 43740,C1(C(N(C2CN(C(C3CCCCCC3)=O)C2)C)=O)CN(S(N)(=O)=O)C1 43741,C1(N(C)C(C2COCCC2NC(C2(F)CCCC2)=O)=O)CCCCC1(C)C 43742,c1(N)ccccc1.C12CN(C1)C(=O)CO2.CC(C)C=CC(=O)N(C)CCNC 43743,N1(C(C=C(CCC)C)=O)CC(C)CCC1COC.C1C(C)(C)C(=O)N1 43744,C1(NC(=O)NCC2CCC(=O)O2)CCC(NC(=O)NCc2ccccc2)CC1 43745,c1(CNC(C2C=CCC2)=O)cccc(C(N2CC(c3cccnc3)C2)=O)n1 43746,N1(C(CNC(C(C)(C)C)=O)=O)CCCN(C(=O)CCc2ncco2)CC1CO 43747,C1(C)(C(N2C(CN(C)C(C3CCCN3C)=O)CCC2)=O)CCOCC1 43748,C1(CNC(CCC(=C)C)=O)CC2COCC2N1C(C1CC2CCCC12)=O 43749,c1(C(=O)NCC(CNC(c2c[nH]c(=NC)o2)=O)F)ccc2nccnc2c1 43750,c1(CC(=O)NC(CNC(C2N(CC)CCCC2)=O)(C)C)ccc(OC)c(Cl)c1 43751,C1(CC)CN(C(c2cc(C)ns2)=O)CC1C(=O)NCC1CSCCO1 43752,c1(C(=O)NC(CNC(C2(COC)C=CCC2)=O)C)nccnc1-n1ccnc1 43753,C#Cc1ccc(CCC(=O)NCC(C)NC(=O)CN2CCOCC2)cc1 43754,N1(C(CC)=O)CC(C(=O)NC(CCC)C(=O)NC)C2(CCC2)C1 43755,c1(C(C)C(=O)NC2CC(n3cc(CO)nn3)C2)ccc(N(C)C)cc1 43756,C1(C2CCCN(C(c3occc3Br)=O)C2)(NC(C(C=C)O)=O)CC1 43757,C1(C(=O)NC2(CC(N)=O)CCC2)CCCN1C(=O)CC1CCC1 43758,N1(C(C(CCC)OCc2ccccn2)=O)CC2(NC(=O)CC(F)(F)F)CCC1C2 43759,Cc1ccnc(C)c1NC(C1CC2CC2N1Cc1cc(Br)cnc1F)=O 43760,c1(C(C(=O)NCCC2N(C(C(F)=C(C)C)=O)CCSC2)C)c(C)nn(C)c1C 43761,O=C1CCC(C(N2CCC(CNC(=O)C(O)CCc3ccccc3)C2)=O)CCO1 43762,c12cc[nH]c1NC2=O.C(CN(C)C)(C(=O)NCC1(CC2CCC2)CC1)OC 43763,c1(CNC2CCC(NC(=O)CC3CCCCO3)C2)cc(F)cc([N+](=O)[O-])c1 43764,C#Cc1cncc(C(=O)NC2CCC2NC(=O)Cc2ccc(F)c(Cl)c2)c1 43765,c1(N2CC(C)CC(OCC)C2)ccc(S(=O)(=O)N2CCSC(C)(C)C2)cn1 43766,n1(CC(=O)NCC(C)(C)CNC(=O)C(C)(C)CF)ccc2cc(F)ccc12 43767,C(c1ccncc1C)=CC(=O)NCCC(C)NC(C(c1ccccc1)OCC)=O 43768,c1(C(=O)NC2C(CNC(C(n3cc(C)nc3)(C)C)=O)CC2)cc2nc[nH]c2cn1 43769,Cc1ccc(C(=O)NCC2CC(F)(CNC(C3(C(C)(C)C)CCCC3)=O)C2)nc1 43770,c1(NC(C2CN(C(CNC(=O)OCC)=O)CC2F)=O)cc(Cl)cnc1C 43771,N1(C(CC2C(C)(C)CC2)=O)CC2(CCOCC2)CC1CNC(c1csc(S)n1)=O 43772,c1(C(N(CC(CNC(C2=C(C)OCC2)=O)(C)C)C)=O)cc(=O)c2ccccc2o1 43773,C1(C(=O)NC2CC(C(N(CC#C)CC3CCCO3)=O)C2)CC1C1(C)COC1 43774,c1(CC)cnccc1C(N1CCCC1C(=O)OC)C(=O)NC(C)CC 43775,C(=O)(CCCCC(F)F)NC1(C)CCCN(C(c2cccc(CS(C)=O)c2)=O)C1 43776,c1(CC(=O)N(CC(O)CN(C)C(C2CC2C(C)(F)F)=O)C)ccnn1C 43777,C(=O)(CCN=c1[nH]ccs1)NCC(CN(C(C1COCCC1(F)F)=O)CC)(C)C 43778,c1(C(=O)NCC(CNC(=O)CC2CCCC2O)CO)nccc2ccncc12 43779,N1(C(CNC(CC)=O)=O)CCN2CCN(C(=O)CC3CCCC(=O)N3)CC2C1 43780,C=CCC(C)(C(=O)NC1CC(NC(=O)CCc2cc(C)n(C)n2)C1)N(C)C 43781,C(=O)(C(CC(C)C)NC(c1ccsc1C)=O)N1CCC(CC(=O)OC)C1 43782,C(CC(C)(C)C(=O)NCC1COCCN1C(=O)C=CC(=O)NC1CC1)OC 43783,C1(NC(C(CC=CCC)C)=O)CC2CCC(C1F)N2C(=O)C(C)(C)Br 43784,C(=O)(C(C)S(C)(=O)=O)N1CCC(N(CC#C)C(c2cccs2)=O)C1 43785,C1(CCNC(C(C)n2cnnn2)=O)CCCN(C(c2cnoc2)=O)CC1 43786,c1(C(=O)NC2C(NC(CCOC(C)C)=O)CC2)cnc(Cl)c(N)c1 43787,C1(NC(CCCCC=CC)=O)CN(C(C2NC(=O)OC2(C)C)=O)CC2(CC2)C1 43788,C1(C(=O)NCCNC(CC2C(C)(C)C2)=O)CC=CC(O)C1 43789,N1(C(CC(=O)OCC)=O)CC2C(N(C)C(c3[nH]nnc3COC)=O)C2C1 43790,C(CCC(O)C(=O)NCCCCn1ccnc1)NC(=O)CN1CC2CC2C1 43791,c1(C(=O)NC(CC)CNC(c2cnc(C)s2)=O)cc2ccc(F)cc2nc1O 43792,c1(CC)nc(CC(=O)NCC2CCCN2C(C2CC(F)C2)=O)cs1 43793,C1(CC)CCN(C(=O)C(C)=CC(C)(C)C)C1C(N1CC(OC(=O)N(C)C)C1)=O 43794,c1(-n2c(C(=O)NCC(C)NC(C3(COC)CCOC3)=O)cnn2)ccccc1F 43795,c1(OC)ccc(CNC2CCC(C(=O)O)C2)c(O)c1 43796,CON(Cc1ccco1)C(=O)C(F)(CNC(=O)CC1CC(SC)C1)C(C)C 43797,N1(C(c2c(COC)cccn2)=O)CC(CC(=O)NCC(C)OC)CC1(C)C 43798,Cc1cc2occ(C(=O)NC34CC(NC(c5cc(C)n(C)c5)=O)(C3)C4)c2cc1C 43799,O=C(C(F)C(F)(F)C(F)(F)F)NCC1(O)CN(C(c2cc(F)c(Cl)cc2F)=O)C1 43800,C1(NC(c2ccc(CNC(C3OCC(C)C3)=O)cc2)=O)CCC(=O)NC1C 43801,c1(N(c2ccc(C(=O)OC)s2)C(C2CCN2C(=O)C2CC2)=O)c(C)cccc1C 43802,N1(C(c2ccn(CC)n2)=O)CC2CCCN(C(C3CC(OC)C(OC)C3)=O)C2C1 43803,C#CCCCC(C)C(=O)NC(c1nccs1)CC 43804,C1(NC(c2n(CCC)nc(C)c2)=O)CC2CN(C(=O)CCC(C)(C)F)CC2C1 43805,S(=O)(=O)(c1cc(C)c(Br)cc1F)NC(C(CCC)OCC)=O 43806,C1(NC(C2CCN(C(CC(C)(F)F)=O)CC2)=O)CCCCCC1O 43807,N1(CC(=O)NC(CC)C(C2CC2)C2CC2)CCC(N2CCC(C)(O)C2)CC1 43808,c1(C(=O)NC23CC(CNC(C(C)SC)=O)(OCC2)C3)ccn2cnnc2c1 43809,N(C(=NCCC(=O)N(C)C)NCC1CC2C=CC1CC2)C1CC(C#C)C1 43810,C(=O)(CCCCC(C)(C)OC)NCC(C(C)C)NC(c1c(OC)c(Cl)ccc1)=O 43811,C(c1cc(F)cc(F)c1)=CC(=O)NCC(CN(C(CCCOC)=O)C)C 43812,N1(C(c2ccn(CCC)n2)=O)CCC2(CCN(C(c3cc(N)ccc3C)=O)C2)C1 43813,c1(-n2cc(CCN(C)CCN3CCNCC3)nn2)c(C(F)(F)F)nc2ncccn12 43814,c1(NC2(CNC(CSc3c(C)cccc3)=O)CCCC2)c(Cl)cccc1[N+](=O)[O-] 43815,N1(C(CCC2CC(NC(c3c(C)n(C)nn3)=O)C2)=O)CCC(N(C)C)C(C)C1 43816,C(=O)(C(F)(F)CN)NCC(Cc1ccccc1)OCC 43817,c1(C(N2CC(NC(C(CC)C(C)C)=O)C2)=O)ccc2c(O)nc(=O)n(C)c2n1 43818,c1(C(N(CCCCN(C(C=CC(CC)=CC)=O)C)C)=O)ccc(F)cc1C 43819,c1(CNc2cccc(P(C)(C)=O)n2)ccc2cc(Cl)ccc2c1 43820,C1(NC(C)=O)CCN(C(=O)NC2COCC2O)CC1 43821,N1(C(c2c(CC)cnn2C)C(=O)NCc2ccccc2)CC(COC)C2(CC2)C1 43822,N1(C(C(CNC(C(C(C)C)OC)=O)(C)C)=O)CC(=O)N2CCCC2C1 43823,C(=O)(CC(CNC(=O)CC1(C)OCCO1)C1CCC1)N(CC(C)C)C 43824,C=CCC(CNC(=O)C(C)c1ccco1)C(=O)NCC1(C(C)C)CC1 43825,Cc1ccc(O)cc1C(N1CCN(C(=O)Cc2ccon2)C(C)C1)=O 43826,CC1(C)CCN2CC1CCNC(=O)C2=O.C(CC(N)=O)NC(=O)COCC1CC1 43827,C=CCCCCC(=O)N1CCC(CF)(NC(c2cnccc2Cl)=O)C1 43828,C1(CNC(C(N2C(CC)CCC2)=O)=O)CSCCN1C(=O)CSCCN(C)C 43829,c1(C(N2CC(CNC(CC=CCC)=O)C(F)(F)C2)=O)cccc2nc(Cl)cn12 43830,S1(=O)(=O)c2ccc(cc2)C(=O)NCCN1.c1(NCC)ccc(C(F)(F)Br)nc1 43831,N1(C(c2cnc(CC)o2)=O)C(CC(=O)NC2C=CCCC2)C2CCCC12 43832,c1(CC(N2CCN(C(CN(C(C)C)C)=O)CC2)=O)cccc([N+](=O)[O-])c1 43833,c1(C(=O)NCC2CC(F)(CNC(CS(=O)(=O)NC)=O)C2)ccc2c(c1)ncn2C 43834,c1(C(CNC(=O)NCc2c(C)nc(CC)o2)N)cccc(Br)c1F 43835,c1(OC)nc(C(=O)NCC(N2CCN(C(c3cc[nH]c3C)=O)CC2)C)ncc1F 43836,C1(O)(C(CNC(CC=C=C)=O)C)CCN(C(=O)CC2(C)CCOCC2)C1 43837,C1(O)(C(=O)NCCN(C(=O)C(c2cccc(C(F)(F)F)c2)(C)C)CC)CC(F)(F)C1 43838,N1(C(c2c(NC)cc(Cl)cc2)=O)CC(CNC(=O)C(C)C(C)C)OC2CCCC12 43839,N#Cc1ccc(F)c(C(N2CCC3CCC23CNC(=O)C=Cc2cocn2)=O)c1 43840,CC1CCN(CCn2ccc(C(F)(F)F)n2)CC1 43841,c1(C(=O)NC2(CNC(=O)CC3(C(F)F)CC3)CCOC2)cc(O)cc(Cl)c1 43842,c1(CC(=O)NC2CC(C)(NC(c3ccsc3Br)=O)C2)nc2ncccn2n1 43843,C1(CN(C)C)CCCC1C(N1CC(NC(=O)C=Cc2cncs2)C1)=O 43844,CC1CN(C(c2cncn(C)c2=O)=O)CCC1NC(c1cc(C2CCC2)[nH]n1)=O 43845,c1(OC)nccc(C)c1NC(=O)CCC(C)NC(C1CCCC(OC)C1)=O 43846,c1(C(=O)NC2C(F)CCN(C(C3(C)CCOCC3)=O)C2)cccc2ccsc12 43847,C(CC(C)C(=O)N(C(C)CNC(C1(C)SCCCS1)=O)C)=CC 43848,C1(NC(C2CC(CCC)C2)=O)CCC2(CC1)CCN(C(c1cccnc1O)=O)C2 43849,c1(C(N2CC(CNC(COCC)=O)(CO)C2)=O)ccc(C)cc1C 43850,C(=O)(CC(C)C(F)F)N1CCCC(N(C(c2nc(SC)sc2)=O)CCF)C1 43851,c1(CC(C)C)cc(C(=O)NC2CN(C(c3ccc(C4CC4)o3)=O)C3CC23)n(C)n1 43852,c1(C(N2C(C)(C(=O)NCc3ccc(O)c(O)c3)CCC2)=O)ccc2nn[nH]c2c1 43853,Cc1cccc2[nH]cc(C(=O)NCCC3(O)CN(C(=O)CCC4CC4(Cl)Cl)C3)c12 43854,N12CC3CC3(C1)C2=O.C(c1ccoc1)=CC(=O)NCCC(=O)NC(C)(C)C 43855,c1(NC(CC)C(C)(C)COC)nc(NC(=O)OC(C)(C)C)nc2ccccc12 43856,c1(CNC2CCN(C(c3c(C)n[nH]c3)=O)CC2F)c(F)cc(Br)cc1F 43857,C(CCO)(C(=O)O)NC(=O)Nc1ccc(Cn2ccnn2)cc1 43858,n1(CC)cnc2c(NC3CCCN(C(=O)Cn4ncc(Cl)c4C)C3)ncnc12 43859,C#CCCCC(C)C(=O)N1CC(C(N)=O)(CNC(c2ccc(Cl)c(F)c2)=O)C1 43860,Cc1cc(C(N2CCC(CCNC(C3CCN(C)C3)=O)C2)=O)cnc1C(F)(F)F 43861,C12(CC(=O)NC3CCCC(NC(C4CCC45CCC5)=O)C3)COC(CF)(C1)C2 43862,Cc1cc(Cl)c(C(=O)NCC2C=CCN2C(=O)CNS(C)(=O)=O)s1 43863,CC(N=c1ccnc(C2CCC2)[nH]1)c1ccccc1C(=O)OCCc1cccs1 43864,CC1=NOC(C)(C(=O)NC2CC(C)(NC(=O)CCc3ccccc3Br)C2)C1 43865,c1(C(C(=O)N(C2CCN(C(=O)C=COCC)CC2)CCC)(F)F)cc(C)ccn1 43866,c1(CCN(C(=O)CCCN(C)C(C2C=CCCC2)=O)C)nccc(O)n1 43867,c1(C(N2CCC(COC)(NC(C3CC=CCC3)=O)C2)=O)ccc(OC)c(Cl)n1 43868,c1(CC(=O)NCC(CO)NC(C(COCC)O)=O)ccccc1SC 43869,N1(C(c2ncc(C)cc2F)=O)CC2CCC(N(C)C(c3occc3C)=O)C2C1 43870,C1(CNC(C2(OC)CCOC2)=O)CC(C)(C)CN1C(c1scnc1Cl)=O 43871,C(=O)(CCS(C)=O)NC(c1ccccc1)CNC(C1C(OC(C)=O)C1)=O 43872,C1(NC(C2C(CNC(C(COCC)C)=O)CCO2)=O)CNC(=O)C1(C)C 43873,C(CCCCC(=O)N(C)CCOCCNC(C1CCC(C2CC2)C1)=O)SC 43874,c1(OC)ccc(C)c(C(N2CC(OCCNC(=O)CN3CC(C)C3)C2)=O)n1 43875,C(=O)(CC(C(F)F)c1ccccc1)N(CCCNC(c1cc(F)n[nH]1)=O)C 43876,CC1(C)C(CNC(=O)NCC2(c3nn[nH]n3)CC2)CC1O 43877,Cc1cc(C(=O)NC(CO)C(=O)NCC2CCC(C(N)=O)CC2)c(O)nn1 43878,N1(C(C(C(C)C)OCC)=O)CC2CCC1C(NC(=O)Cc1n[nH]c(C)n1)C2 43879,N1(C(c2c(C(C)C)onc2)=O)CCC2(CC(C(=O)NCCN(C)C)C2)C1 43880,C1(NC(C(C2CCCN2C(=O)CNC(c2cc(F)c[nH]2)=O)C)=O)CCCCCC1 43881,C1(NC(Cn2nnc(=N)[nH]2)=O)CCCCCN(C(C23CCN(CC2)CC3)=O)C1 43882,c1(OC)c(C(=O)NC2CC(NC(=O)C(C(C)C)NCC(C)C)C2)cc(Cl)cc1C 43883,N1(C(c2ccc(Br)c(Cl)c2)C(=O)NCCC#N)C2CCC1CC(F)C2 43884,c1(NC(C2CCCCN2C(c2cc(Cl)c(Cl)cc2F)=O)=O)cc(F)c(O)cc1Cl 43885,CC1CN(C(=O)COC2CCN(C(=O)C=CC3CCC3)C2)CC(C)(C)O1 43886,C12(NC(c3c(OC)cc(CO)cc3)=O)CCCC1CN(C(=O)CN1CC=CC1)C2 43887,c1(C(=O)NC2C(C)CN(C(C3CC(OC4CC4)C3)=O)C2)ccnc2c1cnn2C 43888,N1(C(C2(C)N(C(C(CC)N(CC)CC)=O)CCC2)=O)CC2CC(N(C)C)C2C1 43889,N1(C(=O)Cc2cc(F)cc(Cl)c2)CCC2OCCN(C(=O)C=CCF)C2C1 43890,C1(C(=O)NCC2OCC(CNC(c3sc(C)c(O)n3)=O)C2)CC2(CCCCC2)C1 43891,C1(C(=O)NCC2CCCCO2)CCN(C(c2cc(Cl)cnc2O)=O)CC1O 43892,c1(C(N(CC(CNC(C2C(CCOC)C2)=O)(C)C)C)=O)cc(C(C)C)nn1C 43893,C1(C(=O)NC2CCCC(CNC(c3c(CC)c[nH]c3)=O)C2)OCCOC1(C)C 43894,CS(=N)(=O)CCNC(=O)C(Cc1cc[nH]n1)NC(=O)CC1COC(=O)C1 43895,N1(C(C(C=C)O)=O)C2CCC1CN(C(c1sc(Cl)cc1Cl)=O)C2 43896,CC1CN(C(C2CCCN2C2CC2)=O)CC(C)N1C(=O)C(F)(F)C(F)(F)F 43897,C(=O)(C(CCC)OCC)N1CCC(C(N2CC(CCC)C2)=O)C1 43898,C#CCC(C(=O)NCCCOCC1CC1)NC(C1CC=CCC1)=O 43899,C1(CC(=O)NC2C(NC(CSCC=C)=O)C2)OCCCC1(C)C 43900,C(=O)(C(O)C(F)(F)F)NC1CC2(C(C(N(C)CC3(COC)CCC3)=O)C2)C1 43901,N1(C(CC)=O)CC2CC1CN2Cc1ccccc1OCc1ccccc1 43902,C1(C(=O)NCC#CCNC(c2cc(C)n(C)c2)=O)CC(c2cccc(F)c2)=NO1 43903,c1(C(N2CCC(CN(C)C(C3CC3CF)=O)C2)=O)cccc2nccn12 43904,c1(CC)ccc(C(=O)NCCC(O)CNC(c2cnc(O)cc2OC)=O)c(Cl)c1 43905,c1(C(=O)NC(c2ccccc2)CCC)ccc(N2CCC(N)CC2)cc1 43906,O(NC(=O)C(C)(C)S(C)(=O)=O)C(CC(C)C)C(=O)N1CCC(C(C)(C)C)C1 43907,n1(C(=O)NCCN(C(c2cc(C(C)=O)[nH]n2)=O)CC)cnnc1O 43908,c1(OC)ccc(NC(=O)NC2CC2c2ccncc2)cc1Br 43909,N1(c2nnc(CC)c(CC)n2)CCC(NC(c2n[nH]c(C)c2O)=O)C12CCCC2 43910,C1(C(N(CC#C)C)=O)CC12CCN(C(=O)CN1CC(C)(C)C1)C2 43911,C(c1cccnc1)=C(C)C(=O)NC1C=CCCC1C(=O)NCCC12CC(C1)C2 43912,C1(NC(c2ccc[nH]2)=O)CN(C(C23CCC(CC2(F)F)C3)=O)Cc2nccn2C1 43913,CCCCCC(F)C(=O)N(CC(N1CC(O)CC1COC)=O)CC1CC1 43914,N1(C(C(C)C)=O)CC(n2cc(C(C)N(C(=O)OC(C)(C)C)C3CC3)nn2)CO1 43915,c1(C(=O)NCCN(C(C2CCc3c2cnn3C)=O)CC)ccc2[nH]nc(O)c2c1 43916,C1(F)(CNC(C2C(CC(C)(C)C)C2)=O)CCN(C(=O)CS(N)(=O)=O)C1 43917,CC(C)(C(=O)NCC(C1CC1)NC(=O)CC1(C(F)(F)F)CC1)c1ccns1 43918,Cc1nn(CC(N2CCC(CNC(c3ccoc3Br)=O)CC2)=O)cc1Cl 43919,N1(C(C=CC)=O)CCC2(CC1)CN(C(=O)C(C)n1cccn1)CC2CO 43920,c1(C(N2CCC(CCNC(C3C(=C)C3)=O)CC2C)=O)ccc2nnc(O)n2c1 43921,C1(CNC(C2(C)CC(C)C2)=O)CN(C(c2ncc(F)cc2N)=O)CC(C)(C)C1 43922,C(=O)(C#CC1CC1)NC(CC)C(=O)N(C1CC(O)C1)C 43923,C(=O)(C(S(C)(=O)=O)C1CC1)NCCC(C)NC(C1(C)CCSCC1)=O 43924,CC1COC2=CNC(=NCC3CN(Cc4ccccc4)CCC3(F)F)NC2=N1 43925,N1(C(=O)C=Cc2ccsc2)CCC2(C1)CN(C(=O)C(F)F)CCO2 43926,C(=O)(C(CC(C)C)NC(=O)OC)NCC(C1(OC)CCOCC1)(F)F 43927,C1(C(N2CC(CC(=O)NCCc3cc(C)n(C)n3)OCC2)=O)CN2CCN1CC2 43928,c1(CCC(=O)NC2CCN(C(CCC(=C)C)=O)C2C)ccc(Br)cc1OC 43929,CCCC(C(=O)NC(C)(C)CNC(c1cccc(COC)c1)=O)S(N)(=O)=O 43930,c1(CC)nnc2cc(NC3(C4CCCN4C(=O)C(C)C(C)S(C)(=O)=O)CC3)ncn12 43931,C1(O)(CCNC(CC2CC(=C)C2)=O)CCN(C(c2cnc(C3CCCO3)s2)=O)C1 43932,c1(C(C(=O)OCC2CCC(F)(F)C2)OC)cccc(CC(F)(F)F)c1 43933,C(=O)(C1=CCCCCC1)NC(C)CCNC(=O)C(n1cc(Br)cn1)C 43934,c1(CNCC(O)CC(F)(F)F)c(O)ccc(F)c1F 43935,CCC(=O)CCC(=O)N1CCOCC(CNC(c2sccc2OCC)=O)C1 43936,Cn1cncc(C(=O)NCC2(NC(=O)C(O)CN3CCCC3)CCOCC2)c1=O 43937,C1(C(N2CCC(n3cc(C(CC(C)C)O)nn3)C2)=O)CCN(C)C(=O)C1 43938,N1(c2cc(NCC(CC)N(C)C)ncn2)CCc2c(F)cc(F)cc2C1 43939,C1(C)(NC(CCCNC(C)=O)=O)CCC(NC(C2(O)CCSCC2)=O)CC1 43940,C(=O)(C1CC(=O)c2ccccc21)N1CCC(NC(=O)Cn2cnnn2)(CF)C1 43941,CN1CCC(NC(C2N(C(=O)Cc3cncn3C)CCC2(C)C)=O)C(C#N)C1 43942,CCC(C)C(C(=O)NC1CCN(C)CC1C)N(C(=O)CCC1CCC1)C 43943,Cc1ccc(C)c2[nH]c(C(=O)NCC3CCC3NC(C3CCS(=O)CC3)=O)cc12 43944,c1(C(=O)NCCCCNC(=O)CCc2cncnc2)c(Cl)ccc2c1OCO2 43945,C12CCCN(C1)C2=O.C=CCC(CNC(C1(C(=O)N(C)C)CC1)=O)NC(N)=O.OCC 43946,c1(C(=O)NC2(CC=C)CN(C(=O)C=CCC)C2)cc2c(s1)COCC2 43947,C1(C)(NC(CN(CCOC)C)=O)CC(NC(c2coc(Cl)c2)=O)C1 43948,c1(C(N2CC(N(C)C(C3(c4cccs4)CCC3)=O)C2)=O)cnn(C)c1N 43949,C(CCCCCN(C)C(c1cc(Cl)no1)=O)NC(C(c1cccc(Cl)c1)C)=O 43950,c1(OC)ccc(CN(C)CC2CCCN(C(C3CC(C)(C)C3)=O)C2)cc1C 43951,C1(C)(CC)CC(C(=O)NC(c2cccnc2)c2nc(C)cs2)CCO1 43952,CCCCCC(F)C(=O)NC(c1cn(C)nn1)C(=O)NCCC1CCCCCC1 43953,c1(C(=O)NCc2cccc(CNC(C=CSC)=O)c2)ccc(C(C)(F)F)nc1O 43954,C1(C(=O)NCCN(C(=O)Cn2nnc(-c3ccsc3)n2)CC)CCC(C)(C)CO1 43955,c1(C(=O)NC2C(CC)CN(C(c3cccnn3)=O)CC2)cccc2nccn12 43956,c1(C(=O)NCC2(C(N3CC(n4ccnc4)C3)=O)CCC2)ccnnc1 43957,c1(CCC(N2CC(NC(C=CCOC)=O)C(C)C2)=O)cc2ccc(O)cc2oc1=O 43958,C(=O)(C(F)(F)C(O)C(C)C)NCCC1=CCN(C(c2c(Cl)cn(CC)n2)=O)CC1 43959,c1(C(=O)OCC)cnc(N2CCS(=O)C(C)C2)cc1C 43960,C1(NC(CC=CCC)=O)CC(NC(=O)Cc2ccccc2F)CC1O 43961,N1(C(CNC(CCC(C)C)=O)=O)CCC2(NC(=O)CC(=O)N(C)C)CC2C1 43962,C1(OC)CC(CNC(c2cc(C(C)(C)C)nn2C)=O)N(C(c2nn[nH]c2Cl)=O)C1 43963,C1(c2c(C(=O)OC)cccc2)CC2CN1N1CC=CC2(CCS(=O)(=O)CC)C1 43964,N1(c2nnc(C)o2)CCC(C(C)NC(C2C3COCC23)=O)CC1 43965,c1(NC(=O)NOc2ccc(Cl)cc2)cnc(Br)cn1 43966,CC(C(=O)NC1CC2CC(NC(=O)C=Cc3cncs3)C2C1)S(N)(=O)=O 43967,c1(C(N2C3CC(NC(C(=O)N(C)C)=O)C(C3)C2)=O)n[nH]c2ccc(Cl)cc12 43968,Cc1cnc2cccc(C(N3CCC(N(C(=O)CC4C=CCCC4)C)C3)=O)c2c1 43969,C1(CN(C(C2C(C)CCC2)=O)C)COCCN1C(C1CC(=O)N(C)C1)=O 43970,C(=O)(C(C)(CO)CO)N1CCCC(C(=O)Nc2c(C(C)=O)cccn2)C1 43971,c1(C(=O)NC(C)CCNC(=O)CC(C)N(C)C)ccc2nccnc2n1 43972,C(CCC(N)=O)(C(=O)N1CC(CCNC(=O)CC2CCCC(C)(C)O2)C1)N(C)C 43973,Cc1ccc(C2(C(=O)NCCNC(C3(C)COC3)=O)CC2)c2ccccc12 43974,C1(NCC2CC(OCC)C2)CCS(=O)(=O)C(C)(C)C1 43975,N1(C(COCC(=C)C)=O)CC(NC(C2CC(n3ccnn3)C2)=O)CCC1C 43976,N1(c2nnc(CCC)s2)CCC(O)(C(C)NC(=O)CN2C(=O)CN(C)C2=O)CC1 43977,c1(C(N2CCC(CNC(C=CC=CC)=O)C(F)(F)C2)=O)cc2c(cn1)CCCC2 43978,O=S(=O)(c1cnccc1N1CCCC(c2nncs2)C1)NCC1(CO)CCCC1 43979,C1(F)(CNC(C(CSC)OC)=O)CCN(C(=O)CC2CC(=O)C2)C1 43980,C1(C(N2CCC(CO)CC2)=O)COCCN1C(C1CC1F)=O 43981,c1(C(=O)NCCN2CCN(C(c3scc(C)n3)C)CC2)cc(C)cc(C)c1N 43982,CC(CC(F)(F)F)C(=O)N1CCN(C(=O)CCCN2CCCC2)C(C)C1 43983,c1(C(=O)NCC(C)(C)NC(=O)Cc2ccoc2)ccc(-c2ccccc2)s1 43984,N1(C(c2c(CC)non2)=O)CCCC(NC(C2CCNC2=O)=O)C1C 43985,c1(C(=O)NC2CC(C)N(C(c3cc4cccnn4c3)=O)C2)ccc2nonc2c1 43986,c1(C(=O)NCC2(CN)CC(F)(F)C2)ccc(NN2CCNCC2)cc1Cl 43987,CC1(C)C(CC(=O)NC2CCC(NC(=O)Cc3cocn3)CC2)CC1O 43988,Cn1cc(S(=O)(=O)CCNC(=O)Cc2ccn(C)c2)cn1 43989,C(C(C)(C)C#CC(=O)NC1CCS(=O)CC1)NC(CN1C(C)CCCC1)=O 43990,C=C(C)C1OCCC1C(N1CC(C(C)NC(=O)Cc2cnc(C)s2)C1)=O 43991,C1(C#CC(=O)N2CCC(CCNC(=O)CCCC(=O)NC(C)C)C2)(CC)CC1 43992,C1(C(=O)NCC(S(C)(=O)=O)CNC(C2CCCCC2O)=O)OCC2COCCC12 43993,C=CCCCC(C)(C)CN=c1[nH]c(C)cc(=NCC2(C)CSCCO2)[nH]1 43994,C(=O)(C(F)C(=O)NCCCOCCNC(C1CCC(N(C)C)CC1)=O)OCC 43995,N(C(=NCCOCC)N1CCC2(CCCCCC2)C1)C(C#C)CC 43996,C1(NC(C2C(C(C)NC(=O)CCc3ccc[nH]3)C2)=O)CCCC(O)CC1 43997,c1(C(=O)NC2CN(C(C(OCC)OCC)=O)C(C)(CC)C2)n[nH]c(C)c1[N+](=O)[O-] 43998,c1(C(N(CC(=O)NC2CC2C(C)(C)C)C(C)C)=O)cnns1 43999,C(C(F)(C(=O)NCc1ccnc(F)c1F)C(C)C)NC(c1c(C(C)C)c[nH]c1)=O 44000,C1(O)(C(C)CNC(c2c(Br)ncn2C)=O)CCN(C(=O)OC(C)(C)C)C1 44001,Cc1cc(C(=O)NCC(C(C)(C)C)NC(c2cccc[n+]2[O-])=O)ccn1 44002,C(=O)(C1CCCc2c1ncn2C)N1CC(NC(c2c(C(C)C)occ2)=O)C(O)C1 44003,C1(N(CC(=O)NC(CNC(=O)COC2CCCC2)C2CC2)C)C=CCCC1 44004,C1(C(N2CCCC(C(F)F)C2)C(=O)NC(C(=O)OC)C)CCCOCC1 44005,N1(C(C)=O)CC(C)CN(C(=O)CCNC(C2(CC=C)CCCC2)(C)C)C(C)C1 44006,c1(CN2C(C(=O)NC(C3CCCCC3)CC)C(O)CC2)ccccc1[N+](=O)[O-] 44007,Cn1c(=O)cc(C(=O)OCc2c(F)c(F)c(Br)c(F)c2F)c2ccccc12 44008,c1(C(=O)NC2(CF)CCN(C(CC3CC(=C)C3)=O)C2)cn2c(C)cccc2n1 44009,C1(CC(=O)NC2CC(CNC(CSC)=O)C2)CSc2ccccc2O1 44010,c1(C(=O)NC2(CNC(C(CC)(C)F)=O)CCCC2)ccc(Cl)cc1Cl 44011,c1(N2CC3CC(NC(C4=C(C)OCCS4)=O)C3C2)nc(Cl)nc(C(C)C)c1C#N 44012,N1(C(C(C)CC#N)=O)CC2CCC(CN=c3nc[nH]s3)(C2)C1 44013,C1(CC(=O)NCC2CCN(C(C3CC4(CSC4)C3)=O)C2)CC2CCC1C2 44014,Cc1cccc(C(=O)NCC2CCC2C(=O)NC(C)(C)CNC(N)=O)c1 44015,C1(CN(C)C)CCCC1C.CC1CN(C)C(=O)C=CC(=O)N1 44016,CCC(CCC(=O)NCC(C)(C)C(F)F)NC(C1(C(C)C)COC1)=O 44017,C1(CNC(C2(C)CC2(F)Cl)=O)C2CN(C(c3ccn(C4CC4(F)F)n3)=O)CC12 44018,C=Cc1ccc(C(N2CCCC(C)(CNC(c3c(Cl)noc3C)=O)C2)=O)cc1 44019,CC1(C)C2CC(C(=O)NCC3CC(F)(CNC(C4CCS(=O)(=O)N4)=O)C3)CC12 44020,CCC(C)C(=O)NCC(N1CCCC1C(=O)NCc1ccn(C2CCC2)n1)=O 44021,c1(C(=O)NC2(C)CCN(C(c3ccn(CC)c3C)=O)C2)cc(O)nc(C)n1 44022,CC(CNC(C1CC1Cl)=O)C(F)C(=O)NCCCN1CCOCC1 44023,c1(C(=O)NCC(CC)NC(=O)Cn2ncccc2=O)ccnc(S)c1 44024,C1(CCNC(CCC=C)=O)CN(C(=O)C(CCC)OCC)CCCO1 44025,c1(C(=O)NCC2CN(C(c3c(C)coc3)=O)C(C)(C)C2)cc(P(C)(C)=O)cs1 44026,C(C(N=c1cnc(CCO)c[nH]1)c1ccccc1)c1c(C)cccc1 44027,N12CCC(C3CC3)C1n1cc(nn1)CC(C)(C)C2=O.C1(SC)CC2C=CC1C2 44028,C1C(CC(C)C)C(=O)N1.C1(CNC(C2CCC2C(N)=O)=O)CCOC1.CC=CC 44029,CS(=O)C1(CNC(=O)NCC2CNC(=O)C2)CCC1 44030,c1(C2(C)CN(C(=O)NCCCc3nccc(C(F)(F)F)n3)C2)ccccc1Br 44031,C1(C(=O)NC(C(=O)NCc2ccc(C)o2)CC2CCC2)CCCC(=O)C1 44032,c1(C(N(C)CC2N(C(c3nnn(CC)c3C)=O)CCOC2)=O)ncc(F)cc1F 44033,C1(C(=O)NC2CC2NC(=O)C(F)(F)C2CCOCC2)(OC)CCSCC1 44034,c1(OC)c(F)ccc(C(=O)NCCN(C(C2CCCCC2)=O)C(C)C)c1F 44035,c1(CC(=O)NC2CCN(C(COCCC)=O)C2)ccccc1CS(N)(=O)=O 44036,Cc1cc(C(N2CCC(NC(C3CC34CCCC4)=O)C(CO)C2)=O)ncc1CO 44037,C1(COC)CN(C(c2nccc(Br)c2C)=O)CCN1C(C1CC2CC2C1)=O 44038,c1(C(N(CCCC(=O)NCCCc2cc(C)no2)C)=O)n[nH]c2c1COC2 44039,Cc1nc2ccccc2n1CC(=O)NC1CC(NC(C2CC(O)C2)=O)C12CCC2 44040,C1(CC#CC)NC(=O)N(C(c2nn(C)cc2O)C)C1=O 44041,C1(C(N2CCC(C#N)C2)=O)(CC)CCN(C(=O)COC(C)=O)C1 44042,c1(C(=O)NCc2ccc(C(=O)NC(C=C)(C)CC)s2)cncc(Cl)c1 44043,CC1C(NC(=O)CCCC(N)=O)CCCN1C(C1CC1c1ccoc1)=O 44044,C1(C(N2CCC(C)(F)C2)=O)(CC)CCCN1C(=O)CCn1cncn1 44045,N1(C(CC#N)=O)CCn2c(CNC(C3CCOC4(CCC4)C3)=O)nnc2C1 44046,c1(CSC)cc(C(=O)NCC2CC(NC(C3CCN(C(C)=O)C3)=O)C2)ccc1F 44047,N1(C(CCN(C(C(CC=C)CC)=O)C(C)C)=O)CC(C2CC2(F)F)C1 44048,C(CC1CCC1)(C(=O)N(CC(C)NC(=O)Cn1cnnc1O)C)NC(C)=O 44049,NS(=O)(=O)c1ccc(C(=O)NCC2CCCCC2NC(=O)CC2NC(=O)NC2=O)o1 44050,Fc1cc(CCC2CC2)ccc1C1CC1c1cccc(Br)c1 44051,C12(CNC(C(CNC(=O)C#CC(C)C)OC)=O)CCC(F)(CC1)C2 44052,C(=O)(C(C)P(C)(C)=O)NCC(CCOC)NC(c1ncccc1CSC)=O 44053,C1(NC(CCCOCCC)=O)CCCN(C(=O)CNC(=O)NC)C1CC 44054,Cn1nc(C(=O)NCCNC(=O)Cc2ccc(F)c(C(F)(F)F)c2)ccc1=O 44055,c1(C(N2CCC(NC(C(CCSC)(C)C)=O)C(C)C2)=O)cc([N+](=O)[O-])cc(C)n1 44056,C(CC1=CCN(C(c2cnn(C)n2)=O)CC1)NC(C(c1ccccc1)NC(C)=O)=O 44057,C1(NC(C=C(C)c2ccsc2)=O)CS(=O)(=O)CC1NC(=O)Cc1cncs1 44058,c1(C(=O)NCC2(F)CCC(NC(CC(CC)OC)=O)C2)c(C)nc(O)nc1C 44059,Cc1c(C(=O)NCCNC(C2OCCC2C(F)(F)F)=O)c(=O)oc2ccccc12 44060,Cc1cc(C(=O)N(CCCC(=O)NC2CC3CC4C(C3)C24)CC2CC2)c(C)nn1 44061,c1(C(=O)NC2CC3(C(NC(Cc4nnc(C)o4)=O)C3)C2)cc(F)cc(Cl)c1 44062,N1(C(C(C(C)C)SCC)=O)CC(CNC(c2cnc(O)c(C)c2)=O)C(C)(C)C1 44063,C12(CNC(=O)C=Cc3cccnc3)CCCC1N(C(=O)C=CC1CCCC1)CC2 44064,C1(NC(c2cc(C)on2)=O)CC1C1CCCN(C(=O)CN2CCN(C)CC2)C1 44065,N1(CC(c2ccc(CNC(C)C)cc2)=O)C(=O)c2cccnc2C1=O 44066,N1(C(C2CC(C)=C(C)CC2)=O)CC2(CCCC(CNC(=O)Cn3nccn3)O2)C1 44067,C1(CC(=O)NCCN(C(CC(=O)NCC)=O)C2CCCCC2)CCOC(CC)C1 44068,C1(C(C(=O)N(CCNC(=O)C(c2ccn(C)c2)C)C(C)C)OC)CCCCCC1 44069,c1(C(=O)NC(CNC(c2c(C)ccc(SC)c2)=O)C2CC2)ccc2c(c1)CCO2 44070,C1(CC)CCN(C(=O)CC=C(C)C)C1C(=O)NCc1nccs1 44071,N1(C(=O)NCC)CCCN(C(CC2CCCC2)C(=O)NC2CCC2)CC1 44072,C1(NC(C(C)=C(C)C)=O)CC(NC(c2cnn(C)c2N)=O)CC1O 44073,C1(CN(C(CSCC(C)=O)=O)C)CCCCN1C(=O)Cc1csc(S)n1 44074,C1(NC(c2cn(CCC)nn2)=O)CCN(C(=O)C(c2ccc(F)cc2)CC)CC1 44075,C(=O)(C1Cc2ccccc21)N(C1CCN(C(C2(C(F)F)CCCC2)=O)C1)C 44076,c1(C(C)NC(c2n(CCCOC)nnn2)c2cc(OC)ns2)cccc(OC)c1 44077,CC(C)(C)C(CNC(C1CCC=CO1)=O)NC(=O)CCN1CCOCC1 44078,C(=O)(CCC(=O)NC1CC(CNC(C2CSCN2C(C)=O)=O)C1)NCC 44079,C(=O)(C1=NN(C)C(=O)CC1)NCCC(C)N(C(c1cncc(C)n1)=O)C 44080,C(C(=O)N1OC2C=CC1CC2)(C1CCOC1)NC(C1C=CCS1)=O 44081,c1(OC)ccc(CC(=O)NCCOCCNC(c2cc(Cl)ccn2)=O)nc1 44082,NS(=O)(=O)CCCC(=O)NCC1(NC(c2cc(C3CCOCC3)no2)=O)CC1 44083,c1(C(CNCC23OCC(C(C)C)(C2)C3)O)ccc(S(C)(=O)=O)cc1 44084,c1(C(=O)NCC(C)(C)NC(c2c(CC)n(C)cc2)=O)oc2ccc(C)cc2c1C 44085,c1(C(N(C2CN(C(c3ccc(N)c(Br)n3)=O)C2)C)=O)n[nH]c2c1CC1CC21 44086,C(=O)(C(CCc1ccc(F)cc1)C(C)(C)C)NCC1C(NC(=O)C2CC2)C1 44087,c1(SC)ccc(C(=O)NCC(C(C)(C)C)NC(C2CCCCC2)=O)c(Cl)c1 44088,c1(C(N2CC(CNC(C(CCC)OCC)=O)N(C)CC2)=O)ccc2cc[nH]c2c1 44089,c1(C(N2CCOCC(CNC(C(C(=C)C)(C)C)=O)C2)=O)c([N+](=O)[O-])cnn1CC 44090,CC1=C(C)CC(C)(NC(=O)CC2(C)CCN(C(=O)CC3(O)CCOCC3)C2)CC1 44091,O=C(C1=CCCCC1)NCCCN(C(c1cccnc1)=O)C1CC1 44092,c1(C(=O)NC(C(=O)NCc2[nH]nc(COC)n2)C2CCOC2)cc(O)cc(F)c1 44093,C1(C)(C(=O)NCCCCNC(c2c(OC)cc(C)s2)=O)CCC(C(F)(F)F)CC1 44094,C=CC(C)CC(=O)NCC1CC(NC(c2ccsc2SC)=O)C1 44095,CC(C)C(CNC(c1cnn2c1OCC2)=O)C(=O)NCCCc1cnccn1 44096,n1(CC)nc(C)c(C(=O)N(CCCCNC(=O)COCc2cccnc2)C)c1Cl 44097,C1(NC(c2ccc(C(C)=O)o2)=O)CCN(C(=O)CCc2cncs2)CC1C(C)C 44098,c1(C(N2CCC(c3ncc(C(=O)O)s3)CC2)=O)cnn2c1CCC2 44099,C1(C(=O)NC(CCSC)C(=O)NC(C)(C)CCCN(C)C)CN(C)CC(C)O1 44100,N1(C(c2cc(C)sc2)=O)CCN(C2CCCN(C(=O)CCOC(C)C)C2)C(=O)C1 44101,C1(C(N(C(C(CC)C)C)C2CC2)=O)CCC2(CC2)N1C(C1CC(C)(O)C1)=O 44102,c1(OC)nn(C)cc1C(=O)NC1CCC(CN(C(=O)C(C)n2ccnc2)C)CC1 44103,C(=O)(C(C)C(C)NC(c1c[nH]cc1C)=O)NC1(COCC)CC1 44104,N1(C(C(CC=C)OC)=O)CCC2(CCC(NC(=O)Cc3ccccc3C)CC2)C1 44105,c1(NC(C2(C3N(C(C(CC)CC)=O)CCC3)CC2)=O)ccc(F)cc1SC 44106,c1(OC)cccc(C(c2nnnn2C2(C)CC2)NCc2cn(C)nc2C(C)C)c1 44107,c1(C(=O)NC(C)CCNC(=O)C(O)c2cnc[nH]2)ccc(Cl)o1 44108,c1(C(=O)NCC(C)NC(c2ccn(C(CC)CC)n2)=O)cc(C)nn1CC 44109,N1(C(C(CCC#C)O)=O)Cc2ccccc2C(NC(c2ccc(Br)o2)=O)C1 44110,c1(CN(CC(N2CCC(O)(CNC(CCC=CC)=O)C2)=O)C)cccc(C#N)c1 44111,c1(NC(c2n(CCCOC)nnn2)(COC)C2CC2)ccc2nncn2c1 44112,N1(C(CCOCCC)=O)CSCC1C(=O)N(CCCF)CC 44113,C(=O)(C1=C(Cl)CCOC1)NCCC(C(=O)Nc1c(OC)cc(F)cc1)(C)C 44114,C1(C(=O)NC2(CC=C)CN(C(=O)Cc3cc(COC)no3)C2)CC=C(C)CC1 44115,N1(C(C(CCC)(C)C)=O)CCC2(CCN(C(=O)CC3CCCCC3(F)F)C2)C1 44116,N1(C(C(CCC)N(C)C)=O)CCC(C(=O)N2CCC23CC(COC)C3)=C(F)C1 44117,C(=O)(CC(C)CC(C)(C)C)NC1(C(=O)NCCC#C)CCN(C)C1 44118,C1(C(=O)NCC(CN(C(c2c(C)cc(C)o2)=O)C)O)CCC(C2CC2)CC1 44119,Cc1nc(C(C)C)ccc1C(=O)NCC(O)CCNC(c1cc(F)cc(F)c1)=O 44120,CC1CCN(C(=O)C2=CCCCC2)CC1CNC(=O)C=Cc1ccoc1 44121,Cc1cc(N2CCn3cccc3C2)nc(=NCCCc2ccc(C)c(C)c2)[nH]1 44122,C#CCC(C)(C)C(=O)NCC(C)N(C)C(C1CC1C#N)=O 44123,N1(C(c2c(C)nns2)=O)CCCC(N(C)C(c2ccc(OCCOC)cc2)C)C1 44124,c1(C(=O)NCCN(C(C2CCN(C(CC)=O)C2)=O)C)nnn(C2CCOC2)c1C 44125,c1(-c2ccc(C(=O)NC3C(C)(C)C3)cc2)ccc2c(n1)CCC2=O 44126,c1(C(=O)NC2CN(C(C3CC3(Cl)Cl)=O)CC2C(F)F)oc2ccccc2c1CO 44127,n1(CC)c2ccccc2c2cc(CN3CC(C)C3(C)C)ccc12 44128,Cn1ncc2nc(Cl)nc(N3CC(NC(=O)CC(C)(C)C(F)F)CC3(C)C)c12 44129,C1(O)(C(=O)NC2CC3(C(NC(c4c(C)c(N)ccc4)=O)C3)C2)CCCC(C)(C)C1 44130,C1(N=c2cc(Br)n(C)[nH]2)(c2n(C(C(=O)OC)C)nnn2)C(C)CCC1 44131,c1(C(=O)NCCSC)cc2cc(-c3cn(C)nc3C)ccc2oc1=O 44132,C1(NC(c2cccc(NC(C)=O)c2)=O)CC(C)CN(C(C2CCC(C)(C)O2)=O)C1 44133,C(=O)(C(C)C(=O)N1CCN(CCCNC(=O)C(C)(C)n2cnnn2)CC1)OC 44134,c1(C(=O)NCCC2N(C(c3c(C)con3)=O)CCOC2)c(Cl)cc(Cl)cc1Cl 44135,C1(C)(C(=O)NCCCN2CCN(C(CCSC)=O)CC2)C(C)(C)C1(C)C 44136,C1(C(N2CCC(OC(C)=O)C2)=O)CCN(C(=O)C(C)(C)CO)CC1(C)C 44137,c1(C(N(C2CC(NC(C(CC=C)OC)=O)C2)C)=O)[nH]nc2ncccc12 44138,c1(CCC)n[nH]cc1C(=O)NCC(CNC(C1CCC(=O)C1)=O)CO 44139,CC1(C)CC(=O)NC1CSCC(CO)C1CCC1.C1(C)(C)CN1 44140,c1(CCC(=O)NCCCC(=O)NCC(CC=C)NC(N)=O)ccc(Cl)c(OC)c1 44141,C1(C(=O)NC2CC(C(C)C)OC2)C=CCN(C(=O)Cn2ccnc2)C1 44142,c1(C(C)NC2CC(CCC(N3CCC(SCC)CC3)=O)C2)ncc(F)cc1C 44143,c1(C(=O)NCCCN(C(=O)CC2C=CCCC2)CC)cc(C(F)F)cs1 44144,Cc1nc2ccc(C(C)NS(=O)(=O)Cc3cc(Cl)ccc3Br)cc2o1 44145,N1(C(c2ncc[nH]2)=O)CCC(C2CCCN(c3nccn4nnnc34)C2)CC1 44146,C#CC1CC(NC(c2cn(CC3CC(N)C3)nn2)C)C1 44147,C#CC1(C(N2CC(C(C)(C)C#N)C2)=O)CN(C(c2cc(OC)ccn2)=O)C1 44148,c1(C(=O)OC)ccncc1NC(C12CC(NC(C3COC(=O)N3C)=O)(C1)C2)=O 44149,N1(C(CCC=CC)=O)CCC2C1CCCN2C(C12CC(c3ccccc3)(C1)C2)=O 44150,c1(NC(C2CC(C)C(C)CC2)=O)cccc2c1CN(c1ccccn1)C2 44151,c1(C(N(C2CCN(C(=O)C(C)CF)C2)CCC)=O)ccc(C2CCOCC2)cc1 44152,CCN=c1ccc(C(=O)NC2CC2NC(c2cc(CC(C)C)c[nH]2)=O)c[nH]1 44153,C1(C)(c2nc(CC)[nH]n2)CCN(N2CCC(C)(C(=O)OC)C2)C1 44154,C1(NC(N2CCCC(C(N(C)C)=O)C2)=O)CCOC2(CCC2)C1 44155,C(=O)(C1CCc2nccn21)NCC(C1CCN(C(C2(C(C)C)CCC2)=O)CC1)F 44156,C1(NC(C=NOC)=O)CN(CC2CC2c2ccc(C(F)(F)F)cc2Cl)CC12CC2 44157,N1(C(Cc2c(C)n[nH]c2C)=O)CC(NC(c2cc(CO)ccc2O)=O)C(C#N)C1 44158,C(c1cccc(CO)c1)=CC(N1CCC(C)(NC(=O)CCCc2cnn[nH]2)C1)=O 44159,N1(C(c2c(CC)ccc(F)c2)C(=O)NCCC2CC2)CCC2OC(=O)OC2C1 44160,c1(C(c2cccnc2)C)noc(COC(=O)CCCN)n1 44161,c1(C(=O)NC(C2CCCC2)CC)cc(CNC(C2CCC(F)CC2)=O)nn1C 44162,C1(C(N(C(C#C)C)C)=O)CN(C(=O)Cc2scnc2C)CCO1 44163,c1(C(=O)NCCCNC(C(C)C2CC2)=O)ccnn1-c1cccnc1 44164,C(=O)(CCCc1nccs1)C(C=CCNC(=O)OCC1(NC(C)(C)C)CCC1)=O 44165,CC1CC(C)N(C(=O)CCCC2CC2)CCN1C(c1oc(S(N)(=O)=O)cc1Cl)=O 44166,C(=O)(CCCCCCn1cc(C2CCC2)nn1)N1CCCC(n2c(C)cnc2)C1 44167,n1(C2(CNCCCN(C(C3CC(OC)C3)=O)C)CC2)cc(C)cn1 44168,Cc1cc2ncnc(N3CCC4(CCN(C(c5ccc(F)c(F)c5)=O)C4)C3)c2[nH]1 44169,C12(COC(C3N(c4cc(N)ncn4)CC(O)C3)=O)CCCCC(=O)N1CCC2 44170,c1(OC)ccc(CN2CCC(C(N3CCOCC3C)=O)C(O)C2)c(Br)c1 44171,c1(C(=O)NC2C(CNC(=O)C3=CCC3)CC2)ccc2oc(=O)oc2c1 44172,C1(CC(c2cnccn2)NCC(=O)Nc2cccc(F)c2)CCCC(F)(F)C1 44173,c1(N2CCC(C(N(C)CC)=O)CC2)ncnc(NC2(C)CCC(C)(C)C2)c1C 44174,n1(C(C)C)cc2ncc(C(N3CCC4(CC3)CN(C(C3CC3Cl)=O)C4)=O)cc2n1 44175,N1(C(=O)Cn2cncn2)CCC2CCC(C1)N2C(c1cc2c(nn1)CCCO2)=O 44176,CC(C)CC(F)C(=O)N1CC(CNC(=O)Cc2ccc(O)cn2)C(C)(C)C1 44177,C=Cc1ccc(C(=O)NC(CC#CC)C(=O)NCCC(=O)NC(N)=O)cc1 44178,c1(NC(C2C(C(=O)OC)C2)=O)sc2c(c1C(N1CCC(O)C(F)C1)=O)CCC2 44179,N1(C(C2C(C(=O)OCC)CC2)=O)CCCC1CC(=O)NC(C(C)C)C1CC1 44180,C1(C(=O)NC(CC=C)C(=O)NC(CCO)C2CCC2)CC2(CCO1)CC2 44181,CC1CCN(C(c2ccn(-c3ccccc3)n2)=O)CC1N(C)C(C1CCCO1)=O 44182,N1(C(C(C(C)C)S)=O)CCn2ncc(C(=O)NCC(N3CCOCC3)C)c2C1 44183,c1(C(=O)NCCCCC(C)NC(c2cocc2C(N)=O)=O)nnc(O)cc1O 44184,C1(CC)(NC(=O)CC2CCCN(C=O)C2)CCCCC1.c12cscc1NC2=O.OC 44185,N1(C(=O)Nc2cnn(-c3ccncc3)c2)CCCC2(C1)CC(F)(F)C2 44186,CCC(C)(CNC(C1(C)CC1(F)F)=O)NC(=O)CCCn1cncn1 44187,C(CCCCC(=O)NCC1CCCC1NC(c1ccc(C(C)C)cn1)=O)=CC 44188,c1(C(=O)NCCCN(C(=O)CCOCC(F)F)C)ccc(-c2nc[nH]n2)nc1 44189,C(=O)(C(O)C(C)(C)C)N(CC(C)O)CCNC(C1CC(O)(CC#C)C1)=O 44190,N1(c2n(CC(=C)C)c(CN3CCCC(O)C3)nn2)CCC(O)CC(C)(C)C1 44191,c1(C(=O)NCC=CCNC(C2C(C)(CC)C2)=O)c(C)nn(C)c1C(F)(F)F 44192,c1(SC)ccc2c(c1)C(NCC1CC(COc3ccccc3)CO1)CCO2 44193,c1(C(N2C(CNC(CCSCCCC)=O)COCC2)=O)ccc2c(n1)CCOC2 44194,C(=O)(CC(C(F)F)C(C)(C)C)NCC1CC(OC)CN1C(=O)CN1CCOCC1 44195,N1(C(Cc2scc(C)c2)=O)CCC(F)(C(N2CC(CN(C)C)C2)=O)C1 44196,C1(CNC(CC2(OC)CCCC2)=O)CC(NC(=O)Cc2cncn2C)CC1O 44197,C1(C(=O)N(CCCCCNC(c2conc2C(C)(C)C)=O)C)(OC)CS(=O)(=O)C1 44198,N1(C(c2c(Cl)ccc(C)c2)=O)CCCC12CCCN(C(c1ccc(=N)[nH]c1)=O)C2 44199,C(=O)(C(C(C)(C)C)NC(C1(C)CC(=O)N(C)C1)=O)N(CCOCC#C)C 44200,C(=O)(C(CC(C)C)C(N)=O)N(C)CC1(O)CCN(C(CC(CC=C)(C)C)=O)CC1 44201,c1(C(=O)OC)ccoc1C(=O)NCC(C)N(C)C(c1csc(C(C)(C)C)c1)=O 44202,C(=O)(C(O)CCS(C)=O)N1CCC(N(C)C(C2(CN(C)C)CC2)=O)CC1 44203,N1(CCNC(CC2(N(C(COCCSC)=O)C)CC2)=O)C(=O)CNC1=O 44204,C1(NC(=O)C=C(Cl)Cl)CCCC12CN(C(c1cn(CC3CC3)nn1)=O)C2 44205,O(N(C)C(=O)CNC(C(C)(C)SC)c1nnnn1C1COC1)CC 44206,CCC(C)(O)C(=O)N(C)C.N1(CC2(C=O)CC2)CCN(C(=O)Cn2cccn2)CC1 44207,c1(SCC(N2CCC(CCCC(=O)OC)CC2)=O)nc2ccccc2n1C 44208,N=c1nc(N2CC(CC(N)=O)C(CC(N)=O)C2)[nH]c(=NCC2CCCC(=O)N2)[nH]1 44209,c1(C(=O)OCC)cc(F)c(C(=O)NC(C(C)NC(=O)C=C(C)C)C(C)C)cc1F 44210,C1(NC(c2ccc(O)nc2)=O)CC2CN(C(c3ccc(S)cc3)=O)CC2C1 44211,C1(C(=O)NCCc2c(CNC(c3c(C)n(C)nc3)=O)nco2)CCC(O)CN1C 44212,c1(C(=O)NCCC2N(C(C(SC)SC)=O)CCCC2C)ccc2occc2c1 44213,C1(NC(CC(C)(C)O)=O)CCOC12CCN(C(c1cc3ccccc3[nH]1)=O)CC2 44214,C12(C(N3C(C(=O)NC(C)CCO)CC(F)C3)=O)CCC(CC1)CC2 44215,c1(C(=O)NC(CC(C)NC(COC(C)=O)=O)C)cc(C)c(Br)o1 44216,N1(C(C(C=C)(C)CC)=O)CC(C)(C)C(NC(C2CC=C(C)CC2)=O)C(C)(C)C1 44217,CCC(CC(=O)N1CCC(OCCCNC(=O)CC2CCOC2C)CC1)SC 44218,N1(C(C(C)Sc2nncn2C)=O)CC(CNC(C2COCCN2C)=O)CC1C 44219,C(=O)(CCCC(=O)N1CC(CNC(=O)CCCCCN(C)C)(OC)C1)OCC 44220,c1(C(N2C(CNC(C3N(CC)CCC3)=O)CC2)=O)c(C)cn(C)c1CC(=O)OC 44221,C(=O)(C1=CCC(C)CC1)NCCC(C)NC(C1(CC(C)C)COC1)=O 44222,C(=O)(CCCCC(F)(F)F)NCC1CN(C(C(CC)C(C)(F)F)=O)CC1(C)C 44223,N1(C(c2c(CC)ncs2)=O)CC2CN(C(c3cc(C)c(OC)c(Cl)c3)=O)CC2C1 44224,CC12CCC(CC(=O)NCCC3(O)CCCN(C(C4(C5CC5)CC4)=O)C3)(CO1)C2 44225,N1(C(C2=C(C)CC2)=O)CC2(CC(NC(=O)C(c3ccnn3C)O)CO2)C1 44226,Cc1nccnc1C(=O)N(CC(C)(C)C(=O)NCC(C)(C)CN(C)C)C 44227,C(C)(CCC(=O)NCC(C)(C)OCCNC(=O)CCNS(C)(=O)=O)SC 44228,CN1CCOc2ccc(C(=O)NCC(O)CNC(C3CC3(Cl)Cl)=O)cc21 44229,C1(NC(C(CCC)c2ccccc2)=O)CN(C(c2ccc(F)cc2)C)CCC1C 44230,c1(C(=O)OC)cccn(CC(N2CCC2CNC(C2(C(C)C)CCC2)=O)=O)c1=O 44231,N1(C(C(CCSC)(C)C)=O)CCC2(CCCN2C(c2ncc(Cl)cc2Cl)=O)C1 44232,N1(C(c2cc(Cl)ccn2)C(=O)NCC=C)CCOC2(CCSC2)C1 44233,C1(C(=O)NC(c2ncc(C)[nH]2)CC)CCN(C(C2CC23CCCC3)=O)CC1C 44234,C(=O)(C#CC(C)(C)O)NCC1CC(COC)CN1C(C1CC2CC1CO2)=O 44235,c1(C(=O)NCC2(C(=O)NC(C(C)(C)O)CCO)CC2)ccn2cncc2c1 44236,N1(C(C(CC)NC(N)=O)=O)CC2(CCN(C(=O)C=C3CCC(C)C3)CC2)C1 44237,c1(OCC)ncc(C(=O)NC2CCC(NC(C3(C)CCOC3)=O)CC2)cn1 44238,C(=O)(C(F)CC(C)(C)NC(=O)Cc1cnn(C)c1)N(C)CCOCCCN(C)C 44239,c1(C(=O)NC(C)(C)CNC(C2CCC(Cn3ccnc3)O2)=O)cc([N+](=O)[O-])n[nH]1 44240,c1(OC)cc(O)c(CNC2(CC(N3CCC(O)C(C)C3)=O)CCC2)c(Br)c1 44241,N1(CC)CCCC(C(=O)NCC2(CNC(=O)CN(C)C3CC3)CC23CCC3)C1 44242,C1(C(N2CCOC(C)(CNC(=O)CSC)C2)=O)(COC)CCCNS1(=O)=O 44243,N1(C(c2cn(CC)nc2)=O)CCCC2(CC(NC(=O)CC3CCCC3C)C2)C1 44244,c1(CC)ccc(CNC(C2CC2CNC(C2(C)CCOC2)=O)=O)cc1 44245,N1(C(C=CCOC)=O)CCC(C(=O)NCC2CN(C)CCO2)C1(C)C 44246,N1(C(c2c(C)c[nH]n2)=O)CC2CCCC2(NC(c2occ3c2CCC3)=O)C1 44247,C1(NC(CCC(=O)NCC)=O)CCN(C(=O)CCc2ccc(F)cc2Cl)CC1F 44248,CC(C)C(C)C(C)CC(=O)NC(C)(C)COCCCNC(c1cnc[nH]1)=O 44249,N1(C(C(CC)(C)C)=O)CC23CCCC2(C1)CN(C(c1cnc(OC)nc1)=O)C3 44250,C(=O)(C(CC)ONC(C1(C)C=CCC1)=O)NC1CC(COC)C1 44251,N1(C(c2ccc(CCC=C)cc2)=O)CC2CC(NC(c3snc(C)c3N)=O)C1C2 44252,Cc1nc2ccc(C(=O)NC(C)CN(C)C(c3cc(C4CC4)ncn3)=O)cn2n1 44253,c1(OCC(=O)N(C(C)CCNC(c2cnc(C(F)F)s2)=O)C)ccc(Cl)cc1F 44254,Cc1ccccc1C(=O)N(C1CCCC(N(C(=O)Cc2ccsn2)C)C1)C 44255,C(=O)(CC(O)CCCCC)NCC(CC=C)NC(=O)CN1CCN(CC)C(=O)C1=O 44256,c1(OC)cc(N)c(Cl)cc1C(N1CC(N(C)C(C23COCC2C3)=O)C2(CC2)C1)=O 44257,c1(C(N(CC(C)NC(C2(C(F)F)CCC2)=O)CC)=O)cc(C)c(Br)c(C)c1 44258,N1(C(C2C(CC)CCN2C(C2CC(F)(CF)C2)=O)=O)CC(CO)CC(C)C1 44259,N1(C(c2cc(CNC(C(CCC)F)=O)on2)=O)CCC(O)C(F)C1 44260,c1(C(N2CCCN(C(C=CCOC)=O)CC2)=O)cc2nc(C)cc(C)n2n1 44261,C(C(O)C(=O)N1CC=CC1)NC(=O)CC1CCCO1 44262,c1(C(N2CC(CNC(COCCOC)=O)C(C)(C)C2)=O)cc2cc(Cl)ccn2n1 44263,N1(C(CC2(OCC)CC2)=O)CCC(C(=O)NC(C)Cc2cccs2)C(C)(C)C1 44264,c1(C(=O)NCCCCCN(C(c2c(C)snn2)=O)C(C)C)cncc(N)c1 44265,Cc1cccc(Br)c1-n1cc(CCCCC(=O)N2CCCC2c2ncon2)nn1 44266,c1(CCC(=O)NC(C2CCN(C(C3C(=C)C3)=O)C2)(C)C)cn(C)c2ccccc12 44267,c1(NC(C2C(NC(CN3CCC(C)C3)=O)COC2)=O)cncc(C2CC2)c1 44268,O(C=CC(=O)N(CCC(C)NC(=O)CC1CC(C)(C)C1)C)CC 44269,CC(C)C(C(=O)NC1CCCN(C(=O)COC(C)(C)C)C1)c1cccnc1 44270,C(C)(CCC(=O)NCC(O)CNC(C1(c2cccs2)CC1)=O)OC 44271,c1(CC(=O)NC2CCN(c3cc(Cl)c(O)nn3)C2)cn2cc(F)ccc2n1 44272,C1(NC(c2cnc(OCC)s2)=O)C2CCN(C(=O)CSc3nncn3C)CCC12 44273,c1(C(N(C2CCCN(C(c3cnsn3)=O)CC2)CC)=O)ccc2c(c1)CCNC2=O 44274,N1(C(C(C)NC(C)=O)=O)CC(O)(CN(C(=O)CC2COCC2O)C)C1 44275,c1(NC(C(N2CC(CC(=C)C)(NC(C3(CCC=C)COC3)=O)C2)=O)=O)ccc(O)cc1 44276,c1(NC(C(=O)NCC(CC=C)NC(=O)C(C)(C)SC)C)ccc(C(F)(F)F)cn1 44277,N1(C(c2c(CNC(C3(C#N)CC3)=O)occ2)=O)CCC(O)(C(F)F)C1 44278,C1(CC)CCC(C)N(C(=O)CCOCCN(C)C(c2nnc(S)n2C)=O)C1 44279,N1(C(C(C(C)C)O)=O)CC2CN(C(C34CSCC3C4)=O)CC2C1 44280,C1(C(=O)NCCC#C)CCN(C(=O)c2cccc(Cl)c2)O1 44281,CC1COc2c(C(=O)NC3C4CC3N(C(c3cc(=O)cc(Cl)[nH]3)=O)C4)cccc21 44282,C1(C)(C(=O)NC(CCC)(C)CC)CN(C(=O)CC2CCCN(C)C2)CC1C 44283,c1(C(N2CCCC(NC(C3(COC)CC=CC3)=O)C2)=O)cc(C)c(C)nc1C 44284,Cc1nc2[nH]c(C(N3CCC4(NC(c5ccc(F)cn5)=O)CC4C3)=O)cc2s1 44285,C1(NC(C(C)(C)OC)=O)CC2CCC1CC2NC(C1(C)CC=C(C)CC1)=O 44286,CC1(C(=O)NCCC2CCN(C(=O)COC3CCC3)C2)CCOC1 44287,Cc1nc2cccc(C(=O)NCC(C)NC(=O)C(F)n3cccn3)c2s1 44288,C12(C(N(C3CN(C(C4(c5cccc(C)c5)CCC4)=O)C3)C)=O)CCC(F)(CC1)C2 44289,C1(CN(C(C(C)C)=O)C)CN(C(C2CCS2(=O)=O)=O)CCO1 44290,c1(NC(C(c2ccccc2F)NC(C(C)=O)=O)=O)cccc2cncc(C)c12 44291,CCCCCC(CC)C(=O)NCC1CC2(CC(NC(C3(CCC)CCC3)=O)C2)C1 44292,Cc1cc(CC(=O)N(CC)CC2CCCC2)n(C)n1.C1(=O)C(C)(C)N1 44293,c1(CC(=O)NCCN(C(=O)C(C)(O)CC)CC)ccccc1S(=O)(=O)C(F)F 44294,C(C(=O)NC12CC(CNC(=O)CSC(F)F)(C1)C2)(c1ccccc1)=C(C)C 44295,Nc1cccc(F)c1C(=O)NCC1CCN1C(=O)C(c1ccncc1)C1CCCO1 44296,C(=O)(CCCC(C)(C)C)N1CC(CCC)C(C(=O)NCC=CCOC)C1 44297,CC(C(C)NC(=O)CC1CC1)S(C)(=O)=O.C1CCC(=O)N1 44298,c1(OC)cc(Cl)ccc1CNC1CC1C(N1CCC2(CC1)CC2)=O 44299,C1(NC(=O)NC2(CN(C)C(C3CSCCS3)=O)CC2)CCCC1c1nc[nH]n1 44300,N1(C(C(C(C)(C)C)N2CCCC2)=O)CCC2(CC1)CC2CNC(c1ccon1)=O 44301,C1(C(=O)NC2C(CNC(=O)CCC3CCCCO3)CCC2)CC2OC1C1CC21 44302,C(=O)(C1COc2ccc(Cl)cc21)NCCN(C(C1CCC1C(F)F)=O)CC 44303,N1(C(CCC(C)(F)F)=O)CCC2(CC(NC(=O)C(C)(F)C(C)(C)F)C2)C1 44304,C1(CC)CN(C(=O)Cc2nccn2C)CCC1NC(c1c[nH]c(C)c1)=O 44305,c1(CNC(C2(C)CN(C(=O)CC3CC4CCC3C4)C2)=O)cnc(C(F)F)nc1 44306,n1(CC)cc(Cl)c(C(=O)N(C(C)CCNC(=O)Cc2ncc(C)[nH]2)C)n1 44307,N1(C(c2cnc(CC(C)C)s2)=O)CCCC(C)(NC(c2cc(F)cc(Cl)c2)=O)C1 44308,c1(OC)cncc(C(=O)NCC2CN(C(=O)CSCc3cccs3)CC2O)n1 44309,c1(C(=O)NCC2N(C(C34CCC(C)(CC3)CC4)=O)CC2)cccc2c1COCC2 44310,C(C(C)C)(C(O)C(=O)NCCCn1cc(CCCC(C)(C)C)nn1)OC 44311,N1(C(C2CCCN(CC)C2)=O)CCCC2CN(C(=O)C(F)CC3CCCC3)CC12 44312,c1(C(N2CC(CNC(C3(CCCC)CCC3)=O)C(C)C2)=O)cc2c([nH]1)CCCC2 44313,O(N(C)C(=O)CN=c1[nH]c(=NC(C)CC2CCCO2)[nH]c2c1COCC2)CC 44314,C=CCCCC(C(=O)NC1CCC(C(N)=O)C1)NC(=O)CC1(OC)CCC1 44315,[N-]=[N+]=NCCCCCCC(=O)NCC1CN(C(=O)CC23CCCC2C3)C1 44316,C1(C)(C(N(C)C)=O)CCCCO1.C1(C)COCC1NC(c1coc(CO)c1)=O 44317,N#Cc1ccc(C(=O)NCC(N2CCN(C(=O)C(F)(F)C(F)F)CC2CF)=O)cc1 44318,c1(NC(C2CCN(Cc3ccc(C)[nH]3)CC2O)=O)cccc2c1OCO2 44319,c1(N(C(C(n2c(CCCC)ncc2)C)=O)CC2CC2)ccc(F)cc1 44320,C(=O)(C1=C(Cl)CCCC1)NC1CN(C(Cc2c(C)scc2)=O)CC(F)C1 44321,C1(CC(N2CCC(CCNC(c3ccc(C(=O)OC)s3)=O)C2)=O)CCN(C)C1=O 44322,Cc1sc(Br)cc1S(=O)(=O)N1CCC2(O)CCOCC2C1 44323,S(=O)(=O)(c1ccccc1)NC(C)C(=O)OCC(=O)Nc1cc(O)ccc1F 44324,N1(C(CCS(=O)(=O)NC(C)=O)=O)CC2CC1CCC2NC(C1(C(F)F)CCC1)=O 44325,N1(C(CC(c2ccc(C)cc2)C)=O)CC2CC(NC(=O)CC3CC=CCC3)C2C1 44326,c1(CC(C(N)=O)NC(C2CCCN2C(c2ncccc2F)=O)=O)ccc(O)cc1 44327,CN1CCOCC1CC(=O)NCc1ocnc1Cn1cc(C2CC=CCC2)nn1 44328,C12(COC)COC(C(=O)NC3CCCCC3NC(c3c(C)coc3SC)=O)(C1)C2 44329,Cc1ccc(C)c(SCC(N2CC3C(C2)N3C(=O)C(C)O)=O)c1 44330,C1(NC(C2CCC(C)O2)=O)COCCN(C(c2cccc(Br)c2F)=O)C1 44331,N1(C(C(SC)SC)=O)CC(NC(=O)Cc2cc(C)on2)CC(C)C1 44332,C#CCC(C)(C)CNC(=O)C(CCOC)NC(c1[nH]ccc1C)=O 44333,c1(OC(C)C(=O)NC(C2CCCN2C(=O)CC2CS(=O)(=O)C2)C)ccc(F)cc1 44334,N1(C(C(N2CCSCC2)C)=O)CC2CCN(C(c3cccc(N)c3)=O)C2C1 44335,C1(C(=O)NCCOCCNC(CC(C(=C)C)OCC)=O)Cc2ccncc2C1 44336,C(=O)(CC(C)CF)NCCCN(C(COCCOCCOCC#C)=O)C(C)C 44337,C(=O)(N=c1c(Br)c[nH]c(C)c1Br)C1N(C(c2c(OC)ccc(C)c2)=O)CC(O)C1 44338,C(N=c1[nH]c(=NCCC=CBr)[nH]c2c1CCCCCC2)C1(C)CCC(=O)N1 44339,c1(C2C(CC(=O)NC(C3(O)CN(C(c4c[nH]nc4Cl)=O)C3)C)C2C)ccccc1 44340,N1(C(c2cc(C)no2)=O)CCC2CCC(C1)N2CC1CCC2CC2C1 44341,O=C1CCc2c(C(N3CCOC(C4CC(F)(F)C4)C3)=O)n[nH]c2C1 44342,c1(C(=O)NC(c2cn(-c3ccc(C)o3)nn2)CCC)ccnn1CCC 44343,C1(C2(NC(C(=C(C)C3CC3)F)=O)CC2)CCCCN1C(=O)CCn1ccnc1C 44344,C1(CN(C)C(C2CC23CCC3)=O)CCN(C(c2ccccc2OCC#N)=O)CC1 44345,C1(NC(C(C)C2CCC2)=O)CN(C(c2cc3cnccc3[nH]2)=O)CC2CCCC12 44346,C(=O)(C(CCC1CCC1)NC(c1c[nH]c(C)c1)=O)NCCOC 44347,C1(NC(c2ccn3nccc3c2)=O)CN(C(=O)CC2CC2(Cl)Cl)CC2(CC2)C1 44348,C(=O)(CC1(O)CCOc2ccccc21)N1CC(C)(C)c2c1cccc2 44349,c1(CCC)cc(C(N2CCC(C(C)NC(C3(CC(C)C)CC3)=O)C2)=O)n(C)n1 44350,c1(OC)cc(C)c(C(N2CC=CC(NC(=O)Cc3ccn(C)n3)C2)=O)cc1Cl 44351,N1(C(C2(NC(C(CC=C)OC)=O)CCC2)=O)CCN(C2CC2)C(C)C1 44352,N1(C(c2c(C)cccc2)=O)CC2CCCC(C1)N2C(=O)COC1CCCCC1 44353,c1(CC)cc(OCCNC(=O)C(CC)c2nc(=N)[nH][nH]2)cc(C)c1 44354,N1(C(CC2(NC(c3cc(CCO)on3)=O)CC2)=O)CC(O)(C(F)F)C1 44355,N1(C(c2cn(CCC)nc2)=O)CCN(C(=O)CCC(C)OCC)CC1CCO 44356,C(CO)(C(=O)NCC1(C(=O)NCC2CCOCC2)CCCC1)NC(N)=O 44357,c1(C(=O)NCC2OCC(CNC(=O)C(Cl)=CCl)C2)cnn2ncccc12 44358,N#CC1CCCC(C(=O)NCC2CC(CNC(C3CC4C=CC3CC4)=O)C2)C1 44359,C12(NC(C34N(C(=O)CN5CCCC5=O)CCC3C4)=O)CCC(O)(CC1)CC2 44360,c1(C(N2CCCCC(NC(C(CC)(C)OC)=O)CC2)=O)c(F)cc(C#N)cc1F 44361,C1(C(N(CCn2ncc(C)c2)C)=O)CC(C)CN1C(c1ccc(O)cc1)=O 44362,C1(CNC(c2cc(OC)ncn2)=O)CCC2(CO1)CC(NC(c1cncs1)=O)C2 44363,c1(C(=O)NCC2(CNC(CCOC)=O)CC23CCC3)cc(OC)cc(C#N)c1 44364,Cc1ccc(NC(C2CC2NC(c2ccc(F)cc2F)=O)=O)cc1Br 44365,CN1CCN(C(C2(O)CCCCC2)=O)CC1C(=O)NCc1ccc(C(N)=O)o1 44366,Nc1cc([N+](=O)[O-])ccc1C(N1CC(NC(=O)Cn2cccn2)C2(CCC2)C1)=O 44367,c1(C(=O)NCC(C)(C2CCC2)NC(C2CC2F)=O)cc(Cc2ccccc2)c[nH]1 44368,C(C(=O)NC(CCSC)C(=O)NCC1C=CCC1)(C(C)C)OCC 44369,c1(OC(c2nc(-c3nccs3)nn2C(=O)NC2CC2)C)ccc(F)c(Cl)c1 44370,C=CCN=c1[nH]cc(C(=O)NC(C2CN(C(=O)CC(C)C)CCO2)C)s1 44371,C=C1CC2CCCC(C1)N2C(C1CC(NC(c2ccc(C)cc2F)=O)CCO1)=O 44372,N1(C(C23CC(C)C2C3)=O)CCC2(CC1)CC2CNC(c1cnn(C)c1Cl)=O 44373,c1(NCC(N)=O)[nH]c(=NCC2CC=CCC2)nc2scnc12 44374,Cc1ccc(N2CCOC(C(=O)NCC3CCN3C(=O)OC(C)(C)C)C2)nc1Br 44375,C#CCC(C)(CC)C(=O)N1CCC(c2cccc(F)c2)(NC(=O)CC(F)F)C1 44376,c1(C(N2CCCC(C(F)(F)F)C2)C(=O)NC2CC(C(=O)OC)C2)cccnc1N 44377,CCC(C)(COC)C(=O)NC(CNC(=O)C1=COCCC1)C1CC1 44378,C12(CC)CN(C(=O)Cn3cnnn3)C(CNC(C3CCS(=O)(=O)N3)=O)(C1)C2 44379,N1(C(C(C)OCCC(C)C)=O)CCC(O)C(NC(=O)CN2CCC(C)(C)C2)C1 44380,c1(-c2cn(CC3N(C(CC(CN(C)C)O)=O)CC=C3)nn2)cccc(C)c1Br 44381,O=C(C1=CCC(F)(F)CC1)N1CCN(C(C2(C3CCCCO3)CC2)=O)C(CO)C1 44382,N1(C(CCC2CCN(C(C(C)C3CCOC3)=O)CC2)=O)CCc2n[nH]cc2C1 44383,CC1CN(C(C2CC(=O)N(O)C2)=O)CCCN1C(c1csc([N+](=O)[O-])c1)=O 44384,C1(CC)CN(C(CCC2CCC2)C(=O)NCc2ccco2)CC1O 44385,C(C(=O)NCC(O)CCNC(=O)CCCc1cccnc1)(C(C)O)NC(C)=O 44386,c1(C(=O)NC2(C(N(CCC(N)=O)CC)=O)CC2(C)C)cnn(C)c1C#N 44387,C(=O)(CC(C)(C)CN(C)C)NC(C(C)C)CNC(c1ccnn1C1CC1)=O 44388,CC1(C)C(CC(=O)NCCCCCO)CCN1C(=O)C(O)CN1CCCC1 44389,Cc1nc(C(N2CC(NC(C3(C(F)F)CCCCC3)=O)C(C(F)F)C2)=O)n(C)n1 44390,CCC(C(=O)N(C(C)C(=O)NCC1CCCCO1)C1CC1)N(C)C 44391,C(=O)(C(F)(F)C(F)(F)C(F)F)N1CCCC(CNC(=O)C(c2ccccc2)F)C1 44392,C12CC(=O)N(C1)CCN2.c1(SCC2C(NC(C3CC(CC)C3)=O)C2)ccccc1 44393,CCC(C)CCC(=O)N1CCCC1CCC1CCN(C(C2CC2(F)F)=O)CC1 44394,Cc1cc2[nH]c(C(=O)NC3C4CN(c5ncnc6cc[nH]c56)CC34)cc2s1 44395,C1(NC(CCC(N)=O)=O)CN(C(c2cnn3c2OCC3)=O)C2CCCC12 44396,C(=O)(CCCCC(N)=O)N1C(C=CC(N2C3CC(=C)C(C3)C2)=O)CCC1 44397,C(=O)(C#CC1CCCOC1)NC1CC2CN(C(c3nc(CC)[nH]n3)=O)CC21 44398,C1(NC(C2CC(N(C)C)C2)=O)COCCC1NC(c1nc(Cl)sc1Cl)=O 44399,C(C1c2ccsc2CCN1C(c1[nH]ncc1C#N)=O)NC(C(CC(C)C)OC)=O 44400,N1(C(c2cn(CCC)nn2)=O)CCN(C(=O)CC(CC)C(C)C)CC2(CC2)C1 44401,CC(C)C(CN(C1CC1)C1CC1)C(=O)NC1CCC(F)(F)CC1 44402,C1(C(=O)NC2CN(C(=O)CN(C(C)C)C3CC3)C2)CCOC(=O)CC1 44403,c1(C(N2CCC(CSc3ccccc3)C2)C(=O)NCC)ccn2nccc2c1 44404,c1(CNC(=O)C(N2CCCC(N3CCNC3=O)C2)=O)ccc(Cl)c(F)c1 44405,C#CC1(C(=O)NCC2CC2Cl)CN(C(=O)CC2CCCC2C)C1 44406,O=C(C1=CCCN(Cc2cc(Cl)ncc2Br)C1)Nc1ccnc(CO)c1 44407,CC1CC(NC(=O)C(F)=CC2CC2)CN(C(=O)C(C)(O)c2ccccc2)C1 44408,c1(OC)nsc(OC)c1C(N1CCC(CCNC(=O)CC2CC23CC3)CC1)=O 44409,c1(OC)ccc(C(=O)NCC(CO)NC(c2c[nH]ccc2=N)=O)c(C)c1 44410,N1(C(C2ON=C(C)C2)=O)CC(N=c2[nH]c3c(C)cccc3o2)C2(CCOCC2)C1 44411,C(=O)(CN=c1cc[nH]cc1)N1CC(NC(C2COCCO2)=O)CC12CCC2 44412,C1(CNC(C(CC)F)=O)CC2(CCN(C(=O)CCc3cc(Cl)no3)CC2)C1 44413,c1(C(=O)NCC(c2ccsc2)O)cc2cccc(Br)c2o1 44414,N1(C(CCCSCC)=O)CCN(CCNC(=O)CC2CC3COCC23)CC1.CC(C)(C)O 44415,C1(NC(c2c(C)[nH]nc2C(F)(F)Cl)=O)CN(C(C2CC2C)=O)CCC1CO 44416,C(C1=NOC2(CNC2)C1)N1C(=O)CN(c2ccc(Br)c(F)c2)C1=O 44417,c1(OC)ccc(CNc2ncnc(NCCC(O)COC)c2C)c(OC(F)F)c1 44418,c1(C(=O)NCC(C)N(C(CC(CC)O)=O)C)nc(O)nc(O)c1N 44419,c1(C(N(C(CCNC(c2c(Cl)cn(CC)n2)=O)C)C)=O)ccc2cnccc2n1 44420,CC1=NNC(=O)C1CC(N1CCOC(CCNC(=O)C(C)(C)C2CC2)C1)=O 44421,C1(CC(=O)NC(CC)(C)CNC(c2cn[nH]c2)=O)Cc2cccc(Cl)c2O1 44422,C1(NC(COCCOCCOC)=O)CN(C(=O)Cc2ccno2)C2(CCOC2)C1 44423,CCCC(O)C(CO)NC(=O)NC(Cc1ccccn1)CO 44424,c1(CC)ccc(OC)cc1C(N1CCCCC1CN(C)C(C1CCCN1C)=O)=O 44425,C1(CNC(C2C(CCC)C2)=O)CCC(CNC(C2CCC3(CC3)C2)=O)CC1 44426,C12(NC(C3CC(=C)C3)=O)CCC(CC1)N(C(=O)C(C)(C)NC(=O)OC(C)(C)C)C2 44427,C(CC1c2ccccc2CCN1C(=O)C(C)C(C)C)NC(CCOCCOC)=O 44428,C12(C(N3CCCC(CNC(Cc4ccc(OC)cc4)=O)C3)=O)CCC(C)(C1)OC2 44429,c1(NCc2c(C)noc2)[nH]c(=NCCn2ccnc2)nc2ncn(C)c12 44430,N1(C(C(=O)Nc2c(C)n(C)nc2)=O)CCOC2(CC1)CCS(=O)(=O)C2 44431,C=C(C)c1ccccc1NC(C1CC12CN(C(c1cc(C(C)C)n(C)n1)=O)C2)=O 44432,C1(NC(c2c(CNC(C(CCOC)C)=O)cc[nH]2)=O)CCn2cncc2C1 44433,C1(C(N(C)C)=O)CCCN(C(=O)C(=O)NC2COCC2OC2CC2)C1 44434,c1(C(=O)NCC2CC(COC)CN2C(C2CC(C)(F)C2)=O)cc2cccnc2s1 44435,CC1(C(=O)NC2CCCC2NC(c2ccc(F)c(F)c2)=O)CCCS1(=O)=O 44436,C1(CN(C(CC2C(CC)C2)=O)C)CN(C(c2ocnc2C)=O)CC12CC2 44437,c1(SC)cc(=NC(=O)C2CCN(C(=O)CC3CC=CCC3)CC2C)[nH]n1C 44438,c1(C(C(=O)NCCCNC(C=CC(CC)C)=O)O)ccc(Cl)c(F)c1 44439,c1(OC)c(C(=O)Nc2cncc(-c3ccc(SC)cc3C)c2)ccc(Cl)c1Cl 44440,c1(C(N2C(C)C(C)N(C(c3nnn(C)n3)=O)CC2)=O)cc(F)cc2ccoc12 44441,C=CCC(C)(C)CC(=O)N1CCN(C(=O)Cc2cc(OC)no2)CC1CF 44442,C12(C(=O)NC(c3c(C)cccc3)C)CC(C)(CN1C(c1cc(O)n(C)n1)=O)C2 44443,c1(NC(C(C)C)CNC(=O)CC2CCCOC2)ncncc1I 44444,c1(CN2CCC(C(=O)Nc3c(C(=O)OC)csc3C)C2)cccc2c1OC(F)(F)O2 44445,N1(C(C(=O)Nc2cccc(C(C)(C)C(F)(F)F)c2)=O)CC(CO)CC(CO)C1 44446,C1(CCNC(C2(C=C)CC2)=O)CN(C(C2OCCC2C(F)(F)F)=O)CCS1(=O)=O 44447,c1(C(=O)NCC2N(C(C(COC)(C)COC)=O)CC2)cc2c(ncn2C)[nH]1 44448,Cc1ccc2c(c1)C(C(=O)NC1CC(NC(=O)Cc3nn(C)cc3Cl)C1)OCC2 44449,C(C(O)C(=O)NC1CC1c1cn(C2CC2c2ccccc2)nn1)SC 44450,Cc1cc(C)c(NC(=O)NCC2CC(c3ccc(C(F)(F)F)cc3)C2)c(S)n1 44451,C1(NC(C(COC)(F)F)=O)CCC(C)N(C(c2ccc(-c3ccco3)[nH]2)=O)C1 44452,O(NC(=O)C(COC)NC(C12CC1CNC2=O)=O)CCOCC#C 44453,N1(C(C2CC(C#C)(O)C2)=O)CC(C)(C(=O)NC2CCOC2=O)CC1(C)C 44454,c1(C(N2CC(CC(=O)Nc3ccc4sncc4c3)C2)=O)c(O)cccc1[N+](=O)[O-] 44455,N1(C(CCCNC(C)=O)=O)CCN(C(=O)C(c2ccc(Br)cc2)C)C(C)C1 44456,n1(CC=C)nnnc1C(c1ccc(-c2ccccn2)s1)NCc1ccc(CC)o1 44457,CCC(C(=O)NCCCOCCNC(c1cncn1C)=O)Sc1nc(=N)[nH][nH]1 44458,C=CCC(CNC(C1C2CCC(C2)C1C)=O)C(=O)N(C1CCN(C(=O)CC)C1)C 44459,C1(CNC(C(C(C)C)C)=O)CN(C(=O)Cc2ccnn2C2CCC2)CC(C)(C)C1 44460,C1(NC(c2ccc(O)nn2)=O)(CO)CCCN(C(=O)Cc2ccc(O)cn2)C1 44461,Cn1cc([N+](=O)[O-])c(C(=O)NCC2(F)CCN(C(=O)CN3CSCC3=O)C2)n1 44462,c1(CC)oc(C(N2CC(CC(=O)NCC(C)CC3CC3)C(C)C2)=O)cc1C 44463,n1(CCC(=O)N(C2CN(C(c3c(C)oc(C4CC4)n3)=O)C2)C)ccc(O)nc1=O 44464,C1(C(N2CCOCC2)C)CCCCN(c2nc(=N)nc(N3CCC(N)C3)[nH]2)C1 44465,C1(NC(C(c2ccccc2Cl)C)=O)CC2(C1)CC(CNC(c1ccc(Cl)o1)=O)C2 44466,C(=O)(C1=CCCC1C)NCC1CC(COC)CN1C(C1OCCC1C)=O 44467,C1(C(C)C)(C(=O)NCCC2CN(C(=O)C(O)C(F)F)C2)CNC(=O)C1 44468,c1(OC)ccc(NC(C2CC3CC3N2C(=O)Cc2ccccc2OC)=O)cc1C 44469,C(CCNC(=O)CC1CC2CC2C1)(C(=O)N1CCOC(CC(C)C)C1)OC 44470,c1(CCC(=O)NC2CC2CNC(c2ccc(-c3cc[nH]n3)s2)=O)nc(O)n[nH]1 44471,c1(C(=O)NC2C(CNC(C3C(CCC)C3)=O)C2)cnnn1C 44472,N1(C(CC=C(C)C)=O)CCC2(CC1)CN(C(C1CC3CC1CC3O)=O)C2 44473,C(C(=O)N1CCC(C)(CNC(=O)C(O)CN(C)C)CC1)(C(F)(F)F)OC(C)=O 44474,C1(NC(C2C3CNCC2C3)=O)CC12CC(=C1CCC1)C2 44475,S(=O)(=O)(c1ccc(F)cc1)NC(CC(=O)N(CC(C)NC(C)=O)CC)C 44476,C1(COC)(CNC(C2OCCC2C)=O)CCN(C(C2CC(OC)C2)=O)C1 44477,N1(C(C2(CC)CCCN2C(C2CCC(N(C)C)C2)=O)=O)CC(C)OC2(CCC2)C1 44478,C(=O)(C(CNC(=O)CCn1cnnc1)C(C)(C)C)NCc1cn(CC)nn1 44479,N1(C(c2c(C)cncc2)=O)CC2(C1)SCCC2NC(=O)CCCCN(C)C 44480,N1(C(COC(C)C)=O)CCC(C=CC(=O)NCC2CC(C)CO2)CC1 44481,N1(C(C(C)NC(=O)OC(C)(C)C)=O)CCC2(CC1)CC2NC(=O)C(C)(F)F 44482,c1(C(=O)NC(C2N(C(C(CC3CC3)OC)=O)CCC2)C)ncc(Cl)cc1F 44483,C(=O)(CC(C)P(C)(C)=O)NC(CCCC)CNC(=O)C(C)(C)OC(C)C 44484,Cc1cc(Cl)c(C(=O)NCC2(F)CCN(C(c3cnncc3O)=O)CC2)cc1C 44485,n1(CC(N2C3CC(CNC(C(C)OC)=O)CC2CC3)=O)cnc2cc(C)ccc12 44486,C(=O)(C1=CCCCC1C)N1C(C(=O)NCCn2ncc(CC)c2)COCC1 44487,c1(C(N(CC)CC2CCCN2C(=O)CN(C)C)=O)ccc2c(c1)CCCCN2 44488,n1(CC(=O)NC2(CO)CN(C(=O)CCCC3CCCC3)C2)nnc(C2CC2)n1 44489,CCCC(CC)C(=O)NC1(CC)CCCN(C(c2ccoc2)=O)C1 44490,c1(C(=O)NC(CN2CCN(C(C(CC)OC)=O)CC2)C)cc(C)ccc1F 44491,CCC(CC(=O)NCC1CC1C(=O)NC(C)CC(F)(F)F)CC(C)C 44492,CC1(NC(=O)C(C2CCN(C(=O)Cc3csnn3)C2)F)CC2(CCC2)C1 44493,C12(CCNC(c3c(C)noc3)=O)CCC(CC1)N(C(c1ccc(F)c(F)c1)=O)C2 44494,c1(COC)ccccc1C(=O)NC(C)C(C)NC(c1cc(Br)cn1C)=O 44495,Cc1cc(F)c(CNC2CN(C(c3cc(Br)nc(Br)c3)=O)CCC2(F)F)cc1Br 44496,Cc1c(C(=O)NCC2(NC(C3CC(=O)CCO3)=O)CCC2)cncc1F 44497,c1(OC)cnc(C(=O)NCC(C)(C)OCC(=O)NCC(N)=O)cn1 44498,c1(C(N2C(CCNC(C(C)OCCCC)=O)CCCC2)=O)cc(F)c(C)cc1Cl 44499,CC1CCN(C(c2cccc3nsnc23)=O)C(C)C1NC(=O)CN1CCOCC1 44500,c1(CCC(=O)N(C)CC2N(C(CC(C)F)=O)CCOC2)nnc(S)nc1O 44501,C1(CC(=O)O)CC2(CCOCC2)CN1Cc1cc(N)c(O)c(F)c1 44502,c1(C(N2CC(CC(C)C)C2)=O)cc(CNC(c2cnco2)=O)on1 44503,c1(N2CC3CN(C(CCCC=C)=O)CC32)ncnc2ccc(OC)cc12 44504,C1(CC(=O)OC)(SCC(=O)NC)CNC(=O)C1.C1(C(=O)O)CCN(C(C)(C)C)C1 44505,C1(NC(C(=O)NCc2ccc(OCCCCOC)cc2)=O)CCC2OCCC2C1 44506,N1(C(=O)CCN2CCOCC2)CCc2[nH]nc(C(N3CCC(Br)C3)=O)c2C1 44507,c1(C(=O)NC2CN(C(c3cc(SC)oc3)=O)C(C)CC2)ccc(P(C)(C)=O)cc1 44508,N1(C(=O)COC2CCCC2)CC(NC(C23CC(CN2C2CC2)C3)=O)CC(O)C1 44509,c1(C(=O)NCC2C(NC(C(C)SC(C)C)=O)C2)cc(C(F)(F)F)ncc1Cl 44510,C12(NC(c3cc(C)n(C4CC4)n3)=O)CCC1CN(C(C1CC(=O)N(C)C1)=O)C2 44511,N1(C(c2c(CC)csc2)=O)CC2CC(C(=O)NCCN3CCOC3=O)CC2C1 44512,c1(C(N2CCC(O)C2C(N2CCC2CO)=O)=O)cccc(Cl)c1F 44513,CC1CCCC(N(C)C(C2CC3(CC(NC(=O)Cn4ccnn4)C3)C2)=O)C1C 44514,C(c1cc(C)c(C)cc1C)=CC(=O)NCC(c1cccc(C)c1)NC(=O)CO 44515,C1(OC)CN(C(=NCCc2sccc2C)NCc2ccco2)CC1O 44516,C1(C(=O)NCCCNC(C(C)C)=O)CC(C)N1C(=O)C=Cc1ccoc1 44517,O=S(=O)(c1cccc2cccnc12)NC1C2CCC1CN(Cc1cnc[nH]1)C2 44518,c1(CC(=O)NC(CNC(c2ccc(C3CC3)o2)=O)C2CCC2)ccc(F)cc1Cl 44519,N1(C(C(CC)N(C)C)=O)CC2C(NC(=O)Cc3ccco3)CS(=O)(=O)C2C1 44520,C1(NC(C2SCCCS2)=O)CCC12CN(C(=O)CCn1cnnn1)C2 44521,c1(C(=O)OC)ccc(O)nc1NC(C)CC(C)NC(C1CCS(=O)(=O)C1)=O 44522,c1(NC(CNC(c2ccc(COC)s2)=O)C)ncc(Br)cc1C#N 44523,c1(CNC(C)=O)c(C)n[nH]c1C(O)CNC(=O)CCC(=O)c1ccc(C)s1 44524,C1(C(=O)NC(C(C)NC(c2ccnnc2)=O)CO)CCCC2(CCCCC2)C1 44525,c1(NC(=O)Nc2c(C)cc(Br)cc2F)c(C#N)oc2ccccc12 44526,N1(C(c2cc(C)nnc2)=O)CCC(NC(=O)CC(C2CC2)C2CC2)CC(C)(C)C1 44527,N1(C(C(=O)NC)=O)CCC(NC(c2cnn(-c3cccc(C)c3)n2)=O)C(C)(C)C1 44528,C1(C(=O)NCc2ncco2)(CC)CCCN1C(=O)CCN(C)C 44529,N1(C(CCC(=O)NCCC)=O)CC2CCCN(C(=O)C=CCOC)C2C1 44530,C1(N(C)C(C2(CCNC(C3(C)CC(F)C3)=O)CC2)=O)CCCC1(F)F 44531,Cc1cnc2ccc(C(=O)NC3CCN(C(=O)CCS(C)(=O)=O)C3)cn12 44532,S(=O)(=O)(c1cnn(-c2ccccc2)c1)N(C1CC2CCC(C1)N2)C(c1ncon1)=O 44533,Cc1ncncc1C(N1CCC(N2CCN(C(C3CCCCN3C)=O)CC2)C1)=O 44534,c1(C(N2CC(CN(C(C3ON=C(C)C3)=O)C)OCC2)=O)cccc2ncc(C)n12 44535,N1(C(CC2CCC(=O)N2)=O)CC2(CCCC2NC(c2cccc(C3CC3)c2)=O)C1 44536,c1(C(N(CC(CC)NC(c2ncc(OCC)nc2)=O)C)=O)c[nH]c2nccc-2c1 44537,C1(CNC(C(CCC)OC)=O)CC2(CO1)CN(C(=O)CC(F)(F)C(C)C)C2 44538,c1(C(=O)NC2C(CNC(c3ccc(C#C)cc3)=O)COC2)cc2cn[nH]c2cn1 44539,C12(NC(N(C)CC3CC=CCC3)=O)CC(NC(=O)OC(C)(C)C)CC1C2 44540,c1(CC)ncnc(N2CC(NC(=O)C(O)CCSC)C2)c1F 44541,CC(C(=O)NCC(c1ccccc1)N(C)C(c1cc(Cl)ccc1Cl)=O)P(C)(C)=O 44542,N1(C(c2ccn(CCOC)n2)=O)C2CC1CN(C(c1ccc(F)cc1I)=O)C2 44543,C1(C)(CC)CCN(C(C2CC2C2CN(C(C3(C)CCCN3C)=O)C2)=O)CC1 44544,N1(c2nc(CC)nc(=N)[nH]2)C2CCCC1CN(C(=O)C=C1CCCC1)C2 44545,c1(C(C(=O)NCC(CNC(c2cc(Cl)ccn2)=O)OC)=O)ccc(Cl)cc1 44546,Cc1cnn(CC(N2CCC3C(NC(=O)CN(C(=O)C(C)C)C)C3C2)=O)c(=O)c1 44547,c1(C(N2CCN(C(COCC=C)=O)C(CO)C2)=O)cnn2cccc(Cl)c12 44548,c1(C(=O)NCC2(CNC(=O)CC(F)F)CCCC2)ccc(O)cc1F 44549,C(C)(C(=O)N(CCNC(C)=O)CC)NC(CC)=O.C12CC(C1)CC(=O)N2 44550,c1(CC)cc(C(N2CCC(CN(C(=O)CC3(C)CC3(F)F)C)CC2)=O)cc(O)n1 44551,C1(N(C)C(c2cnc(Cl)n2C)=O)CCC(C)(C)C1.C12CC(C1)NC(=O)CO2 44552,N1(C(c2ccc(CC)cn2)=O)CCCCC(CCC(=O)NCCC(=O)NC)C1 44553,Cc1ncn(C)c(=O)c1C(=O)NCC1C(C)CCN1C(=O)C(F)=C1CCC1 44554,C1(C(F)F)(CNC(c2csc(CO)n2)=O)CCN(C(C2CC3(CC3)CO2)=O)C1 44555,c1(C(N2C(C)(CC(=O)N(C3CCOC3)C)CC2)=O)cnc(=N)[nH]c1 44556,CCC(C)C(C(=O)NOCc1nc[nH]n1)N(C)C(c1ncc(F)cc1N)=O 44557,C1(CCNC(=O)C(COC)N(C)C)(NC(COCCC)=O)CCCC1 44558,C12(CC)CC(CN)(CO1)C2.C1(C)CCCC1C(=O)NC1CC(C(=O)OCC)C1.OCC 44559,C1(C(=O)NCC2CC(NC(=O)CC3CCCC34CC4)C2)CC2(C1)CC1(CC1)C2 44560,N1(c2n(CCOCCC=C)c(-c3cn(C)nn3)nn2)CC(C)C(F)(F)C1 44561,c1(C(=O)NCC2CC(CC)C2)cc(CNC(c2cccnc2O)=O)ccn1 44562,Cc1cncc(C(=O)N(C)CCOCCCNC(C2CCC(N(C)C)CC2)=O)c1 44563,C(CN=c1cc(C(N)=O)nc[nH]1)(c1ccccc1)N(C)Cc1n[nH]c2c1CCC2 44564,c1(C(=O)OC)ccnc(C(N2CCC(O)(CN(C)C)C2)=O)c1.C12(CC1)CC2 44565,C1(C(N(CCN(C)C(c2cccnc2)=O)C)=O)CCCC2CCCN12 44566,c1(-c2n(C3CCN(C)CC3)nc(-c3ccc(F)cc3)n2)cn(C)ccc1=O 44567,N1(C(C(CC)F)=O)CCC(C2CCCN(C(=O)C=C3CCC(C)C3)C2)C1 44568,CC1CN(C(c2cn(C)[nH]c2=N)=O)CCN(C(=O)C(O)C(F)(F)F)C1 44569,c1(CN2C(CNC(C3CC4CC3C3CC43)=O)CCC2)ccc2nonc2c1 44570,C1(NC(c2cnn(CCC)c2C)=O)CC(C)CN(C(=O)CC2CCCC2(F)F)C1 44571,N1(C(C2(CC)CC2)=O)CCC2(CC1)CC2NC(=O)C(c1cc(C)cc(F)c1)C 44572,c1(SCC)ccc(Cl)cc1C(=O)NCCCN(C(C1(O)CCCC1)=O)CC 44573,C(=O)(CCS(=O)(=O)CC(C)C)N1CCCC(O)(CNC(C(CCC)OCC)=O)C1 44574,Cc1cccc(C(N2CCC(CN(C)C(C3CCS(=O)(=O)C3)=O)C2)=O)c1Cl 44575,c1(C(N2C(C(=O)O)CC(NCCCCS(C)=O)C2)=O)cccc2c1OCCO2 44576,C1(O)(CCNC(CSC(C)(C)C)=O)CN(C(C2CC(n3ccnn3)C2)=O)C1 44577,c1(C(=O)NCC(COC)(F)F)coc2c1CN(C(c1sc(C)nc1C)=O)C2 44578,C1(C(C(=O)NCC2CCN2C(c2cnc(C)cn2)=O)OC)CCC(F)(F)CC1 44579,N1(C(c2cccc(OC)n2)=O)CCc2ccc(C(=O)NCCCC(C)C)nc2C1 44580,CCC(CC)CCCC(=O)N1CC2CC2(NC(=O)Cc2nc(F)c(F)cc2F)C1 44581,c1(OC(COC)C(=O)N2CC(c3ccccc3F)(C)C2)cc(F)cc(F)c1 44582,C(=O)(C(CCOCC)NC(=O)CC1CCOC1=O)NCCOCC#C 44583,c1(C(=O)NC2C3CN(C(CSCCCC)=O)CC32)ncc([N+](=O)[O-])cc1C 44584,N1(C(C(CN(C)C)O)=O)CCC(NC(=O)CCc2cn[nH]c2)C2(CCC2)C1 44585,CC1COCC(CC(N2CCC(CN(C)C(c3cc(F)n[nH]3)=O)CC2)=O)O1 44586,c1(C(=O)Nc2cncc(C(N3CCC(CC(=O)OC)C3)=O)c2)cc(Cl)ncc1I 44587,c1(OCC)cc(N2CCN(C(C3CC(C(C)(C)C)C3)=O)C(C)C2)nc(C)n1 44588,c1(SC)nc(C)c(CCC(=O)N(C2CCN(C(=O)C(C)C#N)C2)C(C)C)c(O)n1 44589,c1(C(N2CC(O)(C(C)NC(c3cc(CC)c(C)s3)=O)C2)=O)cc2ncccc2o1 44590,C(=O)(CCS(=O)(=O)NCC)NC1C(NC(C2N(CCC)CCCC2)=O)CCC1 44591,Cc1cc(Br)cc(C(=O)NC(C2CCCN(c3ccnc(Br)n3)C2)C)c1C 44592,C1(NCC(COCCOC)O)CCN(Cc2nnnn2-c2ccco2)CC1.OC 44593,N1(C(c2ccc(CC)s2)=O)CC2(CCCC2)C1C(N1CCCC(F)CC1)=O 44594,C1(CNC(=O)Cc2cccnc2)CC2(CO1)CN(C(c1cccc(CO)n1)=O)C2 44595,C(=O)(C(C)(C)C(F)F)NCC1C(NC(CC(C)N(C)C(=O)OC(C)(C)C)=O)CC1 44596,CCC(C)(COC(c1nc(C)ncc1Cl)=O)C(=O)Nc1ncccc1C#N 44597,C1(N(C2CCCCCC2)C(C)=O)CCCN(CC2CCC2)CC1 44598,C1(C(=O)NC(CCC)CCCNC(=O)C(C)(C)CN(C)C)CC(C(C)(C)C)=NO1 44599,C1(CC(=O)NCC(C)(C)NC(C(C)C2CC2)=O)COC(C)(C)C1 44600,N1(C(C)=O)CCN(C(=O)NC(c2ccc(C)cn2)C)CC1CO 44601,C12(C(N3CC(CNC(C4(C=C)CCCCC4)=O)C(C)C3)=O)C3CC(CC13)C2(F)F 44602,Cc1nccc(Cl)c1C(=O)NC1CN(C(C23CCC(C(F)F)(CC2)C3)=O)CC1O 44603,c1(C(N2CCCC(NC(C3C(C)CC(C)O3)=O)CC2)=O)ccc(F)c(Cl)c1F 44604,CC1CC(NC(=O)CN2CCCNC2=O)CCN1C(C1CC(=O)N(C)C1)=O 44605,CC1(C)OCC(CC(C(=O)Nc2cccc(C(N)=O)c2)N2CCC(CC3CC3)C2)O1 44606,N1(C(CCC(=O)NCC)=O)CCC(NC(=O)C(c2cn(C)nc2C)O)C(C)(C)C1 44607,N1(C(c2cnc(CC)o2)=O)CCC=CC1C(=O)NCC(C#N)CC 44608,C(=O)(C1=CCC2CCC1N2C(=O)C(C#N)C(C)(C)C)NCC(C)CCO 44609,N1(C(C)C(=O)Nc2cc([N+](=O)[O-])ccc2F)CC(C)OC2(CCCCC2)C1 44610,C(=O)(CCCN=[N+]=[N-])NCC(C)(O)CNC(C1CCCN1S(C)(=O)=O)=O 44611,Cc1cc(Br)c(F)cc1NC(c1cncc(C(F)(F)CF)c1)=O 44612,c1(OCC(=O)NC(C)CC2CCC(=O)N2)ccc(Cc2ccccc2F)cc1 44613,C1(CCNC(CCC=C)=O)CCCN(C(=O)CC2(NC(C)=O)CCCCC2)CC1 44614,C#CCCCCC(=O)NC(C)(C)CN(C)C(c1nc(OC)cc(C(F)(F)F)n1)=O 44615,C(C#CC(=O)N(CCCCO)CC)NC(C1C(=C)C1)=O 44616,CC12CC(C(N3CCC(NC(C4CC4(C)Br)=O)C(F)C3)=O)(C1)C(C)(C)O2 44617,C(=O)(C(O)C(C)CC)N(C(CNC(C=CC(=O)OCCCC)=O)C1CC1)C 44618,C(=O)(C1=NN(C)C(=O)CC1)NCCc1cc(C(N(C2(C)CC2)C)=O)no1 44619,C1(C(=O)NCC2(O)CCN(C(c3ccc(CC)s3)=O)CC2)CN2CCC1(C)CC2 44620,C(=O)(C1=NOC(C)C1C)NC1CC(OC)CN(C(c2n(CC)ccc2)=O)C1 44621,c1(NC(=O)NC2CCC(C(=O)OC)C2)ccc(OC(C)(C)C)cc1 44622,C1(NC(c2cnc(OC)s2)=O)CCC(C)N(C(=O)CC2CCS(=O)(=O)CC2)C1 44623,C(=O)(C#CC(C)(C)C)N1CCC(N(C(c2c(OC)nsc2)=O)C)CC1 44624,C(C)(CC)(CCNC(=O)CC1CCCCC1C)NC(c1c(CC)con1)=O 44625,c1(CCC(N2CCC(CNC(CSCCC)=O)C2)=O)ccccc1F 44626,O(NC(=O)C(F)(F)C(C)(C)O)C(CC(C)C)C(N1CC2CC=CCC2C1)=O 44627,C(N=c1cc(C)nc(NCc2occc2C)[nH]1)C1(COC)CCC1 44628,c1(C(=O)NCC(CNC(C(C(C)OC)N(C)C)=O)CO)cc(C#N)cn1C 44629,N1(C(c2cccc(SCCC)c2)=O)CCN(C(=O)C(C)COC)C(CC)C1 44630,Cc1cc(Cl)ncc1NC(C1CCCCN1C(=O)Cn1cccn1)=O 44631,CCCCCC(=O)N1CC(O)CC1CNC(=O)CC(O)Cc1ccccc1 44632,CCC(C)(C)CCCC(=O)N(C)CCOCCNC(C1CCC2CC1C2(C)C)=O 44633,c1(C(=O)NCC2C(NC(c3c[nH]cc3Br)=O)CCC2)cc2nn[nH]c2cc1F 44634,Cc1ccc(N2CCC(N3CCC(SCCNC(=O)CCC(N)=O)C3)C2=O)cc1 44635,N#Cc1cc(-c2ccc(CNC(c3ccc(OC(F)F)cc3F)=O)cn2)cc(F)c1 44636,C1(CC(=O)NC)CN(C(c2cc[nH]c2C)=O)CCN1C(=O)C=Cc1cccnc1 44637,C1(SC)CCN(c2nnc(-c3ccsc3S(C)(=O)=O)n2C)CC1(C)C 44638,c1(OCC)ccc(C(=O)NCC(C)CN(C(=O)C(C)OCCC(C)C)C)cc1C 44639,C1(CC(=O)N(CC(CNC(C2(C(=O)OCC)CCC2)=O)O)C)C(C=CC)C1(C)C 44640,C(C)(C(C(=O)NCc1cc(O)ns1)NC(c1nonc1C)=O)OC 44641,c1(C(=O)NCC2(F)COCCN(C(C(CC)(C)O)=O)C2)cccc2nc(O)[nH]c12 44642,c1(C(=O)NC2C(CNC(CCCOC)=O)COC2)nccnc1C(N)=O 44643,C(=O)(C(=O)C(F)(F)F)NC1C(C)(C)C1CO 44644,N(C1CCCc2n[nH]cc21)C(C1CC(CNC(COC(C)C)=O)OC1)=O 44645,c1(C(=O)OC)ccnc(C(=O)NC2CN(C(=O)Cc3ccnc(Br)c3)C2)c1 44646,c1(C(N2CCN(C(C3CC(C)C3)=O)CC2CO)=O)cncc(S(N)(=O)=O)c1 44647,c1(CC)cc(NC(=O)C(CNC(c2cnc(C)s2)=O)OC)cc(O)c1 44648,C1(CNC(CC)=O)CCN(C(=O)Cc2csc(NC(=O)C(C)C)n2)CC1 44649,C(=O)(C1Cc2ccccc21)N1CCC(C)(NC(c2c(C)nc(CC)s2)=O)CC1 44650,c1(SC)ccc(C(=O)NC2CC2CNC(C2CC(C)(O)C2)=O)cc1 44651,C1(C(N2CC(C)(C(F)(F)F)C2)=O)CCCN(C(=O)C(F)OC(F)(F)F)CC1 44652,c1(C(=O)NCCC2N(C(CCOCC(C)C)=O)CCC2)ccc(NCCO)cc1 44653,CC1(C)OCCc2cc(C(N3CCS(=O)(=O)C4CCCCC34)=O)ccc21 44654,C1(C(N(CCCC)CCCO)=O)CCCCN1C(C1CCC2CC12)=O 44655,C1(C)(NC(CC(C)c2cccnc2)=O)CCCN(C(c2cnc(O)n2C)=O)C1 44656,C(=O)(C(C)(C)CC(C)C)NCC1(OC)CCN(C(C2(C)CC2C(F)(F)F)=O)CC1 44657,n1(C(C)C)ncc(Cl)c1C(=O)NC1CCC(C)(CN)C1 44658,c1(OC)c(C(=O)NCC2(F)CC(CNC(=O)C3=CCCC3C)C2)cc(Cl)cc1Cl 44659,Cc1nc(C)c(C(N2CCC(C)(CNC(c3scnc3C3CC3)=O)C2)=O)[nH]1 44660,N1(C(C(C(C)C)SCC)=O)CCN(C(C2CC(C)CCO2)=O)CC1CC(F)F 44661,Cc1cc(C(N2CC=CC(NC(C3(C(N)=O)CC3)=O)C2)=O)c2c(c1)CCC2 44662,C12(C(=O)NC3CC(C(F)C(=O)NCCCN4CCCC4=O)C3)CCC(CC1=O)C2 44663,N1(C(c2cc(-c3ccccc3)no2)C(=O)NCC)CCC(n2cc(Br)cn2)CC1 44664,C(=O)(C1=CC(O)C(NC(=O)C2=CCCCCC2)C1)NCC1CCN(C(C)=O)C1 44665,C1(C(=O)NCCNC(=O)Cc2ccsn2)Cc2ccccc2C(=O)O1 44666,N1(C(c2cn(CCN(C)C)nn2)=O)CC(C2CN(C(C3(O)CC(C)(C)C3)=O)C2)C1 44667,C1(NC(Cc2cc(OC)no2)=O)CCCCN(c2nnc(-c3ccon3)s2)C1 44668,n1(CC(=O)NC2(C)CC(NC(c3n[nH]cc3Cl)=O)C2)ccc2ccc(F)cc12 44669,C12(NC(c3ccc(CC)nc3)=O)CC(CNC(=O)Cc3[nH]cnc3C)(C1)OC2C 44670,CN1CC(O)CC1(C)C(=O)NCC1COCCN(CC=Cc2ccccc2)C1 44671,N1(C(C2(C)CCCCO2)=O)CCN(C(=O)CNC(c2ccncc2)=O)C(CO)C1 44672,c1(C(C(=O)NC(C)C)NC(c2c(C)n(C3CC3)nc2)=O)ccc2c(c1)C=CCC2 44673,N1(C(Cc2n(C(C)C)cnn2)=O)CC2C(CNC(=O)CC3CCN(C)CC3)C2C1 44674,C1(C(C(=O)NCCC(=C)C)F)CCN(C(=O)C=CCCC)C1 44675,CC(C)(C)C(CO)C(=O)NC1CCC(NC(c2ccc(F)o2)=O)CC1 44676,C(C(CNC(=O)CCc1ccccn1)S(C)(=O)=O)NC(C(C=C)C)=O 44677,C1(NC(C2CCCC(F)C2)=O)CCN(c2nccc(CO)n2)C12CCC2 44678,C#Cc1ccccc1NC(=O)C(CCC=C)NC(=O)CC(C)C(F)F 44679,C(CCCCC(=O)N(C)CCC1CCCN1C)NC(C1CC(C(C)C)C1)=O 44680,Cc1cc(C(N2CC(NC(C3(C)C=CCC3)=O)C(C)(C)C2)=O)ncc1C(F)F 44681,N1(C(c2c(OC)nsc2)=O)CC(C(=O)NCCC2CCN(C)C2)CC12CCC2 44682,C1(O)(C(N2CCC(C)(c3cn(CCCCF)nn3)C2)=O)CN2CCC1CC2 44683,C1(CNC(C(CCN(C)C)O)=O)CCN(C(c2cn3c(n2)CCC3)=O)CC1O 44684,N1(C(c2nnn(C)c2C(F)F)=O)CCCC2(C1)CN(C(c1csc(C(F)F)n1)=O)C2 44685,C(=O)(CC(C)(C)CNC(C1CC(F)(F)C1)=O)NCC(C)(C)C(F)F 44686,C(CC(=O)NCc1ccc(F)nc1C)(C(C)(C)C)NC(C1CCCN(CC)C1)=O 44687,Cc1cc(S(N)(=O)=O)oc1C(N1CCN(C(=O)COC2CCOC2)C(C)C1)=O 44688,CC1CC(C)(C)CCC1NC(=O)C(=O)Nc1cccc(CN2CCOCC2)c1 44689,C(=O)(C(C)(O)C1CCC1)NCC(C)CN(C)C(C1(Br)CC1)=O 44690,N1(C(CC2(OC)CCC2)=O)CCCCC1C(=O)NC1CC(C)(O)C1 44691,C1(NC(CCc2nnc(C)n2C)=O)CCCC(NC(c2cc(Cl)n(C)n2)=O)CC1 44692,CC1(C(=O)NCC#CC(=O)NCCCC2CCOC2)CCC(=O)C1 44693,N1(C(COc2cc(C)c(F)cc2)=O)CC2CCN(C(c3csnn3)=O)CC2C1 44694,C1(N(C(c2cc(C)n(C3CC3)n2)=O)C)CN(C(=O)C(C)c2cccs2)CC12CC2 44695,c1(-n2cc(N3CCN(C(CCN(CC)CC)=O)CC3)nn2)cnnc(O)c1Br 44696,C(=O)(C(C(C)(C)C)n1cc(C(C)O)nn1)N1C(OC)C(C(=O)OCCN(C)C)C1 44697,c1(C(=O)NC2CCC(NC(C=CSC)=O)C2)c(F)cccc1Cl 44698,C1(CN(C(C2COC(=O)O2)=O)CC)CCCCN1C(C1CC(O)CN1C(C)=O)=O 44699,c1(C(N2CC(C(=O)NC3(C(=O)OC)CC(O)C3)C2)=O)cc(S(N)(=O)=O)sc1Cl 44700,C1(C(=O)NCC(CN(C(C2CCCC(F)C2)=O)CC)(C)C)CC2(CSC2)C1 44701,N1(C(C=CC(C)(C)SC)=O)CCCC12CCN(C(C1CCN(CC(C)C)C1)=O)C2 44702,N1(C(C2CC(OC)C2)=O)CCN(C(c2ccc(SC)s2)=O)C(C)CC1C 44703,C=C(C)CCCC(=O)NC1(CNC(c2cc(F)ncc2OC)=O)CCCCCC1 44704,Cc1cc([N+](=O)[O-])cc(C(=O)NC2CN(C(=O)C3=COCCO3)CCC2F)c1Cl 44705,C(=O)(C1=CCCSC1)NC1(COC)CCN(C(=O)CC2CC23CC3)C1 44706,c1(C(=O)NCc2c(C3CN(C(c4c(C)n[nH]c4)=O)C3)ocn2)coc(C#N)c1 44707,C(=O)(C#CC(C)(C)CNC(c1cnn(C(C)C)n1)=O)NC(C#C)CC1CC1 44708,c1(CNC(N2CCC(c3ccc(OCC)cc3)CC2)=O)ccc(OC)nc1C 44709,C(=O)(C(C)(C=C)CC)NCCC(=O)NC(CC=C)C(=O)OCC 44710,c1(C(N2C(C)CC(CNC(C3CN(c4nnnn4C)C3)=O)C2)=O)ncc(Cl)cc1F 44711,C=C1COc2c(C(=O)NCCC(C)NC(C3(Br)CC3)=O)cnn2C1 44712,C1(C(N(CC(CN(C(CN(C(C)=O)C)=O)C)O)C)=O)CCCCCN1C 44713,CC1COc2ccc(C(N3CCCCC(CNC(c4ccnnc4)=O)C3)=O)cc21 44714,C1(CC(=O)NC2(CC)CCCCC2)CCCN(C(=O)C(O)C2CC2)CC1 44715,C1(COC)(NC(C2C=CC=CC=C2)=O)CCN(C(=O)CCc2cn(C)nc2C)C1 44716,c1(C(N2C(C(N(C3(C)CCCC3)C(C)C)=O)CCC2)=O)ccc(Br)c2cccnc12 44717,C1(CC#C)(C(=O)NCC(O)CNC(c2conc2C2CCCC2)=O)CCCCO1 44718,Cc1cc(=NC(C)c2ccc(Cl)c(F)c2)[nH]c(=NCCOCCCO)[nH]1 44719,c1(CC(=O)NCCC(CNC(C=C(C)C(C)C)=O)O)csc2c(F)cccc12 44720,c1(OC)cccc(C(=O)NCC2(F)CCN(C(=O)CC3C=CCC3)C2)c1F 44721,N1(C(CC(=O)OC(C)(C)C)=O)CCCC12CCCN(C(=O)C(F)(F)C1CC1)CC2 44722,c1(OC(CC)C)cc(CN2CCC(C(=O)N(C)C(C)C)CC2)ccc1OC 44723,C(=O)(C1CCCc2nncn21)N1CCC(C)(N(C(C2CCCC(F)(F)C2)=O)CC)C1 44724,Cc1c(CC(=O)NC(C)(C)CNC(=O)C=Cc2cnccn2)ccc(Cl)c1Cl 44725,C#Cc1ccc(C(=O)NC(C)CCNC(C2CC(CC(C)(C)C)C2)=O)cc1C 44726,Cn1cc(C(C(=O)NC2CCC2(C)C)NC(=O)C(F)C2CCCC2)nn1 44727,CS(=O)(=O)c1cccc(C(N2CCCC2CCCNC(C2CCC3CC23)=O)=O)c1 44728,C1(CC(=O)NC(CN(C(=O)CNC(c2ccc(C)s2)=O)CC)C)CC2CC1C2 44729,N1(CC#C)CCC2(CC1)CC2(C)C(=O)NC(c1cccc(Cl)c1)C 44730,c1(OC)cc(CCC(N2CC(NC(=O)C(N)=O)C(O)C2)=O)ccc1Cl 44731,Cc1cnc2nc(C(=O)NC3(C)CCN(C(c4cc(C)nnc4O)=O)C3)nn2c1 44732,Cc1cc(C)nc(SCC(=O)NC(C)CCCNC(C2(F)CC=CCC2)=O)n1 44733,C=CC1CN(C(C2CC3(CCC3)C2)=O)CC1NC(c1cn(CC)nc1C)=O 44734,C1(C(N(CC(C)C#N)C2CC2)=O)CCN(C(c2ccco2)=O)CC1 44735,n1(CC)cc([N+](=O)[O-])c(C(=O)N(CC(C)NC(=O)Cc2cc(C)cs2)C)n1 44736,C1(NC(C(C)SCC)=O)CN(C(c2cnn(CC3CCC3)c2)=O)CCC1F 44737,C#CCC(C)(C(=O)NC(c1nn(C)cc1O)C)NC(=O)C(C)=CC 44738,c1(N2CC(C)(NC(C3(c4ccccc4)C(C)(C)C3)=O)C2)nnccc1C#N 44739,Cc1ccc(C(F)CC2CCN(C(=O)C(=O)NCCC3CCC3)CC2)cc1C 44740,CN1C(=O)NCC1C(=O)NCCOCCNC(C1OC2CCC1C2)=O 44741,N1(C(C(C2CC(NC(C(CC)=CC)=O)C2)F)=O)CCN(CCO)C(C)C1 44742,C1(C)(CCNC(C2CCC(C)O2)=O)CCN(C(c2cnccc2Cl)=O)CC1 44743,c1(CS(N2CCC(n3c(C)ccc3C)CC2)(=O)=O)c(Br)ccc(F)c1F 44744,C(CCO)(CC(C)C)NC(c1cc(CNC(c2cc(COC)no2)=O)nn1C)=O 44745,C1(NC(Cc2nc(C)on2)=O)CCC(CNC(=O)CCc2ccc(O)cc2)CC1 44746,C(CCS(=O)(=O)C(C)(C)C)NC(=O)NC(c1cccs1)CC 44747,c1(C(N2C(C)C(NC(C3CCC=CO3)=O)CCC2)=O)cc2ccccc2s1 44748,CCC1=C(C(=O)NC2CN(C(=O)CCC3(C#N)CCC3)CC(C)(C)C2)CCCO1 44749,C1(C(=O)NCC(C)(C)CCNC(=O)C(O)C(F)(F)F)CCCC2(CCC2)O1 44750,C#CCCCC(C)C(=O)N1CCCC1(CNC(c1sccc1OC)=O)COC 44751,C(C(C)(F)C(C)(C)F)NC(C1CC(C)N1C(c1ncccc1O)=O)=O 44752,C(=O)(CC(Cc1cccc(F)c1)NCc1cnc(-c2ccco2)s1)OC 44753,c1(OC)cc(CCNC(=O)C(c2ccc(Cl)c(F)c2)O)cc(Br)c1 44754,c1(C(N2C(C)C(NC(c3csc4cncn34)=O)CCC2)=O)cccc2oncc12 44755,S(=O)(=O)(c1ccc(C#N)c(N2CCCC(C)(F)C2)c1)N(CC(C1CCC1)OC)C 44756,Cc1cc(C(=O)NCC2CCN2C(C2C3CCC(F)(F)C23)=O)ncc1Br 44757,N1(C(C2CNC(=O)N2)=O)CC2CCCC1C2c1cn(Cc2c(F)cccc2Cl)nn1 44758,Cc1ccc(F)c(N)c1C(N1CCN(C(=O)CC2CC3(CCC3)CO2)C(C)C1)=O 44759,C(C(=O)N1CC(O)CC1CC(=O)NC1CC(CO)C2CC12)(C(C)C)SCC 44760,N1(C(C(CSC)O)=O)Cc2ccnn2CC(NC(c2cc3ncccc3o2)=O)C1 44761,N1(C(=O)NC2C(OC)(OC)CC2)CCN(C(=O)CCC(C)C)CC1c1cn[nH]c1 44762,N1(CC(=O)OC(=O)C(F)(F)F)CC2(CCC2)CC1C(F)(F)F.CC1(C)C(=O)N1 44763,C(C(CO)C(F)(F)F)NC(c1sc(Cl)cc1Br)c1n(CCOC)nnn1 44764,N1(C(=O)COCC2CCC2)CCOCC1CNC(C1(CO)CCCO1)=O 44765,N1(C(c2c(C)nsc2)=O)CCCC(C)C1CNC(=O)CCc1ccn(C)c1 44766,N1(C(C(C2CC2)OC)=O)CCC(O)(CN(C(=O)C(C)CC(F)F)C)CC1 44767,Cc1c(C(N2CCCCC2C(=O)NCc2cnccn2)=O)ccc2c1OCO2 44768,C12(C(N3CC=CC(NC(C=CC4N(C)CCC4)=O)C3)=O)CCCCC1CCC2 44769,c1(C(N2C(CC(=O)NCCCCOC)CCCC2)=O)cccn2ccnc12 44770,C(=O)(C1CCCc2c[nH]nc21)NC1C(CNC(CSCC(C)C)=O)COC1 44771,C1(NC(C(=O)NCCOC)=O)C=CCN(C(=O)C(O)Cc2ccc(OC)cc2)C1 44772,N1(C(CC(=O)OCC)=O)CC(NC(c2ccc(C(C)=O)o2)=O)CC2(CCC2)C1 44773,C1(NC(c2c(C)nn[nH]2)=O)CN(C(=O)CCN(C)C)CCC1F 44774,Cc1nnc2n1CCC(NC(C1CC(=O)OC1c1cccc([N+](=O)[O-])c1)=O)C2 44775,Cc1ccc(-n2nnc(C(=O)NCC3(F)CN(C(C4CSC4)=O)C3)c2C)cc1 44776,C1(CNC(c2n(C=C)ncc2)=O)CC(C)(C)CN1C(c1cc(C#N)oc1C)=O 44777,C1(N(CCNC(c2ccccc2)C)C(C2(C(=O)OCC)CC2)=O)CCCCC1 44778,C#CC1CN(C(c2sc(Br)cc2C)C(=O)NC(C)(C)CC)CC1O 44779,CC1CN(C(=O)C=Cc2cccnc2)CC(C)N(C(=O)COc2ccccn2)C1 44780,N1(C(C(C=CC)O)=O)CCC=C(C(=O)NC2CCCCCC2)C1 44781,c1(C(=O)NCC2(CNC(C3(C#N)CC3)=O)CCCCC2)ccc2nnn(O)c2c1 44782,N1(C(c2ccc(OC)s2)=O)CC2(CNC(c3snnc3C)=O)CCC1CC2 44783,c1(NC2C(NC(c3c(C)cc(C)o3)=O)CS(=O)(=O)C2)ncc(S(C)(=O)=O)cc1Cl 44784,C(C(=O)NCCC1CCN(C(=O)C(CC)N(C)C)C1)(C(C)C)NC(COC)=O 44785,C=CCC(F)(F)C(=O)N1CCCC1CN(C(=O)Cc1ncoc1C)C 44786,Cc1cc(C(C)NC(N2CCCC2C2CCCOC2)=O)cc(C)c1 44787,N1(Cc2c(C)nncc2)CC2CC1CN2C(=O)CC(=O)N(C)C 44788,C1(NC(c2ccc(CC)s2)=O)CCN(C(C2CC(N(C)CC)C2)=O)CC1CC 44789,c1(C(N2CCN(C(C(CCC)=CCC)=O)CC2C2CC2)=O)ccc(C#N)cc1C 44790,O=C(C1=CC2CC=CCC12)NCC=CCNC(C1(O)CC(F)(F)C1)=O 44791,C1(F)(CNC(C(CSC)O)=O)CCCN(C(c2cccc(C(C)=O)c2)=O)C1 44792,C1(C(=O)OC)COC2(CCN(C(=O)C(O)C(F)(F)c3ccccc3)CC2)C1 44793,c1(C(N2C(C(=O)Nc3c(C#N)cc(Cl)cc3)CCCC2)=O)cc2cc[nH]c2cn1 44794,CC1CCC(NC(c2cnnn2C)=O)CN1C(c1ccc(Cl)c(C(F)(F)F)c1)=O 44795,N1(C(C(F)=C(C)C)=O)CCCCC2(CCN(C(c3ccn(CCO)c3C)=O)C2)C1 44796,C1(C(=O)NCCCCCNC(C(C)OCCOCC)=O)CC2CC1CC2(F)F 44797,N1(c2nc(NCCC(C)F)c3c(n2)scn3)C2CCC1c1cncnc1C2 44798,c1(C(=O)NCC(C)NC(C(C2CCCCC2)OC)=O)c(C)cc(Br)cc1C 44799,N1(C(CC2(C)CCOCC2)=O)C2CCC(C2)C1CC(=O)NCC1CN(C(N)=O)C1 44800,N(C(=NCCN(C)C)NCC1CCS(=O)(=O)N1C)C(C1(C)CCCCC1)C 44801,C1(NC(COc2cc(C)on2)=O)CN(C(=O)C(C)C2CC2)CC1C(F)(F)F 44802,CC1(C(=O)NC(CCCNC(c2cc(Cl)cs2)=O)c2ccccc2)CCC(=O)N1 44803,CC(N=[N+]=[N-])C(=O)N1CCCC1C(C)NC(C1C2CCCOC12)=O 44804,CC(C)(Cc1cnn[nH]1)C(=O)NCCCOC1CCOCC1 44805,C1(NC(C2(CC=C)CCOC2)=O)CCC(C)N(C(c2cnn(C)c2Cl)=O)C1 44806,C1(OC)CCC(NC(=O)C(CC2CC2)NC(c2csc(Cl)c2)=O)C1 44807,C1(C(=O)OC)CCN(C(=O)NCC2(C)CSCCO2)C1C 44808,C1(O)(CNC(c2cc(C(F)(F)F)cc(O)c2)=O)CCCN(C(=O)C=CBr)C1 44809,c1(OC)c(C(=O)NCC2COCCN2C(=O)C(F)n2cccn2)csc1C 44810,C(=O)(CC1=NN(C)C(=O)C1)N1CCC2(C(C(=O)NC(CCOC)C(C)C)C2)C1 44811,c1(N2CC3N(C(=O)Nc4ccccc4Br)C3C2)ncc2ccc(Br)cc2n1 44812,N1(CC2(C)CCC2)CCC(NC(=NCC2CCCO2)NC2CCCCC2)CC1 44813,N#CC1(C(=O)NC2CCCC2NC(=O)C2=CCCSC2)CC12CCCC2 44814,c1(OCC(=O)OC)ccc(S(=O)(=O)NC(C)(C)CCC(=O)O)cc1OC 44815,n1(CC)cc(Br)c(CC(=O)NCCNC(=O)Cc2cncs2)n1 44816,CC(C)(C)CC(CO)NC(=O)CCCNC(=O)CC1CC(C2CC2)C1 44817,c1(CC(C)NC(C)C(c2ccccc2F)O)ccc(C(F)(F)F)cc1[N+](=O)[O-] 44818,C1(C(C)C)CCCN(Cc2cn(-c3ccc(Cl)cn3)nn2)C1 44819,Cc1ccc(S(C)(=O)=O)cc1C(=O)NCCCCC(C)NC(=O)C(C)C1CCC1 44820,c1(NC(C2CC(NCc3cc(C(=O)O)cc(Br)c3)C2)=O)nccc(Cl)c1Cl 44821,O=C(CCS(=O)(=O)Cc1ccccn1)NCC1CC(O)CN1C(=O)C=C(Cl)Cl 44822,N1(CCC)CCCC1C(=O)NCCC(=O)NCc1cc(C(=O)OC)co1 44823,c1(C(=O)NC2(CNC(C3C(C)C3C)=O)CCOC2)csc(=NC2CCCCC2)[nH]1 44824,c1(OC)cc(OC)cc(C(=O)NC(CNC(=O)CC2CC23CC3)CCOC)c1 44825,C1(C(=O)NCC#CCC)CN(C(C2CCCN2C=O)=O)CCN1C 44826,N1(C(Cc2ccc(OCC=C)cc2)=O)CCC(NC(c2cc(C)ns2)=O)C(F)C1 44827,S(=O)(=O)(c1ccc2[nH]c(=NCC(C)(C)C(F)F)sc2c1)NCc1c(OC)nsc1 44828,c1(C(=O)NC(C)CN(C(=O)Cc2c[nH]nc2O)C)ccc(O)cc1F 44829,n1(CC)c(C(=O)NC(C)C(C)NC(c2ccoc2Cl)=O)nc2ccccc12 44830,c1(C(C)N(C(c2cc(C3CC3)[nH]n2)=O)C2CC2)ccccc1F 44831,C1(CC(=O)N(C)Cc2nnc(CC)o2)CCCC(NC(c2cscc2C)=O)C1 44832,c1(C(N(C2CCN(C(C3CCCCO3)=O)C2)CC)=O)cc([N+](=O)[O-])n[nH]1 44833,C#CCC(C)(C(=O)NC1CCCC1)NC(=O)C(C)ONCCOCC1CC1 44834,c1(C(=O)OC)cccc(CC(C)C)c1.CCC1CNC(=O)N1 44835,N1(C(C(C(COC)C)C)=O)CCCC2(C1)CN(C(=O)COc1cccc(F)n1)C2 44836,c1(CC(N2CCC(CN(C(c3cn(CC)nc3C)=O)C)C2)=O)ccc(C)cc1C 44837,c1(C(N2CCCC(CCNC(CC(C)SC)=O)C2)=O)cnn2c1S(=O)(=O)NCC2 44838,c1(C(=O)NC(CNC(c2cc(C)n(-c3ccccn3)n2)=O)C)cccc(N)c1C 44839,N1(C(CC2CCC(C)(C)O2)=O)CCC(C(=O)NC2CC2)CC1(C)C 44840,C1(C(N2C(C(=O)NCCCC(C)O)CCCC2)=O)CC2CC1CC2O 44841,N(C)(S(=O)(=O)N1CC2CC(O)CC(C2)C1)CCCC 44842,N1(C(c2ncnc(C)c2C)=O)CCCC2(NC(C34CC(F)(C3)C4)=O)CC2C1 44843,N1(C(c2n(CC)ccc2)=O)CCc2cc(CNC(C3(CCO)CC3)=O)ccc2C1 44844,C1(CNC(CNS(NC)(=O)=O)=O)CN(C(c2ccc(C)nn2)=O)C2CCCCC12 44845,C(=O)(CCCC(CC)NC(=O)CCC1CCCC1)NC(C#C)(C)C1CCC1 44846,C(=O)(C#CC(C)(C)CNC(=O)C(=O)NCC(F)F)N1CC(C)OCC1 44847,N1(C(C(C)N(C)C)=O)CCCC1(C)CNC(C1CCCC2CC12)=O 44848,c1(C(=O)NC2CCC(NC(Cc3ccn(C)n3)=O)CC2)cccc(S(N)(=O)=O)c1 44849,c1(OC)ccc(-n2nnc(CNC(=O)NC3CC(C(N)=O)C3(C)C)c2C)cc1 44850,N1(C(Cc2nn(C)c(Cl)c2)=O)CCC(C2CN(C(=O)CC(=O)NC3CC3)C2)CC1 44851,C1(CNC(c2ccc(C)o2)=O)N(C(c2ccc(F)c(Cl)c2)=O)CCC1(C)C 44852,Cc1nc2nccc(C(N3CC(NC(=O)CC(O)CN(C)C)C4(CC4)C3)=O)n2n1 44853,N1(C(c2ccc(COC)o2)=O)CCCCC(CNC(c2cc3sccc3s2)=O)C1 44854,N1(C(Cc2ccn(C)n2)=O)CCC(CO)(CNC(C2CCCC23CC3)=O)CC1 44855,S(=O)(=O)(c1ccc(NCCCS(C)=O)c(C#N)c1)N(CC)CC1CC1 44856,c1(C(N(C2CCCC2)CCCNC(C(C)=C2CC2)=O)=O)cccc(C(C)(C)C)c1 44857,Cc1ccc(C(=O)NCc2nc(C(=O)N(C(C)(C)CO)C3CC3)c(C)o2)cn1 44858,c1(C(=O)NCC(C(C)C)NC(=O)C(F)C2CCCC2)cnn2cccnc12 44859,CCC(CC)C(C(=O)NCC(C(C)(C)C)NC(c1cc(O)nn1C)=O)OC 44860,CCC(C(=O)NC(C1(O)CN(C(c2cc(C)cs2)=O)C1)C)N(C)C 44861,N1(C(C2C(=C)C2)=O)CCC2(NC(=O)COc3ccccc3OCC)CC2C1 44862,CCC(CNC(=O)CNC(c1ccccn1)=O)(CC)NC(=O)C(C)C#N 44863,C(CCC(O)C(=O)N1CCCC(O)C1)NC(c1c(CC)ocn1)=O 44864,O=C(O)CC(C(=O)O)NC(=O)NCC12COC(CF)(C1)C2 44865,c1(C(=O)NC2(C)CCCN(C(C(F)=CCC)=O)C2)ccc(CCC)c([N+](=O)[O-])c1 44866,Cn1nnc(C(=O)NCCCC(C)(C)NC(C2CC3(CC3)C2)=O)c1C(F)F 44867,C(=O)(C1=CCCSC1)NCc1cncc(C(=O)NC(CCCC)CC)c1 44868,O=C1C2CC(F)(F)CCN2C(=O)N1CCCn1cc2ccccc2n1 44869,Cc1cn2c(n1)CC(C(=O)NC(C)CC1CN(C(=O)CNC=O)C1)CC2 44870,n1(CC(=O)N(C2CCN(C(CC(C)(F)F)=O)CC2)CCO)ccc(O)nc1=O 44871,c1(-n2cc(COCC3CN(C(C4CC4(Br)Br)=O)C3)nn2)cnccc1C(F)(F)F 44872,C(=O)(CCCS(N)(=O)=O)NC1(CCNC(C(c2ccc(CC)cc2)C)=O)CC1 44873,c1(C(=O)NCC(C(C)(C)C)NC(c2c(OC)cncc2)=O)n[nH]c2c1CCOC2 44874,Cn1nc(Br)cc1C(=O)NCC1(NC(C2CCC(OC(F)F)CC2)=O)CC1 44875,C1(C(C(=O)N(CCNC(c2ccc(C(C)=O)cc2)=O)C2CC2)O)CCC(C)(C)CC1 44876,CC1CN(C(c2cncn(C)c2=O)=O)CCC1N(C)C(c1ccc([N+](=O)[O-])[nH]1)=O 44877,C(C)(CCC(=O)NCCCC1(NC(=O)COCc2ncccc2Cl)CC1)OC 44878,C1(F)(CNC(CCN(C)CCO)=O)CCCN(C(C2CCCC3(CC3)C2)=O)C1 44879,N1(C(C(C)OCCCC)=O)CCCC(CCNC(C2(O)COC2)=O)C1 44880,C1(CN(C(CC2(OC)CCC2)=O)C)CN(C(=O)CC2(OC)CCC2)CC12CC2 44881,N1(C(CC2CC(C)(C)C2)=O)CCN(C(=O)CCCc2ccc(O)nn2)C2CC12 44882,N1(C(c2c(CNC(C(CCSC)O)=O)cnn2C)=O)CCN(C)C(=O)C1 44883,C(=O)(CCCC(F)(F)F)N(C)CCN(C(=O)C(C1CCCCCC1)F)C 44884,c1(CCC(=O)OCC)nc(O)c2c(C)c(C)sc2n1.C1(=O)C(C)N1C(CC)=O 44885,C1(NC(C(CC=C)NC(C)=O)=O)CC2CCC1CN2C(=O)C(C)OCC(C)C 44886,C12(CNC(CC(C(C)C)C)=O)CCC(NC(=O)COC(F)F)(CC1)CO2 44887,N1(C(C2(NC(CCCOC(C)=O)=O)CCSC2)=O)CC(CO)C(C2CC2)C1 44888,C1(CC)(NC(=O)C2=COCC2)CCCN(C(C2(C)CCCCO2)=O)C1 44889,C1(CN(C(C(C)C2CCOC2)=O)C)CCCN1C(=O)CCc1cnn[nH]1 44890,C12(CC(=O)NC3CC(N(C(C(CN(C)C)N(C)C)=O)C)C3)CCC(CC1)C2 44891,C(=O)(CC(C(C)OC)NC(c1c[nH]c(C#N)c1)=O)N(C1CCCCC1)CC 44892,N1(C(=O)Nc2nc(=N)s[nH]2)CCNCC1c1cccc(Cl)c1 44893,c1(C(C)C)ccc(CC(C)NC(=O)CCNc2ccc(-c3ccsc3)cc2)cc1 44894,N1(C(C(COC)(F)F)=O)CCCCC(NC(c2cnn(C)c2C)=O)C1 44895,N1(C(CN2CCN(C)CC2)=O)Cc2nccn2CC(NC(C2CCSCC2)=O)C1 44896,c1(C2(CC(=O)NCC(C(C)C)NC(C3C(CC)OCC3)=O)CC2)ccc(Cl)cc1 44897,C1(C(=O)Nc2cccc(CNC(C(C(=O)OC)OC)=O)c2)CCC2(CC1)CC2 44898,N1(C(C(C2CC2)OCC)=O)CCC(CC(N2CCCC2C(=O)OC)=O)C1(C)C 44899,N1(C(Cc2c(C)nc(C)s2)=O)CCCC(N(C)C(c2cnc(C3CC3)[nH]2)=O)CC1 44900,C(CCC(=O)NOCCCCC)(C(C)C)NC(CCC=CC)=O 44901,N1(C(c2ccc(CC)cc2)=O)CC(NC(=O)COCCOC)C2(CC2)C1 44902,C12(C(=O)NCCC3(O)CCN(C(c4ccc(O)nn4)=O)C3)CCCN(CCC1)C2 44903,C(CC(C(=O)N(CCO)CCN(C)C)NC(=O)CC(O)c1ccccc1)OC 44904,CCC(C)(CNC(=O)CCC1CCCCO1)C(=O)N(C)CC1(N(C)C)CCC1 44905,O=C(C1=CCOC1)NCC1CN(C(=O)COc2ccc(F)cc2)C2CC12 44906,C(=O)(CCCC(=O)C1CC1)NC(C(=O)NCCc1nnc(C)s1)Cc1ccco1 44907,c1(SC)cccnc1C(N1CCC(NC(c2cnc(O)o2)=O)CC1)=O 44908,N1(C(C(CC=CCC)C)=O)CCC2(CCC2NC(c2ccoc2C)=O)CC1 44909,N1(C(=O)OC(C)(C)C)CCCCCCC1CNC(c1cncc(OC(F)F)c1)=O 44910,C(CC1CC1)(CC(=O)NCc1noc(C(N)=O)n1)NC(c1c(C)scc1)=O 44911,CCC(C)C(C(=O)NC(CNC(C1CC(C#N)C1)=O)C1CC1)NC(=O)OC 44912,c1(C(=O)NCC23CC2CN(C(=O)Cc2nc[nH]n2)C3)cc2ccc(F)cc2[nH]1 44913,CC(CC(F)(F)F)C(=O)N(CCCCN(C(=O)C(CO)C(F)(F)F)C)C 44914,c1(OCCOCC)ccccc1C(=O)N(C)CCN(C)C(c1c(C)nsc1N)=O 44915,C1(NC(c2c(COC)scc2)=O)CCN(C(=O)CS(N)(=O)=O)CC1C 44916,c1(CC(=O)NCC2N(C(C(CC)F)=O)CC=C2)cc(C)cc(Br)c1 44917,CCC(O)C(C)(C)C(=O)NC1CC(C(=O)NCC2(CO)CCN(C)C2)CC1O 44918,C(C1CN(C(c2cncc(F)c2Cl)=O)Cc2ccccc21)NC(C(N)=O)=O 44919,c1(CC2CC(c3ccc(-n4cc(C5C(OC)C5)nn4)cc3)C2)cc(F)ccc1F 44920,N1(C(C2N(C(CCOCC)=O)CC2)=O)CCCC1CC(C)(C)C 44921,CC1CC(NC(=O)CCc2ccccc2O)CN1C(=O)C(N)=O 44922,N1(C(C2N(C(c3cc(COC)no3)=O)CC(C)C2)=O)CCC(O)C(C)C1 44923,CC1(C(=O)NC(CNC(c2ccccn2)=O)CO)CCCOC1 44924,C1(NC(=O)CCc2cncs2)CC1C1CCCN(C(c2cc(Cl)cs2)=O)C1 44925,C1(C(N(CCC(O)c2cccs2)C)=O)C(C(=O)N(C)C)C1(F)F 44926,C1(CN(C(C(c2ccccc2)SC)=O)C)CCCN1C(C1CN(C(N)=O)C1)=O 44927,N1(C(C2CC(CCNC(C#CC(C)C)=O)C2)=O)CC(C)(C)CC1CO 44928,N1(C(C2(CC)N(C(c3cc(CC)no3)=O)CCC2)=O)CCCNC(=O)CC1 44929,O=C(C1=NOC(CC2CCCC2)C1)NCC(F)CNC(c1nccs1)=O 44930,N1(C(=O)CC2CCC3CC23)CC23CCCC2(C1)CN(C(c1ccnnc1)=O)C3 44931,N1(C(CC(CNC(=O)CCC(CF)CF)OC)=O)CCCC2CNC(=O)C12 44932,C(CS(=O)(=O)CC(=O)NCC=CC(=O)NC(C)(C)CC(C)(C)C)OC 44933,CC(CC(C)(F)F)C(=O)NCC=CCNC(=O)CCCc1nncn1C 44934,c1(OC)ccc(NS(=O)(=O)NC(=O)NC2CC(F)C2)cc1 44935,C(=O)(C(C)CC1CC1)NCCCN(C(c1ncoc1C1CCC1)=O)CC 44936,C=CC(C)(C)CCN(CCc1ccnn1C)Cc1ccccc1C 44937,C1(NC(=O)C=Cc2ccc[nH]2)COC2(CNC(C3(F)CCOC3)=O)CC1C2 44938,C1(C(=O)NCc2cc(C3CCC3)no2)CCCN(C(=O)C(F)CC2CCOC2)C1 44939,Cc1ccc(C)c(C(=O)NC(C)CC(C)NC(=O)C=Cc2ccc(=N)[nH]c2)c1 44940,N1(C(c2c(C)cccn2)=O)CCCC(C2CC2NC(=O)CCC(F)F)C1 44941,N1(C(CSCC)=O)CC(CNC(=O)C(C(C)(C)C)NC(C)=O)OC2CCCC12 44942,c1(C(=O)OC)cc(F)cc(F)c1NCc1cnc(C(C)(C)C)s1 44943,C1(CC=C)(NC(c2ccc(OC)nn2)=O)CCCN(C(c2ns[nH]c2=O)=O)C1 44944,C=C1CC(N=c2[nH]c(=NCC(=O)N(C)C)[nH]c3cc(C(F)(F)F)ccc23)C1 44945,C#Cc1cc(C(N2CC(CNC(=O)CN3CCCC3C)C(F)(F)C2)=O)cc(F)c1 44946,N1(C(c2cncc(C)n2)=O)CCC(NC(c2ccnc(Cl)c2)=O)C1(C)C 44947,C12(NC(c3cnsc3)=O)CCCN(C(=O)Cc3nc(F)c(F)cc3F)CC1C2 44948,C1(N(C(C(C)SCCCC)=O)C)CN(C(c2cnc(O)cc2OC)=O)CCC1C 44949,N1(C(C(C)Sc2nncn2C)=O)CCC(CO)(CNC(=O)CS(N)(=O)=O)CC1 44950,C(N(CC(C)C#N)N1CCCC(F)(F)C1)c1ccc(C)cc1F 44951,CCS(=O)(=O)c1ccc(S(=O)(=O)N2CCN(C(C3CC3C)=O)CC2)cc1 44952,C1(CC)CN(C(c2cc(C)ncn2)=O)CC1C(=O)NC(CC1CC1)C1CC1 44953,CC(CC(=O)N1CCC(NC(c2ccccn2)=O)C(F)C1)C(C)(C)C 44954,c1(CC(=O)NC(C)(CNC(=O)CCc2ccoc2)C2CC2)ccc([N+](=O)[O-])cc1 44955,N1(C(CCCCOC)=O)CC2CCCC(CNC(=O)Cc3nnc(C)o3)C2C1 44956,c1(CC)cc(C(N2CCC(NC(c3cc(Cl)n[nH]3)=O)C(F)C2)=O)ccc1OC 44957,C(c1ccccc1F)=CCC(N1CCC(NC(c2cc(C#N)no2)=O)(CO)C1)=O 44958,C(=O)(C1OCCc2c(Br)cccc21)NCCCCN(C(C(CC)C)=O)C 44959,C(=O)(C#CC1CCCCC1)NCCCN(C(C1CCC(C)S1)=O)CC 44960,c1(SC)cc(C)nc(N2CCC(CCNC(c3ccc(C(N)=O)[nH]3)=O)CC2)n1 44961,CCCCCCC(=O)NC(C(c1ccccc1)NC(c1ccnn1C)=O)C(C)C 44962,CC(=Cn1ccnn1)C(=O)N1CC2(CCN(C(c3cc4n(n3)CCO4)=O)C2)C1 44963,CCCCC(CC)CC(=O)NCC(CNC(=O)CC=Cc1cccc(F)c1)CO 44964,C1(NCC(c2ccc(C)cc2)C)CCN(C)C(C)C1 44965,c1(CC)cc(S(=O)(=O)NC2COCCC2CCl)c(Cl)cc1Cl 44966,c1(CC)cc(OCC(=O)NC2COCCC2NC(=O)CCCC(C)=O)ccc1Cl 44967,c1(OC)cc(C)ccc1OCC(=O)NC(CNC(c1cn(C)cn1)=O)C(C)(C)C 44968,c1(C(N2C(CNC(C(C)OCC#C)=O)CCCC2)=O)c(F)cc(F)c(F)c1F 44969,O=S(=O)(c1c(Cl)cc(Br)cc1Cl)N1CCCC(c2nc(-c3ccccc3Cl)no2)C1 44970,Cn1nc([N+](=O)[O-])cc1C(=O)NC(C)(C)CNC(=O)C(c1cncn1C)O 44971,C1(CNC(c2c(C)cns2)=O)CC2(CCN(C(C3COCCN3C)=O)CC2)CO1 44972,C1(C(N2CCCC(N(C(c3c(CC)scc3)=O)C)C2)=O)CCc2ncncc2C1 44973,c1(C(N(CC(C)N(C(C(C)n2cnnn2)=O)C)C)=O)c(O)nnc2c1COCC2 44974,C12(NC(C=CC(CC)C)=O)CCC(C1)N(C(c1ccc(OC)nc1C)=O)C2 44975,C1(NC(C(CC)NC(C)=O)=O)CCCN(C(c2cncc(N)n2)=O)C1 44976,C=CC(F)(F)C(=O)NC1CCCC1NC(=O)COc1ccc(C(F)(F)F)cc1 44977,N#CC1CC12CCN(C(=O)C(O)CCNC(c1cc(CO)[nH]n1)=O)CC2 44978,C12(CNC(C=C(C)Cl)=O)CCC(CNC(c3cc(F)cc(C)c3O)=O)(CC1)OC2 44979,c1(CCN(C)C)ccc(C(=O)NCCC(O)CNC(c2cccnn2)=O)cc1 44980,c1(C(C)=O)cncc(C(=O)NC(CNC(=O)CCc2c(C)noc2Cl)CO)c1 44981,N1(C(c2cnc(C)nc2)=O)C2CCC1C(NC(=O)Cc1cc(Cl)cnc1C)C2 44982,CC(C)(C)CCCC(=O)N1CCN(C(c2ccc(C#N)cn2)=O)CC(CO)C1 44983,c1(C(C)NC(c2c(Br)cnn2C)c2n(CCOC)nnn2)ccc(F)cc1 44984,c1(OC)nccc(C(=O)N(C)CC2CCCC2NC(C2C3CCCC23)=O)c1F 44985,CC(C)C(O)C(F)(F)C(=O)NC(C1CN(C(=O)C(C)O)C1)C 44986,C1(NC(c2cn3ccsc3n2)=O)CN(C(=O)C(Cl)=CCl)C2(CCCC2)C1 44987,C(CC)(C(=O)NCC(C)(F)F)N(C(C(F)=CCC)=O)C 44988,Cc1cc(=NC(C)c2ccc(C)o2)[nH]c(=NCCC(=O)N(C)C)[nH]1 44989,C(C1=CCC2CC1C2(C)C)(c1nnnn1C)Nc1cccc(C(C)F)c1 44990,N1(C(Cc2c(C)noc2)=O)CCN(C(C23CC(CO)(C2)OC3C)=O)C(C2CC2)C1 44991,C1(CCC)(NC(C2CCS(=O)(=O)N2)=O)CCCN(C(c2cnsc2)=O)C1 44992,c1(C(=O)NC(CC=C)CNC(c2c(C)ncnc2O)=O)cnc2n1CCCC2C 44993,N1(C(C)Cc2ccncc2)CC(N(C)C(=S)NC(C)(C)C)C(F)(F)C1 44994,c1(CNC(C(CC)N(C)C)=O)ccccc1CNC(=O)CC1CC2CC2C1 44995,c1(C(C)=O)c(C)[nH]c(C(N2CCC(O)C(NC(=O)C=CBr)C2)=O)c1C 44996,c1(SC)ccccc1C(=O)NC(CNC(=O)CCC(=O)OC(C)(C)C)C1CC1 44997,c1(NCC2C(NC(c3ocnc3C(F)F)=O)CCCC2)ncc2cccnc2n1 44998,C1(NC(CC2(CNC(Cn3ncc(CC)c3)=O)CC2)=O)CCCC1N=[N+]=[N-] 44999,n1(CCC)ncc(C(N2CC3C(NC(C4(C5CCCCO5)CCC4)=O)C3C2)=O)c1C 45000,c1(OCC)cccc(OC(=O)C(C2CCCCC2)NC(C2C3CCCC23)=O)c1 45001,N1(C(c2c(OC)cccc2C)=O)CC2CC3CC2C1C3NC(=O)C=C(Cl)Cl 45002,c1(OC(C(C)C)C(=O)NCCC2CCCN2C(=O)C2CC2)ccc(F)cc1F 45003,N1(C(CC(=O)N(CC#C)CC)=O)CC2(CCN(C(C34CCN(CC3)C4)=O)C2)C1 45004,c1(CC(=O)NC2C(NC(C3(COCC)CC3)=O)CCC2)ccc(Br)nc1 45005,c1(C(N(CCC(C)NC(CCCOC(C)C)=O)C)=O)c(F)cc(O)cc1F 45006,CC(C)(C(=O)N1CC2CCC(NC(c3ncsc3Br)=O)(C2)C1)S(C)(=O)=O 45007,c1(C(N2CCC(CNC(c3occc3C3CC3)=O)C2)=O)ccc2c(c1)OCCC2 45008,C1(CNC(c2cn(C(C)(C)C)nn2)=O)CN(C(=O)Cn2[nH]cnc2=N)CCO1 45009,CCC(F)(CNC(=O)CC1CCCCN1C(=O)CCCOC(C)=O)CC 45010,N1(C(C2C(c3ccc(C)s3)C2)=O)CCC(C)C1CNC(C1(C)CCC1)=O 45011,Cn1cnc(C=CC(=O)NCC(c2ccccc2)NC(C2(C(N)=O)CCC2)=O)c1 45012,C1(CNC(C2(C)CC2)=O)CCN(C(=O)C(c2ccc(Cl)cc2)(F)F)CC1O 45013,n1(CC)nccc1C=CC(N1CC(CNC(=O)Cn2ccccc2=O)C(C)C1)=O 45014,C(=O)(C1=COCCO1)NC1C(C2CCN(C(C(CC)=CC)=O)CC2)OCC1 45015,C1(C(C)NC(c2cc(C3CCC3)[nH]n2)=O)CN(C(C2C3CCC2CC3)=O)CCO1 45016,c1(CC)c(C(N2CC(C)(NC(=O)C(CC)NC(N)=O)C2)=O)csc1C 45017,Cc1nc(C(C)C)ccc1C(=O)NC(C)(CNC(C1(F)CCOC1)=O)C1CC1 45018,Cc1[nH]nc2ncc(C(=O)NC3CN(C(C4CCC(=O)C4)=O)CC3O)cc12 45019,C1(C)(C(N(C(C)CNC(=O)CNc2ncccn2)C)=O)CCC(F)(F)C1 45020,c1(C(=O)NCC(C)N(C)Cc2ccc(N(C)C)nc2)c(F)c(F)c(F)c(F)c1F 45021,c1(C(CNC(C2CC=CCO2)=O)NC(C(C)(C)N(C)C)=O)ccccc1F 45022,c1(C(N(C)CC2(O)CCN(C(=O)CSCC(N)=O)C2)=O)oc2ccccc2c1Cl 45023,C1(C(=O)NC(CC)C(=O)NC)Cc2ccccc2CN1Cc1cncc(C)c1 45024,c1(C(=O)NC(C(C)C)CNC(=O)C(C)CF)cccc(N)c1N 45025,N1(C(c2cc(COC)no2)=O)CC(NC(=O)C(O)C2CCC2)CC12CCOCC2 45026,C(CC(C)(C)CC(=O)NCc1nnn(C)c1C(=O)NC1CCN2CCC1C2)OC 45027,N1(C(CSCCNC(C2CC(=O)NC2)=O)=O)CCN2C(=O)NCC2C1 45028,c1(C(=O)NCCNC(C(C(C)C)CN(C)C)=O)cccc2ncnn12 45029,C12(C(=O)NCCNC(C(c3cncnc3)C)=O)C3CCC(CC13)C2(F)F 45030,c1(C(N(CCn2cc(CNC3CCCC3)nn2)CC)=O)ccc(OC)c(F)c1Br 45031,n1(C(C)C)ncc2c1CC(Nc1nccc(N3CCC(SC(F)F)C3)n1)CC2 45032,C1(NC(c2ncn(CC)c2)=O)CC(C(N2CC(c3csc(C)n3)C2)=O)C1(C)C 45033,N1(C(C(CC(C)C)OC)=O)CCC(C)(C)C(CNC(=O)C=CC2CC2)C1 45034,c1(C(N2C(C(C)C)COCC2)=O)cc2ccc(-c3ccc4occc4c3)nc2[nH]1 45035,CC1OC2(CO)CC1(C(=O)NC(C)CN(C)C(C1CC3CCC(C1)C3)=O)C2 45036,C(CCC(c1nnnn1CCC1CC1)NCC1(OC)CCCC1)OCC=C 45037,c1(CC)noc(C(=O)NCC(C2CCC2)NC(C2CC3C=CC2C3)=O)c1C 45038,C1(C2CCN(C(=O)CN3C(=O)CCC3=O)C2)(NC(=O)CCc2ccccn2)CC1 45039,C(=O)(C(CO)NC(C1CC(=C2CCC2)C1)=O)N(CC(C)OC)C 45040,C(CC(F)(F)F)N(C(c1cn(CCNC(c2n[nH]cc2C)=O)cn1)=O)CC 45041,N1(C(c2ccc(C(=O)OC)[nH]2)=O)CCN(C(c2cc(C)ns2)=O)CC(C)(C)C1 45042,CC(Cc1cnc[nH]1)C(=O)NCC(CO)NC(=O)C(C1CCCCC1)O 45043,C1(NC(c2occ3c2CCCC3)=O)COC2(CCN(C(=O)C3=CCSC3)CC2)C1 45044,c1(C(=O)NC(C2CCOC2)C)coc2c1CN(C(c1[nH]ccc1C1CC1)=O)C2 45045,C(c1ccccc1)=CCOCCN(C(C(C1CC1)OC)=O)C.C1CC1 45046,C1(CC)CC(O)CN1C(c1csc(C)c1)C(=O)NC1CCCCC1 45047,N=c1[nH]c2ncc(C(=O)NCC3CCCN3C(=O)COC3CC(F)(F)C3)cc2s1 45048,Cc1occc1C(=O)NCCc1cc(C(=O)NCC(C)(C)C#N)no1 45049,C(=O)(C(CCSC)NC(c1cccnn1)=O)NCC(=O)NCC=C 45050,O=C1CCC(CCC(N2CCCC2CNC(=O)CC2CSC2)=O)N1 45051,C1(SCCN2CCN(C)CC2)CCOCCN1C(c1cc(F)ccc1N)=O 45052,C1(C(N2CCC(CC#C)C2)=O)(NC(=O)CC(C)(O)COC)CCC(C)(C)C1 45053,N1(C(Cn2ncc(CC)c2)=O)CC(C)CC1C(=O)N(C(C)CSC)C 45054,c1(C(N(C(C)CNC(=O)CN2C(C)CCC2C)C)=O)ccc2ncc(=O)[nH]c2c1 45055,c1(C(=O)NC(CNCC)C)ccc(OCCF)cc1.C1(CC(=O)N)CC2CC2C1 45056,N12CC3CCC1C(C3)CN(CCO)CC2=O.c1(CO)cc(-c2ccncc2)no1 45057,CCCCC(C(=O)NCCCC(C)(C)NC(c1cccc(CF)c1)=O)NC(N)=O 45058,C(CC(O)CNC(=O)CNC(=O)C(F)(F)F)NC(CCSCCC)=O 45059,c1(CN=c2cc(C)n(-c3cccc(F)c3)[nH]2)ccc2c(c1)ncn2C 45060,C1(NC(C2CC(=O)N(C3CC3)C2)=O)CCOCC1NC(C1(c2nccs2)CC1)=O 45061,N1(C(C(CC)(C)O)=O)CCC(NC(=O)CCCc2ccc(SC)cc2)C(O)C1 45062,C(CC(C)(C)C)(C(=O)NCCCn1ccnc1)NC(C1C(CC(C)(C)C)C1)=O 45063,Cc1nc(C(N2CCC(OCCNC(c3ccnnc3)=O)C2)=O)n[nH]1 45064,C1(C(N2CC(COC)(NC(=O)CC(C)NC(N)=O)C2)=O)CC2CCC1CC2 45065,C1(O)(C(N2CC(CC(C)NC(=O)Cc3ccsc3)C2)=O)CCCC(C)(C)C1 45066,C1(COC)(CONC(C2CC3CC3C2)=O)CCCO1 45067,C(C)(CCCC(=O)NC(CO)CCC1CC1)NC(c1n(CC)nnc1)=O 45068,Cc1ccc(CN(C2CCCCC2)C(=O)NCc2cccc(C(=O)OC)c2)cc1 45069,c1(C(N(CCC(C)NC(C(C)OCCC=C)=O)C)=O)ccc(C(C)C)s1 45070,C1(C2CCN(C(=O)CC3CCSCC3)C2)(NC(c2cc(C)sn2)=O)CC1 45071,C1(NC(C2N(C)CCOC2)=O)CCCC2CN(C(C3(F)CC4(CCC4)C3)=O)CC12 45072,CN1CCC(F)(F)C(CNC(C23C(C(=O)OC(C)(C)C)C4CC2C3C4)=O)C1 45073,C1(C(=O)NCC(C(N2CC3C(COC)C3C2)=O)(C)C)CCC(C)=C(C)C1 45074,CC(CCNC(=O)CCCCN(C(=O)CC(C)n1cccn1)C)CCO 45075,C=CCC(C(=O)NC(C)CCNC(c1cc2ncccc2s1)=O)C(C)C 45076,C1(NC(CC(C)CF)=O)CCCC12CCN(C(c1cnn[nH]1)=O)CC2 45077,N1(C(C2C(C(C)(C)O)C2)=O)CCC(O)(CCNC(C23CCC(C)(C2)OC3)=O)CC1 45078,c1(NC(C2CN(C(c3nccnc3Cl)=O)CCN2)=O)nc2c(s1)COCC2 45079,CC1CN(C(c2c(F)cncc2Br)=O)CC2(CCN(C(=O)CO)C2)O1 45080,Cc1ccc(CNC(c2cncc(NC(=O)CC(O)c3ccccc3)c2)=O)cn1 45081,C(=O)(C#CC1CCCCC1)N1CCC(NC(C(C)N(CC(F)(F)F)C)=O)C(O)C1 45082,Cc1cc(CC(=O)NCC23CC(NC(=O)C(C(C)C)NC(N)=O)(C2)C3)cc(F)c1 45083,CC(C)CC(C)(CNC(C1(C#N)CC(C)C1)=O)NC(c1ccc(NC=O)cc1)=O 45084,N1(C(C2(N(C)C)CC2)=O)CCN(C(c2cccc(CC#N)c2)=O)CC(O)C1 45085,C(=O)(CC(C)(C)c1ccc(F)cc1)N(C1CC(NC(C2(CSC)CCC2)=O)C1)C 45086,N1(C(c2n(C)nnc2)=O)CCCC(C2CC2NC(C2CCCN2S(C)(=O)=O)=O)C1 45087,c1(C(=O)NC2CC(NC(C3(CC)CC3)=O)C2)cc(=N)[nH]cc1Br 45088,C1(CCC2N(C(CCOC)=O)CCC2)CCN(C(c2cncn2C(C)C)=O)CC1 45089,c1(C(=O)NC2(CNC(CCOCC)=O)CC2)cccc2nn[nH]c12 45090,c1(OC)ccc(CN2CCCC2CC(=O)Nc2cccc(C)n2)c(Cl)c1OC 45091,c1(C(=O)NC23CC(NC(C(c4cccc(C)c4)C)=O)(C2)C3)cc(F)c(N)cc1F 45092,c1(C(=O)OC)cc(NC(c2ccc3c(n2)OCCO3)=O)cc2[nH]ccc12 45093,C1(NC(C2CCC(C)(C)CO2)=O)CC2CCC1CC2NC(=O)CC1CCCOC1 45094,c1(C(=O)NC2CC(CNC(C3CC=CC3)=O)C(O)C2)ccc2oc(O)nc2n1 45095,C=C(C)C1OCCC1CNC(C12CC(CO1)N(C(=O)COCC)C2)=O 45096,c1(C(=O)NC2CC(CCNC(Cc3n(C)cnn3)=O)C2)cc(Cl)cc([N+](=O)[O-])c1 45097,C(C(C)(C(=O)NCCCN(CCCCNC(c1cc(=O)cc[nH]1)=O)C)OC)OC 45098,c1(OC)ncnc(OC)c1CN1CCC(NC(=O)Cn2ccnn2)C1 45099,C1(NC(c2c(C)cccc2F)=O)CC1C1CCN(C(=O)Cc2csc(Cl)c2)CC1 45100,N1(C(C(C)OCCC#C)=O)CCOC(C)(CNC(c2ccc(OC)c(F)c2)=O)C1 45101,C1(C(C)C)N(C(=O)N(C)C(c2ccccc2)c2nc(C(C)O)n[nH]2)CC12CCC2.O 45102,C(c1cn(C)c2ccccc12)=CC(=O)NC1C(C)CN(C(c2cnn[nH]2)=O)CC1 45103,C1(N(C(=O)Cc2cnoc2)CC)CCCN(C(=O)CC2CC(F)(F)C2)CC1 45104,N1(C(c2nc(Br)cs2)C(=O)NCCCSC)CCC(CCO)CC1 45105,C(=O)(CC(O)CC(C)(C)C)N1CCN(C(CCCCN(C(C)=O)C)=O)C(C)C1 45106,C1(S(C)(=O)=O)(C(N2CC(C)N(C(=O)CN3CCSCC3)CC2)=O)CC(O)C1 45107,O=C1OCCC2CN(c3ncncc3-c3ccccc3)CC12 45108,n1(CCC(=O)N(CCF)CCc2ccccn2)cc(COc2ccccc2)nn1 45109,CCCCC(C(=O)NCc1ccnc(O)c1)NC(=O)CC1CC2CC2C1 45110,C1(CNC(C(C2CN(C(C(C(=O)OCC)F)=O)C2)O)=O)OC(=O)NC1(C)C 45111,CC(C)CCC=CC(=O)NC(C)C(=O)NCC(C1CC1)N(C)C 45112,N1(C(C(C)OCCN(C)C)=O)CCC(NC(c2cncc(N)c2)=O)CC1 45113,N1(C(COCCCOC)=O)C2CCC1CN(C(=O)CC(O)CC(C)C)C2 45114,N1(C(C2(C)CC(C)(C)C2)=O)CCC2(CCC(CNC(C3CC3(C)C)=O)OC2)CC1 45115,Cc1cccc(Cl)c1OCC(=O)NC1CN(C(C2CC(C)(F)C2)=O)CC12CC2 45116,n1(CC(=O)Nc2ccnn2Cc2cc(Cl)on2)cc(CCO)nn1 45117,Cc1cc(F)ncc1C(N1CCN(C(=O)CCCCCF)CC1C)=O 45118,N1(C(CCC2CC(OC)C2)=O)CCCCC1CNC(=O)C(O)Cc1ccccn1 45119,NS(=O)(=O)CCN=c1[nH]c(N(C)Cc2ccc(Br)s2)nc2c1CCC2 45120,c1(CN2CC(F)(C(=O)Nc3cc(CC)cc(Br)c3)C2)cc(Cl)c(O)cc1F 45121,N1(C(C(C)=CC)=O)CCN(C(C2(S(C)(=O)=O)CCC2)=O)CC1CC(=O)NC 45122,CC1(C(=O)NC2CCCN(C(=O)C(C)(O)C(F)(F)F)CC2)CCC(F)(F)CC1 45123,CC1CCN(C(=O)CC2C=CCCC2)C1C(=O)N(C)CCC1CCCC1 45124,C1(NC(c2ccc(OC)cc2)=O)CCC(C)N(C(c2ccc(F)c(Br)c2)=O)C1 45125,N1(CC#N)CCCC1C1CCCCN1C(c1cccc2nc(O)[nH]c12)=O 45126,C(CC1CCC1)(C(=O)N(C)CC1CCN(C(=O)Cc2cc(C(C)C)no2)C1)OC 45127,c1(N2CCC(CC=C)(NC(c3cc(C4(C)CC4)n[nH]3)=O)C2)ncnc(Cl)c1CO 45128,C1(C(=O)NC(C2C(C(=O)OC)C2)C)CC2(CCN(C(C3(C)CCC(=O)N3)=O)C2)C1 45129,N1(C(C(C)OCC2CC2)=O)CC(CO)C2(CCNCC2)C1 45130,c1(NC(C2CCC2F)=O)cc(C(F)(F)F)c(Cl)cc1F 45131,C1(NC(C(CC)NC(N)=O)=O)CC2CC(NC(=O)Cc3ccnc(Cl)c3F)C1C2 45132,N1(C(c2c(OC)nccc2)=O)C2CCC1C(C(=O)Nc1ncccc1C(C)=O)C2 45133,c1(C(=O)NC2CN(C(c3n(CC)nnc3)=O)C(CO)C2)ccc2nncn2c1 45134,C(=O)(C1=CS(=O)CCC1)N1CC=CC(NC(CCc2cn(C)nn2)=O)C1 45135,Cc1nn(C)c(-n2ccnc2C)c1C(=O)NC1CCCN(c2ccccc2F)C1 45136,N1(CC(N2CC(n3cccn3)(C(=O)O)C2)=O)CC2(COC2)C1 45137,C1(CN(C(=O)CCC2CCCO2)C)CN(C(c2cccc(O)n2)=O)CC12CC2 45138,c1(CCC(N2CCN(C(C(CC)O)=O)CC2C(C)C)=O)ccc(S(C)(=O)=O)cc1 45139,N1(C(C2(NC(C)=O)CCC2)=O)CCC2(CCCN2C(C2CCCC2C)=O)C1 45140,c1(NC(c2cncc(-c3ccc(SC)cc3)n2)=O)cc(C)c(I)cn1 45141,C(CC(=O)NCCC1=CCCCC1)(C(C)C)NC(C(C1CC1)OCC)=O 45142,c1(C(N(CCC(C)NC(C2CC23CCC3)=O)C)=O)c(Cl)cccc1Br 45143,CCCC(C)CCCC(=O)NC1CCC(C)N(C(=O)C=Cc2nccn2CC)C1 45144,C(=O)(C#CC1CCCOC1)N1CCCCC(CNC(c2ccc(C)c(F)n2)=O)C1 45145,C1(C(=O)NC2CCN(c3nccc4c(Br)cccc34)C2)CC2(CO1)CC1(C2)OCCO1 45146,N1(C(c2cncc(NC(CC)=O)c2)=O)CC2(CCC(NC(c3ccoc3)=O)C2)C1 45147,N1(C(CNC(CCC)=O)=O)CCCC2(C(=O)NC3(c4ncccc4F)CC3)CC12 45148,S(=O)(=O)(c1cccc(N2CCOC(CCOC)C2)n1)NCC=CCCC 45149,C1(N(C(c2c(COC)cco2)=O)C)CCC(NC(C2CC3(CC3)CO2)=O)CC1 45150,N1(C(C(C)OCC=C)=O)CCC2(CCCN(Cc3cc(C)ccc3O)C2)C1 45151,CC1CN(C(=O)CC2OCCC2(C)C)CC1NC(=O)Cc1n[nH]c(=N)s1 45152,c1(CC(N2C(C)CC(NC(C3CCC(C)C3)=O)C2)=O)ccc2sccc2c1 45153,c1(C(C)C)nc(C(=O)N(C2CN(C(=O)C(C)CN3CCCCC3)C2)C)cs1 45154,C1(CNC(CN(CCOCCOC)C)=O)CC2(CO1)CN(C(=O)C=CCOC)C2 45155,S(=O)(=O)(CCC(F)(F)F)NC1(C)CCCN1c1ncc(C#N)cc1Cl 45156,N1(C(c2ncc(C)cn2)=O)CCN(C(c2nccc(Cl)c2C)=O)CC1C1CC1 45157,C1(NC(c2cc(C)c(O)nc2)=O)C2CC3CN(C(=O)CC(C)(C)C(F)F)C1C3C2 45158,N1(C(c2[nH]cc(C#N)c2)=O)CC2(CCC2)CC1CNC(C1(N2CCC2)CCC1)=O 45159,N1(C(CSc2c(C)n[nH]c2C)=O)CC2(CCC2)CC1CNC(C1(F)CCOC1)=O 45160,N1(c2nccc(OC)n2)C2CCCC1CN(C(C1(O)CCOC1)=O)CC2 45161,C(C(=O)N(CCCCN(C(=O)CC1C(=O)NN=C1C)C)C)(C(C)C)OCC 45162,C(C(CC)(CC)C(=O)NC(c1ccccc1)C)NC(C(CC=CC)C)=O 45163,c1(N2CC(C(C)NC(C3(C)CC(O)CN3C)=O)C2)ccc([N+](=O)[O-])cn1 45164,N1(C(c2cc(C)c(C)[nH]2)=O)CCCC2CN(C(=O)C(C)C(O)C(C)C)CCC12 45165,C(C(=O)N1CC(=O)NC(C)C1)(C(C)(C)C)n1cc(C(=O)OC)nn1 45166,C(=O)(CCC(C)(C)NC(=O)CC1CCC(=O)C1)NCCC 45167,c1(CC(=O)N(C2CCN(C(C3CCCN3S(C)(=O)=O)=O)C2)C)ncc(F)cc1F 45168,C(CC(C)C(=O)NC(C)(CNC(=O)COCc1nnc(C)s1)C1CCC1)=CCC 45169,C1(CC=C)(NC(=O)C(CN(C)C)NC(=O)Cc2cnn(CC)c2)CCCC1 45170,c1(OCC)ncc(C(=O)NC2(C)CC(NC(C3CCCCNC3=O)=O)C2)cc1Cl 45171,C#CCC(CC(=O)N1CCCCC1CCO)NC(=O)C(C1CC1)OCC 45172,c1(C(=O)NCc2ccc(-c3ccc(CO)o3)cc2)nc(Br)n2c1CCNCC2 45173,CC1(C)CC(CCNC(C2CCN(C(=O)CS(C)(=O)=O)CC2)=O)CO1 45174,CCCC(CCCNC(c1cscc1OC)=O)NC(=O)C(CC)C(C)C 45175,CCP1(=O)CCN(c2ccc(NC(=O)OC(C)(C)C)nc2)CC1 45176,c1(CNCC(n2cnc(-c3cccs3)n2)C)cccc(Cl)c1 45177,N1(C(CC(=O)NCC)=O)CC2CN(C(=O)CC(C)C(C)C)CC2(C)C1 45178,C1(CNC(CCC=C=C)=O)CC(C)CN(C(=O)CCC)C1 45179,C1(C(N2CC(C=C)C(NC(=O)C3=COCCC3)C2)=O)CC12CCCCCC2 45180,C1(CNC(c2ccn(C)c2)=O)CCC(F)(CNC(C2CC3CCC(C2)S3)=O)CC1 45181,c1(OC)ccnc(CNC(=O)CCCNC(C2CCOC2(C)C)=O)c1 45182,C(=O)(C(C)C(O)C(C)CC)N1CC(C(=O)NCC(CC)N(C)C)C(C)(C)CC1 45183,N1(C(C(CCNC(=O)CC2OCCO2)OC)=O)CCOC(C)(C)C1C 45184,C1(NC(c2nc(C)oc2)=O)CCCCN(C(=O)COCC2CCCC2)CC1 45185,Cc1cc(F)cnc1C1(NC2(c3nnnn3C3CCCCC3)CSCSC2)CC1 45186,N1(C(COC)=O)CCOC(CNC(=O)CNC(c2ccnc(N(C)C)c2)=O)C1 45187,C(C)(C(C)C(=O)Nc1ccsc1CC)NC(c1cn(CC=C)nc1)=O 45188,CCCCCC(C)(C)C(=O)NC1CN(C(=O)C(C)SC(F)(F)F)CCC1C 45189,C1(C(N2C(CNC(C3N(C)CC4(CC4)C3)=O)CCC2)=O)CCC(C2CC2)CC1 45190,N1(C(c2c(C(C)C)nco2)=O)CC(=O)CC1C(=O)NC1CC(F)(F)C1 45191,c1(C(C(=O)OC)NC(C2NCCCC2C(F)(F)F)=O)ccc(F)c(Cl)c1 45192,CC1(C(N2CCC(F)(CNC(=O)C#CC3CC3)C2)=O)CCC(F)(F)CC1 45193,c1(C(=O)NCCCCCNC(c2ccc(OCC)s2)=O)ccn2cccc2c1 45194,C(=O)(C(C)(C)CN1CCCCC1)NC(C1C(C#C)C1)=O 45195,c1(C(C(=O)NC(C)C(=O)OC)N(CCCCCC)C)nn(C)c2c1CCC2 45196,c1(C(=O)NC(c2nc[nH]n2)CC)ccoc1CNC(C1CC1(C)CC)=O 45197,N1(C(CC(CCC)(C)O)=O)CCC2C1CCCN2C(c1cn(C2COC2)nn1)=O 45198,c1(CC(=O)NC(C2CCOC2)CNC(C2(F)CC=CC2)=O)ccccc1Br 45199,CC(C(=O)N1CCCC1CNC(c1ccc(N)c(C(F)(F)F)c1)=O)S(N)(=O)=O 45200,c1(C(=O)NCC2(F)COCCN(C(C=NOC)=O)C2)cnc2scc(C)n2c1=O 45201,C(CN=[N+]=[N-])(C(=O)NCCCc1ccccc1)NC(COCC=C)=O 45202,c1(C(=O)NC(C)CNC(=O)C(c2ccc(C#N)cc2)O)cnn2cccc(Cl)c12 45203,C(CC(=O)CCO)c1cn(C2CCC(NC(=O)C=CC3CCCC3)C2)nn1 45204,c1(NCCCC)ccc(C(=O)NC2(C)CC(NC(=O)CC3CC3)C2)cc1[N+](=O)[O-] 45205,c1(CN2CCCC(C#C)C2)ccc(Br)c(F)c1OC.c12cc(ncn1)CN2 45206,N1(C(c2cn(C)c(=O)cc2)=O)CC2CCC1CC2NC(C1COCCOC1)=O 45207,CC1(C)CCCCC1(CO)NCc1ccc(N)c(F)c1 45208,CC(C(=O)NC(CNC(c1c(F)cncc1Cl)=O)C1CCC1)C(F)(F)C(F)F 45209,N1(C(C)(C)C)CCC(C(=O)NCc2[nH]nc3c2COC3)C(F)C1 45210,CCCCCCCCCCn1nc(C(C)OCC)nc1-c1nnc(C)cc1O 45211,C(C1CCCc2cccnc21)NC(NC(CC)CC)=NCCNC(=O)COC 45212,C1(NC(c2cc(OC)n(C)n2)=O)CN(C(C2CCC(=O)O2)=O)CC(F)(F)C1 45213,c1(C(=O)NC2(C)CCN(C(c3c(CC)c[nH]c3)=O)C2)ccc(N)c(C)c1Cl 45214,CCCCC(O)CNC(C1CCCCN1C(c1ccc(OC)o1)=O)=O 45215,c1(C(N2CC3C(C2)N3C(=O)Cc2ccc(Cl)cn2)=O)cncc2cnccc12 45216,C1(C(N2CC(C(C)(C)C)OCC2)=O)C2CCN(C(=O)Cn3cc(C4CC4)nn3)CC12 45217,N(C(=NCc1cnc(C)cn1)NC(c1ccccc1)C)CC1(SC)CCC1 45218,CN1CCN(C(=O)CC2(NC(=O)CC3CC4CC4C3)CC2)CC(O)C1 45219,c1(C(=O)Nc2nc(C)sc2)cc(-c2cc(OC(C)C)ccc2C)c2cn[nH]c2c1 45220,c12ccc(cc1O)c(=O)[nH]2.N1(C(C(C)(C)SC)=O)CCC(NS(C)(=O)=O)CC1 45221,c1(CC(=O)NC(C2CN(C(=O)Cc3ccon3)C2)C)ccc(Br)cn1 45222,Cn1cc(C(F)(F)F)cc1C(=O)NC1CCC1NC(=O)C1=NOCC1 45223,C(C(F)C(=O)N1CC(OC(=N)O)C1)C1CN(C(=O)OC(C)(C)C)C1 45224,C1(NC(=O)CC23CCCN2CCC3)CN(C(=O)Cn2cncn2)CC1C1CC1 45225,N1(C(CN(C(c2cccc(C#N)c2)=O)CC)=O)CC2(CC(F)C2)C1 45226,C(=O)(CCC(C)(C)NC(C1CCC(O)C1)=O)NCC1CC(C)(O)C1 45227,N1(S(CC#N)(=O)=O)CCC(F)(F)C(C(=O)Nc2ccc3occc3c2)C1 45228,c1(OC)cc(C(N2CC(CNC(c3c(OC)noc3C)=O)C(C)C2)=O)ccc1F 45229,C1(O)(CNC(=O)CCCC2CCCC2)CCCN(C(C2COC(=O)O2)=O)C1 45230,C#CCCC(O)C(=O)NC1(CCC)CCCN(C(=O)Cc2ccnc(O)c2)C1 45231,N1(C(C2(SCC)CC2)=O)CCC(CN(C(=O)C=CC(N2CCOCC2)=O)C)CC1 45232,C(=O)(C(CC1CCC1)NC(=O)CCc1nc(O)n[nH]1)NCC.C12(CC1)SC2 45233,CC1(C)CC(CNC(c2cccnc2)=O)N(C(=O)CCc2cc(Cl)cs2)C1 45234,c1(C(=O)NC2C(NC(C3C(C#N)CC3)=O)C2)ccc(C2CCCCC2)cc1 45235,c1(CCC(=O)OC)ccc(N(CCCCNC(c2nc(=O)n(C)[nH]2)=O)CC)nc1 45236,C(=O)(C(CNC(=O)CCCC1CCCC1)C(C)C)N(CCCOC)C 45237,Cc1c(CC(N2CCC(CCCO)C2)=O)c(=O)oc2cc(N)ccc12 45238,Cc1cc(N2CCC3(NC(C4CC5(CC5)C4)=O)CCCC23)n2nc(C)cc2n1 45239,C=CC1CN(C(C23CCOC(C)(C2)C3)=O)CC1NC(=O)CCc1csc(C)n1 45240,CCC(CC(=O)NC1COCC1CNC(=O)Cc1ccn(C(C)C)n1)C(F)F 45241,c1(C(=O)NC(CC=C)CNC(C2CC(C)=NO2)=O)ccc(Br)c(Cl)c1 45242,C1(CNC(C2=CC(C)(C)C2)=O)CC2COCC2N1C(=O)COc1cccc(Cl)c1 45243,N1(C(C(=O)NCC2CC2)C2CC2(Br)Br)Cc2nccc(Cl)c2C1 45244,c1(CC(C(=O)NC(CCCNC(c2occ(C)c2)=O)C)C)c(C)n[nH]c1C 45245,c1(C(=O)NCC(C)NC(CCn2ncc(C)c2)=O)ccc(Cl)cn1 45246,c1(CC)ccc(C(=O)NCC(C)(C(C)C)NC(=O)CCc2cnc(O)[nH]2)cn1 45247,C1(C(N(C2CCN(C(c3csc(=N)[nH]3)=O)C2)CC#C)=O)CC(C)(C)CCO1 45248,C1(N(C)C(c2cccn2C)=O)CCN(C(C2(C)CCNC2=O)=O)CC1 45249,Cc1cc(-c2nc(C)c(C(=O)N(C)CCN(C(=O)CCC(C)C)C)s2)ccc1F 45250,c1(C(N(C2CCCN(C(CCCC#C)=O)C2)CC)=O)ccc(C)c(Cl)c1 45251,CC#CCC(C(=O)N1CCC1(C)CC)NC(c1cn[nH]c1)=O 45252,c1(C(=O)NC2CC(CNC(C(C)CC(C)(C)C)=O)C2)ccc2c(c1)CCCC2 45253,C1(C)(CNC(C(C(C)C)NC(N)=O)=O)COCCN(C(=O)C2=CCCCO2)C1 45254,C1(C(=O)NC(CC)CNC(c2cc(C(C)C)[nH]n2)=O)CC12CC(F)(F)C2 45255,c1(CC)cc(Br)ccc1C(N1CCCC(N(C)C(c2cc[nH]n2)=O)C1)=O 45256,CC(O)C(C)C(=O)NC(C1CCCN1C(=O)CSCC(N)=O)(C)C 45257,c1(C(=O)NC(c2cccc(C)c2)CNC(C=COC)=O)nn2c(c1C)CCCC2 45258,Cc1cc(C(N2CCC(O)(C(C)NC(C3CC(F)C3)=O)C2)=O)ncc1N 45259,C(C1CN(C(=O)CC)CC1N)=CC.N1(C=O)CCSCCC1C 45260,c1(COC)ncc(C(N2CC(=C(F)CNC(=O)C(C3CCC3)OC)C2)=O)c(O)n1 45261,C=CC1CCCCN1C(=O)CC1(C)CCN1C(=O)C(O)CC1CCCC1 45262,C(=O)(C(F)C(C)(C)O)N1CC(CCC=C)(C(=O)Nc2c[nH]ccc2=O)C1 45263,c1(NC(c2n(CCCSC)nnn2)c2csc(Br)c2)cc(O)c(C)cc1C 45264,N1(CC(=O)NC(CNC(c2cc(C3(C)CC3)n[nH]2)=O)(C)C)CCS(=O)(=O)CC1 45265,c1(SC)ccc(C(=O)NCC(C)(C2CC2)NC(=O)COCC(=O)CO)cc1 45266,c1(CCCOCC)cc(CC2CSCCN2c2ccnc(C)n2)cc(C(F)(F)F)c1 45267,N1(C(C2N=C(C)SC2)=O)CCCOC(CNC(c2cc(C)n(C)c2C)=O)C1 45268,c1(N(CCN(C)C(C2CCC=CCC2)=O)C)cc(C#N)nc(C2CC2)n1 45269,C(=O)(C(C)CC(C)C)N1CCC(C(F)F)(NC(c2c(COC)cccc2)=O)C1 45270,c1(N(CC(O)CC(F)(F)F)CCN(CC)CC)cc(F)cc(F)c1 45271,c1(C(=O)NCC(CNC(C=CC(=O)OCCCC)=O)O)nn[nH]c1Cl 45272,C#Cc1ccc(F)cc1C(=O)NCCOCCNC(c1cc2c(ccn2C)[nH]1)=O 45273,c1(NC(C(F)(F)C2(OC)CCC2)=O)cccc(CNC(=O)Cn2ccnn2)c1 45274,CC1CCC(C)C(C)C1NCC1CCC(=O)N1 45275,C1(CCNC(c2cnc(CC)s2)=O)CCCCN1C(=O)C(C)C1CCC1 45276,C(CC(C(=O)NCC1CCN(C(C)C)C1)NC(c1sccc1Cl)=O)OC 45277,c1(C(N2CC(OCCNC(=O)C(F)CC3CCCC3)C2)=O)ccc2sncc2c1 45278,C12(C(=O)NCC(CC#C)(C)C)CCCC1CCN2C(c1n[nH]cc1C)=O 45279,c1(C(C(=O)NCCC)N(C)CC2CC3CCC2C3)ccc2c(c1)NC(=O)CO2 45280,c1(C(N2CC(C)(C(=O)Nc3ccnc(F)c3)C2)=O)c(F)c(F)cc(F)c1F 45281,Cc1cc(C#N)ccc1NCc1csc(Cl)n1 45282,CC(C)(C(F)(F)F)OCC(=O)NCCOCCNC(C1(F)CC=CCC1)=O 45283,c1(C(N2CCC(CNC(C=CCOC)=O)(OC)CC2)=O)ccc(C)c(C)c1O 45284,N1(c2nnc(C)s2)CC(CNC(C2(C)CC(C)(C)C2)=O)OC2(CCC2)C1 45285,C1(CCCC(=O)OC(C)(C)C)C2CN(C(=O)Cc3ccco3)CC12 45286,c1(C(C(=O)NCCC(C)NC(C2(C(F)F)CC2)=O)=O)cc(F)cc(Cl)c1 45287,C1(C(=O)NCCCSCC)CCCC1CNC(c1nc(Cl)cs1)=O 45288,Cc1noc(C(F)(F)F)c1C(=O)NCC(F)CNC(C1(C2CC2)CC1)=O 45289,c1(CNC(c2ccc(CC)[nH]2)=O)ccc(CN(C(=O)C(C)=C(C)CC)C)cc1 45290,c1(N2CC(COC)C(SC)C2)cc(Br)ccc1S(=O)(=O)NCc1ccc(SC)o1 45291,C(=O)(C1COc2ccccc21)N1CC(CCNC(c2cc(C)n(C)c2)=O)OCC1 45292,Cc1cc(CC(=O)NCCCCNC(=O)CCC(=O)c2ccncc2)c(C)s1 45293,N1(C(c2c(C)nn[nH]2)=O)CCN(C2CCCN(C(=O)C(C(C)C)N(C)C)C2)CC1 45294,C1(C(=O)NC(C#C)CCC)CC(=O)CN1C(C1(C(=O)C2CC2)CC1)=O 45295,N1(C(c2c(COC)noc2)=O)CCC(OC2CCN(C(=O)CCOCN)C2)CC1 45296,n1(C(CC)C)ccc(=NC(=O)C2CN(C(c3ccccc3O)=O)CCC2(C)C)[nH]1 45297,N1(C(C(C2CCCO2)OC)=O)CCN(C(C2CC(=O)C2C(C)(C)C)=O)CC1CO 45298,C1(CNC(C2C=CCN2C(=O)C(O)C2CCCC2)=O)CC2(CCC2)C1 45299,c1(C(c2n(CC=C)nnn2)NCc2ccns2)ccc(C)cn1 45300,N1(C(Cc2ccc(C)s2)=O)CCCC(N(C)C(C2C(C)OC(C)C2C)=O)CC1 45301,C1(C(=O)NCC(C)C(=O)NC2C=CC(C)(C)CC2)CCC(C)(O)CC1 45302,c1(SC)ccc(C(=O)NCCCCNC(=O)C(c2ccccc2)C2CC2)cc1 45303,CC(CS(C)=O)C(=O)N(CCCNC(=O)CNC(=O)CCCCO)C 45304,C(C(C)(C(=O)NCC=CCC(=O)N(CC(C)(C)O)C)OC)OC 45305,C(=O)(C1=CCS(=O)(=O)C1)NCC1(C)CCN(C(=O)Cc2cc(Cl)ccc2O)C1 45306,C(=O)(CS(=O)(=O)c1nccn1-c1ccccc1)N1C(c2n(CC)ncc2)CCC1 45307,c1(NC)cnc(Cl)cc1C(=O)NCC1CCC(NC(C2COCCO2)=O)C1 45308,c1(C(=O)OC)cc(Cl)c(OC)cc1C(C)C.c12ncc(s1)CNC2 45309,C#CC(C(C)(C)C)NC(=O)C(C)(CSC)NC(C1SCC=C1C)=O 45310,c1(-c2cn(C)nc2)ccc(F)c(C(=O)NCc2cn(CC3C4CCCC34)nn2)c1 45311,c1(C(c2nnnn2CC2CCOC2)NCc2ccn(C)n2)c(Cl)cncc1Br.C1CC1 45312,n1(CC)ncc(C(=O)NC(C)CNC(=O)C(C(C)C)NS(C)(=O)=O)c1C1CC1 45313,N1(C(C)=O)CCCC1C(=O)NC(C)(CNC(c1cn(CC(N)=O)nn1)=O)CO 45314,C1(CNC(C(c2cnn(C)c2)C)=O)CCC(NC(=O)Cn2cncn2)CC1 45315,C(=O)(C1=CCCC1C)NC(CCOCC)C(=O)NCCNC(c1ccoc1)=O 45316,C1(C(N(C2CCC(NC(C(CC)=CCCC)=O)CC2)C)=O)CC(C)CC(C)(C)C1 45317,Cc1ncccc1C(N1CC=CC1CNC(C1C(F)(F)C12CC2)=O)=O 45318,c1(OC)ccnc(-c2cn(C3CCN(C(C4(C)C=CCCC4)=O)C3)nn2)c1 45319,c1(-c2ccc(C3N(C(CN4CCC(CC)C4)=O)CCC3)cc2)cc(C)cc(C)c1 45320,c1(OC)cccc2c1OCCCC2NC(=O)C(=O)NC1CCN(C2CC2)C1=O 45321,N1(C(c2c(CC)cco2)=O)CCC(C2CC2)C1C(N1CC(CO)C2(CCC2)C1)=O 45322,N1(C(CCCOC(C(=O)NC2COC2)C)=O)CCCOC(CSC)C1 45323,CC1(C(=O)NC2CC(CNC(C3(C(F)F)CCCC3)=O)C2)CCCNC1=O 45324,c1(CN(C(C2CCCSC2)C(=O)NCCOC)C)c(C)nn(C)c1C 45325,C1(NC(c2nc(Cl)c(Cl)s2)=O)CC2CCC(C1F)N2C(C1CCCSC1)=O 45326,C1(C(N2CCN(C(c3cccc(O)c3)=O)CC2)=O)(OC)CC(C)CC(C)C1 45327,CC1CCC(NC(=O)NC2CN(CC(F)(F)F)C2)C(C)C1 45328,N#CC1CC(C(=O)NCC(O)CNC(C2(CC3CCC3)CC2)=O)C1 45329,C12(C=O)CC(CN(N3CC(C(CC)CC)C3)C1)C2.n1(C(C(=O)N)C)ccnc1C 45330,CCCC(C)CC(=O)N1CCOC(CN(C(=O)CN(C)C2CC2)C)C1 45331,N(C(=NCCC)NCCC(C)Oc1cccc(C(F)(F)F)c1)CC=C 45332,N1(C(c2ccc(C)[nH]2)=O)CC(C(N2CCOCC(N(C)C)C2)=O)C(F)(F)C1 45333,N(C1CN(c2cc(Cl)ncn2)CCc2ccccc21)C(=O)CCc1cnc[nH]1 45334,C1(C(N2C(C)CC(CNC(c3cc(O)nn3C)=O)C2)=O)CCn2c(O)nnc2C1 45335,C(=O)(CC(O)C(C)C)NCC(c1ccc(C)cc1)NC(c1c(CO)noc1C)=O 45336,C12(CNC(=O)C=C3CCCC3)CCCC(CN1C(=O)CSc1ccccc1)C2 45337,c1(C(=O)NC2CCN(Cc3c(C#C)cccc3)CC2O)ccc(O)c(O)c1Cl 45338,c1(CCOC(=O)CNC2CCN(C(c3cnoc3)=O)CC2)ccc2nccn2c1 45339,c1(COC)nc(NCC2CC2C2CCC2)cc(=NCCSC2CCCC2)[nH]1 45340,c1(C(N(CCCNC(C2C(=C)C2)=O)C2CC2)=O)ccc(NC)c(S(N)(=O)=O)c1 45341,N1(C(C(C(C)C)NS(C)(=O)=O)=O)CCC(C)CC1CNC(=O)CN(C)C(C)C 45342,c1(OC)ccccc1C(N1CC(N(C(=O)CCC(C)N(C)C)C)C(O)C1)=O 45343,Cc1[nH]c2c(C(N3CCC(CNC(=O)CC4CC4(Cl)Cl)C3)=O)cccc2c1C 45344,N1(C(C(C(C)(C)O)F)=O)CCC(C2(NC(c3ccnc(C4CC4)c3)=O)CC2)C1 45345,c1(OCC(N2CC(NC(=O)C(=O)NC3CC3)OCC2)=O)cc(F)ccc1F 45346,N1(c2c(OC)cnc(Cl)n2)CCCC(C2CC2NC(c2nccc(Cl)c2F)=O)C1 45347,c1(-c2cn(C3CC(NC(c4cn(CC=C)nc4)=O)C3)nn2)cc(C)cc(C)c1 45348,C1(O)(CCNC(c2c(C)nc(CCC)s2)=O)CCN(C(=O)C(CC)OCC)CC1 45349,N1(C(c2c(C)nc(C(C)C)s2)=O)CCN(C(=O)CSc2nc[nH]n2)C(CO)C1 45350,Cc1cc(N2CC(C)(C)CC2CNC(c2csc(CO)n2)=O)nc(C)n1 45351,c1(C(=O)NC2(C3CC3)CCN(C(C(CC)(C)C#N)=O)C2)cnc2ccncc2c1 45352,C(=O)(C(=O)C(C)(C)CC)NC(C(=O)N(C(C=C)C)C)C(C)C 45353,c1(C(=O)NC(C(C)NC(C2CC(=C)C2)=O)(C)C)cc(Cl)cc(F)c1N 45354,c1(C(=O)NCCN(CCC)C(C2CCCSC2C)=O)occ2c1CCC2 45355,C1(NC(c2ccccc2Cl)(C)CO)CC2CCC(C1)C2N 45356,c1(C(=O)NC2(COC)CN(C(c3n(CC)c(O)nc3)=O)C2)cncc([N+](=O)[O-])c1 45357,C#CC1(NC(=O)C(C2CCC2)NC(=O)C(CC)CC=C)CCCCC1 45358,N1(C(CCc2cn(C)nn2)=O)CC(C)(C)CCC1CNC(C1CCCNC1=O)=O 45359,N1(C(COCC#C)=O)CC(C)(CNC(=O)Cc2cccc(C#C)c2)CC1(C)C 45360,CC(C)CCC(C)N(C(=O)C(C)N(C(C1CCC2CC12)=O)C1CC1)C 45361,c1(C(=O)NC2CC3CN(C(C(CC)=CC)=O)C(C2)C3)ccc2cnnc(O)c2c1 45362,C(C1CCOCC1)=CC(N1CC(COC)(CNC(C2(CO)CCOC2)=O)C1)=O 45363,c1(C(N2C(CN(C(CC=CC=C)=O)C)CC(F)C2)=O)cccc(OC(C)C)c1C 45364,c1(C(=O)NC(C)(CNC(=O)C(O)CN2CCCC2)CO)csc2nnsc12 45365,N1(C(C=C(C)Cl)=O)CC(C)(C)CCC1CNC(=O)CC(O)c1ccccc1 45366,N1(C(c2nnn(C(C)(C)C)n2)=O)CC(NC(c2ncccc2O)=O)CC(F)C1 45367,c1(C(=O)NCC(C)CNC(c2ccnn2CC(F)F)=O)oc2ccccc2c1Cl 45368,C1(F)(CNC(COCCCOC)=O)CCCN(C(C2CCC=CCCC2)=O)C1 45369,C(CC(C(=O)NCCc1nncn1CC)NC(c1cnco1)=O)=CC 45370,N1(C(Cc2nc(C)oc2)=O)CCCC1(C)C(=O)NCC1(C)CCCC1O 45371,c1(OC)ccc(C(=O)NC2CCC2NC(C2CC2c2ccc(F)cc2)=O)c(F)n1 45372,Cc1ccc(F)c(CNC(=O)C(C)Sc2ccc(F)cc2)c1 45373,C1(NC(C(C)OCC#C)=O)CN(C(=O)CCc2cccs2)CC2(CCC2)C1 45374,c1(C(N(CCNC(CC2C(OCC)CC2)=O)CC)=O)ccnn1C1CCOCC1 45375,CC1CC(NC(=O)CCCNC(N)=O)CCN1C(=O)CSC(F)F 45376,c1(-c2ccc(C(=O)NC3C(NC(c4nnn(C)n4)=O)CCC3)s2)cccc(Cl)c1 45377,c1(OC)ccc(F)cc1CC(N1CCN(C(c2ccc(F)s2)=O)CC1CF)=O 45378,N1(C(C(CCN(C)C)O)=O)CC=C(CC(=O)NC(C)(C)C(=O)N(C)C)CC1 45379,CC1(C)CCC=C1C(=O)NC1CN(C(=O)CCC2CCCC(=O)N2)CC12CC2 45380,C(=O)(CC(C(F)F)C(C)(C)C)NC1CCN(C(CCc2ccc(C)s2)=O)C12CC2 45381,N1(C(CCCC(C)C)=O)CC2(C1)SCCC2NC(c1ccc(Cl)cc1)=O 45382,C(=O)(C1=CC2(CCOC2)C1)N(C1CN(C(c2nn[nH]c2Cl)=O)CC1O)C 45383,C(=O)(C(C)CC(=O)OC1CC1)N.C1(OCCSC)CCN(C(=O)CCO)C1 45384,C1(NC(=O)CCc2cncs2)CC12CCN(C(C1CCCOC1)=O)C2 45385,Cc1nn(CC(=O)NCC(C)NC(c2nccnc2Cl)=O)c(=O)n1C 45386,N1(C(CC(C)C2CCCO2)=O)C2CCC1CC(CNC(c1ccc(=N)[nH]c1)=O)C2 45387,N1(C(C2N(C(C)=O)CC(O)C2)=O)CC(NC(c2ccnnc2)=O)C(C)(C)C1 45388,c1(CNC(C(C2CN(C(c3[nH]ccc3C)=O)C2)OC)=O)c(F)cccc1F 45389,N1(C(c2cc3cccc(F)c3s2)=O)CCCC(C2CN(C(C3(F)CC3)=O)C2)C1 45390,c1(C(=O)NC(C(C)C)CNC(C23CC(CN2C2CC2)C3)=O)cnn2cc[nH]c12 45391,C1(C(N(C(C=C)C)C)=O)CCC(CNC(=O)Cc2ccn(CC)n2)C1 45392,C(=O)(C(C)(C)CCC#N)N1CCC(OCC(=O)Nc2ccc(C#C)cc2)C1 45393,C#CC(CC1CCC1)NC(=O)CC1(N(C(=O)CC=CCC)C)CC1 45394,C1(CS(=O)(=O)NCC2CC(C)(C)OC2)CCCC2(CCOC2)O1 45395,Cc1nc(CN(C(=O)CC2(N(C(=O)C(C)C3CC3)C)CC2)C)n[nH]1 45396,C(=O)(C(C)(C)C(=O)N(C)C)NCC1(CNC(c2c(COC)noc2)=O)CCC1 45397,C1(C)(CCC(=O)NCC(C)CN(C(=O)CCOC2CCC2)C)CCC(=O)N1 45398,C1(C(=O)NC(C2CN(C(C(C)(C)OC(C)=O)=O)C2)C)CC1C1CCCC1 45399,c1(C(=O)NC(CC)CNC(C2(Cl)CC2(F)F)=O)cccc(-c2cscn2)c1 45400,C1(CNC(CC2CCCN(C)C2)=O)CN(C(c2cn(C)nn2)=O)C(C)(C)C1 45401,CCC(C)C(O)C(=O)NCCCNC(c1onc(C)c1C)=O 45402,C(=O)(C(CC(C)C)N(C)C)N(CCCCCNC(CCn1ccc(C)n1)=O)C 45403,c1(CC)[nH]nc(C(N2CC(OCCNC(c3cccnc3C(F)F)=O)C2)=O)c1Cl 45404,N1(C(CC2CCN(C)CC2)=O)CC2CCN(C(c3ncc(F)cc3F)=O)C2C1 45405,C(=O)(C(O)CC(N)=O)NC1(CNC(c2c(OC)n[nH]c2)=O)CCCC1 45406,CC1(C)CN(C(=O)CCCC(F)(F)F)C(CNC(=O)CCn2cccc2)CO1 45407,CC1CC(NC(=O)C(=O)NC(C)(C)C(F)(F)F)CN1C(C12CC(F)(C1)C2)=O 45408,c1(C(=O)OC)cc(C(=O)NCC(CNC(c2cc(Cl)c[nH]2)=O)CO)no1 45409,C(=O)(C(C)(O)CCc1ccccc1)NC1CC(NC(C(CC=CC)C)=O)C1 45410,C1(C(=O)NCCC(CNC(CN2CC(C)C2)=O)O)CCCN1C=O 45411,C1(NC(C(N(C)C)C2CC2)=O)CN(C(c2sccc2F)=O)CC(C)(C)C1 45412,CC1CCC(S(C)(=O)=O)CN1c1ncc2ccccc2n1 45413,c1(OC)ccc(F)c(C(=O)NCC(O)CN(C(=O)CC2CCC(O)C2)C)c1F 45414,N12CCCCC(C1)CCC2=O.N1(C(Cc2n(C)ccn2)=O)CCOC(C(N)=O)C1 45415,N1(C(C=C)=O)CCCC2CN(C(c3ccc4cnccc4n3)=O)CC12 45416,C1(NC(C2(C=C)CCOCC2)=O)C2CCN(C(C3(C#N)CCC3)=O)CCC12 45417,CC(C)(C)C(C(=O)NCC1CN(C(=O)CSc2ccccc2)C1)C1CCCCC1 45418,C1(C(=O)OCC)CCCN1S(=O)(=O)N1CCC(C)C1C(F)(F)F 45419,C1(N(C(c2c(COC)cco2)=O)C)CCCN(C(C2CCCOC2)=O)C1 45420,c1(C(C)(C)C)cc(C(=O)NC2CCCC(NC(C3(C)CC=CCC3)=O)C2)ccn1 45421,C1(CNC(=O)Cc2ccsn2)CCN(C(c2ccnn2C2CCCC2)=O)CC1O 45422,C1(C(=O)NC(C(=O)NCC(C2CC2)OC)C2(C)CC2)CC12CCCCC2 45423,N1(C(CN(C2CC2)CC)=O)CCCC1CC(=O)NCC1(C)CCCS1 45424,C1(NC(CCSC)=O)CCN(C(C2CNC(=O)N2C)=O)C12CCC2 45425,CCCCC(CNC(=O)CCCc1sccc1C)NC(C1(C)CC1C)=O 45426,c1(C(N2C(CCCNC(c3c(OC)ccs3)=O)CCC2)=O)cccc2c1CCO2 45427,c1(C(=O)NC2CN(C(c3c(C)sc(Cl)n3)=O)CC2C)ccc2cnoc2c1 45428,c1(OC)cc(-c2cc(C(=O)NCc3cc(F)cc(F)c3)n[nH]2)ccc1F 45429,Cc1nc2cc(C(N3CCC4(CCCN4C(c4ncoc4C)=O)C3)=O)ccc2o1 45430,C1(C(=O)NCC2N(C(CC(C)F)=O)CCCC2)CCCCN1N=O 45431,N(C1CCSc2ccccc21)C(C12C(NC(=O)OC(C)(C)C)C3CCC1C2C3)=O 45432,CC1CN(C(=O)CC2C3CCC(C3)N2C(=O)C(C)OC(C)(C)C)C(C)C(C)(C)O1 45433,c1(C(N2CC=C(CNC(Cn3c(C)nc(C)n3)=O)CC2)=O)cnc2c(c1)COC2 45434,c1(C(=O)NC(CNC(CCCC)=O)C)ccc(OCC)cc1F 45435,N1(C(c2c(CC)ccs2)=O)CCN(C)C(C(=O)NCCc2ccccn2)C1 45436,C1(C(=O)NC(c2cccs2)C)(CF)CCN(C(=O)CNC(=O)C2CC2)C1.CCF 45437,C(=O)(C(C(=O)OC)C(C)(C)C)NC(CC)CNC(C1(n2ccnn2)CC1)=O 45438,c1(SCC)ccc(C(N2CC3CC2C3NC(c2ccc(C(N)=O)nc2)=O)=O)cn1 45439,Cn1cc(C(=O)NCCC2CCN(C(=O)CCCC#N)C2)c(=O)c(Br)c1 45440,NS(=O)(=O)c1ccc(F)c(C(N2CC3(C(=O)NCCCO)CC2CO3)=O)c1 45441,CCC(C)CN=c1[nH]c2c(c(=NCc3nc4c(s3)CCCC4)[nH]1)CCC2 45442,N1(C(C2CC3(CC3)CO2)=O)CCCN(C(=O)C(F)(F)CO)CCC1 45443,C(=O)(CC(Cc1ccccc1)CC)NCCC(=C)CNC(c1cnc(C)[nH]1)=O 45444,C(C(C)(CCO)NC(=O)NC(C1CCOCC1)Cc1nn[nH]n1)OC 45445,c1(C(=O)NC(C2CCN(C(C(CC(C)C)OC)=O)C2)C)ccc(F)c(F)c1F 45446,N1(C(=O)OC(C)(C)C)CC2CCC2(NC2CC(NC(=O)C(Cl)=CCl)C2)C1 45447,N1(C(=O)CSc2ccccn2)CCC(=CCNC(=O)CCC2CC2(F)F)CC1 45448,C1(OCC(=O)N(C(CC)C)C)CN(C(C2(NC(=O)OC)CCC2)=O)C1 45449,N1(C(CC(C)(C)C)=O)Cc2cccc(CNC(=O)CC3CCCCC(=O)N3)c2C1 45450,c1(CCC(N2CC(NC(c3c(OC)ccs3)=O)C2)=O)cccc2ccccc12 45451,S(=O)(=O)(c1cccc(C(=O)NC2CCC2CNC(=O)C(F)=CCC)c1)NCC=C 45452,N1(C(CCC#C)=O)CCOC2(CCN(C(C34CCC(C3)C4(C)C)=O)C2)C1 45453,Cc1ccc2cc(C(=O)NCC3C=CC(NC(=O)C(C#N)C(C)C)C3)[nH]c2c1 45454,c1(C(=O)NCCCC(=O)OCC)ncccc1CC1C(C(NC2=NCCS2)=O)C1 45455,C1(NC(n2cc(C3CCN(C(c4c(CC)csc4)=O)C3)nn2)=O)CCC(CC)CC1 45456,N1(C(c2cc(OC)c(Br)cc2)C(=O)NCCC2CC2)CCC12CCS(=O)(=O)CC2 45457,N1(CCC(=O)NCCC(C)NC(=O)C=CCOC(C)(C)C)CCNC(=O)C1 45458,C(C)(N=c1ccnc(N2CCCC2c2cn(C)nc2NC)[nH]1)c1sc(CC)c(C)c1 45459,Cn1ncc(C(=O)NCC(O)CC(=O)NC2CC2C(C)(C)C)cc1=O 45460,N1(C(CCN(C(CC(C=C)C)=O)CC2CC2)=O)CC2(C1)OC(=O)NC2C 45461,C1(C)(CC)CCCN(C(C2C3CC2N(C(C2CC(=C4CCC4)C2)=O)C3)=O)C1 45462,N1(C(c2ccc(C=CC(=O)OC)o2)=O)CC2OCCN(C(=O)C3CC3)C2C1 45463,CC1CCN(C(C(N2CC(CNC(=O)C(C)(C)CO)C3CC23)=O)C(C)C)CC1 45464,C1(NC(c2ncn(C(C)C)n2)=O)C2CC3C1C3C2C(=O)N(C)CC1CCOCC1 45465,C(=O)(C1=C(Cl)CCC1)N1CC(CN(C(C(CC)(C)C)=O)C)OCC1 45466,c1(OC)cc(C)sc1C(=O)NC1CC(CCNC(C2CCC(C(N)=O)CC2)=O)C1 45467,c1(NC)cc(C(N2CC(c3ocnc3CNC(c3cc(Cl)ns3)=O)C2)=O)n(C)n1 45468,C1(C)(CC)C=C(C(=O)NCCCC(C)NC(=O)C=CCCC=C(C)C)C1 45469,N1(CC(=O)NC(C2(O)CCN(C(=O)CS(C)(=O)=O)CC2)C)C(=O)C(=O)N(C)C1=O 45470,Cn1nc2ccc(Br)cc2c1C1CCCN1C(c1cnc(C2CCCCC2)s1)=O 45471,c1(OC(C(=O)NC2C(NC(Cc3c(C)con3)=O)C2)C)ccc(F)c(F)c1 45472,CS(=O)(=O)c1ccsc1C(=O)NCC1CC(F)(CNC(C2CCCN2N=O)=O)C1 45473,N1(C(CC(CCC)CC)=O)CC2(C1)CN(C(C1(C3CCCO3)CC1)=O)CC2CO 45474,C(C(CC=C)C(=O)NCCC1CC1C(=O)OC)NC(Cn1ncc(C#C)c1)=O 45475,Cc1ccc(C(C2CC2)NC(=O)CC2CCCN(C(c3cnon3)=O)C2)cc1 45476,CC1(C)CCOC1CC(=O)NC1CCN(C(C2CCCC2CF)=O)CC1 45477,C1(CC#C)(NC(=O)C(Cc2cnc[nH]2)NC(C2C3(CC3)C23CC3)=O)CCCCC1 45478,c1(C(=O)NCC2CC2NC(=O)C(O)CC2CCOCC2)cc(Cl)ccn1 45479,N1(C(COCCCCC)=O)CCC2C(CCCN2C(=O)CCC(C)(C)F)C1 45480,N1(CC(=O)NC(C)C)C(=O)C(c2ccccc2)N(C)C1=O 45481,c1(C(c2cccs2)NC(N2C(C(C3CCOC3)=O)CC2)=O)nncn1C1CC1 45482,C1(C(=O)OC)CCN(C(=O)CC(C(F)F)NC(=O)C2CC2)O1 45483,N1(C(C(CC)NC(C)=O)=O)CCC(F)(F)C(NCc2cc(Cl)ccc2Cl)C1 45484,C1(CNC(c2cc(C)sc2)=O)COC(C)(C)CN1C(=O)CCc1cncnc1 45485,C(=O)(N=c1ccn(C)[nH]1)c1ccc(CNC(C2C(C)CC2)=O)o1 45486,CCC(CC)CCCC(=O)N1CCCC(O)(CNC(=O)C(C(C)C)OC)CC1 45487,C(=O)(CS(=O)(=O)CCO)N(CCCNC(c1cn(CC(N)=O)nn1)=O)C(C)C 45488,C1(C(=O)NC(CN(C(c2ccoc2CC(=O)OC)=O)CC)C)C2CCCC12 45489,N1(C(C=CC)=O)CCC(C2CC2)(CNC(=O)CC(C)P(C)(C)=O)C1 45490,C(CCCCC(=O)N1CCC(c2ccccc2C)C1)c1n(CC)ccn1 45491,c1(C(N2CC(OC)CC(NC(COCCC)=O)C2)=O)csc2c1CCC(C)C2 45492,C1(N(C(c2ccc(CCC)s2)=O)CC)CCCN(C(C2(N(C)C)CCC2)=O)C1 45493,Cc1cc(C2CC2)ccc1C(=O)NC(C)CCCNC(=O)C(c1ccnn1C)O 45494,c1(CC(N2CC(N3CCN(C(C4C(C)OCC4)=O)CC3)C2)=O)ccc(F)c(F)c1 45495,c1(NC(c2cn(C(C)C)nc2)C)nc(N2C3CCC2COC3)nc2ncn(C)c12 45496,C1(C(=O)NCC(CNC(C(C)C(F)F)=O)CO)CCC(O)CN1C 45497,c1(C(N2C(C(N(C)CC3(O)CCCC3)=O)CCC(O)C2)=O)ccc2[nH]ccc2c1 45498,C(=O)(C1CCCc2nncn21)N1C(CCNC(C(C)OCCC(C)C)=O)CCC1 45499,CCCC(C(=O)N1CC2CC2(NC(=O)Cc2cncs2)C1)C(C)C 45500,c1(NCC23CC(C(=O)NC(=O)CCN4CCOCC4)(C2)C3)nc2ccccc2s1 45501,c1(C(=O)NC2CC(CNC(c3coc(O)n3)=O)C2)csc2ccc(F)cc12 45502,C1(NC(=O)COC2CCC2)C2CC1N(C(c1conc1-c1ccccc1)=O)C2 45503,C1(CC(=O)NCCN(C(Cc2n(C(C)C)cnn2)=O)C)CCCCN1C 45504,N1(C(C(=O)NCC)CCCCN(C)C)CC2CCC(C1)C2C#N 45505,N1(C(C)C(=O)Nc2ccc(Cl)cc2)CCCN(C(c2cccc(F)c2)CO)CC1 45506,C1(F)(C(=O)NCC(CC=C)NC(=O)C(C)COC)CC2(CCC2)C1 45507,c1(COC(C)C)ccc(C(=O)NC2C3CCN(C(=O)C(C)(C)C#N)C23)cc1 45508,c1(C(=O)NCC2CC(NC(C3(C#C)CC3)=O)C2)cccc(N=[N+]=[N-])c1 45509,c1(-c2onc(C(C(C)C)CCN)n2)c[nH]c2ccc(C(C)C)cc12 45510,C1(NC(CC2C(COC)C2(F)F)=O)CC(Cn2cc(CC(=O)OC)nn2)CC1O 45511,C(CO)(CCCCNC(=O)CC1CCCO1)NC(C1(OCC)CCOCC1)=O 45512,N1(C(C2C(C)OCC2)=O)C2CCC1CN(c1ccnc(C3CCCC3)n1)CC2 45513,c1(C(N(CC(CNC(C(C=C)O)=O)O)C)=O)ccc(CN(C)C(C)C)cc1 45514,N1(C(c2ccc(C)cc2F)=O)CCC2(CC1)CC2C(=O)N(C1CC2CCC1O2)C 45515,C12N(CCCC1(C)C)C2.c1(C(=O)OC)ccc(C(=O)OC)c(OC)n1 45516,Cc1[nH]c(=NC2CC(NC(c3cnc4ccsc4c3)=O)C2)ccc1C#N 45517,N1(C(c2c(CC)cccc2)=O)CC(N(C)C(C2C3CC(F)(F)CC23)=O)C2(CC2)C1 45518,c1(C(N2CCC(N(C(c3sccc3C)=O)CC)C2)=O)cnc(C)nc1C 45519,N1(CC(=O)NC(CNC(COC(CC)CC)=O)C)OC(C)(C)CC1=O 45520,N1(C(c2cc(C)no2)=O)CCC2(CC1)CC2CNC(C1(C2CCC2)CCC1)=O 45521,CCCCCCCC(=O)NC1(c2nnnn2C2COC2)CCCC(C(F)(F)F)C1 45522,c1(CC)ccc(F)c(C(N2CCCC(C)(CNC(c3nnccc3C)=O)C2)=O)c1 45523,C1(NC(C2(CC)CC2(F)F)=O)CCN(C(=O)CCOC(C)C)CC(C)(C)C1 45524,c1(NC2CCC(C(N3CC(C)(NC(C)=O)C3)=O)C2)ccc(C)cn1 45525,CC1C(NC(=O)COc2cc(F)cc(Cl)c2)CCCN1C(=O)CC1(O)CCC1 45526,C1(C(=O)Nc2ccccc2-n2cc(C3CC3)nn2)CCc2ccccc2C1 45527,N1(C(CCC(c2ccc(SC)cc2)=O)=O)CCS(=O)C(C)C1C 45528,N1(CCNC(C(CN(C)C)N(C)C)=O)CCC(NC(=O)C=CC(=O)N(C)C)CC1 45529,N1(C(Cc2cc(C)no2)=O)CCCC(C2CC2NC(c2cncc(C)n2)=O)C1 45530,C(=O)(C1=CCCCC1P(C)(C)=O)NCCCCN(C)C(C1Cc2nccn2C1)=O 45531,c1(C(=O)NCC2CN(C(=O)CC3CCCNC3=O)CCO2)cccc(F)c1O 45532,C1(CC(=O)NC(CC(=O)NC)(C)C)CN(C(=O)CC(C)(C)C)CC12CC2 45533,c1(C(=O)OC)ccc2[nH]nc(C(=O)NCCNC(=O)C(O)C(C)SC)c2c1 45534,C1(NC(N2C(c3ccc(C(F)(F)F)cc3)CC(C)C2)=O)CC(C)N(C)CC1C 45535,C1(C(=O)NC2(OCc3ccccc3)CC2)CCCN1C(C1CCCC1)=O 45536,Cc1cc(C(N2CCCC(CCNC(c3cc[nH]c(=N)c3N)=O)C2)=O)c(C)cn1 45537,C1(C)(C(=O)OC)CN(C(c2ccc(F)s2)C(=O)NCCC2(C)CC2)CCO1 45538,CC(CN(C(=O)CCn1cnnn1)C)C(=O)N(CC(=O)N(C)C)C 45539,N(C(=NCc1ccco1)NC1CCC1)Cc1nc(C(C2CCOCC2)=O)on1 45540,C1(CC)CN(C(=O)Cn2cc(C)cn2)CCC1CNC(=O)CSC 45541,CC1C(NC(=O)C=Cc2cn(C)nn2)CCN1C(=O)CC1OCCO1 45542,Cc1ccc(NC(C2CN(C(=O)CNC=O)CC(C)(C)C2)=O)c(F)c1F 45543,c1(N2CCC(=C)C2)nc(N2CCC(CCN(C)C)CC2)nc2c1ncn2CC 45544,C1(NC(=O)CC2NC(=O)NC2=O)CC12CCN(C(=O)C1=CCOCC1)C2 45545,C=Cc1cncc(C(=O)NCCC2CN(C(=O)C3=C(C)OCC3)CC(C)O2)c1 45546,C(=O)(C(C(=O)OC)OC)N1C(C(C(=O)N(CCCC=C)CC)(C)C)CCC1 45547,C1(CC(=O)NC(CC=C)C)CCCN(C(=O)C(C)(CO)OC)CC1 45548,c1(COC)cc(C(=O)NCC2C(C(N3CC(COC(C)C)C3)=O)C2(C)C)no1 45549,C=C(C)C1CN(C(=O)CC2CCCN(C(=O)Cc3cnns3)CC2)CCO1 45550,c1(CN2C(CNC(=O)C=Cc3cccnc3)CCC2)cc(Br)ncc1Br 45551,N1(C(CC(C)CF)=O)CCN(C(c2cccn2Cc2cccs2)=O)C(C)C1 45552,CCC(O)(CC(=O)NC1CCC1CNC(=O)Cc1ccon1)c1ccccc1 45553,C1(CC(=O)NCCOCCOCCNC(=O)Cc2ccc[nH]2)CC(O)C12CCC2 45554,c1(NC(C(C(C)OC)NC(c2csc(=N)[nH]2)=O)=O)cnn2c1CCCC2 45555,C#CCC(C)(C)C(=O)N1CC2(CNC(=O)C(F)(F)CC)CCC1C2 45556,C(CC(C)C)(C(=O)NCCC1(OC(C)=O)CN(C(=O)C(=O)NC(C)C)C1)OC 45557,c1(C(=O)NC2CC(CNC(CCNC(C)=O)=O)C2)ccn2nnnc2c1 45558,N1(C(C(C)CNC(=O)CN(C)C)=O)CCCC(O)(CO)C1 45559,C1(C(=O)NCCN(CCC)C(C2(C)C(C)(C)C2(C)C)=O)CC2CCC(C1)C2O 45560,CC1CN(C(=O)CC(C)c2ccccc2)CC1NC(=O)CC(F)(F)Cl 45561,c1(CNCC23C(CN(C(C4CCCSC4)=O)C2)C3)cccc(F)c1Cl 45562,O=C(C1=C(Cl)CCCC1)NCC1(NC(C23CSCC2C3)=O)CCOCC1 45563,N1(C(c2oc(C)c(CO)c2)=O)CCN(C(=O)CN2CC3CC3C2)C(C)C1C 45564,C(=O)(C1=CCC(F)(F)CC1)N1CC(CNC(=O)C=CC2CCCO2)OCC1 45565,CP(C)(=O)CCC(=O)NCC1CCOC1C(=O)NCC#CC#CCO 45566,C1(CC(=O)NC2(c3onc(C)n3)CC2)C2CCC1CN(C(C1CCCCO1)=O)C2 45567,C1(NC(C2CCC=CO2)=O)CN(C(=O)CCC2CCCO2)C2CCCCC12 45568,c1(C(N2CC(C)(NC(=O)Cc3cccnc3)C2)=O)cncc(N)c1 45569,N#CC1(C(=O)NCc2csc(C(N3CCC(C4CCCO4)C3)=O)c2)CCCC1 45570,C1(F)(CNC(=O)CCCN2CCCCC2)CCN(C(=O)CC2CCC(=O)N2)CC1 45571,C#CCC(C)(CC)C(=O)NCC(C)CNC(c1nccn1C(C)C)=O 45572,C1(CCNC(C(F)=CCC)=O)CN(C(=O)CCN2C(=O)CCC2=O)CC(C)O1 45573,c1(NC(c2n(CCCSC)nnn2)c2nc(C)cs2)ccc(Cl)c(NC(C)=O)c1 45574,N1(Cc2nc(C)sc2)CCCC(NC(=O)N(C)CC2COCCO2)C1 45575,N1(C(CP(C)(C)=O)=O)CCN(C(=O)CCCn2cccn2)CC1c1cn[nH]c1 45576,C(C)(CCC(=O)N1CCC(C(C(C)C)NC(=O)COCCN(C)C)CC1)SC 45577,c1(C(=O)NC(C)CCCNC(=O)C2CC2)cnccc1C(F)(F)F 45578,c1(CNC(=O)COC2CC(F)(F)C2)n[nH]c2c1CN(C(=O)C1=CCOC1)CC2 45579,N1(C(c2cc(OCC)cc(F)c2)=O)CCC2(CCCN(C(=O)C(C)(C)CF)C2)C1 45580,c1(SC)ccc2c(c1)CC(C)N2C(c1c(NC(=O)OC(C)(C)C)cccc1)=O 45581,Cc1ccc2oc(C(=O)N(C3CN(C(c4cn(C)c(C(F)F)n4)=O)C3)C)cc2n1 45582,C12(C(N(CCN(C)C)CC)=O)CCC(CC1NC(c1cc(OC)n[nH]1)=O)C2 45583,Cc1cc(C(N2CCN(C(=O)C=CC(=O)OC(C)(C)C)CC2C)=O)ccc1[N+](=O)[O-] 45584,CC(CCNC(C1(CNC(=O)CC2CCC(C)C2)CCCC1)=O)C(C)(C)C 45585,Cc1cccc(Cl)c1S(=O)(=O)N1CCN(Cc2cc[nH]n2)C2CC12 45586,C1(C(=O)NC(CNC(C(C)SCC)=O)CC(C)C)COC2COCC12 45587,C1(C(=O)NC2CCN(C(C=CCC)=O)C2C(C)C)CCc2nnc(O)n2C1 45588,C1(C(=O)NC2CC(NC(C(CCC)NC(C)=O)=O)C2)CC2CCCC(C1)C2 45589,n1(CC)nc(C2CC2)cc1S(=O)(=O)NC1(CC2CC2(Cl)Cl)CCCC1 45590,N1(C(c2cnc(NC(C)=O)o2)=O)CC(NC(=O)C(C)(C)N2CCCCC2)C2CC12 45591,C1(C(N2CCOC(CC3CC3)C2)=O)CCOCCN1C(=O)CC1CC=CCC1 45592,C1(Cc2nc(C(C)Sc3ccccc3)n(-c3ccccc3)n2)CCC(F)(F)CC1 45593,N1(C(CC(CC)C)=O)CC(NC(C2CC3CCC2CC3)=O)CC(C)(C)C1 45594,c1(-c2scc(C(=O)NCCCCC#C)n2)cnn2c1CCCC2 45595,N1(C(=O)CN2CC3CCC2C3)CC2CC(NC(C34CSCC3C4)=O)CC(C2)C1 45596,CCC(C(=O)NC1CCSC12CN(C(c1cnn(C)c1C)=O)C2)C(C)(F)F 45597,C12(C(N3CCC(N(CC#C)C(C4CCC(C)O4)=O)CC3)=O)CCC(N=[N+]=[N-])C1C2 45598,CCCCCC(O)C(=O)N1CC(O)(C(C)NC(=O)CN2C(=O)CNC2=O)C1 45599,CS(=O)(=O)c1ccsc1C(=O)NC1C2CC1N(C(C1(C#N)CC13CCC3)=O)C2 45600,C(=O)(C(O)C(C)(C)C)NCCn1cc(C(N(CC#C)C)=O)nn1 45601,C1(CN(C(=O)CN2CCOCC2=O)C)CCCN(C(C2CCCS2(=O)=O)=O)C1 45602,c1(C(=O)NCC(=O)NC23CCC(C2)N(C(C2CCO2)=O)C3)cc(Cl)ccc1Cl 45603,C(=O)(C1=COCCO1)N1CCC(CCCCCNC(C2CCCS2)=O)CC1 45604,c1(C(=O)NCC2N(C(C(C)(Cl)Cl)=O)CC2)cc(C2CC2)oc1C1CC1 45605,Cc1cccnc1C(=O)NC1CCCN(C(=O)C(O)c2ccsc2)C1 45606,C1(C(=O)NCCCNC(C(C)Oc2ccc(F)cc2)=O)CCc2ncccc2C1 45607,C1(C(=O)OCc2nnnn2-c2ccccc2)CCc2cc(F)ccc2O1 45608,CCCC(C(=O)N1CCCC1(C)c1cn(Cc2cnco2)nn1)OC 45609,N1(C(c2c(C)occ2)=O)CCCCC1C(=O)CCc1cn(-c2cccc(Cl)c2)nn1 45610,CC(C)(C)C(C)(C)C(=O)NC1CCC(NC(c2[nH]nnc2C2CC2)=O)CC1 45611,C1(C(=O)NCC=CCNC(C(c2c(F)cccc2F)C)=O)CC2CCCC(C1)C2 45612,c1(C(=O)NC(C(C)NC(c2c(COC)cccc2)=O)(C)C)nccc(OC)c1F 45613,c1(C(C)(F)F)cncc(C(=O)NC2(C)CC(NC(=O)C(F)C3CCOC3)C2)c1 45614,C1(C(N2CC3(C(NC(c4c(C)nsc4)=O)CCC3)C2)=O)Cc2ccccc2CO1 45615,Cc1ccc(C=CC(N2CC=CC(C(=O)NCC3CCOC3C)C2)=O)cc1 45616,C(C1COC(C)(C)O1)=CC(=O)NC1CC(C)(NC(C(C=C=C)C)=O)C1 45617,c1(CC)cnc(Cl)nc1N(C)CCN(CCOC)C(C1CCC2CC2C1)=O 45618,CCCC(CCC)=CC(=O)NC1CN(C(=O)Cc2ncccc2C)C2CC12 45619,Cc1ccccc1C(=O)NC1CCOC(C2CCN(C(c3cncs3)=O)CC2)C1 45620,c1(C(N2CCC(CNC(C(C)OC)=O)(CO)C2)=O)c[nH]nc1[N+](=O)[O-] 45621,N1(C(CNC(CCC)=O)=O)CCC(NC(C2CC2c2c(F)cccc2F)=O)C(C)C1 45622,c1(CC(C(N2CC(n3cc(CN)nn3)(C(=O)OCC)C2)=O)C)ccc(O)c(F)c1 45623,Cc1ccc2nc(C(=O)NC3(CNC(c4nc(C)oc4C)=O)CC3)c(N)n2c1 45624,c1(OC(CC)C(=O)NCCNC(=O)CC(F)F)ccccc1C(C)C 45625,C=C(C)CC(C(=O)NC(c1cncs1)C)NC(C1CC2CC(=O)C1O2)=O 45626,C(N=c1[nH]c(=NCCc2csc(O)n2)[nH]c2cc[nH]c12)c1nccc(NC)c1 45627,C12(C(=O)NCCC(O)C(F)F)CCC(CC1)N(C(C1(CO)CCCCC1)=O)C2 45628,C(C(C(=O)N(C)CC1(CO)CC1)NC(=O)CC1CCC1)SC 45629,c1(CC(=O)NC2C3CN(C(c4c(C)cc[nH]4)=O)C2C3)ccc2c(c1)CC(C)O2 45630,C1(C(=O)NC(CNC(c2cc(Cl)c(Cl)[nH]2)=O)CO)CCC2CC2CC1 45631,c1(C(=O)NC(CC=C)CNC(=O)C(c2ccc(Cl)cc2)O)c[nH]c2nccc-2c1 45632,c1(OC(C)C)cnc(C(=O)NC2CCC(CNC(c3cc(N)ccn3)=O)C2)cn1 45633,C(=O)(C1=CCN(C(c2cc(O)cs2)=O)CC1)NC(CC(CC)C)CO 45634,CCCC(CC(=O)NC1CCC(OC)CC1)NC(c1cc(C#N)cn1C)=O 45635,c1(OCC(=O)NCCCN(C(=O)CCc2ccncc2)CC)cnn(C)c1 45636,C(=O)(CS(F)(F)(F)(F)F)NCC1(C)CCN(C(C(C)OC)=O)C1 45637,CN1CCC(NC(=O)CC(C)(C)C#N)C12CCCN(C(C1CSC1)=O)C2 45638,Cc1c(C(=O)NC(C)(C)CNC(=O)CC2(O)COC(C)(C)C2)cc(N)cc1O 45639,c1(OCC)ccc(C(=O)NCc2cccnc2CNC(=O)C(C(C)C)OC)cn1 45640,Cc1ccnc2ccc(CN3CCC(CCNC(=O)COc4ccsn4)C3)cc12 45641,c1(C(=O)NC2(C)CC(NC(=O)CCCc3cccs3)C2)ccc([N+](=O)[O-])cc1 45642,N1(C(C(c2ccc(CC)s2)=O)=O)CCN(C(c2ccon2)=O)CC1C 45643,C1(CC)CC2(CCN2C(c2cn(C)nc2Cl)C(=O)NC2CCCC2)C1 45644,C1(C(=O)NCC(CC)C)CCN(C(c2cc(C)cc(C)c2)=O)CC1(C)C 45645,N1(C(CC(C)O)=O)CC2CCC(N(C(=O)CCc3cnn(C)c3)C)C2C1 45646,CCC(C(=O)NC(CNC(c1cccc2c1CCO2)=O)CO)C(C)(F)F 45647,c1(CC(=O)NCC=C2CCN(C(C3CN(C)C(=O)C3)=O)CC2)ccnc(Cl)c1F 45648,C1(C(=O)NC2(CNC(c3csc4nccn34)=O)CCCC2)CCCCC12CCC2 45649,CCCCCCC(C)NC(=O)C(=O)Nc1cc(-c2ccccc2)nn1CC 45650,N1(C(c2cncc(NC)c2)=O)CCC(CCNC(c2coc(Cl)n2)=O)C(F)(F)C1 45651,Cc1c(C(=O)NCc2csc(CNC(=O)C(C)C3CC3)n2)sc2cccc(F)c12 45652,C=CCCCCC(=O)NCC(C)NC(=O)CCCSCc1ccccc1 45653,CS(=O)c1ccc(CC(N2CCC(NC(C3CC(C)(F)C3)=O)C2)=O)cc1 45654,N1(C(C2CC(NC(=O)C=CCN3CCC3)C23CCC3)=O)CCc2nc(O)[nH]c2C1 45655,N1(C2CCN(C(C(C)(C)OC)=O)C2)CCN(C(=O)CC2(C(F)(F)F)SCCS2)CC1 45656,c1(C(C(=O)NCCC(C)NC(=O)CC2OCCC2(C)C)O)cccc(Cl)c1 45657,C1(C(=O)NC2C=CC(C(=O)NN3CC(CC4CC4)C3)C2)CC2(C1)CC2(F)F 45658,C1(C(=O)Nc2ncc(Br)cc2OC(F)(F)F)CCc2n[nH]cc2C1 45659,c1(CC)ccc(NC(c2c[nH]nc2CNC(c2cnc(C)nc2C)=O)=O)c(F)c1 45660,Cc1nccnc1C(=O)N(C)CCNC(=O)CC(C)Cc1cccc(F)c1 45661,N1(C(c2ccc(COC)o2)=O)C2CCC1(CNC(C1CC(SC)C1)=O)CC2 45662,C12(CC(=O)NCCC3CCN(C(=O)CCc4ccncc4)C3)CCC(CC1)OC2 45663,Cc1c(C(N2CCCC(N(C(=O)C#CC3CC3)C)C2)=O)cc(N)cc1O 45664,C(CC1CCCO1)N=c1[nH]c2ccc(S(=O)(=O)N3CCCC(CO)C3)cc2[nH]1 45665,CC1(C)COC(C(=O)NCC2CCC(C(=O)NCCCN3CCCC3=O)CC2)C1 45666,C(=O)(C(C)(O)C1CC1)NCC(C)CN(C)C(c1n[nH]cc1Br)=O 45667,N1(CCCc2ccc(C)cc2)C(=O)CN(Cc2ccc(F)cc2F)C1=O 45668,C1(F)(C(N(CC)Cc2cccs2)=O)CCN(C(=O)Cc2nccn2C)C1 45669,n1(C(C)C)ncc(Cl)c1C(=O)NCC1CCC(F)(CNC(C2(C(N)=O)CC2)=O)C1 45670,N1(C(C(C)(C)n2cc(Cl)cn2)=O)CC2C(C(=O)NCCC3(C)CC3(F)F)C2C1 45671,C1(CCCC)CN(C(C2CC=CCC2C(=O)OC)=O)CCN1C(=O)C(C)CC 45672,c1(CC(=O)N(C(CNC(CSC)=O)C)CC)cc(Br)ccc1Cl 45673,c1(C(=O)NC2CCC(N(C(c3ccc(COC)o3)=O)C)C2)nc(C)ccc1F 45674,C(CC(=O)N=c1cc[nH]cc1O)C1N(Cc2c(OC)nccc2)CCC1 45675,C1(COC)(Nc2ccccc2C(=O)NCC(C)C(C)(C)C)CC2(C1)OCCO2 45676,c1(OC(C)C(N2CC(O)(C(C)NC(=O)C3=CCC3)C2)=O)cccc(F)c1 45677,c1(C2CCCN(C(c3ccsc3Br)C(=O)NCCC#N)C2)ccc(F)c(F)c1 45678,n1(CC)cnc2c(NCCCC(C)NC(=O)COc3ccon3)nc(Cl)nc12 45679,CCCCS(=O)(=O)CC(=O)NC1CN(C(=O)COc2c(Cl)cccc2Cl)CC1C 45680,C(CCc1ccco1)(C(C)(C)C)NC(C(COCC)n1cc(C2(C)CC2)nn1)=O 45681,C1(CNC(C2(SC)CC2)=O)CCCCN(C(c2ccc(N)cc2Cl)=O)C1 45682,CN=c1[nH]cc(C(=O)NC(C(N2CC3C(CO)C3C2)=O)C2CCC2)o1 45683,c1(C(=O)NCC2CC(C)(C)CN2C(c2cnccn2)=O)cc2ccccc2[nH]1 45684,c1(SCC(N2CC3C(NC(Cc4c(CC)con4)=O)(C3)C2)=O)cc(F)ccc1F 45685,Cn1ccc(C(=O)NCC2CCN(C(C3(n4cc(Br)cn4)CC3)=O)C2)cc1=O 45686,C1(C(=O)NC(C)(C)CNC(=O)CC2SC(=N)NC2=O)CS(=O)(=O)CCO1 45687,c1(OC)cc(C(N2CC3CC(NC(C4CCOC4)=O)C3C2)=O)ccc1C 45688,Cc1ccc(C2(CNC(=O)Nc3cccc(C(F)F)c3)CCC2)c(F)c1 45689,N1(C(c2ccc(C)cc2C)=O)CCCC(F)(CNC(=O)C(O)C(C)(C)C)CC1 45690,C1(C(=O)NCc2cc(C)nc(C)c2)N(C(=O)CC2CC(C)C2)CCCC1(C)C 45691,N1(C(C(CCNC(C(CC=C)NC(C)=O)=O)O)=O)CCC12CN(C)C2 45692,c1(CC)ccnc(C(=O)NC(CNC(C2CC23CC(OC)C3)=O)CC(C)C)c1 45693,C1(CNC(CCC=C)=O)(C(=O)OC(C)(C)C)CCN(C(=O)C(O)CC(=O)OC)CC1 45694,N1(C(CCC(=C)Br)=O)CC2CC(C1)CN(C(=O)CCC(CC)OC)C2 45695,CCCC(C)(C)C(=O)N1CCCCC(CNC(=O)C(O)CCSC)C1 45696,C1(CNC(C2CC(SC)C2)=O)CCCCCN1C(c1cc(N)ccc1C)=O 45697,c1(OCC)ccc(C(=O)NC2CCCCC2CNC(c2ccnnc2O)=O)nn1 45698,C12(C(=O)NC3C(CNC(C(OC)OC)=O)C3)CC3CC(F)(C1)CC(F)(C3)C2 45699,c1(-c2cc(CN(c3cc(C)cc(C)c3C)C)cc(C)c2)ccc2cncn2c1 45700,C(C)(CC(=O)NC(c1nocc1C(=O)N(C)Cc1ccn(C)n1)C)SC 45701,Cn1ncc([N+](=O)[O-])c1N1CC(CCNC(c2cc(-c3ccncc3)no2)=O)C1 45702,CC12CC(CCO1)N(C(C1(NC(c3ccc(C#N)s3)=O)CC1)=O)C2 45703,n1(CC(=O)N(CC(C)(C)NC(C2C(OCC)C2)=O)C)c(C)cc(O)cc1=O 45704,N1(S(CCOC)(=O)=O)CCC2(CCN(Cc3ccn4ccnc4c3)CC2)CC1 45705,C(=O)(CCCS(N)(=O)=O)N1CC(NC(C2(C#C)CCC2)=O)C(C)C1 45706,c1(C(=O)NCC2(C)C(NC(CP(C)(C)=O)=O)CCC2)ccc2nsnc2c1 45707,Cc1cnc(C(C)(C)NC(C2CS(=O)(=O)C2)=O)s1 45708,n1(CC)ccc(C(=O)N(CCCNC(c2cc(C)cs2)=O)CC2CCCC2)n1 45709,C1(C(=O)NCCN(C(=O)CC2CCC(C)CC2)CCOC)CCN(C)C(C)C1 45710,C(C(C)CC(F)(F)F)N(C(N1C(CCC(C)C)CCC1)=O)CCO 45711,Cc1ccc(F)cc1C(=O)NCC(O)CCNC(c1csc(C(F)F)n1)=O 45712,C#CCC(CC)NC(=O)CCNC(C1(CO)CCCC1)=O 45713,C1(NC(CC2C(=O)NCC2)=O)CCN(C(C2CC3C=CC2C3)=O)C12CCC2 45714,C1(CN(C(C(n2c(C)ccn2)C)=O)C)CN(C(=O)CC2CCCC2)CC12CC2 45715,c1(C(=O)NC2CCCN(Cc3ncc(C)nc3)C2C)cnc2c(C)cccc2c1 45716,S(=O)(=O)(c1cccnc1N1CCS(=O)CC1)NCC(c1ccc(F)cc1)CC 45717,N1(C(C=C(CC)CC)=O)CCN(C(c2cc(N)c(Cl)cn2)=O)C2(CC2)C1 45718,N1(C(c2coc(Br)n2)=O)CC(F)(F)CC1CNC(C1(F)CCOC1)=O 45719,C1(NC(c2cn(C)nn2)=O)CCN(C(=O)C(=Cc2cccc(F)c2)F)C12CC2 45720,C1(OCCC)CN(N2CC(OCCN(C)CC)C2)C1 45721,CN1CC2(CC2)CC1C(=O)NC1CC(O)CN(C(C2(C3CC3)CC2)=O)C1 45722,CCCCCCCCNC(=O)CC1CC(F)CN1C(c1cc(F)c[nH]1)=O 45723,c1(SC)cncc(C(=O)NCC=C2CCN(C(=O)CCn3cc(C)cn3)CC2)c1 45724,C#Cc1cc(OC)cc(C(=O)NC(C)(C)C(C)CCC)c1 45725,C1(NC(CCCOCC=C)=O)CCC(CC(=O)NCc2ccc(C)s2)CC1 45726,c1(C(C(N2CCC(NC(C34CC(F)C3C4)=O)C2)=O)O)ccccc1Cl 45727,C1(C)(C(=O)NCCc2ccc(C)nc2)CN(C(c2ccsc2)=O)C(C)(C)C1 45728,N1(C(Cc2c(C)noc2)=O)CCC(NC(c2cccnc2)=O)C1Cc1ccccc1 45729,C1(NC(C2CC3CCC2CC3)=O)CN(C(=O)C(C2CCCCC2)O)CC2(CC2)C1 45730,C1(C(N(C(C(=O)NC(c2cn(C)nc2)CO)CO)C2CC2)=O)CCCCNC1=O 45731,Cc1ccccc1C1(C(=O)NC2COCC2NC(C23CCC2C3)=O)CCOCC1 45732,C12(C(=O)NC3CC(NC(c4nc(CCC)oc4)=O)C3)COC(CCO1)C2 45733,c1(NC(C2(Cc3cncc(C)c3)CC2)=O)nn(C)c(Cl)c1-c1nn[nH]n1 45734,N1(C(CNS(CCCOC)(=O)=O)=O)CC2CC1CC2NC(c1ccc[nH]1)=O 45735,C(C)(C)(C(F)(F)F)OCC(=O)N(C(C)CN(C(=O)Cn1cc(C2CC2)cn1)C)C 45736,N1(C(C=CC2C(C)C2(Cl)Cl)=O)CC2(CCN(C(c3cc(C(N)=O)no3)=O)C2)C1 45737,c1(OC)cc(NCC2CC(NC(C3CN(C)C(=O)N3)=O)C2)nc(OC)n1 45738,C=C1CCN(C(=O)CC2(C=C)CN(C(=O)C(O)C3CC3)C2)CC1 45739,C12(OC)CN(C(=O)OC3CCCC(CS(=O)(=O)NC(C)(C)C)C3)C(CO)(C1)C2 45740,C1(NC(C2(C=C)CCC2)=O)CCN(C(c2c(C(F)(F)F)cnn2C)=O)CC1F 45741,Cc1c(CNC(C2CCCN2C(=O)C(C)(O)C2CC2)=O)nnn1C 45742,Cc1nn(C)cc1CN(C(=O)C(C1(O)CN(C(C2CC2C(N)=O)=O)C1)F)C 45743,N1(C(CC(=C)C)=O)CC(O)CC1CNC(C1CC(=O)N(c2ccc(C)cc2)C1)=O 45744,C(=O)(C1=CCCCCC1)N1C(C)CC(CC(=O)NCC2COCCOC2)C1 45745,C1(NC(CCC(C)OCC)=O)CCN(C(=O)C(COC)COC)CC12CCC2 45746,C(=O)(C1=C(C)OCCS1)N1CCCC(C(=O)NC2(SC)CCC2)C1 45747,N1(C(C(=O)NCC(C)NC(=O)C(N2CCC(C)C2)=O)C)CCOCC1 45748,C1(OC)CC(NC(=O)CCCCCc2ccccc2)CN(C(=O)CC(C)F)C1 45749,N1(C(C(CC)C(C)C)C(=O)NCCSC)CCC2(CC1)C(C)(C)C21CCC1 45750,CC#CCCC(=O)NCC(C)(O)CNC(C1COCCN1CC(F)(F)F)=O 45751,N1(Cc2c(OC)cccc2)CCc2sc(-c3cncc(F)c3)nc2C1 45752,c1(CN2C(c3cc(C)nn3C)CCC2)cc(C2CC2)[nH]c(=N)n1 45753,C12(C(N(C)CC3CCN(C(=O)C(O)CF)C3)=O)CCC(C(F)F)(CC1)CC2 45754,CON(CCO)C(=O)C(CCOCCO)NC(c1ccc(C)cc1O)=O 45755,N#Cc1ccc(NC(C23CC2CN(C(c2cc(O)ncn2)=O)C3)=O)c(I)c1 45756,C1(C(N2CCC(CC)C2CNC(c2ccncc2Cl)=O)=O)CC2CCC(C1)C2O 45757,c1(C(N2C3CCC(NC(C=C(CCC)CCC)=O)(C3)C2)=O)cccc2ccnn12 45758,c1(C(=O)NCCC(C)N(C(c2[nH]cc(C)c2C)=O)C)onc2ccccc12 45759,c1(C(=O)N(C2CC3CC3C2)c2ccccc2)cccc(C(F)(F)F)c1Br 45760,CC(C(=O)NCC1CN(C(=O)Cc2nnc(S)n2C)CCO1)S(N)(=O)=O 45761,C12(NC(C(C)Cc3ccc(Cl)cc3)=O)CCC(C1)N(C(=O)CCC1CCCC1)C2 45762,O=C(C#CC1CCC1)NCC1(CNC(c2ccc(C(F)F)o2)=O)CCC1 45763,Cc1cc(Cl)c(C(=O)NCC2(O)CN(C(=O)C(c3ccncc3C)C)C2)c(Cl)c1 45764,Cc1cn2c(CC(=O)NC(c3ccc(F)cc3)CNC(c3ccsn3)=O)csc2n1 45765,C(CC1=CCN(C(c2n[nH]c(C)c2N)=O)CC1)NC(C1(CC)CCOCC1)=O 45766,C1(NC(CC2(C)CC2)=O)CCN(C(C2CC3(C2)CC3(F)F)=O)CC1F 45767,C#Cc1cc(CNCCNC(=O)C(C)c2cccs2)cc(F)c1 45768,N1(C(CCC=C(C)C)=O)CC(NC(C2(CO)CCCC2)=O)CC12CCOC2 45769,C(=O)(CC(C)C(C)(C)NC(=O)CC1CCCSC1)N1CCC(C#C)(O)C1 45770,N1(C(c2cn(C)nc2-c2ccncc2)=O)CC2CCCC1(CO)C2 45771,C1(NC(C(CC)Sc2ccccc2)=O)CCOCC1NC(C1(CC=CC)CC1)=O 45772,c1(C(C23CC(CO2)C3)N(C(C(=O)NCC(CSC)(C)C)=O)C)ccccc1Br 45773,c1(OC)ccnc(NCc2c(C(=O)CN3CC(CO)OCC3C)cccc2)c1 45774,C1(c2c(C(=O)OCC)nco2)CCCN(CCCCCn2cc(C(C)OC)nn2)C1 45775,Cc1nc(C(N2CC(OCC3CCN(C(=O)Cc4ccccc4)C3)C2)=O)c(C)[nH]1 45776,C(=O)(CCCC(C)(C)C)NC(CC#C)CC(=O)NC(CC1CC1)CC 45777,C1(CNC(C2(C(=O)NC)CCC2)=O)CC2CN(C(C3CCOC3)=O)CC12 45778,CC(CNC(=O)C(=O)NCC(F)F)(C1CC1)NC(=O)COC1CCOC1 45779,C1(CC#C)(C(N2CCCC2CNC(C2COCCO2)=O)=O)CCCCC1 45780,O=C1CC2(CCN(C(C3CC(NCc4nc(O)n[nH]4)C3)=O)CC2)CN1 45781,C12(CNC(c3c(OCC)nccc3)=O)CCCC1N(C(=O)CSC(F)F)CCC2 45782,N1(C(COC)=O)CCN(C(C2CCn3cc(C)nc3C2)=O)C2COCC12 45783,C1(NC(C2(OC)CC2)=O)CC(C)N(C(c2cccc(OCC3CC3)c2)=O)C1 45784,c1(C(=O)NCC2CCN2C(=O)COc2ccsc2)ccncc1F 45785,C12(C(=O)NCCC3OCCN(C(C4CN(CC)C(=O)C4)=O)C3)CC(C1)S(=O)(=O)C2 45786,c1(C(N(CC(C)(C)CNC(=O)CC2(COC)CC2)CC)=O)cn2cc(C)sc2n1 45787,Cc1ccc(C(N2CC3CCC(C2)N(C(c2conc2C)=O)C3)=O)c([N+](=O)[O-])c1 45788,c1(C(=O)NC2(CO)CN(C(c3ccnc(C)n3)=O)C2)cccc2nccn12 45789,C1(CNC(=O)NC(C2(CCO)CC2)C)CC(OC(C)(C)C)C1 45790,N1(C(C(C#C)(C)C)=O)CCC2C(CCCN2C(c2ccc3c(c2)CCOC3)=O)C1 45791,c1(C(=O)OC)ccc(CC(N)C(N2CCN(Cc3ccsc3)CC2)=O)cc1 45792,C1(C(=O)NCC2CN(C(c3cc(OC)n(C)n3)=O)C2)CCCC(C)(C)O1 45793,Cc1nn2ncccc2c1C(=O)NCCC(C)N(C(=O)CC(C)(C)F)C 45794,CCC(CNC(c1nccnc1C)=O)(CC)C(=O)NC1CC(C)(C)OC1=O 45795,Nc1nc(C(N2CC3CC(NC(c4cc(CCCO)on4)=O)C2C3)=O)ccc1O 45796,c1(CCC(=O)NC2CC(F)(CNC(c3nc(COC)sc3)=O)C2)ccc(Cl)nc1 45797,C1(C(N(C)CCC2CCOCC2)=O)(CO)CCN(C(=O)CC2CCOC2=O)C1 45798,Cc1c(C(N2CCOCC2C(N2CCOCC2CO)=O)=O)ncn1C 45799,C(C(=O)N1CCC1C(=O)NCCc1ccnc(C)c1)(C(C)C)NC(C)=O 45800,Cc1ccc(C(=O)NC2CC(NC(C3(N(C)C)CC3)=O)C23CCC3)c(Cl)c1Cl 45801,C=C(Br)CCC(=O)NC1CCC(CNC(=O)C=C(C)C)C1 45802,C1(NC(=O)Nc2ccc(-c3[nH]c(=NC)sc3)cc2)CCC2CC2CC1 45803,C(=O)(C(=O)C(C)CC)N(C(C(=O)NCC(C=C)(C)C)C)CC 45804,c1(C(=O)NCCC(=O)NCCOC2CC2c2cscn2)ccoc1C1CC1 45805,C1(O)(CN(C(=O)CC2CC23CC3)C)CCN(C(=O)Cc2cccc(Cl)c2)C1 45806,C(=O)(CCC(=O)NCC1CN(C(=O)CN2C(C)CCC2C)CC1C)NC 45807,N1(C(Cc2ccc(C)s2)=O)CC(NC(c2cc(C(N)=O)n(C)n2)=O)CC(C)C1 45808,CC1CN(C(c2ccc(CN(C)C)o2)=O)CC1CNC(c1ccsc1C#N)=O 45809,CC1CC(C(N2CCC(NC(c3nsnc3O)=O)C(C)C2)=O)CC(C)O1 45810,S(=O)(=O)(CCC(=O)NC1CC(NC(=O)C(O)C(C)(C)C)C(O)C1)NC 45811,N1(C(COC(CC)C)=O)CCC1C(=O)NCCC1(CO)CC1 45812,c1(NC(C2CC(NC(c3nc(CC)oc3C)=O)C(O)C2)=O)ccc(O)c(CO)c1 45813,N1(C(c2c(SC)cccc2)=O)CC2CCN(C(=O)C(F)n3cccn3)CC2C1 45814,Cc1ccc2c(N3CCCC4(CC4)C3)nc(=NCC3CCOC(CO)C3)[nH]c2c1 45815,c1(C(=O)NC2CCCC(NC(C3N(CC)CCC3)=O)C2)cc(C#N)oc1C 45816,CC1CCc2ncc(C(N3CC4CC(C3)CN(C(=O)CC#N)C4)=O)n2C1 45817,N1(C(c2nc(N(C)C)oc2)=O)CCCC1(C)CNC(=O)CCS(C)=O 45818,C1(CNC(C(CC)C)=O)CCN(C(=O)Cc2cccc(NC(C)=O)c2)C1(C)C 45819,C12(C(=O)NCC(N(C(=O)C3=CCCSC3)C)C3CC3)CC(C)(C1)OC2(C)C 45820,C1(C(N2CC3C(NC(C(=O)NCCOC)=O)C3C2)=O)CC(C)(C)CCO1 45821,C1(CC)CCCC1C(=O)NC12CC(C(N3CCC3(C)C(=O)NC)=O)(C1)C2 45822,Cc1ccc(CCC(N2CC3CC2(CNC(C2CC2C)=O)C3)=O)c(C)c1 45823,CC1CN(C(=O)CC2CN(C)C2)CCN1C(c1coc(C2CCC2)n1)=O 45824,Cc1ccc(C(=O)NCC2(O)CN(C(=O)C(C)N3CCC3)C2)o1 45825,c1(C(N(CCCCN(C(C(c2ccnn2C)C)=O)C)C)=O)cc(O)nn1C 45826,C1(N(C(CSCC)=O)C)CCC2(CC1)CCN(C(=O)CC1CCCC(C)(C)O1)C2 45827,c1(C(N2CC(C(=O)OC)C2(C)C)=O)cc(F)cc2nc(S)[nH]c12 45828,c1(C(N2CC(NC(C3CCCN(C(=O)OC)C3)=O)C2)=O)ncc(Cl)cc1F 45829,N1(C(CC2CCN(C(CC(COC)(C)O)=O)C2)=O)CC2(COCC(=O)N2)C1 45830,c1(NC(C(c2c(Br)cn(CC)n2)N(C(C)C(=O)OC)C)=O)cccc2cnccc12 45831,c1(OC)cc2cc(C(=O)COC)sc2cc1N(C1CCNCCC1C)C 45832,n1(C2(N3CC(C(N4CCC4C(F)F)=O)C3)CC2)cc(Br)nn1 45833,c1(CNC(N2CC(C)(CCc3ccccc3)C2)=O)ccc(Cl)cc1F 45834,c1(C(N(C2CCN(C(c3ccco3)=O)CC2)CC#C)=O)csc2c1CCCC2 45835,c1(SC)cc(C)ccc1C(=O)NCC(C(C)C)NC(=O)C(C)C(F)F 45836,N1(C(C2N(C(C)=O)CCOC2)=O)CCCN(C(c2ccc(Cl)o2)=O)CC1C 45837,n1(CC)cc(-c2n[nH]cc2C(=O)NCC(C)N(C(=O)C(C)NS(C)(=O)=O)C)cn1 45838,C1(NC(c2c(CCC)occ2)=O)CN(C(c2ccnc(S)c2)=O)C2(CCOC2)C1 45839,CN1N=C(C(=O)NC2CCN(C(c3cc(F)cs3)=O)CC2(C)C)CCC1=O 45840,C1(NC(Cc2c(C)nc[nH]2)=O)CC12CCC(NC(=O)CCC1(C)CC1)CC2 45841,C1(F)(C(N2CCC(NC(c3cc(OC)nn3C)=O)C2)=O)CC2(CCC2)C1 45842,C=C=C(C)CC(=O)N(C1CN(C(c2cc(-c3ccn(C)c3)[nH]n2)=O)CC1O)C 45843,N1(C(=O)CCc2cc(Cl)sc2Cl)CCC2(CCCN2C(=O)C(F)F)C1 45844,N1(C(C(c2cn(C)nc2)=O)=O)CCc2ccccc2C1CCNC(C1(Br)CC1)=O 45845,N1(C(CSCCOC)=O)CCC2CCN(C(=O)COCCCN(C)C)CC2C1 45846,CCCCC(O)C(=O)N(C)CC1CCCN1C(c1csc(-c2cocn2)n1)=O 45847,O=C(CS(=O)(=O)CCO)NC1CCC(CNC(c2ccc(F)cc2F)=O)C1 45848,n1(CC(=O)NCC(CC)NC(=O)Cc2ccn(C)n2)c(-c2cccs2)nnc1S 45849,C(=O)(C(C)C(F)(F)C(F)F)NC1CC(CNC(COCCOCC#C)=O)C1 45850,Cc1ccc(C(=O)NC(C(N2CC(C(N)=O)C3(CC3)C2)=O)c2ccoc2)cc1F 45851,C1(C(N(CCCn2ccnc2)C(C2C(C)C2)=O)=O)CCCCC1(C)C 45852,CC1CCc2ccccc2N1N(CC(=O)O)C(C1CCCC(CN)O1)=O 45853,C1(OC)(CNC(c2nocc2C)=O)CCN(C(C2COCCC2C)=O)C1 45854,N1(C(c2c(N)cccn2)=O)CC2CC(NC(=O)CCSc3ccccc3F)C1C2 45855,Cc1ccnc(C(=O)NC2CC2CNC(c2ccc(Cn3cccc3)cc2)=O)c1 45856,c1(OC)cccc(NC(=O)CC(C=O)NC2(C)CC(C)=NO2)c1 45857,C1(NC(CCCCCC#C)=O)CCN(C(=O)CC(C(F)(F)F)OC)C12CCCC2 45858,c1(CCC)ccc(CC(N2CC=CC(NC(c3cnc[nH]3)=O)C2)=O)cc1 45859,C1(CNC(C=C(C)C)=O)(NC(C2CNC(=O)N2)=O)CCC(F)(F)CC1 45860,c1(CC(=O)NCC2(COC)CCCN2C(=O)C=C2CCC2)ccc(Cl)nc1C 45861,CCC(CC)C(F)C(=O)NCC1CN(C(C2CC3(CCC3=O)C2)=O)C1 45862,c1(C(N(C(C)C(C)C)CC)=O)cc(C(F)F)cc(C)c1 45863,N1(C(Cc2c(CC)nccc2)=O)CCCC(COC)(NC(=O)C(O)COC)C1 45864,N12CCSCC1NC2=O.c1(C2CN(C(c3cnn[nH]3)=O)C2)ncccn1 45865,N1(C(c2n(CC)ncn2)C(=O)NC2CCCC2)CCCC(O)(C(N)=O)C1 45866,S(=O)(=O)(c1ccc(Br)cc1NCc1ccccc1F)N(C)Cc1ccc(C)nc1 45867,CCC(CC)(CCNC(=O)CN1CCCCC1)NC(c1csc(C)n1)=O 45868,C1(NC(C(=O)NCC(c2ccc(OC)cc2)N)=O)CCc2cn(C(C)C)nc2C1 45869,c1(-c2scc(OCC)c2)cccc2cc(C(N3CCCC4CCCCC34)=O)sc12 45870,C1(C(=O)NCC(C2CC2)NC(c2cc(C)sc2)=O)CC2CC1CC2O 45871,C(=O)(C(CNC(=O)CCNC(=O)N(C)C)N(C)C)N1CCC(CCN(C)C)C1 45872,C1(NC(c2c(C)nc(O)[nH]2)=O)CN(C(=O)C(C)C2CCC2)C(C)(C)C1 45873,c1(C(=O)NCCN(CC(C)O)C(c2c(C#C)cn(C)n2)=O)cn2cc(C)sc2n1 45874,c1(C(=O)NCCN(C(C2CN(CCC)C(=O)C2)=O)C)cccc(F)c1O 45875,c1(NC)cc(C(=O)NC2CCN(C(c3cccc(F)n3)=O)CC2CO)cc(Cl)n1 45876,c1(N2C(CCOC(c3ccc(OC)cc3F)=O)C(C)CC2)nc(Cl)nc2[nH]ccc12 45877,C1(NC(c2n(C)cc(NCc3cnc(N(C)C)nc3)n2)=O)CCC(C2CC2)C1 45878,c1(C(=O)NC2(CNC(C=COCC)=O)CCOCC2)ccc2n[nH]cc2c1 45879,c1(CC(=O)NCCCNC(c2ccsc2Cl)=O)cc(Cl)ccc1O 45880,C(=O)(CCOC(C1CN(C(C2CCC2)=O)C1)=O)OC(C)(C)C 45881,N1(C(C23CCC(OC)C2C3)=O)CCN(C)CC1C(=O)NCCCCCN(C)C 45882,N1(C(c2c(C)cc[nH]2)=O)CCCC2CCN(C(c3csc4c3CCCC4)=O)CC12 45883,C1(CCN(C)C(C2(C3CC3)CCCO2)=O)CCN(C(C2C(Cl)(Cl)C23CC3)=O)CC1 45884,C1(NS(CC=C)(=O)=O)CN(C(C2CCCN(C)C2)=O)CCC1F 45885,Cc1ccc(C#N)cc1NC(C1CCN(C(C2CCOC2(C)C)=O)CC1(C)C)=O 45886,C(=O)(CC(C)CC(F)(F)F)N(C(c1ccn(C(C)C)n1)C)C(C1CCCCC1)=O 45887,Cc1ccc(NC(=O)NCC2CC2)c(C(N2CCNCC(C(=O)O)C2)=O)c1 45888,c1(C(c2n(CC=C)nnn2)NCC(CO)C(C)(C)C)ccc2c(c1)CCO2 45889,c1(CC(=O)NC2C(NC(CC(=C=C)C)=O)CCC2)c[nH]c2c(F)cccc12 45890,N1(C(CCCCC)=O)CCc2nc[nH]c2C12CCN(C(c1cccc(N)c1)=O)C2 45891,CC1(C)C2CCC1(C(=O)NCC1CC(F)(CNC(C3CC34CC4)=O)C1)CC2 45892,CC(C(=O)N(C)CCOCCCN(C)C(C1(C#N)CC1(C)C)=O)C(F)F 45893,Cc1ccc2[nH]cc(CNC(C3(N(C(=O)CN4CCC(=O)CC4)C)CC3)=O)c2c1 45894,C1(CNC(c2nsnc2O)=O)CN(C(C2(F)CCOC2)=O)CCC1(F)F 45895,c1(C(N2CCC(C(N(C3(CO)CCC3)CC)=O)C2)c2ccccc2)ccccc1 45896,Cc1cc(F)cnc1C(c1nnnn1CCCOCC1CC1)NCCCC(F)(F)F 45897,C1(c2cn(C3N(C(CC(C)F)=O)CC3)nn2)CCCCC1C 45898,c1(CC(=O)OC(CCC=C)C)cc(Cl)cc2ccccc12 45899,c1(OCC(=O)NC(CNC(C2(NC(C)=O)CC2)=O)C(C)C)ccc(F)c(F)c1 45900,c1(CC)cc(C(=O)NCCC2CC(OC)CN2C(c2cnco2)=O)oc1CC 45901,Cc1ncsc1C(=O)N(C)Cc1cocn1 45902,c1(C(=O)NCC2(NC(C3C(C)(C(F)F)C3)=O)CCC2)ccnc(-n2cccn2)c1 45903,C(C(=O)NNC(=O)C(C)(C)CCCCNC(=O)C(O)C1CC1)OCC 45904,C(=O)(CCCCN(C)C(c1ccc(C)nc1)=O)NCc1scc(C)c1 45905,C(=O)(C#CC1CCCOC1)N1CC(C)N(C(c2coc3ccc(F)cc23)=O)CC1 45906,C1(O)(CCNC(=O)CSC2CCS(=O)(=O)C2)CCCN(C(C2(O)COC2)=O)C1 45907,c1(C(=O)NC2C(SCC=O)C2)ccncc1.C1(CC(=O)NC)CCCCC1 45908,C1(CC(=O)NCCCN(C(c2cccc(COC)c2)=O)C)OCCCC1(C)C 45909,N1(C(CCOC)=O)C2CCC1(CNC(=O)Cn1cc(C3(O)CCC3)nn1)CC2 45910,C1(C(=O)NCCc2cc(C)nn2C)CCN(C(c2ccccn2)=O)CC1O 45911,N1(C(=O)CC2CCCCC2)CCCC(C2CN(C(c3cc(F)ccc3Cl)=O)C2)C1 45912,C(=O)(CC1OCCc2ccsc21)NC1(CCNC(=O)Cc2cncnc2)CCC1 45913,N1(C(c2cccc(C(C)(C)C)n2)=O)CC(C2CN(C(C3(C)CC(C#N)C3)=O)C2)C1 45914,C1(C2CC2)(CNC(C(C)OCC(C)C)=O)CCN(C(=O)CCCn2cncn2)C1 45915,C1(NC(=O)CC2CCN2C(=O)C=Cc2nccs2)CC(=O)N(C2CCCCC2)C1 45916,C12(C(N(CCNC(=O)C(c3ccc(Cl)cc3)(F)F)CC)=O)CCC(CC1)OC2 45917,C(=O)(C1CSc2ccccc21)NCc1c(OCC#C)nccc1 45918,N1(C(CC(c2ccc(F)cc2)NC(C2CCCCO2)=O)=O)CC2OCCOC2C1 45919,N1(C(C2(OC(C)=O)CC2)=O)CCC(C(N2CCOC(CN(C)C)C2)=O)C(C)C1 45920,C(C(C)(C)CNC(=O)CC1CCC(C)O1)N(C(COCC(=O)NC)=O)CC 45921,C=C(C)CCCC(=O)N1CCC(C(C)(C)NC(=O)C(CC)c2cccnc2)C1 45922,C12(C(=O)NCC(C)NC(=O)Cn3ncnn3)CC3CC(C(=O)N1)C2C3 45923,C=CCC(CNC(C1(CO)CCC1)=O)C(=O)N1CCOCC1CC 45924,Cc1cccc([N+](=O)[O-])c1NC1CC(CCNC(C2CC3(CSC3)C2)=O)C1 45925,C=CCC(CC)C(=O)N1CCN(C(=O)COc2cccc(F)c2F)CC1COC 45926,N1(C(c2c(O)ccc(C)c2)=O)CCC(C(=O)NCC(c2cnc[nH]2)C)CC1(C)C 45927,C1(N(C(c2c(CC)ncs2)=O)C)CCN(C(=O)Cc2cc(C(=O)OC)cs2)CC1 45928,CCC(C(=O)NC(C)CCNC(c1cccc(N2CCCC2=O)c1)=O)C(C)O 45929,C=C(Cl)CC(C(=O)NCCCOCC(F)F)NC(c1cc(C)ncn1)=O 45930,c1(CNC2(Nc3cc(C(=O)NCCC)n(C)c3)CC2)cccc(O)c1C(=O)OC 45931,c1(CC)nc(N2CC(OCCN)C2)cc(Cl)n1 45932,Cc1ccc(C)c(CC(N2CCC(CNC(=O)C=C3CC3)C(C)C2)=O)c1 45933,C1(C(=O)NCC(C2CC2)NC(=O)CCc2ccccc2F)CCC2(CC1)CC(=O)C2 45934,c1(C(N(CCNC(c2c(CC)n(CC)nc2)=O)C(C)C)=O)cccc(C)c1F 45935,C(=O)(C(F)CC(C)(C)NC(C1(CO)CCCC1)=O)NC1CC(CCOC)C1 45936,CC(CC(F)(F)F)C(=O)N1CCC(C(C)(C)NC(=O)C(F)C(C)(F)F)C1 45937,CC1CC(CNC(=O)CC2(C)CC2(Cl)Cl)CN1C(c1n[nH]c(=N)s1)=O 45938,c1(NCCNC(C(=O)NC(CC)(C)COC)=O)cnc(C)n1-c1ccccc1 45939,N1(C(C2(CCC)CCC2)=O)CC2CCCC2(NC(=O)C=C(Cl)Cl)C1 45940,N1(C(C(N2CCCC(CC(=O)OCC)C2)=O)=O)CCCNC(=O)C1CC 45941,C1(SC)CCN(C(=NCCCCl)NCC(=O)N(c2cnc(C)c(C(C)=O)c2)C)C1 45942,c1(COC)ccc(C(=O)NCC(C2CCC2)NC(c2oncc2C)=O)cc1 45943,C1(NC(c2n(CC)ccc2)=O)CC2(C1)CC(NC(=O)CC(O)c1ccccc1)C2 45944,N#Cc1c(Cl)nsc1NC1CCN(CCNC(=O)CNc2ccccc2)C1 45945,C=CC1(C(N2CCC(O)(CCNC(c3scc(C)c3C)=O)C2)=O)CCCC1 45946,c1(C(N(C(c2n(CC)ccn2)C(=O)O)C)=O)cc(C)cc(O)c1 45947,N1(C(C(C)NC(C)=O)=O)CCOC(CCNC(=O)CC2CC(C)C2)C1 45948,Cc1oc(C2CC2)nc1N(S(=O)(=O)CC1CC1C)C 45949,C(C(=O)NC(C)CC)(C(C)CC)N(C(c1cc(CC)on1)=O)C 45950,c1(C(N2CCC(CNC(C3CC4(CC4)C3)=O)C23CC3)=O)cc2c([nH]1)CCCC2=O 45951,C#Cc1ccc(CNc2cccnc2C(=O)NC(c2ccccc2)CN(C)C)s1 45952,N1(C(c2cc(C)cc(O)c2)=O)CCC(C2(NC(C3(C(C)C)CC3)=O)CC2)CC1 45953,Cc1cncc(C(N2CCC(O)(C(C)NC(=O)CCc3ccncn3)C2)=O)c1 45954,C1(N(C(CCN(CCCCC)C)=O)C)CCC(NC(=O)C(O)CC)CC1 45955,c1(CNC(C(N(C(CN(CCC)C)=O)C)C2CC2)=O)cnc(C)cn1 45956,N1(C(=O)CO)CC2CCN(C(c3nn[nH]c3Cl)=O)CCC2C1 45957,c1(C(N2CC(NC(=O)Cc3ccnc(F)c3)C(O)C2)=O)cc2c(nn1)CCCC2 45958,c1(C(N2C(CNC(CC3C(C)=NNC3=O)=O)C=CC2)=O)cc(C)ccc1F 45959,c1(NC(=O)C(F)CC2CNC2)cnccc1CO 45960,C1(CNC(C(C)OCC#C)=O)CCCN1C(c1c[nH]nc1-c1cccnc1)=O 45961,N1(Cc2ncc(C(=O)NC(c3nc(C)oc3)C)cn2)CCC(CN(C)C)CC1 45962,c1(N2CCN(C(=O)C=Cc3ccccn3)CC2)ncnc2c(Cl)cc(Cl)cc12 45963,N(C(=NCC1CC1)N1CCC(C2CCCN2CC)C1)Cc1ccccc1NCC 45964,CC#CCCCCN=c1ccc2cc(S(=O)(=O)N(C3CCN(C)C3)C)ccc2[nH]1 45965,c1(CC)ccc([N+](=O)[O-])cc1C(N1CCC12CN(C(C1CCCNC1=O)=O)C2)=O 45966,C(=O)(C(C(C)(C)C)c1ccccc1)NC(C(C)NC(=O)CCC1CCCC1)CO 45967,N1(C(c2n(C(CC)CC)nc(C)c2)=O)CCCC(NC(c2coc(C)n2)=O)CC1 45968,C1(NC(=O)NC(C)(C)CC(N2CCCCC2c2ncc[nH]2)=O)CCN(C)CC1 45969,C#CCC(C)(C(=O)NC1(C)CCSCC1)NC(=O)CC(C)(O)COC 45970,C1(NC(c2occ(C)c2)=O)(CO)CCN(C(c2ccc(CC(C)(C)C)cc2)=O)C1 45971,N1(C(C2OCCN(C(C3(CC(C)C)CCC3)=O)CC2)=O)C2CCC1CN(C)CC2 45972,c1(C(N(CC(COC)C)C)=O)cn2c(n1)CCN(c1ncnc3cc[nH]c13)CC2 45973,C(=O)(C#CC1CCOCC1)NCC(C(C)C)NC(C1CC(=O)N(C2CCC2)C1)=O 45974,c1(C(=O)NCC2C(NC(=O)Cc3cscn3)CC2)cc2ncccc2s1 45975,N1(C(C(C)NC(N)=O)=O)CC2(CC(NC(=O)C(C)(C)NS(C)(=O)=O)C2)C1 45976,CCCCC(CC)CC(=O)NC(C(C)N=c1[nH]ncs1)c1ccccc1 45977,C1(F)(CNC(C(C)=C(C)C)=O)CCCN(C(C2(C)CC(C)C2)=O)C1 45978,c1(C(N2C(CNC(=O)C=CC3CCCCC3)CC3CC32)=O)cc(=O)cc(Cl)[nH]1 45979,c1(Cc2n(CCCOC)c(N3CCC(CS(N)(=O)=O)C3)nn2)c(O)cccc1F 45980,C(C(C)(C(=O)NCC=C1CCN(C(c2nn(C)cc2SC)=O)CC1)OC)OC 45981,C(c1ccccc1)=CCC(N1CCC(CN(C(C(COCC)C)=O)C)C1)=O 45982,N1(Cc2noc(CCC)c2SCC[Si](C)(C)C)Cc2c(ccc(F)c2Br)C(C)(C)C1 45983,C(=O)(CCC(C(C)C)NC(c1c[nH]c(C)c1)=O)N1CCCC(OC)CC1 45984,N1(C(C)C)CC(C(=O)OCc2ccccc2C(F)(F)F)CC1=O.C1(C)C(=O)O1 45985,Cn1ncc(C(=O)NC2CC3CC(NC(C4OCC4(C)C)=O)C2C3)c1S(N)(=O)=O 45986,C=CCC(F)(F)C(=O)NC1CN(C(=O)COCCOCCO)C2CC12 45987,c1(Cn2ccc(C(N3CCC(c4ncc(C)cn4)CC3)=O)n2)ccc(Cl)c(F)c1 45988,Cc1ccc(SCC(=O)NCCCCC2CN(C(c3snnc3C)=O)C2)cc1 45989,CC1(C)CC(NC(=O)CCCNS(C)(=O)=O)CN1C(c1nc(Cl)ccc1N)=O 45990,C1(C(=O)NCCc2nc(C)[nH]n2)CCCC(NC(=O)C(F)CC2CCOC2)CC1 45991,N1(C(COCC(=O)OC)=O)CCC(C(C)(C)C)(CNC(C2CC(C)(F)C2)=O)C1 45992,CC1CC(CNC(=O)C(O)C2CCCC2)CN1c1nccc(C2CCCC2)n1 45993,N1(C(C(CCCC)C)=O)CCCC2CN(C(C3(CCOC)CCCC3)=O)CCC12 45994,C1(C)(CCC(=O)N(CCC(C)(C)C)C)CCCN1C(=O)CCc1ncnn1C 45995,C1(CNC(C2(OC)CC(CF)C2)=O)CC(=O)N(C2CN(C(=O)C=C(C)C)C2)C1 45996,c1(CCNC(CCc2cc(C)on2)=O)c(C)n[nH]c1C 45997,N1(C(c2nccc(CC)c2)=O)CCN(C(C2CC(C)=NO2)=O)C(CC(=O)NC)C1 45998,N1(CCCCCCCOCCOCC)CCN(CC(=O)NCC=CCl)CC1 45999,Cc1ccc2nc(C)c(C(=O)N(C3CCN(C(C4CC(Cl)(Cl)C4)=O)C3)C)cc2c1 46000,C1(C(=O)NC2CN(C(c3c(O)ccc(CC)c3)=O)CC2O)CCc2cnnn2C1 46001,c1(OC)ccc(C(=O)N(C)C(c2nn(-c3ccccc3)nc2C)C)cc1[N+](=O)[O-] 46002,CCCCC(C)CCC(=O)N1CC2CCC1CC2NC(=O)C(C)OCC 46003,C1(CNC(C(C=CC)O)=O)CC(C)CCN1C(=O)CNC(c1ccc(C)s1)=O 46004,c1(C(CC(=O)OC)NC(c2c[nH]cc2C)=O)cccc2ccccc12 46005,C1(N(c2n(C)ncc2Br)C(C2NCCC2O)=O)CCC2(CC1)CNC2 46006,N1(C(CC(C)N2CCCC2)=O)CC2C(C(=O)NCc3nn[nH]n3)C2C1 46007,c1(CC(=O)NCC(C(=O)NC(C23CC(CO2)C3)C)O)ccnc(O)c1 46008,C1(NC(c2c(OC)nsc2)=O)CCC12CN(C(=O)CCc1csc(=N)[nH]1)C2 46009,N1(C(c2cncc(NC(CN(C)C)=O)c2)=O)CCN(C=O)CC1 46010,c1(CC(=O)NCC=CC(N2CCC(CF)CC2)=O)ccc2c(c1)CC2 46011,N1(C(C2(N(C)C)CCC2)=O)CCN(C(c2ccn3nccc3n2)=O)C2(CCC2)C1 46012,N1(C(C2(CCCC)CCC2)=O)CCC2(CCCN(C(=O)CNC(=O)OC)C2)C1 46013,C(=O)(C(C(C)C)NC(=O)C(CC)n1ccnc1)NC(CC#C)CC 46014,Cc1cc(C(=O)NCCOc2ccccc2C(=O)O)c(F)cc1Cl 46015,C1(CC(C)NC(c2cc(F)n[nH]2)=O)CCN(C(C2(C)CC=CC2)=O)CC1 46016,N1(C(CC(=O)OC)=O)CCC2(CC1)CC(NC(=O)C(CC1CCCC1)C(C)C)C2 46017,Cc1ccc(F)c(CC(=O)NC2CCC(NC(=O)C(F)C3CCC3)C2)c1 46018,C1(C(=O)NCC(O)CNC(C2CCC(c3ccccc3)C2)=O)(CC)CCCC1 46019,N1(C(C)=O)CCC2(CCOCC2)C(NC(c2coc3c2C(=O)NCCC3)=O)C1 46020,c1(CN(C)C(C2CC(NS(C)(=O)=O)C2)=O)ccccc1CNC(=O)C(C)(C)OC 46021,C1(C(N2CC(CC(C)NC(C3=C(C)OCC3)=O)C2)=O)CCc2nc(O)[nH]c2C1 46022,CCCCCCCC(=O)N1CC2CCC(NC(=O)CCN(C)CC)(C2)C1 46023,c1(C(=O)NC2(CN(C)C(c3ccc[nH]3)=O)CC2)ccnc(Cl)c1N 46024,CC1CCC(CN(C)C(C2(CNC(C3CCCC(CF)C3)=O)CCC2)=O)CC1 46025,C1(NC(C2CCC(C)CC2)=O)COC2(C1)CN(C(c1ncnc(O)c1Cl)=O)C2 46026,c1(C(N2CCC3CN(C(C4C(C=C)OCC4)=O)CC32)=O)cnc2ccccc2n1 46027,c1(OC)cc([N+](=O)[O-])ccc1CN=C(NCC(F)F)NC1CCCCC1C 46028,C(=O)(C1=CCC(NC(=O)C(n2cc(-c3sc(C)nc3C)nn2)C)C1)OC 46029,CCC(Cc1ccccc1)C(=O)NC(c1nc(C(C)C)no1)C 46030,N1(C(C2(C)CC2(F)Cl)=O)C(CNC(C2CCCO2)=O)CC2COCC12 46031,c1(-c2cn(CC)c(=O)cc2)ccc2ccc(C(=O)Nc3ccc(Br)nc3)nc2c1 46032,CC(C)CC(C)CC(=O)N1CCC(N(CCO)C(c2c(Cl)cccc2Cl)=O)CC1 46033,CC(CN=c1[nH]c(=NC(C)c2nccs2)[nH]c2ccc(Cl)cc12)N1CCCC1 46034,N1(C(C2C(=O)NCC2)=O)CC(CO)C2(C1)CN(C(C1CCn3ncnc3C1)=O)C2 46035,C(=O)(C(C)CC(F)(F)F)NCC1CC(OC)CN1C(c1c[nH]nc1C)=O 46036,C(=O)(CS(=O)(=O)CC(=O)OC)N1C(CNC(C(CC)=CC)=O)C(C2CC2)CC1 46037,c1(C(=O)NC(CCCCNC(C)=O)C)cnc2c(C)cnn2c1 46038,C1(C(=O)Nc2cc(OC(C)C)n[nH]2)COCCC1c1nc(C2CC(F)(F)C2)no1 46039,C1(C(=O)N(CC(C)(O)C2CC2)C)(CC)CCN(C(=O)C(C)CC)CC1 46040,c1(C(=O)NCc2ccc(-c3nn[nH]n3)nc2)cccc2[nH]ncc12 46041,c1(-c2cn(CCCCNC(c3c(C)coc3)=O)nn2)cccc(C(F)(F)F)n1 46042,N1(C(C2(F)C(C)C2)=O)CC2(CCCCN2C(=O)CCOCC(F)(F)C(F)F)C1 46043,c1(NC(c2c(C)nccc2)C)[nH]c(=NCC2CC2(Cl)Cl)nc2scnc12 46044,C1(NC(c2nccc(C)n2)=O)CCC2CCN(C(=O)C=Cc3ccc(C)o3)C12 46045,c1(NC(C2(C)CS(=O)(=O)C2)=O)ccc(S(=O)(=O)c2ccccc2)nc1 46046,N(C(=NCCC(C)(C)S(C)(=O)=O)NCC(F)F)CC1CC(N(C(=O)OC)C)C1 46047,N1(C(C=CCOC)=O)CC(CNC(c2cnc(C3CC3)nc2O)=O)OC(C)(C)C1 46048,c1(OCC(=O)NC(C(C)NC(C2CCCCC2)=O)C)cccc(Br)c1 46049,CC1(C)CC(CC(=O)NC(CO)C2CCC2)CN1C(=O)CC1CC(=O)C1 46050,c1(CCCC(=O)NCC2CC2NC(C2CC3(CC3)C2)=O)ccc(Cl)c(Cl)c1 46051,c1(C(N2CC3CN(C(=O)CCN4CCOCC4)CC32)=O)cnc2ccccc2n1 46052,N1(C(CN(C(C(C)=O)=O)CC2CCCCC2)=O)CCSC(C)(C)C1 46053,C1(CC(=O)NC2CC(C(C)NC(=O)C=Cc3nccs3)C2)CCN(C)C1=O 46054,C1(NC(c2ncn(C(C)(C)C)n2)=O)CCN(C(C2(C)CC2(Cl)Cl)=O)CC1(C)C 46055,c1(C(N2C(C)CN(C(=O)C(F)(F)CO)CC2)=O)cc2n(n1)CCCC2=O 46056,C1(C(=O)NC(c2ccc(Cl)nc2)CNC(=O)C=C2CCC2)CCOC(=O)N1 46057,C1(C(=O)N(C2CCC(NC(=O)CNC(c3cnoc3C)=O)C2)C)(OC)CC(C)C1 46058,Cn1cnc2cc(C(=O)NC3C4CC3N(C(=O)C(C)(Cl)Cl)C4)ccc12 46059,C1(NC(C(C)N2CCC2)=O)CN(C(=O)Cc2ccno2)C2(CCOCC2)C1 46060,c1(OC)ccc2c(c1)C(NC1=NCCCN1)CCO2 46061,CN1CC(O)CCC1C(N1CC2(CNC(c3cnn[nH]3)=O)CC1CO2)=O 46062,C1(Nc2c(-c3ccc(F)c(N4CCCC4)c3)cccc2)CNC2(CCOC2)C1 46063,N1(C(COC(C)(C)C)=O)CC2CCN(C(C3CC=CC3)=O)C2C1 46064,C1(CNC(c2ccc(O)nc2)=O)CC2(CCN(C(C3(CF)CC3)=O)CC2)CO1 46065,Cn1cnc2sc(C(=O)NCCC3CCN(C(C4(O)CCCCC4)=O)C3)cc12 46066,c1(C(=O)NCC2N(C(Cc3c(O)nc(=N)[nH]c3)=O)CC2)cc2ccc(Cl)nc2s1 46067,N1(Cc2c(C(=O)OC)csc2)CCOCC1c1cccc(F)c1 46068,C1(N(CC(C)C)CC(=O)NCc2ccccc2)CCCC(N)C1 46069,C1(CC=C)(NC(c2ncoc2C2CCC2)=O)CN(C(=O)Cc2ccnn2C)C1 46070,C(=O)(C1CCCc2n[nH]cc21)NCC(C)NC(C1CC(C)(c2ccccc2)C1)=O 46071,CC1CCN(C(=O)CCCc2ccncc2)CC1CNC(c1ccc[n+]([O-])c1)=O 46072,N1(C(c2c(C)csc2)=O)CC2CC(NC(=O)Cc3cc4ccccc4o3)C(C2)C1 46073,Cc1ccccc1N1CC(C(=O)N(CCCNC(=O)CC(C)F)CCO)CC1=O 46074,C=CCC(C(=O)NCCC(C)NC(c1cnn(C)c1CC(=O)OC)=O)C(C)(C)C 46075,CC1(C)CCN(C(c2ccc3sncc3c2)=O)CC1NC(c1cncnc1)=O 46076,c1(C(C(=O)NCCNC(C(COC)COC)=O)C)ccc(S(C)(=O)=O)cc1 46077,CCC(=O)CCC(=O)N1CC(C)(CCC(N2CCC(N(C)C)(CC)C2)=O)C1 46078,CC(C)CC(O)CC(=O)NCSC1(O)CC2CCC1CC2 46079,O=C1C(=CC2CCOC2)Cc2c(Cl)ccc(Br)c21.C(=O)C=CC=CC=CCO 46080,C(=O)(CCC(=O)NCC1CC(O)CN1C(=O)CCOc1cccc(Cl)c1)OCC 46081,c1(C(=O)NCC2(NC(C3CC3F)=O)CCOC2)cc(Cl)cc(C(F)(F)F)n1 46082,c1(C(=O)NCC(CC)(CC)NC(C2C(C)C2C)=O)cc(F)c(F)cc1Br 46083,CC1(c2ccc(NC(C3CN(c4ncncc4I)C3)=O)cc2)NC(=O)NC1=O 46084,c1(C(=O)OC)ccccc1CCC(=O)NCC1(F)CN(C(=O)Cc2ccon2)C1 46085,c1(CNC2CC(NC(C(C(C)c3ccccc3F)O)=O)C2)cc(C#N)ccc1F 46086,C(CC(C(C)(C)C)NC(=O)Cn1ncn(C)c1=O)N(C(C(CC#C)C)=O)C 46087,C(CCC(C)(C)C(=O)NCC(C)CCCO)NC(c1c(C)ncnc1)=O 46088,CCCS(=O)(=O)C(C)C(=O)NC1CN(C(=O)CCCCCN(C)C)C2(CCC2)C1 46089,C1(NC(c2oc(C)c(Br)c2)=O)CN(C(=O)CCCCCNC(N)=O)C2(CCC2)C1 46090,N1(C(C2(C(=O)NC)CC2)=O)CCC2(CCCN(C(c3ccn(C)n3)=O)C2)C1 46091,c1(C(=O)NC2CC(CO)N(C(C3(C(N(C)C)=O)CC3)=O)C2)ccc2nn[nH]c2c1 46092,c1(C(=O)NCC2(O)CN(C(c3ccc(CC4CC4)s3)=O)C2)ccnc(Cl)c1Cl 46093,C1(C(N(C2CCN(C(=O)Cc3cncc(C)c3)C2)NCC)=O)CCCC2(CC2)C1 46094,N1(C(C(C(C)C)NC(C)=O)=O)CCC12CN(C(=O)C(C)NC(=O)C1CC1)C2 46095,C1(NC(c2cc3sccc3[nH]2)=O)CC2(NC(C3CC4CC4C3)=O)COC1C2 46096,C12(C(=O)NCC(CC)O)CC(C)(CN1C(c1cc(COC)no1)=O)C2 46097,C(=O)(C1CCc2nccn21)NC1(C(=O)NCCc2ccns2)CCN(C)C1 46098,C#Cc1ccc(C(=O)NC2CN(C(C3(C(=O)NC(C)C)CC3)=O)C2)cc1F 46099,C1(C(=O)NC2(c3ccn(C)n3)CC2)(NC(CC=CCC)=O)CCN(C)C1 46100,c1(OC)ccc(CN(C(C2C3CCOCC23)C(=O)NC)C)c(OC)c1 46101,N1(C(Cn2nc(C)c(Br)c2)=O)CCOCC(NC(C2(F)CCCCC2)=O)C1 46102,CC(C(=O)NO)NC(C1CC(C)N1C(=O)CCC1CCCCC1)=O 46103,N1(C(c2ncc(OC)nc2)=O)C2CCC1CN(C(C1CCC3(CCC3)C1)=O)C2 46104,C1(CNC(CCCCSC)=O)CCC2(CN(C(c3cccc(C)c3C#N)=O)C2)O1 46105,C1(C(=O)OC)C=CCCN1C(=O)CCC1(C)CN(C(=O)CCOC(C)C)C1 46106,C1(C(=O)NCC(C)(CO)NC(c2ccc(C)cc2)=O)CCCC2(CCC2)O1 46107,N1(C(=O)C=Cc2ccc(C(F)(F)F)cc2)CCOC2(C1)CN(C(C1(O)CC1)=O)C2 46108,CC(=O)CCC(=O)N1CCC1(C)CC(=O)NC1CCC(C(N)=O)CC1 46109,c1(CNC(CCC2N(C(CN(C)C(=O)C3CC3)=O)CCC2)=O)cccc(O)n1 46110,C1(C(=O)NC(C(=O)NCCN(CCOC)C)CO)CC2(C1)CC2(F)F 46111,c1(OC)cccc2sc(NC(C3CC4CCCC4N3C(N)=O)=O)nc12 46112,C(CCCCC(=O)NCC1(O)CCN(C(c2scnc2CC)=O)C1)OCC 46113,C(=O)(C(C)(C)C(O)C(C)C)N1CC2C(NS(CCOC)(=O)=O)C(CC2)C1 46114,C1(NC(C2C(C)(C)C2)=O)CCC2(CCN(C(c3ccc4cc[nH]c4n3)=O)C2)C1 46115,C1(C(N2CCN(C(CC(=O)NCC)=O)C(C(C)C)C2)=O)CC2OC(C)(C)OC2C1 46116,O=C1CC(C(=O)NC2CC3(C2)CC3C(N2CCn3nccc32)=O)=NN1 46117,C1(NC(C(C)c2ccsn2)=O)CCCN(C(=O)Cc2cccc(Br)c2)C1 46118,Cc1cc(CC2CCCCN2C(=O)C(C)N(C)CCC2(O)CCCCC2)n(C)n1 46119,N1(C(C2(C)C(C)C2)=O)CCC(C2CC2)(CNC(c2ccc3[nH]ccc3n2)=O)C1 46120,C(=O)(C(F)CC(CC)CC)N1CCC(C(N(C23CCN(CC2)CC3)CCC)=O)CC1 46121,N1(C(C=CC=CC)=O)CCC2CC2(C(=O)NCc2n[nH]c3c2CCC3)CC1 46122,c1(OC)cc(Br)ccc1C(CO)NC(=O)NCc1oc(C)cc1C 46123,NC(=O)CC(C(=O)NCCC1CCCCC12CC2)NC(=O)CC1CCSC1 46124,c1(C(N2CC(CNC(C3C(OCC)C3)=O)(OC)C2)=O)c(O)nnc2c1COCC2 46125,c1(C2(CNC(c3ccsc3)CO)CCC2)ccccc1Cl 46126,C1(NC(C2CCC(=C)CC2)=O)C(C)CCN(C(c2ccc(Cl)c(F)c2F)=O)C1C 46127,C(=O)(C1=CCC(C)(C)CC1)NC(C(C)(C)NC(Cc1c(O)ccc(C)c1)=O)C 46128,c1(C(=O)NCC2C(C(=O)Nc3cnc(OC)nc3)C2)coc2c1COC2 46129,C(=O)(CCCC(F)(F)CO)NC1CC2CN(C(c3cncc(C#N)c3)=O)C1C2 46130,c1(OC(C)C)ccc(CC(=O)N(C2CCC(CNC(=O)CC(C)C)CC2)C)cc1 46131,c1(NC(CSCCC)=O)ccc(CNC(=O)CCCOC2CCN(C)CC2)cc1 46132,c1(CCOC)nc(=NC2CCCC(NC(C3(O)CCSCC3)=O)C2)s[nH]1 46133,Cc1cc([N+](=O)[O-])c(C)cc1C(N1CC2CN(C(c3ncccc3F)=O)C2C1)=O 46134,C(C(CNC(=O)CC(C)C1CC1)S(C)(=O)=O)NC(C1(CC=C)CC1)=O 46135,N1(C(c2c(C)[nH]cc2)=O)C(C(=O)N(C(C)C)Cc2ccco2)CCC1C 46136,O=C(C1CCCc2cncn21)NCC1(O)CN(C(=O)C(Cl)=CCl)C1 46137,c1(N2CC(C)=C(C)C2)nc(N(C)CCNS(C)(=O)=O)nc2cc[nH]c12 46138,C1(NC(CNC(C(CC)C)=O)=O)CN(C(c2ccn(C)c2)=O)C2(CCCCC2)C1 46139,c1(C(=O)NCC(C)CNC(c2ccc(C(F)F)o2)=O)c(F)cc(Cl)cc1F 46140,Cc1ncc(C(=O)N(CC(C)N(C(=O)CN2CC3CCC2C3)C)C)cc1N 46141,Cc1c(NC2CCN(CC(F)(F)F)C2)ncnc1N(C)CCOC1CC1 46142,c1(N2CCC(N(C)C(c3ccc(O)nn3)=O)C2)nnccc1C#N 46143,C1(C(=O)NCCC(CNC(CN(C2CC2)CC)=O)O)CCCC(C)(C)O1 46144,c1(OC)ccc(C(N2CCCC2CC(C)O)C(=O)NCC2CCCO2)cc1Cl 46145,C(=O)(CC(C)(C)CC(F)F)NCC1N(C(c2ccc(CC)cc2C)=O)CCC1C 46146,c1(-n2c(-c3cnc(F)c(C)c3)nc(COCC)n2)c(C)cc(C)cc1C 46147,c1(C(=O)NC(c2c(NCc3nccc(C)c3)cccn2)=O)ccc2nc[nH]c2c1 46148,c1(CC)nc(C)c(C(N2CCC(C)(CNC(=O)CCC(=O)N3CCCC3)C2)=O)o1 46149,C(=O)(C1CCCn2nccc21)NCC1C(NC(CN(CC(C)(C)C)C)=O)C1 46150,c1(NC(=O)NCc2ccc(CC)s2)cnccc1C(F)(F)F 46151,c1(C(=O)NC2CCC(CNC(C(N3CCNC3=O)C)=O)C2)ccc(F)cc1N 46152,n1(CC(=O)N(C(CNC(Cn2cc(C(C)=O)nn2)=O)C)C)ncccc1=O 46153,C#Cc1cnn(C)c1C(N1CCC(F)(CNC(c2cncn2C2CC2)=O)C1)=O 46154,CC1CC(NC(=O)Cc2cc(F)ccc2Cl)CCN1C(c1cnn2ccsc12)=O 46155,c1(C(=O)NCC(CC)(CC)Nc2cncc(C#N)n2)ccc2nc[nH]c2n1 46156,c1(CC(C)C(=O)N2CCCC2CN(C)C(c2cc(F)c[nH]2)=O)ccc(F)cc1F 46157,C(=O)(CCC(C)NC(=O)NCCCNCCN1CCCC(C)C1)OC 46158,C1(NC(CCC(=O)NCCC)=O)CCCN(C(c2ccccc2SC)=O)CC1F 46159,c1(C(CC)C(=O)N(C(C)CN(C(=O)COCC(=O)NC)C)C)c(C)noc1C 46160,C12(C(=O)OC(C)(C)C)CC3CC(CC(C3)C1)C2.CC1CC(C)OC1C(=O)NC 46161,C1(C(N(CC(C(C)C)OC)C)=O)C=CCN(C(=O)CCn2ccnc2C)C1 46162,c1(C(=O)NC2CCCC(NC(C3N(C)C(=O)CC3)=O)C2)ccc2c(c1)CCCC2 46163,C1(CNC(CC(C)O)=O)CCCCN(C(c2ccc(Cl)o2)=O)CC1 46164,N1(C(c2ccc(C)o2)=O)CCC(NC(=O)C(C2CCCN(C)C2)(C)C)C1C(C)C 46165,c1(OC)ccc2[nH]cc(C(N3CC(CNC(c4ccnn4C)=O)C(C)C3)=O)c2c1 46166,c1(C(=O)NC2CN(C(C=C(CCC)C)=O)C(C)C2)cc2c(OC)cccc2[nH]1 46167,O=C1COc2ccccc2CN1C1CN(S(=O)(=O)c2scnc2C2CC2)C1 46168,C1(CNC(C=C(C)C)=O)(CNC(=O)CC2CCC(=O)N2)CC12CCC2 46169,CCCC(C(=O)N1CCN(C(C23CCCN(CC2)C3)=O)CC1C(C)C)C(C)C 46170,N1(C(c2cnn(CC)c2Br)=O)CC(C)CCC1CNC(C1CCCCC1)=O 46171,c1(OCCC)ccc(-c2ccc(CC(N3CCOCC3)=O)cc2F)cc1C 46172,CC1(C)CN(C(=O)C=Cc2ncc[nH]2)C1C1CCN(C(=O)CSC2CC2)CC1 46173,C(=O)(CS(=O)(=O)CC1CCCN1)C(c1cn(CCS(CC)=O)nn1)(C)C.N 46174,N1(C(C(N)=O)=O)CC2(C1)SCCC2NC(=O)Cc1ccccc1O 46175,CC(CCCNC(c1csc(F)c1)=O)NC(=O)C(c1ccccc1)F 46176,NC(C(=O)NCC1(F)CCCNC1)C1CCc2ccccc21 46177,C1(CC)CCCN(C(C2CN(C(C)C)C2)=O)C1C(=O)NC1CN(C)CCC1O 46178,C1(SC)CCCCN(C(C2CCN(C(=O)c3ccc(=N)[nH]n3)O2)=O)C1 46179,Cc1cccc(C(C)N(C)Cc2cc[nH]c2)c1C 46180,C=CCCC(C(=O)NC1(CO)CC(OC)C1)NC(=O)C=Cc1cscn1 46181,c1(C(N2CCCC(O)(CNC(c3c[nH]c(=N)o3)=O)C2)=O)cc(=O)n2nccc2[nH]1 46182,C1(NC(CN(CCC)C(C2CN3CCN2CC3)=O)=O)CCCCC1C#N 46183,C1(C(NOCCCOCC)=O)CCN(C(=O)Cc2c[nH]nc2C)C(C)C1 46184,N1(C(c2ccc(CSC)o2)=O)CCC(C)C(N(C(=O)Cc2ncoc2C)C)C1 46185,CC1CCC(C(=O)NCCN(C(=O)COc2cnn(C)c2)C2CC2)CC1 46186,C(CC(C(=O)NC1CCCN(C(c2csc(C(F)F)n2)=O)C1)OC)OC 46187,CC1(C)OC(=O)NC1C(=O)NC(c1cccc(Cl)c1)CNC(=O)CCC(N)=O 46188,c1(OC)c(C(=O)N(C2COC3CCCCC23)N(c2ccc(C)o2)C)sc2nccnc12.C(C)=O 46189,C=C(C)CC(C(=O)NC12CC(NC(=O)C(C)NC(C3CCCC3)=O)(C1)C2)OC 46190,N1(C(C2CCC(=O)N2)=O)CCC2(CC2NC(=O)C2=C(Cl)CCC2)C1 46191,N1(CCC(=O)N(C(C)CNC(C2(N(C)C)CCCCC2)=O)C)CCSC(C)(C)C1 46192,C1(C(=O)NCC(C)(C)Nc2nc(C3CCCC3)ns2)CCc2c[nH]nc2C1 46193,C1(=O)C(CCC2OCCO2)SN1c1nc(C)cs1.C(C(=O)OC(C)(C)C)(OC)OC 46194,C1(C)(CNC(Cc2cn(C)nc2)=O)CCCN1C(=O)C=CI 46195,C=C(Cl)CC(C(=O)N(C1CC(C#N)C1)C)NC(=O)CNC(=O)C(C)CC 46196,C1(CNC(=O)NCC(c2cnn(C3CC3)c2)(C)C)CCCC(C2CC2)O1 46197,C1(C(=O)NCC(CC=C)NC(=O)C(c2ccc(F)cc2)CO)CCS(=O)(=O)CC1 46198,C1(CC(=O)N(CC(=O)NCCSCCC=C)CCC)CCC(=O)C1 46199,C1(C(=O)NC2CCC(NC(c3cn(C)nc3Cl)=O)CC2)COC2(CCC2)CO1 46200,c1(CC)ccc2c(Cl)c(C(=O)NC(CNC(C3(C#N)CC(C)C3)=O)CO)sc2c1 46201,CN1CCCC(CC(N2CCC(CO)(NC(=O)COCc3ccccc3)C2)=O)C1 46202,c12cc(F)c(F)cc1NC2=O.C(=O)(C(C)(C)C)NCCNC(C=C(C)C(F)F)=O 46203,c1(C2(C(=O)NCCNC(C3C=CCN3)=O)CC2)cccnc1 46204,N1(C(C(CC#C)O)=O)CCC2CCC(C1)N2C(c1ccc(Cl)cc1Cl)=O 46205,C1(CCC)CN(C(C2(C)CCNC2=O)=O)CCN1C(c1nnn(C(C)C)c1N)=O 46206,C(=O)(CCC(C)C)NC(C)=O.c12sccc1C(=O)NC1CC(C1)N(C)C2=O.CO 46207,c1(C(=O)NC2CN(C(CCCC(=O)OC)=O)C2)cc(O)nc(OC)n1 46208,C1(NC(c2cc(Br)no2)=O)(CO)CN(C(c2ccnn2CC(F)F)=O)C1 46209,N1(C(c2c(CC)n(C)cc2)=O)CC(C)CN(C(c2cc(=O)cc(Cl)[nH]2)=O)CC1C 46210,CCCCCCCCC(C)CC(=O)N1CC(CO)(NC(=O)C=C(C)C)C1 46211,C1(CNC(C2(COC)CC2)=O)CC2CCC1N2C(=O)C(c1ccccc1OC)C 46212,N1(C(C2C(C)C2)=O)CC(NC(=O)CCc2cnccn2)C2(CCS(=O)(=O)CC2)C1 46213,N1(C(C2(COC)CC=CC2)=O)CC(CCNC(c2nn[nH]c2Cl)=O)OC(C)C1 46214,Cc1c(C(C)N(C)C)cccc1Br.c12cn(nn1)C1(CC1)C(=O)N(C)C2C 46215,C=CCC(C)(CC)C(=O)N1C2CCC(C2)C1CC(=O)NCCn1cnccc1=O 46216,C1(OC)(CNC(C2(CCl)CN(C(=O)CC(C)O)C2)=O)CCOC1 46217,C1(CC(=O)N(CC(N2CC(O)(CC=C)C2)=O)CC2CC2)CCC(=O)NC1 46218,c1(NC(C2(C)CN(Cc3cncnc3)C2)=O)ccc(F)c(F)c1Br 46219,C1(NC(=O)C(F)=C2CCC2)CCN(C(C2CC(O)(C(F)(F)F)C2)=O)CC1CO 46220,C1(NC(c2c(COC)cco2)=O)CCCCC1CNC(c1cc[nH]c(=N)c1)=O 46221,C1(C(CC)C)CCCCN1C(C=Cc1ccccc1)C(=O)NCCCSC 46222,c1(C(N2CC(C(=O)NCC3C(OCC)CCC3)C2)=O)cc(CS(C)(=O)=O)c(C)s1 46223,N1(C(=O)CCCF)CCN(C(=O)COc2cc(F)cc(Cl)c2)CC(O)C1 46224,C12(C(=O)NC3(C(COC)OC)COC3)CC(C(C3(C(N)=O)CC3)=O)(C1)C2 46225,c1(OC(C)=O)nc(N2CCN(CCNC(c3cc(C)c(Cl)s3)=O)CC2)ncc1Br 46226,N1(C(CCC2CCC(C)O2)=O)CCC2CC(CNC(c3cnoc3)=O)CCC2C1 46227,c1(C(C(=O)NCCCC)N(C)Cc2cccc(C)c2F)c2c(nn1C)CCSC2 46228,C1(C(N2CCC(C(C)C)(C(=O)NC(C)CC(C)(C)O)C2)=O)CCC2(CC1)CC2 46229,CCCCC(C)(F)C(=O)NC1CC1CNC(=O)C=Cc1ccc(Br)s1 46230,Cc1ccc(OC(C)C(N2CC(CNC(C3(C#N)CCCC3)=O)C(C)C2)=O)cc1 46231,c1(N(CCNC(c2cc(C)sc2)=O)C2CC2)ncnc2cnn(C)c12 46232,CC(C)CC(C)CC(=O)NCc1cc(C(=O)Nc2cncc(C(C)C)c2)ccn1 46233,c1(OCC)ccccc1S(=O)(=O)Nc1cc(C)nn1C1CCCCC1 46234,N1(c2ncnc(=N)[nH]2)CCc2c(CNC(C3CCCC(C(N)=O)C3)=O)cccc2C1 46235,C1(C)(CNC(C(C=C=C)C)=O)CN(C(c2nc(O)nc(O)c2OC)=O)C(C)(C)C1 46236,CC(C)(C(=O)N1CC2CCC2(NC(=O)CC(O)C(Cl)(Cl)Cl)C1)S(C)(=O)=O 46237,CCCCCC(F)C(=O)NC(Cc1cnc[nH]1)C(=O)NC1CC(C)(C)OC1(C)C 46238,c1(C(=O)NC2C(C)CN(C(=O)CCN3C(=O)CCC3=O)C2)cc[nH]c2nccc1-2 46239,Cc1ccc(-c2ccc(-c3nc(-c4ccc(N)cc4)nn3CC(F)F)o2)cc1 46240,N1(C(CCOC)=O)CCC(O)(CNC(c2cnc(-c3ccccc3)s2)=O)CC1 46241,C(=O)(CS(=O)C(F)(F)F)N1C(CN(C)C(C23CCC(F)(CC2)CC3)=O)CCC1 46242,c1(CNC(c2nc(C)oc2)=O)nc(CNC(=O)CC(C)CF)cc(O)n1 46243,CCCC(C)C(=O)N1CC(CO)(CNC(C2CCCCC2)=O)C1.c12conc1C2 46244,N(C1COCc2ccccc21)C(=O)C(c1ccccc1)Sc1ccc(Cl)cc1 46245,C1(CC(=O)N(CCNC(=O)C(C2CCOCC2)O)CC2CC2)CCCCC1(F)F 46246,c1(OC)cc(C(=O)NCC(CO)NC(c2nnn(C)c2C)=O)cc2c1OCO2 46247,N1(CCC(=O)NC(C)(CNC(=O)C=C(Cl)Cl)Cn2cccn2)CCC(O)CC1 46248,N1(C(CCCN(C(=O)OC)C)=O)CCC(NC(C2CCCC2C)=O)C2(CCC2)C1 46249,c1(NCCOC)cc(=NCC2CC(OCc3ccccc3)C2)[nH]c(C2CC2)n1 46250,CC1CC(C2CN(C(=O)C(CC(F)F)N(C(=O)CCc3nc(O)n[nH]3)C)C2)=NO1 46251,N(C(=NCCc1nnc(C)n1C)N1CC(C)N(CCOC)C(C)C1)C(CC)C 46252,CC1(C)C(CNC(=O)Cc2ccnc(F)c2F)CCN1C(C1CSC1)=O 46253,Cc1cc(=NC(=O)C(=O)NCC2(CNC(C3CC34CCCC4)=O)CCC2)[nH]o1 46254,c1(OC)cc(C=CC(=O)NCC2(C)CCN(C(=O)C(CO)N(C)C)C2)sn1 46255,c1(C(=O)NC(CNC(=O)CC2CCCC2)CO)csc2c(Cl)cccc12 46256,N1(C(C(C)(C)c2nccs2)=O)CCN(C(=O)CSC2CCCCO2)CC(O)C1 46257,c1(CC(=O)NC2(CO)CCCN(C(=O)CCOC3CC3)C2)ccc2c[nH]nc2c1 46258,C1(C(N2CC(C)(C#N)C2)=O)CN(C(C2CC3COCC3C2)=O)CC12CC2 46259,N1(C(C(CC=C)C)=O)CC2(C(=O)NC3CN(C)CC3C)CCC1CC2 46260,C(CCC1CC1)(C(=O)NC1CC1c1ccco1)NC(C(C)n1ccnn1)=O 46261,Cc1cc(C(=O)NCC2CCCC2C(=O)NC(c2ncc[nH]2)C)ccc1O 46262,Cc1nc[nH]c1CN(C(=O)CCCn1cc(C(C)O)nn1)C 46263,Cn1cc(C(C)(C)C(=O)NC2CCC2NC(=O)CC2(c3ccon3)CC2)cn1 46264,c1(C(N2C(C3(O)CN(C(CC=CC=C)=O)C3)CCC2)=O)cnc(C)c(C)c1 46265,C(=O)(C1OC(=O)c2ccccc21)NCCN(C(=O)C=Cc1cnn(C)c1)C(C)C 46266,N1(C(C2C(C)C2)=O)CC23CCCCC2(C1)CN(C(C1(C#N)CCOC1)=O)C3 46267,C1(C(N2CC(NC(C3C4CS(=O)(=O)CC34)=O)C2)=O)CC2COCC(C1)C2 46268,c1(C(=O)NC2CCN(S(CCCC)(=O)=O)C2)cc(Br)c(O)c(Br)c1 46269,c1(C(N2C(C)CC(NC(c3c(CC)nccc3)=O)C2)=O)cccc2cccc(C)c12 46270,N1(C(CC(C)(C)C)=O)CCCOC(CNC(C2CC2c2c(F)cccc2F)=O)C1 46271,N1(C(C2N(CC)CC2)=O)CC=CC1(C)C(=O)NOCC1CC1 46272,C(CCN=C(NCc1ccc2c[nH]nc2c1)NCC1CCCC(C(F)F)C1)SC 46273,c1(CC(=O)NC2(CC)CCN(C(c3cncn3C)=O)CC2)cnn2ccccc12 46274,C(=O)(C(C)(C)CS(C)(=O)=O)NC1C(C)CCN(C(c2ncnc3sccc23)=O)C1 46275,c1(C(=O)NCC2N(C(C3(C(=O)OCC)CCO3)=O)CC2)c(C)cccc1Cl 46276,N1(CC(C)(C)C2CC2)CCC(C(N)=O)CC1.C1(CC(=O)N(C(C)C(N)=O)C)CCN(C)C1 46277,C1(NC(c2n(C)c(S)nc2)=O)CN(C(c2c(F)cncc2Cl)=O)CC1(C)C 46278,n1(CC)nnc(C)c1COC(c1ncc(CC2CCN(C)CC2)s1)=O 46279,Cc1ccc(C(=O)NC23CC2CN(C(C2(C)CC=CC2)=O)C3)c(Cl)c1 46280,c1(NC(CN2CCN(C(C(F)=CCC)=O)CC2)=O)ccc(C#N)cc1 46281,C1(NC(C(C)(Cl)Cl)=O)COC2(CCN(C(=O)COc3ccc(C#N)cc3)C2)C1 46282,c1(C(N2C(C)CCN(C(CC(C=C)(C)O)=O)CC2)=O)ccnc2ccc(Cl)cc12 46283,c1(C(=O)NCC2N(C(CNC(=O)OC)=O)CC(O)C2)cc(N)ccc1F 46284,C1(C(=O)Nc2c(C(N3CCC(CN(C)CC)C3)=O)[nH]cc2)CC12CCCCC2 46285,c1(C(=O)NC2(C)CC(NC(C3N(C(C)=O)CCC3)=O)C2)c(C)nn(C2CC2)c1Cl 46286,c1(C(=O)NC2CCN(C(C3(CCC)CC3)=O)CC2CO)n[nH]c2c1CCSC2 46287,C1(NC(c2cncc(C)n2)=O)(CNC(=O)C(F)C(C)C)CCC(F)(F)CC1 46288,C(=O)(CS(=O)C(F)(F)F)NCC(CCNC(C(CC)SC)=O)(C)C 46289,c1(CC)ccc(C(=O)NC2CCC(CNC(c3ccc([N+](=O)[O-])[nH]3)=O)C2)c(C)c1 46290,C1(NC(C(C)N(CCC)C(c2cc(C(F)F)[nH]n2)=O)=O)CC2(CCOC2)C1 46291,Cc1noc2[nH]c(=N)c(C(=O)NCCCC3CCCOC3)cc12 46292,Cn1cc(CC(O)C(=O)NCC2CC(NC(=O)CC3CCC=CCC3)C2)cn1 46293,N1(C(C(C)C)=O)CC(O)(CNC(=O)CCCN(C)C(C)C)C1 46294,N1(C(CCSCC)=O)CC2CCN(C(c3ccc(OC)c(N)c3)=O)CC2C1 46295,N1(C(C(=O)NCCCC)CC(C)CCC)CCC=C(c2ccco2)C1 46296,c1(C(N2C(C(N(CCCC)CCO)=O)CC3CC32)=O)cc([N+](=O)[O-])c(Cl)cc1Cl 46297,CC1CCCN(C(c2cc(-c3ccccc3)no2)=O)C1CNC(=O)CNC=O 46298,c1(OCC)ccc2[nH]cc(CN3C(=O)CCN(CCCCF)C3=O)c2c1 46299,c1(C(N2CC(NC(C(C)CC(C)(C)C)=O)C2)=O)cccc2c1C(=O)NC2 46300,C(=O)(CCCC(C)C)NCC(CCCC)NC(=O)Cc1csc(COC)n1 46301,c1(C(=O)NCC2C(NC(CCC(C)(C)OC)=O)CCCC2)cccc2ccnn12 46302,C1(NC(=O)CNC(c2ccccc2)=O)CC2CN(C(c3coc(CO)n3)=O)CC12 46303,CC1=C(C)CC(C)(C(=O)NCC2(CNC(C3CC(=O)N(C)C3)=O)CCC2)CC1 46304,CC1CCc2cc(C(=O)NCCN(C(=O)CC3(O)CCCCCC3)C)ccc2N1 46305,O=C(C1=CCN(C(C2CC2C2CCCC2)=O)C1)NCCN1CC2CC2C1 46306,c1(OCCOC)cc(OC)ccc1C(=O)NCC(C)(C)c1ccsc1 46307,N1(C(c2ccc(COC)o2)=O)CCN(C(C2CC(S(C)(=O)=O)C2)=O)CC1CO 46308,c1(NC(C)C)cnc(NC(=O)NOCCOCCO)cn1 46309,c1(CC)nc(C#N)cc(=NC(C)c2ccc(NC(=O)C(C)CC(C)CC)cc2)[nH]1 46310,c1(CC)ccc(C(C)C(N2CCC(N(C(=O)CSCC(F)(F)F)C)C2)=O)cc1 46311,c1(C(=O)NCC2CCC(NC(C3(OC(C)=O)CC3)=O)C2)cnc2c(C)cccn12 46312,CC1(C)CCC(F)(F)CC1C(=O)NC1CN(C(c2cc[nH]c2)=O)CCC1CO 46313,C1(CNC(C(=O)NCC)=O)C2CC1N(C(c1csc(-c3ccc(C)o3)n1)=O)C2 46314,C(C(C)(O)CC(=O)N1CCCCC1CNC(c1cc(C)sc1Br)=O)OC 46315,N1(C(c2cc(CC)oc2C)=O)CCCC2(NC(c3cn[nH]c3)=O)CCCC12 46316,Cn1cc(C(=O)NC2CC(NC(=O)Cc3cc(O)nnc3O)C2)c2ccccc12 46317,C(=O)(C(CC(C)(C)C)N1CCC(c2nc(C3CC3)no2)C1)NCCCSC 46318,c1(-c2cc(CNc3scc(OC)n3)on2)cccc(OC)c1OC 46319,C1(NC(c2c(C)nc(COC)s2)=O)CCN(C(=O)Cc2c[nH]nc2C)CC1CO 46320,Cc1cc(C(N2CCC(OCCNC(=O)Cn3cccc3)C2)=O)nn1C(C)C 46321,c1(C(=O)NC2C(C)CCN(C(C(COC)C)=O)C2)cc2cccc(Cl)c2nc1C 46322,C1(C(=O)NC(CCCNC(C(CSC)OC)=O)(C)C)Cc2cc(Br)cnc2C1 46323,C1(C(N(C2CCN(C(C3CC34CCCC4)=O)CC2)C)=O)CC(O)CN1C 46324,C1(CNC(=O)C=CBr)CCC(F)(CNC(=O)CCc2ncccn2)CC1 46325,N1(C(C2(C)CCNC2=O)=O)CCCC(NC(=O)CNC(c2ccccc2)=O)CC1 46326,C1(C(N2CCCC(NC(C(c3c(C)n[nH]c3C)C)=O)C2)=O)Cc2cscc2C1 46327,c1(CC)nc(C)[nH]c1C(=O)NC1CN(C(c2ccn(C3CCCC3)n2)=O)C2CC12 46328,c1(C(=O)NCCC(C)(C)NC(=O)CC(C)(C)C#N)cnn2c1OCC(F)C2 46329,CCCCC(CN=c1[nH]nc(CC)o1)NC(=O)C1=CCC1 46330,c1(C(=O)NC2CCC(N(C(CC)C(=O)NC)CC)CC2)cccc(Cl)c1O 46331,c1(CC(=O)N(CCOC)CCNC(=O)C(F)C2CCOC2)ncoc1C 46332,C(=O)(C1CCc2nccn21)N(CC(C)NC(CCn1c(C)ncc1)=O)C 46333,Cc1[nH]c2ccc(Br)cc2c1CCNC(=O)Cn1cc(Br)c(=O)c(I)c1 46334,C=C(C)CC(C(=O)NC1CCCN(C(C2CCCN2N=O)=O)C1C)NC(C)=O 46335,Cc1cccc(F)c1C(=O)NC1CCC(NC(C2(F)CC=CC2)=O)C1 46336,C(C(C(=O)NC(Cc1ccco1)CO)N(C)C)NC(C(C1CCC1)OC)=O 46337,Cc1cnc(C(=O)NC(C)(C)CNC(=O)CCc2cnc(C)nc2O)c(Br)c1 46338,c1(C(=O)N(C2CCS(=O)(=O)C2)C(c2nocc2C(=O)O)C)n[nH]c2ccccc12 46339,C1(NC(CCOCC#C)=O)CN(C(c2c(C)noc2CC)=O)CCC1CO 46340,N1(C(C(N2CCNC2=O)C)=O)CCC(C(=O)NCCN2CC3CC3C2)C1 46341,C1(CC(=O)NC(C2CCN(C(=O)C(C)C(C)C)CC2)(C)C)(COC)CCOCC1 46342,C1(CNC(c2ccn(CC)n2)=O)CN(C(C23CCC(CC2O)C3)=O)CCN1C 46343,C(=O)(CC(CC(C)C)NC(C)=O)NC(CC)CN(C(=O)C1=CCCOC1)C 46344,C(=O)(CCCS(C)(=O)=O)N1CCCC(C)(NC(=O)CC(C)(C)c2ccccc2)C1 46345,n1(CC)nc(C(C)C)cc1C(=O)NCCN(C(c1cc(C(N)=O)n(C)n1)=O)CC 46346,C1(CCOC)CCCCN1C(C1CN(C)NC1=O)=O 46347,c1(C(N(CC(C)NC(c2ccn(COC)n2)=O)C)=O)cn(C)nc1Br 46348,C(=O)(C1=NOC(c2ccc(Cl)cc2Cl)C1)N1CC(C)C(NC(=O)C2CC2)C1 46349,c1(C(N(C(CC)C(=O)OC)C)=O)coc2c1CN(C(=O)C(c1cncnc1)C)C2 46350,C(C(CC(C)C)NC1C(C)CCN1C(=O)COCC1CC1)NC(C)=O.c1c(=O)n1 46351,CC(C(CO)NC(C1CCO1)=O)NC(c1cc(Cl)ns1)=O 46352,c1(OC)cc(NC(=O)C(=O)NC(C)Cn2cnnc2)ccc1C(C)(C)C 46353,CCC(CC(=O)NCCC(=O)NCC(C)(O)C(C)C)C1CCC1 46354,C1(C(=O)NC(C2CCN(C(=O)CC34COCC(C3)C4)C2)C)C2CCCCCC12 46355,C1(C(C)NC(=O)C=CC(=O)NC2CC2)CCCCN1C(C1CC2CC1C2)=O 46356,c1(C(=O)NC(C)C(C)(C)NC(c2ccn(CCO)c(=O)c2)=O)cc(O)cc(O)n1 46357,C(C)(c1ccco1)=CC(=O)N(C(C)C(=O)NC1CCC(C(N)=O)CC1)CC 46358,CCCCC(CC(=O)NC(CSC)CC)NC(=O)C=C1CCC(C)CC1 46359,C(=O)(CC1COCc2ccccc21)NC(C1CN(c2cc(Cl)ncn2)CCO1)C 46360,C(=O)(CCCC(C)(C)C)N(C1CCN(C(=O)CN(c2ncccn2)C)CC1)CC 46361,O=C(C#CC1CCCO1)NC1CCN(C(=O)Cc2nsc3ccccc23)CC1F 46362,C(C)(C(=O)N(C(C)C(=O)N(C)CCn1cnnc1)C)N(C(C)=O)C 46363,C1(CNC(C(C)=CC)=O)CCCCN1C(c1cn(C)nc1COC)=O 46364,CCC(CNC(C1CCOC(C)C1)=O)(CC)C(=O)N1CC2(C1)CC2(F)F 46365,N1(C(c2cccc(OCC#C)c2)C(=O)NC2CCCCC2)CCOCC(C)C1 46366,C(=O)(C(F)C(C)(C)O)N1CC(CCO)(NC(C2C(C(=O)OC)C2)=O)C1 46367,C1(CNC(C2N(CC)CC2)=O)CN(C(c2c(Cl)c(C)nn2C)=O)CCC1(F)F 46368,S(=O)(=O)(c1ccccn1)NC1CC(C(N2CCN(C(C)C)CC2C)=O)C1 46369,N1(C(CC(CC(C)(C)C)O)=O)CC(CNC(C2(F)CC2)=O)CC12CCOCC2 46370,c1(CC)ncncc1C(=O)N(CCCNC(C1CCN1S(C)(=O)=O)=O)C(C)C 46371,C#Cc1ccccc1CN=C(NCC(F)F)NCC1(OCC)CCOC1 46372,N1(C(C2(CCOC)CC2)=O)CC=CC(NC(C23CCCC2(C(N)=O)C3)=O)C1 46373,C1(NC(Cc2cc(C)nn2C)=O)(CNC(C2COC(=O)N2)=O)CC2CCC1CC2 46374,CC(C)CCCC(=O)N(C1CCN(C(C2CC(C)CCC2C(C)C)=O)C1)CCO 46375,c1(CC(=O)N(C(C)CCNC(=O)Cc2cccnc2F)C)c(F)cccc1F 46376,C(=O)(CCCS(C)(=O)=O)NCC1C(C)(C)N(C(=O)C(=O)Cc2ccccc2)CC1 46377,N1(C(c2sc(C)c(C)c2C)C(=O)NCCOC)CC2CCC(C1)C2O 46378,N1(C(c2cnc(C)o2)=O)CC(NC(=O)C(C)Cn2ccnc2)C2(CCCC2)C1 46379,NS(=O)(=O)c1ccc(C(=O)OCc2ccccc2C(=O)C(F)(F)F)cc1 46380,C1(C#N)(C(=O)NCCCN(C)C(c2cn(C)c(=O)n2C)=O)CC12CCCC2 46381,C1(C(N(CC(=O)NCC(CSC)(C)O)CC2CC2)=O)C2CC(=O)CC12 46382,N1(C(C(C)NC(C)=O)=O)CC2CCN(C(=O)CCN3CCOCC3)C2C1 46383,CCC(CC(=O)NC(C)CCN(C)C(c1cc(C2CC2)ccn1)=O)C(C)C 46384,C(N=c1[nH]nc(C(N)=O)s1)C1(NC(c2n(CC#N)ncc2)=O)CCCCC1 46385,c1(C(=O)NC(CN(C(C2(C(F)F)CC(=C)C2)=O)C)C)nc2ccccc2n1CC 46386,c1(C(=O)NCC2CCCN(C(C(C(=O)OCC)F)=O)C2)ccnc2nc(C)nn12 46387,CCCC(C)C(=O)N1CCC(N(C(=O)CCC#N)CC2CC2)C1 46388,CCCCCCC(=O)N1CCC(O)C(C(=O)NCc2csc(C3CCCO3)n2)C1 46389,C1(NC(c2ccc(N(C)C)nc2)=O)(CO)CCCN(C(=O)Cc2ccsc2Cl)C1 46390,c1(CC)ncc(C(=O)NCC(N2CCN(C(C3CNC(=O)N3)=O)CC2)C)c(O)n1 46391,C1(C(=O)NC2CCCN(C(COCCCOC)=O)CC2)Cc2ccccc2S1 46392,c1(C2(C(=O)NC3CCC(CCNC(CCC#C)=O)C3)CC2)cccc(F)c1C 46393,c1(CC)nc(=NCCOCCNC(c2ccn3nnnc3c2)=O)s[nH]1 46394,C(C)(C)(CN=c1[nH]c2cc(Br)ccc2o1)NC(Cc1c(C)noc1Cl)=O 46395,c1(CC(=O)NC2C(C)(C)C(CNC(=O)COc3ccsn3)C2)ccc(F)c(Cl)c1 46396,O=C(N=c1[nH]c2sccc2s1)c1cncc(NC(c2ccccn2)=O)n1 46397,CC(COc1ccccc1)C(=O)NNC(=O)CN(C)C 46398,C#Cc1cnc(C(=O)NCC2C=CCN2C(c2cc3nc[nH]c3cn2)=O)c(C)c1 46399,S(=O)(=O)(c1ccc(Cl)s1)NC(C)C(N1CCC(N2CCCC2)CC1)=O 46400,N1(C(C=C)=O)CCOC(C(C)NC(C)=O)C1.C(c1ccco1)=C(C)Cl 46401,C1(C(=O)NCC2(O)CN(C)C2)CSCCN1C(C1CCC(O)CC1)=O 46402,C(=O)(C1=CNC2=NCCC2=C1)N1CCN(C(C2C(OCC)C2)=O)CC1C1CC1 46403,c1(N2CCCC(C)(CNC(c3n(CC)ccc3)=O)C2)ncnn2cccc12 46404,C1(CCNC(C2CC(=C)C2)=O)CCN(C(=O)CNS(=O)(=O)CCOCC)C1 46405,C(c1ccc(S(=O)(=O)NC2CC2)cc1)=CC(N1CC(NC(C(CC#C)O)=O)C1)=O 46406,Cc1nn(C)c(C(F)F)c1C(=O)NCCNC(C12CCCC1CCC2)=O 46407,CCCS(=O)(=O)N(C)CCOCCNC(C1(C(C)C)CCC1)=O.C1(O)CN(C=O)C1 46408,C1(CNC(CCSC)=O)CCN(C(C2(C3CCCCO3)CCC2)=O)CC1C 46409,c1(C(=O)NCC(C)C)ccc(F)c(NC(=O)CCc2ccccc2Br)c1 46410,N1(c2nnc(CCOC)s2)CCCCC(NC(c2cccc(=O)n2C)=O)C1 46411,N1(C(CCCNC(=O)OC)=O)CC2(C1)CN(C(=O)CC1CC(C)(C)CO1)C2 46412,C1(NC(CCc2cnc(C)s2)=O)C=CCN(C(C2C(C)(C)C2(F)F)=O)C1 46413,c1(CNC(C2C(O)CCN(C(CCC=C)=O)C2)=O)ccc2nc[nH]c2c1 46414,N1(C(c2cnc(C)n2C)=O)CCC2(NC(=O)CCc3cncnc3)CCCC12 46415,N1(C(c2c(OCC)nccc2)=O)CCC(C)(C(=O)Nc2nc3sccc3s2)CC1 46416,N1(CC(=O)NCC2(C)CCCN2C(=O)CS(C)(=O)=O)C(=O)C2CCCCC2C1=O 46417,C1(C(=O)NC(CC)(C)C2CC2)C2CC1N(C(=O)C(=Cc1cn[nH]c1)C)C2 46418,C1(C(=O)N(C)CCN(C)CCO)(CC)CCN(C(c2cc(O)nn2C)=O)C1 46419,c1(C(=O)NCC2CCCC(C#C)C2)coc2c1CN(C(=O)Cc1cncnc1)C2 46420,C1(CNC(C(=O)NCC2CC2)=O)CC12CCOC2.c12occc1C(=O)NC2 46421,C(=O)(C(C(C)(C)C)SC)N(C(CN(C(c1c(OC)cccn1)=O)C)C)C 46422,C1(C(N(CCNC(=O)CC2COC3CC2C3)CC)=O)(OC)CCCCCCC1 46423,C1(C(N)=O)CN(C(C2CC3CC3N2C(=O)CCCN2CCCC2)=O)CCO1 46424,N#Cc1ccc(C2CC2CNC(C2CCOCC2)C(F)F)cn1 46425,Cn1ccnc1C(N1CCC(n2cc(CCN(S(C)(=O)=O)CCN)nn2)C1)=O 46426,N1(C(CC2(OC)CN(C(C3(n4cccc4)CC3)=O)C2)=O)CC(C#N)(C(C)C)C1 46427,C1(CCNC(CC2CN(C)C2)=O)CCN(C(=O)C(N)=O)C1 46428,C1(C(=O)NCC2(C(C(C)C)O)CC2)CCC=CCC1 46429,c1(C(N(C(C)C)CCN2CC=CCC2)=O)cccc(C#N)c1.C1(C)C(=O)N1 46430,c1(C(=O)NCC2CCN2C(c2cc[nH]c3nccc2-3)=O)cc(F)c(F)c(Cl)c1F 46431,c1(C(N(C2CN(C(C3CN(C(N)=O)C3)=O)CC23CC3)C)=O)n[nH]c2ccc(F)cc12 46432,C(N=c1[nH]c2cccc(F)c2s1)C1C(C)CN(C(c2cc3n(n2)CCCC3)=O)C1 46433,CCC(C)(C)CCCC(=O)NC1CN(C(=O)C(COC)N(C)C)CCC1(C)C 46434,CC1(COC(c2ccc3ncc(Br)n3c2)=O)COCC2CCCN12 46435,C(c1ccc(OC(C)C)cc1)=CC(=O)NC(CN(C(CC(=O)NC)=O)C)CC 46436,C1(c2cn(Cc3cnn(CCCOC)c3)nn2)(C(=O)OC)CCOC1 46437,C12(C(N(CCCN(C(C3(COC)CC3(F)F)=O)C)C)=O)CCC(COC)(CC1)C2 46438,N1(C(CCOCCOC)=O)CC2CCN(C(C3(C)CCCN3C)=O)CCC2C1 46439,c1(OC)ccc(N2CCCC2=O)cc1.N12CCC(CC1)CC(=O)NCCCC2=O 46440,C(C)(C)(CC(C)NC(=O)CCN(C(c1ccc(C)s1)=O)CC1CC1)OC 46441,c1(C(N2C(C)CN(C(c3csc(C#N)c3)=O)C(C)C2)=O)ccc2c(c1)CCN2C 46442,C1(N(C(c2cnc(C(C)C)s2)=O)CC)CCCN(C(C2(C#N)CCOC2)=O)CC1 46443,N1(C(C(CC=C)OC)=O)CCC(CNC(c2cnc(COC)nc2O)=O)C(C)C1 46444,c1(C(=O)NC2C(C)(C)CN(C(=O)C(F)C(C)(C)O)CC2)ccc(O)c([N+](=O)[O-])c1 46445,C1(O)(C(=O)NCCCN(C(c2cc3ccncc3o2)=O)CC)CCCC(C)CC1 46446,N1(C(Cc2nc(COCC)on2)=O)CCOC(CCCNC(C2CC2(C)C)=O)C1 46447,c1(CCC(=O)NCCC(C)NC(C2CC2c2cnn(C)c2)=O)c(F)cccc1Cl 46448,CCC(CC)(CO)C(=O)NCC(C)(F)CNC(c1ccc(N)cc1F)=O 46449,Cc1cc(C(N2CCN(C(=O)Cc3cnsc3)C3CC23)=O)c(C)nc1C 46450,C#CCC(C)(C)C(=O)NC1CCCCC1NC(=O)Cc1ccsc1C 46451,c1(CC)nn(C)c(CC)c1CNC(c1ccc(F)cc1)c1nnnn1C1CCC1 46452,N(C(=NCC1CCC(=O)N1C)NC1CCC(O)CC1)C(COC)C 46453,C1(CNC(=O)CC2CCC(C(F)(F)F)O2)CCN(C(C2C3CNC(=O)C23)=O)CC1 46454,Cc1cc(=NCC2CCOC2)[nH]cc1S(=O)(=O)N1CCCC1 46455,c12ccc(cc1)NC(=O)C(=O)O2.c1(SCC)ccccc1OCCCCC 46456,c1(C(=O)NCCCN(C(CSCC#C)=O)C)ncc(C)cn1 46457,C(CCCC(=O)N1CC(C(=O)NC(c2ccccn2)C)CCC1C)(OC)OC 46458,Cc1cc(C(=O)NCc2nc(C(N3CC(N4CC(F)C4)C3)=O)c(C)o2)c(O)nn1 46459,C1(C(N(CCCNC(=O)CC2CCCC2(F)F)C)=O)CCN(C)S1(=O)=O 46460,C(=O)(CCC1=CCCCC1)NCC(C(=O)NC1CN(C)CC1O)O 46461,C1(N(S(c2c(C)onc2)(=O)=O)C)CCc2ccccc2C1 46462,C(=O)(C1=NOC(CNC(c2cncc(O)c2)=O)C1)NC(C#C)C1CCC1 46463,CC(C)(CNC(=O)CC1CCCC(C2CC2)O1)CCNC(=O)Cc1ccns1 46464,N1(C(=O)NC2CC(COc3ccccc3)C2)CCCC2(CCCNC2=O)C1 46465,N(C(=NCCC12CCC(CC1)OC2)N(C)Cc1cnn(C)c1)CCC(=O)NC 46466,N1(C(c2cc(C)no2)=O)CC(C)(C)CC1CNC(c1nnc(C)cc1O)=O 46467,C1(C(=O)NC(c2cc(C)on2)C)CCN(C(C2CN(C)C(=O)N2)=O)CC1O 46468,c1(C(=O)NCC2C(C)(C)N(C(=O)CC3CCCO3)CC2)cnn2cccnc12 46469,Cc1cccc2cc(CN3CCCC3NC(C)COc3cccc(F)c3)cnc12 46470,CC#CCCC(=O)NCC(C)NC(=O)C(C)CC1CCCCC1 46471,c1(NC(C2CSCCN2c2ccncn2)=O)cc(Br)cc2cn[nH]c12 46472,C12(NC(CC(C)NC(=O)C#CC3CC3)=O)CCC(CC1)C2(C)C 46473,C1(C(=O)NCCC2(OC)CN(C(=O)Cn3cccn3)C2)CCOC(=O)N1 46474,C1(NC(C(=O)N(C2CC(CNC(C3CC3)=O)C2)C)=O)CC(C#N)C1 46475,Cc1c[nH]nc1C(=O)NC(CO)C(=O)N1CCCC1 46476,C(=O)(CCC1CCc2ccccc21)N1CCN(C(c2c(C)scc2)=O)CC1CF 46477,N1(CC)N=C(C(=O)N2CCCC2C(C)(C)CNC(=O)CC2CC=CC2)CCC1=O 46478,C(=O)(C(CC1CCOCC1)NC(=O)C=CC1CCC1)NC(C(C)F)C 46479,Cc1cc(C(=O)NCCC2CCCN2C(=O)C=CC2CCOC2)c(Cl)cc1Cl 46480,c1(C(=O)NCCN(CCC)C(C2CCCCC2C(=O)OC)=O)cnn(C)c1CC 46481,CC(C)(C)S(=O)Cc1cccc(NC(=O)COC2CC2(F)F)c1 46482,N#Cc1ccc(C(=O)NCC2(CNC(C34COCC3C4)=O)CC2(F)F)[nH]1 46483,c1(CNC(C=C(CC)CC)=O)cccc2c1CN(C(C1(COC)CCC1)=O)C2 46484,CCC1CN(C(C23CC4(F)CC(F)(C2)CC(C3)C4)=O)Cc2ccccc21 46485,CCC(C(=O)OC)C(=O)NCCCN(C(C1CC2CCC1O2)=O)CC 46486,N1(c2nccc(Br)c2)CCC2CCCCC2C1 46487,CCC(C)CC(C(=O)Nc1cnc(Cl)c(C)c1)NC(c1cnn(C)n1)=O 46488,c1(C(=O)NCCNC(c2cnn[nH]2)=O)ccc(-c2ccccc2)cn1 46489,CC1CCCC(C(N2CCCCC2CNC(c2cc(=O)n(C)cn2)=O)=O)CC1 46490,C1(C(C)C)CC(CC(=O)N(C)CCN(C)C(c2c[nH]c(C(F)(F)F)c2)=O)CCO1 46491,c1(OCC#C)ccc(C(=O)NCC2CN(C(C3(O)CC(C)(C)C3)=O)CC2O)cc1 46492,CC1CCOC(c2nnc(CCCCCS(C)(=O)=O)o2)CN1c1nnn(C)n1 46493,Cc1cc(C#N)cc(C)c1C(=O)NC1CCN(C(c2ccc(Cl)[nH]2)=O)CC1 46494,c1(OCC(N2CCN(c3ccc(C(F)(F)F)cn3)CC2)=O)ccc(F)cc1O 46495,c1(OC)ccc(N(C(=O)CC2CCCN2C(C)=O)CC2CCN2C(C)(C)C)c(C)c1 46496,Cc1ccc(Br)c(NC(c2cc(-c3cccc(N4CCOCC4)c3)cs2)=O)c1 46497,N1(C(C2CC2NCc2c[nH]nc2-c2ccccc2)=O)CCN2CCCCC2C1 46498,N1(C(c2cc(SC)oc2C)=O)CCC2(CCCN(C(=O)C=C3CC3)C2)C1 46499,Cc1nn(C)c(C)c1C(N1CC2C(CNC(C3CN(C)CC(C)O3)=O)C2C1)=O 46500,O=S(=O)(c1[nH]c(=NCC2C(F)(F)C23CCCC3)ccc1Br)NC1CC=CCC1 46501,Cc1cc(C(=O)N(CCN(C)C(c2scnc2C2CCCC2)=O)C(C)C)no1 46502,C1(CN(C(=O)C(C2CC2)NC(C2(C(N)=O)CC2)=O)C)CC1(C)C 46503,c1(C(N2CCC(CNC(C(CC3CC3)OC)=O)C2(C)C)=O)cccc2ccnn12 46504,c1(C(=O)NCC2C(C)CCN2C(=O)CSc2ccc(O)cc2)ccc(F)cc1Cl 46505,N(C)(S(C)(=O)=NS(=O)(=O)c1[nH]c2ccc(Cl)cc2c1Br)CC#C 46506,O=C(NNc1cc(C(F)(F)F)ccn1)c1cnc(C2CCC2)[nH]c1=O 46507,C1(NC(N(CCC)CCC)=O)(Cc2ccc(F)cc2)CCNCC1 46508,N1(C(C(C(C)O)(C)C)=O)C2CCC1CN(C(c1cn(C3CC3)nn1)=O)CC2 46509,C1(C(N2CC(CC(C)NC(=O)C=CCN3CCOCC3)C2)=O)CCC2CC1CO2 46510,CC(C)(C(O)C(F)F)NC(C1CN(C(c2cc(Cl)c[nH]2)=O)CC12CC2)=O 46511,Cc1cc(=O)oc(C)c1C(N1CC(NC(C2COCCN2CC2CCC2)=O)C1)=O 46512,CCCC(CCC)C(=O)NC1CN(C(c2cc(C)c(OC)c(Cl)c2)=O)CC1C 46513,C#Cc1ccc(C(=O)NCCC2(C)CCN(C(c3cncc(OC)c3)=O)C2)cc1 46514,c1(C(=O)NC2C(c3ccc(Br)cc3)(CC)C2)ccc(S(C)=O)c(F)c1 46515,C1(C(N2CCC(O)(CC)CC2)=O)CN(C(=O)Cc2cccc(F)c2)CCC1(C)C 46516,N1(CC(=O)NC(C(=O)N(CCOCC)CC)C2CCCO2)CCC(=O)CC1 46517,Cc1nc(C)n(CCC(=O)NCC2CCN2C(=O)C(N2CCOCC2)C2CC2)n1 46518,N1(C(c2ccn(COC)n2)=O)CC(OC)CC1CCNC(c1nocc1Cl)=O 46519,N1(C(c2c(C)ccnc2O)=O)CCCCC(NC(c2cn(C)nn2)=O)CC1 46520,C(=O)(CC1CCOc2ccccc21)NCC1C(NC(CCN(C)CCO)=O)CC1 46521,N1(C(C(c2ccc(F)cc2)C)=O)CC2CC1C2NC(=O)CS(C)(=O)=O 46522,CCC(CC(=O)N1CCC(CN=c2nc(C3CC3)[nH]s2)(C)C1)C(F)F 46523,C1(CCC)(NC(=O)Cc2ccc(F)cc2)CCN(C(c2nnc(S)n2C)=O)CC1 46524,Cc1c(C(C(C)C)NC(N2CCOC(c3ccccc3)C2)=O)oc2ccccc12 46525,c1(C2C(=O)N2)ccc(-c2ccccc2)o1.C1(N(C)CC2CCOC2)CCCCC1 46526,N(C1CC2(CN(C(c3ccnn3C)=O)C2)n2ccnc21)C(CC(=O)NCC#C)=O 46527,C(=O)(CC(O)C(C)C)NC1CCC(CC(=O)NCc2cc(C)ncn2)CC1 46528,c1(C2(C(=O)NC(CNC(CSC(C)(C)C)=O)CO)CCC2)ccc([N+](=O)[O-])cc1 46529,Nc1ccnc(C(N2CCC(F)(CNC(=O)CC3CSCCS3)C2)=O)c1Cl 46530,CCCCC(C(=O)NOC(C)CC)NC(c1nonc1N)=O 46531,c1(C(N2CCC(CN(c3nnc(C(C)C)o3)C)C2)=O)c(Cl)cccc1Cl 46532,N1(C(c2c(C)cccc2)=O)C(C(=O)O)CCCC1C 46533,C(=O)(C1CCCc2scnc21)N1C(C)CN(C(=O)COC2CCCCC2)CC1 46534,c1(CC(=O)NCCC2CC(NC(c3cn(C)[nH]c3=N)=O)C2)nsc2ccccc12 46535,c1(C(=O)NC2C(C=C)CN(C(=O)COCCC)C2)cc(S(N)(=O)=O)c(C)s1 46536,c1(C(=O)NCC2N(C(C(F)OC)=O)CCC2C)cc(O)nc(C2CC2)n1 46537,N1(C(C=C(C)CNC(C2CCC(C)(C)C2)=O)=O)CC=C(CO)CC1 46538,CCC(C)CCCCC(=O)NCC(Cc1ccccc1)C(=O)N1CC(C)C(C)C1 46539,C(CC(C)C(C)C)NC(C(CN(C)C)NC(Cc1scc(C)c1)=O)=O 46540,c1(C(N2CC(NC(c3c(C)ccs3)=O)C(C3CC3)C2)=O)cc2nc(Cl)ccc2o1 46541,N1(C(CC=CCC)=O)CCn2c(CNC(C3C(Cl)(Cl)C34CC4)=O)nnc2C1 46542,C1(CNC(c2c(C)con2)=O)CCN(C(C2CCOC2)=O)CC1C1CC1 46543,N1(C(C(C)N(C)C)=O)CCCN(C(c2cc(C(F)(F)F)ns2)=O)CC1C 46544,c1(CN2CC3(CCC(C(=O)Nc4ccnnc4)O3)C2)ccc2nc(O)[nH]c2c1 46545,CCP(=O)(CC)c1ccccc1C(N1CCCC1CNC(=O)CCC(N)=O)=O 46546,Cc1oc(C(C)C)cc1C(=O)NCCC1CCCN1C(C1CC(O)C1)=O 46547,Cc1ncnc(C(=O)NCC2CCC(NC(c3c(C)nn(C)c3Cl)=O)C2)c1C 46548,Cc1oc2ncnc(O)c2c1C(=O)NC1CCN(C(c2cc(Cl)no2)=O)CC1O 46549,n1(CCN(C)C(C2(C(F)(F)F)CCO2)=O)cc(C2CCCCO2)nn1 46550,c1(OC)cc(NC(=O)NCC2(O)CCOCC2)ccc1F 46551,C(C)(CC(C)N=c1c(C#N)c[nH]c2ccccc12)NC(C1CC(CC)OCC1)=O 46552,n1(CCC)ccc(-c2nc(-c3ccc(C(F)(F)F)o3)no2)n1 46553,c1(CC)nc(N2CCCC(NC(=O)C(C)Cc3c(C)n[nH]c3C)C2)cc(Cl)n1 46554,N1(C2CCN(C(=O)CC3COCCO3)CC2)CCN(C(c2cnns2)=O)CC1=O 46555,C1(NC(C2(CCC)CC2)=O)CC2CC(C1)N(C(c1cc(CC(=O)OC)on1)=O)C2 46556,C1(NC(c2c(C)noc2N)=O)CN(C(c2ccccc2)=O)C2(CCOC2)C1 46557,CC(C)CCCC(C)C(=O)NC1CCC(C)N(CC(=O)NC(C)C)C1 46558,N1(C(=O)CCCn2cncn2)CC2CC2(C(=O)NC2CC23CCC3)C1 46559,C1(C(=O)NC2CN(C(C)C)CC2C)(CC)CCCN1C(=O)CS(C)(=O)=O 46560,CCC(C)C(C)CNC(C1CC(=O)CN1C(=O)CC1CCC(C)CO1)=O 46561,c1(C(N2CC(N(C)Cc3ccc(Cl)s3)C2)=O)cc(O)cc(Cl)c1 46562,c1(C(=O)NC2C(CNC(CN(C(C(C)C)=O)C)=O)COC2)cnn2cccc(Cl)c12 46563,c1(C(=O)OCC(=O)Nc2c(C)cccn2)cccc2c1C(=O)OC2(C)C 46564,C(=O)(CC1=CCCCC1)NC(C(C(C)C)C)CNC(=O)NC1(C)CC1.C(C)(C)(C)O 46565,N1(C(Cc2c(C)nc[nH]2)=O)CCC2CCN(C(=O)CNC(N)=O)CC12 46566,c1(C(=O)NC2C(CNC(C=COCC)=O)COC2)cccnc1Sc1cc[nH]n1 46567,N1(c2nccc(SC)n2)C2CCC1CN(C(=O)C(C)Cn1ccc(C)n1)CC2 46568,n1(CC)c(=O)nc(O)c2c(C(=O)OCCCCCC(F)F)cc(C3CC3)nc12 46569,C12(C(N(C(CCNC(C(C=C=C)C)=O)C)C)=O)CC3CC1C2C3(F)F 46570,c1(C(N2C(C)C(NC(=O)C(O)Cc3cnc[nH]3)CC2)=O)ccc([N+](=O)[O-])c(O)c1 46571,C1(CC(=O)NCCS(N)(=O)=O)C2CCCC2N1C(=O)COC1CCC1 46572,c1(C(=O)OC)ccc(C(=O)NCCCC(C)(C)NC(C2CCS(=O)(=O)N2)=O)cc1 46573,C1(NC(C(C2CCC2)OC)=O)CC(O)(CNC(C2CCCN2C(N)=O)=O)C1 46574,C(=O)(C1=CC2CCCC12)N1CC(CC(C)NC(C2(CCOC)CCCC2)=O)C1 46575,C(C(C(C)C)NC(=O)CC1(OC)CN(C(=O)CC(C)n2cccc2)C1)OCC 46576,C(=O)(CC(C)(C)C(=O)NC1CN(C(c2cn(C(F)F)cn2)=O)C1)OC 46577,c1(NS(c2ccc(C)cc2)(=O)=O)ccc(C2=CCC(O)CC2)s1 46578,C1(COC)(CNC(=O)CCN(C)CCO)CCN(C(C2CCCC2C)=O)CC1 46579,CC(C)C(O)C(=O)N1CC(NC(C2(O)CC(CF)C2)=O)C(O)C1 46580,c1(C(N2C(C(C)NC(=O)Cc3ccno3)CCC2)=O)cc(Cl)ccc1Cl 46581,c12cc(oc1C)C(=O)NCCNC2=O.c1(COCC)ccsc1C(=O)OC 46582,c1(C(=O)NCC2(F)CN(C(C(N=S(C)(C)=O)=O)=O)C2)ccc(F)c2ccccc12 46583,c1(C(N2CCC(NCc3cn(CC(=O)NC)nn3)CC2)C)ccc(F)cc1F 46584,C1(CC)(CC)CCCN(C(=O)CC2CCN2C(c2ccc(O)cn2)=O)C1 46585,CCCC(C(=O)NC1C2CN(C(c3cnn4ncccc34)=O)CC12)C(C)C 46586,c1(C(N2CCCC(CCNC(CCC=CC)=O)C2)=O)cc(N)c(C)cc1C 46587,c1(C(=O)NCCNC(C2CCCN(C(C)=O)C2)=O)ncc(Br)cc1F 46588,CCC(CC)C(F)C(=O)N(C)CC1COCCN1C(=O)CCc1csnn1 46589,c1(OC)ncc(C(=O)NC2CCC(N(C)C(c3cnc(CC(C)(C)C)o3)=O)C2)s1 46590,c1(C(=O)NC2CC(O)(CNC(C(C)OCCC#C)=O)C2)cc(F)c(F)c(F)c1 46591,N1(C(C=C(C)C)=O)CC2CC(F)(F)CCC2(NC(c2cc(Cl)cnc2O)=O)C1 46592,c1(NC(=O)C(=O)NC2CCSC2)ccccc1.C12CC(C1)N2 46593,N1(C(CN(CCC#C)C)=O)CCN(C(=O)CCS(=O)(=O)CC)C2CC12 46594,N1(C(C(C)(C)SC)=O)CC(NC(C2CN(C3COC3)C2)=O)C(SC)C1 46595,c1(C(=O)O)cc2cc(CNc3ccc(C(F)(F)F)cc3F)sc2s1 46596,Cc1oc2c(F)c(F)c(F)c(F)c2c1C(=O)NC1CC1(C)C(F)F 46597,N1(C(COC2(C)CN(C(C3N(C)C(=O)OC3)=O)C2)=O)CCc2n[nH]cc2C1 46598,C1(CC(=O)NC)CN(C(=O)CCSC)CCN1C(=O)CCC1CCC1 46599,c1(CC)ncccc1NC(=O)CCC1(NC(=O)CCCF)CCC1 46600,C(=O)(C1CCCc2ncccc21)NCC1(F)CN(C(C2(C)CCCC2)=O)C1 46601,c1(C(=O)NC2C3(CCN(C(C(CC)O)=O)CC3)C2)c(C)nc2ncccn12 46602,CN1CC(C(=O)NCC23CC(NC(c4ccnc(C(N)=O)c4)=O)(CO2)C3)CC1=O 46603,N1(C(Cc2n(C)ncc2)=O)CC2CC2(C(=O)NCC(F)CO)C1 46604,CC1CCN(C(=O)CC(C)n2cccn2)C(C)C1NC(c1ccccc1F)=O 46605,c1(C(N2CCC(N(C(C(C)NC(CC)=O)=O)C)C2)C)ccccc1Cl 46606,c1(N2CCC(C(=O)Nc3nccnc3F)C2)ncnn2cc(Br)cc12 46607,C1(C)(CC(=O)N(CC(CNC(c2nccc(CC)c2)=O)O)C)CCS(=O)(=O)N1 46608,CCC1CC(=O)N1C.C(=O)(CCCN(C)C(C)C)N.C(C)(CCC)C(C)C 46609,N1(C(C2(C(C)C)CCCN2C(=O)C(C2CCCCC2)C)=O)CC2CCCC(C2)C1 46610,C1(C(=O)NCC2(O)CCN(C(C3CCCC(F)C3)=O)C2)CCC2C(CC1)C2(F)F 46611,C1(NC(c2nc(CNC(c3cc(OC)nn3C)=O)oc2)=O)CCCCC1N=[N+]=[N-] 46612,c1(CC)nc[nH]c(=NCCC2CC2(C)C)c1F 46613,C1(c2ccccc2)(C(=O)NC(CNC(CSCC)=O)CO)CCOC1 46614,CC1C(C(=O)NCC2(CNC(=O)CCc3nc(O)n[nH]3)CC2)=Cc2ccccc21 46615,c1(COC)cc(C(=O)NC2CC2CNC(c2cncnc2)=O)cs1 46616,c1(C(=O)NC2CC(NC(C(F)=CCC)=O)C23CCC3)c(F)ccc2nc[nH]c12 46617,C1(CNC(c2n(CC)ncc2)=O)CCN(C(=O)CCOC2CCOC2)CC1(F)F 46618,N1(C(C2CCC(CC)CC2)=O)CC(CC(=O)NCCc2cncn2C)CC1(C)C 46619,N1(C(C)=O)CCOC(C(N2CCC(NC(=O)C(F)(F)c3nccs3)C2)=O)C1 46620,c1(C(=O)NC2CN(C(C3CCC3Cc3ccccc3)=O)C2)ccnc(S)c1 46621,C1(CNC(CSCCC(C)C)=O)CCN(C(C23COC(CF)(C2)C3)=O)C1(C)C 46622,Cc1cc(CC(N2CCC(C)(CCNC(C3CCS(=O)(=O)N3)=O)C2)=O)n(C)n1 46623,N1(C(C2(CCC)CCC2)=O)CCC2C(NC(=O)CCC3CC(F)(F)C3)C2C1 46624,C12(C)CCN(CC1)C2=O.C1(C(C)=O)CCCN(c2ncc(I)cn2)C1 46625,C(=O)(N1CC2COCC2O1)C1OCCC(NC(=O)C=C2CCCCC2)C1 46626,c1(C(=O)NC(C2CN(C(c3nccnc3Cl)=O)C2)C)cncc(C2CC2)c1 46627,N1(C(CC=C=C)=O)CCCCCC1C(=O)N(C)CC1CCCN1C 46628,S(=O)(=O)(c1c[nH]c2cc(F)ccc12)Nc1c(C)ccc(-n2cnnn2)c1 46629,c1(CC)ccc(C(=O)N(C)CCOCCC(=O)NOC2CCOC2)cc1 46630,n1(CC(=O)NCC2N(C(CCCCC=C)=O)C3C(C2)C3)ncn2nccc2c1=O 46631,C(=O)(C(O)CCNC(=O)CN1CC2CC2C1)NCCCNC(N)=O 46632,c1(C(=O)Nc2nc3c(s2)CCCC3)c[nH]c2cc(-c3ccc(O)nc3)cnc12 46633,c1(C(C(=O)NC(C)(C)CC)N(C2C3CCCC23)CC)cc(C)nnc1C 46634,N1(CC)CC2C=CC1C(CO)C2.N12CCC(CC1)ONC2=O 46635,c1(C(=O)NC2CC(C)(COC)N(C(c3[nH]nnc3C)=O)C2)ccn2ncnc2c1 46636,c1(N(CCCNC(=O)NC2(CSC)CC2)C)ccccc1 46637,N#Cc1ccccc1C1CCN(C(c2cc(C(F)F)on2)C(=O)NCC(F)F)C1 46638,Cc1ccn(CC(=O)N(C(C)CNC(=O)COc2c(C)occc2=O)C)c(=O)c1 46639,N1(C(c2ccc(C)s2)=O)CC2CC(C1)CN(C(=O)C(C)C(C)O)C2 46640,C(=O)(C(C)(CC)CO)NCCC1N(C(c2cnc(CC)s2)=O)CCOC1 46641,C(CS(=O)(=O)CC(=O)NC(C(=O)Nc1cncc(Cl)c1)C1CCOC1)OC 46642,N1(c2nccc(C#N)n2)CC2(CCCC2NC(=O)CN2CC3CCC2C3)C1 46643,CC(O)(C(=O)NCC1(NC(c2cnn(CC3CCCO3)c2)=O)CCC1)C1CCC1 46644,C1(NC(c2n[nH]c(C)c2Cl)=O)CCC2(CC1)CCN(C(c1ccc(CO)s1)=O)C2 46645,c1(C(=O)NCCC2(C(N(CCCCC)C)=O)CCCC2)nc(=N)cc[nH]1 46646,c1(C(=O)NC(C)CN(C)C(c2ccc(-c3cccs3)[nH]2)=O)ncc(F)cc1N 46647,C1(C(N(C)CC2CCN(C(=O)CCc3ccccc3)C2)=O)CCC(F)(F)CO1 46648,c1(C(N2CC(NC(c3cc(CC)no3)=O)C(C)C2)=O)c(C)nc2sc(C)nn12 46649,O=C(C1CCc2ccccc21)N1CC2CC1CN2C(c1cc(F)cc(F)c1F)=O 46650,C(CCCCCCCO)=CC(=O)NC1(CNC(C23COCC2C3)=O)CCOC1 46651,N1(C(C(C)c2cccs2)=O)CCC(O)CC1C(N1CCC(c2ccco2)C1)=O 46652,C1(C(=O)NCC2(NC(C(CCC)F)=O)CCOCC2)CN2CCC1CC2 46653,N1(CCN(C)C(C2CC(F)(F)C2)=O)CCN(C(c2ccnn2C)=O)CC1 46654,N1(C(COC2CC(NC(C(C)OC(C)(C)C)=O)C2)=O)CC2CN(C)CC2(C)C1 46655,CC(CNC(=O)CCc1cscn1)(CO)NC(=O)Cn1cccn1 46656,c1(C(=O)NCC(CNC(C(CC)N(C)C)=O)(C)O)cc(N)c(C)c([N+](=O)[O-])c1 46657,Cc1oc(C(=O)NCC2CCCN2C(=O)C=Cc2cccn2C)cc1S(C)(=O)=O 46658,c1(C(=O)Nc2c(C(=O)OC)nn(CC(F)(F)F)c2)c(C)cc(C)nc1C 46659,C=CCCCCC(=O)NC(C(=O)NC1CC12CCC2)c1cccs1 46660,Cc1cccc(C(CNC(=O)COCCOC)NC(C2CCS2(=O)=O)=O)c1 46661,N1(c2nccc(OCC)n2)CCC(NC(C2C=CC(=O)N=N2)=O)C(F)C1 46662,c1(NCC2(OC)CCCSC2)nc(=NCC#CCCO)[nH]c2c(C)nn(C)c12 46663,NC(=O)CCC(=O)NCC1CCN1C(C12CCC1C2)=O 46664,c1(C(N2CC(C(N)=O)(CNC(C(COC)OC)=O)C2)=O)cc2c(cc1N)OCO2 46665,C1(CN(C)C(c2nocc2Br)=O)CCCN1C(=O)CC1C=CCC1 46666,CCCCC(CNC(=O)CC1(N(C(=O)C(C)n2ccnc2)C)CC1)CCC 46667,C(=O)(C1=Cc2ccccc2C1)NC1C2(CCN(C(CN(CC)CC)=O)C2)CCC1 46668,CCCCCS(=O)(=O)CC(=O)N(CC(C)O)CCNC(=O)CC(C)C(F)(F)F 46669,N1(C(CSCC#C)=O)CCCC2(CCCCC2NC(c2cnn[nH]2)=O)C1 46670,C1(NC(c2nc(C)oc2)=O)CC1C1CCN(C(=O)C(C)CC(F)F)CC1 46671,C1(c2ncc(C)cn2)CCN(N(CC2CCOCC2)Cc2ccc(Cl)cc2)CC1 46672,C(C(=O)N1CCCC(C(=O)NOCC(O)CO)CC1)(C(C)(C)C)OC 46673,C1(C(N2CCC(NC(C(C(C)C)NC=O)=O)C2)=O)CC2C=CCC(C1)C2 46674,CP(C)(=O)C1(O)CCN(C(c2ccccc2Cl)C(=O)NCC2CC(F)(F)C2)CC1 46675,C1(NC(c2c(C)cn(C)n2)=O)CC2CC1CN(C(=O)C(C)(C)C(F)(F)F)C2 46676,c1(CC(CC)NC(=O)CCn2cc(-c3cc[nH]n3)nn2)ccccc1Cl 46677,C(C(CNC(c1cnc(S)n1C)=O)S(C)(=O)=O)NC(CC(C)F)=O 46678,Cc1ccc(C)n1CC(N1CCCC1CCNC(c1cc(C(F)(F)F)cs1)=O)=O 46679,N1(C(=O)Cc2cccnc2)CC2(CCN(C(C3CCCN3C(=O)C3CC3)=O)C2)C1 46680,c1(C(=O)NC(C(=O)NC(C)CNC(c2cocn2)=O)C)ccc2ccccc2c1 46681,C1(NC(C2COCCN(C(C3(OC)CCCC3)=O)C2)=O)CC(C)N(C)CC1C 46682,c1(OC)cccc(CNC(=O)C(O)C2CN(C(=O)C(C)(C)C#N)C2)c1 46683,N1(C(Cn2c(C)cc(C)n2)=O)CCC2C(C1)NC(=O)CN2C(=O)CC1C=CCC1 46684,C1(NC(c2cc(O)ccc2I)=O)CC2(C1)CN(C(=O)Cn1cccn1)C2 46685,C1(NC(C(C)O)=O)(CO)CN(C(=O)CC(C)n2cccc2)C1 46686,c1(CC)nc(C)oc1C(=O)NC(C)(C)C(=O)NCc1sc(C)nc1C 46687,C(=O)(C(C)(C)C(=O)N1CCCC(N(C(=O)CC2(C#N)CCC2)C)C1)N(C)C 46688,C1(N(C(=O)Cn2cccn2)Cc2cc(Cl)ccc2F)CCC12CCNCC2 46689,CC1CC(C(=O)NCCOCC2CCC2)CN(C(=O)CCn2cnc(=N)[nH]2)C1 46690,N1(C(c2c(CCC)nco2)=O)CCCC(C(N2CC3CCC3(C)C2)=O)(CC)C1 46691,N1(C(CN2C(C)CCC2)=O)CC(O)CC1CNC(C1COC1)=O 46692,C(=O)(C(F)C(C)(C)O)NC1(C)CN(C(CC(C)Cc2ccccc2)=O)C1 46693,c1(C(=O)NC(CNC(CC2(OCC)CC2)=O)CC(F)(F)F)ncnc2sccc12 46694,Cc1cnc(Cl)[nH]c1=NC(=O)c1cnc2n[nH]c(-c3ccnc(F)c3F)c2c1 46695,c1(C(=O)NC2CC(CNC(C(C)(C)CF)=O)OCC2)cc(Cl)c2n[nH]cc2c1 46696,C(C(C)C)(C(O)C(=O)NCCC1(O)CCN(C(c2cnn(C3CC3)c2)=O)C1)OC 46697,C(CC(C)C(=O)NCC(c1ccccc1F)NC(C1CCC1(F)F)=O)=CC 46698,CCC(C)(O)CCNC(=O)C(C(C)OC)NC(=O)CN1CCC(=O)CC1 46699,c1(N(CC(CN(C(C(CC)NC(N)=O)=O)C)O)C)cc(Cl)nc(CS(C)(=O)=O)n1 46700,C1(NC(C(=O)NC(C)C)=O)CN(C(c2ccc(Br)s2)=O)CC2(CCC2)C1 46701,CC(C(=O)Nc1cnoc1C1CCOCC1)C(C)O 46702,N1(C(CC)=O)CC(C)CN(C(=O)CCc2n[nH]c3c2CCCC3)CC1C 46703,c1(CC(=O)NCC2CCCCC2F)ccc(F)cc1.C12(COC)CN(C1)C2=O 46704,C1(C(=O)NC2CCC(F)(F)C2)CC(F)(F)CN1S(=O)(=O)CCBr 46705,c1(C(=O)NC2(C)CN(C(c3sc(Cl)cc3Cl)=O)C2)cn2c(n1)CCC2 46706,Cc1nc2ccnn2c(C)c1C(=O)NCC1COCC1NC(=O)CCC(F)F 46707,N(C(=NCCc1ccc2occc2c1)N1CCN(CC2CCCO2)CC1)CC=C 46708,c1(CC(N2C(C)CC(NC(c3cnc(S)n3C)=O)C2)=O)cnc2c(=O)[nH]ccn12 46709,N1(C(C(CCC)NC(C)=O)=O)CCOC2(CCCN(C(=O)C(O)C(C)(C)C)C2)C1 46710,C(C(C)CC(=O)N1CC(OC)CC1CCNC(=O)Cc1cncn1C1CC1)OC 46711,N1(C(c2n(C)nc(Br)c2)C(=O)NC2CCC2)CC(C(N)=O)C2(CC2)C1 46712,CC(CCc1ccccc1F)C(=O)NCC1CCCN1C(c1c[nH]nc1Cl)=O 46713,N1(C(CCC(CC)C)=O)CCC2(CCC(NC(=O)C(F)CC(C)C)CC2)CC1 46714,C1(C(N(CCCCNC(c2cc(COC)on2)=O)C)=O)CN(C)CCO1 46715,Cc1nn2cc(C(N3CC(CNC(c4cc(C(N)=O)no4)=O)C4CC34)=O)nc2s1 46716,N1(C(Cc2cc(C)no2)=O)CC(CNC(=O)CSCc2csc(=N)[nH]2)CCC1C 46717,C1(C(=O)NCCC(C)NC(C2(F)CC2)=O)CC(C)N(C)C1 46718,N1(C(c2cnc(CC)[nH]2)=O)CC(CNC(=O)CCn2ccnc2)C(O)C1 46719,c1(NC(CC2CC(NC(CC3CC(CC)C3)=O)C2)=O)cccc(F)c1C 46720,c1(OC)ncc(C(N2CC(CCNC(C3CCC(C)O3)=O)C2)=O)cc1C 46721,c1(CC(C)C)occc1C(=O)NCC(C(C)C)CCN(C)C.C(=O)(COCCO)N 46722,C1(CNC(c2ccc3nn[nH]c3c2)=O)CN(C(c2cc(Cl)no2)=O)CCC1(F)F 46723,N1(C(c2cnc(C(C)OC)s2)=O)CC2C(NC(=O)Cc3cscn3)C2C1 46724,c1(NC(=O)NCC(c2cccc(Cl)c2)SC)cc(C(F)F)c(F)c(F)c1 46725,CC1(C)CN(C(=O)CCC2CC2(Cl)Cl)CC(CNC(=O)C=Cc2cscn2)O1 46726,C1(N(CC#C)C(c2nocc2Cl)=O)CCN(C(C2(O)CCC2)=O)CC1 46727,N#Cc1ccc(C(O)C(=O)OCC2CCC2c2ccccc2)cc1 46728,O=S(=O)(c1ccc(Br)cc1NC1CCCn2ccnc21)N1CC2CCC1CC2 46729,N1(C(C2C(C)(NC(Cc3nc(C)oc3)=O)CCCC2)=O)CCCC(C2CC2)CC1 46730,c1(C(=O)NCC)snnc1CCNC(=O)COC1CCC1.C1CS1 46731,c1(C(N(CCNC(c2cccc(N(C)C)c2)=O)CC)=O)ccc2nc(S)[nH]c2c1 46732,c1(C(=O)NCCCN(C(C2CCC(C(N)=O)O2)=O)CC)cc(OC)cnn1 46733,N1(C(CNC=O)=O)CCOC2CN(C(C3C4CC5C(C4)C35)=O)CC12 46734,CC1=C(C(=O)N2CC3(CC(NC(c4cc(C#N)ccc4N)=O)C3)C2)CCCC1 46735,N1(C(Cc2nc(C)sc2C)=O)CCCC(NC(C23CC(C2)C(C)O3)=O)CC1 46736,N1(C(CC2(C(=O)OC)CCC2)=O)CC2CCC(N(C)C(C3CC3F)=O)C2C1 46737,C(=O)(C(C(C)C)OC)N(CC(=O)OCCC)C(C)C.C1(=O)CC(C)=CCN1 46738,N#CC1(C(N2CC(O)(CNC(=O)CC3CCCCC3O)C2)=O)CC12CCOCC2 46739,c1(Nc2n(CC#C)cnc2-c2ccc(F)cc2)c(OC)ncc(Br)c1C 46740,N1(C(CCc2c(C)ncs2)=O)CC=C(CCNC(=O)CCCC2CC2)CC1.C=O 46741,C(=O)(CC1COc2cc(O)ccc21)NC(CCC(C)(C)C)C(N)=O 46742,C(=O)(C1=CCC(NC(=O)C(C)(C)C(=O)OC(C)(C)C)C1)NCP(OCC)(C)=O 46743,c1(NCC(=O)NCC2CN(C(CSCCCC)=O)C(C)C2)ccc(Cl)cc1Cl 46744,CC1CCC(C(=O)NCc2nc(CNC(=O)C=Cc3ncc[nH]3)cs2)C1 46745,C1(NC2(c3n(C(C)C)nnn3)CCN(CC(F)(F)F)CC2)CN2CCCC2CO1 46746,C=CCC(C)(CC)C(=O)NCC1CCC1C(=O)Nc1ccc(C)cc1CO 46747,C1(CNC(C2(CSC)CCC2)=O)CN(C(c2sccc2F)=O)CC12CC2 46748,C12CC1CN(C(C1(CNC)CCC1)=O)C2.Cc1nc(CNC(CCS)=O)cs1 46749,CCC(O)C(C)C(=O)N1CCCCC1CCNC(C1CCCCN1CC(F)F)=O 46750,N1(C(=O)NCc2nc(CCC(=O)OC)[nH]n2)CCC(F)(C#N)C1 46751,CCCCC(CNC(C1CCC(CN2CCOCC2)O1)=O)NC(=O)CC1CCC1 46752,CC1CCc2c(C(N3CC(NC(C4CCC(C)(O)CC4)=O)C(C)C3)=O)csc2C1 46753,Cc1cc(C(=O)N(C(CNC(c2cccc(O)n2)=O)C2CC2)C)n2nccc2n1 46754,c1(C(N2C3CC(NC(C=CC)=O)CC2CC3)=O)ccc(=O)n2c1CCC2 46755,Cc1cc(C(=O)NC2(C)CCC(NC(=O)C(C)SC3CC3)CC2)n2nccc2n1 46756,C(=O)(C(F)(F)C(C)O)NCC1CC(NC(C2(COC)CC2)=O)C1 46757,CC1CCCC(CNC(C2(NC(=O)Cn3cc(Br)cn3)CC2)=O)O1 46758,CC(C)C(O)CC(=O)N(CCC(N1CCCC(C)(N(C)C)C1)=O)C(C)C 46759,C1(CCNC(C(CC)OC)=O)CCCN(C(=O)CC2C(=O)NN=C2C)CC1 46760,CC1CC(NC(=O)CCS(N)(=O)=O)CCN1C(C1CC2(C1)CC2(F)F)=O 46761,c1(CC)cc(C(=O)NCC=CCNC(=O)C(F)(F)c2ccnn2C)oc1CC 46762,Cn1ncc(CNCCN2CCN(C(c3ccoc3)=O)CC2)c1C1CC1 46763,C(=O)(C(C)CC(C)(C)C)NCC(C)(C1CCC1)NC(CCc1ccnc(C)n1)=O 46764,N1(C(C2C(C)(C)CCC2)=O)CC2C(C(F)(F)F)CC2(NC(=O)Cc2cc[nH]n2)C1 46765,C1(C(=O)NCC(C2CCN(C(c3cnc[nH]c3=N)=O)CC2)C)CCCCC12CC2 46766,c1(C(N2CCC(C(CNC(C3(COC)CC3)=O)F)CC2)=O)cccc2cnsc12 46767,c1(C(=O)NCCCNC(CC2(C)CC(F)(F)C2)=O)cc2ccccc2[nH]c1=N 46768,c1(C(=O)NCC(C)(CC)NC(CCC#CC)=O)cc2ccccc2nc1C(F)F 46769,C1(C(C)(C)CNC(=O)CCCc2cncs2)CCN(C(C2CCOC(=O)N2)=O)CC1 46770,C1(Cc2onc(CN3C(=O)COCC3)n2)CCC2(CCNC2)CC1 46771,c1(C(C(=O)NCCC)N(CCOC)Cc2cccnc2)cn(C)cn1 46772,CCC(CC(=O)NC1CCN(C(C2CN(C(=O)NC)C2)=O)CC1)C1CCC1 46773,CC1OCCC1CC(=O)NOCC(=O)NCC1(CCCO)CC1 46774,C1(CC(=O)NC2CCN(C(c3c(F)ccc(O)c3F)=O)C2)CCC2(CCC2)CO1 46775,C(=O)(CCCCCn1cnnn1)NC12C(CN(C(c3cccc(OC)c3)=O)C1)C2 46776,C1(NC(c2cc(SCC)ncc2)=O)CC2CN(C(=O)C=CCO)CC12 46777,CC1=NOC(=O)C1CC(=O)NC1CCC(NC(=O)CSc2nncn2C2CC2)C1 46778,O(P(=O)(OCC)C1(C)CCCN1C(=O)Nc1nc2cc(Cl)ccc2n1C)CC 46779,CCC(CN(C)C)CC(=O)N(C)CC1(O)CCN(C(c2cncn2C(C)C)=O)C1 46780,N1(C(CC2(CC=C)CCCC2)=O)CCC2CCN(C(C3C=CCC3)=O)C2C1 46781,c1(NC(C2CSCCN2Cc2scc(Br)c2Br)=O)ccc(O)cc1Br 46782,c1(C(N2C(C)CC(CNC(=O)CSc3nncn3C)C2)=O)ccc2c(c1)CCN2 46783,C1(NC(c2c(C)n[nH]c2)=O)COCCN(Cc2ccc(Br)cn2)C1 46784,c1(C(N(C)CC2CCN(C(c3cn(C(F)F)cn3)=O)C2)=O)ccc2c(c1)COC2 46785,N1(C(C(C)=CC)=O)CCCC(C)(NC(=O)Cn2nnc(-c3ccco3)n2)C1 46786,c1(OC)ccc(C(=O)NC2CCCC2NC(=O)C(O)CC(F)F)cc1OC(F)F 46787,N1(C(Cn2ncc(C#C)c2)=O)CC2CCOCC2(NC(=O)CC(C)(C)CC)C1 46788,c1(N2CCC(CNC(C3CC4CC3C3CC43)=O)C2)ncnc(Cl)c1F 46789,c1(C(=O)NCCN(C(=O)C(C(C)C)c2ccncc2)CC)cc(Br)nn1C 46790,C1(NC(C2(C(C)C)COC2)=O)CC(CNC(=O)C(C)CC2CC2)CC1O 46791,N1(C(C(CC)=CC)=O)CC(OC)C(NC(=O)CC2(CO)CC2)C1 46792,C1(C(C)C)CN(C(=O)CC(C)(C)C(F)F)CCCN1C(=O)CCCCC1CC1 46793,N1(C(COCCCOC)=O)CCOCC(C(=O)Nc2cc(Cl)ccc2C)C1 46794,C1(CC(C2CC3(OCCC(N)C3)C2)=O)CCC2(CCCC2)CC1 46795,CC1CCCC1N(CC(C)(C)CNC(=O)C(=O)Nc1ccn(C2CCC2)n1)C 46796,c1(C(=O)NCC#CCNC(CN(CCC#C)C)=O)csc(O)n1 46797,Cc1ccc2cc(Cl)cc(C(=O)NCCn3cc(-c4csc(C)n4)nn3)c2n1 46798,c1(C(N(CC(O)CNC(=O)C(N)=O)C)=O)cc([N+](=O)[O-])c(N(C)C)cc1F 46799,C12(C(=O)NC3CC(CNC(C4(OC)CCCCC4)=O)C3)CCC(C)(CO1)C2 46800,C1(C(=O)NC(C(N2CCC(CN=[N+]=[N-])C2)=O)C2(C)CC2)CC=CC(O)C1 46801,c1(CCOC)ccc(N(C(c2ccc(CC3CC3)cc2)C(=O)NC(C)C)C)cc1 46802,N1(C(C(C=C)(C)C)=O)CCC2(CCCN2C(C2CCC3(CCOC3)O2)=O)CC1 46803,c1(NC(CC2N(C(CNc3ncc(C)s3)=O)CCC2)=O)ccc(-c2ccco2)cc1 46804,C(=O)(CC(C)C(C)(C)NC(C1Cc2ccccc2C1)=O)N1C(C)C(=O)NCC1 46805,c1(C(=O)NC2C(NC(C3N(C)CCCC3)=O)CCCC2)cccc(=S)n1O 46806,c1(OC)cc(-c2cc(C3CCCN3)nn2C)cn(C)c1=O 46807,c1(C2C(C)C2)ncc(C(=O)N(C)CCOCCCNC(=O)C(C)(C)F)s1 46808,C1(NC(c2cccc(SC)c2)=O)CC2(NC(c3c(Cl)n[nH]c3C)=O)COC1C2 46809,C(C(=O)N1CCC(NC(C2CC2F)=O)C1)(C(C)(C)C)NC(=O)OC 46810,N(C1CCCc2c[nH]nc21)C(C(C1CC1)NC(c1cn[nH]c1)=O)=O 46811,C(CC(C(=O)NC(CC1CC1)CC1CC1)NC(=O)CCC1CCC(=O)C1)OCC 46812,C12(C(=O)NCCN(C)C(C3(C)C=CCCC3)=O)CCCC1C2Br 46813,C(=O)(CCCCCNC(C1CC(=O)C1(C)C)=O)NC(C(=O)OC)C(C)C 46814,C(C(=O)NCCC1CCN(C(=O)CNc2nccs2)C1)(C(C)C)N(CC)CC 46815,O=C(CC(F)(F)F)NCC1CCCCC1NC(c1ccc(OC(F)(F)F)cc1)=O 46816,N1(C(C(C2CCC2)OC)=O)CCC12CN(C(=O)CCCSc1ccccc1)C2 46817,c1(C(N2CCCC(C(C)NC(C34CC(C)(C3)C4)=O)C2)=O)ccc(F)c2occc12 46818,C(=O)(C1CCCc2ncccc21)N(CCNC(C1(CC=C)CC1)=O)C(C)C 46819,C(=O)(C(F)(F)C(C)O)NC1CC(CCNC(c2ccc(CCC)[nH]2)=O)C1 46820,c1(C(=O)NCC(CC=C)NC(C2C(C)C2C)=O)coc2c1NC(=O)CCC2 46821,CC1CN(N(C)Cc2ccc(CBr)cc2)CCC1C(F)(F)F 46822,C1(CNC(CCCOC)=O)CC(C)(C)CN1C(c1ccc(C(=O)N(C)C)nc1)=O 46823,c1(C(=O)NC(C(C)C)CCNC(=O)CCCN(C)C)ccc2c(c1)C=CCC2 46824,C1(C)(C(=O)NCC(n2cc(-c3cc(CC)on3)nn2)C)COCCO1 46825,c1(C(N2CC(CCCCNC(CC(=C)Br)=O)C2)=O)[nH]c(C)nc1C 46826,N1(C(c2c(OC)n[nH]c2)=O)CCC2(CC2C(=O)NCC(C)(C)CN=[N+]=[N-])C1 46827,C(=O)(C(C)CCCOC)NC1C(CC)CN(C(c2cnn(C3CCC3)c2C)=O)C1 46828,C(CC(C)(C)C)N(CC(=O)NCC1CCCN1C(=O)CCC1CCOCC1)C 46829,c1(SCC(=O)NC2CCN(C(C3CCC3C(F)F)=O)C2)cccc(F)c1 46830,CC1(C(=O)Nc2ccnc(-c3nn[nH]n3)c2)CCCCCCC1 46831,c1(C(N2C(C)CC(NC(C3CC3(C)C)=O)CC2)=O)cc(F)c(O)c(F)c1 46832,c1(NC(C2C(CNC(c3c[nH]nc3Cl)=O)CC2)=O)ccc2n[nH]cc2c1 46833,C1(NC(C23CCC(NC(c4c(CC)n[nH]c4)=O)(CC2)C3)=O)CCN2CCCCC12 46834,C#CCCCC(c1ccc(Br)cc1)NC(c1cc(-c2ccc(F)cc2)n(C)n1)=O 46835,c1(C(=O)NC2CCN(C(c3cnc(-c4ccoc4)s3)=O)CC2)cnn2c1OCC2 46836,c1(C(N2CCS(=O)CC2C)C(=O)NCCCOC)cc(F)c(Br)cc1F 46837,C1(CC)CCC(C)CN1C(C1CCN(C(=O)C=CCN2CCC2)C1C)=O 46838,CCC(CC(=O)NC(CNC(=O)COc1cc(C)on1)C1CCC1)C(C)C 46839,c1(C(=O)Nc2ccc(C(N(C(C)C)C)=O)nc2)ccc(Br)cc1C(F)(F)F 46840,c1(C(=O)NC2CCN(C(C(CCC)OC)=O)CC2(C)C)cc2c(C)cccn2n1 46841,C1(NC(Cc2cc(C)ns2)=O)CN(C(=O)CCSc2ccccc2)CC1C 46842,C1(N(C(=O)CC2COC(=O)C2)C)CCN(C(c2cnc[nH]2)=O)CC1 46843,c1(C(N(C(CNC(C(C2CCOC2)OC)=O)C2CC2)C)=O)cn2cccnc2n1 46844,N1(C(CCC#C)=O)CC2(CCOCC2)CC1CNC(c1cnc2sc(C)cn12)=O 46845,c12ccccc1S2.C(CCCCC(=O)NOC(C)CC)NC(C(C)OCC=C)=O 46846,C1(C(=O)N(CC(C)(C)CNC(C2C(C)(C)C2(C)C)=O)C)(OC)CCC(C)(C)C1 46847,C1(NC(C(CC)COC)=O)CN(C(c2cnc(OC)nc2)=O)CC1S(C)(=O)=O 46848,c1(CCC(=O)N(C2CCCN(C(C3CCOC3)=O)C2)C)cn2ccccc2n1 46849,C1(CC)CC2CN1N1CCC(C1)NC(=O)O2.c1(C=O)ccncc1SC.O 46850,C1(N(C(Cn2c(C)cnc2)=O)C)CN(C(=O)CCOc2ccccc2O)CC1O 46851,N1(C(C(C)NS(C)(=O)=O)=O)CCC(CNC(c2sccc2C(F)F)=O)C(O)C1 46852,Cc1cc(C(N2CC3CC3C2C(N2CCCC(O)(C(C)C)C2)=O)=O)cc(C)n1 46853,CCCCC(CC)C(=O)NCCOCCCN(C)C(C12CC(C(F)F)(CO1)C2)=O 46854,C1(NC(c2cc(C)c(Br)o2)=O)CN(C(=O)CNS(N)(=O)=O)CC1C1CC1 46855,N1(C(c2n(CC#C)ccc2)=O)CCN(C(C2CCCS(=O)(=O)C2)=O)C(C(C)C)C1 46856,Cc1nc(C(=O)NC2CCC2NC(c2csc(Cl)c2)=O)c(C)s1 46857,C#CC1(C)COCCN1C(=O)CCn1cc(-c2cnn3c2NCC3)nn1 46858,N1(C(c2n(C)nc([N+](=O)[O-])c2)=O)CCCC2(CCCCC2NC(=O)CO)C1 46859,CN1CCCC(C(=O)NCC(C2CCN(C(c3ccnnc3O)=O)CC2)(C)C)C1 46860,C1(CC(N2CC=CC(NC(c3c(C)cco3)=O)C2)=O)CCCC(F)(F)C1 46861,CC1=CC(C)C(c2cn(CC3(F)CCN(C(=O)CCC4CC4)CC3)nn2)CC1 46862,C1(CC(N2CCC(CN(C(CCC(C)N(C)C)=O)C)CC2)=O)CC2(CCO1)CC2 46863,C1(CNC(c2c(COC)scc2)=O)CCC2(CCN(C(=O)CC(C)C)CC2)CO1 46864,CC1CN(C(=O)C(CNC(=O)CC2C=CCC2)N(C)C)CCS1=O 46865,C1(O)(CNC(c2ccn(CCOC)n2)=O)CCCN(C(=O)C(C)NC(C)=O)C1 46866,C1(N(C)C)CCC(n2cc(CN(CC3CC(O)C3(C)C)CC3CC3)nn2)CC1 46867,c1(C(=O)NC(C)CN(C(C2CN(CC)C2)=O)C(C)C)cc(C(C)C)[nH]n1 46868,C1(N(C(C(C2CC2)OC)=O)C)CCC(NC(c2nnsc2C(F)F)=O)CC1 46869,C1(C(C)(C)C)CC(C(=O)NCC(C)(C)CNC(C2CC2c2ccccn2)=O)=NO1 46870,c1(OC)cccc(C(=O)NC2CCN(C(C3(C#N)CCCO3)=O)C2)c1C 46871,CC1(CC(=O)NC2CC(F)(CNC(=O)COCCCF)C2)Oc2ccccc2O1 46872,Cc1cccc(C(=O)C(=O)NC2CCN(C(c3cnc(C4CC4)o3)=O)C2)c1 46873,C12(C(=O)NCC(CC)NC(=O)C(F)Cc3ccccc3)CC3CC1C2C3 46874,N1(C(c2n(CC)ccc2)=O)CCOC2CN(C(=O)C(c3ccccc3F)C)CC12 46875,CCC(C)C(C(=O)N(C)Cc1nccn1CC)NC(C1CCCSC1C)=O 46876,C(CCC(C)(C)NC(=O)C=C(Cl)Cl)NC(C=CCCC(C)C)=O 46877,c1(C(=O)OCC)cnc(SC)[nH]c1=NCCCN(C(=O)CC(C)(F)F)C 46878,c1(C(=O)NC(CN(C(=O)C(C2CCOCC2)O)CC)C)cc(C(C)C)n(C)n1 46879,c1(C(N2C(C)(CC)CC(NC(=O)CC3=CCCC3)C2)=O)nc2c(s1)COCC2 46880,CN1CCc2cc(C(N3CCC(N(C(=O)C=CS(C)=O)CCO)C3)=O)sc2C1 46881,CC(C)C#CC(=O)NCC1(C(N)=O)CN(C(C2CC(O)C(F)C2)=O)C1 46882,C1(C)(C(=O)NCC(N(C(C(C)n2cccc2)=O)C)C2CC2)CCCS1(=O)=O 46883,C12(CCNC(=O)Cc3ccccc3F)CCC(C1)N(C(c1ns[nH]c1=O)=O)C2 46884,C1(CC(C)NC(C2(CC#C)CCC2)=O)CCN(C(=O)CNC(C)=O)CC1 46885,C12(C(N3CC(SC)C(NC(=O)CC4CCCN(C)C4)C3)=O)CCC(CC1)CC2 46886,C1(C(N2CC(O)(C(C)NC(c3cc(OC)no3)=O)C2)=O)Cc2cc(C)ccc2O1 46887,c1(C(=O)NC(C)CCF)ccc(CNC(C2CC2F)=O)nc1 46888,C1(NC(CCSCCC)=O)CC(C)N(C(=O)C(=O)NCC(F)F)C1 46889,C12(NC(CCCC#C)=O)CCN(C(c3cnoc3C(C)C)=O)CCC1C2 46890,C(=O)(C1OC(=O)c2ccccc21)N1CC(NC(CCC)=O)C(C)(C)CC1 46891,CCCC(CNC(=O)C(CC)OC)C(=O)NC1CCN(CCC)C1 46892,c1(C(N(C(CNC(C)=O)Cc2ccccc2)C)=O)ccc(CO)cc1OC 46893,C(CC(C(N)=O)NC(C(C)(C)C1CCCC1)c1nnnn1CCCF)OC 46894,C1(NC(C(=O)N(C)C)=O)CC2CCC1N(C(c1ccccc1Cl)=O)C2 46895,c1(CC)ocnc1C(=O)N(CC(C)CNC(=O)Cn1cnnc1O)CC 46896,N1(C(C2N(CC)C(=O)CC2)=O)CCCC(NC(c2cnc(C)n2C)=O)C1C 46897,C1(C)(NC(C2N(C(CC3COCC(C)O3)=O)CCC(O)C2)=O)CCCCC1(C)C 46898,S(=O)(=O)(c1sc2cc(F)ccc2c1C)NCC(C(CC)C)C 46899,C=C(Cl)CC(C(=O)NCc1cnc(F)c(C)c1)NC(=O)C(C)C(F)(F)F 46900,c1(NC(COC)CC(C)C)cc(N(CC(C)CO)C)nc(C)n1 46901,NC(=O)CCCC(=O)N1CCC(CO)C(NC(c2cc(C3CC3)nc(O)c2)=O)C1 46902,CC1CCN(C(C2(CC#N)COC2)=O)CC1CNC(=O)CCC(C)(C)F 46903,C1(C(=O)NC2(CNC(Cc3n(C)ncc3)=O)CCC2)CC2CCCCN2C1 46904,Cc1c(C(N2CCC(NC(c3cncc(Cl)c3)=O)C2C)=O)ccn1CCO 46905,C1=CC(=O)Nc2c(OC)ccc1c2.O(NC(=O)CCC1CCCCC1)CC 46906,CCC(C(=O)OC)C(=O)NCc1cc(C(=O)N(CC)CC)on1 46907,c1(CC(N2CC(CNC(c3c(C#C)c[nH]n3)=O)OCC2)=O)ccc(Br)cc1C 46908,Cc1csc2ncc(C(=O)NC3CN(C(=O)C(c4ccc(Cl)s4)=O)CC34CC4)n12 46909,Cn1nc(I)cc1NC(=O)NCC1(C)CC(F)(F)C1 46910,c1(CCC)nc(C)c(C(N2CC(CNC(C3(C#N)CCC3)=O)CC2C)=O)o1 46911,C1(OC)CC(C)N(C(=O)C(=O)NCCCc2nn[nH]n2)C(C)C1 46912,c1(C(=O)NC(CN(C(C2(COC)CCCO2)=O)C)C)cc(Cl)c(N)cc1OC 46913,C#Cc1ccc(CN2CCOC(CNc3nccc(C#N)n3)C2)cc1 46914,N1(C(c2n(C)c(S)nn2)=O)CCCN(C(c2ccc(N)cn2)=O)CC1 46915,C1(C(=O)NCC(C)(CO)NC(=O)CN2CC3CC3C2)CCC(=O)NC1 46916,N1(C(COC(C)C)=O)CCCC2CN(C(=O)CN3CCN(C)CC3)CCC12 46917,N1(C(C(CC)(C)C)=O)CCC2CN(C(c3c(OC)ccnc3F)=O)CCC2C1 46918,C(CC(C)C)(C(=O)OC)NC(C(c1ncoc1C)N(C(C#C)(C)C)C)=O 46919,n1(CC)nc(C(N2CC(NC(=O)CCc3ncccn3)CC2C)=O)cc1O 46920,N1(C(C2C(C)=CCS2)=O)CC2CC1C2CNC(c1nnc(C)s1)=O 46921,c1(CC)nn(C)c(C(=O)NCC2CCN2C(c2cc(C(F)(F)F)c[nH]2)=O)c1Cl 46922,Cc1nc2ccnn2cc1C(N1CC(NC(=O)C=CCF)C(C)C1)=O 46923,c1(C(=O)NC23CC(NCc4cc(Br)cs4)(C2)C3)cc(Cl)cnc1O 46924,c1(C(=O)NCC2(F)CC(CNC(c3sc(CC)c(C)c3)=O)C2)cc(N)cc(F)c1 46925,c1(N2CCC(O)(C(C)NC(c3cncc(Cl)c3)=O)C2)ncc2c(n1)CCCCC2 46926,N1(C(C(=O)NC(CC)C)CC2C=CCC2)CCC(CCC(C)O)CC1 46927,C1(NC(=O)CCCn2ccccc2=O)CN(C(=O)Cn2nccn2)CCC1CO 46928,c1(C(=O)NC2CN(C(CSc3ccc(OC)cc3)=O)C2)nc2cccnc2s1 46929,C(=O)(C(O)CCCNC(=O)CC1CCOC1(C)C)N(C1CCN(CC)C1)C 46930,S(=O)(=O)(c1cccc(Cl)c1Cl)N1CC2(CC(NC(c3c(OC)cccn3)=O)C2)C1 46931,Cc1c(C(=O)N(CC(C)NC(=O)CCC=CBr)C)ccn1C 46932,N1(C(C23C(NC(C(CCC)C#N)=O)CC(CC2)C3)=O)CCOC(C)(C)CC1 46933,c1(CC)ncc(C(=O)NC2(CCNC(=O)CN3CC4CC4C3)CCCC2)c(O)n1 46934,c1(C(=O)NC2CCN(C(C(F)=CC)=O)CC2(C)C)cc2c(nc1O)CCCC2O 46935,Cc1nnc(N(C2COC2)C(C2(C)CCCC2(F)F)=O)nc1C 46936,c1(NC(c2n(CC)nnn2)c2ccccc2)cc(CO)ccc1OCC 46937,N1(C(CC2(CC=C)CCCC2)=O)C2CCC1C(CNC(c1cc(C)ns1)=O)C2 46938,c1(CC)cc(C(=O)NCCC2(CNC(=O)COCC(=O)NCC)CC2)on1 46939,c1(C(N2CC(NC(C(C)(F)c3ccccc3)=O)C(O)C2)=O)cccc(Cl)c1Cl 46940,CCCC(C(=O)NCC(CO)NC(c1c[nH]nc1C1CC1)=O)N(C)C 46941,CCCCC(O)C(C)C(=O)N(CC(=O)NCC1CC2C=CC1O2)C 46942,c1(C(=O)NC(C)C(CO)NC(=O)C(C)(C)F)cnc(C2CC2)nc1O 46943,N1(C(C2CCC(=C)CC2)=O)CCCC(C)(NC(=O)CC2CCC2(F)F)C1 46944,c1(C(=O)NC2(C(N3C(CC(C)(C)C)CC3)=O)CC2(C)C)cnn2c1CCC2 46945,C=CCCC(=O)NCCC(C)N(C)C(c1occc1Cl)=O 46946,c1(OCC)ccc(C2CCN(C(=O)C(N3CCOC(CN(C)C)C3)=O)C2)cc1 46947,C(=O)(C(F)CCCCCCCC)NC1CCCN(C(CC2CC(=C)C2)=O)C1CC 46948,c1(CNC(C2(C)CC2F)=O)nc2c(s1)CN(C(c1cc3sccc3[nH]1)=O)CC2 46949,C1(C(N(CC(CC)NC(CC(C=C)(C)C)=O)CC)=O)CCC2(CC1)CNC(=O)C2 46950,c1(C(=O)NC2CCN(CCNC(CCC)=O)CC2)c[nH]c2c(Cl)cccc12 46951,C1(C2CCC2)(CNC(C2C(=C)CC2)=O)CCN(C(c2cnc(O)c(C)c2)=O)CC1 46952,C1(CNC(c2ncn(C)c2)=O)C2CN(C(c3ccccc3C3CC3)=O)CC12 46953,C#CCC(C)(C(=O)NC(C(O)CO)C1CC1)NC(C1COCOC1)=O 46954,c1(C(=O)NC(CCCNC(c2cc(OC)c(C)cc2)=O)C)cc2n(c1)CCCC2 46955,CC(CC1=CCCCC1)(C(=O)O)NC(=O)COCCn1cc(CNCCO)nn1 46956,CCCC(CCCNC(c1c(C)nn(CC)c1C)=O)NC(=O)Cc1nonc1C 46957,N(C(=NCC(C)Oc1ccc(F)cc1)NCC(F)F)CCSCC 46958,c1(N2CCN(CC)C(C)(C)C2)nc(=NC)[nH]c(=NCCCC(=O)NC2CC2)[nH]1 46959,C(=O)(CCC(=O)c1cnn(C)c1)N(CCCNC(c1c(COC)cco1)=O)C 46960,C1(NC(c2cc(C)oc2C)=O)COC2(C1)CN(C(c1c(C)ncn(C)c1=O)=O)C2 46961,C12(CNC(C(F)(F)C3(OC)CCC3)=O)CCC(NC(=O)CC3CC34CC4)(CO1)C2.SC 46962,C(CC(=O)N1CC2CC1CN2C(=O)CC(C)(C)C(F)F)(C(F)(F)F)OC 46963,c1(SC)cc(C(N2CC(N(C(=O)Cc3cc(C#N)cs3)C)C2)=O)ccc1[N+](=O)[O-] 46964,C=CC(C)(CC)C(=O)NC1CCOC(C(=O)NOCC(F)(F)F)C1 46965,c1(N(C(C)=O)C)cccc(C(=O)Nc2ccn(C3CCNC3)n2)c1 46966,c1(C(C)=O)cc(C(=O)NCC2CN(C(c3ccon3)=O)CCCO2)c(C)nc1C 46967,N1(C(Cc2c(C)non2)=O)CC(C)(C)CC1CNC(C1CCC1(C)C)=O 46968,CCCCCCCCC(=O)NC(C)(C)CC=CC(=O)N(CC(C)C#N)C 46969,C1(NC(CS(=O)(=O)NCC)=O)CCCC12CN(C(=O)C=Cc1ncc(C)[nH]1)C2 46970,C(=O)(C1=NNC(=O)CC1)N1C(C)CCC(NC(c2cc(SC)oc2)=O)C1 46971,C(=O)(C1=CCC(C)(C)CC1)NCC1CCC(CNC(c2ncn(CC)n2)=O)CC1 46972,c1(NC(C2N(C(c3cc(C(C)C)no3)=O)CC(O)C2)=O)ncc(Br)nc1C#N 46973,C=C(C)C(CC(=O)NCCN(C(c1cc(F)ncc1OC)=O)CC1CC1)OCC 46974,C(CCCO)N(C(C1(NC(=O)CC2(CSC)CC2)CSC1)=O)CC 46975,c1(CC)ccc(O)c(C(=O)NC2CC(CNC(c3cnc(O)c(OC)c3)=O)C2)c1 46976,C#Cc1ccc(Br)c(C(=O)NCC2CN(C(c3cc(C)oc3C)=O)C3CC23)c1 46977,c1(OC(=O)NCC(=O)NCC(C)N(C)C)cc(C(F)(F)F)ccc1O 46978,C1(C(=O)NCc2c(SC)cccc2)CCCCC1(C)CNC(C1CCC=CO1)=O 46979,C(=O)(C(C(=O)NC(C(=O)N(CC(C)(C)O)C)C1(C)CC1)OC)OC 46980,C(C(O)(C(F)(F)F)c1ncc(C)o1)NC(=O)NC1CN(C(CC(=O)OCC)=O)C1 46981,C(=O)(C(F)C(F)(F)C(F)(F)F)N1CC2(CC(NC(=O)CC3CC34CC4)C2)C1 46982,C(=O)(C1OC(=O)c2ccccc21)NCCCNC(CSC(=N)N)=O 46983,N1(C(c2cn(CCOC)nn2)=O)CCC(C)(NC(=O)C(C)n2cncn2)CC1 46984,N1(C(c2cc(C3CCCC3)[nH]n2)=O)CC2CCC(C1)N2C(C1C2CCC1CC2)=O 46985,c1(C(C(=O)NCCCN(C(Cc2c(C)cc(C)s2)=O)C)O)ccc(Cl)c(Cl)c1 46986,C1(=CCNC(C(C)CO)=O)CCN(C(=O)C(c2ccccc2)N(C)C2CC2)CC1 46987,C1(NC(CC2CN(C(C(=O)NCC)=O)CC2C)=O)CCN(C)CC1C 46988,CCC(CC)(CC)C(=O)NCCN(C(=O)Cc1cnc(C)[nH]1)Cc1ccccc1 46989,N1(C(C2CN(C)C2)=O)CCn2c(-c3ccc(Cl)cc3)nnc2C1 46990,CC1CN(C(c2cn(CCO)nn2)=O)CCCN1C(=O)CC1CCCNC(=O)C1 46991,C(C1CCCn2cc(C(C)(C)C)nc21)NC(C(CC)c1nn[nH]n1)=O 46992,c1(C(=O)OC)cc(CC(=O)NC(C)(CNC2CCCN2C=O)CO)ccc1C 46993,CCCC(C(O)C(=O)NCc1c(C)noc1C)NC(=O)CCC(C)CN(C)C 46994,N1(C(CNS(NC)(=O)=O)=O)CCN(C(c2n[nH]cc2C(=O)OC)=O)CC(CO)C1 46995,c1(NC(N2C(COC)CCCC2)=O)cc(C)c(Cl)c(C)c1 46996,c1(COC)cccc(CS(=O)CC(=O)NCc2ccc(C)nc2)c1 46997,c1(CNC(C2(CC)CCCCC2)=O)ccc2c(c1)CN(C(=O)CCC(C)SC)C2 46998,c1(C(N2CC(CC=C)(C(=O)NCC(C)CCCO)C2)=O)nc(C)ccc1C 46999,CCC(C)C(C)C(=O)NC(C)(C)CN1CCN(C(c2ccnc(OC)c2)=O)CC1 47000,N1(C(Cc2cc(CC)no2)=O)CC2CC2(CN2CCCC(C(=O)NC)C2)C1 47001,c1(C(=O)NCCC2CN(C(C3C(OCC)C3)=O)C2)nccn2ccnc12 47002,C1(N(C(CCOCCOC)=O)CCF)CCCN(C(=O)CCC2(C#N)CCC2)C1 47003,N1(CC(C)C)CCCC(C(=O)N(CC(C)(C)CNC(C2CCNC(=O)C2)=O)C)C1 47004,C(CN=[N+]=[N-])(C(=O)NCC(C)S(N)(=O)=O)NC(C(N1CC(C)C1)C)=O 47005,C(CCO)(C(F)F)NC(=O)C(O)CN1CCCC1.CC(C)(CNC(=O)COC)N 47006,C1(NC(C2(CC)CCC2)=O)CCCC(N(C)C(c2cc(-c3ccoc3)[nH]n2)=O)C1 47007,c1(C(N(C)CC2CCCN2C(C2CCCC2(C)C)=O)=O)cc2c(s1)CCC2 47008,c1(C(N(CCNC(c2cnc(COC)s2)=O)C2CC2)=O)ccnc(S(N)(=O)=O)c1 47009,C1(C(N2CCOCC2)=O)Cc2nccnc2CN1C(=O)C1=NOCC1 47010,C(=O)(C(C)(C)CC(C)(C)C)NCC(C)NC(=O)Cc1csc(N2CCNC2=O)n1 47011,N1(C(C(C)N(C)C)=O)CCCCC1CNC(=O)CCNC(C1CC2(CC2)C1)=O 47012,C(=O)(C(CC(C)C)ONC(=O)CCC1CCOC1)N(CC(=O)NC)CC=C 47013,C(=O)(CCCCCn1cnnn1)NC1CCCN(C(c2ccc(OC)cc2)=O)C1 47014,c1(NCC2C(OCC)CN2C(=O)C(O)C(C)C)cc(P(C)(C)=O)ccn1 47015,c1(C(=O)NCC(C)CN(C)C(C2(N(C)C)CCC2)=O)occc1C1CC1 47016,N1(C(Cc2c(C)nc[nH]2)=O)CC(NC(=O)C(C)C(C)(F)F)CC2(CC2)C1 47017,CC1CCN(C(=O)COC2CCC2)C1C(=O)NCc1ccc(F)cc1 47018,c1(C(=O)NCC2CC(C)(C)N(C(=O)CO)C2)cc(Br)c2nccn2c1 47019,C(=O)(CCCC(=O)N1CC2(CCNC(=O)CN(C)CCO)CCC1C2)NCC 47020,c1(C(=O)NCCOC2CN(C(C3OC4CCC3C4)=O)C2)ccc(F)c(F)c1 47021,c1(C(=O)NC2C(C)N(C(c3cccc(Cl)n3)=O)CC2)c(F)ccc(F)c1N 47022,C1(CNC(c2c(C)csc2)=O)C(C2CC2)CCN1C(=O)CC(C)C(F)(F)F 47023,c1(C(=O)NC(C)(C)CNC(=O)C(C2CCCCC2)F)ccc(OCC(N)=O)cc1 47024,c1(C(=O)NCC(C)(CC)NC(C(CC)=CC)=O)cccc2c1ccn2C(C)C 47025,C1(C2CCN(C(c3ns[nH]c3=O)=O)C2)CCCCN1C(c1cscn1)=O 47026,CN(C1CN(C(=O)CCCC2CCC2)CCc2ccccc21)C(=O)C1CC1 47027,C(=O)(C(C)(C)CC(C)(C)C)NCCC1(CNC(c2nccc(C)n2)=O)CC1 47028,CCC(N=c1cc(NCCOCC2CCCCO2)nc(C(C)C)[nH]1)C(C)C 47029,c1(C(=O)NC2CCC(n3cc(C4(O)CCCCC4)nn3)CC2)nc[nH]c2nccc1-2 47030,C(=O)(C(F)n1ccnc1)N(C(C)C(=O)NCCNC(N)=O)CC 47031,C1(CNC(=O)C#CC2CC2)COCC2(CCN(C(C34CC(F)(C3)C4)=O)C2)O1 47032,N1(C(C2(CCN=[N+]=[N-])CC2)=O)CC(=O)NCC1C(N1CCNC(=O)C1)=O 47033,c1(C(=O)NC(CC(C)NC(c2c(NC)cccc2)=O)C)c(F)cc(C)cc1Cl 47034,C(C)(C(C)C(=O)NCC1(C2CCC2)CC1)NC(C(C=C)C)=O 47035,c1(C(=O)NC2CCC(CNC(C(N)=O)=O)C2)cccn2c(CC(C)C)nnc12 47036,N1(CC)CC(NC(=O)Cn2cc(CNC(c3nc(C)c(C)s3)=O)nn2)C(C)C1 47037,C1(NC(=O)CC2CC2)CCCCN(C(C2CC3(C2)CC2(CC2)C3)=O)CC1 47038,c1(NC(C2CC2Cl)=O)cccc(Oc2cccc(F)c2)c1 47039,Cc1cn2c(n1)C(C)N(C(=O)CC1CC3(C1)CN(C(=O)OC(C)(C)C)C3)CC2 47040,c1(C(=O)NCCN(CCC)C(C)C)cnn(CCNC(=O)CCN2CCCC2)c1 47041,N1(C(C(C)OC)=O)CCCN(C(c2nc(Br)c(C)s2)=O)CCC1 47042,N1(C(CCCC=C)=O)CCC(C)N(C(C2CC(C)(C)CN2C)=O)CC1 47043,C1(C(=O)NC(C)CN(C)C(C23CC(C2)C3)=O)CCCC(C)CC1 47044,c1(C(N2CCC(C)(CNC(C3CC(OC)C3)=O)C2)=O)ncc(Br)cc1F 47045,n1(C(C)(C)C)cc(CC(=O)NC(C)(CNC(=O)Cc2ccsn2)C2CCC2)cn1 47046,c1(OC)cc(F)cc(C(=O)NCC(O)CNC(C2(C)CC(C)OC(C)C2)=O)c1N 47047,c1(C(=O)NC(CN(C(=O)CCc2cccnc2Cl)CC)C)ccc(Cl)c(C)c1O 47048,N1(C(c2cc(OC)n[nH]2)=O)CC(NC(C2(CO)COC2)=O)CC12CCOC2 47049,CC(C(=O)N1CC(C(C)NC(=O)CSCc2ccccn2)C1)C(C)(C)C 47050,c1(N2CC(C(=C)C)OCC2)cccc(S(=O)(=O)NC2CC23CC(OCC)C3)n1 47051,C(CCCC(CO)NC(c1occ(C)c1C)=O)NC(Cc1c(SC)cccc1)=O 47052,N1(CCNC(C(c2cncnc2)N(C(C2CCCOC2)C)C)=O)CCOCC1 47053,Cn1nc2c(cc1=O)CC(c1nc(CC3=CCCCC3)no1)CC2 47054,c1(CNC(CCn2cc(C3CCN(C)C3)nn2)=O)ccc2c(n1)OCCO2 47055,C#Cc1ccnc(C(=O)NCC(O)CNC(=O)COCC2CCCCO2)c1 47056,c1(CCC(=O)NC(C)CCCNC(=O)C=CC2CCC2)c(F)cccc1Cl 47057,CC1CN(C(CCc2ccc(Cl)cc2)C(=O)NC2CC2)CCN1CCC(C)(C)C 47058,C1(C(c2ccc([N+](=O)[O-])cc2)NC(c2c(OC)nccc2)=O)CC(C)(C)CCC1O 47059,C1(C(=O)NC2CC2)CCN(C(=O)C(c2cccnc2)O)C1.c12sccc1C(=O)N2 47060,CC1CCCC1CC(=O)NCCOC1CCN(C(=O)C(c2ccc(Cl)s2)=O)C1 47061,c1(C(N2CC(CC)C(NC(=O)C#CC3CCOC3)C2)=O)cc(OC)c(C)c(OC)c1 47062,C1(CN(C(=O)CC2CCOCC2)CC)CCCN(C(=O)CS(N)(=O)=O)C1 47063,C(=O)(C1Cc2c(Cl)cccc21)N1CC(S(N)(=O)=O)C(NC(=O)CC(F)(F)F)C1 47064,c1(CC)c[nH]nc1C(=O)NCC1CC1CNC(c1cnn(CCOC)c1)=O 47065,C(C)(C)(CC(=O)NCC(C)(CNC(c1cc(C)n(C)c1)=O)OC)OC 47066,C1(NC(CC#N)=O)CCN(C(c2cnc3n2CCS3)=O)CC12CCC2 47067,c1(C(N2CC3CN(C(CN(C)CC)=O)CC3C2)=O)cc2c(F)ccc(F)c2[nH]1 47068,N#Cc1cccc(N2CCN(C3CCN(C(=O)NC45CCC(C4)C5)C3=O)CC2)c1 47069,CC1(NC(c2cnn(C3CCC3)n2)=O)CCN(C(C2(n3cccn3)CCC2)=O)C1 47070,c1(-c2cnc(OC)c(CN3CCC(Br)C3)c2)cc2cc[nH]c2cn1 47071,N1(C(C(=O)NCCC2(C)CC2)CC2CCC3CC23)CC2CCCCC12C 47072,C1(NC(C(C)C)=O)CC(CNC(=O)COCCSc2ccccc2)C12CCC2 47073,N1(C(c2cccc(C)n2)=O)CCC2C(NC(c3sc(N(C)C)nc3Cl)=O)C2CC1 47074,C1(Nc2nccc(C)n2)CC(NC(=O)CCC2CC2)C12CCOCC2 47075,N1(C(c2ncn(C)c(=O)c2)=O)CCC(CNC(C2COCC2(C)C)=O)C(F)(F)C1 47076,c1(CN2C(c3nnc(C(C)C)o3)C(C)(C)C2)cc(C(=O)O)cc(Br)c1C 47077,CC(C)CCC(C(=O)NC1CCS(=O)CC1)NC(C1CC2(CCCO2)C1)=O 47078,C1(CC(=O)NC(COCC)C(=O)NCCC(=O)N(C)C2CC2)CC=CCN1C 47079,c1(C(=O)NCC2CC(C)N(C(c3cccc(CO)c3)=O)C2)ccc(Cl)c(C#N)c1 47080,c1(CC)cscc1C(=O)NCCC1(CNC(=O)CCCc2ccc(C)s2)CC1 47081,c1(N2CCC(NC(C(CC)C)=O)C(F)C2)nc(C)nc(C)c1F 47082,c1(NC(C=CCOC)=O)c(F)cc(F)c(F)c1F 47083,C1(C(=O)NCCCCn2cc(C(CC)(O)CC)nn2)(OC)CCCC(C)(C)C1 47084,CCC(CN(C)C)CC(=O)NC1CCCCC1CNC(c1nn(C)c(C)c1Cl)=O 47085,Cn1c(C(=O)NCC2COCC2NC(=O)Cn2ccc(C(F)(F)F)n2)nnc1S 47086,N1(C(c2nc(NC(C)=O)sc2)=O)CC(C)(C)CCC1CNC(=O)C=C1CCC1 47087,C(=O)(CC1OCCc2sccc21)N1C(c2cn(-n3ncc(COC)c3)nn2)CC1 47088,c1(OCC)ccc(C(N2CCOCC2)CNC(=O)C(C)NC(C)=O)cc1C1CC1 47089,c1(C(N2C(CNC(C3C(C#C)C3(C)C)=O)CC(C)(C)C2)=O)cc(F)c(F)cc1F 47090,C(=O)(CN=c1cc[nH]cc1)N1CC=C(C(=O)N2C(CC)CC(O)C2)C1 47091,c1(C(N2CC(OCCNC(C3=C(C)CCC3)=O)C2)=O)cc2ccc(O)nc2s1 47092,C1(OCC)CN(C(N2CCCCC2C(=O)NC)=O)CC1C(=O)OC(C)(C)C 47093,c1(C(=O)NC2CC(CNC(C(COCC)(C)C)=O)C2)ccnc(O)c1Br 47094,CCCCCCCC(O)CC(=O)N1CCNC(C(=O)NC2(CC#N)CCCC2)C1 47095,CCC(CC)CC(=O)N1CCC(C)(NC(=O)C(O)CC(N)=O)C1 47096,c1(C(C(=O)NCC2CC2)N(CC(C)Cn2cccn2)CC)cccc2c1OCO2 47097,C12(CNC(c3c(CSC)cccn3)=O)CCC(CC1)N2C(C1C=CCC1)=O 47098,c1(OC)ccc(F)cc1C(=O)NCCC(C(C)C)N(C)C 47099,C1(C)(CC)CC(NC(=O)CC2CCCCC2)CN1C(=O)CC1(OC)CCOCC1 47100,CC(CC(=O)N(CC(C)(C)CNC(=O)C(N1CCN(C)CC1)C)C)CC(F)(F)F 47101,N1(C(C2(C#C)CN(C(=O)CC(C)(C)OC)C2)=O)CCC2C(CCN2C)C1 47102,CCC(CC(C)C)C(=O)N1CC(CN=c2nc[nH]s2)C(C)(C)C1 47103,C1(NC(CCCC)=O)CC2CCC(C1F)N2C(c1ccc2c(c1)CCN2)=O 47104,C(=O)(C1=CC2(CCNC2)C1)N1CCC(C(N(C(C)C)C(C)C)=O)CC1 47105,C12(CNC(C(C)CN(C)C)=O)CC(CCO1)N(C(=O)C(CO)C(F)(F)F)C2 47106,c1(NC)ccc(C(N2CC(CNC(=O)Cn3cccn3)C3(CC3)C2)=O)cc1F 47107,N12CCC(O)(C1)C2=O.N1(CC(=O)Nc2cn(C)nn2)C(=O)CSC1=S 47108,c1(C(N2C(C(C)NC(C3(C)CC(C)C3)=O)CCC2)=O)cn2ccccc2n1 47109,N1(C(=O)C(=Cc2c[nH]cn2)F)CCN(C(=O)CNC(=O)CC2CCC3CC23)CC1 47110,c1(OC)cc(C(N2CCC(C)(NC(=O)CC3CCC3(C)C)C2)=O)ccc1F 47111,O(N=C(C(=O)Nc1cccc(C)c1)c1ncc(C)[nH]1)CCN(C)C 47112,C=CC1(c2cn(CCCF)nn2)COCCN1C(C1CC1(C)C(=O)O)=O 47113,C1(NC(C(C)Cc2ccccn2)=O)CN(C(c2ccc(F)c(I)c2)=O)CC12CC2 47114,c1(CC)sc(C(=O)N(CC(C)NC(=O)CCC(C)N(C)C)C)cc1C 47115,C1(NC(c2ccc(Cl)nn2)=O)CCCN(c2ccccc2)C1 47116,C1(NC(C2CC2(F)F)=O)CCC2CN(C(C3(CF)CC3)=O)CCC2C1 47117,c1(OC)ccc(CCC(N2CC(CNC(C3CCCO3)=O)C(F)(F)C2)=O)cc1Cl 47118,C(CNC(C1CN(C)C(=O)N1)=O)(CC(=O)NC1(CO)CC(C)C1)OC 47119,N1(C(c2ccc(OC)s2)=O)CCC(N(C)C(c2ccn3nccc3n2)=O)C2(CC2)C1 47120,[N-]=[N+]=NCCCCCC(=O)NCC1CCC(NC(c2ccc(C(N)=O)o2)=O)C1 47121,CC1(C)CCC(C(=O)NCCCC2CN(C(c3cccnc3O)=O)CCO2)CC1 47122,CCC(C(=O)NC1CCC(C)N(C(c2cc(Cl)ccc2O)=O)C1)C(C)C 47123,C1(O)(CNC(C2(C#C)CC2)=O)CCCN(C(=O)C(C)NC(c2ccoc2)=O)CC1 47124,C(CC1c2ccccc2CCN1C(=O)C(O)C(C)C)NC(C(Br)=C(C)C)=O 47125,C(=O)(CCCC(=O)NC(C)C)N(C(CNC(CSc1nc(C)[nH]n1)=O)C)C 47126,CCC(C)(CCC(C)C)C(=O)NC1COCC1NC(c1cncc2nc[nH]c12)=O 47127,CC(O)CCCCCC(=O)OCC1CCCCN(c2ccc(Br)cc2)C1=O 47128,C=C(C)CCCC(=O)N(C1CCN(C(c2ccncc2N)=O)CC1)CC(C)C 47129,CC(C)(C(=O)N1CCC(Nc2ccccc2)CC1)S(C)(=N)=O 47130,c1(CNCc2cccc(-c3cccc(O)c3F)n2)cnn2c1CCCC2 47131,CC1=C(C(=O)N2CCN(C(c3cscn3)=O)C(CCO)C2)CCS1(=O)=O 47132,S(=O)(=O)(c1cn(C)cn1)NCC1C(NCCNC(CCc2c(C)noc2Cl)=O)C1 47133,Cc1c(C(=O)NC(C)(C)C(C)NC(=O)C(C)CC(F)F)nn(C)c1N 47134,N1(C(C(CCOC)C)=O)CCC12CN(C(=O)Cc1c(C)cccc1Br)C2 47135,C(CCCCC(=O)N1CCCC1C(C)(C)O)N(C(C(C)CC1CCC1)=O)C 47136,CC1COC2(C1)CN(C(C1CCCN1C(C1CC(CF)C1)=O)=O)C2 47137,N1(C(CC2(NC(c3ccnc(C)c3N)=O)CC2)=O)CC(C)C12CCOCC2 47138,c1(CCC(=O)N(C2CCN(C(c3cc(C)c[nH]3)=O)CC2)CC)cc(F)ccc1F 47139,CC1(C(=O)NC(CNC(C2CCCO2)=O)CO)CCC2CC2C1 47140,C1(C(N(CC(C)NC(c2cccc3nonc23)=O)C)=O)CNc2ccccc2O1 47141,c1(OC)cc(C)sc1C(=O)NC(C1CN(C(=O)CCCC2CCCC(=O)N2)C1)C 47142,C(=O)(CCCCCNC(=O)CC1CC(F)CN1C(c1cc(O)nc(Cl)c1)=O)OC 47143,c1(OC)c(C(=O)NCC(C)NC(c2cnc(Cl)s2)=O)csc1Cl 47144,c1(SC)c(C(=O)NC2COCC2CNC(C2Cc3cscc3C2)=O)cccc1F 47145,C(=O)(C(C#N)C(C)(C)C)N1CCC(OC)(CNC(=O)CCOCC(F)(F)F)C1 47146,C1(C(=O)OCC2CC2)(CCN(C)C)CC=CC1.CC1C(=O)N(C2CC2)CCN1 47147,C(c1ccc(F)cc1F)=CC(=O)NCC1(OC)CCN(C(C2COC(=O)N2)=O)C1 47148,C(=O)(C(O)c1ccco1)NCCCOCCCNC(C1C(CCC)C1)=O 47149,C1(NC(c2ccc(NC)nc2)=O)CCC(C)N(C(=O)CCSC)C1 47150,S(=O)(=O)(c1ccc2nc(C)oc2c1)Nc1c(C)cc(Br)c(S(N)(=O)=O)c1C 47151,C(=O)(C(O)C(F)(F)F)N1CCC(C)(CCNC(c2ccc(C#C)o2)=O)C1 47152,C(CN=c1[nH]c(=NCc2cnc(O)[nH]2)c2sccc2[nH]1)C1C(C)C1 47153,C(C(=O)N1CCCc2nccn21)C1(C(CC2C(C)(C)C2)=O)CC1 47154,c1(-n2cc(CCCNC(C3C(C(=O)OC)(C(C)C)C3)=O)nn2)cccc(C)c1Br 47155,C(C)(N=c1[nH]c(=NCC(C)c2nccs2)c2[nH]ccc2[nH]1)c1nc(C)[nH]n1 47156,C1(C(=O)OC)CC=CCN1C(=O)COC1CCN(C(=O)C(C)(C)CF)C1 47157,C1(NC(c2n(CC)ncc2)=O)CC12CC(NC(=O)C(O)C(C)C)C2 47158,Cc1csc(=NCC(=O)N2CC3C(CNC(=O)CSC4CCCCO4)C3C2)[nH]1 47159,C1(NC(c2ccc(CC)[nH]2)=O)CCN(C(c2cc(C(C)(C)C)oc2C)=O)CC1F 47160,c1(OCCC)ccc(C(N2CC(C)(NC(C3CCCCCC3)=O)C2)=O)cc1 47161,N1(C(CC(=O)OC)=O)CC2CC1C2NC(c1nscc1Br)=O 47162,C1(C(N(C(C)C(N)=O)CCOC)=O)C2CCC1(c1cccnc1)C2 47163,N1(C(Cc2ccn(CC)n2)=O)CC2(CCC(CNC(=O)CC(C)n3cccn3)O2)C1 47164,CS(=O)CCCCNC(C1(CNC(C2CCOC2)=O)CC=CC1)=O 47165,C#Cc1cnc(NCC(CNC(c2ccccc2C)=O)Cl)nc1 47166,c1(CNC(C2N(C(C(C(C)C)F)=O)CCCC2)=O)ccc(CO)c(F)c1 47167,C(C1=CCN(C(c2ccnc(C(N)=O)c2)=O)CC1)NC(C(CC)NC(N)=O)=O 47168,C(C(C)C(F)C(=O)NCc1cc(C)no1)NC(c1c(OC)nn(C)c1)=O 47169,Cc1ccnc(C(=O)NCC(C2CCCC2)NC(c2conc2C(C)C)=O)c1N 47170,C(CCC(O)C(=O)NC(C)C(O)C(F)F)NC(COCC)=O 47171,C1(C(=O)NC2C(C(N(C(C(=O)OCC)C)C)=O)COC2)CC2(CCCO2)C1 47172,N1(C(c2nccc(C)n2)=O)CCC2(CC1)CC2CNC(=O)C=CS(C)=O 47173,Cc1cc(C(N2CC(CCO)(NC(=O)C(C)SC(F)(F)F)C2)=O)cnc1C 47174,C(C(C)CC(=O)Nc1ocnc1C(=O)NC)NC(c1n(CC)ccc1)=O 47175,C1(C(=O)NC2C=CCC2)(NC(C2CCCSC2)=O)CCOCC1 47176,c1(C(=O)NCC2CCC(NC(C3N(CCC)CCC3)=O)C2)c(C)ccc(F)c1N 47177,C1(CC(=O)OC2(CC3CC3)CC2)CCN(CCCF)C1.c1(O)ccccc1 47178,CCCCCCCCC(C)CC(=O)NC12CC1CN(C(=O)CCSC)C2 47179,n1(C(C)C(=O)NC2CCOCC2NC(=O)C2=CCC2)cnc2ccccc12 47180,C(=O)(C(C)P(C)(C)=O)N1CCC(N(C(CC(C)OC)=O)Cc2ccccc2)CC1 47181,c1(C(=O)NCC2(O)CC(CNC(C=C(CC)C)=O)C2)cc(C)c(C(N)=O)cn1 47182,C1(C(N2CCC(C)(NC(C)=O)C2)C(=O)NCCCOCCO)CC2C=CC1CC2 47183,N(C)(S(=O)(=O)N(C)C)CC(N1C(CN(C(c2ncn(C(C)C)n2)=O)C)CCC1)=O 47184,Cc1cccc(N)c1C(=O)NCC1CCCCN1C(=O)CCNC(=O)CO 47185,c1(N(CCCNC(CCC(C)(C)F)=O)CCO)ncc(Br)cc1C#N 47186,CC(C)CCCC(=O)NCC(CC(=O)Nc1cscc1C1CC1)C1CCC1 47187,C(=O)(CC(O)CC1CCNCC1)N(c1ccccc1)CCOCCC(C)C 47188,Cc1cc(C(N2CC=CC2CNC(=O)C(c2cccc(Cl)c2)C)=O)ccn1 47189,N1(CC)CCCN(C(=O)CONC(C2CCOC(C(=O)OCC)C2)=O)CC1 47190,CCC1=NOC(C(=O)NC2CC(NC(C3(CC(=O)NC)CCCC3)=O)C2)C1 47191,c1(C(N2CCCC3CNCCC3C2)=O)c[nH]c2ccc(F)cc2c1=O 47192,N1(C(c2c(C)nc[nH]2)=O)CCC(C)N(C(c2ncnc(C)c2C)=O)CC1 47193,Cc1ncc(C(N2CC(C(=O)NC3(CCO)CCOC3)C3(CC3)C2)=O)cc1C#N 47194,C1(CNC(c2c(C)nc(O)[nH]2)=O)CC2CCCCC2N1C(C1CCSC1)=O 47195,C1(C(=O)NC2CCCCN(C(c3ccc(Cl)cc3O)=O)C2)CC2CCCCCC12 47196,C=CCC(C)C(C)(c1nnnn1-c1c(C)cccc1C)NCCC1CC1.C1CS1 47197,CC1CCN(C(C2(N3CCCC3)CC2)=O)CC1CNC(=O)CNS(=O)(=O)C1CC1 47198,C(C1=NOC2CN(C(=O)CC3CC3)CC12)NC(c1cc(C)nnc1O)=O 47199,c1(CC(N2CC(NC(C=C(C)C(C)C)=O)C(C)C2)=O)cn2ccsc2n1 47200,N1(C(CC=CCNC(c2csc(Cl)c2)=O)=O)CCCC2(CC2)C1 47201,C1(C(=O)NC2(C(=O)NCC)CC2)CCCC(NC(C2(O)CC2)=O)CC1 47202,C#CC1(CNC(=O)COCC2(F)CC2)CCCC1 47203,C1(C(=O)NCC2C3CN(C(C(c4ccc(C)o4)C)=O)CC32)CCN2CCOCC12 47204,c1(C(NNC(c2c(C)scn2)=O)=O)cc(Cl)cnc1F 47205,C(=O)(C(CC1CCOCC1)NC(=O)CCc1cc(C)on1)NC(CC)C1CCC1 47206,CC1CC(C#N)(C(=O)NC2CC(NC(C3(Cl)CC3(F)F)=O)C2)C1 47207,N1(C(C(=O)NCC)=O)CC(C(=O)N(CCCOC)C)C(C2CC2)C1 47208,CCC(C(=O)N1CC2CC1C2CNC(c1cccc(F)c1F)=O)C(C)O 47209,c1(OCCCOC)ccc(C(=O)NCCN(C(c2ncccc2O)=O)CC)cn1 47210,N1(C(c2cn(CC=C)nc2)=O)CCC(NC(=O)C(F)C(C)(C)O)CC1C 47211,N1(C(c2nncc(OC)c2)=O)CCC(N(C)C(C2SCCS2)=O)C(C)C1 47212,C1(C(=O)NCC2(F)CC(NC(c3occ4c3CCC4)=O)C2)CCCC2(CCC2)O1 47213,N1(C(C(C)(C)NC(=O)OC)=O)CCC(NC(=O)C(C)(C)C)C(O)C1 47214,C1(CC(=O)NC2CC(CNC(CCCNC(C)=O)=O)C2)COCC(C)(C)O1 47215,N1(C(c2ccc(F)c(C)c2O)=O)CC2(C1)CN(C(=O)CCCF)CC2CO 47216,C(CN=c1[nH]c(=NC)[nH]c(=NCC=CC2CC2)[nH]1)c1c(OC)c(C)c(C)cc1 47217,N1(C(CC2(NC(C)=O)CC2)=O)CCOC(C(C)NC(c2cc(Cl)cnn2)=O)C1 47218,c1(OC)cccc(=NC(=O)Cc2csc(C(=O)Nc3cc(Br)c(C)cc3F)n2)[nH]1 47219,c1(OC)ccc(OC)c(CC(C)C(=O)OCC(COCc2ccccc2)(C)O)c1 47220,C(N=c1[nH]c(N2CCc3nc(O)[nH]c3C2)nc2ccccc12)C1(C)C(C)(C)C1 47221,n1(C(CC)C)ncc2cc(C(=O)NCC3CCN3C(c3ccncc3)=O)cnc12 47222,CC1CCN(C(c2cc(Cl)cs2)=O)C1C(=O)N(C1CC=CC1)C 47223,CCCCCCCC(=O)N1CCCC1C(C)NC(c1c(Br)c(C)nn1C)=O 47224,C1(C(N(CC(O)CNC(C2CC23CCCCC3)=O)C)=O)CCC(=C(F)F)CC1 47225,C1(CC=C)(NC(C2CC2(F)F)=O)CC2CCC(C1)N2C(=O)Cc1c(C)noc1Cl 47226,C1(C(=O)NC(C2N(C(c3cc(COC)[nH]n3)=O)CCCC2)C)CCC2(CC1)CC2 47227,C(C(O)C(F)(F)F)N(C(C(C)N(C(=O)CC1(CNC(C)=O)CC1)CCC)=O)C 47228,c1(CCC(=O)NC2CC(C)N(C(=O)CC#N)C2)cc(F)ccc1Br 47229,N1(C(C2CCN(C)C2)=O)CC=CC(C(N2CCN(CC(N)=O)CC2)=O)C1 47230,C1(C(N(CCCF)CC)=O)CC2CC2N1C(C1CC=C(C)CC1)=O 47231,N1(C(CC2(CNC(C3CCN(C)CC3)=O)CC2)=O)CCCC(F)CC1 47232,C(=O)(C1=NOC(CNC(=O)C=C2CCOCC2)C1)N1C(CC(C)C)CCCC1 47233,N1(C(CCC(=C)C)=O)CCC(C2CC2)(CNC(=O)CC2C(C)(C)C2(C)C)C1 47234,N1(C(c2cnc(C)nc2)=O)CC2CC(C)N(C(C3CCCOC3)=O)C2C1 47235,c1(C(=O)NC(C(C)NC(C2(CC)CC(C)(C)C2)=O)C)ccc(C(F)(F)F)c(F)c1 47236,N1(C(C(=O)NCC)=O)CCCC(N(CCCC)C(C2(CN(C)C)CCC2)=O)C1 47237,c1(CCC)cc(C(=O)N(CC(C)CNC(=O)CC(CC)C2CCC2)C)ccn1 47238,Cn1ncc(C(=O)NC2CCCCC2NC(=O)CCc2ncccn2)c1Cl 47239,c1(C(C)C)nnc(SCCCCCN2CCOCC2)n1-c1ccc(F)cc1 47240,C1(C(N(C)Cc2cc(OC)c(Br)cc2)=O)CC(c2ccccc2F)=NO1 47241,C1(C(NC(=NCc2ccsc2)NC2CCCCC2)C)CN2CCCC2CO1 47242,c1(C(=O)NCC2(O)CC(C(=O)NCC(C3CC3)OC)C2)cc(C)oc1C 47243,c1(CC(=O)NC23C(CN(C(C4(OC)CCOC4)=O)C2)C3)nsc2ccccc12 47244,N1(C(C2CCCCC2)=O)CC(C(N2CCC2CO)=O)C(F)C1 47245,c1(C(=O)OC)coc(C=CC(=O)NC2CCC(N(C)C(c3cc(C)sn3)=O)C2)c1 47246,C1(C(C)NC(=O)CC2(CN(C)C)CCC2)CCCN1C(=O)CSc1n[nH]c(O)n1 47247,C1(NC(CS(CCC)(=O)=O)=O)CCC2CCN(C(c3ccc(O)cc3Cl)=O)C1C2 47248,c1(C(C)NC2CC2C(=O)OC(=O)NC(C)(C)C)ccc(-c2ccccc2)s1 47249,C1(n2cc(CC(C)(C)CO)nn2)CCC(NC(c2[nH]nnc2C2CC2)=O)CC1 47250,c1(C(N(CCCCN(C)C(c2csc(-c3cn[nH]c3)n2)=O)C)=O)cncc(F)c1 47251,N1(C(=O)OC)CCC(CNC(C2CCCN2C(=O)CC2CC2C(F)(F)F)=O)CC1 47252,CCN=c1[nH]cc(C(=O)N(CCCNC(C2CC2[N+](=O)[O-])=O)C)s1 47253,C1(N(C(CCOc2cccc(C)c2)=O)C)CN(C(c2csc(=N)[nH]2)=O)CC12CC2 47254,CC(C)(C#N)CC(=O)NC1CC(NC(C2CCC=CCC2)=O)C(O)C1 47255,c1(C(C)=O)cccc(C#CC(=O)OCC2CCC3(CCCCCC3)O2)c1 47256,C1(N(C2CC2)Cc2cnc(C)n2-c2ccccc2)CC(C)CC(C)C1 47257,c1(OCC)ccc(-c2cccc(C3(C(=O)NCCCOCC)CC3)c2)c(F)c1F 47258,C1(CC)(CC)CC(NC(C2CCCOCC2)=O)CN1C(c1ccc(OC)cn1)=O 47259,N1(C(C(C)NC(C2CCC2)=O)=O)CCCC(O)(CNC(=O)Cn2nccn2)C1 47260,c1(OC)ccnc(O)c1C(N1CC(NC(=O)Cc2cnsc2)C(C)C1)=O 47261,Cc1cc(C(N2CCN(C(C3CCCO3)=O)CC2)C(=O)NC2COC2)cc(F)c1 47262,C1(S(C)(=O)=O)(C(=O)NC(CNC(C(C)=C2CC2)=O)CC(C)C)CCC1 47263,N(C1CC(C)(C)c2ccccc21)Cc1c(Br)cc(OC)c(OC)c1O 47264,c1(C(=O)NCCCN(C(=O)CNS(=O)(=O)N(C)C)CC)cc(S(C)(=O)=O)cs1 47265,C(=O)(C(C(C)(C)O)NC(c1ncncc1N)=O)N1CC(C)SCC1 47266,CCC1=C(C(=O)NCC(F)CNC(=O)CCCOC(C)C)SCCO1 47267,C1(C)(CNC(CC(=C)C)=O)CN(C(c2cc(F)c(C(C)=O)cc2F)=O)C(C)(C)C1 47268,n1(C2CN(C(CCN(C(CCC)C)C)=O)C2)cc(C2COCC2O)nn1 47269,c1(CNC(C(C2CN(C(Cn3nnc(C)n3)=O)C2)N(C)C)=O)cc(C)oc1C 47270,c1(CCC(N2CC(O)(CCNC(=O)C(C3CCCCC3)F)C2)=O)cncc(F)c1 47271,CCCC(C(=O)N1CC(=O)CC1C(=O)N(C)CCc1cnccn1)OC 47272,c1(C(N2CCC(O)(CNC(c3cnn(C(F)F)c3)=O)C2)=O)noc2ncccc12 47273,c1(C(=O)NC(C(=O)OCCC)C)cn(CC2CCOC2)nn1 47274,c1(OCC)ccc(C(=O)NC(c2ccccc2)(C)CNC(C2CCCO2)=O)cn1 47275,c1(CNC(CC2C3CN(C(C(n4ccc(C)n4)C)=O)CC32)=O)ccc(F)cc1F 47276,CN1CCC(C)(C(=O)NCCCCCN(C(=O)C(O)CC2CCOCC2)C)C1 47277,Cc1ccc(CC(N2CCC(C)(C(=O)N(C)Cc3nncn3C)C2)=O)cc1 47278,C12(CNC(c3n(C(C)C)ncc3)=O)CC1CN(C(C1CCCC1C(F)F)=O)C2 47279,C1(N(CCCC)C(c2n[nH]cc2Cl)=O)CCN(C(c2cc(OC)cs2)=O)CC1 47280,C#CC1(C(=O)NCC(CC(C)C)N(C)C)CCN(C(=O)CNC(=O)CN(C)C)C1 47281,Cc1ccc(C(C)C)cc1OCC(N1CCSCC1NC(=O)OCCO)=O 47282,N1(C(=O)COc2cccnc2)CCC(F)(F)C(Nc2ncc3c(n2)CCC3)C1 47283,C=C(C)CC(C(=O)NC1CCCCC1N=[N+]=[N-])NC(=O)C(C1CCOCC1)F 47284,c1(OC)noc(C2CC2)c1C(=O)NCC1(NC(C2(C#N)CC2C)=O)CC1 47285,CN1N=C(C(=O)NCC2(CNC(c3cc(CCO)on3)=O)CCC2)CCC1=O 47286,N1(C(c2c(CC)con2)=O)CCC(CF)(NC(=O)C(C)CSC)C1 47287,C1(O)(CCNC(Cc2n(C)cnc2)=O)CCN(C(c2cnn(CCF)c2)=O)CC1 47288,C12(C(N(C(C3CCCCC3)C)C)=O)CC(CO1)N(C(c1ccc(Cl)cn1)=O)C2 47289,N1(C(c2ccnnc2NCC(=O)NC2CCC2)=O)CCc2ccccc21 47290,N1(CC(=O)N(CCNC(=O)CCc2ncc[nH]2)CC)CCc2sccc2C1 47291,C=C(C)c1cccc(NC(C2CC(=O)CN2C(=O)C(C(C)(C)C)OC)=O)c1 47292,c1(NC2CCN(C(c3cccc(C)c3)=O)C2)ncc(C)c(SC(C)C)n1 47293,c1(-c2ccc(CN3CC(CC)C3)cn2)ccc(OC)c(F)c1F 47294,Cc1c(CCC(N2CCOCC2CNC(=O)C(C)C)=O)c(O)nc2[nH]nc(O)c12 47295,CC1(NC(c2coc(Br)c2)=O)CCN(C(c2ccc(C3(C)CCO3)cc2)=O)CC1 47296,N1(C(c2c(C)nco2)=O)CC(C)(CNC(=O)CC2CCCC(=O)N2)CC1(C)C 47297,c1(C(=O)NC(C)C(C)(C)NC(C23CC(C)C2C3)=O)cc(Br)cc2nc(O)[nH]c12 47298,C12(C(N3C(C)CC(NC(C(C4CCCCC4)C)=O)C3)=O)CCC(F)(CC1)CC2 47299,CC(C)CC(C)(CNC(=O)Cc1cccc(O)c1)NC(c1ccn(C2CC2)n1)=O 47300,N1(C(C(C2CCCO2)NC(C2CCSCC2)=O)=O)C2CCCC1COC2 47301,CC(C)(C)CC(=O)N1CCC(C(C)C(=O)N2CCC2C2CCC2)CC1 47302,C=C=CCC(=O)NCC1COCC1NC(=O)CCc1cc(OC)no1 47303,c1(N(CC(C)NC(Cc2nc(C)sc2C)=O)C)nc(Cl)ncc1Cl 47304,Cc1cc(-n2ccnc2)ccc1C(=O)NCCN(C(=O)C(F)C(F)(F)F)C(C)C 47305,C1(NC(c2ccn(-c3ccc(Cl)c(F)c3)n2)=O)CCCCCC1c1ccccc1 47306,c1(C(=O)NC2C(NC(c3c(CC)cno3)=O)CC2)ccccc1-c1ccccc1 47307,Cc1cc(=NCC2(CCCO)CCCC2)[nH]c(NC(c2cccnc2)C)n1 47308,CN1CCC(n2cc(C3CCCN3C(=O)Cn3cnc(C(=O)O)c3)nn2)C1=O 47309,CC(CNC(=O)OCc1ccn(C2CCC2)n1)(CO)CO 47310,C1(C(N(C2CCN(C(c3ncsc3C)=O)C2)CC)=O)CCCC2CC12 47311,N1(C(C(CC)OC)=O)CCC2(CCN(C(c3occc3C3CC3)=O)C2)C1 47312,c1(OC)ccc(F)c2[nH]c(C(=O)NCC(C)(CO)NC(=O)CC(C)O)cc12 47313,c1(C(N(C(CNC(C2(CC=C)CCC2)=O)C2CC2)C)=O)cn(C2CCCC2)nn1 47314,c1(N2CCCC(CS(N)(=O)=O)C2)cccc(S(=O)(=O)NCc2cscc2Cl)n1 47315,C1(C)(CNC(c2c(CC)con2)=O)CN(C(=O)CC(C(F)(F)F)OC)C(C)(C)C1 47316,C1(NC(c2cc(C(C)C)[nH]n2)=O)CCN(C(c2cn(C)ccc2=O)=O)C1(C)C 47317,C1(C)(C(=O)NCC(CN(C)C(c2ccnc(-c3ccco3)c2)=O)O)CCC(=O)C1 47318,c1(CC)cc(C(=O)NC(C2CCN(C(=O)COC(C)C)C2)(C)C)c(C)o1 47319,C1(C)(CNC(C(C)NC(C)(C)C)=O)CCN(C(=O)CC23CCCC2C3)CC1 47320,N1(C(=O)Cc2nc[nH]n2)CCOC2(CCN(C(C3CC4CCC3O4)=O)C2)C1 47321,CC(C)C(CN(C)C)N=c1nc(N2CC3CCC3C2)c2c([nH]1)CCS2 47322,Cc1nc(Cl)[nH]c(=NC2CC(NC(=O)C(C)n3cnnn3)CC23CCC3)c1Cl 47323,Cn1nc(C(N2CCC(NC(c3ccncc3)=O)C23CCC3)=O)c2c1CCC2 47324,CC(CC(C(=O)N1Cc2cncnc2C(C)(C)C1)Nc1ccccc1)CC(C)(C)C 47325,C1(C(=O)NCCC(=C)CNC(c2csc(C)n2)=O)CC(=O)N(C2CCCCC2)C1 47326,C1(OC)CN(C(C2CC(C#N)C2)=O)CC1NC(C1(c2ccccc2F)CCC1)=O 47327,c1(CNCC2CCC(C(F)(F)F)CC2)csc2ccc(Br)cc12 47328,Cc1cnc(NC(C2CSCCN2Cc2c(C)cccc2Br)=O)c(Cl)c1 47329,c1(C(N(CCCNC(C(CCCCCC)C)=O)C)=O)cc2n(n1)CC(C)NC2=O 47330,C(C(CC1CC1)C(=O)NC(C)(C)C(C)O)NC(Cc1c(C)occ1)=O 47331,C(=O)(CC(C(F)F)NC(c1n[nH]c(O)n1)=O)NCCC(CC)(C)C 47332,Cc1cc(C(=O)NCC2CCC2NC(C2CCCO2)=O)n(C(F)F)n1 47333,C1(C)(C(N2CCC(=CCNC(COCCCCC)=O)CC2)=O)CCC(=O)NC1 47334,CCC(C(C)O)NC(c1ccoc1CNC(=O)COCC(C)C)=O 47335,C1(NC(c2sc(CC)c(C)c2)=O)CN(C(=O)C(F)(F)C(C)O)CC1C1CC1 47336,Cc1c(CNC(=O)NCC2(F)CCCCC2)cccc1F 47337,CS(=O)c1cccc(NC(c2noc(C(N)C3CC3)n2)C)c1 47338,C=CC1(C2(C(=O)NCCCCN(C(=O)CSc3cccs3)C)CCC2)CCC1 47339,C(c1cccnc1C)=CC(=O)NCC(C(C)C)NC(C(CC)c1ccccc1)=O 47340,CC1CC(NC(c2cncc(O)c2)=O)CCN1C(c1cccnc1Cl)=O 47341,Cc1[nH]c(C#N)cc1C(N1CC(CC(N2CC3(CCC3)C2)=O)C(C)C1)=O 47342,N1(C(c2c(C)ncnc2)=O)CCC(F)(C(=O)N(CCCC(O)CO)C)CC1 47343,c1(CCC(=O)OCCc2c(C(F)(F)F)cccc2F)ccc2ccccc2c1 47344,c1(NC(C2ON=C(C)C2)=O)ccc(NC(=O)CN2C(=O)CCCC2=O)cc1C 47345,C#CCCCC(C)C(=O)N1C(C(=O)NCc2cccc(CC)c2)CC1C 47346,N1(C(c2c(C)csc2Cl)=O)CCC2(CC(NC(c3c(C)ncnc3C)=O)C2)C1 47347,C(CC(O)C(=O)NCCCCC(C)NC(c1ccc(NC=O)cc1)=O)SC 47348,N1(C(c2c(C)nc(C(C)C)cc2)=O)CCC2(NC(=O)CN(C)CCO)CCCC12 47349,Cc1nn(C)c(C)c1S(=O)(=O)NC1CCN(CC2(C)NC(=O)NC2)CC1 47350,c1(OCC#C)ccc(C(=O)NCC2(NC(=O)C(C)SCC)COC2)cc1 47351,c1(C(=O)NCCCC(C)NC(CC2C(OC)COCC2)=O)nc2cnccc2s1 47352,c1(C(N(C(c2ccccc2)CNC(C2CNC(=O)C2)=O)C)=O)cc2cccnn2n1 47353,C1(C(N(CCNC(C2CCCSC2)=O)Cc2ccccc2F)=O)CC2CCC1C2 47354,C1(CC(=O)NC2(CC=CC)CCC2)CCCN1C(C1COCCO1)=O 47355,CC(C(=O)NC1C2CCOC2C12CCCC2)N1C(=O)COc2ccccc21 47356,Cn1cnc2c1CCCC2C(=O)NCC1(F)CN(C(=O)CCC2CCOC2)C1 47357,C1(C)(NC(C2(C#C)CCC2)=O)CCN(C(=O)CNC(=O)CNC(C)=O)C1 47358,Cc1cc(CC(N2CC(O)CC2CC(N2CCC(C)(N(C)CC)C2)=O)=O)nn1C 47359,C=Cc1ccc(C(=O)NC2CC(O)CN(C(C3(O)CC(C)(C)C3)=O)C2)cc1 47360,c1(C(=O)NCC2CCCN(C(C(C3CCC3)OC)=O)CC2)nc2ccccn2n1 47361,C1(C(N(CCC)CC)=O)CCCN(C2CCCCC2OC)CC1 47362,N1(C(C(CCSC)(C)C)=O)CC2CC(C1)CN(C(C1CC3CC(=O)C1C3)=O)C2 47363,C1(OC)CC2(C1)CC2NC(=O)C(C1(O)CCC1)NC(=O)C=Cc1cc[nH]n1 47364,C(CC(O)CC(=O)NC1CCC(N(C(=O)C(C)n2cncn2)C)CC1)SC 47365,N1(C(Cc2c(C)nccc2)=O)CCC(O)(CNC(c2ccc([N+](=O)[O-])o2)=O)CC1 47366,c1(CSC)cccc(C(=O)NC(c2cn(CC3CCOCC3)nn2)C)c1 47367,N1(c2c(-n3c(C)cc(C)n3)cccc2)CCCC(C(=O)NCC=CCN)CC1 47368,C1(CC(=O)N(C2(C#C)CC2)C)CC(O)CN1C(=O)CN1CCCC1 47369,c1(C(C)=O)cc(C(=O)NCC23CC(NC(c4ccoc4C)=O)(C2)C3)n(C)c1 47370,N1(C(c2n(C)c(S)nc2)=O)CC2CN(C(c3coc(C(F)(F)F)n3)=O)CC2(C)C1 47371,C1(C(N(CCCN(C)C)CCNC(c2ccncc2)=O)=O)CCC(=O)N2CCCC12 47372,C1(C(N2CC(CC)OCCC2)=O)C2CCCC2CN1C(c1ccc([N+](=O)[O-])[nH]1)=O 47373,C1(CNC(=O)C(=O)NCC2CC=CCC2)CCC(C2CC2)O1 47374,CCC(N)CCC(=O)N1CCC12CC(c1cn(C(C)CO)nn1)C2 47375,C1(NC(CNC(=O)CC(F)(F)F)=O)CCN(C(=O)CSc2nnc(S)s2)CC1O 47376,c1(C(=O)NCCC(CNC(=O)Cc2c(Cl)cnn2C)OC)ccc(F)cn1 47377,C(=O)(C(F)C(F)(F)C(F)(F)F)N1CCC2CCC(NC(C3CC(C)(C)C3)=O)C1C2 47378,C1(C(=O)NC(c2ccccn2)C)CN(C(C23C=CC(CC2)C3)=O)CC1(C)C 47379,c1(OCC)ncc(C(=O)NCCC2(NC(=O)C(C)(F)F)CCCC2)s1 47380,N1(C(=O)OC(C)(C)C)CCSC(C(=O)OCC2CCCO2)C1 47381,C1(CC=C)CCCCN1C(=O)CN(C(C1(CO)CCCCO1)=O)CC 47382,CC12CC(C1)C(C(=O)NCC1(O)CC(NC(c3cncc(C4CC4)c3)=O)C1)CO2 47383,N1(CCNC(C(C)(C)c2cscn2)=O)CCN(C(=O)C(O)CC2CCCC2)CC1 47384,C1(CNC(C(C)Oc2ccc(C)cc2)=O)CN(c2ncnc(=N)[nH]2)CCN1C 47385,c1(CN(C)CC2CC2)ccccc1Nc1ccccc1 47386,CCCCC(O)C(C)C(=O)N1CC2CCC(C1)N2C(c1cnn(CC)c1C)=O 47387,O=C(N1CC(n2cc(-c3cnc(C4CC4)s3)nn2)CO1)c1cccnc1C1CC1 47388,c1(CC(=O)NC2CC(C(C(=O)N(C(C(C)C)C)C3CC3)F)C2)cncnc1 47389,c1(C(c2nnnn2C2CCOC2)NC2(CC)CC2)cc(C)ccc1Cl 47390,C=CCCC(C(=O)NOCCF)NC(C1CC=CCO1)=O 47391,C(=O)(CC(C)(C)C(F)(F)F)NCC1N(C(C(C(=O)OCC)F)=O)CC2(CC2)C1 47392,S(=O)(=O)(C(Cl)(Cl)Cl)N(CCCC)C(C1(NCCC#C)CC1)=O 47393,N1(C(Cc2c(C)nn(C)c2)=O)CCC(C)C(CC(N2CCC(SCO)CC2)=O)C1 47394,N1(C(COCC=C)=O)CC2CC(C(=O)NCCOCCC3CC3)C(C2)C1 47395,CCCCC(C)CCC(=O)NC1CN(C(=O)CC23CCC(CC2)OC3)CC1O 47396,C12(C(N3CC(C(N)=O)(CNC(c4ccccc4)=O)C3)=O)CC(C(F)F)(CO1)C2 47397,N1(C(CCOC(C)=O)=O)CC(NC(=O)CN2CCC(C)(O)C2)CC(C)(C)C1 47398,C1(NC(CC(C)N)=O)CCCN(C(=O)Nc2ccccc2)C1 47399,C(CNC(=O)CCCc1cnn[nH]1)(CC(=O)N1CCC(N(C)C)C1)OC 47400,C1(NC(c2c(SC)cccc2)=O)CC2CN(C(=O)CCc3cn(C)nn3)CC12 47401,Cc1sc(C)c(S(=O)(=O)N2CCC(C)C2C)c1C(=O)O 47402,N1(C(=O)CCCc2ncco2)CCC(CO)(CNC(=O)C(F)OC(F)(F)F)C1 47403,Cc1cc(-c2nc(CC(F)(F)F)nn2CCCN(C)C)nc2ccccc12 47404,N1(CC)C(=O)CCC1CC(=O)NC1(C)CCN(C(=O)CCc2nccn2C)C1 47405,C(=O)(C1CCc2c[nH]nc21)N1C(C)C(NC(c2ccc(C(N)=O)nc2)=O)CCC1 47406,c1(-c2scc(C(=O)NC(c3ccc(Cl)cc3)CF)n2)ccc2c(c1)OCO2 47407,C(C)(C(O)C(=O)NCC1CCC(CNC(c2ccncc2C2CC2)=O)CC1)OC 47408,N1(C(c2c(C)nsc2)=O)CC(C2CCCN(C(=O)C(C)(F)F)C2)C1 47409,CCCCC(O)C(=O)N1CC2C(C(=O)NCCn3cccc3)C2C1 47410,C1(C(=O)OC)(NC(N2CCN(c3cn(C)nc3)CC2)=O)CC(O)C1(C)C 47411,c1(C(=O)NCC2(CNC(c3sc(C)c(O)n3)=O)CCC2)c(O)cccc1Cl 47412,c1(NCC(N(C)C(c2ccncc2F)=O)C2CC2)ncc2scc(Br)c2n1 47413,N1(CCCNC(C)CCC(F)F)CC2C3C=CC(CC3)C2C1 47414,N1(C(CC=CCC)=O)CCCOC(CCNC(C2(C)CN(C(C)C)C2)=O)C1 47415,C1(C(=O)NCC(C)N(C(C2CC(NS(C)(=O)=O)C2)=O)CC)CCCC(=O)N1C 47416,N1(C(C2(CC)CCN(C(CCC3CC(OC)C3)=O)CC2)=O)CC2COCC(C2)C1 47417,O(C1CCCC(=O)c2ccccc21)CC(N)(CC(F)(F)F)C(F)(F)F 47418,c1(CC#N)ccnc(NCC2CCCCN2C(=O)CSc2ccc(F)cc2)n1 47419,S(=O)(=O)(c1ccc([N+](=O)[O-])cc1Cl)N(CC(=O)NCCNC(COCCC)=O)C 47420,C(CCCCCC(=O)N(CCCCCO)C)n1cc(CC)nn1 47421,C1(CC=C)(NC(=O)C(O)C2CC2)CCCN(C(=O)CCCN(C)C)C1 47422,C1(C(N2CC(CC=C)(NC(=O)Cc3ncc(C)s3)C2)=O)COC(C)(C)CO1 47423,C1(C(N(CC(N2CCCC2)C)C)=O)CSCCN1C(C1(Cl)CCCCC1)=O 47424,Cc1cc(C2CC2)cnc1C(=O)N(C)CCNC(=O)CCc1ccccc1O 47425,N1(C(C=C(C)C)=O)CCC2(C(=O)Nc3ccnn3CCCO)CC2C1 47426,N1(C(Cn2ncc(CC)c2)=O)CC(O)CCC1C(=O)NCc1ccc(F)c(F)c1 47427,c1(C(N2C(CNC(CCN(C(CCC)C)C)=O)CCC2)=O)ccc2nonc2c1 47428,CC(C)(O)C#CC(=O)NCCCNC(c1ccc(CO)cc1)=O.C12(CC1)C(=O)N2 47429,CC(C)C(C(=O)N(CC(C)CNC(C12CC(CC(F)F)(C1)C2)=O)C)n1cnnc1 47430,CC1(C)COC(C(N2CC(C)(NC(=O)CCC(N)=O)C2)=O)CO1 47431,N1(C(c2nc(OC)c(F)cn2)=O)C2CCC1CN(C(=O)Cc1cnc(C)[nH]1)CC2 47432,C1(C(N(CC(C)NC(c2cncc(C(C)C)c2)=O)CC)=O)COC2(CO)CC1C2 47433,N1(C(C2CCCO2)=O)CCCC2C1CCCCN2C(=O)COc1cccnc1 47434,N1(CC2CN(C(c3cc(COC)sc3)=O)C2)CCN(C(c2ns[nH]c2=O)=O)CC1 47435,C1(C(=O)NC2C(NC(C3CC(N(C)C)C3)=O)CCCC2)CCc2nnc(O)n2C1 47436,C1(NC(CCc2cn(C)nc2)=O)CN(C(=O)CSc2nncn2C(C)(C)C)CC1O 47437,C1(C(=O)NC2CC(C(N)=O)C2)CCN(C(=O)CC2CCCC2N(C)C)O1 47438,c1(CC(C(=O)OCC(N2CCC(C(F)(F)F)C2)=O)O)cccc(Br)c1 47439,N1(C(C(CCCC)F)=O)CCC2(NC(=O)CN(C3CCCC3)C)CCCCCC12 47440,C(=O)(C(CC(F)F)N(C)C(c1ccc(C#N)cn1)=O)NCC(C1CCCC1)C 47441,N1(C(c2nc(CC)oc2)=O)CCC2(C(=O)NCCn3ccc(C)cc3=O)CC2C1 47442,C#CC1(O)CC(C(N2CCC(N(C(=O)CC(C)(O)C3CC3)CC)CC2)=O)C1 47443,C1(CC(=O)O)(NCC2(CC=C)CCOC2)CCN(C(=O)OC(C)(C)C)CC1 47444,C(=O)(CCC(C)C#N)N1CCN(c2nnc(-c3c(C)nc(Cl)s3)n2CCC#N)CC1 47445,Cc1conc1C1CN(C(=O)CC2CC(NC(C3(CO)CCOC3)=O)C2)C1 47446,C#CCCCC(C)C(=O)NC1CN(C(C2(n3cccn3)CC2)=O)CC1C(F)(F)F 47447,C1(C)(CNC(C=C(COC)C)=O)CCN(C(C2CC(C)C(C(=O)OC)O2)=O)CC1 47448,C(CCCCC(=O)NC1CCN(C(c2cnoc2-c2cccs2)=O)CC1C)SC 47449,C1(C(N2CCCC(c3n(CC)cnc3)C2)=O)Cc2c(C)cccc2O1 47450,C12(CNC(CC3N(C)CCC3)=O)CCC1CCN2C(=O)CC1=CCCC1 47451,c1(NCC(N2CCC(NC(C3CCCSC3)=O)C(O)C2)=O)ccccc1[N+](=O)[O-] 47452,c1(CC)ncoc1C(=O)NCCCC(=O)NCC(c1ccccc1)F 47453,c1(C(=O)Nc2sc(C(C)=O)c(C)n2)cc(O)ccc1Br 47454,C1(CC(C)=O)(C(=O)OC)CCN(C(CCCC)C(=O)NCCC#C)CC1 47455,C(=O)(CS(=O)(=O)C(C)(C)C)N(CC)CC1CCN(C(c2ccn(C)c2)=O)CC1 47456,C1(CCNC(c2sccc2C2CC2)=O)CCN(C(C2(CF)CC2)=O)C1 47457,C1(NC(C(C)C2CCCO2)=O)CN(C(C2CCCS2)=O)CC(C)(C)C1 47458,N1(C(C2(OCC)CCC2)=O)CCN(C(CNC(C2(C)COC2)=O)C(F)(F)F)CC1 47459,C(=O)(CCCC(F)(F)F)N1CC(C(=O)NCCCOCC2CCC2)CC(C)C1 47460,C(CCC(C)C)(C(=O)NCCC1CC(C)C1)NC(C1CC=C(C)CC1)=O 47461,C1(C(=O)NCC2(CC)CCCC2)CC2CN(C(=O)C(C)n3ccnc3)CC2C1 47462,C1(NC(CCC(=O)N(CC)CC)=O)CCN(C(c2nn(C)cc2Cl)=O)C12CCC2 47463,c1(-c2n(CC=C)c(N3CCC(=Cc4cccs4)CC3)nn2)n[nH]c2c1CCOC2 47464,c1(OC)cc(C=CC(=O)NCC2CC2NC(C2(n3cnnn3)CCCCC2)=O)sn1 47465,C1(C(=O)NC(COC(C)C)C(=O)NC2CC3CCC(C2)S3)CC12CCCCC2 47466,N(C1CCc2cccnc21)C(CCOCCNC(C1CN2CCC1C2)=O)=O 47467,C1(NC(C(C)NC(c2ccoc2)=O)=O)CCC(NC(c2scnc2C(F)F)=O)C1 47468,c1(C(N2C(C)CN(C(=O)CC#N)CC2)=O)cccc2c1CC(=O)N2C 47469,C1(C(=O)NC2C(NC(c3n(C)cc(C#N)c3)=O)CCCC2)CCc2nccn2C1 47470,C(=O)(C(C)CC(C)C)NC(CCC(=O)N(CCC)CCC)C 47471,c1(CC(N2C(C)CC(NC(c3ccc(C#N)[nH]3)=O)C2)=O)ccc2c(c1)CCC2 47472,c1(C(N(CC(=O)NC2CC(C(C)(C)O)C2)CC#C)=O)nccc2[nH]ccc12 47473,C=CC(C)(O)C(=O)NCC(CNC(c1sccc1Cl)=O)OC 47474,C(=O)(C(F)(F)C(F)(F)C(F)(F)C(F)F)N1CCCC(NC(C(C=C)O)=O)C1 47475,N1(C(C2(C)CC2(F)Cl)=O)CCC2(CCCC2NC(c2cnc(O)nc2O)=O)CC1 47476,C=C(C)C1OCCCC1C(=O)N(CCNC(=O)C(C)n1cccn1)CC 47477,C(CCC(C)CC(=O)NCC1CCC(NC(=O)CCc2ncc[nH]2)C1)=C(C)C 47478,c1(CC(C)C(=O)N2CCC(NC(=O)Cn3nnnc3C3CC3)C2)cccc(Cl)c1 47479,CC1CN(C(=O)C(O)c2ccsc2)CC1NC(c1ncccc1N)=O 47480,N1(C(c2cc(CNC(c3c(C)cc(C)s3)=O)ncc2)=O)CC2(CCC(=O)O2)C1 47481,C#CCCCC(C)C(=O)NC12CC1CN(C(c1c(F)ccc(OC)c1F)=O)C2 47482,c1(C(C)C)ccc(C(=O)NCC(C)NC(=O)CCC2CCC(O)CC2)cn1 47483,c1(CN(C)C)ccc(C(=O)NCC2CCCCN2C(C2CC3CCC2O3)=O)cc1 47484,c1(OC)ccc(C(N2CC(OCCNC(=O)C(N)=O)C2)=O)c2ccoc12 47485,N1(C(CSCC(C)C)=O)CC(CNC(=O)CN2CCN(C3CC3)C2=O)CCC1C 47486,C12(NC(Cc3nnc(C)o3)=O)CCN(C(=O)CC3CC(F)(F)C3)CC1C2 47487,Cc1c(C(=O)NC23COC(CNC(=O)Cc4csc(S)n4)(C2)C3)cnn1C 47488,C(=O)(Nn1cccn1)c1[nH]c(=N)sc1.c1(C2N(S(=O)(=O)N)C2)ccccc1F 47489,C(=O)(C(C#N)C(C)(C)C)NCC1(F)CCC(NC(COCCOC)=O)C1 47490,c1(NC(C2N(C(c3ccc(Cl)cc3)=O)CCC(=C)C2)=O)cnc2c(c1)CCC2 47491,Cc1ccc2c(C(N3CCC(CNC(=O)CC(O)C(C)(C)C)C3)=O)c[nH]c2c1 47492,c1(C(N2CCC(C(=O)N(C)C)CC2)C(=O)NCCCSCC)c(Br)cnn1C 47493,N1(C(CSCC=C)=O)CCCCC12CC(NC(c1ncsc1C(C)C)=O)C2 47494,N1(C(Cc2cn(CC)nn2)=O)CCC(CNC(c2ccc(I)cc2)=O)(OC)C1 47495,C1(C(N)=O)CC(C(=O)NCCCNC(=O)CSCC2CC2)=NO1 47496,N1(c2n(C)c(C3CCN(S(C)(=O)=O)CC3)nn2)CCC2(CCCCO2)C1 47497,N1(C(CC(=C=C)C)=O)CC(NC(=O)C(C)SC)C(N=[N+]=[N-])C1 47498,C1(C(=O)NC2(C)CC(NC(C3CCC(C)CC3)=O)C2)CCn2c(O)nnc2C1 47499,Cn1nccc1CCC(=O)NC1CCCC1NC(c1coc(Cl)n1)=O 47500,Cc1cc(=O)cc(CNC(C2CN(C(c3sccc3C#N)=O)CCO2)=O)[nH]1 47501,C1(NC(C(CC)C#N)=O)CC(O)(C2CCN(C(c3csc(C)n3)=O)CC2)C1 47502,N1(C(=O)Nc2cc(C(=O)OCC)n[nH]2)CC2CC2(CC)C1 47503,n1(CC(=O)Nc2c(F)cc(I)cc2F)ccc(=NC(=O)c2cc[nH]c2)nc1O 47504,c1(C(N2CCC(NC(c3cc(CO)ccc3O)=O)CC2)=O)cn2c(n1)CCC2 47505,C1(CC(N2CC3(CNC(CCOC)=O)C(C2)CCO3)=O)CCCC2CCCCC12 47506,N1(C(C(CC#C)(C)C)=O)C2CCC1C1CC1(NC(C1CCC(=O)N1CCC)=O)C2 47507,c1(C(N2CC3(C(N4CCCC(O)(CO)C4)=O)CC2CO3)=O)cc(F)ccc1F 47508,c1(C(=O)NCC2(NC(=O)CC3CCOCC3)CCOC2)nc[nH]c2nccc1-2 47509,N(C(=NCCCc1ccc(O)cc1)NCc1ccccc1)CC(COC)F 47510,C12CCC13CN(C3)C(=O)C1=NNC(=CC(c3cccs3)=CC=CC(=O)N2)C1.CC=C.CC 47511,N1(C(CC(=O)OCC)=O)CC2(CCCC2)C1C(=O)NC(c1nccn1C)C 47512,C1(c2cn(CC(=O)NC)nn2)CCCCN1C(=O)COCC1CCCO1 47513,S(=O)(=O)(c1cc(C)cnc1NC(CCO)c1ccco1)NC(CCCC(=C)C)C 47514,C(=O)(C(C(CC)CC)N1CCOCC1)NCCN(C(C1C(C=C)C1)=O)CCC 47515,C1(NC(C2C(=C)CC2)=O)CN(C(c2cc(Br)cn2CC)=O)CC1F 47516,C(C)(C)(CC(=O)NC(Cc1cn[nH]c1)C(N1CCC(O)(CC(C)C)C1)=O)OC 47517,C1(C(=O)NC(C)CN2CCN(C(c3ccon3)=O)CC2)CC12CCCCC2 47518,c1(CC)cc(NC(C2CCCCC2(C)NC(=O)CP(C)(C)=O)=O)cnc1C 47519,c1(C(N2CCC(C)(NC(Cc3nc(C)sc3)=O)C2)=O)cnn(C)c1C#N 47520,c1(C(=O)NC(CNC(c2cnc(CC)s2)=O)C(C)C)cnn2ccnc(N)c12 47521,N1(C(c2ccc(C(C)(F)F)nc2)=O)CC2=C(C1)CN(C(=O)Cc1cc[nH]c1)C2 47522,C1(C(=O)OCc2cnc(C#N)s2)CC2(CCC(F)(F)CC2)CO1 47523,C(=O)(C#CC1(CC2CCC2)COC1)NN1CC2CCC(NCC)C2C1.C(=O)(NC)O 47524,c1(C(=O)NC2CN(C(CC3(C)CCCO3)=O)CC23CC3)c[nH]c2ccc(F)cc12 47525,C#CCCCC(=O)NCCN(C(=O)C=CCCC=C(C)C)CCOCCC 47526,C1(NC(C2CCCOC2)=O)CC2(C1)CC(C(=O)NCC(O)C(F)F)C2 47527,CC1(F)CN(C(=O)Cc2ccon2)CCN(C(=O)CCS(C)(=O)=O)C1 47528,C(=O)(C1CCCn2cnnc21)NCCC1N(C(c2ncn(CC)n2)=O)CCSC1 47529,c1(C(N(C)CC2(O)CN(C(C(C)COc3ccccc3)=O)C2)=O)ccc(O)nn1 47530,Cc1ccc(N)c(C(N2CC(C)(C)CC2CNC(c2cn(C(F)F)cn2)=O)=O)c1 47531,C(=O)(C(C)(C)C1=CCN(C(=O)CCCCC(C)CC)C1)N1CC(C#C)(F)C1 47532,c1(Cc2onc(C(=O)NCC)n2)cccc(Br)c1O 47533,C1(CNC(C=CC=CC)=O)CN(C)CCN1C(C1CCCN1CC(C)C)=O 47534,N1(CC)CCc2c(NC3CC3(c3ccccc3F)C)cccc2C1 47535,c1(CC(=O)N(C2CN(C(=O)C(O)C3CC3)C2)C)ccc(S(N)(=O)=O)s1 47536,c1(CNC(C(C2CCN(C(C(OC)OC)=O)C2)C)=O)cnn(C)c1O 47537,CCC(F)(C(=O)OC)C(=O)N1CCOC(CN(C(=O)Cc2cnoc2)C)C1 47538,CC(N=c1[nH]c(=NCc2cc[nH]n2)c2ncccc2[nH]1)C(F)F 47539,C1(NC(c2ccc(C(F)F)o2)=O)CCCC12CCN(C(=O)CCc1ncc[nH]1)C2 47540,c1(C(=O)OC)cn(C)nc1C(=O)NCC1CC1CNC(C1CCCCC1C)=O 47541,N1(C(c2c(C)ccnn2)=O)CC(NC(c2ncccc2F)=O)CC12CCOC2 47542,C1(NC(CCC(N)=O)=O)CCN(C(C2CN(C3COC3)C2)=O)C(C2CC2)C1 47543,c1(C(=O)NC(CNC(CC(CC)C(C)C)=O)C)c(O)cnc2cc(F)ccc12 47544,CC(C)(O)C(F)(F)C(=O)Oc1ccc(NC(c2sc3cnccc3c2Cl)=O)cc1 47545,N1(C(C(C)CSC(F)(F)F)=O)CCC(CF)(NC(=O)C(=O)NCCC(N)=O)C1 47546,c1(C(N(CCOCCN(CC(=O)NCCC)C)C)=O)ccc(C(C)=O)o1 47547,N1(C(CC2(OC)CCC2)=O)C(C(=O)NCC(=O)OC(C)C)CCC1C1CCCC1 47548,N1(C(=O)NCC(=O)Nc2c(C)cc(Cl)cc2)CC23CCCC2(C1)C3 47549,C(=O)(C(C(F)(F)F)C(F)(F)F)NCCC1N(C(c2ncn(CC)c2)=O)CCOC1 47550,Cc1cc([N+](=O)[O-])ccc1C(=O)NC1CCC1NC(=O)C(=O)NC(C)C 47551,Cc1ccc(C(=O)NC2CCC2CNC(C2COCCO2)=O)cc1Cl 47552,C1(C)(C(=O)NCC(C)=CC(N2CCC3CC23C)=O)CC(=O)N(C)C1 47553,C1(C(N(CC(C)NC(C=CC)=O)C)=O)CCCN1CC(C)C 47554,N1(C(c2cc(CC)on2)=O)CCCC(O)(CNC(=O)CCC2CCN(C)C2)CC1 47555,C1(c2ccc(C)o2)CCCCCN1C(=O)Cc1ccccc1C(N)=O 47556,C1(NC(C2(N(C)C)CCOCC2)=O)CN(C(C2CC2(C)C)=O)C(C)(C)C1 47557,CC1CCCC=C1C(=O)N1CCCN(C(C2CNC(=O)C2)=O)CCC1 47558,C(C)(C(C)(C)NC(c1cccn1C1CCCC1)=O)NC(C(C)n1cncn1)=O 47559,c1(CCCC(=O)NC2C(NC(C(CCC)NC(N)=O)=O)C2)cc(O)ccc1C 47560,CCC(C(=O)N1CCC(NC(=O)CCOCc2ccccc2)C1C1CC1)C(C)C 47561,N1(C(c2cc[nH]c(=NC)c2N)=O)CCC2(NC(=O)C(O)C3CC3)CCCCCC12 47562,C(C(C)(C(=O)NCCC1CCSC1)NC(c1ccc(F)cn1)=O)SC 47563,C1(N(C(CCOCC#C)=O)C)CN(C(=O)CCCCC)CCC1O 47564,CC(C)(O)CCC(=O)NCCC(F)Cn1cc(CN2CCNC(=O)C2)nn1 47565,c1(C(=O)NCCC2CN(C(C3C(C)C3C)=O)C2)n[nH]c(C2CC2)c1Cl 47566,C(CCN(C)C(C12CCCC1C2(F)F)=O)(C(C)(C)C)NC(C=CC=CCC)=O 47567,c1(C(=O)NCC2OCCC(NC(=O)CCF)C2)ccc2c(c1)C(=O)CCCC2 47568,c1(OCC(=O)OC)c[nH]nc1C.C1(C(=O)OC)CC1(Cl)C(=O)O 47569,C1(C(=O)NC(C#C)CC2CC2)CCCCCC1NC(C1(C)CNC(=O)N1)=O 47570,C(=O)(CCCCCCCC(=O)NCCNCc1ccc2cn(C)nc2c1)OC 47571,C(CN=c1[nH]c(=NC2CC2)[nH]c2ccsc12)N(S(=O)(=O)c1cccs1)C 47572,C1(NC(c2nc(C)n(C)c2)=O)CC12CCN(C(=O)C=CC1CCCC1)C2 47573,C(C1=NOC2CN(C(c3ocnc3C(F)(F)F)=O)CC12)NC(CCCC(=C)C)=O 47574,C(=O)(CC(C)(O)C1CC1)N(C1CN(C(c2cscn2)=O)C1)C 47575,Cc1[nH]c(C(=O)NCc2ncccn2)c(C)c1C(=O)NCc1cncn1C 47576,N1(C(c2cc(C)[nH]c2C)=O)CCCC(C)(NC(c2cnoc2C)=O)C1 47577,c1(C(N(C2CCN(C(c3ccc(Cl)cc3F)=O)C2)C)=O)c(Br)ccc2c1OCO2 47578,N1(C(C(C)CSC(F)(F)F)=O)CCCCC(NC(c2cn3ccnc3s2)=O)C1 47579,c1(N(CC(O)CF)C)ccc(S(=O)(=O)NCc2ccc(S(C)(=O)=O)s2)cc1F 47580,n1(C(COC)CNC(=O)CC2CC(SC)C2)cc(C2(C3CC3)CC2)nn1 47581,C1(C(N(CCCNC(C=CCCC)=O)CC2CCCC2)=O)CC12CCCCCC2 47582,c1(C(=O)NC2CCC(CCNC(C3CC3F)=O)C2)cncc(-n2ccnc2)n1 47583,N1(C(C2(C(N(C)C)=O)CC2)=O)CCn2ncc(CN(C)C(C3CCSC3)=O)c2C1 47584,Cc1ccc(C(=O)NC2CC2NC(c2cccc(F)c2O)=O)c(O)n1 47585,C(=O)(CC1=CCOCC1)NCC1CCC(C(N2C(CC)CCC2)=O)CC1 47586,CCC(C)C(O)CC(=O)NCc1ccc(C(=O)NCC2CCC3(CC3)C2)cn1 47587,Cc1ccn2c(C(N3CC4CC3C4NC(=O)CC(O)CN(C)C)=O)cnc2c1 47588,n1(CC)cc(Cl)c(C(N2CCC(O)(CN(C)C(C3(C)CSC3)=O)C2)=O)n1 47589,c1(C(=O)NCC2(NC(=O)CC3CCC(O)C3)CCOCC2)cnc2[nH]nnc2c1 47590,c1(C(=O)NCC=CCNC(C(CC)(C)C#N)=O)nc2ccc(Br)cn2c1F 47591,C1(C(C)C)(C(=O)Nc2cnsc2)CCN(C(c2ccncc2O)=O)C1 47592,C12(C(N(C(c3cn(-c4ccccc4)nn3)C)C)=O)CCCCC(=O)N1CCC2 47593,c1(C(N2C(C(=O)Nc3cnccc3I)CC(C)C2)=O)ccc(Cl)c(C(F)(F)F)c1 47594,CCCC(C(=O)N1CC2CC1C2CNC(=O)CCc1cc(C)n(C)n1)OC 47595,C1(C(N2CCN(C(c3occ(C)c3)=O)CC(O)C2)=O)Oc2ccccc2OC1C 47596,N1(c2cc(C)nc(N3CCC(C4CCCO4)C3)n2)CCC2(CCOC2)CC1 47597,C1(CNC(C2(COC)CN(C(c3c(C)ncs3)=O)C2)=O)CCCN(C)C1=O 47598,c1(C(N(C2CN(C(=O)COCCCF)CC2F)C)=O)cccc(Cl)c1F 47599,c1(OC)cncc(C(N2CC(CNC(=O)CC3(C#N)CC3)CC2C)=O)n1 47600,C1(N(C(CC=CC=C)=O)CCOC)CCN(C(C2CCCCN2C(C)=O)=O)CC1 47601,c1(C(N2CC(O)(CCCOC(C3CN(CC)C(=O)N3)=O)C2)=O)ccc(=N)[nH]c1Cl 47602,C1(NC(C2CC(C#C)(O)C2)=O)CCCC2CN(C(c3cc(C)nnc3O)=O)CC12 47603,N1(C(CCCC#C)=O)CCC2(NC(c3n[nH]cc3COC)=O)CCCCCC12 47604,c1(C(N(CC(CC)NC(c2cccn2Cc2ccncc2)=O)C)=O)cc(C)sn1 47605,c1(C(N(C)CCOCCNC(C2CCCN2S(C)(=O)=O)=O)=O)cc(Cl)n(C)n1 47606,c1(CC)ncc(NC(=O)NC2CCN(CC3CCOCC3)CC2)c(C)n1 47607,CC1CCC2CN1CCCNC2=O.C(C)(C)(C)OC(=O)N.C1(O)CC1 47608,c1(C(N2CC(CNC(CC(C)(C)C)=O)OCC2)=O)cc(Cl)ncc1O 47609,C1(CC)CN(C(c2c(F)cccc2Cl)=O)CCC1NC(=O)CCCC(N)=O 47610,Cc1cnc(CCNC(C2C3CN(C(=O)CCCc4cnn[nH]4)CC23)=O)cn1 47611,c1(C(N2C(CNC(C(C)NC(CC)=O)=O)CC2)=O)c[nH]cc1-c1cnn(C)c1 47612,N1(C(C2C(C)=CCS2)=O)CCC(NC(=O)CC2CS(=O)(=O)C2)C(C)(C)C1 47613,CC1(C)CC(NC(=O)CC2(C3CC3)CC2)CN1C(=O)CC1CN2CCC1CC2 47614,C1(C2CC2)(NC(c2cc(C)c(O)nc2)=O)CCN(C(=O)C(C)(O)CC(C)C)C1 47615,N1(C(C(C2(O)CCCCC2)NC(C(C(C)C)C2CC2)=O)=O)CC(C(N)=O)C2(CC2)C1 47616,C(C)(c1cccc(Cl)c1)=CC(=O)NC(CC)CN(C)C(c1cccc(C)c1F)=O 47617,C12(CCNC(=O)NCc3cn(CCC)nc3)CCC(CC1)CC2 47618,CON1CCC(NC(C2(NC(=O)CC3CC4CC4C3)CC(F)C2)=O)CC1 47619,C(=O)(C(C)(C)C(=O)NC1CC1CNC(=O)Cc1ccc(Cl)nc1C)OCC 47620,c1(COCC(N2CC(C)S(=O)CC2)=O)nc2ccccc2s1 47621,N1(C(CC(C(=C)C)OC)=O)CCc2sccc2C1CNC(C1C2CC3C(C2)C13)=O 47622,C1(C(N(C(C2CCOCC2)C)C)=O)CCCC(NC(=O)Cc2cccnc2O)C1 47623,C1(CC(=O)N(C(C)CN(C(=O)CN2CCCC2=O)C)C)CC=CCN1C 47624,N1(C(C(C)Oc2cccc(Cl)c2)=O)CC2CCN(C(C3CC=CC3)=O)CCC2C1 47625,c1(CC#N)cccc(C(=O)N(CCNC(=O)CC2CC3(CC3)C2)C2CC2)c1 47626,c1(C(=O)NCC#CCNC(c2sccc2Cl)=O)ccc(Br)cc1Cl 47627,N1(C(C(=O)NC(c2cccc(OC)c2)CF)=O)CC2CC(C)C2C1 47628,c1(C(=O)NCCC(C)N(C(=O)CC2OCCC2(C)C)C)cc2c(F)cccc2s1 47629,C1(OC)(CNC(=O)Cc2ccc(F)cc2F)CCN(C(=O)CSSC)CC1 47630,CC(CN(C)C)CCC(=O)N(CCCN(C(=O)C(c1ccc(F)cc1F)=O)C)C 47631,C(=O)(CC(C(C)(C)C)NC(c1c[nH]c(=S)cn1)=O)NC(CCC)C(F)(F)F 47632,N1(C(C(CC)(C)C#N)=O)CCC=C(C(=O)NOC(c2ccccc2)CCOC)C1 47633,CC#CCC(C(=O)N(C1CCN(C)C1)C)NC(=O)CCC(C)(C)OC 47634,n1(CC)ccc(C(N2CC(NC(=O)Cn3ccnn3)CC2C)=O)cc1=O 47635,N1(C(C2OCCN(C)C2)=O)CCN(C(c2cnn(C)c2Cl)=O)CC(CO)C1 47636,N1(C(COCC(C)C)=O)CC2CC1CCC2NC(=O)CSCc1cscn1 47637,CN1CC=C(CCNC(=O)C(C2CCCO2)NC(=O)CNC=O)CC1 47638,c1(NC(CCC(=O)NCCCC(CCC)N)=O)ccc2c(c1)OCCO2 47639,C1(C)(CC(=O)NCC2CN(C(CNC(C)=O)=O)C2)CCCO1 47640,C1(O)(C(=O)NC2COCCN(C(c3cnc(C)s3)=O)C2)CCCC(C)CC1 47641,N1(C(CN(CCC)C(c2cc(COC)on2)=O)=O)CCCC2(CC2)C1 47642,CC1CCCN(C(=O)C(N2CC(CNC(=O)CCC3CC3)C(C)C2)=O)C1 47643,C1(CNC(Cc2c(C)con2)=O)CCCN(C(C2CCC(C(C)C)CC2)=O)C1 47644,c1(C(N2CC(C)(C(N(C3C(C)CC3)C)=O)C2)=O)ccc(N)cn1 47645,c1(C2(C(N(C3CCN(C(C4CC4Cl)=O)CC3)C)=O)CC2)ccc(Cl)cc1 47646,C1(C(N2CC(C(C)NC(C(c3ccccc3)OC)=O)C2)=O)(CO)CC=CC1 47647,C1(C(=O)NCC(CCNC(C(N2CCOCC2)C)=O)O)CCCC(F)(F)C1 47648,C1(C)(C(N2C3C(NC(CC4(OC)CCC4)=O)C(C3)C2)=O)CCC2(CC1)OCCO2 47649,c1(C(N2CCC(CC)C2)C(=O)NCSc2ccccc2)ccc2cc(Br)ccc2c1 47650,CC1(CNC(c2cccc(O)n2)=O)CCCN1C(=O)CCc1cnc[nH]1 47651,S(=O)(=O)(c1cccnc1NCC1(CC#N)CC1)NCC(CCOC)(C)C 47652,C1(C(N2C(CN(C(=O)Cc3nncn3C)CC)CCC2)=O)CC2C=CCC(C1)C2 47653,c1(C(NC(NCc2cn(CC)nc2)=NC)C)cccc(NC2CC2)c1 47654,c1(CC)ccc(C(=O)NC2CCC(CCNC(=O)Cn3cnc(=N)[nH]3)C2)nc1 47655,C(=O)(C1CC(=O)Nc2ncccc21)NCC(C)(C)NC(c1cnc(C2CC2)s1)=O 47656,C(=O)(C(C)(C)CCCNC(c1coc(C(N)=O)c1)=O)NC1C(O)CCC(C)C1 47657,C(=O)(C1CCc2c[nH]nc21)NC1CC2CC(NC(CCNC(=O)NC)=O)C2C1 47658,C1(CNC(c2nccc(C)c2)=O)CN(C(=O)C(F)=C2CCC2)CC(C)(C)C1 47659,c1(NC(CC)=O)cncc(C(N2CC(NC(c3cccnn3)=O)C(C)C2)=O)c1 47660,N1(C(C)=O)CCCC1C(=O)N(CC(C)O)CCNC(=O)C(C)OCC(F)(F)F 47661,C1(C(=O)NC2CC(C)N(C)C2)CN(Cc2cn(CCF)nn2)CCC1O 47662,C1(NC(c2cncc(CO)c2)=O)CC12CC(NC(c1cc(C3CC3)ccn1)=O)C2 47663,c1(C(=O)NCC2C3N(C(C(C)O)=O)CC(CC3)C2)ncnc2c1ncn2C1CC1 47664,c1(C(=O)NCC(C)(C2CCC2)NC(CN(CCOC)C)=O)cccc(C(F)F)c1 47665,N1(C(c2c(O)ccc(C)c2)=O)CC2(NC(C3CCCCS3)=O)CCC1CC2 47666,C(=O)(CC(O)CN(C)C)NCC(C)(C1CC1)NC(c1cc(C)[nH]n1)=O 47667,N1(C(Cc2cc(C)no2)=O)CC2CCCC(NC(=O)C(C)CC3CCC3)(C2)C1 47668,C1(CC(=O)N(CC#C)CC)CCCN(C(c2ccc(SC)o2)=O)C1 47669,C(=O)(CS(=O)(=O)C1CC1)NCC(C1CCN(C(COCC=C)=O)CC1)O 47670,O=C1OCCC12CCN(Cc1nnc(C(F)(F)F)o1)C2 47671,CC1(C(=O)NC2CCOC2)CCCN1C(=O)CCC1CCOCC1 47672,N1(C(C(CCC)F)=O)CCN(C(=O)CC2COC(=O)C2)CC1CCC 47673,C1(CNC(C(CC2CCC2)OC)=O)CN(C)CCN1C(=O)CC1CC1 47674,C(c1cccc(Cl)c1Cl)=CC(=O)NCCCCCCNC(=O)CC1CCOC1 47675,CONC(=O)C(=O)NCC(C1CC1)NC(c1nnc(S)n1C)=O 47676,C1(c2nn[nH]n2)(C(N2C(C(=O)NC(c3cccs3)COC)CSC2)=O)CCOCC1 47677,N(C(=NCCCN1CCOCC1)NCC(=O)NOC)CCN(C(=O)OC)C 47678,c1(C(=O)NC(CC)CCC(=O)NCC(N2CCOCC2)=O)ccc2c[nH]nc2c1 47679,n1(CCNC(C2CC3CC3N2C(=O)Cc2cccs2)=O)cnc2ccccc12 47680,CCC(CC(=O)NCC(C)(O)C1CCCC1)NC(=O)C(C)OCCOC 47681,C(=O)(C(COC)NC(C1CC(OC)C1)=O)N(C1CCN(C(C)(C)C)C1)CC 47682,c1(OC)cc(C(N2CCC(O)(C(C)NC(=O)C=Cc3ccco3)C2)=O)ncn1 47683,C(C1CCCN1C(=O)CN1CCCCC1C)=CC(=O)NCc1n(CCC)cnc1 47684,c1(C(=O)NC(C)CCNC(=O)CSC(F)(F)F)cnn(CC(F)(F)F)c1 47685,c1(C(=O)OC2CN(CCC)C(=O)C2)c(C)nn2c1CN(C(=O)OC(C)(C)C)CC2 47686,c1(C(N2CCCC(C)(C(=O)NCCC[Si](CC)(C)C)C2)=O)cnc(O)cc1O 47687,n1(CCCC)nc(C(=O)N(C)CC2(CO)CC2)ccc1=O.C1(=O)C(OC)N1 47688,c1(CC)c(C(N2CC(c3ccccc3C(=O)O)(O)C2)=O)cnn1C1CCCC1 47689,C1(CNC(C(CCCC)NC(N)=O)=O)CC2(CCC2)CN1C(=O)CCC(C)OC 47690,N1(C(c2c(C)snn2)=O)CCCC(CNC(C2CN(C3CCOC3)C2)=O)C1 47691,C1(C(=O)NCC2(CN(C(CC3CC(OCC)C3)=O)C)CC2)CC2CCC1NC2=O 47692,C1(F)(C(=O)NC2CCC(C(N(C(c3ccccn3)C)C)=O)C2)CCOCC1 47693,Cc1nccnc1C(=O)NCCC(C)(C)NC(C1CC(F)(CF)C1)=O 47694,c1(C(N2CCC(NC(C3C(CC)C3)=O)C2)=O)cccc(OC)c1Cl 47695,c1(CC(C)C)ccc(C(C)C(=O)N(CCCN(C)C(c2csc(Cl)n2)=O)C)cc1 47696,C12(NC(c3nc(Br)n4ccsc34)=O)CCCC(CN(C(=O)CO)C1)C2 47697,N1(C(c2c(OC)cncn2)=O)CCC(F)(F)C(CNC(c2cc(Cl)c[nH]2)=O)C1 47698,S(=O)(=O)(c1ccc(F)cc1)Nc1ccc(NCC(N2CCOCC(O)C2)=O)cc1 47699,c1(OC)cc(F)c(C(=O)Nc2cccc(NC(C3CC4(CC4)C3)=O)c2)cc1F 47700,C#Cc1cccc(C(=O)NCC2(OC)CN(C(C3CCC(C)CC3)=O)C2)c1 47701,N1(C(CCc2cccc(OC)c2)=O)CCC2CN(C(C3CCCS3)=O)CC12 47702,C1(C(=O)N(C(=O)Cn2ccnc2)CCCC2CCCCC2)CC(F)(F)C1 47703,c1(CC(=O)N(CCNC(c2c(C)ccnc2)=O)C2CC2)ccc2ccccc2c1 47704,CC1(C)CC(CC(N2CC(O)CC2CNC(C2CC=CCC2)=O)=O)CC(C)(C)O1 47705,c1(CC)ccsc1C(=O)N(CC(C)C(=O)N(CC(CC)OC)C)C 47706,C1(CC(=O)NCC(C#C)CC2CC2)CN(C(=O)Cn2c(C)ccc2C)C(C)(C)C1 47707,CC1(C)CC(CNC(C2CC=CCO2)=O)N(C(c2ccnc(C#N)c2)=O)C1 47708,Cc1[nH]nc(C(N2CCCCC2CN(C)C(c2cc(C#N)on2)=O)=O)c1F 47709,N1(C(c2c(CC)n(C)cc2)=O)CC2CN(C(C34CC(CC)(CO3)C4)=O)CC2C1 47710,N1(C(c2c(C)nns2)=O)CC2(CCN2C(c2ncn(C)n2)=O)C1 47711,c1(C(C(=O)NC(C)CN(C(=O)CCc2cnn[nH]2)C)O)ccccc1C(F)(F)F 47712,C1(NC(c2nc(C)sc2)=O)CC(C(NC[Si](C)(C)C)=O)C1(C)C 47713,Cc1cc(CC(=O)NC2CCN(C(c3csc(Br)n3)=O)CC2)nn1C 47714,N1(C(c2nc(C)sc2C)=O)CCCCC(CNC(C23CC(CO2)C3(C)C)=O)C1 47715,N1(c2cc(C)nc(N(C)CCc3nccc(O)n3)n2)CCc2nc(Br)sc2C1 47716,N1(C(CCC(=O)N(C)C)=O)CCC2CN(C(C3CCn4nnnc4C3)=O)CC2C1 47717,c1(C(C)C(=O)NCC2CCCC2NC(=O)Cc2cc[nH]c2)ccc(N)cn1 47718,c1(CN=C(NC(CC)CC)NC2CCSC2C)ccc(F)c(Cl)c1 47719,C1(C2CCCCO2)(C(=O)NC2CC(NC(c3ccn(CC)c3C)=O)C2)CCCO1 47720,CCC(C)C(C(=O)NCC=CCNC(c1ccc(C2CCC2)nc1)=O)OC 47721,C=CC(O)(C(=O)NC1CCN(C(=O)C(=O)NCCOC)CC1O)C(F)(F)F 47722,c1(NCC(=O)N(c2ccc(C(CC)C)cc2)C)cc2oc(C)nc2cc1Cl 47723,C(=O)(C(O)CC[S+](C)C)NC1C(NC(c2ncc(C)c(C)c2)=O)CCCC1 47724,CC1CC(N=c2nc3c(cnn3C)c(NCc3ncoc3C(F)(F)F)[nH]2)CCO1 47725,C1(C2CCC2)(C(=O)NCC(C)(C)OCCNC(C2CCC(F)(F)C2)=O)CCC1 47726,C=CCCCCCCC(=O)N1CC(CN(C(=O)CC2CCOCC2)C)C2(CC2)C1 47727,c1(C(=O)NCC=CCNC(=O)CC23CCCC2C3)cc2cccnc2o1 47728,C1(NC(C2(CC#C)CC2)=O)CC=C(C(=O)NC2CC3C(C2)C3(F)F)C1 47729,CC1CCc2ncc(C(N3CCCC34CCN(C(c3ccccc3)=O)C4)=O)n2C1 47730,C1(NC(=O)Cc2cc[nH]n2)COC2(CCN(C(c3cnc4c(c3)CCC4)=O)C2)C1 47731,Cn1cc(Cl)cc1C(=O)NCc1ccoc1C(=O)NC1CCCC(F)C1 47732,N1(C(C(=C)F)=O)CCC2CN(Cc3ccc(Br)cc3O)CC12 47733,CCC(CC)(CCNC(=O)C(C(C)(C)C)SC)NC(=O)COC(F)F 47734,N1(C(C(N2CCCC(C)C2)=O)=O)CCCC2(NC(C3CC4CCC3C4)=O)CC2C1 47735,c1(NC)ncccc1C(=O)NCCC(O)CNC(=O)CCC1CC(C)C1 47736,c1(C(=O)NC2CC(NC(C=CCOC)=O)C2)cc2c(nc1O)CCCC2O 47737,C1(NC(C(CSC)C)=O)CCC2(CCN(C(c3ccoc3Cl)=O)C2)C1 47738,CN1CCC(N(C(c2csc(C(F)(F)F)c2)C(=O)NC2CC2)C)C1 47739,c1(C(=O)NC(C)(C)CCNC(=O)C2=C(Cl)CCOC2)c(N)c(F)cc(F)c1F 47740,c1(OC)ccc(C(=O)NCC2(CNC(C3CC34CC4)=O)CCC2)c(Cl)n1 47741,CCCCCC(O)C(=O)N1CC2=C(C1)CN(C(c1ncc(Br)cc1N)=O)C2 47742,c1(C(=O)NCC(C)N(c2ncc(C)c(O)n2)C)ccc2nnc(O)n2c1 47743,C#Cc1nccnc1NC(C1CC1NC(c1cnc(C(F)(F)F)cn1)=O)=O 47744,C(=O)(C(O)C(F)(F)F)N1C(C(N2CCC(C(C)C)C2)=O)C(C)C1 47745,CC(C)CC(C(N)=O)NC(c1n[nH]c2c1CCC2)=O 47746,CC1CN2CCN1C(C(=O)NC(C)(C)CNC(=O)CCCN1CCCC1)C2 47747,c1(OC(C)C)ccc2c(c1)CCN(C(=O)C(=O)NCC1CCCCC1C)C2 47748,CCC(C)(O)C(=O)N1CCN(C2CCCC2NC(=O)C=CC2CCCCC2)CC1 47749,CC1(C)CC(NC(c2ccc([N+](=O)[O-])s2)=O)CN(C(=O)Cc2cc[nH]n2)C1 47750,C(=O)(C#CC1CC1)N(C1CCN(C(CN(C)CC2CCC2)=O)C1)C 47751,N1(C(C2N(C)CCCC2)=O)CCN(C(=O)CSc2ccncc2)C(CF)C1 47752,C(C(C)N=c1[nH]c(=N)[nH]c(=NCC(F)(F)c2cccc(F)c2)[nH]1)(C1CC1)OC 47753,c1(C(N2CC(C)C(CNC(C3CC34CCCC4)=O)C2)=O)ccc(F)c2c1OCC2 47754,CC1(C(=O)NCC(C2CCCC2)NC(c2cc(Br)no2)=O)CC(F)C1 47755,N1(C(C(COC)C)=O)CCC2(CCCN2C(c2cncc(OC(F)F)c2)=O)CC1 47756,C1(NC(c2c(CC)scc2)=O)CC(CNC(c2cn(C)nc2OC)=O)C1(C)C 47757,C1(C(N(C(CNC(c2cc(C)nc(C(F)F)n2)=O)C)C)=O)CCn2nccc2C1 47758,Cn1ccc2cc(C(N3CCC(NC(c4ccc(F)o4)=O)C34CC4)=O)ccc12 47759,C1(NC(c2nc(CC)sc2)=O)CN(C(=O)Cc2cc[nH]c(=N)c2)CC2(CC2)C1 47760,N1(C(C(CC(=C)C)NC(=O)Cn2cc(C#N)cn2)=O)CC2(CC(CO)CO2)C1 47761,c1(C(=O)NC(C)(C)CNC(C23CCCN2CCC3)=O)ccc2c(c1)NC(=O)CC2 47762,c1(OC)ccc(C(N2CCCC2CN(C(=O)CC2CCCC2C)C)=O)cc1 47763,C1(NC(C(CCC)CNC(=O)C(CO)OC)=O)CC(C2CCCC2)C1 47764,C1(C)(C(N2CC(C(C)(C)O)(CNC(C(C)OCCC=C)=O)C2)=O)CC2CC2C1 47765,C12(C(=O)NC3CC(CC(=O)NCC4CCCCC4O)C3)CCCC1C2(F)F 47766,CC1(C(=O)NC2C=CC(CC(=O)NCCn3cncn3)C2)CCCOC1 47767,c1(OC)cc(C(=O)NC2CC2NC(=O)CC2OCCO2)c2ccccc2c1 47768,C1(c2nc(COC)nn2C2CCOC2)CCN(c2ccccc2)S1(=O)=O 47769,C1(c2n(CCC)nnn2)(NC(c2cccc(Br)c2)C)CNC(=O)C(C)(C)C1 47770,c1(C(N2C(C)CC(NC(c3nn[nH]c3Cl)=O)C2)=O)nccc2ncccc12 47771,c1(C(=O)NC2CC(NC(CN(C3CCC3)C)=O)C2)c(F)cccc1F 47772,c1(-c2c(OCC)cccc2)cnc(C(=O)Oc2ccccc2)cc1OCCOC 47773,C1(CNC(C2CCC(CC)O2)=O)CCCN(C(=O)Cc2cncnc2O)CC1 47774,c1(C(=O)NC(CC)CNC(=O)CC2CCCOC2)cccc(N)c1C 47775,C1(F)(CNC(C2(C(C)C)CCC2)=O)CCN(C(C2CC(F)(CO)C2)=O)C1 47776,N1(CCC(CC(=O)OCC)(C)C)CC23CCCC2(C1)CN(C)C3 47777,C1(C#N)(C(N2CCC(CC=C)(NC(=O)C=CCC)CC2)=O)CC2CCC1CC2 47778,C12(CC(=O)NCC3CCC(C)S(=O)(=O)C3)CC3CC(C1)CC(Br)(C3)C2 47779,C(=O)(C(C#N)C(C)C)NC(C(=O)NC(c1scc(C)n1)C)C 47780,C1(C#N)(C(N2CCN(CCCNC(C(C)C(F)F)=O)CC2)=O)CC2CC2C1 47781,N1(C(c2cnc(OCC)s2)=O)CCC(C(C)NC(=O)COc2cnn(C)c2)CC1 47782,CC1CC(C)C(C(=O)NC2CCN(c3nccc(-c4ccccc4F)n3)CC2)O1 47783,N1(C(c2c(C#C)c[nH]n2)=O)CC(=O)NCC1C(=O)NC1CCCC12CC2 47784,S(=O)(=O)(c1c[nH]c(C(N2C3CCC2CN(C(c2ccon2)=O)C3)=O)c1)N(C)C 47785,N1(C(=O)NCC(N2C(C)CC3(CC3)C2)=O)CC2(CCN(C)CC2)C1 47786,CN1CCC2CCC(C1)N2C(=O)Nc1cccc(Oc2ccccc2)c1 47787,C(=O)(C(C)(C)S(C)(=O)=O)NC(C1CCCN(C(=O)COC(F)F)C1)C 47788,C1(NC(C2(C)CC2(F)F)=O)CCC(NC(=O)C(c2ccccc2)=O)CC1 47789,Cn1ccc2cccc(C(=O)NCC(O)CCNC(C3(C)CC3(F)F)=O)c12 47790,CCC(CC(=O)N1CC(F)CC1CO)NC(=O)C=Cc1cn(C)cn1 47791,CC1CCCN(C(=O)CC2CCCC2)C1CNC(c1csc(C(C)(F)F)n1)=O 47792,c1(OC)ccc(-c2onc(C(=O)NC3CC(CNC(=O)CSC)C3)c2C)cc1 47793,c1(CSC(C(=O)N(CC(CC)NC(=O)C(F)=C(C)C)C)C)ccc(F)cc1 47794,C(CC(C)CN=C(NCc1nsc2ccc(Cl)cc12)NC(c1cccs1)C)OC 47795,Nc1cnc(C(=O)NCC2(NC(C34CC(F)(C3)C4)=O)CCCCC2)cn1 47796,C(=O)(CC(C(F)(F)F)NC(c1sccc1F)=O)NCC1C(C(C)C)C1 47797,c1(C(C)C)oncc1C(=O)NCC1CCN(c2ccccc2)C1 47798,c1(C(=O)NC2(C(=O)NC(C=C)C3CC3)CC2C)cc(CO)[nH]n1 47799,CN1C(C)(C)C(Nc2ccnc(CO)n2)CS1(=O)=O 47800,N1(C(C(CCCC)O)=O)CC2CCC1C(NC(=O)C(C(=O)OCC)OC)C2 47801,C1(NC(C2N=C(C)SC2)=O)CC1C1CCCN(C(c2cc(C3CC3)ccn2)=O)C1 47802,C1(NC(N)=O)CC(=O)NC1=O.C12CCN(C1)N(CC(C)C)C(=O)C2.CCN 47803,C(=O)(CC(C)Cc1ccccc1)N(CCNC(c1c(COC)cc[nH]1)=O)C1CC1 47804,c1(OC)ccc(CCNC(=O)C(=O)N(CCO)CC2(C)CCCC2)cc1C 47805,c1(C(=O)NCC2(F)CCN(C(C3CCCOC3)=O)CC2)cnc2ccnn2c1O 47806,C1(CNC(CCN(CCC)C)=O)CC(CNC(=O)C(C)(C)NCC)CO1.[SH](C)(=O)=O 47807,N1(C(C2(C)CCN(C(C3CC(=O)CS3)=O)C2)=O)CCCc2occc2C1 47808,N1(C(c2c(C)n(C3CC3)cc2)=O)CC(NC(=O)CCc2ccccn2)C(C)(C)C1 47809,C(=O)(CCCCCF)N(C(C)C(=O)NC(C)(C)CCCO)CC 47810,C12(C(N3CCCC(NC(C(c4cccc(OC)c4)O)=O)C3)=O)CC(N=[N+]=[N-])C1C2 47811,C=CC(CC)CC(=O)NCC1CCC(NC(c2cnn(CC(F)(F)F)c2)=O)CC1 47812,C(=O)(CS(=O)(=O)C1CC1)NCC1C(NC(C(C)Cc2ccncc2)=O)C1 47813,C(CN=c1nc2cccc(Br)c2c[nH]1)C1CCN(C(c2c(C)noc2)=O)C1 47814,N1(C(C2C(C=C)CC2)=O)CC(CO)C2(C1)CN(C(c1cnc(O)c(F)c1)=O)C2 47815,C1(NC(=O)C=C(Cl)Cl)CCCCCC1NC(C1CC2CCC(C1)C2)=O 47816,CCCCCC(C1CC1)NC(=O)CNC(c1ccc(C)nc1)=O 47817,c1(NC(C2N(C(C(C)O)=O)CC2)=O)nc(Cl)ccc1F 47818,CC(C)C(CCN(C)C(c1csc(CO)n1)=O)NC(C1(O)CC1(C)C)=O 47819,CC(C)(C)CC(O)CC(=O)NC(CCF)C(=O)NCc1ccc(C(N)=O)o1 47820,C1(C(NNC(C=Cc2c(C)cccc2)=O)=O)C2CCCCCCC12 47821,C(=O)(C(C)CCCOC)N(C(C)CNC(=O)CCCCSC)CC 47822,C1(c2nnnn2C2CCC2)(Nc2ccc(C(C)(C)CO)cc2)CC2CCOC12 47823,N1(C(CC2CC(CC)C2)=O)CCOC2CN(C(C3CC3CC)=O)CC12 47824,CC1COCC(CC(=O)N(C2(C(N3CC(O)(c4cc[nH]n4)C3)=O)CC2)C)O1 47825,C(=O)(C1=CC2(CCOC2)C1)N1C(C(=O)NCc2ccc(O)c(F)c2)CC2CC21 47826,c1(C(=O)NCC(CC=C)NC(=O)Cc2ccc(F)c(F)c2)onc2c1CCCC2 47827,CCC(C)CC(C)C(=O)NC1(CNC(=O)C(C)(C)Oc2cccc(Cl)c2)CC1 47828,C(CC(=O)NCC1=CCN(C(c2sc(C#N)cc2Cl)=O)CC1)(C(N)=O)NC(C)=O 47829,c1(C(=O)NC2C3N(C(C(CCCC)O)=O)C(CC3)C2)cc2c(C)cccn2c1 47830,N1(C(CNC(CC)=O)=O)CCC(O)(CCNC(c2c[nH]nc2C)=O)CC1 47831,Cc1cc(OCC2CCCO2)ccc1NC(=O)NC1CCC2COC1O2 47832,c1(C(=O)NCC(CNC(c2cc[nH]c2)=O)F)cccn2cc(C(F)(F)F)nc12 47833,CC1CN(c2nnnn2CCC2CCCCC2)CCCO1 47834,Cc1cccc(C2CC2C(=O)Nc2cn[nH]c2)c1.N12CCC1CNCC2=O 47835,C(=O)(CCCCC(=O)NCCC1CCCN(c2nccc(C)n2)C1)NC 47836,N1(C(c2cnc(C)nc2C)=O)CC(NC(C2(Cl)CC2)=O)C(N=[N+]=[N-])C1 47837,c1(C(=O)NCC2(C)C(C)CN(C(c3cc(C#N)c[nH]3)=O)C2)cc2ncccn2n1 47838,c1(CC(=O)NC2CC3(CN(C(C(C=C)O)=O)C3)OC2)c[nH]c2ccc(Br)cc12 47839,N1(C(C(N2C(C3C(C)(O)CCCC3)CCC2)=O)=O)CCCc2ncc(F)cc21 47840,C=CCC(C)(C)CCNC(c1cc(Cl)cc(OC)n1)c1nnnn1CCCCCC 47841,C12(NC(C3(CC)CCN(C(c4c[nH]nc4C)=O)C3)=O)CC1COC2(C)C 47842,C1(NC(C2C(=C)CC2)=O)CC2CC(NC(=O)CCC3CCOCC3)C1C2 47843,C12(NC(=O)OC(C)(C)C)CCCN(C(=O)C(Cc3cccnc3)C3CCCC3)C1C2 47844,C1(CNC(=NC)NCCC(C)SC)CNCC(C)(C)O1 47845,C1(CCCC)(C(N2CCC(C(C)NC(=O)CC)C2)=O)CCCC1.C1(C)C(=O)N1 47846,CC(c1cccnc1)=CC(=O)NCC1(CO)CCCO1 47847,C(=O)(C1=Cc2ccccc2C1)NC(CC)CNC(c1c(C)nsc1Br)=O 47848,C(=O)(CC1=CCCCC1)N1C(C)CCC(NCc2cnccn2)C1 47849,C1(C(=O)NC(C(C)NC(=O)Cc2nnn(C(C)(C)C)n2)CO)CC12CCCCC2 47850,CC1(C(=O)NCc2ncccc2O)CCCN(C(C2CCOC2C2CC2)=O)C1 47851,C(=O)(C1=NOC(C)(C)C1)NCCCCCCN(C(C(CC#C)C1CC1)=O)C 47852,C(CC1=CCN(C(=O)CC2CCNC2=O)CC1)NC(c1n(C)c(Cl)cn1)=O 47853,C1(C(C)(C)C)CCCCN1C(=O)Cn1nccn1.n12cc(nn1)C2 47854,c1(C(=O)NC(CCCCNC(c2ccn(COC)n2)=O)C)ccc(S(C)=O)cc1 47855,c1(CC(N2C(CN(C)C(C3CC3(Cl)Cl)=O)CC(F)C2)=O)ccc2c(c1)COCC2 47856,C1(NC(C2N(CC)CCC2)=O)CC2(CCN(C(=O)Cn3nc(C)nc3C)C2)C1 47857,c1(C(=O)NCC(CNC(=O)CCC2CCC(=O)N2)OC)ccn2cncc2c1 47858,c1(C(=O)NCc2ccc(C(=O)NC(c3cccs3)(C)C)o2)cccc(F)c1O 47859,CCCCC(CC)C(=O)N1CCCN(C(c2ccc(Cl)nc2O)=O)CCC1 47860,N1(C(CCC#CC)=O)CCC(NC(c2nn(C)c(Cl)c2C(F)(F)F)=O)C(C)C1 47861,O=C1CC(C2CC2)(C(=O)NC23CCC(NC(=O)C=CBr)(CC2)C3)C1 47862,C1(C(=O)NCCOCCNC(n2cccc2)=O)(CO)CCCO1 47863,c1(C(N2CCn3ncc(I)c3C2)=O)cc(C(F)(F)F)nc2ccccc12 47864,C(=O)(C(F)(F)C(C)(C)O)N(C1(CC(=O)N2C(C)C2=O)CC1)C.CO 47865,C(=O)(CC(O)CC(C)(C)C)N1CCC(C(C)C(=O)NC2CCOC2(C)C)CC1 47866,n1(CC(=O)OC)cc(CNC(=O)NC(C2CCCCC2)c2ccccc2)nn1 47867,c1(CC)cccc(F)c1C(=O)NC(C)CNC(=O)C(C)Cc1cccc(Cl)c1 47868,N1(CC(=O)NC(CN(C(C=CC(=O)N(C)C)=O)C)(C)C)CCCC1C(N)=O 47869,c1(OC)ccc2c(c1)CC(C)CC2NC(N1CCCC(n2cnc(C(N)=O)n2)C1)=O 47870,N1(C(C(C)Oc2ccc(F)cc2Br)=O)CC2CCN(C(C3CC3F)=O)CC2C1 47871,C1(N(C(CCN(C(=O)CC2CCOC2(C)C)CC=C)=O)C)CCCC(C)(C)C1 47872,C1(C(=O)OC)C(C)OCCN1C(CCc1cccc(Cl)c1)C(=O)NCC#N 47873,c1(C(N2C3CN(Cc4cccc(OCC)c4Cl)CC23)=O)ccc(NCC)cc1Cl 47874,Cc1nc(C(=O)NCC2(F)CC(NC(=O)CC3CCCCC3)C2)c2ccccn12 47875,N#Cc1cc(C(=O)NCC2(NC(c3cn(C4CC4)nn3)=O)CCOC2)on1 47876,n1(CCNC(N2CCCC(N3CCCC3=O)CC2)=O)cccc(C(F)(F)F)c1=O 47877,Cc1nn(C)cc1CN(C(=O)C(=O)N(CCCCC(=O)O)C)C 47878,C1(C(=O)OC)CC(SCC(N2CCN(C(c3ocnc3C)=O)CC2)=O)C12CCC2 47879,C(=O)(CCC1=CCc2ccccc21)NC1C(CNC(c2nnc(C)s2)=O)C1 47880,c1(C(C)(F)F)cccc(C(=O)NCC(CO)NC(c2cccn2C2CC2)=O)c1 47881,N1(C(c2ccc(C)[nH]2)=O)CCCCC(CCC(N2C3CCC2COC3)=O)C1 47882,C1(NCC(N2C(C(=O)OC)CC2C)=O)CCCN(C(=O)C=CCN(C)CC)C1 47883,Cc1cc(Nc2cc(NC(C)CN3CCCCC3)ncn2)cc(C)c1 47884,c1(NC(C2CCCN(C(C3CC(=O)NCC3)=O)C2)=O)ccc(F)c(CO)c1 47885,C1(COC)CN(C(c2ccc(-c3ccccc3)cc2Cl)=O)CC(C)O1 47886,C1(CC=C)(NC(=O)COC2CCCC2)CCN(C(c2ccccc2C(C)=O)=O)C1 47887,Cc1ccc(C(=O)NC2CC(N(C(=O)CCc3cscn3)C)C2)c(F)c1C 47888,C(CCN(C)C(C12CC(C1)C(C(F)(F)F)O2)=O)(C(C)C)NC(CC1CC(=C)C1)=O 47889,N1(c2nc(C)cc(C)n2)CCC2(CC1)CN(Cc1c(F)cccc1I)C2 47890,N1(C(C(CC(C)C)C)=O)CCC(C2CCCN(C(=O)CC3SC(=N)NC3=O)C2)C1 47891,C1(C(N2CCN(C(c3cccc(C)n3)=O)C(CO)C2)=O)CCc2nc(C)nn2C1 47892,CC(C)(CN=C(NC(C1CC1)C1CC1)NC1CCC(F)(F)C1)OCCOCCSC 47893,C1(NC(COCCCC)=O)CN(C(=O)C(n2nc(C)cc2C)C)CC1SC 47894,C(=O)(CCC(=O)C(C)(C)C)NC1CCC(CCC(=O)NCC(N(C)C)C2CC2)C1 47895,Cc1ccccc1OCC(=O)NC1COCC1C(=O)NC(CO)C(C)C 47896,C(=O)(C(CC(C)C)C(C)C)N1CC(OC)C(C(=O)NCC2CC3(CCC3)CO2)C1 47897,c1(C(=O)NCC2C(CNC(c3cc(OC)n[nH]3)=O)C2)cc2c(cc1O)OCO2 47898,C=CCCC(CC(C)C)C(=O)NC1CN(C(=O)Cc2ncccc2C)CCC1O 47899,CCCC(CCCO)C(=O)N1CCN(C(C2CCCN(C(C)=O)C2)=O)C(C)C1 47900,CN(S(N)(=O)=O)C.c1(C=O)cn(C2CC(C(=O)NCCc3cncnc3)C2)nn1 47901,CCCCCCC(C(=O)NC1(C)CCN(C(=O)C(C)(C)C2CC2)C1)NC(C)=O 47902,c1(C(N2CC3C(CNC(C=C(C)C(=O)O)=O)(C3)C2)=O)ccnc(Cl)c1C 47903,Cc1nc(F)ccc1NC1(c2nnnn2C2CCOCC2)CCN(C2CC2)C1 47904,C1(CNC(C2(OCC)CCCC2)=O)CCCC(NC(=O)COC(C)(C)C)C1 47905,N1(C(C(C)(C)C2CCOCC2)=O)CC2CCCC(NC(c3cnsc3)=O)C2C1 47906,c1(C(=O)NCC23C(CN(C(c4cn(CC=C)nn4)=O)C2)C3)cccn2cnnc12 47907,CCC(C)C(C)C(=O)N1CC(O)(CNC(c2csc3nnsc23)=O)C1 47908,C(CC(C(=O)NOC(CO)C(C)C)NC(C1CC(C(C)C)C1)=O)=CC 47909,CCC(C(=O)NCC(CNC(=O)C=CCO)OC)Sc1nc(=N)[nH][nH]1 47910,N1(NC(C2CCCCC2)(C)C)CC(=O)N(Cc2ccc(CSC(F)F)o2)C1=O 47911,c1(CC)cc(N2CC(C3CC3)CC2C2CC2)n2ncc(Br)c2n1 47912,C1(NC(c2nc(OC)c(F)cn2)=O)CCN(C(=O)CC(=O)NC2CC2)CC1C 47913,C1(C(=O)NCc2c(C)noc2)C2CCN(C(=O)CCC(C)CN(C)C)CC12 47914,C1(NC(C(CC)NC(N)=O)=O)CC2CCC1C(NC(C1CC(CN(C)C)C1)=O)C2 47915,C(C)(C(C)(C)NC(=O)Cc1ccn(C2CCCC2)n1)NC(CSC)=O 47916,CC1CCN(CCC(=O)NCC2C(C)CCN2C(c2cc(C#N)on2)=O)CC1 47917,c1(OC)cc(OC(C)(C)C)ccc1NC(=O)NCCCC(C)C1CN(C(C)=O)C1 47918,CC(C)C(C)CC(=O)NCC1(C(C)(C)O)CN(C(=O)CC2OCCO2)C1 47919,C(c1ccc([N+](=O)[O-])s1)=CC(=O)N(C)CC1CCCCN1C(=O)C1=COCCC1 47920,Cc1oc(C(C)(C)C)cc1C(=O)NCC1CC1NC(c1cnoc1C(C)C)=O 47921,c1(C(N(C2CCN(C(Cc3cc(C)nc(O)c3)=O)C2)C)=O)coc2ccccc12 47922,N1(C(c2nn(C)c(C(N)=O)c2)=O)CCN(C(=O)Cc2ccsn2)C2CC12 47923,CCC(CC(=O)NC(CNC(c1ccc(Cl)s1)=O)CC)C(C)C 47924,N1(C(=O)CC2CCOCC2)CCCCC2(CCN(c3nnco3)C2)C1 47925,C1(CS(C)(=O)=O)CN(C(=O)C=CC2CCCO2)CCN1C(=O)C(Cl)=CCl 47926,CC(CN(C(=O)C(CCN(C)C)NC(C1CC(O)C(F)C1)=O)C)C(C)(C)C 47927,c1(C(N2CCC(N(C(C3C(COC)C3)=O)C)C2)=O)cc(C2CC2)oc1C1CC1 47928,N1(C(C(C)(C)N(C)C)=O)CCC(C2CCCN(C(C3CC3C(C)(F)F)=O)C2)CC1 47929,c1(OC)cc(-c2cnc3cc(C(N4CCOCC4)=O)[nH]c3c2)cc([N+](=O)[O-])c1 47930,C1(CNCc2cccc(OCCCC)c2)CCCC1C1CC1 47931,C1(NC(c2cc(CC)[nH]n2)=O)CCCCC1NC(=O)C=CC(C)C 47932,N1(C(C(CC(C)C)F)=O)CCC2CCC(C1)N2C(c1cccc(SCC#N)c1)=O 47933,N1(C(C2N(C(C3C(C(=C)C)OCC3)=O)C3CCC2C3)=O)CCc2ccc(F)cc21 47934,C(CC1c2ccccc2CCN1C(c1ccon1)=O)NC(=O)C(C1CC1)C1CC1 47935,CC1CN(C(c2nocc2C(C)(C)C)=O)CC(CCNC(=O)C2=CCSC2)O1 47936,c1(NC(C)CCC2CCCO2)cc(NCC(C)(C)CN2CCCCC2)ncn1 47937,C1(CNC(C=NOC)=O)CN(C(=O)CNc2cccc(Cl)c2)CC12CCC2 47938,CCCC(CC1CCCC1)C(=O)NCC(C)(C)CNC(c1c(C)cccc1F)=O 47939,c1(C(N)=O)ccccc1C(=O)NC1CCC1CNC(=O)C(C1C=CCC1)=O 47940,C1(C(=O)NCC=CBr)CCCN(C(=O)CCC2CCCO2)CC1 47941,Cc1ncc(C=CC(=O)NCC2CCCN2C(=O)C=CC(c2cnn(C)c2)=O)s1 47942,c1(CCC)ccc(C(=O)N(CCC(C)NC(=O)CC2CCCO2)C)s1 47943,C1(CNC(C=CC(C)(C)SC)=O)CCCN(C(C2(C)C=CCCC2)=O)C1 47944,CC(C)C(O)C(C)(C)C(=O)NCC1CCC(NC(=O)CN2CCC(O)CC2)CC1 47945,Cc1cc(C(=O)NC(C2CCN(C(c3ccn(C(C)C)c3C)=O)C2)(C)C)ccn1 47946,c1(NCC(C(C)(C)C)SC)ncnc(NCCc2nc(C)cs2)c1C 47947,C1(NC(c2ncc(CC)s2)=O)CC2CCC(C1)N2C(c1cnc(OC)nc1C)=O 47948,N1(C(C(C(C)C)C)=O)CCC(CNC(=O)CN2CCCS2(=O)=O)C12CC2 47949,C1(CNC(C2C3CNCC23)=O)CCN(C(=O)CCC2CCCC2)CC1 47950,c1(C(N2CC3(CN(C(C(C(C)(C)C)OC)=O)C3)C2)=O)cc(Cl)cc(Cl)c1Cl 47951,O=C1CNC(=O)c2cc(C(=O)NCC(CNC(=O)C(F)(F)CO)CO)ccc2N1 47952,c1(NC(CC(CC)O)=O)ncc(-c2ccc(N(C)C)c(C)c2)cc1O 47953,C1(NC(c2c(COC)cco2)=O)(CO)CCN(C(c2ccsc2SC)=O)C1 47954,c1(CNC(CN(C(COC2(C#C)COC2)=O)C)=O)c(C)noc1CC 47955,c1(C(=O)NC2(CN=c3[nH]nc(C)s3)CCCCC2C)cnc2nncn2c1C 47956,N1(C(CSc2ccc(OC)cc2)=O)CCCC(C)C1CNC(c1ccncc1)=O 47957,CN1CCN(C(c2ncncc2F)=O)C(CNC(C2(F)CCOCC2)=O)C1 47958,Cc1nccn1CCCC(=O)NCC1CCN1C(=O)C(F)CC1CCCC1 47959,c1(C(=O)CC2C(CNC(c3cc(SC)c(C)o3)=O)C2)cnc(CC2CC2)nc1C 47960,Cc1ncc(NC(=O)C(C)(C)C2CCN(C(c3cc(F)c[nH]3)=O)C2)c(C)c1C 47961,Cc1nc(NC2CN(C(c3c[nH]c4c(Cl)cccc34)=O)CC2C)c2sccc2n1 47962,c1(CC)cnc(C)c(NC(=O)COC2CCN(C(=O)C=CCOC)C2)c1 47963,C1(NC(CN(C(C)C)C)=O)CCN(C(=O)C(C)(C)C2(C)CC2(F)F)C1 47964,N1(C(C(CCCC)C)=O)CC(NC(=O)CCC2CCC(C)O2)CC2(CC2)C1 47965,N1(C(C(CC#C)O)=O)CC(NC(c2cc(C)ccc2NS(C)(=O)=O)=O)CC(F)C1 47966,c1(CCC(N2C(C(C)NC(C(C)=C3CCCC3)=O)CCC2)=O)ccc(N)c(F)c1 47967,CC(C)CC(CNC(C1CCN(CO)CC1)=O)C(=O)NC(C1(CO)CC1)C 47968,c1(OC)ccc(S(=O)(=O)N(c2cc(C3CC3)nn2C)C2CC3CCC2C3)cc1Cl 47969,c1(C(=O)NC2C(NC(=O)CSc3nc[nH]n3)C2)cc(F)cc(F)c1 47970,c1(NCCC(=O)N(CC(C)Cn2cccn2)C2CC2)cnc(C#N)cn1 47971,N1(CCC(=O)N(C)CC2(CNC(C3CC34CC(O)C4)=O)CC2)CCCC(N(C)C)C1 47972,C1(NC(COCC(C)C)=O)CCN(C(C2CN(C3COC3)C2)=O)C(C)C1 47973,C(=O)(C(CNC(=O)CCC1CCCCC1)OC)N(C1(C#C)CC1)C 47974,C(CCc1c[nH]nc1-c1ccccc1)(C(=O)O)OC(CC(C)O)=O.C(C)(C)(C)OC(N)=O 47975,C=CC(C)CC(=O)N1CC2(NC(=O)CSc3ccccc3)CC1C2 47976,c1(CC)onc(C(N2CCC(NC(=O)CCc3cnn[nH]3)C2C(C)(C)C)=O)c1C 47977,c1(C(N(CCNC(C2C(C)C2C)=O)C2CC2)=O)cnc2ccc(F)cc2c1 47978,CC(C)CS(=O)(=O)CCC(=O)N1CC(CC(C)NC(=O)CCn2ccnn2)C1 47979,C(=O)(C#CC1(C)CCCO1)N1CC(N2CCN(C(C3(F)C(C)OCC3)=O)CC2)C1 47980,N1(C(C2(OC)CCSC2)=O)CCN(C(c2ccnc(C3CC3)n2)=O)C(C(F)F)C1 47981,C12(CNC(C(N)Cc3ccc(OC(F)(F)F)cc3)=O)CCCCC1CCC2 47982,C1(NC(CN(C(=O)Cn2c(C)ccc2C)CC#C)=O)CCn2ncnc2C1 47983,c1(OCCNC(c2n(CCC)nnn2)c2cc(C3CC3)no2)cc(F)cc(F)c1 47984,N1(C(c2ccc(CC)[nH]2)=O)CC(C)(C)CC1C(=O)NCCC1CCCN(C)C1 47985,c1(C(=O)NCC2CN(C(c3n[nH]c(CC)c3C)=O)C2)nnc(O)nc1O 47986,C(C(C)(C)CC(=O)N1CCCCC1CNC(C1CCN(C)C1)=O)OC(C)=O 47987,c1(C(=O)NCCNC(c2cn(C)c(Br)c2)=O)ccnc(Cl)c1O 47988,CCC(C)C(O)CNC(C1CCC(n2cc(C3(O)CSC3)nn2)CC1)=O 47989,N1(C(CCc2ccc(C)nc2)=O)CCN(C(=O)CC2CCCC2)C2CC12 47990,c1(C(=O)NC(CNC(c2n[nH]c(CC)c2Cl)=O)(C)CO)cc(F)cc(Cl)c1O 47991,CON(C)C(=O)CSC1CCN(C(=O)Cc2nnnn2C2CCCC=C2Br)CC1 47992,C1(CC(=O)NCC2N(C(C(C)CC3CCCC3)=O)CCC2)COCCOC1 47993,c1(CC)c(C(=O)NCC(C(C)C)NC(=O)CCC(C)(C)C#N)cnc2ncnn12 47994,c1(C(=O)NC2CCC(C)(CNC(C3(CCOC)CC3)=O)C2)nn(C)c(C)c1Cl 47995,C1(CNC(c2c(CC)ocn2)=O)C(C2CC2)CCN1C(c1scnc1C1CC1)=O 47996,C=CCCC(F)(F)C(=O)N1CC(N(C(=O)CC(C)(C)C(F)F)C)C2(CC2)C1 47997,N1(C(C(CC)n2cccn2)=O)CCC(C(F)CNC(=O)C(C)(C)F)CC1 47998,C1(SC)CN(C(=O)Cc2occc2C)CC1NC(=O)C(C)CNC(C)=O 47999,C(C(=O)NC1CC(F)(F)C1)(C1=NOC2CC12)N1C(CC#N)CC(F)(F)C1 48000,N1(C(C2CC(SC)C2)=O)CCC(C(C)(C)NC(C2CC(C)C2)=O)C1 48001,c1(NC(C2OCCN(C(C(C=C)O)=O)C2)C)ncc(C)c(C)n1 48002,C1(CNC(CCCCC)=O)CCC(C)CN1C(c1ccc(Cn2cccn2)o1)=O 48003,C1(NC(CCC#CC)=O)CCCCN(C(=O)CCCNC(C)=O)C1 48004,C1(CNC(c2conc2C(F)(F)F)=O)CN(C(c2n[nH]cc2Cl)=O)CC1O 48005,C(=O)(CC(C)(C)N(C)C)NCC(CC=C)NC(=O)Cn1cc(Br)c(C)n1 48006,Cc1cc(C(C)C)ccc1C(=O)NC(C1CCN(C(=O)CC2CCOC2)CC1)C 48007,C1(CC)C(NC(C2CC2CF)=O)CCCN1C(c1ccc(CN(C)C)o1)=O 48008,c1(C(=O)NC(CN(C(c2cc3cccnc3[nH]2)=O)CC)C)cnn2cccnc12 48009,N1(CC)CCOC(C(N2CCCC(CNC(c3ncoc3C(C)(C)C)=O)C2)=O)C1 48010,Cc1cc2ncc(C(=O)NCCC3CC(NC(C4(C)CC4(Cl)Cl)=O)C3)c(C)n2n1 48011,CC1(C(=O)NOCc2cccc(F)c2)CCN(C(c2nccnc2N)=O)CC1 48012,C(=O)(C1=CCC(C)(C)CC1)NC(CC#C)C(=O)NC1(C)CCC(C)(C)C1 48013,C=C(Cl)CC(C(=O)NC1CC(C)(O)C1)NC(c1cc(Cl)cn1C)=O 48014,N1(C(c2ncn(C)n2)=O)CC2CCCC(C1)N2C(=O)CC=C(Cl)Cl 48015,CCC(C)C(C(=O)NCc1cnn(C)c1O)N(C(=O)C#CC(C)(C)C)C 48016,Cc1ccc2c(CN3CCC(CC(=O)Nc4c(C)cccc4Br)CC3)c[nH]c2c1 48017,C1(NC(=O)CN2C(=O)CNC2=O)CCC12CN(C(c1ccnn1CC(F)F)=O)C2 48018,N1(c2sc(C#N)c(Cl)n2)CCc2sc(C(=O)NCCCOC(F)F)cc2C1 48019,CC(C)CCCCC(=O)NCC=CC(=O)NC(C1CCOCC1)C 48020,N1(C(c2c(C)cccc2F)=O)CC(NC(=O)C=CC2CCCO2)CC2(CCC2)C1 48021,c1(C(=O)NC2C(C(=O)NCCCN3CCOCC3)COCC2)cc2occc2[nH]1 48022,C1(C(=O)NC(C=C)C2CC2)CCC(C)(C)N(C(=O)CCC(C)CN(C)C)C1 48023,CCC(C(=O)N1CC(N2CCCC2)C1)NC(=O)COC1CCCC1 48024,N1(C(=O)NCC(=O)Nc2cccc(Cl)c2)CCC2(NC(c3cccs3)=O)CC2C1 48025,c1(C(c2nnnn2CCCC)NC(C=C)C)nnc(CC)s1 48026,C=C1CCN(C(=O)C(C)CN(C)C(C2(C)CC=CCC2)=O)CC1 48027,c1(C(C)O)ccc(C(=O)NC(C2CN(C(=O)COCP(C)(C)=O)CCO2)C)cc1 48028,N1(C(C=Cc2ccc(C)s2)=O)CC(C)CCC1CNC(=O)CC1(C)CCOC1 48029,C1(C(N(CCNC(CN2CC(CC)C2)=O)CC2CC2)=O)CCc2ccnn2C1 48030,C(C(N=c1ccnc(NCCCn2cccn2)[nH]1)C1CCCO1)SC 48031,C1(NC(C(C)C2(O)CCC2)=O)CC(C)(NC(=O)CC(C)N(C)C)C1 48032,CCC(CN=c1ccc(Br)c(S(=O)(=O)N2CCC2c2cc(C)cc(C)c2)[nH]1)OC 48033,C(=O)(C(O)C1=CCCCC1)NCC(CO)NC(c1c(C)nc(CC)s1)=O 48034,c1(C(C)(C)C)ncc(NC(C2CCN2Cc2ccc(Br)o2)=O)cn1 48035,CCCC(CCCNC(=O)COc1ccsc1)NC(=O)C=Cc1c(C)coc1C 48036,N1(C(C2C=C(C)CS2)=O)CCC(NC(C2CCS2(=O)=O)=O)C1C1CC1 48037,CC(C)CC(O)CC(=O)NCc1nocc1C(=O)NOCC(=O)OC(C)(C)C 48038,CC1CCC(c2nnnn2C2COC2)(NCc2cscn2)C1 48039,c1(C(=O)NC2CCN(C(C=C(C)C(C)(C)C)=O)C2C)cc2cccc(C)n2n1 48040,c1(CC(N2C3(CNC(=O)CCC4CCC4)CCC3CC2)=O)cc(F)c(F)cc1F 48041,n1(CC(=O)NC2C(C)N(C(=O)C=CC3CC3)CC2)sc(=O)c2ccccc12 48042,c1(-n2c(C)nnn2)cc(C(=O)NCCCNC(=O)CSC2CC2)ccc1Cl 48043,N1(C(C2CC(C#N)(OC)C2)=O)CC(C(=O)N(CCC(F)(F)F)C)OC(C)C1 48044,C1(CC(C)C)CCN(C(C2CCN(C(=O)CCc3cn(C)cn3)C2)=O)C1 48045,C1(NC(C2(CCC=C)CN(C(c3cc[nH]c3)=O)C2)=O)CCn2cncc2C1 48046,c1(CC(=O)NC(C(=O)N(CC)Cc2ccncc2)C2CCOC2)cncnc1O 48047,C1(C(=O)NCCC(=O)NCC#C)COC2(C1)CN(C(c1cnc(OC)nc1)=O)C2 48048,c1(C(=O)NC2C(C)CCN(C(c3nc(C)oc3C)=O)C2)c(C)nc2sc(C)nn12 48049,N1(C(CC2N(C(C3=CCCCC3C)=O)CC(C)(C)C2)=O)CCCC2C(=O)NCC12 48050,c1(C(N2C(CC)C(O)CC2)C(=O)NC2(C)CC2)cc2c(s1)CCOC2 48051,C12(CCNCC1)C(=O)N2.N1(CC)CCC1(C)CCO 48052,C(=O)(C(F)C(C)CNC(c1ccc(O)cn1)=O)N(CC(C1CC1)OC)C 48053,C12(CNC(=O)C=CC(F)(F)F)CCC1CCN2C(=O)CCN1CCCC1 48054,C(=O)(CC(O)C(C)(C)C)N1CCC(NC(Cn2c(C)ccn2)=O)C1C 48055,N1(C(C2N(CC)CCC2)=O)CCC(C)(CNC(c2sncc2C)=O)C1 48056,C1(CCOC)(NC(=O)C2=C(Cl)CC2)CCN(c2ccnc(C)n2)CC1 48057,c1(OC)ccc(CN2CCC2(C)C(N2CCOC(c3ccccc3)C2)=O)cc1 48058,c1(C(N2C(CN(C(CC(C)C3CC3)=O)C3CC3)CCC2)=O)c(C2CC2)cnn1C 48059,C1(C(=O)NC2CC(NC(=O)COc3cccc(Cl)n3)C2)CCN(CCO)C(=O)C1 48060,C(CC(O)CC(=O)N(C)CCN(C(=O)C(C)(F)CC)C)SC 48061,[N-]=[N+]=Nc1ccnc(COC(C2CC(O)CN2C(=O)OCc2ccccc2)=O)c1 48062,c1(C(=O)NCCCC(CCC)NC(c2cc[nH]c2CC)=O)cnc2ncccn12 48063,Cc1nc2ccc(C(=O)NC(C3CCN(C(c4nccn4C)=O)C3)(C)C)cc2s1 48064,C(C)(CNC(c1ccn(C)c1)=O)(CC(C)C)NC(Cc1nc(C(C)OC)sc1)=O 48065,N1(C(C2CC(=C)CN2C(=O)Cc2cc(Br)ccc2Br)=O)CCC(O)C(C)(CO)C1 48066,c1(CC)nc(C)oc1C(N1CC2C(N(C(=O)C(CC)SC)C)C2C1)=O 48067,Cc1cc2c(C(N3CCC(CNC(=O)CSC(F)F)CC3)=O)cccc2[nH]1 48068,C1(C)(C(=O)NC2CCN(CCC)C2)CCCN(c2cc[nH]c(=N)n2)C1 48069,c1(N2CC(CNC(C(CC)N(C)C)=O)OCC2)cc(C)c([N+](=O)[O-])cn1 48070,n1(CCOCC)c(N2CCOC(C)C2)nnc1C1(OC)CC1 48071,Cc1nc(C(=O)NCC(C)(C)CN(C)C(C2CCSC(C)C2)=O)cn1C 48072,CC1(F)CN(C(c2cccc([N+](=O)[O-])c2)=O)CCN(C(c2cccc(=O)o2)=O)C1 48073,C1(CC=O)C(=O)N(C)C(C)(C(=O)NCCOC(F)F)C1CC 48074,Cc1ncc(N)cc1C(=O)NC1COCC1NC(=O)Cc1cc(C2CC2)nn1C 48075,Cc1cccc(Br)c1S(=O)(=O)NCCCc1ccc([N+](=O)[O-])cc1 48076,CN1C(C(=O)NCC2CC3(CC3)CN2C(=O)CC2(O)CCCC2)CCS1(=O)=O 48077,c1(NC(c2n(CCC)ncc2)=O)ccc(NC(=O)C(C2(O)CCCC2)F)cc1C 48078,Cc1ncnc(O)c1C(=O)NCC1CC(NC(c2cnc(Cl)s2)=O)C12CCC2 48079,C(CC(=O)NCCS(C)(=N)=O)(C(F)F)NC(Cc1cc(C)n(C)n1)=O 48080,C1(O)(CCNC(C2(CC=C)CCOC2)=O)CCN(C(=O)Cn2ncc(Cl)c2C)C1 48081,c1(C(C2CCOC2)OC)nc(-c2cccs2)nn1-c1ccnc(F)c1 48082,C(=O)(C(F)(F)CC(C)C)NC1(COC)CCN(C(=O)Cn2cc(Cl)cn2)C1 48083,C1(CN(C)C(C2CCN(c3ncccn3)C2)=O)CCCOC1 48084,C(CS(=O)(=O)CC(=O)NC(CCSC)C(=O)NC1CCC=CCCC1)OC 48085,N1(C(C2C(CC)C2)=O)CC(CNC(c2cccc(CC)c2N)=O)CC12CCC2 48086,c1(CN(C)C)cnc(O)cc1C(F)(F)F.C12CC(C1)NC2=O 48087,C(C(C)(C(=O)NC(C1CCN(C(=O)C=Cc2ccncn2)C1)(C)C)OC)OC 48088,N1(C(C2(C)C(C)OCC2)=O)CC(C2(NC(c3cnnn3C)=O)CC2)C1 48089,C1(C(N(CCC(=O)NC2CC2CN(C)C)CC)=O)CC=CCC1 48090,CCC1=NOC(C(=O)N(CC(C)NC(c2cccc(C(C)(F)F)n2)=O)CC)C1 48091,N1(C(C(C2CCOCC2)C)=O)CCC(C)(C(=O)Nc2cccc(C(F)F)c2)C1 48092,Cc1nc(CC(N2CCC(CO)(NC(C3CCC(=O)O3)=O)C2)=O)c(C)s1 48093,C1(OCC)CN(C(c2nccn2CC)=O)CC1OC.c1(O)cncc(CNC(C)=O)n1 48094,c1(CC(C)C)c[nH]c(C(=O)N(C)CCN(C(=O)CC2C=CCC2)C)c1 48095,c1(C(N(C2CCN(C(C3CC=CC3)=O)C2)CC)=O)cc(C(C)C)nc(O)c1 48096,O=C(C(O)C1=CCCCC1)NCC1CCN1C(=O)Cc1ccc(C(F)F)cc1 48097,CCCC(O)CC(=O)NCC(C1CCCC1)NC(=O)C(c1cccc(F)c1)C 48098,Cc1ncncc1C(N1CC(NC(C2OCCC2C)=O)C(C)C1)=O 48099,C(N=c1[nH]c(N2CC(CO)C3(CCC3)C2)nc2c1COC2)c1c(C)cncc1 48100,c1(C(=O)NC(CC=C)CNC(=O)CCC=C=C)c(C)[nH]c2ccc(OC)cc12 48101,c1(CC)c(C(N2CCC(C3CCCN3C(c3[nH]ncc3C#N)=O)C2)=O)cnn1C 48102,c1(C2(NC(C(C)c3ccco3)=O)CC2)ccc(C(=O)O)cc1 48103,CC1CCCN(CC(=O)NC2CCCCNCC2)C1CCO 48104,N1(C(C)C)C(=O)COCC1C(N1CCC(CNC(=O)C2=CCOCC2)C(C)C1)=O 48105,C(CCCCC(=O)N1CCN(C(C)C)CC1)NC(Cc1cccc(C)c1)=O 48106,N1(C(CN(CCC)C)=O)CC(C)C(NC(c2nccc3occc23)=O)C(C)C1 48107,N1(C(C(CC)C2CCOCC2)=O)CCN(C(=O)CCCCCSC)CC2(CC2)C1 48108,N1(C(C#C)=O)CCc2c(C(=O)Nc3ccc4nc(C(C)C)[nH]c4c3)n[nH]c2C1 48109,Cc1cc(F)sc1C(=O)NCc1cccc(CN(C)C(c2nnn(C)c2N)=O)c1 48110,C1(CC(N2CC(CCNC(=O)CCn3cccc3)OCC2)=O)CCCCCCC1 48111,N#Cc1cn(CC(=O)NC2CN(C(C3NC(=O)C4CC34)=O)C2)c(=O)nc1O 48112,c1(C(=O)NC(CN(C(C)C)C)C)ccccc1NC(=O)C(C)NC(N)=O 48113,C1(CCC)(C(=O)O)CCN(C(c2nnccc2C)c2nnc(C)o2)CC1 48114,C1(NC(CC(c2ccc(F)cc2)C)=O)CCCN(C(=O)CC2COC(=O)N2)CC1 48115,c1(C(N2CCC(C(=O)OC)(OC)C2)=O)ccc(Cl)nc1Cl 48116,C(=O)(CCCCCN(C)C)NC1CC(F)(CNC(c2ccnc(CC(C)C)n2)=O)C1 48117,Fc1cccc2c1OCC2Nc1cc(NC2CCC=C2Br)ncn1 48118,c1(C(N(CCC(C)NC(C(C(C)C)O)=O)C)=O)ccc(F)c(C#N)c1 48119,c1(C(N(C(C)CNC(=O)CC2CCC3CC23)C)=O)ncc(C2CC2)cc1F 48120,Cc1ccc(C(=O)NC2CC(NC(C3(c4ncco4)CC3)=O)C23CCC3)nc1O 48121,c1(C(=O)NC2COCCN(C(C3(C(F)(F)F)CC3)=O)C2)cccc2c1OCCC2 48122,C1(CNC(C2CC(CC)OCC2)=O)CC2CCC1N2C(C1CNC(=O)N1)=O 48123,Cn1cnc2c(NC3(C4CN(C(=O)CC5CCC(C)(O)CC5)C4)CC3)ncnc12 48124,c1(COC)ncsc1C(N1CCCC1CNC(=O)CC1CC(OC(C)(C)C)C1)=O 48125,C1(OC)CCN(C(c2c(C(=O)OCC)[nH]cc2C)=O)C(c2ccccc2)C1 48126,CC1CC(C(=O)NC2CCCCC2NC(c2cn(CCC3CC3)nn2)=O)CN1C 48127,C(=O)(C(O)C(F)(F)F)NCCC(CNC(c1n(CC)ncc1)=O)O 48128,N1(C(CC2C(NC(C(C(C)(F)F)F)=O)CCCC2)=O)CCCC12CCOCC2 48129,c12ccc(cc1)CN(CC)CC(C)NC(=O)CC2.C1(C)(C(=O)OC)CC1(F)F 48130,c1(CCC)ccc(C(c2nnnn2C2CC2)NCC2CCCOCC2)cc1 48131,C1(C(=O)NCCCC(C)NC(C(C2CCCCC2)OC)=O)CN2CCCN1CC2 48132,C1(CC)(CC)C(OC)CC1Nc1cccc(Oc2c(NC)cccc2)c1 48133,c1(C(=O)NC(C(CO)NC(C(CSC)C)=O)C)ccc(Br)c(SC)c1 48134,C1(C(=O)NCC(CC(F)(F)F)NC(C#CC(C)(C)O)=O)CCn2cncc2C1 48135,N#Cc1ccnc(N2CC(OCCNC(C3COC4(CCC4)C3)=O)C2)c1[N+](=O)[O-] 48136,c1(C(C)NC(C2(C(C)(C)C)CCNC2)=O)ccc(F)cc1 48137,Cc1ncc2cc(C(N3CC4CC(NC(=O)CCc5csnn5)C3C4)=O)ccn12 48138,C1(C2CC2)(CNC(C(N2CCC(C)CC2)=O)=O)CCN(C(C2(C)COC2)=O)C1 48139,C1(CNC(C2C(CC)CCC2)=O)CN(C(=O)C=Cc2cnc(C)s2)CCCO1 48140,c1(CC(=O)NCC(CC)(C)NC(=O)CCC=CC(C)C)ccc(OC)cc1C 48141,N1(C(C2CCC(=O)NC2)=O)CCOC2CN(C(c3cnc4ccccn34)=O)CC12 48142,c1(C(=O)NCC2OCC(CNC(CCC)=O)C2)cc2cccc(Br)c2cn1 48143,N1(C(c2ccno2)=O)CC2C3CCC(C2C1)N(c1nc(Cl)nc2[nH]ccc12)C3 48144,c1(NC(c2n[nH]cc2I)=O)ccc2c(c1)CN(C(=O)Cc1cncnc1)C2 48145,C1(C)(C(=O)NC2CC(CCNC(C3(OC)CCC(C)C3)=O)C2)C(C)(C)C1(C)C 48146,Cc1cccc(CC(=O)N(C2CCC(NC(=O)Cc3nccn3C)C2)C)c1 48147,C(=O)(C(F)CCC(C)C)N1CCN(C(C2N(CC)CCOC2)=O)CC1C 48148,C(=O)(C(CC(C)C)C(C)C)NC1CC2(C(C(N(CCOCC)C)=O)C2)C1 48149,C1(CC(=O)NC(CNC(C(c2cnn(C)c2)C)=O)(C)C2CC2)CNC(=O)C1 48150,c1(C(=O)NC2CCC(n3cc(COC)nn3)CC2)c(F)ccc(SC)c1F 48151,N1(C(CCC(=C)C)=O)CCC(NC(=O)CN2CCC(C(N)=O)CC2)CC1C1CC1 48152,c1(C2CCCN(C(=O)NCC3CC3)C2)cccc(OCCc2ccn(CC)n2)c1 48153,C1(CSC)CCCN1C(=O)C(Cc1cc[nH]n1)NC(c1ccoc1)=O 48154,Cc1nc(S)nc(C)c1CCC(=O)NCCN(C(C1CCN(C)C1=O)=O)CC1CC1 48155,C1(C(CC)C)CCN(C(=O)COC2(C)CN(C(=O)C(O)CC)C2)CC1 48156,c1(NCc2cnc(CC)s2)ccc2c(c1)CN(C(c1cnc(C)c(C)c1)=O)C2 48157,N1(C(CNC(CC)=O)=O)CC2CC(NC(c3ccn(C4CCCC4)n3)=O)C(C2)C1 48158,N1(C(C)=O)CS(=O)(=O)CC1C(=O)NCC1CN(C(=O)Cc2cn3ccsc3n2)C1 48159,c1(N2CCC(CCNC(C(CNS(C)(=O)=O)N(C)C)=O)C2)ccncc1[N+](=O)[O-] 48160,N1(C(C(F)OC)=O)CCC2CCN(C(C3CN4CCN3CC4)=O)CC12 48161,c1(CC)nn(C)c(C(=O)NCC2CN(C(c3ccc(SC)o3)=O)CCC2C)c1Cl 48162,C1(C(=O)NCC(CN(C(C(C=C)(C)C)=O)C)C)CC(C2CCOCC2)=NO1 48163,c1(NC(C2(O)CCOC2)=O)cc(=NCC23CC(C(=O)OC)(CO2)C3)[nH]cn1 48164,C1(CNC(c2cnnc(O)c2)=O)CC2CCCCC2N1C(c1ncc(F)cn1)=O 48165,c1(CNC(=O)C(=O)Nc2c(C(=O)OC)scc2C(=O)OC)ccc(F)c(OC)c1 48166,C(CCCCCC(=O)Nc1cncc(C#N)c1)NC(C1(OCC)CCOC1)=O 48167,CCC(CC)C(C)C(=O)NCC1(C)CCCN(C(C2(C3CCC3)CCC2)=O)C1 48168,C#CC1(C(N(C)C[Si](C)(C)C)=O)CCN(C(=O)CCC2CCCO2)C1 48169,N1(C(C2(CC)CCCCO2)=O)CC(NC(=O)CCCC2CCCC2)CC(F)C1 48170,N1(C(C2CC3CC3C2)=O)CC=C(CC(=O)N2CCC3CC23)CC1 48171,c1(C(C=CC)O)nnc(N2CCN(C(c3cccs3)=O)CC2)n1CC(C)C 48172,c1(C(=O)NCC2N(CC(=O)NC(N)=O)CCC2)ccn2ccnc2c1 48173,C1(C(C(=O)N(C(C=C)C)C)C)CCCN(C(=O)C=CC(=O)NC(C)C)C1 48174,c1(OC)ccc2c(c1)OC(CN1CC(COC)OC(C)(C)C1)O2 48175,c1(OC)cc(N)ccc1C(=O)NC1C2CN(C(C3(C)C=CCCC3)=O)CC12 48176,C1(NC(Cc2nn(C)c(C(F)(F)F)c2)=O)(CO)CCC(C(=O)O)CC1 48177,c1(C(N2CC(NC(C3C(C)C3C)=O)C3(C2)CC3)=O)cc2cc(F)ccc2[nH]c1=O 48178,c1(C(=O)NC2CN(c3ccnc(C4CCCC4)n3)C2)cc(F)c(OCF)c(F)c1 48179,CCCCC(O)C(C)C(=O)NCCC1CCCCN1C(c1cccn1C1CC1)=O 48180,Cc1cc(CC(=O)NC(C)C(C)(C)NC(=O)Cc2csc(Cl)c2)n[nH]1 48181,N1(C(c2cccc(CC)n2)=O)CCC2C(CCCN2C(=O)Cc2cn[nH]c2)C1 48182,N1(C(c2ccn(CCNC(CCN(CCC)C)=O)c2)=O)CCC12CCC(C)CC2 48183,C1(F)(CNC(c2n(CC)ncc2Cl)=O)CCN(C(C2CC3CC3CC2C)=O)CC1 48184,c1(C(C)C)nc(=N)[nH]c(=NCCCCNC(=O)CN(C2CCSC2)C)[nH]1 48185,N1(C(C(C)n2ccnn2)=O)CC2(CCC(CNC(=O)CCF)O2)C1 48186,C(=O)(C1CCCc2ncnn21)OCC.C12CCN(C(=O)C(=O)N(C)C)C1CN2 48187,C1(CNC(c2on(C)c(=O)c2)=O)(CO)CCN(C(=O)Cc2cnns2)CC1 48188,C(=O)(C1=NOC(C)C1C)N1CC(N(C(C(C)C)=O)C)C(O)C1 48189,c1(OCC)cc(NC(C2CCCN2C(=O)CC2CC2(C)C)=O)cc(Cl)n1 48190,C1(C(=O)NCC(C)(C)NC(C2(F)C3CCCCC23)=O)CC2(C1)CC21CCC1 48191,CC(CN(C)C)C(=O)N1CC(O)(C(C)(C)CNC(=O)C=CCN2CCCC2)C1 48192,C1(C(=O)NC(C)CN(C)C(c2cnncc2O)=O)CN(C)CCN(C)C1 48193,CC1=C(C(=O)NCC2CCC(NC(C3OC(C)CC3C)=O)C2)CCCO1 48194,Cc1nc(Cl)nc(N2CCCC(C(C)NC(=O)C=Cc3ccncc3)C2)c1F 48195,CCS(=O)(=O)CC(CO)NC(=O)NCCCc1scnc1C 48196,C1(CC(=O)NCCC2CCN(C(=O)CN3CCCC3)C2)CCC2(CC1)OCCO2 48197,Cn1cncc1C=CC(=O)NCCN(C(C1CC1c1cccnc1)=O)C1CC1 48198,C(=O)(C1CCS(=O)(=O)c2ccccc21)NCC(CNC(Cc1ccc(C)s1)=O)C 48199,Cc1ncccc1C(=O)NCc1cc(C(=O)NOCCCN(C)C)co1 48200,N1(C(c2ccc(NC)cc2)=O)C(=O)CCC(N(CC(C)C)C)C1=O 48201,c1(C(=O)NC2C(NC(C(C)(C)n3ccnn3)=O)C2)cc(F)c(Cl)cc1Cl 48202,N1(C(CC(C)c2cccnc2)=O)CC2CC2(CNC(=O)CN(C)C(N)=O)C1 48203,CCCCC(CC)CC(=O)NCC1CCC2CN(C(C3CSC3)=O)CCC2C1 48204,C1(O)(C(C)NC(=O)COC2CCCC2)CN(C(=O)CCc2nccs2)C1 48205,CC(C)C(O)C(=O)N(C(C)CCNC(=O)CCc1cnco1)C 48206,C(C)(CCC(=O)N(CCCNC(=O)Cn1nc(C)cc1C)C1CC1)SC 48207,C(C(CC(C)C)C(=O)N1CCN(C(c2cc(CC)c(CC)o2)=O)CC1CF)CC 48208,C1(O)(CNC(c2nc(CNC(CS(=O)(=O)NC)=O)oc2)=O)CC2CCC1O2 48209,C12(NC(=O)CNC(c3cscn3)=O)CCCN(c3ccn4nccc4n3)CC1C2 48210,Cc1cccc(CNC2CCN(C(c3cc(C(=O)O)ccc3F)=O)C2)c1C 48211,n1(CC(=O)NC2C(SC)CN(C(C3(CO)CCCC3)=O)C2)nc(C)c(Cl)c1C 48212,CC1CC(C(N2CCCCC2C2CCOC2)C(=O)NC2CCOCC2)CC(C)C1 48213,Cc1nc(O)c(C(=O)NCC23CC2CN(C(C2(CO)CC2)=O)C3)c(C)c1[N+](=O)[O-] 48214,N1(C(CNS(NC)(=O)=O)=O)CCCC2CCN(C(c3nocc3C)=O)CC12 48215,c1(C(=O)NC2CCN(C(c3cscc3C3CC3)=O)C2)ccc(SC(F)(F)F)nc1 48216,c1(C(=O)Nc2scc(COC)n2)cc(Br)cnc1C(F)(F)F 48217,C1(NC(CC=CC)CO)CCOC2(CCOCC2)C1 48218,N1(C(CCC(=C)C)=O)CC(CNC(=O)CCCC)CC12CCOCC2 48219,Oc1nc2ccccc2cc1NCCN1CCCC1 48220,N1(C(C(N2CC(C)CC(C)C2)=O)=O)CCn2c(cnc2C(N2CCOCC2)=O)C1 48221,N1(CC)C(=O)CCC1C(=O)NC(C)(C)CNC(=O)C=C1CCSCC1 48222,CCC1(C(=O)NCC(CC)NC(=O)Cc2ccsc2C)CCCc2ccccc21 48223,Cc1nn(CC(=O)NCC2(O)CCN(C(=O)CC3(C)CCC3)C2)c2ncccc12 48224,C1(C(=O)NC2C(CNC(c3cnoc3-c3ccoc3)=O)CC2)CC2(C1)CC2(F)F 48225,c1(C(=O)NCC(CNC(C(C(C)(C)C)SC)=O)F)cc(Cl)c2n[nH]cc2c1 48226,Cc1cc(Cl)cc(C(N2CCOC(CN(C)C(c3ccc(F)s3)=O)C2)=O)c1N 48227,CC1CCC1C(=O)NC(C(=O)NCC=CCl)C1CCCC1 48228,c1(C(N2CC(F)(CNC(C(C(C)C)NC(C)=O)=O)C2)=O)ccc(Br)c(C)n1 48229,CCCCCC(C)(C)C(=O)NC1CCOC(CNC(C2CCC2COC)=O)C1 48230,c1(CC)cc(Br)cc(C(=O)NCC2CCN(C(=O)CCC(F)F)C2)c1N 48231,c1(OC)ccc(F)cc1CNC(=O)NCC1CC2(CCC2)CN1 48232,Cc1ccc(CC(=O)NC(C2CN(C(C3CC3(C)C)=O)C2)C)cc1Cl 48233,C1(C(=O)OC)CCCC1NC(=O)NCCNC(c1sncc1C)=O 48234,Cc1cccnc1C(=O)NC(C)(CNC(c1cc(CC(C)C)nn1C)=O)C1CC1 48235,CC1(C(=O)Nc2cc(O)ncn2)CCN(Cc2cccc(F)n2)CC1 48236,c1(NC(N2CCOCC2)=O)ccc(S(=O)(=O)NC2CCCn3ccnc32)cc1Br 48237,c1(C(=O)NC2CC3CN(C(C(CC)(F)F)=O)C(C2)C3)cc(S(=O)(=O)NC)oc1C 48238,C1(NC(CC2(CC)CCC2)=O)CC(C)(NC(=O)CNC(=O)NC2CCCCC2)C1 48239,N1(C(C(C)(C)C)=O)CCCC(F)(CNC(c2cccc(C3CC3)c2Cl)=O)C1 48240,c1(CCC(=O)NCCCCNC(=O)CC2CCC2C2CC2)c(Cl)cccc1Cl 48241,c1(C(=O)NC(C2CCCN(C(C3=C(C)OCC3)=O)C2)C)cc2c([nH]1)CCOC2 48242,N1(c2ccc(C#C)cc2)CCC2C(CCN2S(=O)(=O)CCCCCCC)C1 48243,C(=O)(CS(=O)(=O)Cc1cccs1)NCCOC1CCN(C(C(CC=C)C)=O)C1 48244,C1(C=C)(C(N(C(C(=O)N(C(CCSC)C)C)C)C2CC2)=O)CCCCC1 48245,c1(CN(C(C2CC(=O)C2)=O)C2CC2)c(F)cccc1F 48246,N1(C(=O)CN2CC3CC3C2)CC2CCCN(C(C3CCC(F)C3)=O)C2C1 48247,CN1CC(C(=O)NCC2CC2CNC(C2(C(F)F)CC(F)(F)C2)=O)NC1=O 48248,C(C(=O)NNc1ccc(S(=O)(=O)N(C)C)cc1)(C(C)(C)C)n1cc(COCC)nn1 48249,C12(NC(C3CC(C)OCC3)=O)CCC(CC1)N(C(=O)CN1CCOCC1)C2 48250,N1(C(C2C(C)CCC2)=O)CC2CCC1CC2NC(c1cnn(C)n1)=O 48251,c1(C(=O)NC2CN(C(c3cnsn3)=O)C3(CCC3)C2)cc2ccnc(Cl)c2s1 48252,Cc1nc2cc(C(=O)NC3(CNC(C4CCN(CC(F)(F)F)C4)=O)CC3)[nH]c2s1 48253,c1(C(=O)NCCCCN(C(c2cc(C(C)=O)on2)=O)C)cc(C)c(Cl)cn1 48254,c1(N2CCC(F)(CNC(CC(C)(C)OC)=O)CC2)ncc(C#N)cc1F 48255,N1(C(C(C)CC2CCCC2)=O)CCCCC1CCNC(=O)C1=CCOC1 48256,n1(CCO)ncc(-c2noc(C3(CO)CC3Cc3ccccc3)n2)c1N 48257,CCC(CNC1(c2nnnn2C2CCCC2)CCC(C2OCCO2)C1)(CC)SC 48258,N1(C(C2N(CC#C)CCC2)=O)CCC(NC(C2C(C)OC(C)C2C)=O)C(F)C1 48259,CP(C)(=O)c1ccc(C(N2CCC(CNC(=O)C3=CCCCC3)C2)=O)cc1 48260,c1(C(=O)NCC2(N(C)C(C3CSC3)=O)CC2)cnc(C2CC2)s1 48261,c1(OC)ccc(F)c(C(=O)OCCO)c1.c12cnc(nc1)N1CC(C1)C(=O)N2 48262,C1(C(=O)NCCN(C(CCN(CC)CC)=O)CCC(C)C)CCCCC(F)(F)C1 48263,c1(OCC)ccccc1COCC(O)CN(C)Cc1cccnc1-n1cccn1 48264,N1(C(=O)NCC2(CO)CC2)CCCC2(NC(=O)CCc3cccc(F)c3)CC2C1 48265,c1(C(N(C2CN(C(c3cnns3)=O)CCC2O)C)=O)ccc2cccnn12 48266,CC1N(C(C2CC23CC(NC(C2(N(C)C)CCC2)=O)C3)=O)CCCC1(C)C 48267,CC(CCNC(=O)CNS(N)(=O)=O)CCNC(=O)C(C)(C)C1CCOCC1 48268,C1(C(=O)NC2CC2(F)F)CC12CCN(C(=O)Cc1cccc(Br)c1)CC2 48269,CC(CC(F)(F)F)C(=O)N1CC(CCNC(c2cc(=O)cc(Cl)[nH]2)=O)C1 48270,C1(C(=O)NCC(C)(C)OC)CN(C(C2(C#N)CCCC2)=O)CC(C)(C)C1 48271,C1(C(N2CCCCCC2CNC(=O)C(F)(F)c2cn[nH]c2)=O)CCCCC1(F)F 48272,c1(C(=O)NCCN(CC(C)O)C(c2c(C)n(C)nc2)=O)cccn2c(C)cnc12 48273,CC1(NC(=O)Cc2csc(C(F)(F)F)n2)CN(C(=O)CC2CC3(CC3)C2)C1 48274,N1(C(C2C(CC(C)C)C2)=O)CC2CN(C(=O)Cn3ccccc3=O)CCC12 48275,C1(CNC(C(CC)(CC)CO)=O)CCN(C(C2CC2C(=O)OC)=O)CCC1(F)F 48276,CCCCCCC(C)C(=O)N1CC2CN(C(c3cc(Cl)cc(OC)c3N)=O)C2C1 48277,Cc1nc[nH]c(=NCC(C2CC2)NC(c2c(C)oc(C)c2C)=O)c1C#N 48278,c1(CC(N2CC(NC(CC(C)(C)O)=O)C(C)(C)CC2)=O)ccc2cccnc2c1 48279,C12(CNC(C3CN(C4CCC4)C3)=O)CCCC1N(C(=O)CC1OCCO1)CCC2 48280,N1(C(C(COC)COC)=O)CCN(C)C(C(=O)NCCCN(C)C(C)=O)C1 48281,CCCC(C)(C)C(=O)NCCC1(C)CCN(C(c2ccc(OC)cc2)=O)C1 48282,N1(C(C(C#C)(C)C)=O)CC(NC(c2ccccc2C2CCOC2)=O)C(N=[N+]=[N-])C1 48283,CCCC(C)CCNC(=O)C(C1CCN(C(c2ccccc2O)=O)CC1)C 48284,C1(N(C)C)CCCC(C(=O)OC(C)(C)C)C1.N12CCC(C1)N(C)C(=O)CC2 48285,N1(C(C(CNC(C(C=C=C)C)=O)C)=O)CCN(C)C(C)C1 48286,c1(C(N2CC3C(CNC(=O)C(F)(F)C4CC4)C3C2)=O)cnc2cccnc2c1 48287,Cc1cc(C(N2CCCC2C2CCCCCC2)=O)ncc1-c1nn[nH]n1 48288,C(=O)(CC(C1CC1)C1CC1)NCC1CCCCO1.C12CC1C(=O)NC2C 48289,C1(C(N(CCC#C)C)=O)CCC(C2CC2)N1C(c1cc(Cl)cs1)=O 48290,N1(C(c2cn(CC)nn2)C(=O)NCC2CCCO2)CC2(CO)CC2(C(F)(F)F)C1 48291,C1(C(N(C(C(=O)NC2CCN(CCC)C2)CC)C)=O)CC12CCCCC2 48292,N1(C(C=C(CCC)C)=O)CCC(C2CC2)C1CNC(=O)Cc1c(C)cccc1C 48293,N1(C(Cc2ccc(CC)c(F)c2)=O)CC(C2CN(C(C34CC(OC)C3C4)=O)C2)C1 48294,c1(-c2c(C(N3CCOC4CC34)=O)n[nH]c2)cccnc1-c1ccccc1 48295,C(=O)(C(C)CC(C)(C)C)N1CC(F)CC(NC(c2ccc(OC)cc2C)=O)C1 48296,C#CCC(CC(=O)NC(CC)C(C)(C)C)NC(C1CS(=O)C1)=O 48297,c1(CNC(C=C2CCC(C)CC2)=O)nc2c(s1)CCN(C(=O)Cc1cncs1)C2 48298,C(CC1CCC1)(C(=O)NC(C)(C)C)N(CCCF)C 48299,N1(CC(=O)N=c2cco[nH]2)CC2CCN(C(c3nc[nH]c3C(F)(F)F)=O)CCC2C1 48300,C12(C(=O)NCC(CNC(c3ccn4ncnc4c3)=O)O)CCC(O)(CC1)CC2 48301,C1(CCC(=O)NC(C#C)C2CC2)CCCN(C(=O)CC(O)c2ccccc2)C1 48302,C1(CNC(C(C2CC2)OC)=O)C(C)CCCN1C(=O)C(=Cc1ccc(C)cc1)C 48303,C1(NC(c2c(C)nc(C3CC3)[nH]2)=O)CC2CC(NC(=O)C(O)CC(C)C)CC2C1 48304,C1(NC(c2nn(C)c(C(N)=O)c2)=O)CC2CCC(C1)N2C(=O)C(O)C1CCC1 48305,C1(C(=O)NCC2(F)CN(C(C(c3ccccc3)=O)=O)C2)CCC2C(CC1)C2(F)F 48306,N1(C(c2cc(C)ncn2)=O)CCC(C2CCN(C(=O)Cc3ccccc3C)C2)C1 48307,C(=O)(CCCC(C)(C)C#N)NCC1C(C(=O)NCCc2cnc(C)[nH]2)C1 48308,C1(C(=O)NCC(C(=O)OCC)C)N(C(c2cncc(C)n2)=O)CC12CCCC2 48309,Cc1n[nH]c(C)c1SCC(N1CCCC(CN(C(=O)C(C)CC2CCC2)C)C1)=O 48310,C1(CNC(c2c(C)nn(C)c2)=O)CC(C(=O)NC2CCC(C)(C)C2)=NO1 48311,CCC(C)(COC)C(=O)NCC(C1CC1)N(C(=O)Cn1cccc(C)c1=O)C 48312,c1(CC(=O)NC2CCC(NC(Cc3c(Cl)cn(C)n3)=O)C2)cc(F)ccc1Cl 48313,S(=O)(=O)(c1cc(Br)cc2c1OCC2)NC1C(C(=O)NCc2ccc(C)cc2)C1 48314,Cc1c(C(=O)NC(CNC(C2CC3(CCC3)C2)=O)C(C)C(C)C)cc(O)cc1N 48315,CC(C(=O)N1CCCN1C(=O)Oc1ccccc1C(F)(F)F)C1CCCNC1 48316,C(=O)(C1CCCc2c[nH]nc21)N1CC(CNC(CC(C=C)C)=O)C1 48317,C12(CNC(C3C(OC)CCC3)=O)CCC1CN(C(=O)Cc1cccc(F)c1F)C2 48318,c1(N(CC(=O)NCCC)C)nc(=NC)nc(N2CC(N(C)C)C(C)(C)C2)[nH]1 48319,C12(C(=O)NCCCOC(=N)O)CC(CN1C(=O)CC1CCOC1)C2 48320,O=C(C#CC1CCOCC1)NCC1CN(C(c2ccc(C(F)F)o2)=O)CC1(F)F 48321,c1(CC)cc(F)c(C(=O)NC2(C)CN(C(=O)C(CC)n3cncn3)C2)cc1F 48322,C1(CC)CN(C(=O)Cc2cc(C)n(C)n2)CCC1CNC(=O)C(CC)(CO)OC 48323,c1(NC(c2n(C)ncc2)C2CC2)ccc(S(=O)(=O)N2CCC2C(N)=O)c(Br)c1 48324,CC(CS(C)(=O)=O)C(=O)NCCN(C(=O)C=Cc1cnccn1)CC1CC1 48325,S(=O)(=O)(c1cc(-c2ccccc2)no1)C1(N(C)C2CC2)CCC1 48326,C#Cc1cccc(C(=O)NC2CCN(C(C3CCCCN3N=O)=O)C2C)c1C 48327,c1(C(=O)NC(C(C)NC(c2c(C)nns2)=O)(C)C)cc(C2CCCCC2)n(C)n1 48328,C(=O)(C(C)(C)C(C)NC(=O)CCc1cn[nH]c1)NC(c1nccc(O)n1)C 48329,S(=O)(=O)(c1ccccc1C(=O)NC1CC1)Nc1c(C(=O)OCC)n(C)cn1 48330,CC(C)CC(O)C(=O)N1CCN(C(=O)Cn2ccnn2)CC1c1cccc(F)c1 48331,CC(C)CC(C)(O)CNC(c1cc(CNC(=O)C=CC2CCOC2)ccn1)=O 48332,c1(C(N2C(C(N(C)Cc3scc(C)n3)=O)C(C)CC2)=O)ncn2c1CCC2 48333,CCCC(CNC(c1cc(C)[nH]c1C)=O)C(=O)N1CC(C)(CO)C1 48334,C1(CNC(CSCC#C)=O)C(C2CC2)CCN1C(c1cnc(-c2ccsc2)s1)=O 48335,C1(C(N(CCNC(CCOCC)=O)C(C)C)=O)CCC(N2CCOCC2)CC1 48336,C=CCCCCCCCC(=O)N1CC2(CCCC(CNC(C3(O)CCC3)=O)O2)C1 48337,Cc1cc(Br)cnc1C(=O)NCC1CN(C(c2ccc(Cl)o2)=O)CC1C 48338,C(=O)(C1=NN2CCCN=C2N1)NC1C(NC(Cc2cc(C)sc2)=O)CCCC1 48339,c1(NC(C)=O)nc(C(=O)NCC(C)NC(C2CC23CC3)=O)cs1 48340,c1(C(=O)NC(CNC(c2cc(CC)c(CC)o2)=O)C(C)C)c(F)ccc(C)c1F 48341,N1(C(C2(CC(C)C)CCC2)=O)CC(NC(=O)Cc2coc(C(F)F)n2)C(C)C1 48342,C1(C)(C(=O)NCC(C)NC(c2cnn(-c3ccccn3)c2)=O)CC=CCO1 48343,N1(C(c2c(CCC)nco2)=O)CCC(N(C)C(C2(N3CCCC3)CCC2)=O)CC1 48344,c1(C(N(C2CCN(C(c3ccc(CC)s3)=O)C2)CC)=O)c(OC)nsc1OC 48345,C1(OC(CCCOCC(C)C)=O)CCCC(C(C)(C)C)CC1 48346,C(C(=O)NCCC1CN(C(c2cnccc2Br)=O)C1)(C(C)(C)C)NC(C)=O 48347,N1(C(C(C)(CO)NC(C)=O)=O)CC(NC(c2ccn(CC(C)C)n2)=O)C2(CCC2)C1 48348,C(CO)(C(C)NC(=O)C(n1nnnc1C(C)(C)C)C)NC(C1CC(=C)C1)=O 48349,C(C(C)C(C)C(=O)NCCOCCN(C)C(c1cc(C)nn1C)=O)OC 48350,C1(COCC)CN(C(C2CCN2C(C2CCCO2)=O)=O)CCO1 48351,C1(Cl)(C(=O)NCCN(C(c2nocc2C2CC2)=O)CC)CC12CCC2 48352,N1(C(c2cccc(CC)c2N)=O)CC2CCCC(C1)N2C(C1COCCC1C)=O 48353,C1(C(=O)NCCCOCC(C)C)CN(C(=O)C(C)S(C)(=O)=O)CC1(C)C 48354,C=CCC(CC)C(=O)NCC=CCNC(C1CCCN1Cc1ccc(C)cc1)=O 48355,c1(C(=O)OCCC(CCC)C)ccc(C(C)(C)C)c(F)c1 48356,c1(-c2cn(CCNC(C34CC(CO3)C4)C)nn2)ccc(Cl)cc1OC(F)(F)F 48357,c1(NC(CC)CC(F)(F)F)ncccc1S(=O)(=O)NC(c1nncs1)C 48358,Cc1nccc2c(=O)c(C(=O)NC3CCC4(CNC4)OC3)c[nH]c12 48359,c1(CNC(=O)CCNC(=O)CCCn2cncn2)cccc2cncn12 48360,c12nc(C)c(o1)C(=O)NC2.C(CCCCC1CC1)NC(COCC)=O 48361,C(N=c1[nH]c(=NC(C)CC(C)(C)N(C)C)c2ncccc2[nH]1)c1sc(C)c(Br)n1 48362,C1(CC(=O)NC2CCN(CCC)C2)CN(C(=O)CC2CCCC2)CCO1 48363,Cc1cn2c(n1)CCC(C(=O)NC1CCC1NC(c1ccccc1[N+](=O)[O-])=O)C2 48364,C(=O)(C(C)(C)CC(=O)OCC)N1CCC(N(C(C(CC(=C)C)C)=O)CCC)C1 48365,C(CCCC(=O)NC1CCOCC1C(=O)N(CC1=CCCOC1)C)(OC)OC 48366,c1(C(N(CCNC(=O)CCCn2ccnc2)CC)=O)c(F)ccc2cnn(C)c12 48367,C(C(=O)NC(C)CN(C)C(c1nc(C)nn1C)=O)(C(C)(C)C)NC(=O)OC 48368,Cc1csc2c(C(N3CC4CC(NC(=O)Cn5cnnn5)CC3C4)=O)ncnc12 48369,C(=O)(C(O)CCC(F)(F)F)N1C(C(C)C)C(NC(C2CCSC2)=O)CC1 48370,C1(C(=O)NC2CC(CCNC(C3CCC(OC)CC3)=O)C2)CCc2nncn2C1 48371,c1(C(N2CCC(N(C(=O)CC(C)F)CC)CC2)=O)ccc(-n2cnnn2)c(C)c1 48372,C1(C(=O)NCCC2CN(C(C3(C)CCC3)=O)C2)CC12CCCCC2 48373,c1(OCC(=O)NC2CCC(F)(CNC(C(C)SC)=O)C2)cccc(Cl)c1Cl 48374,C1(C(N2CC(C(C(=O)N(CCCN=[N+]=[N-])C)OC)C2)=O)CCCC(=O)C1 48375,N1(CC(COCC(C)C)O)CCC(N(C)C(c2cnoc2)=O)CC1 48376,C(=O)(C1=CC2C=CC(C1)C2)N1CC(CC(=O)NC(C)C2CC2)OCC1 48377,C(C1CCCC1)=CC(=O)N(C1(CC(=O)NCC(CO)C2CCC2)CC1)C 48378,N1(C(C(C)NC(CC)(C)C)=O)CC(C)C(NC(C2C3CC4C(C3)C24)=O)C(C)C1 48379,Cc1ccc(=O)n(CC(=O)NCC2(O)CN(C(C3CCN(C)S3(=O)=O)=O)C2)n1 48380,c1(CC(=O)OC(C=C)Cc2nccn2C)c(C)cc(C)cc1C 48381,c1(N(CC=C)C)ncccc1S(=O)(=O)NC(c1ccccc1F)C.C1CO1 48382,CC1(CNC(C2CCCC3(CC3)C2)=O)CN(C(c2cn3ccnc3s2)=O)CCO1 48383,C1(NCCOC)C2CCCN(CC(=O)N(C)CCN3CCNC3=O)C2C1(C)C 48384,c1(C(Cc2ccccc2)NC(C(=O)N(CC(C)OC)C)=O)ccc(Br)cc1 48385,C12(NC(c3n[nH]c4c3COC4)=O)COC(C1)C(NC(c1cc(F)c[nH]1)=O)C2 48386,c1(CC(N2CC(CCCC)N(C(=O)COCC)CC2)=O)ccc2c(c1)CCN2C 48387,N1(C(CC(CCC)O)=O)CC2CCC(C1)C2NC(c1cc(C)on1)=O 48388,c1(NC(c2c(C)nns2)=O)cnc(F)cc1C(=O)Nc1cccc(CCO)c1 48389,C1(NC(C2CCCC(O)C2)=O)CN(C(c2ccsc2C(F)(F)F)=O)CCC1CO 48390,Cc1ccc(F)cc1N(C)C(C1CCCN(C(c2ccn(C(C)C)n2)=O)C1)=O 48391,N1(C(c2cc(CC)sn2)=O)CCCC(C(=O)NCC2CCN2C(C)(C)C)C1C 48392,C(=O)(CS(=O)(=O)Cc1cccs1)NC(CNC(C(C)=C1CCC1)=O)(C)C(C)C 48393,C1(NC(C(C)OCCCCCC)=O)CN(C(=O)C(F)OC)CCC1(C)C 48394,CCC(C)(CNC(C1CCC(CNC(=O)C2=C(Cl)CC2)C1)=O)C(N)=O 48395,c1(NC2CCC3C(C)(C)C2C3)nc2c(c(=NCCC(O)C3CC3)[nH]1)CCCCCC2 48396,C1(NC(C(=CC(F)(F)F)C)=O)CCN(C(C2CC(=O)OC2(C)C)=O)C12CCC2 48397,c1(C(=O)NCCC2N(C(C3(OC(C)=O)CC3)=O)CCC2)cnc2onc(C)c2c1 48398,c1(OC)nccc(C(=O)NCC2(C(=O)Nc3c(C)nn(C)c3C)CC2)c1F 48399,C(=O)(C(C)CS(C)(=O)=O)N1C(COC)CN(C(=O)CCc2nncs2)CC1 48400,c1(CN(CCCC)C(c2ccsc2C(=O)O)=O)ccc(F)c(C)c1 48401,N(C1CCCc2c[nH]nc21)CC.c12cc(cc(F)c1)C(N(CCC#N)C)C(=O)N2 48402,C1(CNC(C2CCCC(C)C2)=O)CC2(CC2)CN1C(=O)CCCN1CCCC1 48403,c1(N2CCC(C)(COC)C2)ccc(Br)c(S(=O)(=O)NCCC(C)CCO)n1 48404,N1(C(C2CC(OC)C2)=O)CCCC(C)(NC(=O)COCc2ccncc2)C1 48405,CS(=O)(=O)c1nc(Cl)cc(=NC2CCCCC2NC(C2CCCOCC2)=O)[nH]1 48406,CC(C)(C)C(CO)C(=O)NCC(F)CNC(=O)CCc1cccc(C(F)(F)F)c1 48407,C(=O)(C(F)C(F)(F)F)N(CCCN(C(C(N1C(C)CCC1C)C)=O)C)C 48408,c1(C(N(C(C)CN(C)C(c2ccc(CO)c(F)c2)=O)C)=O)sccc1S(C)(=O)=O 48409,C1(NC(c2nsnc2O)=O)CC(O)(C2CCN(C(c3ccccc3)=O)CC2)C1 48410,CCCC(CC)CC(=O)N1CC2CCN(C(=O)CCn3nc(C)nc3C)C2C1 48411,c1(C(N2C(CNC(CC(C)n3ccnc3)=O)COCC2)=O)ccn2c1CCCC2 48412,N1(Cc2scc(C)n2)CCC2(CC1)CN(C(C1(C)CCOC(C)C1)=O)CC(C)O2 48413,C1(C(N2CCCC(C)C2)=O)CCN(C(=O)CCCC2CCC2)C12CCC2 48414,N1(C(CC(CC)O)=O)CCCC(C2CC2NC(c2cc(C)nn2CC)=O)C1 48415,N1(C(C2CCCCC(=O)N2)=O)CCCC12CCN(C(C1(F)CC=CCC1)=O)CC2 48416,C1(C(=O)NC2CCN(CC(=O)Nc3ccccn3)CC2)CCc2ncccc2C1 48417,C(CC(O)C(=O)NC(C1CCN(C(=O)COC2CCN(C)CC2)C1)(C)C)SC 48418,C(=O)(C(O)C(C)(C)C)N1CCN(C(CNC(C(C2CCC2)OCC)=O)C)CC1 48419,c1(NC(Cc2cccc(-c3ccc(OC)c(OC)c3)n2)=O)c(Cl)nc(C)nc1Cl 48420,C1(C(=O)NCC(C)(F)CNC(C2CC(F)C2)=O)CCOC1(C)C 48421,CC(C)(C)CC(O)CC(=O)NCCCC1(CNC(C2(C#N)CCC2)=O)CCCC1 48422,C1(C(N2CC(CC(=O)OCC)C2)=O)CN(C)CCN1C(=O)CCc1ccco1 48423,c1(NC(C(CC)(F)F)=O)cc(NC2CCC2OC(C)(C)C)cc(C)c1 48424,C(=O)(CCC(C)NC(C1CN(C(=O)C(C)c2cc[nH]n2)CC1C)=O)OC 48425,C(=O)(C(CC1COCCO1)C(F)(F)F)N(C1CN(C(c2ccn(C)n2)=O)C1)C 48426,c1(C(=O)NCC2C(NC(C(CCC)C(C)C)=O)C2)cc([N+](=O)[O-])ccc1CC 48427,N1(C(=O)OC(C)(C)C)CCOC(CCSc2cnoc2-c2ccc(Cl)s2)C1 48428,C1(NC(CN(CCC)C)=O)CCN(C(c2cccc(N)c2C)=O)CC1O 48429,CN1CC=C(CC(=O)N2CCC3CCN(C(=O)CN4CCCNC4=O)C3C2)CC1 48430,c1(OC)nc(N2CCN(C(c3cc(Cl)c(Cl)s3)=O)CC2C)ncc1Br 48431,C1(CNC(c2ncc(C)cc2C)=O)CC2CCCC2N1C(c1cc(Cl)ns1)=O 48432,N1(C(C(CSC)OC)=O)CCC(C2CCN(C(c3cnc(C(C)C)s3)=O)CC2)C1 48433,C(=O)(CC(O)CNC(c1conc1C)=O)N(C)Cc1cnc(C)s1 48434,C(CC(N)=O)(c1cn(CCS(C)(=O)=O)nn1)NC(C(C)SCC)=O 48435,N1(C(C(CC)C(C)C)=O)CCC(CNC(c2csnc2C)=O)C12CCC2 48436,C1(COC)(NC(=O)CNC(c2cccs2)=O)CN(C(c2cocn2)=O)C1 48437,NC1(C2CCN(C3(C(=O)NC4CCCCC4)CCC3)CC2)CC1 48438,C(=O)(CCS(=O)(=O)NC)N1CC(C)(NC(C2N(CC)CC2)=O)C1 48439,C1(NC(c2ccsc2)=O)CCCCC1C(=O)Nc1ncccc1-c1ccccc1 48440,c1(C(=O)NCC2CC(F)(CNC(Cn3c(C)ccn3)=O)C2)ccnc(CO)c1 48441,C1(C(=O)NCCNC(c2c(C)nsc2NCC2CC2)=O)Cc2cc(F)cc(F)c2O1 48442,C(CC(C)C)(CS(C)(=O)=O)NC(c1cn(CCC)nc1C)c1nnnn1C1CC1 48443,C1(NC(c2c[nH]nc2-c2ccoc2)=O)CCCCN(C(=O)C(F)(F)C(F)F)CC1 48444,Cc1ccc2c(N3CCOC(CC(N4CCNC(=O)C4C)=O)C3)ncnc2c1 48445,C12(C(=O)NC(CC)CNC(=O)COc3cccc(Cl)c3)CCC(COC)(CC1)C2 48446,c1(C(N(C2CC2)Cc2cn(-c3c(C(=O)OC)scc3)nn2)=O)cc(=O)n(C)cn1 48447,c1(C(=O)OC)c(C(=O)NC(C)C(C)NC(=O)CC2(OC)CCCC2)n[nH]c1C 48448,C1(NC(c2c(CC=C)cccc2)=O)CC(C)CN(C(=O)C(C)(O)C2CC2)C1 48449,N1(C(c2ccn(COC)n2)=O)CCCC12CCCN(C(=O)C(C)CC(C)(F)F)C2 48450,C12(C(=O)NC(c3cnc(C)s3)C)C(NC(=O)Cn3cnnn3)C3CC1C2C3 48451,c1(C(=O)NCC2(O)CCCN(C(COC(CC)C)=O)C2)ccc(C#N)c(O)c1 48452,C=CC(C)(C)C(=O)NC(CSCC)C(=O)NCCN1CCCC(C)C1 48453,Cc1nc2ccccc2cc1C(N1CCC1C(=O)Nc1ccc(N)c(C)c1C)=O 48454,CN1CCCC(CNC(=O)C(O)CNC(c2ccccc2F)=O)C1 48455,c1(C(=O)OC)ccc(NC(c2cc(NC(=O)CC(C)C)n(C(C)C)n2)=O)cc1 48456,C1(C)(CNC(C(CC)OC)=O)CN(C(c2ccc(F)c(Cl)c2F)=O)C(C)(C)C1 48457,Cc1cc(C(=O)N(C(C)(C(=O)N2CC(OC(=N)O)C2)C2CC2)C)nn1C 48458,n1(CC(=O)N(CC(CNC(c2cnn(CC)c2C)=O)O)C)nc(C)c(Cl)c1C 48459,C1(C(N(CC(C2CCC2)OC)C)=O)CCCCC1(C)NC(c1cnc[nH]c1=N)=O 48460,N1(C(C(C2CCCO2)OC)=O)CC2(C1)CN(C(c1ccc(Cl)cc1F)=O)C2 48461,C12(CNC(c3ccc(Cl)[nH]3)=O)CC(CO1)N(C(c1cc(CF)on1)=O)C2 48462,C=C(CNC(C1CC(C)CO1)=O)CCNC(C1CN(C(=O)OC(C)(C)C)C1)=O 48463,N1(C(CC2C(C)CCCC2)=O)CCC=C(C(=O)NCCN(C)C2CC2)C1 48464,Cc1ccc(F)c(O)c1C(N1CC(CNC(=O)CCc2ccon2)C(C)C1)=O 48465,C1(n2cc(CC(C)(C)O)nn2)CCCCCN1C(=O)CCC12CCC(CC1)C2 48466,c1(C(C(=O)NCCCOC)N(C2CN3CCC2CC3)C)ccc(F)c(Br)n1 48467,C1(CC(=O)N(CC(C(=O)NCC(C(=O)NC)O)C)C)NC(=O)NC1=O 48468,CC1=C(C(=O)NC2CCOCC2NC(C2CC(CN(C)C)C2)=O)CCS1(=O)=O 48469,C12(C(N3CC=C(CNC(c4c(CC)cccn4)=O)CC3)=O)CCCN1CC(O)C2 48470,CCC(C)C(=O)C(=O)N1CCC(C)(C(=O)NCC2CCCC2)C1 48471,c1(C(=O)NC2C(C)(C)CN(C(C3(F)CCOCC3)=O)C2)c(F)ccc2occc12 48472,C(C(C)(CC(C)C)NC(=O)C(C)N(C)C)NC(C1(CC)CC1)=O 48473,Cc1c(C(=O)NC2CC2NC(c2ccc(C(F)(F)F)o2)=O)cnn1C1CC1 48474,N1(Cc2n(C)cc(C(F)(F)F)n2)CCC(O)C(CC(=O)O)(N(C)C)C1 48475,c1(C(N2CCC(OC)(CNC(C3(C)CCSCC3)=O)C2)=O)ccc(=O)n(C)c1 48476,C=C(CNC(C1C(O)CCN1C(c1cccc2occc12)=O)=O)C1CCOCC1 48477,C12(NC(=O)COC3CC3)CCC(C(=O)NCC(O)C3CCC3)(CC1)C2 48478,N1(C(c2cnn(CC(F)F)c2)=O)CCC12CN(C(C13CCCCC1C3)=O)C2 48479,N1(C(c2ccc(C(N)=O)nc2)=O)CCCCC(NC(C2C=CCS2)=O)C1 48480,N1(C(C2N(C(C3C(C)CCC3)=O)CSC2)=O)CCCCC12CC2 48481,C1(C(=O)NC(C2CCCC2)C#C)CCC2(CC2)N1C(=O)CC1(OC)CCC1 48482,N1(C(Cn2ncc(C)c2)=O)CCC2(CC1)CC2NC(C12CCC1C2)=O 48483,c1(N2CCC(C(=O)OC(C)(C)C)CC2)nccc(NCCN2CCCC(O)C2)n1 48484,c1(OC)cccc(C(N2CCCCC2CCNC(=O)C=CCOC(C)(C)C)=O)c1 48485,c1(C(C(=O)NC2CCC(N(C(=O)C(C)(C)CF)C)C2)=O)c[nH]c2cc(F)ccc12 48486,CN=c1nc(C(N2CC(NC(=O)C(C)(C)C(F)(F)F)CC(O)C2)=O)cc(C)[nH]1 48487,N1(C(C2CC(=C)C2)=O)CCC2OCCN(C(=O)CCc3ccc(SC)cc3)C2C1 48488,N1(C(CC=CC)=O)CCCC2(CCC2NC(C2CCCCO2)=O)C1 48489,n1(CCC(=O)NCCC(C)NC(c2c(C(=O)OC)scc2)=O)c(C)csc1=O 48490,c1(C(N2CC(C)C(CCNC(c3cccc(F)c3)=O)C2)=O)cncc([N+](=O)[O-])c1 48491,C1(NC(c2cc(SC)oc2)=O)CC(NC(=O)C2=CCCOC2)C12CCOCC2 48492,N1(C(CCCNC(=O)OCC)=O)CC2CCC1C(CNC(C1CCC1C)=O)C2 48493,C1(NC(CC(C)OC)=O)CCN(C(=O)C(C)Sc2ccccc2)C12CC2 48494,C1(c2n(C(C)C)nnn2)(NC(CC(N)=O)C2CCOCC2)CCOCC1 48495,C(=O)(C(Cc1ccoc1)NC(=O)C(F)=CC1CC1)N(CC(C)OC)C 48496,c1(CC)nnc(N2CC3(CN(C(=O)CCCn4cccn4)C3)C2)c(C#N)c1CC 48497,C1(CNC(CC=C)=O)CC2CCC(C1)N2C(=O)CS(=O)(=O)NC1CCC(C)CC1 48498,CC1(CNC(=O)Cn2ccc([N+](=O)[O-])n2)CN(C(c2cccnn2)=O)CCO1 48499,C1(CNC(CCc2cccc(OC)c2)=O)CN(C(=O)Cc2cc[nH]c2)CCCO1 48500,c1(C(=O)NC(CNC(C(C)Cc2cnc[nH]2)=O)C2CCC2)ccc2oncc2c1 48501,c1(C(=O)NC2C(NC(C3(COC)CCCCO3)=O)CC2)cc(C)ccc1C 48502,N1(C(c2nnn(CC)c2C)=O)CCC(NC(C2(Cl)CC2(C)C)=O)CC(O)C1 48503,C1(NC(c2cnc(CCCC)s2)=O)CN(C(C2(CC)CCNC2=O)=O)CC1C 48504,N1(C(CC2(NC(C3(C)CCC(=O)N3)=O)CCC2)=O)CC2CCC2(C)C1 48505,C1(C(N2C(C)C(NC(C3C4COCC34)=O)CCC2)=O)CCC(C2CC2)CC1 48506,S(=O)(=O)(c1ccc(N2CCC(CO)CC2)c(C#N)c1)N1CCC(C)C(CO)C1 48507,CC1CSCCN(C(=O)CC2CCCC(NC(=O)C(c3ccnn3C)O)C2)C1 48508,C1(NC(Cn2cc(CNC(C3CC(C)OC3)=O)nn2)=O)CC(C)(C)C12CCC2 48509,C1(C(N2CC(CNC(Cc3cn(C)nc3)=O)OCC2)=O)CC2C=CC1C21CC1 48510,c1(OC)cc(C(=O)NC2C3CN(C(=O)C=CSC)CC23)cc2nc(O)[nH]c12 48511,c1(C(=O)NC2CC3(C(NC(CC4N(CC)CCC4)=O)C3)C2)ccn2c1CSCC2 48512,c1(C(N(CC(CC)NC(=O)CC#N)C)=O)cc(C)c(F)cc1Br 48513,Nc1ccc(C(=O)NC2CCCN(C(c3cncc(F)c3Cl)=O)CC2)nc1Cl 48514,C=Cc1cnn(C)c1C(N1CCN(C(C2(C)CC2(Cl)Cl)=O)C(C)C1)=O 48515,N1(C(Cc2cccc(COC)c2)=O)CCN(C(=O)CCCCSC)C2COCC12 48516,N1(C(C2CC(C(=O)O)CN(C(=O)OC(C)(C)C)C2)=O)CCC(NC(C)C)C(O)C1 48517,CC1CN(C(c2ncn3c2CCC3)=O)CCCN1C(c1cccc(N)c1O)=O 48518,N1(C(C2OCCN(CC)C2)=O)CCN(C(c2scc(C)c2C)=O)CCC1C 48519,C(=O)(C1=C(Cl)CCCC1)N1C(C)CC1C(=O)NC1(CO)CCCCC1 48520,CCCC(C)CC(=O)N1CCCCC(N(C)C(c2cc(C)n(C3CC3)c2C)=O)C1 48521,N1(C(c2ccc(CN(C)C)cc2)=O)CCC=C(CNC(=O)CC2CCC3CC23)C1 48522,c1(C(C)C)nc(NCCCC(C)C)cc(=NCC2CCCC(CO)C2)[nH]1 48523,c1(C(=O)NCc2nc(CNC(CCc3nc(=N)[nH][nH]3)=O)sc2)cccnc1S 48524,N1(C(C2N(C(Cn3nc(C)oc3=O)=O)CCC2(C)C)=O)CCC2(CCCCO2)C1 48525,Cn1nnc2c(C(N3CCC(NC(C4CCC(F)CC4)=O)C3)=O)ccnc12 48526,c1(C(C(N2CC=CC(OCC)C2)=O)NC(CCN(C)CC)=O)c(C)cccc1Br 48527,N1(C(C(OCC)OCC)=O)CCC(F)(C(=O)NCC(C)(C)CN2CCCC2)CC1 48528,Cn1nc(Br)cc1NC(C1CCCN1C(=O)COc1ccccc1)=O 48529,C(N=c1[nH]c2ncc(Cl)cc2o1)c1c(C)c(C(F)(F)F)n[nH]1 48530,c1(C(=O)NCCC(C)NC(C2C3CCCCCC23)=O)c(F)ccc(F)c1Cl 48531,Cc1ccc(CCCC(=O)NC(C)(CNC(C2CCCCC2O)=O)C2CC2)cc1 48532,C1(C)(C(N2CCC(NC(CC(C)(C)OC)=O)(CO)C2)=O)CCC(F)(F)CC1 48533,c1(C(=O)NCCCOCCOCCOC)cc(C)nc2c1c(C)nn2C 48534,c1(C(=O)NC2CC(NC(C(Cn3ccc(C)n3)C)=O)C2)nccc(F)c1Cl 48535,C1(CNC(COCCOCC#C)=O)(CNC(=O)C(C)SC)CCOCC1 48536,C1(C(N2C(CCCNC(CCC=C)=O)CCC2)=O)CCOC(C)(C)C1 48537,Cc1cc(C(N2CC(C(C)NC(c3cc4occc4s3)=O)C2)=O)cc(N)c1O 48538,C1(COC)(NC(c2cc[nH]c(=N)c2)=O)CCN(C(=O)C(C2CCOCC2)C)CC1 48539,C1(NC(CCSCC(C)C)=O)CCC2CCN(C(c3c[nH]ccc3=O)=O)C12 48540,c1(C(c2nnnn2C2COC2)NCC(C2CCSCC2)(C)O)cccc(CO)c1 48541,N12CC3CCC1CN3CC1(CC(=C)C1)C2=O.C1(C(=O)OC)CCCO1 48542,CC1(NC(c2nccnc2Cl)=O)CCCN(C(c2ccc(=O)oc2)=O)C1 48543,C12(C(=O)NCC3(CNC(C4N(CCC)C(=O)CC4)=O)CCC3)CCCC1OCC2 48544,C1(C(C)(C)C)CCCN(C(=O)C(CO)NC(C2CC(F)(CF)C2)=O)C1 48545,N1(C(C=CCC)=O)CC(CNC(c2cccs2)=O)CC12CCOCC2 48546,c1(C(=O)NC(CN(C(=O)CN2CCC(C)C2)CC)C)sc2cc(F)ccc2c1C 48547,c1(CC(=O)NC(C(C)NC(=O)Cn2cncn2)CO)coc2ccc(F)cc12 48548,c1(C(=O)NCC2(O)CCCN(C(c3cc(Cl)no3)=O)C2)ccc2c(c1)CCCO2 48549,N1(C(CC=C=C)=O)CC(NC(=O)C(CC)CC)C(S(C)(=O)=O)C1 48550,CCCCCC(C)(C)C(=O)NC1CN(C(c2c[nH]c3cccnc23)=O)CC1CO 48551,CC1CN(C(=O)OC(C)(C)C)CCS1(=O)=O.C12(F)CN(C1)C(=O)N2 48552,c1(OC)ccccc1OC1CCN(C(=O)C(=O)NCC2(C)COC(=O)N2)C1 48553,C(=O)(CCCCCC(C)C)N1C(C)CCC(NC(C2(CC=C)CC=CC2)=O)C1 48554,N1(C(C2N(C(COCCC=C)=O)CCSC2)=O)CCc2nocc2C1 48555,C(c1ccc(C)c(C)c1)=CC(=O)NC1C2(CC(NC(C(CC3CC3)OC)=O)C2)C1 48556,Cc1cc(C(=O)NCC2(C)CC(NC(C3(C)CC3)=O)C2)sc1Br 48557,Cc1ccc(C(N2CCN(C(=O)C(C#N)C(C)C)C(C3CC3)C2)=O)nc1O 48558,Cn1ncc2c1CCCC2N=c1[nH]c(=NCC2SCCS2)[nH]c2cc[nH]c12 48559,C1(CCO)CCN(C(=O)NC2(CNC(=O)OC(C)(C)C)CCCCC2)CC1(C)C 48560,c1(N2CCN(CC)CC2)nc2cccnc2c(=NCC2CCCC(F)(F)CC2)[nH]1 48561,c1(C(=O)Nc2cccc(NC(CC3C(CC)C3)=O)c2)c(Br)c(C)nn1C 48562,C1(C(N2CC(OCC#C)C2)=O)CCC(C)N(C(=O)C(O)Cn2cncn2)C1 48563,C1(F)(C(N2CCC(NC(Cc3c(C)con3)=O)CC2)=O)CS(=O)(=O)CC12CCC2 48564,c1(C(N2CCC(CC)C2CNC(=O)COCC2CC2)=O)cnc2nccn2c1 48565,Cc1cc(F)sc1C(=O)NC1CCC(CCNC(c2ccc(C3CC3)o2)=O)C1 48566,C1(NC(C(c2ccccc2)OC)=O)CN(C(=O)Cc2ncncc2Cl)CCC1F 48567,c1(NC(C2CC(F)(F)C2(F)Cl)=O)ccc2c(c1)CCCC2 48568,c1(C(c2n(CCOCC)nnn2)N)cnc2c(c1)CCC2.C(CCO)CC1CCC1 48569,c1(C(=O)OCC)ccc(CCNC(=O)C(=O)NC(C)C(C)(C)C#N)cc1 48570,N1(CC(N2CC(NC(=O)OC(C)(C)C)OCCC2)=O)CCCC2(CC2)S1(=O)=O 48571,CCCCCCC(=O)N(CCNC(c1sccc1C1CC1)=O)CC 48572,C1(NC(CC2C(C#N)C2)=O)C2CN(C(c3cnn(-c4cccnc4)c3)=O)CC12 48573,Cc1cc(C(N2CCCC(NC(C3C=CCC3)=O)C2C)=O)c(O)c(C)n1 48574,c1(OC)cccc(C)c1C(N1CC2CC1(CNC(C1CC13CC(O)C3)=O)C2)=O 48575,N1(C(C(CCSC)O)=O)CCCC2(CCC(=O)N2)C1 48576,C1(NC(C(CC)N(C)C)=O)CCN(C(=O)Cn2cnnc2)C12CCC2 48577,n1(CC(=O)NCC2CC(NC(=O)CCc3cnoc3)C2)ccccc1=O 48578,C(C)(C(C(=O)N1C(CO)CC1C)C(C)C)NC(C1ON=C(CC)C1)=O 48579,CCC(COC)(CC)C(=O)N1CC(CC(=O)NCC(C)O)(OC)C1 48580,c1(C(=O)NC(C2CCCO2)C)ccnc(CNC(C2(C(N)=O)CC2)=O)c1 48581,c1(NC(c2c(NC(C(CCC)C)=O)ccs2)=O)ccc(Cl)cc1Br 48582,c1(C(=O)NC2CC(CNC(C(n3ncc(C)c3)C)=O)C2)ccc2cccnc2c1 48583,CC1CN(C(c2nnn(C)c2C(F)F)=O)CCC1NC(=O)C=Cc1ccccc1 48584,C#CC1(O)CCN(C(C2CCCC(NC(=O)CNC(=O)NC)C2)=O)C1 48585,C1(CCC=C)CCCN(C(C23CC2CCN3C(=O)C(=O)NOC)=O)C1 48586,CC1CN(C(c2cncn(C)c2=O)=O)CCC1N(C)C(c1ccc(CO)cn1)=O 48587,CC(C(C(=O)O)NC(=O)CC1CCN(C(=O)OC(N)=O)C1)OC(C)(C)C 48588,C=CCC(CC)C(=O)N1CC2(CC(CC(N3CCC(c4ccon4)C3)=O)C2)C1 48589,c1(C(=O)NC2C(C)CN(C(=O)CC(C)(F)F)C2)ncnc2c1c(Br)cn2C 48590,C12(C(N(CC(=O)NC(c3cnccn3)C)CC3CC3)=O)CCCC1C2(F)F 48591,c1(C2C(C(=O)NCCCOCCNC(C(CC#C)O)=O)C2)cccc([N+](=O)[O-])c1 48592,CC1CCCC(NC(=O)C(C)CN(C)C(c2cnn(C3CC3)c2)=O)C1 48593,c1(NC(C23CC(CNC(CCCOCCC)=O)(C2)C3)=O)ccc(OC(C)C)cc1 48594,c1(C(=O)OC)cn(C)[nH]c1=NC(=O)N1CCC(OCCCO)CC1 48595,c1(C(N2CC(NC(CN(C3CC3)CC)=O)C(C)C2)=O)c(C(F)F)nn(C)c1C 48596,N1(C(COC)=O)CC(CNC(c2c(F)ccc(Br)c2F)=O)C2(CCC2)C1 48597,c1(C(N2CC(CC(C)NC(=O)CSC(C)(C)C)C2)=O)cnc(C(F)(F)F)c(F)c1 48598,C(=O)(C1=CCN(C(C2CCNC(=O)C2)=O)CC1)NCC(C)(C1CC1)OC 48599,C(CCCCC(=O)NCC1C(C)CCN1C(=O)CC1(C)CC1(Cl)Cl)OCC 48600,C(=O)(CC(CC)SC)N(CCC)CCNC(=O)COCCF 48601,C1(CNC(C(CC)OC)=O)(NC(C23CC(C(=O)NC)(C2)C3)=O)CC(F)(F)C1 48602,CCC(CCOC)C(=O)N1CC(CN(C(=O)C(C)(C)n2cnnn2)C)C2(CC2)C1 48603,N1(c2cc(C(=O)OC)nc(Cl)n2)CC2(C1)SCCC2NC(=O)Cc1n[nH]c(C)n1 48604,c1(NC(=O)NC)ccc(NC(C2(NC)CC2)=O)c(OC2(C)CCC2)c1 48605,C1(C)(CN(N(CCC)CC)C)COCCC1NC(=O)OC(C)(C)C 48606,N1(C(C(C)(C)OCC)=O)CC2CCC(N(C(=O)CCS(C)=O)C)C2C1 48607,c1(CNC(C(C)O)=O)cccc2c1CCN(c1cccc(Cl)c1[N+](=O)[O-])C2 48608,c1(C(=O)NC2CC(C)(CNC(=O)CNC(=O)NC3CC3)C2)ccc2nccn2c1 48609,Cc1cc(=NC(C)CCCC(F)(F)F)[nH]c(=NCC2CC23CCC(O)CC3)[nH]1 48610,C1(C(=O)NCC(C(C)C)CO)C2CC3C(C2NC(c2ccccn2)=O)C13 48611,c1(C(=O)NC2CN(C(c3cc(C)ns3)=O)CC(F)(F)C2)cnc2ncnn2c1C 48612,c1(CC(=O)NC2C(C)CN(C(=O)CCCCN(C)C)C2)ncn2c1CCC2 48613,CCC(C)(C(=O)N1CCC(OCCNC(=O)C(C)(C)n2ccnn2)C1)OC 48614,C(=O)(C(C)(C)C1=CCSCC1)NC1CCN(C(c2c(Cl)ccc(OC)c2)=O)C1 48615,O=C(CCCC(F)F)NCC1CCN1C(c1ccc(CO)nc1)=O 48616,C1(=CCNC(c2ccc(SC(F)(F)F)cc2)=O)CCN(C(=O)C(O)CF)CC1 48617,Cc1ccc(C)c(C(=O)NC(C2CCCN2C(=O)CC(=O)NC2CC2)C)c1 48618,N1(CCc2nn[nH]n2)CCN(C(c2ccccc2)C2CC2c2ccsc2)CC1 48619,C1(C(=O)NC(c2ccccn2)(C)C)CCCCC1NC(C1CNC(=O)C1)=O 48620,c1(C(N(CC=C)CC)=O)ccnc2nc(=NC(=O)C(C)C(=O)OC(C)(C)C)[nH]n12 48621,N1(C(C(CCC(C)C)O)=O)CCC2(CC1)CC(C)N(C(=O)CCCC1CCC1)C2 48622,C(=O)(C(C)CC(C)CC(C)C)NCC1(C)C(C)CN(C(C(C(CC)(C)C)O)=O)C1 48623,CCC(CC(=O)N(C1CC(NC(=O)Cc2cc[nH]n2)C(O)C1)CC)C(C)C 48624,CC(C(=O)OC(C)(C)C)C(=O)N1CC=CC1CNC(=O)C=Cc1nccs1 48625,C1(C(=O)NC2(CC=C)CN(C(=O)C(C)C)C2)C2CC2C2CC12 48626,Cc1noc(C)c1CC(C)C(=O)NCC1CCN(C(=O)CCc2cccnc2)C1 48627,C(C1CSc2ccccc21)NC(=O)Nc1cn(CCOC2CCCCC2)nn1 48628,c1(C(c2n(CCCSC)nnn2)NCCN(S(C)(=O)=O)C)cc(F)cc(C#N)c1 48629,C(C)(CN=c1ccnc(N2CCOC(C)(c3cccs3)C2)[nH]1)n1c(C)cc(C)n1 48630,C=CCC(CNC(c1cc(C)cc(C)n1)=O)C(=O)NC(C)CN1CCCC1 48631,c1(CN2CCCC(NC(CCC(C)C)=O)CC2)cc(Cl)c(O)cc1F 48632,Cc1cc(F)ccc1C(=O)N(CC(C)C(=O)N(C)Cc1cccc(F)c1)C 48633,c1(C(N(CCC(C)NC(C2(OCC)CCOCC2)=O)C)=O)cc(F)c(Cl)cc1F 48634,Cc1cc(C(F)(F)F)sc1C(N1CC(C)C(F)C1)C(=O)NC1CCC1 48635,Cc1cc(=NCCN(C)C(C2Cc3cccc(C)c3O2)=O)[nH]c(C)n1 48636,C1(CC(=O)NCC(C)(C)CC2CN(C(c3ccncn3)=O)C2)CCC=CCC1 48637,Cc1ccc(-c2ccc(C(N3CCC(O)(CN)C3)=O)cc2)cc1Br 48638,C1(NC(c2ccc(C#C)cc2)=O)CN(C(c2ccc[nH]2)=O)CC12CCC2 48639,N1(C(=O)NCC(Cc2ccc(OC)cc2)OC)CCC(O)C2(CCC2)C1 48640,Cc1ccc(C)n1CC(N1CCC=CC1C(=O)NOCC1CCOCC1)=O 48641,N(C(=NCC1CN(C)S(=O)(=O)c2ccccc21)N1CCCC2(CCOC2)C1)C(C)C 48642,c1(CNC(CCOCCN(C)C)=O)cn(C2CN(C(c3nocc3Cl)=O)C2)nn1 48643,N1(CCC(=O)NC(C)CCCNC(c2sccc2F)=O)CCCC(N(C)C)C1 48644,CC1CCC(C)N1CC(=O)NC1(C)CCN(C(c2c[nH]nc2C2CC2)=O)C1 48645,N1(C(C=CC)=O)CCC(C2CCCN(C(=O)CS(=O)(=O)CC(F)(F)F)C2)C1 48646,CC(C)CCCCCC(=O)N(C1CCC2CN(C(c3ncc[nH]c3=O)=O)CC12)C 48647,c1(C(N2CC(O)CC(NC(c3cc(C)[nH]n3)=O)C2)=O)csc2cc(Cl)cnc12 48648,CCC(CC)(C(=O)N1CCCC(c2ccc(NC(C)=O)c(Cl)c2)C1)OC 48649,N1(C(c2cn(CC)nc2C)=O)CCN(C(c2ccc(N)c(C)c2F)=O)C(C)C1C 48650,CC#CCC(C(=O)NCC(O)COC)NC(=O)Cc1cccs1 48651,CS(=O)(=O)C(C(=O)N1CC(NC(=O)Cc2cccc(C3CC3)c2)C1)C1CC1 48652,c1(OC)cnc(Cl)cc1C(N1CCC(NC(=O)C(C)(Cl)Cl)C(C)C1)=O 48653,C1(C(C)(C)C)(CNC(C(C)OCC)=O)CCN(C(C2CCC(N(C)C)CC2)=O)C1 48654,C(=O)(C1=NOC2(CCC2)C1)N1CC(C)N(C(=O)CCP(C)(C)=O)CCC1 48655,c1(C(N(CCOC)C)=O)n[nH]c2cc(C(=O)N=c3[nH]nc(C4CC4)o3)ccc12 48656,C1(CNC(CC2CCN(C)C2=O)=O)CN(C(c2cnc(S)[nH]2)=O)CC12CC2 48657,C(=O)(C1(C)CCc2ccccc21)N1CCC(C)N(C(C2CC23CCOC3)=O)CC1 48658,C(=O)(CCC(=O)NN(C)C)NC(CC#CC)C(=O)NCc1oc(C)nc1C 48659,N1(C(CCCCCCC)C(=O)NC(C)(C)CC)Cc2ccccc2CC1(C)C 48660,CC1(C)CC(CNCCc2c(F)cccc2F)CCO1 48661,Cc1ccc(C(N2CCCC(NC(=O)C=CC(=O)OC(C)(C)C)C2CO)=O)c(Cl)c1 48662,C(CCCN=c1[nH]nc(C2CCCC2)s1)NC(c1cnn(CC2CCCO2)c1)=O 48663,N1(Cc2c(C)sc(C(=O)O)c2)CC(F)(C(=O)O)C2(COC2)C1 48664,C1(NC(C2N(C(c3c(C)csc3)=O)CC(O)C2)=O)CNC(=O)C12CC2 48665,CCC(CC(=O)NCC(C(C)C)NC(c1cccc(O)c1F)=O)C(F)F 48666,c1(CC)cccc2c3c([nH]c12)C(CC)(CC(=O)NC(C)CC1CCCO1)OCC3 48667,N1(C(C(=O)NCC2C(F)(F)C23CC3)=O)CC(=O)NCC12CC2 48668,S(=O)(=O)(c1ccc(Cl)nc1)N(C1COC2(CCNCC2)C1)CCCNC(C)=O 48669,Cc1n[nH]cc1C(=O)NCCCOCCNC(=O)CNC(N)=O 48670,n1(CC)ncc(C(N2CC(NC(=O)C(C)c3ccsc3)C2)=O)c1C(F)(F)F 48671,CC1=C(C)CC(C)(C(=O)NC2C=CCN(C(c3ncsc3S(N)(=O)=O)=O)C2)CC1 48672,C=CCCCCC(=O)NCC1CCC(Cn2cc(C(=O)O)nn2)CC1 48673,C(=O)(C1=CC2C=CC(C1)C2)NCC(C(NOCCC(C)O)=O)O 48674,N1(C(c2cc(C)no2)=O)CCC(C)C(CNC(=O)CCCOC(C)(C)C)C1 48675,C1(C(N2CC(C3CN(C(CNC(C)=O)=O)C3)C2)=O)Cc2cccc(Cl)c2C(=O)O1 48676,C(=O)(CCCCC(N)=O)NC1CC(N(C(C(CC(C)C)NC(C)=O)=O)C)C1 48677,Cc1ccc(C(c2nnnn2C2CC2)NCc2ccc(CS(N)(=O)=O)cc2)cn1 48678,Cc1cccc(C)c1OCC(=O)NC1CCN(C(=O)CC2CCC2)C1C(C)(C)C 48679,C1(CC(=O)N(CCNC(c2sccc2C(F)F)=O)CC)SC2=NCCN2C1=O 48680,c1(CC(N2C3(CN(C(c4c(C)nns4)=O)C3)CC2)=O)n[nH]c2ccccc12 48681,c1(Sc2nnc(N3CCC(OCC)C3)s2)ccc(Cl)cc1 48682,C(CCCC(=O)N1CCC1C1CCCC1)NC(Cn1c(C)ccn1)=O 48683,c1(C(=O)NC2C(CNC(CCC3(C)CC3)=O)CCC2)ccc2cnoc2c1 48684,C1(NC(=O)C2=NOCC2)CC2(CCN(C(C3CCCCC34CC4(F)F)=O)CC2)C1 48685,CC1COCCC1N(C(=O)C(C1CCCO1)NC(=O)CCC1CCC(=O)C1)C 48686,N1(C(CCC(OC)O)=O)CCCCC(C2CN(C(C)C)C2)C1.C(C(C)(C)OC)N 48687,C=CCC(C(=O)NC(CC(N)=O)C(=O)Nc1cc(C)cc(O)c1)C(C)C 48688,N1(C(c2ccc(Cl)s2)=O)CCC(C2CCN(C(C3(O)CC3)=O)CC2)C1.C(=O)C1CC1 48689,c1(NC(C(COC(C)C)NC(C(CC)OC)=O)=O)ccc(OC(C)C)c(C)c1 48690,c1(OC)cnc(C(N2CC3C(CNC(C4(CO)CC4(F)F)=O)C3C2)=O)nc1 48691,N1(C(CC(C)(F)F)=O)CC2COCCC2(NC(c2ccnc3[nH]cnc23)=O)C1 48692,c1(C(=O)NC(C(C)NC(C23CC(O)C2C3)=O)C)ccc(Cl)cc1 48693,C1(NC(CC(COC)(C)O)=O)C2CC(O)C1N(C(=O)CCCc1cccs1)C2 48694,N1(C(c2ccc(CSCC)cc2)=O)CCN(C)C(CNC(=O)C(C)CCO)C1 48695,n1(CC)ncnc1C(C)NC(c1ccccc1)c1nnnn1Cc1cccs1 48696,N1(C(C=C(C)C(C)(C)C)=O)CC2CCC2(CCNC(=O)C=Cc2cccn2C)C1 48697,C(=O)(C(C(F)(F)F)=Cc1ccccc1)N1C(CNC(c2c(C)csc2)=O)CCC1 48698,n1(CC(=C)C)nnnc1C(c1nc(C2CC2)cs1)NC(C1CCC1)C1CC1 48699,C1(C2CCC2)(C(=O)NCCCC2(NC(=O)CC3CCCC(=O)N3)CC2)CC1(F)F 48700,n1(CCCC)nc(C)c(C=CC(=O)N(CC(C)C(=O)OC)CCC)c1Cl 48701,C1(COCC)C(C)CCCN1C1(CNC(=O)OC(C)(C)C)CC1.c1cnc(C#N)s1 48702,Cc1cnoc1C(=O)NCC1(NC(C2CC(CC3CC3)C2)=O)CCC1 48703,N1(C(C2CCN(CC(C)C)CC2)=O)CCC(NC(=O)CCC(C)(C)C)C(C)(C)C1 48704,C1(C(N2CC(CC(C)C)OCC2)=O)CC(O)CCN1C(c1cc(O)cc(F)c1)=O 48705,N1(c2ncc(CCCOC)cn2)C2CCC1C(NC(=O)OC(C)(C)C)C2.CC 48706,C(CC(CNC(=O)C(C)(C)C1CCCCO1)NC(C1(OC)CC1)=O)OC 48707,N1(C(C(C2CCCC2)OC)=O)CCC(N(C(=O)C(O)C(C)C)CCO)CC1 48708,Cc1cc(C(N2CC(CC(C)NC(c3cccc(=S)n3O)=O)C2)=O)c(F)cc1F 48709,c1(OC)cccc2c(C(=O)N(CC(C)NC(=O)Cc3cncc(O)c3)C)csc12 48710,S(=O)(=O)(c1ccc2c(c1)CC(C(=O)O)C2)NC1CCC(C(C(=O)OC)(C)C)CC1 48711,c1(C(=O)NC(C(N2CC3(CCC(=O)N3)C2)=O)C2(C)CC2)cccc2cncn12 48712,c1(C(=O)NCC(C)NC(=O)C(O)CC2CCOCC2)cc(Cl)ccc1C(F)(F)F 48713,C1(C(N2C(C)CCC(CNC(=O)CCc3ccoc3)C2)=O)CC2CCC(C1)C2O 48714,CN1CC(NC(C2C3CC3CN2C(c2nn(C)cc2Cl)=O)=O)CC1=O 48715,C1(CCNC(C(F)=CCC)=O)CCN(C(C2CC2C#N)=O)CCC1(F)F 48716,C(=O)(CCCC(=O)N1CC(C)(CCC(=O)Nc2cnc(F)cc2C)C1)OCC 48717,C1(OC)CCCC(CNC(C2CC(C)N2C(c2cscc2Cl)=O)=O)C1 48718,N1(C(C(C)CC2CCC2)=O)CC2CC(CNC(c3cnc(S)[nH]3)=O)C2C1 48719,c1(OC)cc(CCCNC(C2CCCC2)C2CCC2)cc(OC)c1O 48720,C(CC(C(=O)N1CCC(NC(=O)N(C)C)C1)NC(C1CCOC1C1CC1)=O)SC 48721,c1(C(=O)NC2C(CNC(C(CC)NC(N)=O)=O)CC2)cc2nc(=O)ccn2[nH]1 48722,C1(N(C(COC)=O)C)CCCC(N(C)C(c2cn(C3CC3)cn2)=O)C1 48723,C1(C)(CNC(CCc2n(C)cnn2)=O)CCN(C(C23CCCCC2C3)=O)CC1 48724,CC1CC(NC(C2COC(=O)N2)=O)CN1C(C1CCN(C2CC2)CC1)=O 48725,N1(C(COC(C)(C)C)=O)CCC(N(C(=O)CC2C=CCCC2)CC2CC2)C1 48726,c1(OCC)ncc(C(N2CC(NC(=O)CCCC3CC3)CC(C)C2)=O)cc1Cl 48727,N1(C(C(C=C)O)=O)CCCN(C(c2nc(OC)c(C)s2)=O)CC1C(C)C 48728,C1(C#N)(C(=O)NC2CCC(NC(c3cccc(CC)c3)=O)CC2)C(C#N)C1(C)C 48729,C1(C(=O)NC2CCC(NC(=O)Cc3csc(Cl)n3)C2)CCOC(=O)N1 48730,CCC(C)CCC(=O)NC(C)C(C)(C)C(=O)NCCN(CC(F)F)C 48731,C1(N(C(C(C)=C2CCC2)=O)C)CCN(C(=O)Cn2ncccc2=O)CC1C 48732,C(CCC)(C(=O)NC1COCC1CNC(C1CSCCS1)=O)=CCC 48733,N1(C(c2n(CC)ccc2)=O)CCCC12CCN(C(=O)CC1CC3CCC1O3)C2 48734,C1(C)(C(=O)NCC(C(CC)C)C)CCN(C(C2(CN(C)C)CC2)=O)CC1 48735,c1(C(=O)CN2CCC3(CCC(=O)N3)C2)cc2c(cn1)OCCC2 48736,CC(CN(C)C)CC(=O)N1CCC(CC(=O)NC2CC(CN(C)C)C2)CC1 48737,Cc1cc(Br)ccc1CC(=O)NCC#CCNC(c1cc(C2CC2)nn1C)=O 48738,C1(C(=O)NC2(C(N(C)C)=O)CCCCC2)CC2CCC1N2C(=O)COC(C)(C)C 48739,CCC(CCCC(=O)NC1CCCC1)NC(=O)CN(C)C(C)C 48740,c1(CC)cc(C)c(C(=O)NCC(=O)NCCCN(C(=O)C2=CCCC2)C)o1 48741,N1(C(C2(CCCC)CC2)=O)CCC2(NC(c3cc(-c4ccc(C)s4)[nH]n3)=O)CC2C1 48742,C(=O)(C(O)CC(C)(C)C)NC(CC)CNC(=O)C=Cc1ccc(OCC#N)cc1 48743,C1(O)(CNC(C2(CCC=C)CC2)=O)CCCN(C(c2nnc(O)nc2O)=O)C1 48744,C1(CC(=O)NC2(c3ccnc(Cl)c3)CC2)CCN(C(C2NC(=O)NC2=O)=O)CC1 48745,c1(CC(=O)Nc2cc(Cl)c(Br)cc2O)cc2ccccc2nc1O 48746,n1(C(C)C)cccc(C(=O)NCc2cn(CCNC(C3CC(F)C3)=O)nn2)c1=O 48747,c1(C(=O)NC2CCN(C(C(C=C)O)=O)CC2)ccc(Cl)c(OC)c1 48748,CCC(C)C(O)C(C)C(=O)N1CCCC(C(=O)N(C)CC2(CO)CC2)CC1 48749,c1(C(=O)NC2CCN(C(C(C3CCC3)OC)=O)C2C2CC2)ccc(C)c(C)n1 48750,N1(C(CN(C)CC)=O)CCC(COC)(NC(=O)COc2c(Cl)cccc2Cl)CC1 48751,C1(C(=O)NCCCN(C(=O)CC(C)(C)F)C)CCCCC1(C)C 48752,C1(NC(C2COCCO2)=O)C2CC3CN(C(=O)C#CC4CC4)C1C3C2 48753,N1(C(CC(CN(C)C)O)=O)CCCCCC(Nc2ncc(C#N)cc2C(N)=O)C1 48754,N1(C(c2c(OC)ccnc2)=O)CC(NC(=O)Cc2csc(C)c2)CC(F)(F)C1 48755,C(=O)(C1CC(=O)c2ccccc21)NCC(C)NC(c1c(C)cc(C)[nH]1)=O 48756,N1(C(c2cc(C)ns2)=O)C2CCCC1CC(NC(c1c(C)[nH]c(C)c1C)=O)C2 48757,c1(C(=O)NCCOCCN(C(C(COC)(C)OC)=O)C)c(C)cccc1[N+](=O)[O-] 48758,CCCC(C(=O)OC)C(=O)N(C(C)CNC(c1cccn2cnnc12)=O)C 48759,N1(C(C2CC(=C)C2)=O)CCC2(C1)CN(C(=O)C(C1CCC1)OC)CCO2 48760,c1(C(=O)NC2C(NC(Cc3cn(C)nc3)=O)CCC2)ccc2cnnc(O)c2c1 48761,C(=O)(CCC(C)(C)C(=O)NC1CC1NC(C1CCCc2ccccc2O1)=O)OC 48762,N1(C(C(CCC)N(C)C)=O)CC2(C1)CN(C(c1cc(OC)cc(=O)o1)=O)C2 48763,C1(CNC(c2ccnc(-n3ccnc3)c2)=O)CN(C(C2CCOC2=O)=O)CCO1 48764,c1(SC)cc(C(N2CCC(C3OCCO3)C2)=O)co1 48765,c1(C(=O)NCC2C(CNC(CNS(CC)(=O)=O)=O)C2)csc(SC)n1 48766,N1(C(CCC(C)C)=O)CC2CCC(NC(c3cccc(CN=[N+]=[N-])c3)=O)C2C1 48767,CCC(C)(C)CCN=c1[nH]c(N2CC(CCOC)OC(C)C2)nc2ccccc12 48768,CC(C)C(=O)C(=O)NC(c1ccnn1C)C(N1CCC(OCCO)C1)=O 48769,N(C(=NCc1ccnn1C)N1CCOC(C2CCC2)C1)CC(CC)(C)C 48770,C1(NC(Cc2cc(C)ns2)=O)CN(C(=O)C(O)CC(=O)OC(C)(C)C)CCC1F 48771,c1(NC(N(c2cc(OC)ncn2)C2(CO)CNC2)=O)cc(C)cc(C)c1 48772,Cc1cc(C=CC(=O)NC2CC(NC(c3csnn3)=O)C23CCC3)c[nH]c1=N 48773,c1(C(=O)NC2CC(C)(NC(c3cc(C)oc3C)=O)C2)nccc2ncccc12 48774,c1(C(N2CC3C(CNC(c4cc(O)ccc4F)=O)(C3)C2)=O)ccc(I)cc1Br 48775,Cc1scc(C(N2CCC2CNC(=O)C(c2ccccc2)OC(C)(C)C)=O)c1C 48776,C1(C(N2CC(OC)C2)=O)CC(C)CN1C(=O)CCC1CC1(F)F 48777,CCC(CC(=O)NCC(C1CCN(C(c2cc(C)c(C)o2)=O)CC1)(C)C)C(C)C 48778,CC(CCC(=O)NCC1(CNC(C2(F)CCOC2)=O)CCC1)c1ccccc1 48779,CC1CCN(C(=O)C(C)NC(C2CC2C)=O)CC1.c12cn(nn1)CC(=O)NC2 48780,C1(C(=O)NCC(CC)NC(C2(N(C)C)CC2)=O)CCc2cc(OC)ccc2C1 48781,C1(NC(C2CCN(C)C2=O)=O)CC2CC1N(C(=O)CSc1nc[nH]n1)C2 48782,N1(C(c2nn(C)c(F)c2)=O)CCCC1C1CCCN1C(c1n[nH]c2c1CCC2)=O 48783,CC(C)C(C)C(CNC(c1csc(-c2ccsc2)n1)=O)NC(C1OCCO1)=O 48784,N1(C(C(CC(=C)C)C)=O)Cc2ccnn2CC(NC(c2cc(CC)oc2C)=O)C1 48785,O=C1CSC2(CN(C(C34CCC(CC3)N(C(c3nocc3Cl)=O)C4)=O)C2)N1 48786,c1(CNC(C(C2(O)CCC2)NC(=O)Cc2cccs2)=O)ccc(Cl)nc1 48787,Cc1ccc(NC(=O)C(CC2CC2)NC(=O)CC2CCN(C)C2=O)cc1C#N 48788,c1(C(=O)NCCN(C(C(CC)n2cccn2)=O)C(C)C)c[nH]cc(F)c1=O 48789,c1(C(=O)NCCC2N(C(C(N)=O)=O)CC(F)(F)C2)cc(Cl)cc([N+](=O)[O-])c1 48790,N1(CC)CC(C(=O)N2CCC(C)(NC(=O)CS(=O)(=O)CC)C2)c2ccccc21 48791,Cc1nc2c([nH]1)CC(C(N1CCC13CN(C(C1CC4(CC4)CO1)=O)C3)=O)CC2 48792,C=CC1CCCN(c2ncccc2CNC(c2scc(C(=O)OC)c2C)=O)C1 48793,C1(=CC(=O)NC2CC(O)CN(C(=O)CC3CCOCC3)C2)CN2CCC1CC2 48794,CC1CN(C(=O)C(C2CCCCCC2)O)CC(C)N(C(c2cc(C#N)c[nH]2)=O)C1 48795,Cc1nc(NCc2cccc3c2CNC3=O)cc(=NCC2CCCC2N(C)C)[nH]1 48796,c1(OCC(=O)NC(C2CCOC2)CNC(c2c(C)nc[nH]2)=O)cc(F)cc(Cl)c1 48797,c1(C(=O)NC2CCCN(C(C(CCC)CC)=O)CC2)cccc2c1CC(C)(C)C2 48798,C1(OC)CC(CC(=O)NC2(CNC(c3cnc(C)cc3C)=O)CC2)C12CCC2 48799,N1(C(c2n[nH]cc2Br)C(=O)NC(CC)(C)C)CCCCC12CCN(C)C2 48800,C1(COC)OCCC1C(=O)NCCOCCN(C)C(c1cc(C(C)(C)C)on1)=O 48801,c1(C(=O)N)ccc(C2CC2)o1.C1(CCNC)CCCO1.C1(=O)C(c2ccoc2)N1 48802,Cc1oc2cc(C(=O)NCCN(C)C(C3(O)CC3(C)C)=O)[nH]c2c1C 48803,N1(C(C2CN(C(C3CCCCS3)=O)CC23CCC3)=O)CCc2ccc(F)cc21 48804,C=CCC(C)(O)C(=O)NC(C)C(=O)NCC(C)(C)C1CCCO1 48805,C(=O)(C1CCCc2nc[nH]c21)N(C1CCCN(C(C(COC)(C)C)=O)C1)CCO 48806,CC(C)CC(CCO)NC(C1CCC(NC(c2ccnn2C(F)F)=O)C1)=O 48807,c1(C(=O)NCCC(C)N(C(C(CC)n2cccn2)=O)C)cc(C)nc(N(C)C)n1 48808,N1(C(=O)OC(C)(C)C)CCN(c2nccn2-c2ccccc2)CC1CO 48809,N1(C(CCC=CC(C)C)=O)CCC(NC(C2CCCC(O)C2)=O)CC1 48810,c1(CNC2CC(C(=O)NCc3cnc(Cl)nc3Cl)C2)c(F)cc(Br)cc1F 48811,N1(C(C(CC)=O)=O)Cc2ccccc2C1C(=O)Nc1nc2ccccc2nc1OC 48812,C1(NC(C(CC=C)OC)=O)CC2(C1)CC(C(=O)NCC1C(C)C1C)C2 48813,C1(CC)CC(O)CN1C(c1occc1CNC(=O)CSCC(N)=O)=O 48814,CC(F)(F)CC(=O)NCC1CCN(C(=O)CN2CCCCC2=O)C1 48815,C1(NC(CSCC)=O)CCCCC1CC(=O)NOCC(O)C(C)(C)C 48816,C(CN=C(NCc1ccco1)NC(c1ccccc1Cl)C)N(CC)CC 48817,C(CCC(C)(C)C(=O)NCc1cc(Cl)ccn1)NC(C(C(=O)OCC)CC)=O 48818,C(=O)(CCCC(=O)NCC1CC(CN)C1)C(c1cccc(NC(=O)C2CC2)c1)=O 48819,N1(C(c2cn(C)nn2)=O)CCCC2(CCC(NC(=O)C(=O)N=S(C)(C)=O)C2)C1 48820,CC1CC2(CCN(C(=O)CS(N)(=O)=O)CC2)CN1C(C1CNC(=O)O1)=O 48821,CC(CC(=O)NCC1CC1c1cncs1)n1ccnc1.C12(CC1)C(=O)N2 48822,Cc1n[nH]c(C)c1SCC(=O)NC1(CNC(=O)C(C)c2cncs2)CCCCC1 48823,CC1(NC(c2nnnn2Cc2cccs2)c2cnc[nH]2)CC2(C1)CC2(F)F 48824,C#CCC(CC#C)C(=O)NCC1(C)CN(C(C2(C)CCC2)=O)CC1C 48825,N1(C(c2n(CCC)ncc2)=O)CC2CC1CN2C(c1c(Cl)sc(C)c1C)=O 48826,N1(C(CSCC#C)=O)CCC=CC1C(N1CC(C(C)C)C1C(C)C)=O 48827,Cc1cc(C)c(C(=O)NC2CC3CC2N(C(C2CCC2(C)C)=O)C3)c(C)c1Br 48828,C1(C(=O)NCCC(C)(C)NC(C2CCCC2C(F)F)=O)(OCC)CCOCC1 48829,N1(C(C2(C)COC2)=O)CCCC(CCCCNC(C23CCCC2(C(N)=O)C3)=O)C1 48830,N1(C(C(=Cc2ccccn2)C)=O)CC2CCC(CNC(C3(F)CCOC3)=O)C2C1 48831,Nc1cc(C(=O)NC2CC(CNC(c3ccc(Cl)cn3)=O)C23CCC3)cnc1N 48832,C(=O)(CS(=O)(=O)C1CCCC1)NCC1(C)CCCN1C(C1CCCC12CC2)=O 48833,C=CCCCCC(=O)NC1CC(O)CN(C(c2ccccc2NC)=O)C1 48834,Cc1nc(C)c2c(C)c(C(=O)NCC(C)(C)NC(=O)C(C)C(C)O)sc2n1 48835,C(c1ccc(C)cc1)=CC(=O)NCCO.N12CCC(CC1)C2=O.C1(C)(CC)CC1N 48836,c1(C(=O)NC2CCC(CNC(C3CCCC(C)O3)=O)CC2)cc2ccccn2n1 48837,c1(CN2CC3(CC(C(N4CC(C(N)=O)OCC4)=O)C3)C2)c(Br)cc(F)c(F)c1F 48838,N1(C(C(C)=C(C)C)=O)CCC2(CCN(C(=O)C(=O)Cc3ccccc3)C2)C1 48839,C#CCCCCC(=O)NCc1cc(C(=O)NCC2(C3CC3)CCCO2)n(C)n1 48840,c1(C(=O)NC2C(C(C)C)CN(C(=O)C3=CCCS3)CC2)n[nH]c2ccccc12 48841,C1(CCC(=O)NCc2c(CC)c[nH]n2)CCCCN(C(=O)C2=C(Cl)CC2)C1 48842,C=C(Cl)CC(C(=O)NCCCN=[N+]=[N-])NC(c1ccncc1OC)=O 48843,c1(CNC(C2CCCSC2)=O)nc2c(s1)CCN(C(C1CCCN1C1CC1)=O)C2 48844,c1(CN2CC(C(=O)NC(C3(C(F)(F)F)CC3)=O)SCC2)nccc2occc12 48845,C1(NC(C2(OCC)CCC2)=O)CCN(C(=O)Cc2ccc(C)s2)CC1F 48846,CC(C)S(=O)(=O)C(C)C(=O)N1CC(CNC(c2cc3ccccc3[nH]2)=O)C1 48847,CCC(C)C(C(=O)N1Cc2conc2C1)N(CCOc1ccccc1)C 48848,C1(CNC(=O)NC2C(C)CCN(Cc3ccccc3)C2)CCc2scnc2C1 48849,C1(C(=O)NC(C)CCNC(c2conc2C(C)(C)C)=O)CCN(S(N)(=O)=O)CC1 48850,C1(OCC)CCCCC1OC(c1c(Br)cnn1C)=O 48851,C12(NC(c3c(C)nc(N(C)C)s3)=O)CCCC1CN(C(c1ccc(=O)oc1)=O)C2 48852,c1(CNC(CCOC(C)C)=O)ncccc1C(=O)NC1CCC1 48853,CCCCC(F)C(=O)N(C1CCCN(C(=O)C(C)(C)OCC)C1)C 48854,N1(C(C(CCC)(C)C)=O)CC2(C(=O)NCc3nc(C)ns3)CCC1CC2 48855,c1(NC2CCCN(C(CC(CCC)CC)=O)C2)nccc(C)c1[N+](=O)[O-] 48856,C1(C(=O)NCCOCCC#C)(CC)CCCN1C(=O)C=CCC 48857,CC1CCC(CNC(c2csc(=N)[nH]2)=O)CN1C(=O)CC1(O)CCCCCC1 48858,C(CCCCC(=O)NCC1(NC(c2csc(C)c2N)=O)CCC1)OCC 48859,CCC(CNC(c1cnn(C)n1)=O)(CC)NC(=O)Cn1ncnn1 48860,C(=O)(CC(F)(F)CC(=O)N1CC(NC(c2ccc(C)cc2)=O)C(C)C1)OC 48861,c1(CC)ccc(C=CC(=O)NC2(CNC(C3(C)CC3C)=O)CCCC2)o1 48862,C1(C(=O)NCCC(C)NC(C2(CCCC)CC2)=O)CCCCN1c1ncccn1 48863,C(C)(CCC(=O)N1CC2C(NC(C3CC(=O)N(C4CCCCC4)C3)=O)C2C1)OC 48864,CCC(CC(=O)NC(CN(C)C(c1cccc(C(C)C)n1)=O)CC)OC 48865,C(=O)(C1CCCn2nccc21)NCC(COC)NC(=O)Cc1ccc(F)cc1F 48866,N(C1CCc2cccc3cccc1c23)C1CCN(N(C)C)CC1.C=O 48867,c1(OC)c(C)cc(C(=O)NCCC(C)NC(C2(C(C)(C)C)CCC2)=O)cc1Cl 48868,C1(O)(C(C)NC(c2n(CC)nnc2)=O)CCN(c2ncncc2C#N)CC1 48869,c1(C(N2CCC(NC(C(CC)C)=O)C2Cc2ccccc2)=O)ncc(N)cc1Cl 48870,CCCC(C#N)C(=O)N1CCN(C(c2ccncc2Cl)=O)C(C2CCC2)C1 48871,c1(C(=O)NCC2N(C(CN(C)C(c3ccccn3)=O)=O)CC2)cnn(C2CC2)c1 48872,N1(C(c2ccc(CC)[nH]2)=O)CCOCC1CNC(=O)C(c1ccc(OC)cc1)O 48873,N1(C(CC(=O)NCC)=O)CCC2(CCC(CNC(=O)Cc3cnc[nH]3)O2)CC1 48874,C1(NC(C(C)CO)=O)CN(C(=O)C(C)(C)c2ccn(C)n2)CC2CCCC12 48875,c1(C(=O)NCC(CNC(C=C(C)C(C)(C)C)=O)O)cncc2nc(O)[nH]c12 48876,c12cc(nn1C)C(=O)N1CCC1C(=O)NC1(CCCC1)C(=O)OCC2.CCS 48877,C1(CNC(C2(COC)CC2)=O)CCN(C(c2ccc(C(C)(F)F)cc2)=O)CC1C 48878,CCCC(C)(O)C(=O)NCC1CCCN(C(c2cc(C(F)(F)F)nn2C)=O)CC1 48879,N1(C(C(Cc2ccoc2)NC(C2OCC(C)(C)C2)=O)=O)CCC(C2(C)CC2)CC1 48880,C1(CC(=O)N(C(C)C2CC2)CC)CN(C(=O)CCCC2CCCO2)CCO1 48881,c1(CC)ccc(OCC(=O)NC2(CO)CN(C(=O)CCn3cnnn3)C2)cc1 48882,c1(-n2ccc(C(=O)NCC(C)N(C(=O)CC(C)SC)CC)n2)ccc(F)cc1F 48883,C1(O)(CCNC(C2COCCC2(F)F)=O)CCCN(C(=O)CCc2cnoc2)C1 48884,C1(NC(Cc2ccc(C)nc2)=O)CCN(C(=O)CC2OCCCO2)CC1(C)C 48885,c1(COC)cccc(NC(=O)C(N2CC(CCN)C(C)C2)=O)c1 48886,N1(C(c2c[nH]cc(C)c2=O)=O)CC(NC(=O)Cc2nc[nH]n2)C2(CCCC2)C1 48887,C(=O)(C(F)(F)C(F)(F)C(F)(F)F)N1CC(O)(CCNC(C2CCN(CC)C2)=O)C1 48888,CC(C)C(C(=O)NOCCCN(C)C)C(C)NC(=O)CP(C)(C)=O 48889,C(=O)(C(F)(F)C(F)(F)C(F)(F)F)NC1C(NC(CC(CC)C(F)F)=O)COC1 48890,C=CC(C)(CCOC)C(=O)NC1CCC1C(=O)NCc1ncoc1C1CC1 48891,C1(C(=O)NCCN(C(C(CC=C)CC)=O)CCCCCC)CC2CCCC(C1)C2 48892,N1(C(C(C)NC(C)=O)=O)CC(NC(=O)C(C)Cc2c(C)n[nH]c2C)C(C)(C)C1 48893,c1(CNC(C(F)=CCC)=O)cc(C(N2CC(CO)(COC)C2)=O)no1 48894,c1(C(N(CCOCCNC(C(CCC)C#N)=O)C)=O)c(F)ccc(F)c1Cl 48895,C#CCCC(O)C(=O)N1CCC(F)C(NC(c2ccc(Br)c(O)n2)=O)C1 48896,Cc1cc(C(N2CCC(C)(C)C2CC(=O)NOCC(C)(C)C)=O)nc(O)c1 48897,C1(CNC(=O)CCN2CCCCC2)COCCN1C(=O)COC(F)(F)F 48898,C#CCCCCCCC(=O)NC(C1CC(NC(c2nccc(OC)c2N)=O)C1)C 48899,C1(CC=C)(C(=O)NC(C(=O)NCCSCCOC)C2CC2)CCOC1 48900,CC(C)CCC(=O)N1C(CNC(c2ccc(N3CCCC3=O)cc2)=O)CC2CC12 48901,N1(CC(=O)NC2CCCC2C(=O)Nc2ccc(F)cc2)CCC(C(=O)O)CC1 48902,C1(C(=O)NCCN(CCC)C(c2cc(N)ccn2)=O)(CC)CC(C)(C)C1 48903,c1(C(=O)NC2CCC(C)(CNC(CC3(CSC)CC3)=O)C2)cc(C#N)[nH]c1C 48904,C#Cc1ccc(C(=O)NC2CC(C)(NC(c3cccc(C(C)C)n3)=O)C2)cc1F 48905,N(C(=NCCCSC)NCC(O)COc1ccc(Cl)cc1Cl)CC(=C)C 48906,C=C=CCCC(=O)NC(C1CCN(C(c2nccc(C(F)(F)F)n2)=O)C1)(C)C 48907,c1(C(=O)NC(C2CCCN(C(c3csc(C4CC4)n3)=O)C2)C)c(O)cccc1Cl 48908,N1(C(CCC(=C)Cl)=O)CCC(C(=O)NC(C(C)C)C2CCC2)C(C)(C)C1 48909,CCCCCC(O)CC(=O)NC1CCC(NC(c2nc[nH]c3ncnc2-3)=O)C1 48910,C1(CNC(CN(C2CCC2)C)=O)CCC2(CCC2)CN1C(=O)C(O)C(C)(C)C 48911,Cc1cccc2c1C(NC(C1(N(C)C)CCSC1)=O)CC2 48912,c1(-c2nc(C)[nH]n2)ccc(C(N2CC(NC(c3cc(Cl)ns3)=O)C(O)C2)=O)cc1 48913,n1(C(C)C)ncc2cc(C(N3CC4CC3CN(C(C3CCSC3)=O)C4)=O)cnc12 48914,C1(CCCC)CCCCN1C(=O)CC1CCCN1C(=O)C(C(C)C)N(C(C)=O)CC 48915,c1(OC)cc(C(=O)NCC(CC(C)C)NC(=O)C=CC2CCOC2)n(C)n1 48916,N12CCCC(CC1)NC(C)CC2=O.C1(CC)CCC(CC(=O)OC(C)(C)C)CC1 48917,N1(C(=O)CC2(NC(=O)CN3CC4CC4C3)CCC2)CCc2ncncc2C1 48918,c1(C(=O)OC)cn2c(n1)CCCN2C(=O)Cc1nc(Cl)n(C)c1C 48919,CC(C)CCCCC(=O)N1CCCC1C1(O)CN(C(=O)C(=O)NC(C)C)C1 48920,C1(COC)(NC(=O)CCC2CCCO2)CCN(C(=O)C(OC)OC)C1 48921,C#CCC(C)(CC)C(=O)NCC1(O)CCN(C(=O)COCCCC)C1 48922,Cc1cc(NC(=O)CC2COCCO2)ccc1NC(=O)CNS(=O)(=O)C1CC1 48923,C(=O)(CCC1C(=O)Nc2ccccc21)N1CCC(NC(C2COC2)=O)C1 48924,c1(OC(C)C(=O)NCCC(C)N(C(=O)CNc2cccnc2)C)ccccc1Cl 48925,C(=O)(C1CCc2nccn21)NCC1CC(OC)CN1C(c1cc2occc2[nH]1)=O 48926,N1(C(=O)CCc2ccon2)CCC(NC(C2CC(n3ccnn3)C2)=O)CC(O)C1 48927,C(CCCC(=O)NOCCO)N(C)C(c1ccc(F)c(O)c1)=O 48928,C(C)(C)(CCCC(=O)N(CC(C)C(C)C)C)NC(c1c(C)ccnc1)=O 48929,C1(NC(c2c(OC)cnc(Cl)c2)=O)CC2CCC(C1)N2C(C1(C#N)CCC1)=O 48930,N1(C(c2cnc(SC)s2)=O)CC2(CCN(C(c3ccncc3N)=O)CC2)CC1C 48931,O=S(=O)(c1cnccc1N1CC2C3CCC(C3)C2C1)NC(CF)CF 48932,C1(NC(CC2(C)CCOCC2)=O)CC(C(=O)NCc2nnc(O)o2)=CC1O 48933,c1(N(C(CCO)C2CC2)C)ccc(S(=O)(=O)NC2CCOCC2)cc1Cl 48934,Cc1ccc2occ(C(=O)NCC3CN(C(C4C(C)C4C)=O)CC(C)(C)O3)c2c1 48935,N1(C(c2cc(C)c(F)c(C)c2)=O)CCN(C(=O)C(O)C(F)F)C2CCCC12 48936,c1(C(N2CCC(CCNC(C(C)c3ccco3)=O)C2)=O)ccc2nc[nH]c2c1F 48937,C1(CNC(N(CCCC)Cc2ccco2)=O)CCC(Oc2ccncc2)C1 48938,C(C)(CC(=O)N(C1CCN(C(=O)Cc2csc(NC=O)n2)C1)CCO)OC 48939,Cc1snnc1C(=O)NC(CC1CCOCC1)C(=O)NCCC(C)N(C)C 48940,C(=O)(CN1C(=O)CCc2ccccc21)NC(C)CCN(C)C(c1ccnnc1)=O 48941,CC1CCCn2ncc(C(=O)NCC3(O)CC(NC(c4ncc[nH]c4=O)=O)C3)c21 48942,N1(C(CCCOCC=C)=O)CCC(C)(CCNC(=O)COc2ccon2)C1 48943,C#Cc1ccc(C(C(=O)OC(c2conc2CC)=O)NC(=O)OC(C)(C)C)cc1 48944,CCCCCCCCCC(CC)C(=O)N1CC(C2CN(C(=O)CCCOC)C2)C1 48945,c1(CNC(=N)NC2CCN(c3ccc(F)cc3)C2=O)ccc(Cl)cc1Cl 48946,CCCC(CCCNC(=O)CCNC(=O)C1CC1)NC(=O)CC1CCCO1 48947,C1(C(=O)OC)CCC(C)N(C(=O)Nc2cnc(C(F)(F)F)cn2)C1 48948,c1(CC)cccc(NC(C2(C)CCCN2C(=O)C(c2ccc(C)o2)C)=O)c1F 48949,N1(Cc2n(CC)ncn2)CCCCC(NC(=O)CC2COC(=O)C2)C1 48950,C12(NC(C(CC=CC)NC(c3ccnn3C=C)=O)=O)CCC(C1)OC2C 48951,C1(C)(C(=O)NCC(C)O)CC12CCN(c1cc(C#N)ccn1)CC2 48952,N1(C(c2cc(CCC)on2)=O)CC2CCN(C(=O)CCCCC(C)=O)CC2C1 48953,N1(C(C=C(C)Cl)=O)CCCC(CN(C)C(C2CCC2C(c2ccccc2)=O)=O)C1 48954,Cc1ncccc1CCC(=O)N(CC(O)CN(C)C(C1C=CCS1)=O)C 48955,N1(C(CSCc2n(C)c(O)nn2)=O)CCC2(CC1)CC2(C)C(=O)NC1CC1 48956,C12(NC(C(CCSC)NC(C)=O)=O)CCCC1CN(C(c1ccoc1C)=O)C2 48957,C(=O)(CCCCCC(C)O)NCCC1(NC(c2c(CC=C)cccc2)=O)CCC1 48958,C(=O)(C(C)(C)CCC#N)N(CC(C)(C(C)C)NC(C=NOC)=O)c1ccccc1 48959,c1(CC)cccc(NC(=O)C(Cn2cncn2)NC(c2nonc2N)=O)c1C 48960,C(c1cc2ccccc2o1)=CC(=O)NCCC(C)N(C(C1C(C)C1C)=O)C 48961,O=C(C(=O)C(F)(F)F)NCc1cn(C2CCN(C(=O)C(O)c3ccsc3)C2)nn1 48962,N1(C(C=NOC)=O)CC2(CC(NC(c3cc(Cl)ns3)=O)c3nccn32)C1 48963,CC(C)(C)C(=O)NCCCC(=O)NCC1CC1CNC(=O)Cn1cccn1 48964,C1(CC(=O)NC2CCC(CNC(C(CC)N3CCCC3=O)=O)C2)CCCOCC1 48965,N1(C(C2(C3(C)CC3)CC2)=O)CC(C(=O)NC2(C)CCSC2)C2(CCC2)C1 48966,N1(C(C(COC)(C)C)=O)CC2(C)CC1(C(=O)NC(C)CCC1CCCO1)C2 48967,C(=O)(C1(C)CCOc2ccccc21)N(CCNC(C(CCCC)CC)=O)C 48968,C1(COC)CC(C(=O)O)N(C(=O)Cn2cc(C(O)C(C)(C)C)nn2)C1 48969,C(=O)(C(CCCC)NC(C1CCCS1)=O)N1C(C=C)CCC1 48970,Cc1nc(C(N2CCCC(NC(=O)C(C)Cc3ccnn3C)C2)=O)c(C)s1 48971,C#Cc1ccc(CC(=O)NC2CC(NC(C3CCCS3)=O)C2)cc1 48972,C#CCCCCCCC(=O)N1CC2(CC(CC(N3CCOCC3C3CC3)=O)C2)C1 48973,N1(C(C2C3COCC23)=O)CCC(CNC(CC2CCN(CCC)C2)=O)CC1 48974,C12(C(=O)SC)CCC(NC3CC(N(C(CC4C(C(=O)OC)CC4)=O)C)C3)(CC1)C2 48975,NC(=O)N=Nc1ccc(C(=O)NCC2CC(NC(C3CCCN3C=O)=O)C2)cc1 48976,n1(CC)nccc1C(=O)N(CCNC(=O)CN1CCCC1CO)CC 48977,Cn1nc(-c2nc(-c3ccc(C(F)F)cc3)nn2C2CSC2)c2c1CCCC2 48978,N1(C(CC(CNC(=O)CC=C(Cl)Cl)OC)=O)CC(C)(C2CCC2)C1 48979,N1(C(Cc2ccc(C)o2)=O)CC(NC(c2cncn(C)c2=O)=O)CC1(C)C 48980,c1(OC)ccc(F)cc1CNCC1CCCN1C(c1cccc(Br)c1OC)=O 48981,CC1CN(C(c2cnnn2C)=O)CCC1C(N1CCCC(C)(CO)C1)=O 48982,n1(CC=C)cccc1C(=O)NCC(C)NC(=O)Cc1ccoc1C 48983,Cc1noc2nc(C(C)C)cc(C(N3CCCC(S(N)(=O)=O)CC3)=O)c12 48984,C1(NC(C2CN(C)C(=O)C2)=O)CC2CCCC(C1)N2C(c1cccn1C)=O 48985,C1(C(N(C(CNC(C(C)=CC)=O)C)C)=O)CCCCCS1(=O)=O 48986,c1(C(=O)NCC2(C)CCCN2C(=O)C2=C(Cl)CCCC2)cc(F)cc([N+](=O)[O-])c1 48987,c1(C(N(C(C)CNC(=O)C(F)Cc2ccccc2)C)=O)cccn2ccnc12 48988,CN1CCn2ncc(C(N3CCCN(C(c4cc(Cl)ccc4F)=O)CCC3)=O)c21 48989,n1(CC)ncc(CNC(C2(C)CCN(C(=O)CN=[N+]=[N-])C2)=O)c1C 48990,CC(C)(CCCF)NC(C1(C2CCCN2C(=O)CC=C(Cl)Cl)CC1)=O 48991,C1(C(=O)NCCOC(C)=O)CCN(C(c2cc(C)c(C)cn2)=O)CCO1 48992,c1(C(N2CCC(O)(CNC(CN3C(C)CCC3)=O)C2)=O)cc2scnc2[nH]1 48993,Cc1ccc(C(c2nnnn2CC2CC2)NCCc2scnc2C)s1 48994,N(C(=NCCOCC1CC(SC)C1)NCC(C)C)C1CCN(C(=O)OCC)CC1 48995,C1(C(C)(C)C)(CNC(CC=C)=O)CCN(C(=O)Cc2ccnc(OC)c2)C1 48996,N1(C(COc2ccc(CC)cc2)=O)CCCN(CCNC(=O)C(F)CC)CC1 48997,C(=O)(CCCCC(C(F)(F)F)NC12CC1CN(C(=O)OC(C)(C)C)C2)OC 48998,N1(C(C(C=C=C)C)=O)CCCN(C(c2cnc(C)s2)=O)CC1C(C)C 48999,C#Cc1ccccc1CC(N1CC(CNC(=O)CC(=C)Br)CC1C)=O 49000,c1(CN(CCCNC(c2ncccc2C2CC2)=O)CC)ccc2n[nH]cc2c1 49001,NC(CCC1CC1)C(=O)N1CC(N2CCCC2)C1 49002,Cn1cc(NC(=O)C(=O)NC2CCCC(CC(=O)NC3(CO)CCC3)C2)c(O)n1 49003,C1(C(=O)NCC(C(=O)OC)Cc2cccc(C)c2)CC2CNCC1O2 49004,C(C(C)(C)CC(=O)N(CCCNC(C1CCCN1S(C)(=O)=O)=O)CCO)OC 49005,c1(OCC(N2CC(CCC(=O)NCC)OCC2)=O)c(C)cccc1Br 49006,c1(NC(C23C(CN(C(c4cc(OC)c(I)cc4)=O)C2)C3)=O)ccc(F)cc1C#N 49007,n1(CC)c(C(=O)N(C2CCCCC2)CCNC(=O)CCOC2COC2)cnc1O 49008,C1(C(N)=O)CCCC(C(N2CC(OCCNC(c3cnnn3C3CC3)=O)C2)=O)C1 49009,C(=O)(C(C(C)C)C(C)C)NC1(CCNC(c2c(C)cc[nH]2)=O)CCC1 49010,N1(CC(C)NC(C2ON=C(C)C2)=O)CCN(C(=O)C=C(Cl)Cl)CC1 49011,C(C#CCN=c1[nH]ccc(=NC2CCN(C3CCCCC3)C2)[nH]1)OC 49012,Cc1cc(Br)cc2c1CN(C(=O)Nc1cnc3c(c1)CCOC3)CC2 49013,CC1ON=C(C(=O)NCC2CN(C(=O)C(N)=O)CCO2)C1C 49014,CCC(C)C(C(=O)NC(C)CN1CCN(C(=O)CC2CC(C)C2)CC1)NC(N)=O 49015,N1(C(C(C)C2CCC2)=O)CC2CCC(C1)C2CNC(=O)C(O)CC(F)(F)F 49016,C1(C(=O)NCC2=NOC(C)C2)CCCCCC1NC(c1nccs1)=O 49017,C12(NC(c3cnco3)=O)CCCC1N(C(c1cc(-c3ccccc3)co1)=O)CC2 49018,C12(NC(CCS(C)=O)=O)CCOCC1CN(C(C1(c3cc[nH]n3)CC1)=O)C2 49019,C=CCC(C(=O)NC(C1(O)CN(C(c2cccc3ncsc23)=O)C1)C)C(C)C 49020,N1(CC(=O)NC2C3CN(C(c4[nH]n(C)c(=O)n4)=O)C2C3)CCC(=O)NC1=O 49021,c1(C(N2CC(NC(c3c(CC)onc3)=O)C3(C2)CC3)=O)ccc2n[nH]cc2c1F 49022,C1(C(N(OC)CC2CC2)=O)CC(C)CN(C(=O)C#CC(C)(C)C)C1 49023,C1(C(N2C(CNC(=O)Cc3cccnc3)COCC2)=O)CCc2ccccc2C1 49024,CC1CN(C(=O)C(F)=CCCF)CCC1N=c1cc(C(N)=O)nc(Cl)[nH]1 49025,CS(=O)(=O)c1cc(C(=O)NC2C=CCN(C(=O)Cc3nc[nH]n3)C2)cs1 49026,c1(C(=O)NC2(c3ccccc3)CCN(C(C(C=C)O)=O)C2)cc(C)nnc1O 49027,C1(C(=O)NCC(CC)NC(=O)CCc2cn(C)nn2)CCCC1c1ccccc1 49028,C(=O)(C(C)(C)C#N)NCCC1(C(=O)NC(C(C)C)CO)CC1 49029,c1(C(N(C2CCN(C(C3(O)CC3(C)C)=O)C2)C)=O)cc(C(F)F)cc(Cl)c1 49030,N1(Cc2c(C)nccc2)CC2(CCC(C(=O)Nc3oncc3C#N)O2)C1 49031,Cc1nn(CC(F)(F)F)cc1C(N1CC2C(NC(=O)CC3CSCCS3)C2C1)=O 49032,C(CCCCC(=O)N(C(C)CNC(C1CC(OC)C1)=O)C)=CC 49033,C(C(C)(CO)NCCCNC(=O)COc1cccnc1)NC(=O)OC(C)(C)C 49034,CC(N=[N+]=[N-])C(=O)N1CC(CC(F)C(=O)NCC(c2ccccc2)F)C1 49035,CC1CCCC=C1C(=O)NC1CCN(C(=O)CC(F)(F)C(F)F)CC1(C)C 49036,c1(OC)cc(C(=O)NCC(O)CNC(C23CC(CO)(C2)OC3C)=O)cc(OC)n1 49037,c1(CNC(C(N2CCC(CCC(=O)OCC)C2)=O)=O)ccc(F)cc1CC 49038,N1(C(C2N(C(c3c(C)c[nH]c3)=O)CC2)=O)CCC2(CCCO2)C1 49039,C=CC1CCN(C(C2CCN2C(=O)C(C)SCC)=O)CC1 49040,C(CCC(C)C)(C(=O)N(C)CCc1ncccn1)NC(C1C(CCC)CCC1)=O 49041,CCS(=O)(=O)C=CC(=O)N1CCC(C)N(C(c2cc[nH]c2C2CCCC2)=O)CC1 49042,C1(OCC)CC(CNC(=O)CNC(=O)Cc2cc[nH]n2)C1 49043,C(c1cn(C)cn1)=CC(=O)NC(C(=O)NC(c1onc(C)n1)CO)CO 49044,C(=O)(CC1=NN(C)C(=O)C1)NCC1ON=C(C(=O)N(C2C(C)C2)C)C1 49045,N1(C(c2c(CC)cns2)=O)CC(O)CCC1C(=O)NCCn1ncnn1 49046,C(=O)(NNC(=O)C1CCCS1)NC(Cc1cc(C)[nH]n1)C 49047,C1(S(N)(=O)=O)(C(N(CCCNC(c2cc(C3CCOC3)[nH]n2)=O)C)=O)CCCC1 49048,N1(C(C(CC)(C)O)=O)CCCCC2(C1)CN(C(c1nn(C)cc1Cl)=O)C2 49049,c1(C(=O)NC(CCNC(C(CCCC)O)=O)(C)C)cc(=O)c2cc(F)ccc2o1 49050,C1(C2CCCN(C(=O)CCc3ccsc3)C2)(NC(=O)C(O)Cc2cnc[nH]2)CC1 49051,Cc1cc(=NCC2CC(C)CC(C)C2)[nH]c(=NCCS(=O)(=O)C(F)F)[nH]1 49052,N1(C(C2(COCC)CC2)=O)CCOCC(C(N2CCC(C)(C)C2)=O)C1 49053,C1(C(=O)NCC(CN(C)C(c2c[nH]cc2C(C)(C)C)=O)O)C2CCCC12 49054,CCCCCC(O)C(=O)N1C(C)C2CC1C2NC(C1(C(F)(F)F)CCCCC1)=O 49055,c1(C(N(C2CCCN(C(=O)C=C3CC3)CC2)C)=O)ccc(N)c(Br)n1 49056,CCC(C)(C)CC(=O)N1CCOC(C)(CNC(=O)CC(C)OC)C1 49057,c1(C(=O)NCC2(NC(c3ccc4c(c3)NCC4)=O)CC2)cnc2[nH]ccc2n1 49058,N1(C(C(C2CCOCC2)C)=O)CCOCC(CNC(C2CC(=O)N(C)C2)=O)C1 49059,c1(OC)ncc(Br)cc1CN(C1CCN(C(C2CCN(C)C2)=O)C1)C 49060,C=CCC(CC(C)C)C(=O)N1CC(NC(C2(C#N)CC(C)C2)=O)CC(C)(C)C1 49061,C1(C2CCOCC2)(C(=O)NCC2N(C(CCCN(C(C)C)C)=O)CC(O)C2)CC1 49062,N1(C(CCCC)=O)CC(=O)NCC1C(N1CCCC(C)(CCC)C1)=O 49063,Cc1sc(O)nc1C(=O)NCCC1CCCN(C(C2(N3CCCC3)CC2)=O)C1 49064,CC(C)CC(C)CC(=O)NC1(C)CCN(C(C2(C#N)CC2)=O)C1 49065,c1(C(N2CC(OC)(CNC(c3ccoc3)=O)C2)=O)cnc2ncnn2c1C(C)C 49066,C1(C(=O)Nc2cnn(C)c2Cl)CNC(=O)CN1C(c1n[nH]c2c1CCC2)=O 49067,c1(C(N(C)CCOCCC(=O)NC2CCCCC2(F)F)=O)cccc2occc12 49068,C(C(C)(O)CC(=O)NC(CNC(c1cc(C(C)C)ccc1C)=O)CC(C)C)OC 49069,N1(C(C2(F)CCN(C(Cc3ncc(C)nc3)=O)C2)=O)CCOC(C)CC1 49070,CC#CCCCC(=O)NC1CCC1CNC(c1ncn(CC)n1)=O 49071,CCC(CC(=O)NC(C)CC(C)NC(c1c(C)cncc1C)=O)C(C)(C)C 49072,C(=O)(CC(C)C)NC(C(=O)N(CCOC)CCOC)c1cccs1 49073,C1(C(=O)NC(C2CCCC2O)C)C=CCN(C(=O)CC2CC(=O)NC2=O)C1 49074,N1(C(=O)OC)CCCC1C(=O)N(C1CC(NC(c2cn(C(C)C)cn2)=O)C1)C 49075,c1(CN2CC(CNC(C3(CC)CCNC3=O)=O)OCC2)c(F)cccc1Cl 49076,Cc1ccc(C)c(C(=O)NC2CC3CC2N(C(C2(O)CC2(C)C)=O)C3)n1 49077,C(=O)(C#CC1(C)COC1)N1C(C)CCC(C(=O)NC(CC)CO)C1 49078,C1(CNC(=O)CCCC2CCC2)CC2(CCC2)CN1C(=O)Cc1ccncc1Cl 49079,N1(C(CNC(CCC)=O)=O)CC(F)CC1CNC(c1c(C)ncn1O)=O 49080,c1(C(N2CCC(C)(CCNC(CCOC(C)=O)=O)C2)=O)cnc2ccncc2c1 49081,n1(CCC(=O)NC2CC(NC(CN3CCC(C)(C)C3)=O)C2)cc(S(N)(=O)=O)cn1 49082,C(=O)(NNc1cc(F)cc(F)c1)N(CCN)CCc1ccccc1 49083,c1(CNC(c2csc(CO)n2)=O)cccc(NC(C2CCC(O)C2)=O)c1 49084,N1(C(C2N(C(CNC(=O)NC)=O)C(C(C)C)CC2)=O)CCOCC1C(N)=O 49085,CS(=O)(=O)c1cscc1C(=O)NCC(CO)NC(C1(F)CC=CCC1)=O 49086,c1(C(=O)NC2CC(CCC(=O)N3CC(C(F)(F)F)C3)C2)cnn2ccccc12 49087,c1(C(C)C)cc(S(=O)(=O)N2Cc3nncn3C(C)C2)cc2ccccc12 49088,CC(C)CC(C)(O)C(=O)N1CCCC(CNC(=O)C#CC2CCC2)C1 49089,Cn1ncc(CC(=O)NC2CCC(NC(c3ccon3)=O)C2)n1 49090,c1(OC)ccc2c(c1)C(NC(=O)NCC1(SC)CC(C)(C)C1)CCC2 49091,CCC(C#N)C(=O)NC1CC(CNC(=O)C(c2ncccc2F)(F)F)C1 49092,C(=O)(C(CNC=O)c1ccccc1)NCC#CCNC(C(C)C1CC1)=O 49093,CC1(C(N2CCCC(O)C2)=O)CCCN(Cc2nc(Cl)sc2Cl)C1 49094,c1(C(=O)NC(CN(C(c2c(CC)non2)=O)CC)CC)coc2ccccc12 49095,c1(C(C(=O)NCCOCC)N(c2ncc(Cl)s2)C)ccc(C#N)cc1 49096,c1(C(N2CC3(C(NC(C(CCC)C)=O)CC3)C2)=O)ccc2cc(C)cn2c1 49097,n1(CCC(=O)NC2CN(C(c3c(C)ncnc3)=O)C2)cc([N+](=O)[O-])nc1C 49098,c1(C(N2C3C(C(=O)NC4CCN(CC)C4=O)C(C3)C2)=O)ncc2ccccn12 49099,C1(CN(C(COCC(=C)C)=O)C)C2CN(C(C3CC3c3ccc(Cl)cc3)=O)CC12 49100,N1(C(C(CC)SC)=O)CC(CNC(=O)CSC(F)F)C(F)(F)C1 49101,C(C(=O)N(C1CCN(C(c2cnn(C3CCC3)c2C)=O)C1)C)(C(C)C)SC 49102,c1(NC2CCC(SCC)C2)ccc(S(=O)(=O)NCc2nnc(C)o2)cc1C#N 49103,C#CCC(C)(C(=O)Nc1nccnc1CC)NC(=O)C(=O)NC(C)C 49104,C1(C(N(CCN(C(C(CC)(C)O)=O)CC)C(C)C)=O)CCc2ncnc(C)c2C1 49105,C(=O)(C(F)(F)C(F)(F)F)N1CC(NC(c2c(C)ncs2)=O)C(C)C1 49106,C(=O)(C(C)(C)C(C)O)NCc1ccc(N(C2(C3CCCCO3)CC2)C(C)=O)cn1 49107,c1(OC)ccc2cc(C=CC(=O)NC3CCN(C(=O)C(C)C)C(C)C3)ccc2c1 49108,C#Cc1ccc(CNC(C2(N(C)C(C3CCSC3)=O)CC2)=O)cc1 49109,C#Cc1ccc(C(=O)NC(C(N2CC3CC3(COC)C2)=O)C2CCC2)c(C)c1 49110,CCCCCS(=O)(=O)CC(=O)N1CCCC2(NC(c3ccc[nH]3)=O)CC2C1 49111,O=C(CCC(CF)CF)NC1COCC1CNC(c1cncc([N+](=O)[O-])c1)=O 49112,CCCCC(C(=O)NC1CCC(CCC(=O)N(CCC(=O)OC)CC)C1)C(C)C 49113,C(=O)(CS(=O)(=O)C(C)C)N(C)CC1CCN(C(c2c(CCC)nco2)=O)CC1 49114,N1(C(c2cnn(CC)c2C)=O)CCN(C(=O)Cc2ncc(C(C)=O)s2)C(C)C1C 49115,C(N(C)N1CC2(C=Cc3ccccc3O2)C1)C1(SCC)CC1 49116,c1(NC2CC(C)N(C(c3cccc(C4CC4(F)F)c3)=O)C2)ncc2ncnc-2[nH]1 49117,c1(C(=O)NCCCCC(CO)NC(C2CC(OC)C2)=O)cccc2c1OCC2C 49118,C1(NC(=O)C(F)OC(F)(F)F)(CO)CCCN(C(C2(Cl)CC2)=O)C1 49119,c1(C(=O)NC(C(=O)NC2(C(C)C)CC2)Cn2cncn2)c[nH]nc1[N+](=O)[O-] 49120,c1(OC)nc(N2CC3(CCN(C(c4cncc(C)n4)=O)C3)C2)ncc1C#N 49121,NCC(Cc1ccccc1)C(=O)N1CCCCC1c1ccc(-c2ccccc2)o1 49122,N1(C(C2=NOC(C)C2)=O)CC2CCOC2(CNC(=O)CCC(=O)c2ccc[nH]2)C1 49123,Cc1nc(CC(=O)NCC(CO)NC(=O)CCC2CCC(=O)N2)co1 49124,N1(C(c2c(C(=O)OC)cco2)=O)CCC2(NC(C3CCCOC3)=O)CCCC12 49125,c1(OC)ccc(C(N2CCC(NC(c3ccnc(Br)c3)=O)C(O)C2)=O)cc1O 49126,C(=O)(CC(O)CN(C)C)N(C1CCN(C(c2ccc(-c3cc[nH]n3)s2)=O)C1)CC 49127,C1(CC(=O)NCC(C)N(C(c2cccc(C3CCC3)c2)=O)CC)CC(C)(C)CO1 49128,c1(C(=O)NC(CC)CNC(=O)CC2COC(=O)C2)nnc2n1CCCCC2 49129,C(c1ccc([N+](=O)[O-])s1)=CC(=O)NC1CC(O)(CNC(CS(N)(=O)=O)=O)C1 49130,C(C(=O)NNC(=O)c1ccc(I)c(I)c1)c1ccc(C)cc1 49131,CC1CCCCC1(CNC(c1ccc(=N)[nH]c1)=O)NC(C1(CN(C)C)CC1)=O 49132,N1(C(C=CSC)=O)CC(CO)C(C(F)(F)F)C1.c12cc(on1)CNC(=O)C2 49133,c1(OC)ccccc1CC(=O)NCC1(F)CC(NC(c2conc2C2CC2)=O)C1 49134,C1(NC(CCOC(CC(C)C)C)=O)CN(C(=O)COC(C)(C)C)CC1C(F)F 49135,N1(C(c2c(C)ncn2C)=O)C2CCC1CN(C(=O)Cc1ccncc1Cl)C2 49136,CC1CC(CNC(C2(C)CCSCC2)=O)CN(C(=O)CCc2cn(C)nn2)C1 49137,C1(CNC(C=CCC)=O)CCCC2CN(C(c3ccc(CSC)cc3)=O)CC12 49138,N1(C(C(COC)OC)=O)CC2CC(NC(c3sc(C(C)C)nc3C)=O)CC1C2 49139,N1(C(C(CC)C)=O)CCN(C(C23COCC(C2)C3)=O)CC1CC1CC1 49140,c1(CC)cc2c(CC(=O)NCC(C(C)C)NC(=O)CC3COCCO3)csc2s1 49141,c1(NCC2CCCN(CCC(=O)OC)C2)cc(OC)ccc1[N+](=O)[O-] 49142,C1(NC(c2c(OC)cccc2)=O)CCCN(C(=O)C(=O)CC(C)C)C1C 49143,C1(CNC(CC2ON=C(C)C2)=O)CCC(N(C)C(c2cncs2)=O)CC1 49144,c1(C(N2C(COC)(CNC(c3occc3C)=O)CCC2)=O)csc(=NC2CC2)[nH]1 49145,C(=O)(C1CCSc2ccccc21)NC(CC=C)CNC(=O)CCCC(=O)OCC 49146,C(=O)(CCC(C)(C)C)NC1C(C)CN(C(C2(N(C)C)CCCC2)=O)C1 49147,C(=O)(C#CC1CCOC1)NCC(CC)NC(c1ncsc1S(N)(=O)=O)=O 49148,c1(C(=O)OC)ncc[nH]c1=NCC1(CNC(c2cnc(C(C)C)s2)=O)CC1 49149,C1(CNC(C2(CC)CC2)=O)(C)CCCCC1.C1(N)CCSC1.C1(=O)C=CC(=O)N1 49150,N1(C(C2C(NC(=O)CC3CC4(CC4)C3)C=CCC2)=O)CCc2ccsc2C1 49151,c1(C(N(CCOC)CCNC(C2CC(C)(C)C2)=O)=O)cc(F)ncc1OC 49152,c1(C(=O)NCC2CCC(C(N3CC(C)(O)C3)=O)O2)occ2c1CCC2 49153,c1(NC(C(c2ccco2)NC(COC(CC)CC)=O)=O)ccc(F)cc1O 49154,N1(C(c2cc(CC)[nH]n2)=O)CCCC(CCC(=O)NCC(C)C(C)C)C1 49155,C1(C)(C(=O)NCC2N(C(c3n(CC)cnn3)=O)CCC2)CCCN1C(=O)C1CC1 49156,Cc1[nH]c(C#N)cc1C(=O)NC1(C)CC(NC(C23CCCC2C3)=O)C1 49157,c1(OC)cnc(C(=O)NC(CNC(=O)CCc2nc(C)no2)C(C)C)cn1 49158,CC(C)(C)C(O)C(=O)N1CCCCCC1CNC(c1cnc2sccn12)=O 49159,CCCC(O)C(=O)N1CCC(C)(NC(=O)Cc2nc(C)sc2C)C1 49160,c1(C(=O)NCC2CC(CNC(=O)COC3CCOCC3)C2)ccc2ccoc2c1 49161,CCC(CC)(CC)C(=O)N1Cc2occ(C(=O)NCC3CC(F)(F)CO3)c2C1 49162,CC1(C)C(NC(C2(CO)CCOCC2)=O)CC1CNC(=O)Cc1cncnc1 49163,C1(C(N(C)Cc2cnc(C)s2)=O)CCC(C)(C)N(C(c2c[nH]nc2Cl)=O)C1 49164,N1(C(c2cc(C)on2)=O)C(CN(C)CCO)CC2CC12 49165,C(=O)(C1=CCC2CCC1N2C(c1n[nH]c2ccccc12)=O)NCCCC(C)CO 49166,C1(CNC(CCCCOCC)=O)N(C(=O)C=C2CCC(C)CC2)CCCC1(C)C 49167,C12(CNC(c3ccc(OC)nc3)=O)CCCN(C(=O)CCCc3nccs3)C1C2 49168,C(=O)(C(O)CC(C)(C)C)NC(C(C)NC(=O)CSc1nccn1C)C 49169,C12(CC(=O)NCCSCC#C)CCC1CN(C(C1(OC)CC(C)(C)C1)=O)C2 49170,CCC(C)C(O)C(C)C(=O)N1CCN(CCNC(c2ccc([N+](=O)[O-])o2)=O)CC1 49171,C#Cc1cnn(CC(N2CCC(NC(=O)CCc3cc(C)on3)C2CC)=O)c1 49172,C(CC(C)N(C)CCOCCCCC)OCCOC 49173,C=C(C)C(CC(=O)N1CCCCC1CNC(c1csnc1C(=O)OC)=O)OCC 49174,C(=O)(C(C(C)C)NS(N)(=O)=O)N1CCC(CNC(C(CSC)O)=O)C1 49175,Cc1cncc(CN(C2CCCC2c2nc[nH]n2)C(C23CC(CC(F)F)(C2)C3)=O)c1 49176,O=C(CC1CC(NC(c2ccc([N+](=O)[O-])cc2)=O)C1)N=c1cc(C2CCOC2)[nH][nH]1 49177,C(=O)(C(C)C(C)S(C)(=O)=O)N(CCCNC(c1ccc(NC(=O)OC)cc1)=O)C 49178,C(=O)(C1CCc2ccccc21)NC(C(C)(C)NC(Cc1c(C)con1)=O)C 49179,C1(C(N(C)CC2(C)CCC2)=O)CCCN(C(C2(C)CCCOC2)=O)C1 49180,C1(C(=O)NCc2c(C(=O)NC3(C(C)(F)F)CCC3)c[nH]n2)CCNC(=O)C1 49181,c1(CCC)cc(C)c(Nc2cccc(NC(C)=O)c2)cn1 49182,N1(C(=O)CCOC2CCC2)CC2(CC2)CC1CNC(C1(CC2CC2)CCC1)=O 49183,Cc1cccnc1C=CC(=O)NCC(C)CN(C(=O)CN1CCC(F)CC1)C 49184,CS(=O)c1ccc(C(N2CCC(C)(C)C2CNC(=O)Cc2nc[nH]n2)=O)cc1 49185,C1(O)(CCNC(c2n[nH]c(CC)c2Cl)=O)CCCN(C(=O)C(C)(C#N)CC)C1 49186,C(=O)(C1COc2ccc(Cl)cc21)NC1C=CCN(C(COC2(C)CCC2)=O)C1 49187,CC(C)(O)CCCNC(=O)CC1CCN(C(C2(CF)CC(=O)C2)=O)CC1 49188,c1(OC)ccc(C2(C(=O)NC3CN(C(C4CC(OC)C4)=O)C3)CCC2)cc1 49189,C(C1=NOC2(CCC2)C1)NC(C(C)CNC(=O)C(C)NC(N)=O)=O 49190,c1(CCC(=O)NC(C2CCCN2C(c2cnc[nH]c2=N)=O)(C)C)ccc(Cl)nc1 49191,C1(C(N2C3CN(C(c4ccc(N)cn4)=O)C(C3)C2)=O)CC(c2ccncc2)=NO1 49192,NS(=O)(=O)CCCC(=O)NCC1CCCCN(C(C2CCCCO2)=O)C1 49193,N1(C(C(CC)OC)=O)CCOC(C2CN(C(=O)CCc3cc(C)no3)C2)C1 49194,C(=O)(CCCC(=O)NCCNC(C)=O)N1CCN(C(C(CN(CC)CC)F)=O)CC1 49195,C(=O)(C(C)(C)C(=O)N1CC2(C(N3CC(F)C3)=O)CC1CO2)N(C)C 49196,C(F)(F)(C(=O)NOC(c1ccccc1)C)C12CCC(OC)(C1)C2.c1(C)ccccn1 49197,CN1CC(C)(C(=O)NCC2CN(C(=O)CCc3cnc(O)[nH]3)CCO2)CCC1=O 49198,C(N=c1[nH]cnc2c(Br)cccc12)C1CN(C(c2c(OC)nsc2)=O)C(C)C1 49199,C1(NC(C2CCC=CCCC2)=O)CCCOC12CCN(C(c1cnoc1)=O)CC2 49200,n1(CC(=O)NC2CCC(CNC(CC3CC(CC)C3)=O)CC2)ccc(O)nc1=O 49201,C(C)(C)(CCC(=O)NC(Cc1ccco1)C(N1CCCC(CN=[N+]=[N-])C1)=O)OC 49202,N1(C(=O)CSCC(F)(F)F)CCN(C(C2(Cc3cccs3)CC2)=O)CC1CCO 49203,C1(C(=O)NCCC(CC)CO)CN(C(C2CC(C)CCO2)=O)CC(C)(C)C1 49204,c1(NC(=O)NC2CCN(C3CC3)C2)ccc2c(c1)C(=O)NCCO2 49205,Cc1c(NC(=O)NC2OCC3CCCC23)cccc1N1CCNC1=O 49206,C1(CNC(c2cc(C)ncc2C)=O)CN(C(=O)C(C)N(C)C)C2(CCC2)C1 49207,O=S(=O)(c1[nH]c(=NCC2CC2C2CCC2)ccc1Br)N1Cc2cccc(Cl)c2C1 49208,c1(C(N(C2CCN(C(C(CC#C)O)=O)C2)C)=O)cc(S(=O)(=O)NC)c[nH]1 49209,CC(C)C(C(=O)NCc1cnn(C(C)C)c1)c1ccnc(N(C)C)c1 49210,Cc1nccnc1N1CCN(c2nnc(C3CCOC3)n2CC2CC2)CC1 49211,C1(C(CC)CC)C(=O)OCCN1CC(CCCC)CC.C(CCF)CC 49212,C1(NC(=O)C2=CCCC2)CC(O)CN(C(C2CC(O)(c3ccccc3)C2)=O)C1 49213,CC(C)(C)C(CCc1ccc(F)cc1)C(=O)N1CCNC2(CC2)C1 49214,C(=O)(C(C)(C)Cc1cccc(Cl)c1)N1CC(F)(CNC(C2C(CC)C2)=O)C1 49215,C1(NC(C2(C)CC2(Cl)Cl)=O)CCCN(Cc2cn(Cc3csc(Br)n3)nn2)C1 49216,N1(C(C(CC#C)C)=O)CCC(NC(=O)C2=C(C)OCCS2)C(F)(F)CC1 49217,c1(-c2cn(CCN(C(=O)C(c3cccnc3F)(C)C)C)nn2)cnccc1Cl 49218,c1(C(=O)NCC2N(C(CCN(CC)CC)=O)CCN(C)C2)cc2ncccc2o1 49219,c1(C(=O)NC2CN(C(c3cc(CC)c(CC)o3)=O)C2)c(N)ccc(F)c1F 49220,N1(C(C=CCC)=O)CC2CC(NC(c3cn(C)nc3-c3cccnc3)=O)C1C2 49221,C(C)(c1cccnc1)=CC(=O)N(C(C)CNC(C1(C)CC=CCC1)=O)CC 49222,C=CCC(CC(=O)N1CCSC(C)(C)C1)NC(C1CC2(CCO1)CC2)=O 49223,CCN=c1cc(C(N2CCCC(NC(=O)C3=C(C)CC3)C2)=O)cc[nH]1 49224,C1(C(=O)NC(c2ncnn2C)C)CCN(C(=O)CN2CCSCC2)C(C)(C)C1 49225,CSC1=C(C(=O)N2CCN(C(=O)CCC#N)CC2C2CC2)CCCC1 49226,C1(CC(N2CC(C(N(c3ccn(C)n3)CC)=O)C2)=O)CCCC(C)O1 49227,N1(C(CCCCC(N=[N+]=[N-])=O)=O)CCC2(CCC2)C(CNC(C2C=CCC2)=O)C1 49228,N1(C(C(C(C)(C)C)(C)C)=O)CCC(NC(c2ccc(N)cc2O)=O)C(F)(F)CC1 49229,c1(C(=O)NCCC(C)(C)NC(c2cc(OC)no2)=O)ncccc1SC 49230,N1(C(CCSCC)=O)CCN(C(C2(C)CC2)=O)CC1c1nccn1C 49231,C1(OC)CC(CCN(C)C)N(C(C2CCN(c3ccncc3)C2)=O)C1 49232,c1(CCC(N2CCC(c3cn(CC=C)nn3)C2)=O)cc(OC)c(Cl)cc1OC 49233,C(CCCC(=O)NC12CCC1CN(C(=O)CC(C)n1ccc(C)n1)C2)(OC)OC 49234,N1(C(C2(C)COCCO2)=O)CC2=C(C1)CN(C(=O)CNC(c1ccco1)=O)C2 49235,N1(C(CCc2ncn(C)c2)=O)CC(F)CC1CC(=O)NC1(n2cccn2)CC1 49236,c1(C(N2CCC(N(C(=O)CSc3nncs3)C)C2)=O)ncc(C(F)F)cc1F 49237,c1(Cn2cc(C3CCN(C(c4nc(CCC)oc4)=O)C3)nn2)cc(F)cc(Cl)c1 49238,N1(C(C2N(N=O)CCC2)=O)CC2CCCC(C1)N2C(c1ccn2ccsc12)=O 49239,c1(OC)ccc(C(=O)CSC(C(C)C)C(C)(C)O)c2c1C(=O)CO2 49240,c1(C(=O)NCC(CN(C(C(C)(C)OC)=O)C)C)cccc2nn(C)nc12 49241,N1(C(C2(OC)CC2)=O)CCC2(CC1)CCN(C(c1c(C)ccnc1Cl)=O)CC2 49242,n1(CC(=O)N(CC(CN(C(CC(C)n2ccnc2)=O)C)O)C)cnc([N+](=O)[O-])c1 49243,c1(CC(=O)NCC2(CC)CCOC2)ccc(NC(=O)C(C)CC2CCCC2)cc1 49244,Cc1nc2cccc(C(=O)NCC34CCCC3CCN4C(c3cnsn3)=O)c2[nH]1 49245,N1(C(C2CC(CC)C2)=O)CCCC(O)(CN(C(=O)CCC(C)C)C)C1 49246,C1(NC(CC(=O)OCC)=O)CN(C(C2CC(=O)NC2(C)C)=O)CC2(CCC2)C1 49247,c1(C(N2C(CCCC)CN(C(=O)CC(C)C(C)C)CC2)=O)cc(F)cc(N)c1F 49248,[N-]=[N+]=NC1COCC1NC(C1CN(C(C2(N3CCCC3)CC2)=O)CC12CC2)=O 49249,N1(Cc2cc(OC)cc(Cl)c2)C(=O)C2C(C)CCCN2C1=O 49250,C1(C(=O)NCc2cnc(C)s2)CN(C(=O)CC2CCOC2)CC1(F)F 49251,c1(C(N2C3C(NC(C4CCN(CCC#C)CC4)=O)C(C3)C2)=O)c(C)ncnc1O 49252,c1(C(=O)NCC2CCCN(C(c3c(OC)ccs3)=O)C2)ccc([N+](=O)[O-])c(F)c1 49253,c1(NC(C2CCN2C(=O)C(c2ccccc2)=O)=O)c(Cl)ccnc1Cl 49254,N1(C(=O)Cc2c(F)cccc2Cl)CC2CCC(C1)N(C(c1ccns1)=O)C2 49255,C1(NC(c2cccc(C)n2)=O)CC2CCC1CN2C(c1ccnn1C1CC1)=O 49256,Cc1cc(Cl)c(C(=O)NCc2ccc(CNC(=O)CC3CC3(C)C)cc2)s1 49257,CCCC(C#N)C(=O)NC(c1cnn(C)c1)C(=O)NCC(C)CCC 49258,N1(C(CC(n2c(CC)ncc2)C)=O)CC2(CC(NC(C3CCOC3C)=O)C2)C1 49259,C1(F)(CNC(c2cc(C)c(O)nc2)=O)COCCN(C(=O)C(C)(C)F)C1 49260,c1(C(=O)N(C2CC2)CC2CC2)ccc2cc[nH]c2c1Br 49261,CC1CCC(C)(C(=O)NC2CC3(C2)CN(C(c2cc(C(F)F)no2)=O)C3)C1(C)C 49262,Cc1cc(F)cnc1C(=O)NC1(CO)CCN(C(C2(N(C)C)CC2)=O)CC1 49263,C(=O)(C(C(C)(C)O)NC(C1CCCN(C)C1)=O)NCCC1C(C)C1 49264,C(=O)(CCCC(F)(F)F)N1C(CCC)CN(C(=O)COC2CCCC2)CC1 49265,CCCC(CC(=O)N(C)CC1(N(C)C)CCC1)NC(c1cc(Cl)c[nH]1)=O 49266,N1(C(CCCCC(=O)OC)=O)CCC2(CCC(NC(=O)CCCSC)CC2)C1 49267,c1(C(N(CCC(=O)N(CCOC)C)C2CCC2)=O)ccnc(C)n1 49268,N1(C(C(C)(C)CF)=O)CC2(CCN(C(=O)CCCC3CCCCC3)C2)C1 49269,N1(C(c2cnc(C(C)C)[nH]2)=O)CCOC(C)(CNC(=O)C(F)(F)C(F)F)C1 49270,C1(NC(=O)Cc2coc(CF)n2)CN(C(=O)Cc2cccs2)C2(CCCCC2)C1 49271,c1(CNC(C(C)OC(C)(C)C)=O)ccc(C#N)cc1O.C12CC(C1)NC2=O 49272,c1(C(N2CC(C(C)NC(c3occc3Br)=O)C2)=O)cc(N)c(F)cn1 49273,C12(C(=O)NC(c3cccs3)C)CCC(CN(C(=O)CCCCCC#N)C1)C2 49274,C1(C(N(CC(CC)OC)CC)=O)CCN(C(=O)CC2CCCO2)O1 49275,N1(C(c2c(NC)n(C)nc2)=O)C(CC(=O)N(C)CC2(N(C)C)CC2)C2CCCC12 49276,N1(C(C=CC(C)NC(=O)C(F)CC2CCOC2)=O)CCCCCC1 49277,CCC(C)(CC)C(=O)N1CCC(N2CCN(C(=O)CCCNC(N)=O)CC2)C1 49278,C(=O)(C1CCc2nccn21)N1CCN(C(C2C(C)(C)COC2)=O)CC1CO 49279,c1(C(N2CCC3(C(=O)NC4CCN(CC)CC4)C(C2)C3)=O)c(Cl)ccc(F)c1Cl 49280,CC1CC(C)OC1C(=O)N(C(C)CCNC(c1ccsc1C(F)F)=O)C 49281,C=CCC(C(=O)NC(CNC(=O)C(c1ccccc1)C)C(C)(C)C)NC(C)=O 49282,c1(C(=O)NCCOCCNC(c2ccn(CC)n2)=O)ccc2ccsc2c1 49283,C1(CC(=O)NCC2N(C(c3c(C)nn(C)c3Cl)=O)CCC2)CCC2(CCC2)CO1 49284,C(C(C)(C)CC(=O)NC(C1CCCC1)CO)NC(C1(CC)CCCC1O)=O 49285,c1(CN(C2CCNCCC2C)C(c2c(C)cccn2)=O)ccc(F)c(Cl)c1 49286,C(=O)(C1CCCc2nn(C)cc21)NC(C(C)C)(C)CNC(c1ccc(Cl)o1)=O 49287,C(CC(C)(C)C(=O)N1C2CCC(C2)C1CNC(=O)Cn1[nH]cnc1=N)SC 49288,c1(C(N2CC=C(CNC(C3C(C)(Br)C3)=O)CC2)=O)[nH]nc2ncnc(O)c12 49289,C1(c2nc(CCCCC)nn2-c2ccc(N(C)C)c(Cl)c2)CCC2CC1C2(C)C 49290,CN1C(=O)c2ccccc2C1CC(=O)N1CCc2cc(O)c(C(=O)O)cc2C1 49291,C1(S(=O)(=O)NC(C2CCOC(=O)N2)=O)(COC)CC1C 49292,N1(C(C2CC=C(C)CC2)=O)CC2(C(N3Cc4c[nH]nc4C3)=O)CCC1CC2 49293,C(=O)(CCCCCN(C)C)NCCCN(C(C1CC=C(C)CC1)=O)C(C)C 49294,c1(C(N2CCN(CC(C)(C)NC(=O)Cn3ccnn3)CC2)=O)nnc(O)cc1O 49295,C(C(=O)N1CC(CO)(NC(=O)CCCCN2CCOCC2)C1)(C(C)C)SC 49296,C1(NC(C2C(CC)C2)=O)CCC(NC(=O)CCOc2ccc(Cl)cc2)CC1 49297,N1(C(C2C(=C)CC2)=O)CCCC(C2CN(C(c3nc[nH]c3C(C)(C)C)=O)C2)C1 49298,C1(C(=O)NCCn2ccc(C(N3C(C(C)C)CCC3)=O)c2)CCC(=O)N(C)C1 49299,c1(CCC)ccc(C(N2CCC(CF)(NC(=O)N(C(C)(C)C)C3CC3)C2)=O)cc1 49300,C(=O)(C1=CC(O)CCC1)NC1CCN(C(C2CC(C)(C(=O)OC)C2)=O)CC1 49301,Cc1csc2c(N3CC4CN(C(c5cc(Cl)cc(Cl)c5O)=O)C4C3)ncnc12 49302,c1(CN2CCN(C(=O)CCc3cccc(F)c3)C3C2C3)cccc([N+](=O)[O-])c1Cl 49303,C1(NC(c2cn(CC)nc2C2CC2)=O)CCN(C(=O)Cc2ccns2)CC1C 49304,N1(c2cc(SC)ncn2)Cc2ccccc2C1C(=O)N.NC1CCc2cccnc21 49305,c1(CN2C3C(C(N4CCC(C(N)=O)CC4)=O)C(C3)C2)c(F)cc(Br)cc1F 49306,c1(C(CNC(=O)CC2CCCCC2)O)cccc(-c2cccnc2)c1 49307,N1(C(c2c(N)ccc(C(C)C)c2)=O)CCC2CN(C(c3nccn3C)=O)CCC12 49308,N1(C(c2c(C)ccn2C)=O)CC(CCNC(c2oc(CO)cc2C)=O)OC(C)C1 49309,c1(C(=O)NCC2CCCC(NC(C3C(CC)CCO3)=O)C2)cc2c[nH]cnc-2n1 49310,Cc1c(C(N2CCC(C(=O)NCCc3noc(=O)n3C)(CO)C2)=O)nnn1C 49311,Cc1cc(C(=O)NC(C)CCNC(=O)C2=CCCC2)cc(Cl)c1 49312,c1(CC)ccc(CNC2CC2NC(=O)Nc2cccc(F)c2)cc1 49313,C(=O)(C(C)(C)C1=CCN(C(C2COCC(C)O2)=O)C1)N(CC(CC)OC)C 49314,C(=O)(C(C)(O)CC(C)C)N1CCN(C2CCN(C(CS(=O)(=O)NC)=O)C2)CC1 49315,c1(C(=O)NCc2cccc(F)c2)ccc(F)c(S(=O)(=O)N2CCC2)c1 49316,N1(C(C=C(CC)CC)=O)CC2CC(NC(c3ccnnc3S)=O)CC2C1 49317,C1(C(=O)NC2(CC=C)CN(C(C3(CF)CC3)=O)C2)CCCCC1C1CC1 49318,Cc1c(NC(=O)C(=O)N(C2CCN(CC3CC4(CO)CC3C4)C2)C)cccc1F 49319,CC1CC(CCNC(c2ncoc2-c2ccco2)=O)CCN1C(=O)COCCF 49320,C(=O)(C(F)CCC(C)C)NC(CC)CC(=O)NCCCC(C)O 49321,C1(CC)CN(C(=O)C(O)C(C)(C)C)CCC1NC(c1cc(O)ccc1C)=O 49322,N1(C(C(C)=C(CC)C)=O)CCC2(CCN(C(=O)C(C)(C)C(F)F)C2)C1 49323,C1(NC(c2c(C)scn2)=O)CCCC(N(C)C(C2CCC(C)CC2)=O)C1 49324,C1(C(=O)NC2CC3C=CC2C3)CCCN(C(=O)CN2CSCC2=O)CC1 49325,c1(CNC(c2cnc(C)n2C)=O)ccc(CNC(c2c(C)ncn2O)=O)c(F)c1 49326,c1(C(N2CC(NC(c3nc(Cl)cs3)=O)C(O)CC2)=O)csc(=NC2CC2)[nH]1 49327,Cc1cnc2cccc(C(N3CC(NC(=O)COCCCF)CC(F)C3)=O)n12 49328,CC(C)(C)CCC(N)CNCc1cnccc1Cl 49329,C(=O)(CCCS(C)(=O)=O)NCC1(F)CC(NC(C(c2c(C)cccc2)C)=O)C1 49330,c1nc(N2CCCCC2)[nH]c(=Nc2nnnn2C2CC2)n1 49331,N1(C(CCCO)C(F)(F)F)CCc2cc(Nc3ncccn3)ccc21 49332,CC1=C(C(=O)N2CCC(NC(=O)CC3(O)CCOC3)C(CO)CC2)CCS1(=O)=O 49333,C1(C#N)(C(=O)OCc2cc(C)c(Cl)cc2)CCCCCCC1 49334,c1(CC(=O)NCCOC2CCN(C(C(C)=CC)=O)C2)nn(C)cc1Br 49335,Cc1cn(C)cc1C(=O)NCC(C(=O)N(CCC(=O)NC1CC1)C)N(C)C 49336,N1(C(CCn2c(C)nc(C)n2)=O)CCC2CCN(C(C3CCNC3=O)=O)CC2C1 49337,C1(NC(c2c(CC)nc[nH]2)=O)CCN(C(=O)Cc2cnn(C)n2)C12CCCC2 49338,C(=O)(C1=NN(CCO)C(=O)CC1)N1C(C)C(CC2CC2)CCC1 49339,CC(C(=O)NC1CC(CNC(C2CCC2c2ccccc2Cl)=O)C1)C(F)F 49340,N1(C(c2ccc(CN(C)C)o2)=O)CCC2(C1)CN(C(C1CC(Cl)(Cl)C1)=O)C2 49341,c1(OC)ccc(CC(=O)NC2CCCC2NC(C2CN(C)CCO2)=O)cc1Cl 49342,CCC(C(=O)N1CCN(CC(=O)N2CC(c3nncs3)C2)CC1)C(C)C 49343,C(C(=O)NOCCCC1CC1)(C1CC1)OC(C)C.c1(C=O)csnn1 49344,c1(CC)onc(C)c1-c1ccc(O)cc1.c12ccc(cc1)C(C)NC(=O)OC2 49345,C(=O)(CC(C)(C)C(F)F)NC1C(NC(C(C)S(N)(=O)=O)=O)CCC1 49346,CN1CCN(C(c2cc3occc3s2)=O)C(CNC(c2ccc(O)c(N)c2)=O)C1 49347,Cc1nc(O)[nH]c1C(=O)NC1(CN(C(=O)Cc2csc(C(F)(F)F)n2)C)CC1 49348,N1(CC(=O)N(C)CC2(NC(C3CCC(CC)O3)=O)CC2)CCC(=O)NC1=O 49349,C#CCCCCCCC(=O)NC1CC(F)CN(C(=O)C(c2ccc(C)o2)C)C1 49350,N1(C(C(C)NC(COC)=O)=O)CC2CCC(C1)C2NC(=O)CC1CC=CCC1 49351,c1(C(=O)NCC2(C)CCN(C(C3(OC)CC3)=O)C2)c(C)nn(C)c1OC 49352,c1(CN2CCC(C(=O)Nc3cc(C(=O)OC)cc(Cl)c3)C2)c(F)cc(O)cc1F 49353,Cc1cc(C)c(C(=O)NCCCCN(C(=O)COCCOCCO)C)s1 49354,c1(NC(C(C)(N(C)C(c2ccnnc2)=O)C2CC2)=O)ccc(O)c(=O)cc1 49355,c1(C(=O)NC2CN(C(C(C=CC)O)=O)CC2O)cnc2c(c1)COCC2 49356,C(CC(=O)N1CC2CC2(CO)C1)(C(F)F)NC(CC1C=NN(C)C1=O)=O 49357,C1(O)(C(C(=O)NC(c2ccc(C)s2)C)NC(c2cc(CC)on2)=O)CCCCC1 49358,c1(CC)cc(C(=O)N(CC(C)(C)C(=O)NC(CO)C(=O)OC)C)nn1C 49359,C(C)(CCC(=O)N1CC(O)(CNC(C2CC(=O)N(C(C)C)C2)=O)C1)SC 49360,C(=O)(CC(C)P(C)(C)=O)N(CC(C)(C)NC(C=C(C)c1ccsc1)=O)C 49361,C1(CC)CN(C(CC(C)C)C(=O)NCCCF)CCN1CC(C)O 49362,C(=O)(C(C)C(F)(F)F)NCCN(C(=O)C(C)COC)CCC 49363,c1(N2C(=O)C2)ccc2nn[nH]c2c1O.C1(C(C)(C)C)CCC(C(=O)CC2N=N2)CC1 49364,C1(CC)CN(C(=O)C(C)c2cccs2)CCN1C(c1cnc(O)c(F)c1)=O 49365,N1(CCO)CCCOC1=O.C(=O)(CCCc1cccs1)C(C1CCN1)=O 49366,C(=O)(CC(CC(C)C)NC(C1CCC(C)=C(C)C1)=O)N(CC)CC1CCCC1 49367,C1(C(=O)NC23C(CN(C(c4cc(C)[nH]n4)=O)C2)C3)CCc2ccc(F)cc2C1 49368,c1(C(=O)NC(CC)CNC(c2cscn2)=O)cc(N)c(N)cc1F 49369,N1(C(CCN(CCCCC)C)=O)CCN(C(C2CC2OC)=O)CC1C1CCC1 49370,c1(OC)ccc(CC(N2CCC(CNC(C34CCC(CO3)C4)=O)C2)=O)nc1 49371,c1(C(N2C(COC)CN(C(=O)C=C3CCC(C)C3)CC2)=O)cc(S(C)(=O)=O)co1 49372,C1(COC)CN(C(=O)CC2CCCC2)CCN1C(C1CCCC(=O)N1C)=O 49373,C12(NC(c3ncn(CC)c3)=O)CCCC(NC(c3ccsc3C)=O)(C1)C2 49374,c1(C(=O)NCC2(NC(COCC)=O)CC3CCC2C3)ccc2snnc2c1 49375,C12(C(=O)NCCCc3ncco3)CCC(CC1)N(C(=O)C=CC1CCOC1)C2 49376,C(=O)(CCCS(=O)(=O)NC1CC1)N1CCN(C(CN(S(C)(=O)=O)C)=O)C(CF)C1 49377,S(=O)(=O)(CC(=O)NC1CCN(CC2CCCC2(C)CCOC)CC1)N(CC)CC 49378,C1(C(=O)OC)CC(n2ccnn2)CN1S(=O)(=O)CCC(=O)OC 49379,c1(OC)cccc(C=CC(=O)NC(C)CC(C)NC(c2ccc(C)nc2C)=O)c1 49380,c1(C(=O)NC2CC(CC(=O)NC(C=C)(C)C)C2)cn(C)nc1SC 49381,c1(C(=O)NCCCCNC(C2C(C(=O)NCC#C)C2)=O)cccc(C(N)=O)c1F 49382,c1(CC)nc(C(=O)NCC2COCC2NC(=O)Cn2cc(Cl)cn2)co1 49383,C(C)(C)(CCC(=O)N1CCN(C(c2sc(C)cc2Cl)=O)C2CC12)OC 49384,c1(C(N2CC(F)CC(C(=O)Nc3c(C#N)nccc3)C2)=O)cccc([N+](=O)[O-])c1 49385,c1(C(=O)NCC2(OC)CN(C(=O)C(C)(CO)OC)C2)nc2ccccc2cc1Cl 49386,C1(C2(O)CN(C(C3(CF)CC3)=O)C2)(CNC(C2CC2C2(O)CCC2)=O)CC1 49387,C1(CN)CCCN1C(=O)CC1(CNC(=O)Cc2ccn(C3CCCC3)n2)CCC1 49388,c1(C(=O)NCC2CN(C(c3c(SC)snn3)=O)C2)nnn(C2CCCC2)c1C 49389,N1(C(C(CC)O)=O)CCN(C(=O)C(F)(F)c2csc(Cl)n2)C2(CCC2)C1 49390,C1(C(=O)NCCn2ncc(CC)c2)C=CCCN1C(c1cn(CC)nn1)=O 49391,c1(C(=O)NC(C(C)(C)NC(Cc2c(C)nsc2)=O)C)cc(C(F)(F)F)cc(Cl)c1 49392,C(N=c1[nH]ccn2cnnc12)c1c(OC(F)F)ccc(F)c1 49393,C1(N(C(c2nc(C(C)OC)oc2)=O)C)CCN(C(=O)COC2CCOC2)CC1 49394,C=Cc1cnn(C)c1C(N1CC2CC1CC2NC(=O)C(=O)C(C)(C)C)=O 49395,CC1CC(CNC(=O)Cn2ccnc2)CN1C(=O)OC(C)(C)C.c12ccc(o1)C2 49396,Cc1ccc2c(c1C)OCCC2NC(=O)NC1(C)CCC(=O)N1C 49397,C(CCC(O)C(=O)Nc1ccc(C)nc1)NC(C(C)=C1CCCC1)=O 49398,n1(CCOc2c(C)cccc2)nc(C2CCCO2)nc1C1CCCn2ccnc21 49399,c1(CC)ccc2cc(C(=O)NCC(C(C)C)NC(=O)C(CO)NC(N)=O)[nH]c2c1 49400,C1(C(=O)OC)CC(F)(F)CCN1C(=O)OC(C)(C)C.C1(OC)CCN2C1C2=O 49401,C#CCC(C(=O)N(CC(C)N(C(=O)Cc1csc(Cl)n1)C)C)C1CC1 49402,N1(C(c2nc(C)[nH]n2)=O)CCC2(NC(=O)C(=Cc3c[nH]cn3)F)CCCC12 49403,c1(C(C)C)nocc1C(N1CCCC1CN(C)CCOCCO)=O 49404,c1(C(=O)OCC)[nH]c2ccc(NC(c3c(Cl)cc(COC)cc3Cl)=O)cc2c1C 49405,C1(C(NOCCCN(C)C)=O)CC(N(C(=O)Cc2cccnc2C)C2CC2)CCO1 49406,N1(C(C2(F)C(C)C2)=O)CCC2(CCC2CNC(c2ccc[nH]2)=O)CC1 49407,CC(C)CC(=O)NCC1CCN(C(C2CNC(=O)N2)=O)C1 49408,CC(C)CCCOCC(=O)N(CCCN(C)C)CCNC(C1CC1Br)=O 49409,C1(OC)CCC12CC(C(=O)NCC13CC(CO1)N(C(=O)CC1CSC1)C3)C2 49410,c1(C(=O)NCC2CC3(CC(NC(CCSCC(N)=O)=O)C3)C2)cnc2n1CCCC2 49411,CC(C)(C(=O)NCC1(NC(=O)CC2(n3cccn3)CC2)CC1)c1ccns1 49412,c1(CC(=O)NCC2CCN(C(C3CNC(=O)N3)=O)C23CC3)ccc(Cl)c(Cl)c1 49413,Cn1nc(CC(=O)NC(C)(CNC(C2CC23CCC3)=O)CO)cc1C(F)(F)F 49414,c1(OC(C)CNC(=O)NCc2nc(-c3ccccn3)no2)ccccc1Br 49415,N1(C(C(n2c(C)ncc2)C)=O)CC2CCC2(CNC(c2cc(Cl)n(C)n2)=O)C1 49416,c1(C(=O)NC(CNC(c2c(C)cno2)=O)C(C)(C)C)c(Cl)ccc2ccoc12 49417,C1(C)(C(=O)NCc2ccc(C(N(C)Cc3n(CC)ccn3)=O)s2)CCOC1C 49418,c1(C(=O)NCC2C(NC(CCN3C(C)CCCC3)=O)C2)ccc2n[nH]cc2n1 49419,c1(C(c2nnnn2Cc2cccs2)NC(C(C)(C)OC)C)cnc(Cl)n1C.C1CC1 49420,n1(C(C)C)nncc1C(=O)N(CC(C)NC(=O)CN1CCCC1)C 49421,N1(C(C(C)=C(C)C)=O)CC(C)(C)OCC1CNC(c1cccc(O)c1)=O 49422,C1(CNC(C#CC2(CC)CC2)=O)CCC(C)(C)CN1C(c1csc(C2CC2)n1)=O 49423,C=CCC(C(=O)NC1CCSC12CN(C(c1ccc(Cl)o1)=O)C2)C(C)C 49424,N1(C(C(CCC)N(C)C)=O)CC(NC(c2cccc(C(=O)OC)n2)=O)C(C)(C)C1 49425,C1(c2c(CC)cccc2)CCCN(c2nnc(-c3ccnc(C)c3)o2)CC1 49426,n1(C(C)C)nnnc1C(C1CCCC1)NC(c1cccnc1)c1ncsn1 49427,C(=O)(C(C)(C)CCCF)N(CCCCCNC(C(C(C)C)OCC)=O)C 49428,CC12CCC(C(=O)NCC#CCNC(=O)C(C)(C)n3cc(Br)cn3)(CC1)CO2 49429,C1(C(N(C(CC(C)C)C)C)=O)C2CN(CC(=O)OCC3CCC3)CC12 49430,N1(C(c2ccn(CCOC)n2)=O)CCC2CN(C(C3CC4(CC4)CO3)=O)C2C1 49431,C1(C(N2C(CC)CNC(=O)C2)=O)CCN(C(=O)C(C(C)C)C2CCC2)CC1(C)C 49432,c1(C(N2CCN(c3c(Br)cnc(C)n3)CC2C)=O)ccc(Br)c2ccccc12 49433,c1(SC)ccccc1C(N1CCOC(CCCNC(C2CCCN2C=O)=O)C1)=O 49434,N1(C(=O)CC2CC(F)(F)C2)CCCC1C1CCCN1C(C1SCCCS1)=O 49435,C1(CC(=O)NC(CCNC(C(C)O)=O)C)CC(F)(F)C1 49436,C1(CNC(C(C)(C)F)=O)CC2(CCN(C(c3ccc(N)c(Cl)c3)=O)C2)CO1 49437,N1(C(CC(=O)OC(C)(C)C)=O)CCC(NC(C2CC2(F)F)=O)C12CCCC2 49438,CCCC(C)CC(=O)NC1CCC12CN(C(c1cc(C)cc(F)c1)=O)C2 49439,C(=O)(C(O)C(C)(C)C)NCC1(OCC)CN(C(=O)C2=CCCCC2)C1 49440,c1(C(=O)NC(CNC(C2N(S(CCC)(=O)=O)CCC2)=O)C(C)C)nccc(C)n1 49441,C(=O)(C1=C(C#N)CCC1)N(C(C)CNC(C1CCCN1N=O)=O)CC 49442,CCC(C)(CO)C(=O)NC(CNC(c1cncc(F)c1)=O)C(C)(C)C 49443,c1(C(N2C3CCC(CNC(C(C)(C)SC)=O)(C3)C2)=O)ccc2c(c1)COC2 49444,c1(C(N2CCC(C(F)F)CC2)C(=O)Nc2ccc(F)cc2)ccc2c(n1)CCC2 49445,N1(C(C(c2cnn(C)c2)C)=O)CCC12CN(C(c1cc(O)cc(Cl)c1)=O)C2 49446,c1(OC)ccccc1SCNC(=O)C(c1sc(Br)cc1C)N(CC(C)(C)C)C 49447,CCCCC(C)C(=O)NCC(C1CC1)NC(=O)C(F)(F)c1nc(C(F)(F)F)cs1 49448,C1(NC(CNC(C=NOC)=O)=O)CCC=CCC1 49449,CCCS(=O)(=O)CC(=O)NC(C)CC(C)NC(=O)COc1ccc(Cl)cn1 49450,N1(C(CCNC(=O)CO)=O)CCCN(C(c2cc(-n3cnnc3)ccn2)=O)CC1 49451,C=C(C)c1ccccc1NC(c1cc(CNC(C2C3CC(=O)CC23)=O)no1)=O 49452,N1(C(c2c(CC)cns2)=O)CCOCC(C(N2CC=CC2C(=O)NC)=O)C1 49453,CN1CCCC(CCC(=O)N(C)CCC2CCN(C(C3(O)CCC3)=O)CC2)C1 49454,c1(CC2N(CC(=O)N(CC)CC3CC3)CCC2)cccc(C)c1.C(=O)(CO)N 49455,C#Cc1ccc(C(=O)NCCC2CC(NC(c3ccc(C#N)o3)=O)C2)cc1C 49456,C(C(C)CC(=O)N(C1CC1)C1CC1)NC(CC=CCC)=O 49457,c1(C(=O)NC(CN(C)C)C(=O)NC2CCC(C)(C)C2)ccc([N+](=O)[O-])o1 49458,N1(C(c2cc(CC)nn2C)=O)CC(C(=O)NC(CO)C(N)=O)C(C2CC2)C1 49459,C1(C)(C(=O)NC(CN(C(C(CC)F)=O)CC)C)C(C)(C)C1(C)C 49460,Cc1cc(C(N2CC3C(NC(=O)CC4CCC(C)(C)C4)C3C2)=O)n(C)n1 49461,CCC(C(F)(F)F)NC(c1ccn(CCNC(C2COCC(C)O2)=O)c1)=O 49462,CC(C)C(C(=O)N1CCC(NC(C2CC3(CC3)C2)=O)C1)n1cncn1 49463,c1(-n2c(-c3ccc(C(CC)(C)C)cc3)nc(CC3CC3)n2)ccc(F)c(Cl)c1F 49464,c1(C(N2CC3C(CNCc4ccc(C(N)=O)cc4)(C3)C2)=O)ccc2scnc2c1 49465,c1(OC)ccc(C(=O)N(CCC(C)NC(=O)CC2CCC(=O)N2)C)c(O)c1F 49466,CCC(C)(C)C(C)CC(=O)NCCC(C)NC(c1ccc(OCCOC)nc1)=O 49467,C1(CNC(CNC(C)=O)=O)C2CN(C(c3cnn(-c4cccc(Cl)c4)c3)=O)CC12 49468,C1(C(=O)NCc2nc(-c3ccc(C)cc3)oc2)CN(C)CC(C)O1 49469,N#Cc1ccc(C(N2CC(CO)(NC(=O)C=Cc3cscn3)C2)=O)s1 49470,C1(NC(C2(CC(=O)OC)CC2)=O)CC(C(=O)NC2CNC(=O)C2(C)C)=CC1O 49471,c1(C(=O)NCCCC(C)NC(=O)CC(=O)N(C)C)ccccc1NC(=O)C(C)C 49472,C1(C(=O)NC(CNC(=O)CCCC2CCCC2)C2CC2)CCCC(CC2CC2)C1 49473,c1(C(=O)NC2(n3cccn3)CC2)cc(O)nc2c1CN(C(C1(F)CC1)=O)CC2 49474,C1(NC(C=NOC)=O)CCC(O)CN(C(=O)CC(C(F)F)n2cccn2)C1 49475,C(=O)(CC(C)CCC=C(C)C)NCC1CCN(C(C2CC(C(=O)OC)C2)=O)CC1 49476,CCC(CC(=O)NC(CNC(c1coc(C2CC2)n1)=O)C(C)C)OC 49477,C1(C(N2CC(CNC(=O)C=CC3CCCC3)C(C)C2)=O)(OC)CCC(C)CC1 49478,CCCCC(C(=O)NO)NC(=O)NC1CCOCC1F 49479,C1(C(N(C(C)C(F)F)C)=O)CCC2CCCCN2C1 49480,c1(OC)cccc(C(=O)N(CCCNC(=O)CCc2ccc(F)cc2)C)c1OC 49481,c1(COC)nc(NCC2CC(=O)N(C)C2=O)cc(=NCc2cccs2)[nH]1 49482,c1(C(N2CCC2C(=O)NC2CC2)=O)ccnc(CC(F)(F)F)c1.C12(CC1)C(=O)N2 49483,S(=O)(=O)(c1ccc(F)c(C(=O)O)c1)CN1CC2CN(Cc3n(C)cc(Br)n3)C2C1 49484,c1(C(=O)NC(Cc2ncn(C)n2)C(=O)O)ccc(CO)cc1 49485,c1(C(N(C2CCN(C(=O)COCc3ccncc3)C2)C)=O)ccn(CC2CC2)n1 49486,N1(C(c2cc(-c3cccs3)on2)=O)CC2(CCN(C(C3(C(F)(F)F)CC3)=O)C2)C1 49487,C1(C(=O)NCC2N(S(CCOCC)(=O)=O)CC(OC)C2)Cc2ccccc2C1 49488,C1(C(c2nnnn2C2COC2)NC(=O)CC(C)OCC)(OCC)CCCC1 49489,N1(C(COCCC)=O)CC2(CC1CNC(=O)Cc1cc(C)[nH]n1)CC2(F)F 49490,c1(C(=O)NCC2CC(C(N(C3C4CCCC34)C)=O)C2)cc(C(N)=O)[nH]n1 49491,C1(C2CCCN(C(c3csc(=N)[nH]3)=O)C2)(NC(CCC(=O)NCCC)=O)CC1 49492,C(=O)(CCCCCC)NCC12OCC(N(C(CC(=C)C)=O)CC)(C1)C2 49493,c1(C(=O)NC(CC)CNC(=O)C(C)c2cncs2)ccc(F)cc1OC 49494,C(=O)(CCC(=O)c1cc(C)sc1C)NCCN(C(=O)CC1CCS(=O)(=O)C1)CC 49495,CC(C)CC(F)(F)C(=O)NC1CC1CNC(c1ccc(Cl)c(F)c1N)=O 49496,O=C(CC(C(F)F)NC(C1(F)CC1)=O)NCC1(F)CCOCC1 49497,CN1CCC2C(CCN2C(=O)CCC2(NC(=O)COc3ccccc3)CC2)C1 49498,C1(C(=O)NC2(C(=O)N(CC(=O)NC(C)(C)C)C)CCN(C)C2)CCCC1C1CC1 49499,C(=O)(N1CCC(C(=O)NCC(F)CO)O1)c1nc(=N)[nH]cc1 49500,C1(NC(c2c(CC)cco2)=O)CN(C(=O)CCc2ccccc2F)CCC1C 49501,C1(C2CCC2)(CNC(c2csc(CNC(COC3(C)CCC3)=O)n2)=O)CC1 49502,C(=O)(N=c1[nH][nH]c2cccnc12)C1CCC(NC(c2ccccc2O)=O)C1 49503,C(=O)(CCC(F)(F)F)NC1CC(O)(CNC(c2c(CC)oc(C)c2)=O)C1 49504,C(=O)(C1CCc2c(Br)cccc21)NCC(CC)NC(c1cc[nH]c(=N)c1)=O 49505,N#Cc1c(C(=O)NCC2(O)CCN(C(=O)C(=O)NCC(F)(F)F)C2)cccc1F 49506,c1(C(N2C(CC(=O)NCC(C)S(N)(=O)=O)CCCC2)=O)cn(C)ccc1=O 49507,N1(C(C=CC)=O)CCC(C)(CNC(c2ccc(C(=O)NC)nc2)=O)C1 49508,Cc1cc(F)c(C(c2nnnn2C2CCCCC2)NC2CC(C)C2)c(Br)c1 49509,c1(OC)ccc(CCC(=O)N(C)CC2CCCN(C(C3(SC)CC3)=O)C2)cn1 49510,C(=O)(CCS(N)(=O)=O)NCC(C)(C)OCC(=O)N(C)Cc1nccn1C 49511,C(=O)(CCCCC(C)(C)C)NCC(C)(CC)NC(CCC(=C)Br)=O 49512,CCCCC(CNC(c1cc(Cl)ccn1)=O)CCC 49513,C1(C(N2CC(C)C(CCNC(=O)CCCCCF)C2)=O)CCc2c[nH]nc2C1 49514,c1(CC)nnc(C)cc1C(=O)NC(C)(CNC(c1cc(C(F)F)[nH]n1)=O)CO 49515,Cc1cc(O)ncc1C(=O)NC1C2CC1N(C(=O)CN1CCC(=O)CC1)C2 49516,Cc1nc2sccn2c1C(=O)NC1CN(C(c2cc[nH]c2)=O)CC1C 49517,C1(C(=O)NC(C)C(=O)NO)CCC(C)(C)N(C(=O)CC2CCCCCC2)C1 49518,C(=O)(CCC(=O)Nc1nccs1)NCC(C)N(C)C(c1cccc(O)c1)=O 49519,N1(C(CC(C)CF)=O)CCN(C(=O)CCC2OCCO2)C(CF)C1 49520,c1(C(=O)NC2(C)CC(C(=O)Nc3cnc(OC)nc3)C2)nccc(C)c1F 49521,c1(OCC(=O)NCC2N(C(CSCC(C)C)=O)CCC2C)cc(Cl)cc(Cl)c1 49522,Cn1cc(C(F)=CC(=O)NC2CC(NC(c3conc3C3CCCC3)=O)C2)cn1 49523,C(=O)(C(CC(C)C)C(C)C)NCCC1OCCN(C(CC2(NC(C)=O)CC2)=O)C1 49524,c1(OC)ccc(NC(C2CC23CCN(C(c2cnnc(O)c2)=O)C3)=O)c(CO)c1 49525,c1(C(=O)NCCC2N(C(Cn3ncc(C)c3)=O)CCC2)cncc2cnccc12 49526,C12(NC(=O)Nc3ccc(OCCO)nc3)CCC(O)(CC1)C2 49527,CCCCCC(F)C(=O)N1CCC(c2cn(Cc3n[nH]cc3C)nn2)CC1 49528,C1(CC)CC(NC(=O)CC(C)(C)NC(C2CC(CF)C2)=O)CCO1 49529,C1(CNC(CNC(C)=O)=O)CN(C(=O)C(C)(C)N(C)C)CC(C)(C)C1 49530,C#CC1CCCN(C(=NCCOC)NCC(CC(C)(C)C)C(=O)NC2CCC2)C1 49531,C1(SC)CN(C(=O)C(N2CCCC(C)C2)=O)CC1NC(c1cncc(C)c1)=O 49532,C=CC(C)(CC)C(=O)NC1CCCC1NC(c1c(C)coc1-c1ccccc1)=O 49533,N1(C(C(C(=O)OCC)F)=O)CCN(C)C(C(=O)NCC2=CCCC2)C1 49534,c1(OC)ccc(CC(=O)N(C)CC2CN(C(=O)Cc3ccsc3)CCO2)c(F)c1 49535,c1(C(C)OCC)nc(CC(C)CN(C(=O)C=C2CC2)C)cs1 49536,C(=O)(NNc1ccc(S(=O)(=O)C(F)F)cc1)c1c(OC)c(F)c(F)c(F)c1 49537,N1(C(C2OC3CCC2C3)=O)CC2=C(C1)CN(C(C1(n3cnnn3)CC1)=O)C2 49538,C1(C)(C(=O)NC2(CC(=O)OC)CCC2)CCCN(C(c2cccnc2Br)=O)C1 49539,N1(C(c2ccc(C(=O)OC)s2)=O)CCC2CCN(C(C3CC4CC4C3)=O)CC12 49540,c1(C2(C(N3CC4CCN(C(=O)C=CCO)C4C3)=O)CC2)nccc2ccccc12 49541,C(C)(CCCCNC(=O)C(C)c1cccs1)NC(C1N=C(C)SC1)=O 49542,C1(C(=O)NCCOC(C)(C)C)CC2(CCN(C(c3ccnc(Cl)c3)=O)CC2)CO1 49543,c1(C(=O)NC(CCOC)CNC(C2(C)CC=CC2)=O)ccc2cnn(C)c2c1 49544,CC1(C(=O)NCC(N2CC(N(C)C)C(O)C2)=O)CC2CCC1C2 49545,CON(CCC(=O)NC1CCC(=O)N(C(C)C)C1)C(=O)c1cccc(C)c1F 49546,c1(C(=O)OCC)cc(C(=O)NC23CC(NC(=O)CN(C)C4CC4)(C2)C3)ccc1Cl 49547,Cn1ccc2cccc(C(N3CC4CCC(Nc5ncc(O)cn5)C4C3)=O)c12 49548,N1(C(c2cnc(SC)s2)=O)CCN(C(C2CCCC2c2cnn(C)c2)=O)CC1 49549,C1(CNC(C2CC(C)SCC2)=O)CCCC2CN(C(=O)Cc3ccn(C)n3)CC12 49550,n1(-c2cn(CC)nc2)nc(CCOCC2CC2)nc1-c1coc(C2(CC)CC2)n1 49551,C(=O)(C(C(C)CC)CNC(=O)C(C(CC)CC)OC(=O)OC(C)(C)C)NCC#C 49552,C1(CNC(c2cc(CCC)ncc2)=O)CCN(C(=O)C(C2CC2)OC)CC1O 49553,c1(C(C)(C)OC)nc(=NC(=O)N2CCC(C)(NC(C)=O)CC2)s[nH]1 49554,Cc1ccnc(CNC(=O)C(O)CCNC(C2CCCCCN2C)=O)c1F 49555,Nc1ncccc1C(N1CC2C(CNC(c3cc(=O)cc[nH]3)=O)C2C1)=O 49556,C(=O)(C(O)CC(F)(F)F)N1CCCC(N(C(COCc2ncc(C)o2)=O)C)C1 49557,c1(NC(c2coc(Cl)c2)=O)cccc(NC(C2(C3CCCO3)CCC2)=O)c1 49558,C1(NC(CC(C(=C)C)OCC)=O)COC2(C1)CN(Cc1sccc1Cl)C2 49559,N1(C(C(CC=C)C)=O)C2CCC1CC(C(=O)NC1(C(=O)OC)CC1)C2 49560,c1(C(=O)NC2(CNC(=O)C(=O)NC3CC3)CC2)ccnc2c1CCC2 49561,C1(C(N2CCN(C)C(CO)C2)=O)CN(C(c2cc([N+](=O)[O-])c[nH]2)=O)CCC1(C)C 49562,CN=c1nc(N2CCC(C(C)COC)CC2)[nH]c(N2CCOCC(C)C2)n1 49563,N1(C(c2c(C(C)C)ocn2)=O)CCCC(NC(=O)C(C)c2ccco2)CCC1 49564,CCC(CC(=O)NC(C1CN(C(=O)C=Cc2ccc(C(F)F)o2)C1)C)OC 49565,C1(CNC(c2ccco2)=O)COCC2(CCN(C(=O)CC3CC4(CC4)C3)CC2)O1 49566,c1(OC)cc(C(=O)NCC2(F)CC(CNC(=O)CN3CCOCC3)C2)ccc1Cl 49567,Cc1cnc(Cl)c(CCNC(=O)NC(c2cccc(SC3CC3)c2)C)c1 49568,N1(C(C2N(C)CCOC2)=O)CC2CCN(C(c3ccc(Cl)c(Cl)c3)=O)C(C2)C1 49569,C(CN=C(NCC(C)C)N1CCC(=C(F)CBr)CC1)c1c(OC)ccc(F)c1 49570,C(=O)(CS(=O)(=O)C1CC1)NC1CCCC(NC(=O)COc2cccnc2)CC1 49571,N1(C(COCC#C)=O)CCC2C(NC(c3sc(-c4ccccn4)nc3C)=O)CC12 49572,C(=O)(C(C)(F)C(=O)NC(C)C(=O)N(CCC(F)CN=[N+]=[N-])C)OC 49573,c1(SC)cn(C)nc1C(N1CCCC(C(C)NC(C2(O)CCOCC2)=O)C1)=O 49574,N1(C(C(=O)NC2CC2)=O)CC2CN(C(c3ccc(-c4nnco4)cc3)=O)CCC12 49575,N1(C(Cc2cccc(COC)c2)=O)CCC(NC(C2CCCC23CC3)=O)CC1C 49576,c1(CNC2C(F)(F)CCN(C(c3ccncc3F)=O)C2)cc(F)ccc1[N+](=O)[O-] 49577,C(=O)(CCCCCN=[N+]=[N-])N1CC(N(C(C2CC(C(C)C)C2)=O)CC)C1 49578,Cc1ccc2cc(C(=O)NC3CCCC34CCN(C(C3(CO)CC3)=O)C4)[nH]c2c1 49579,C1(NC(C(=O)NCC)=O)CC(C)(NC(C2CCCN2S(C)(=O)=O)=O)C1 49580,CC(C)(C(=O)NCc1nnc(C(F)F)o1)NC(C12CC(CO1)C2)=O 49581,N1(C(COCCOC)=O)CC=CC1CNC(=O)CN1CCC(C)C1 49582,Cc1ccn2ncc(C(=O)NCC3CN(C(C45CC(C)C4C5)=O)C3)c2n1 49583,c1(C(=O)NCCN(C(C(COC)CC(C)C)=O)C)n[nH]c2nccc(Cl)c12 49584,CC1CN(C(C2CCCS2)=O)CC1NC(C1(F)CCOC1C)=O 49585,N1(C(C=CC2N(C(CN(CCC)C)=O)CCC2)=O)CCN(C)C(=O)C1C 49586,c1(C(N2C(C(=O)O)CC(=C)C2)=O)c(-c2nn[nH]n2)cccc1Br 49587,C(CS(=O)(CCO)=NC(=O)c1ccc(-n2cccn2)cc1)NC(=O)OC(C)(C)C 49588,CC1CN(C(=O)CC(C(F)(F)F)NC(=O)CC(C(Cl)Cl)N(C)C)C12CCOCC2 49589,C12(C(=O)OC)CC(C(=O)NCC3CCC(NC(=O)CCc4ccncn4)C3)(C1)C2 49590,c1(C(N2C(CCNC(=O)C=Cc3cc[nH]n3)CCCC2)=O)cnc2c[nH]nc2c1 49591,C1(n2cc(C#CCNC(=O)CC)nn2)CCOC2(CCOCC2)C1.C1CC1 49592,c1(CN)cccc(C(N2CCCCC2c2ccc(F)cc2)=O)c1 49593,N1(C(c2c(CC)ccs2)=O)CCN(C(C2CCN(C)CC2)=O)C(CF)C1 49594,c1(CC(N2CC(C)N(C)CC2)=O)c[nH]c2ccc(-c3cncc(N(C)C)c3)cc12 49595,c1(C(=O)NC2C3(CC(NC(Cc4cnc(C)[nH]4)=O)C3)C2)ccc(N)c([N+](=O)[O-])c1 49596,c1(C(C)(O)CCC(=O)NC(c2ccccc2)C2CC2)cccc([N+](=O)[O-])c1 49597,C#Cc1ccc(F)c(C(N2CC3CCC2(CNC(=O)Cc2ccsc2)CC3)=O)c1 49598,C1(NCC2CCN(C(C)C)C2)CCCCN1C(c1ccn(CCF)n1)=O 49599,O=C(C#CC1CCCO1)NCC(c1ccc(F)cc1)NC(c1cc(Cl)no1)=O 49600,C1(N(C(C(CC)C)=O)C)CCCCN(C(C2CC=CC2)=O)C1 49601,C12(OC)CC(C(=O)NCC(C)(C)NC(c3cccc(F)c3)=O)C(C1)C2 49602,c1(C(N2CCN(CC(N3CCOCC3)=O)CC2)=O)n[nH]c2c1CCC(F)(F)C2 49603,c1(C(=O)NCc2nc(C(N3CCCC3c3ncc[nH]3)=O)co2)c(O)cccc1Cl 49604,c1(-c2nc(C(C)OC)nn2CC2CCOC2)cc(=O)c2ccccc2o1 49605,c1(OC)ccc(C2(CNC(=O)NC3(C)CCCNC3=O)CCCC2)cc1OC 49606,C1(NC(C(CCC)OCC)=O)CCN(C(c2cc(C)n(C(C)C)c2)=O)CC1F 49607,N(C1CCOc2ccccc21)(CCCN)C(=O)NC1CCOCC1F 49608,CC1Cn2nc(C(=O)NC3CCN(C(c4occ5c4CCC5)=O)C3)cc2C(=O)N1 49609,c1(CC(C)C(=O)NCC#CCNC(C2CC3(CCCO3)C2)=O)ccc(C#N)cc1 49610,C1(C(N2CC(CNC(C=C(C)C)=O)OCC2)=O)CCN(C)S1(=O)=O 49611,c1(NC(C(C)C)C(C)NC(=O)Cc2cnccc2Cl)ncnc2c1cnn2C 49612,Cc1cc(Cl)c(Br)cc1C(N1CCCC1C(=O)Nc1nc(C#N)cs1)=O 49613,C=CC1(C(N2CCC(C(F)(F)F)C2)=O)CCN(C(C2CCC2C)=O)C1 49614,N1(C(COCCCC)=O)CC2CCC1C(CNC(=O)CCCc1cnn[nH]1)C2 49615,N1(C(c2ncn(CC)n2)=O)CC(CNC(=O)C=Cc2ccsc2)C2(CCC2)C1 49616,c1(C(N2CC3CCC3(C(N3CCC(O)C3)=O)C2)=O)cccc2ncsc12 49617,C1(CC)(NC(C2C=CCC2)=O)CCN(C(=O)C(C(C)C)OC)CC1 49618,n1(CC)ccnc1C=CC(=O)NC1CC1CNC(C1COCCO1)=O 49619,c1(OC)ccc(CCC(=O)NCC2CCC2NC(C2CC3C=CC2O3)=O)c(F)c1 49620,N1(C(c2c(OC)ccc(C)c2)=O)CCC2C(CCN2C(c2cnncc2C)=O)C1 49621,c1(CC)nc(C)c(C(=O)NCC(C2CCCN2C(C2CCCOC2C)=O)(C)C)s1 49622,N1(C(C2(C)CCCCC2)=O)CC(CO)C2(CCN(C(C3COCCO3)=O)CC2)C1 49623,C1(CNC(C2(C)CCNC2=O)=O)CN(C(c2c[nH]nc2Cl)=O)C2(CCC2)C1 49624,c1(CC)ccc(O)c(C(=O)N(C(C)CCNC(C2CCC2(C)C)=O)C)c1 49625,C1(CC)C(NC(=O)COc2cccc(C)c2)CCN1C(c1ccsn1)=O 49626,N1(C(c2ccc(C(CC)=O)cc2)=O)CCN(C(=O)C(C)C(C)O)CC1CC(F)F 49627,C1(N(C(C2C(CNC(c3c(CC)non3)=O)OCC2)=O)C)CCC(O)CC1 49628,CCCC(C)(O)C(=O)NCC(CC)NC(=O)Cc1ccc(OC)c(OC)c1 49629,N1(C(c2cc(C)c(O)nc2)=O)CCC=C(C(=O)N2CCCCC2C#N)C1 49630,C12(C(=O)NC(COc3cccc(C(=O)OCC)c3)C)CC=CC(C1)OC2 49631,c1(OC)ccc(CC(N2CC3C(N(C(=O)CN4CC(C)(C)C4)C)C3C2)=O)cn1 49632,CC1=C(C(=O)N2CCC(CC(N3CC(Nc4ccccn4)C3)=O)C2)CCO1 49633,CCCC(CCO)NC(=O)C(CC)NC(=O)C#CC(C)C 49634,C(c1cccc(Cl)c1)=CC(=O)NC(C1CCN(C(c2cc(C)c(C)[nH]2)=O)C1)C 49635,N1(C(C=C(C)Cl)=O)C2CCC1CC(N(C)C(c1ccncc1Br)=O)C2 49636,S(=O)(=O)(c1ccc(C(N2CCC(C(C)NC(c3cc[nH]c3)=O)C2)=O)o1)NC 49637,c1(CN2C(C(C)C)CN(C(=O)C(C)(C)Br)CC2)ccc2nc(O)oc2c1 49638,C1(C)(CNC(CC2C(OC)CC2)=O)CCN(C(=O)CC2CCC(=O)NC2=O)CC1 49639,C1(CCOC)(NC(=O)CC2(CO)CC2)CCN(C(C2CC2C(C)O)=O)CC1 49640,N1(C(C(COC)N(C)C)=O)CC(CNC(=O)CCn2ccc(C)n2)C2(CC2)C1 49641,c1(CC(N2CCC(CNC(c3ccnn3CCl)=O)C2)=O)cccc(C(F)(F)F)n1 49642,CC(C)C(O)CCNC(C1CC=CCN1C(C1CC2C=CC1O2)=O)=O 49643,C(C(CNC(=O)CC1CCC(=O)N1C)C(F)(F)F)NC(c1c(SC)nn(C)c1)=O 49644,Fc1cccc2c1CN(c1nccc(=NCCN3CCCS3(=O)=O)[nH]1)C2 49645,n1(CC)ccc(C(=O)N(CC(C)O)C)n1.c1(OCC(=O)NCC(CO)N)cnn(C)c1 49646,c1(OCC(N2CCC(N(C)Cc3cccnc3O)C2)=O)cc(F)cc(Cl)c1 49647,CCC(C)C(=O)N(C)CC1(O)CN(C(C2C=C(C)CS2)=O)C1 49648,c1(C(N2CC(NC(C(CCC)O)=O)C(OC)C2)=O)cnc2c(c1)CNC2=O 49649,Cc1ccc(CC2(C(N)=O)CC3CCC2CC3)c2c1N(c1ccncn1)CCC2 49650,c1(NCC(C)CCCO)[nH]c(=NC2CC3(CCCC3)C2)nc2c1ncn2C 49651,CC(C)CCCC(C)NC(=O)CN1CCN(C(C2C=CC=CC=C2)=O)CC1 49652,N1(C(c2c(C)csn2)=O)CCN(C(c2ccc(F)cc2O)=O)C2CCCC2(C)C1 49653,N1(C(C2(COC)C=CCC2)=O)CCCC(NC(c2nnsc2SC)=O)C1 49654,CC1=C(C(=O)NC(CNC(c2cc(C(F)(F)F)n[nH]2)=O)CC(F)(F)F)CCCO1 49655,N1(C(Cn2c(C)ncc2)=O)C2CCC(C2)C1CNC(C1COC2(CCC2)C1)=O 49656,N1(C(Cc2ccc(OC)nc2)=O)CC(C2CCCN(C(=O)C(C)(C)C(C)O)C2)C1 49657,N1(C(c2n(CC#C)cnn2)=O)CCC2C(C(=O)N(CC(=O)NCC)C)C2C1 49658,Cn1ccc(C(N2CC(C)(NC(=O)CC3(O)CCOC3)C2)=O)c1C1CCC1 49659,C1(NC(C2CC2(F)Cl)=O)CCN(C(=O)C(C2CCCC2)C2CCCC2)CC1 49660,N1(C(C2CC(SC)C2)=O)CC2CC2(NC(=O)COCc2cccc(OC)c2)C1 49661,C1(SCC(CCNC(C2C(C)CN2C(=O)NC(C)(C)C)=O)F)CCC(C)(C)CO1 49662,c1(C(N2CC(NC(C3(OC)CCOC3)=O)C2)=O)cc2c(C)c(Cl)ccc2[nH]1 49663,N1(C(CCC2CC(OC)C2)=O)CCCN(C(c2cc(C#N)ccc2C)=O)CC1C 49664,Cc1cc(N2CCOCC2)cc(NC(c2ncc(F)cc2N)=O)c1 49665,C1(CNC(c2ncn(CC)n2)=O)(CO)CCCN(C(C2CCCC(F)C2)=O)C1 49666,c1(N(C2CCCO2)C(N(C2CN(C(=O)OC(C)(C)C)C2)C)=O)ccc(F)c(F)c1F 49667,c1(C(=O)NC2CC(CNC(Cc3c(C)nsc3)=O)C2)coc2c1CCCC2 49668,C1(C(=O)NCCC(C)NC(c2nc[nH]c2C(C)(C)C)=O)CCCCN1S(N)(=O)=O 49669,CC1CCN(C(=O)C(N2CCC(C)(c3ccccc3)C2)=O)CC1C 49670,CC1=NOC(C)(C(=O)NCCC(=O)NCCS(C)(=N)=O)C1 49671,C1(CC(N2C(CNC(CSC)=O)COCC2)=O)CN2CCN1CC2 49672,Cc1ccc(NC(C2CCN(C(C(=O)NCCC3(NC(C)=O)CC3)=O)CC2)=O)cc1 49673,c1(NCC(CC)Oc2ccccc2)nc(N(CC(Cl)Cl)C)nc2ncn(C)c12 49674,CC1CC(=O)NCC1C(N1CC(C(C)NC(c2cc(Br)c[nH]2)=O)C1)=O 49675,CC1CC(NC(c2cc(CF)on2)=O)CN(C(c2c[nH]nc2C2CCC2)=O)C1 49676,C12(NC(c3c(C)cc(C)s3)=O)CCOC(CNC(C3CCC(=O)NC3)=O)(C1)C2 49677,CCCC(C)(O)CC(=O)NCC1CC(F)CN1C(=O)Cc1nccs1 49678,Cc1oc(C(=O)NCCC2(O)CN(C(c3ccc(C(C)C)cn3)=O)C2)cc1CO 49679,C#Cc1ccc(CC(N2CCOC(C)(CNC(c3cnnc(O)c3)=O)C2)=O)cc1 49680,c1(C(N2CCC(NC(c3n(C)nc(C4CCC4)c3)=O)C2)=O)c(F)cc(Cl)cc1F 49681,c1(C(N2CCCC(O)(CNC(CCCOC)=O)C2)=O)cc(OC)cc([N+](=O)[O-])c1 49682,CC1CC(C)(C)CN1CCO.c12cn(nc1C1CCCCC1)CCNC2 49683,Cc1c(Br)sc(CNCC(=O)CC(C)C)c1Br 49684,c1(C(N2CCC(OC)(CNC(c3cocn3)=O)C2)=O)ccc(F)c(CSC)c1 49685,N1(C(CCCCN(C(c2cnn(C=C)c2N)=O)C)=O)CCC2(CCC2)C(O)C1 49686,N1(C(C(C)SC(C)C)=O)CCC2C(C1)CN2C(=O)CCCc1ccc(Cl)c(Cl)c1 49687,c1(N2CCCC(NC(C)=O)C2)ncnc(NCC2CCCC2(C)C)c1C 49688,C1(C(=O)NCCC2CCCN2C(=O)C2CC2)CCN(C(c2n[nH]cc2F)=O)CC1 49689,C1(N(C)C(C2CC23CCC3)=O)CC2CC1N(C(c1ccc(N)cc1F)=O)C2 49690,C1(CNc2c(Br)cnc(C(=O)OC)n2)(OC)CC(C2CCC2)C1 49691,N1(C(c2c(SC)ccs2)=O)CCOC2(CCN(C(C3CCOCC3)=O)CC2)C1 49692,C1(NC(c2cnsn2)=O)CC12CCC(NC(c1cccc(F)c1Cl)=O)CC2 49693,Cc1cnc(C(N2CCC(C)(C(N3CC(N4CCCC4=O)C3)=O)CC2)=O)c(F)c1 49694,Cc1oc([N+](=O)[O-])cc1C(=O)N(CCCNC(=O)C=CC1CCCN1C)C(C)C 49695,CN=c1nc(C(=O)NCCC(C)(C)NC(=O)CSCCC(C)C)cc(C)[nH]1 49696,c1(C(N2CCC3(C2)CC3(F)F)C(=O)NC2(C)CC2)cnc2ccc(Cl)cn12 49697,C1(COC)(CNC(C2CCCCC2O)=O)CCCN1C(=O)CC1(C)OCCO1 49698,c1(CCNC(C2(CNC(=O)COC3CCOC3)CC(=C)C2)=O)ncc(C)cn1 49699,C#CCC(C)(C)C(=O)OCC1CCC(NC(c2n[nH]cc2OCC)=O)C1 49700,N1(C(c2cc(Cl)c(Br)s2)C(=O)NCCOCC)CC2CCCC1C2CSC 49701,c1(OC)ccc(NCC(Cc2ccc(N(C)C)cc2)N(C)C)cc1OC 49702,O=C(CCCCCCCO)NC1CC(CC(=O)NCc2nnco2)C1 49703,c1(C(=O)NC(C)CCNC(C2(F)CCCC2)=O)cc(Cl)cc(Br)c1N 49704,N1(C(C2CC(OC)C2)=O)CC2CCC(NC(c3c[nH]cc(F)c3=O)=O)CC2C1 49705,C1(NC(C2CCC(C)C2)=O)CN(C(C2C3CCCC23)=O)CCC12CCC2 49706,n1(CC(N2CC(CC(C)NC(C(C=C=C)C)=O)C2)=O)ccc2ccccc2c1=O 49707,C(=O)(CC(C)(C)Cn1ccc(C(=O)O)n1)NC(N1CC(=O)CCC1=O)C 49708,c1(CCC)onc(C)c1C(=O)NC1CN(C(=O)CCc2ccc(OC)cc2)C1 49709,C1(NC(C=CCOCCOC)=O)COCCN(C(c2cnc(S)n2C)=O)C1 49710,C=C(C)C(CC(=O)NC1CN(c2nc(SC)ns2)CCC1C)OCC 49711,C12(C(N(C3CCN(C(c4ccc(Br)cn4)=O)CC3)CC)=O)CC(C)(C1)OC2C 49712,c1(CC)cccc(C(=O)N(C(C)CN(C)C(C2(Br)CC2)=O)C)n1 49713,C(CCCC(C)(C)C(=O)NNC(=O)c1csnn1)NC(c1cc(CC)nc(Cl)c1)=O 49714,N1(C(Cc2cnc(C)[nH]2)=O)CC2CCC(C1)C(NC(C1CCC3CC13)=O)C2 49715,CC1CC(C)CN(C(=O)CC2CC(NC(=O)CN3CCCCC3C)C2)C1 49716,C(=O)(C(O)CC(F)F)NC(CC)CNC(=O)Cc1cc(-c2ccccc2Cl)on1 49717,c1(C(=O)NCC(CCNC(CC(C)(C)C)=O)(C)C)cc2ccccc2cc1N 49718,C(=O)(C1=C(F)CN(C(=O)C(C)C(C)CC)CC1)NC1CCN(OCC)CC1 49719,N1(C(CCCCOCC)=O)CCN(C(c2cn(CCO)nc2C)=O)C(C2CC2)C1 49720,c1(C(N2CCC(c3cccc(F)c3)C2)=O)cn2ccnc2s1 49721,C1(NC(C2CCC(C)O2)=O)CCCC(C(N2CCOC(C3CCC3)C2)=O)C1 49722,c1(OC)cnc(F)cc1C(=O)NC1(CNC(c2nnsc2C)=O)CCCCC1C 49723,Cc1ccc2c(C(N3CC(CC(C)NC(C4(S(N)(=O)=O)CC4)=O)C3)=O)coc2c1 49724,C1(C(=O)NCCC(=C)CNC(=O)CCOCC(F)(F)C(F)F)CCCC(C)C1 49725,c1(C(N(C(C)CNC(=O)C(C)=CC2CC2)CC)=O)ccc(C(N)=O)nc1 49726,C1(C(N(CC)Cc2ccsc2)=O)(CC)CCCN(C(c2ncc(C)cc2F)=O)C1 49727,c1(C(=O)NCC2(CNC(c3c(CC)ocn3)=O)CC2)ccc(F)c(C2CC2)c1 49728,n1(CC(=O)NC23CCN(C(c4ccc[nH]4)=O)CC2C3)nc2n(c1=O)CCCCC2 49729,C(CC(C)C(=O)N(C1CCC(CNC(c2cc(Cl)cs2)=O)CC1)C)=CC 49730,C1(C(N2CC3(OCC(NC(CCSCCC)=O)C3)C2)=O)CCc2nncn2CC1 49731,C1(C(N(C)Cc2ccc(CC)o2)=O)CCCN(C(=O)COC(C)=O)C1CC 49732,CCC(C)(CNC(=O)C(F)OC(F)(F)F)C(=O)NCC1(CN=[N+]=[N-])CC1 49733,c1(C(=O)NC(c2ccccc2)CNC(c2cn(CC)nn2)=O)cccc(SC)n1 49734,CC12CCC(C(=O)NCCC3CN(C(C4CCCCCC4)=O)C3)(CC1)CO2 49735,c1(CC)ccc(F)cc1C(N1CCCC1C1(O)CN(C(C2CC2(Cl)Cl)=O)C1)=O 49736,c1(CS(N2CCC(NS(CCC)(=O)=O)C2)(=O)=O)cc(F)ccc1Br 49737,C1(CC(=O)N(C(c2ccccn2)C)C)CCCN(C(C2CCCO2)=O)CC1 49738,N1(C(c2cc(C)nn2C)=O)CCn2nc(C(=O)NC3CCC(CO)CC3)cc2C1 49739,C1(NC(=O)OC(C)(C)C)CC2CCC1(Nc1cnc(O)nc1O)C2 49740,c1(CC)c(C(=O)NC2CCCC2CNC(=O)Cc2csc(C)c2)csc1C 49741,N1(C(C(C)SCCCC)=O)C2CCC1C(C)C(NC(c1nc(C)oc1C)=O)C2 49742,c1(OC(C(=O)N(CC(C)NC(=O)C(C)n2ccnn2)CC)C)ccc(C)cc1 49743,c1(C(N2CC(F)(CNC(c3cc(C(F)F)no3)=O)C2)=O)nccc(F)c1Cl 49744,N1(C(=O)NCc2c(OCCOC)cccc2)CCCC(CO)CC1 49745,C(=O)(C(CNC(=O)Cn1ccnn1)N(C)C)N(C(C(C)SC)C)C 49746,N1(C(CN(C(c2cnc(O)cc2C)=O)CC)=O)CCSC(C)C1C 49747,c1(CC(=O)NC(C)CC2CN(C(C3CC(C)(O)C3)=O)C2)cc(F)ccc1Br 49748,Cn1cccc1C=CC(=O)NC(CNC(C1CSC1)=O)C1CC1 49749,O=C(C(O)CC(F)F)Nc1ccc(N2CCCNC2=O)nc1 49750,C1(C(=O)NCCOCCNC(c2nn(CC)nc2C)=O)C2CS(=O)(=O)CC12 49751,N1(C(c2nc(CC)oc2)=O)CC(OC)CC(NC(c2cccc(C)c2)=O)C1 49752,C1(C(N(C)CC2(NC(C(C)Oc3cccc(C)c3)=O)CC2)=O)CC2(CCCC2)C1 49753,C(CCCCCNC(=O)CCc1cccnc1Br)N(C(C1C(=C)CC1)=O)C 49754,C(=O)(CCCN(C)N=O)N1CC(CCCNC(CCC2CC(OC)C2)=O)OCC1 49755,c1(CC)cnccc1C(=O)NC1CC(C(=O)NCC(c2ccccc2)F)C1(C)C 49756,N1(C(CCNC(=O)OC(C)(C)C)=O)CCC2(CC(NCC3CC(F)(F)C3)C2)C1 49757,C=CC(CCC)CC(=O)NC(C(=O)NC1CCCCCC1F)C(C)(C)C 49758,N1(C(c2cn(CC)nc2)=O)CCCC(C(C)NC(c2c[nH]c(C(=O)OC)c2)=O)C1 49759,c1(OC)cc(C(N2CC3C(NC(=O)CN4CC(C)C4)C3C2)=O)c(OC)cc1Cl 49760,c1(C(N2CCN(C=O)CC2)C(=O)Nc2ccc(OCF)cc2)cc(Cl)c(Cl)c(Cl)c1 49761,N1(C(c2cc(C)nc(O)n2)=O)CC23CCCC2(C1)CN(C(C1(C)CCCO1)=O)C3 49762,N1(C(c2nc(C(N)=O)sc2)=O)CC2(COC(CNC(c3coc(Cl)n3)=O)C2)C1 49763,NCCCC(N)C(=O)N1CCC(CC(=O)NC2CCC(O)C2)C1 49764,C(=O)(CC(F)(F)C(C)(F)F)N1C(C)CCC(CNC(=O)CCc2cnc[nH]2)C1 49765,N1(C(C=C(C)C(C)C)=O)Cc2n[nH]cc2C1C(=O)N1CCC(C)(NC(C)=O)C1 49766,c1(N(C)CC2CCSCC2)nc2c(c(=NCC3(CO)CC3(C)C)[nH]1)CSC2 49767,C(=O)(C1=NOC2COCC12)N1C(C(=O)NCc2nn(C)cc2CO)(CC)CCC1 49768,Cc1nc(C2CCC2)sc1CC(=O)N(CCCNC(C1CC1CF)=O)C1CC1 49769,N1(C(CCC(CC)=O)=O)CC2(CCCC2NC(=O)C=CC2CCCN2C)C1 49770,c1(C(N(C2(CC(N3C(C(C)O)CC3)=O)CC2)C)=O)cc(C(N)=O)co1 49771,CC(CCCNC(=O)C(C)c1ccsn1)NC(=O)CSC(C)(C)C 49772,C1(NC(C2(C)C=CCC2)=O)COCCN(C(c2ccsc2-n2cnnn2)=O)C1 49773,N1(C(C=CC)=O)CC(F)(n2cc(COCCO)nn2)C1 49774,n1(CCC)cc(C(=O)NCCCC2CCCN2C(C2CCS2(=O)=O)=O)nn1 49775,N12CCC(CC13CCC3)NC2=O.N1(C(c2nc(C)cs2)CC)CCC(C)C1 49776,C1(C(=O)NCC2CN(C(Cc3cc(C)on3)=O)C(C)C2)CCC2(CCOCC2)O1 49777,c1(NC(c2cccc(NC)c2)=O)c(OC)nc(Cl)nc1C.C(=O)(CC(C)SC)NC 49778,c1(OC)ccc(CNC(CC(C)OC)c2nnnn2C2(C)CC2)c2ccccc12 49779,C=Cc1ccc(C(N2CCN(C(C3C(F)(F)C34CC4)=O)C(CO)C2)=O)cc1 49780,CC1OCCCC1C(N1CCC(CCC(=O)NCCCN2CCOCC2)CC1)=O 49781,C1(C2CC2)(C(N(CC(C(C)C)C)C)=O)CN(C(C2CCCSC2C)=O)C1 49782,c1(C(N2CC(CC=C)(NC(C3CC=C(C)CC3)=O)C2)=O)ccnc(OCC)c1F 49783,n1(CC)ncc(C(=O)NCC2CCN(C(=O)CN(C(=O)COC)C)C2)c1C1CC1 49784,C1(NC(C(C)Oc2ccccn2)=O)(CNC(C2(C(N)=O)CC2)=O)CCOCC1 49785,c1(C(C)=O)cc(=NCCCOCCNC(c2nc(Cl)sc2Cl)=O)[nH]cn1 49786,Cc1nn2cccnc2c1C(=O)NCC1COCC1NC(c1nc(O)sc1C)=O 49787,N1(C(C2CCC(=O)N2)=O)CCN(CCO)CC1.C1(NC)CC(OCF)C1 49788,n1(CCC)nnnc1C(c1ccc(CCC)s1)NCCc1ccoc1 49789,c1(C(=O)NC(C)CN(C(=O)Cc2ccc(F)cc2)C)c(F)ccc(Cl)c1F 49790,CC1CN(C(=O)C=C2CCN(C)C2)CCCN1C(=O)CN1CC(=O)N(C)C1=O 49791,c1(OCC(=O)NCC(C)N(C)C(c2ccc(CC#N)cc2)=O)ccc(Cl)cn1 49792,C1(C(=O)NCC2(C=C)CCOCC2)CCN(C(C2(F)CCOC2)=O)CC1(C)C 49793,Cc1cccc2c(C(=O)NCC3CC3NC(=O)CSc3cccc(Cl)c3)n[nH]c12 49794,N1(C(CN2C(C)CCC2C)=O)CCC2(CCCN(C(=O)CCCCF)C2)C1 49795,c1(C(N2CC(NC(=O)COc3ccc(Br)cc3)C2)=O)ccc2nncn2c1 49796,N#Cc1cc(CN2CC(O)(CNC(c3ccc(Cl)c(O)c3)=O)C2)ccc1Cl 49797,C12(C(N3C4C(NC(c5cc6c(s5)CCC6)=O)C(C4)C3)=O)CCC(O)(CC1)CC2 49798,C1(CNC(CNC(CNC(C2C(C)(C)CCO2)=O)=O)=O)CC2CCCC2C1 49799,N1(C(c2c(C)nccn2)=O)CCC(NC(=O)COC2(C)CCC2)C12CC2 49800,CC1(C)COCCC1C(N1CCC(CCNC(=O)C=CC2CC2)C1)=O 49801,CN1CC2(CCN(C(=O)CC3CCN(C(c4cccc(C5CC5)c4)=O)C3)CC2)C1 49802,C1(C(N2CC(C)(C(C)C)OCC2)=O)COC2(C1)CC1(CN(C(=O)OC(C)(C)C)C1)C2 49803,N1(C(C2C(NC(C(C)n3ccnc3)=O)C3CCC2C3)=O)CCc2nc[nH]c2C1 49804,Cc1cccc(CC(C(=O)NCC2CCCC2)NC(=O)OC(C)(C)C)c1.C(C)(C)(C)O 49805,c1(NC(CSc2ccc(C)cc2)C)ccc2ncc(I)n2c1 49806,c1(C(C)(F)F)csc(C(=O)NC2(CO)CN(C(c3csc(Cl)c3)=O)C2)n1 49807,N(C(=NCc1cnn(C)n1)NCC(F)F)C(C)CCc1ccccc1 49808,c1(C(=O)NC2C(NC(CCOC)=O)CCC2)cc2c(cc1Br)OCO2 49809,c1(CC)ccc(NC(=O)C(C)=CCNC(=O)CC2C=NN(C)C2=O)c(F)c1 49810,N1(C(C2C=CC=CC=C2)=O)CC2CC1CN2C(c1cc(C2CC2)nc(O)c1)=O 49811,CC1CC=C(C(=O)NCC23CCC(CC2)N(C(C2CC4CC2CC4O)=O)C3)CC1 49812,C(=O)(C1=C(c2ccccc2)CCC1)NCC(CC)(C)NC(c1cnnc(C)c1)=O 49813,CC1CCC(CCNC(=O)C(Cc2ccoc2)NC(C2CCC(O)C2)=O)CC1 49814,C(C)(CCC(=O)N(CCCNC(=O)Cc1cnc(C)o1)C)SC 49815,c1(NC)ccc(NCCCCC(=O)N(C)CCNC(=O)NC(C)(C)C)cc1C 49816,C(C(C(C)C)NC(c1ccccn1)=O)(C1CCCCC1)NC(CCCC)=O 49817,CN1CC(F)CC1C(N1CCC(C(C)(C)NC(=O)CC2CNC(=O)O2)C1)=O 49818,Cc1cnc(NCC2CCCCC2C(=O)NC(c2ccc(Cl)cn2)C2CC2)c(C)c1 49819,N1(C(C(C2CCN(C(c3cc(C(C)=O)on3)=O)C2)C)=O)CCc2nnnn2CC1 49820,CCC(CNC(C1(F)C(C)(C)C1(C)C)=O)N=c1[nH]nc(C(F)(F)F)s1 49821,N1(C(C2CCC(C)O2)=O)CCCC2C1CCN2C(c1cccc2c1CC(=O)N2)=O 49822,c1(CC)sc(C(=O)NCC2(C)CCN(C(=O)C(c3cccnc3)C)C2)cc1C 49823,CC1CCC(CC(=O)N(C)CC2(CNC(=O)C=Cc3cc[nH]c3)CC2)C1 49824,c1(C(CNCCOc2ccc(C(=O)OCC)cc2)C)cc(F)cc(F)c1 49825,C1(C(=O)NCCOCCC#C)C2CC3C(C2NC(=O)C(C)(C)Cl)C13 49826,C1(C)(CC)CC(C(=O)NC(C)CNC(=O)CC#N)CCO1 49827,c1(C(N(C(CNC(CCc2ncc(C)[nH]2)=O)C2CC2)C)=O)ncccc1C(F)F 49828,Cc1nnn(C)c1C(N1CCC(C)(CNC(c2ccccn2)=O)C1)=O 49829,c1(C(=O)NC2CCN(C(C(C)=CC)=O)C2CC)cnn2cccc(Cl)c12 49830,C1(C(N2CC3(CN(C(C4C(c5ccn(C)n5)C4)=O)C3)C2)=O)CCC2(CCOC2)O1 49831,C#CC1CN(C(=O)CN(C)C(C)C)CCN1C(=O)CC1(C2CC2)CC1 49832,N1(C(c2ccncc2Br)C(=O)NCc2cccc(OC)c2)CCCC(O)CC1 49833,CC1(C(=O)N(CC(O)CO)C2CC2)CCN(C(=O)C(=O)NC2CC2)CC1 49834,CC(O)C(C(=O)N1CCN(C2CCC2)CC1)NC(=O)CC1CC2C=CC1C2 49835,CC(C)(C)C(CNC(c1ccc2cc[nH]c2n1)=O)C(=O)N1CC2(CCC2)CC1CO 49836,C1(NC(c2cc(C)ns2)=O)CC2C1CCN2C(c1cnn(C(C)C)c1C)=O 49837,c1(C(N2C(C)(CNC(CC(CC)OC)=O)CCC2)=O)ccc2c(c1)CNC2=O 49838,Cc1cc(C)c(C(=O)NCC2CCC(NC(=O)CSC(C)C)CC2)c(O)n1 49839,N1(C(C2C(=C)CC2)=O)CCN(C(c2cc(C(C)C)on2)=O)C(c2ccccc2)C1 49840,C1(CCOC)(NC(=O)CSc2nncs2)CCN(C(c2ccc(CO)cn2)=O)C1 49841,CC1CC(CO)(O)C1.c1(CC(=O)NCC=C(C)C)cccs1 49842,N1(C(c2c(C)nn(C)c2C)=O)CC(C)OC2(CCN(C(=O)CC3CSC3)CC2)C1 49843,Cc1ccc(C(=O)NCC2(O)CC(NC(C3CCN(C)C3=O)=O)C2)cn1 49844,C1(NC(=O)COC2CC2)CC2CN(C(c3cc(Br)c(F)cc3F)=O)CC2C1 49845,C1(CNC(=O)C(F)C(F)(F)F)CC2CCC(C1)N2C(c1ccc2c[nH]nc2n1)=O 49846,S(=O)(=O)(c1ccc(=NCCOCCO)[nH]c1)NCCCN1CCOCC1.CN1CC1 49847,C1(C(C)(C)CNC(C2(CO)CCCC2)=O)CCCCN1C(C1CCOCC1)=O 49848,N1(C(C2C(CC)CCO2)=O)CCCC(C(=O)NCC(=O)OC(C)C)CC1 49849,C1(n2cc(-c3c(C)nccn3)nn2)CC2CCC1(NC(=O)Cn1cc(Cl)cn1)C2 49850,N1(C(c2c(NC)ccc(Cl)c2)=O)CCC=C(C(=O)N(C)Cc2ccncc2)C1 49851,N1(C(C23CC(n4cc(CCSC)nn4)C2C3)=O)CCN(CCN(C)C)CC1 49852,C1(NC(C#CC2(C)CC2)=O)CN(C(C2CC3(CCC3O)C2)=O)C2(CCC2)C1 49853,C#CCC(C(=O)NC)NC(c1cc(CNC(c2nccnc2C)=O)[nH]n1)=O 49854,C1(O)(CNC(CCOCCN(C)C(c2ncc[nH]2)=O)=O)CCOC1 49855,c1(C(=O)NCC(CNC(=O)C(O)C(F)(F)F)OC)cccc(S(C)(=O)=O)c1 49856,C1(C2CC2)(NC(c2c(C)nc[nH]2)=O)CCN(C(=O)CC2OCCOC2(C)C)C1 49857,c1(OC)cccc(CN2CCC(CNC(c3c(C4CC4)noc3C)=O)CC2)c1 49858,CC1(C)CC(F)(F)CCC1C(N1CCOC(CCNC(=O)C2=CCC2)C1)=O 49859,n1(CC)cc(C(=O)NCC2C3CC2N(C(=O)CC2CCSCC2)C3)c(C)n1 49860,c1(OC)ccc(F)c(C(=O)NC2CCCCC2NC(c2cccnc2)=O)c1F 49861,C1(C(=O)Nc2cn(CC(=O)OC)nc2)CCC(NC(=O)CNC=O)CC1 49862,Cc1cc(C(N2CCCC(CNC(=O)CC3OCCCC3(C)C)C2)=O)ccc1N 49863,C1(C(N2CC(C(=O)NCc3ccnc(Cl)c3)(CC)C2)=O)C2CCC(F)(F)C12 49864,C1(NC(C2(COC)C=CCN2C(=O)CCc2ccc[nH]2)=O)CCCCCC1(C)C 49865,c1(C(N(CC(C)NC(C2CCC3(CCC3)O2)=O)C)=O)csc(S(C)(=O)=O)c1 49866,CC1(C(=O)NCCNC(=O)CCc2nc(O)n[nH]2)CCc2ccccc21 49867,C1(C(N2CC(F)(CNC(C(C)(C3CC3)OC)=O)C2)=O)CCC(C)(C)OC1 49868,c1(CC(=O)NC(C#C)(C)C2CCC2)c(C)nn(C)c1Cl 49869,N1(C(c2cnc(C(=O)OC)o2)C(=O)NCC=C)CCOC(C)(C2CC2)C1 49870,C1(n2cc(CNC(C)=O)nn2)CCN(C(c2ocnc2C)=O)CC1 49871,c1(SC)nc(=NC2CCCN(C(c3ccccc3C(C)(F)F)=O)C2)s[nH]1 49872,C1(CNC(CCC(C2CCC(C)CC2)=O)=O)C(C)CCCN1C(=O)CSC(F)F 49873,c1(C(N(CC(CC)NC(CC2(OCC)CC2)=O)C)=O)cnn(CC)c1 49874,N1(CCCCCCC)C2CCCC1COC2 49875,C=CC1(CC)COCCN1C(c1ncc(Br)cc1Cl)C(=O)NC(C)(C)C 49876,c1(C(N2CC3CN(CC)CC3C2)C(=O)NC2(C)CC2)cc2ccccc2nc1C 49877,Cc1ccc(CC(N2CC3(CNC(c4ccc(C)n4C)=O)CCC2C3)=O)cc1F 49878,Cc1cc(C=CC(=O)NC2COCC2CNC(=O)CCc2cccs2)on1 49879,N1(C(C(COC(C)C)(C)C)=O)CCCC(NC(c2cnc(O)c(F)c2)=O)C(F)C1 49880,c1(C(=O)NC(C)CCCCNC(=O)C2CC2)coc2c1COC2 49881,N1(C(CCC=C)=O)CC2(CCC2)CCC1CNC(=O)CCCF 49882,N1(Cc2c(F)cc(OC)c(I)c2)CCC(C)(C)CC(C)(C)C1 49883,N1(Cc2cc(C)c(Br)cc2C)CCC2CN(c3ncc4[nH]cc(I)c4n3)CC2C1 49884,C1(NC(C2CCC(OC)CC2)=O)CCN(C(=O)C(c2ccnn2C)O)CC1O 49885,N1(C(C2C(=C)C2)=O)CCN(C(c2ncc([N+](=O)[O-])n2C)=O)C2(CCC2)C1 49886,c1(SC)cccc(F)c1C(=O)NC1CCN(C(=O)CCC(C)(C)C)C1(C)C 49887,c1(C(=O)NC2C(NC(c3cc(C)nn3C)=O)CC2)c(C)nc(O)nc1C 49888,C1(CC=C)(NC(=O)CC2CCCOC2)CCCN(C(c2ccc(CC)[nH]2)=O)C1 49889,c1(C(CCOCC)NC(=O)C(C)O)cc(C(F)(F)F)ccc1C(F)(F)F 49890,c1(OC)cc(C=CC(=O)NCCOCCCNC(=O)CCCCC#N)ccc1F 49891,c1(C(=O)NC(C)(C)CCCNC(=O)CN2CCCCC2)nccc(Cl)c1Cl 49892,c1(NC(C2CSCCN2Cc2cc(F)c(O)c(Br)c2)=O)ncc(Br)cc1[N+](=O)[O-] 49893,C(=O)(CCCC1CC1)N(C1CCN(C(c2cc(-c3ccccn3)ns2)=O)C1)C 49894,C1(C(N2C(C)(C)CC(NC(c3cc(Cl)ccn3)=O)C2)=O)CN2CCCCC2CO1 49895,c1(NS(CC)(=O)=O)ccc(C(=O)NC(CNC(C2(C)CCNC2=O)=O)CO)cn1 49896,c1(C(=O)NC(CNC(c2cc(CSCC)on2)=O)C2CCC2)cc(Cl)ccc1O 49897,c1(CONC(C2C(CNC(c3ccc(CC)[nH]3)=O)CCCC2)=O)ccc(O)c(C)c1 49898,C1(CNC(C(CC)(C)OC)=O)C2CCC(C2)N1C(=O)CCc1ccc(Cl)cc1 49899,c1(CC)ccc(C(=O)NCC(C2CC2)N(C(=O)C(N2CCNC2=O)C)C)[nH]1 49900,N1(C(C(CCCC)C)=O)CC2=C(C1)CN(C(C1CCCCC1CC)=O)C2 49901,Cc1cc(Cl)c(C(=O)NC(C2CN(C(c3cnc(S)nc3)=O)CCO2)C)cc1N 49902,N1(C(c2ccc(SC)o2)=O)CCC(NC(=O)Cc2sc(C)nc2C)CC1C1CC1 49903,N1(C(CCC=CC(C)C)=O)CCN(CCNC(C2(C)CC=CCC2)=O)CC1 49904,C1(NC(c2c(C)ncc(C)c2)=O)CCCC12CCN(C(c1cn[nH]c1)=O)C2 49905,c1(C(N(C(CCNC(c2c(C)nn(CC)c2Cl)=O)C)C)=O)cccc2c1CCN2 49906,c1(C(C)NC(=O)CN(C(=O)CCC2CC2(F)F)C)nncn1C 49907,C(=O)(C(F)(F)CC)NCCC(C)N(C(C1N(C(CC)=O)CSC1)=O)CC 49908,C1(C(=O)NCC(C(C)C)NC(=O)CCn2cccn2)CCC2(CC2)C1 49909,c1(C(=O)NC2CC(C(C)NC(c3cccs3)=O)C2)nc(O)nc(O)c1N 49910,c1(-c2scc(C(N3C(CNC(COCC=C)=O)CC3)=O)n2)ccc(O)cc1 49911,c1(C(=O)NC2(COC)CCN(C(c3ccccc3)=O)C2)ccc(=O)n(C)n1 49912,N1(C(C2(CC)COC2)=O)CCCC1(C)C(=O)NC(c1ccc(F)cc1)CO 49913,C(CC(F)F)(C(=O)NCC(=O)NC1CCCC1)N(C(c1cncc(CC)c1)=O)C 49914,C(C(=O)N(CCCCCCNC(=O)C=C1CCC(C)C1)C)(C(C)C)OCC 49915,C1(C)(C(N(CCC)CCNC(c2ccc(Cl)o2)=O)=O)SCCCS1 49916,C1(NC(C2CC(CNC(C3C(C)CCOC3)=O)C2)=O)CCCCC1N=[N+]=[N-] 49917,Cc1nn(C)c(Cl)c1C(=O)NC1CCCN(C(c2scnc2C2CC2)=O)C1C 49918,c1(N2CC(C)OCCC2)nc(N2C3CCC2COC3)nc2c1COC2 49919,c1(N2CCC(NC(c3c(C)cc(OC)cc3C)=O)C2)ncnc2cc(C)[nH]c12 49920,C1(CC)CN(C(c2scnc2C)=O)CCN1C(c1nocc1Br)=O 49921,C#Cc1cnc(C(=O)NC(CC2CCC2)C(=O)N(CCC=C)C)c(C)c1 49922,C1(CCC)CN(C(c2cnc(Br)c(OC)c2)=O)CCN1C(=O)CCSC 49923,C(=O)(CC(CC1CC1)NC(C1(CC)CCOC1)=O)NCC(CC)O 49924,N1(C(C2(C)CC2)=O)CC2(C1)CN(C(c1csc(Cl)c1Cl)=O)CC2CO 49925,c1(C(=O)NCC(C)NC(c2ccnc3c2CCC3)=O)cc(C#N)c(F)cc1F 49926,C1(OC)CN(C(c2c(Cl)cccc2Br)=O)CCC1NC(C1C2COCC12)=O 49927,C1(C(=O)NC(CNC(COCCC)=O)C)CCCN1C1CC1 49928,N1(C(c2c(F)ccc(C)n2)=O)CC2CCN(C(=O)CCC3CCC(C)O3)CC12 49929,N1(CC(N2CC(O)(CNC(C3(c4cccnc4)CCCC3)=O)C2)=O)CSCC1=O 49930,N1(C(c2c(C)n[nH]c2)=O)CC2(CC(CNC(=O)CCc3ccc(F)nc3)C2)C1 49931,N1(Cc2cnc(SC)nc2)CCCC(C(=O)Nc2cc(I)ncn2)CC1 49932,C(C(C(=O)N(CCC1CC1)CC)NC(c1ccc(CC)s1)=O)OCC 49933,C1(C(=O)NCC2C3CN(C(=O)CCN4CCOC4=O)CC23)CCc2cnnn2C1 49934,c1(C(=O)NC2C(C)(C)CN(C(=O)CC3OCCO3)C2)cnc2nccn2c1 49935,CC1CC2(CC(C(=O)NCCC3CCC(NC(=O)CCN4CCCCC4)C3)C2)C1 49936,Cc1cccc(OCC(=O)NC2(COC)CN(C(c3ncccc3F)=O)C2)c1C 49937,c1(C(N(C(CNC(C(C)OC)=O)C)C)=O)ccc(F)c2c1OCC2 49938,CC(C)C(O)C(C)(C)C(=O)NC1CCN(C(=O)C2=CCCC2)CCC1CO 49939,Cc1ccc(F)c(CNC2(c3nnnn3CCN3CCOCC3)CC2)c1Br 49940,c1(OC)ccc(CC(=O)N(C(c2cn(-c3ccccc3)nn2)(C)C)C2CC2)c(C)c1 49941,C(N=c1ccnc(C(N)=O)[nH]1)C1CCCC(NC(CCNC(C(C)(C)C)=O)=O)C1 49942,C1(NC(c2coc(Cl)n2)=O)C2CC3CN(C(=O)C4=CCCSC4)C1C3C2 49943,C(=O)(CCCCCC(C)(C)C)N(CCCNC(CCc1ccc(C)s1)=O)C1CC1 49944,c1(OC)ncc(F)cc1C(N1CC2CC(NC(c3ccc(C)s3)=O)C1C2)=O 49945,N1(C(CCCCCC#N)=O)CCCC(C2(NC(=O)C=C3CCC3)CC2)C1 49946,CN1CCN(C(c2ccc(F)s2)=O)CC1C(=O)NCC1CCC(C)(C)O1 49947,c1(C(N(C(CC)C(=O)NCCOC(=N)O)C)=O)cccc2cc[nH]c12 49948,C(=O)(C1=CCCCCC1)NCC1(OC)CCN(C(CSCCCC)=O)C1 49949,C(=O)(CC(CC=C)NC(c1ccnc(O)c1F)=O)NC(C#C)CC1CCC1 49950,C(=O)(C(F)(F)C(O)C1CC1)NC1C(NC(=O)COc2ccccc2)COCC1 49951,c1(OC)cccc(NC(=O)COCCNC(c2csc(C(F)F)c2)=O)c1C 49952,c1(CC(=O)NC(CC)CN(C(C2(O)CCC2)=O)CC)ccc2scc(C)c2c1 49953,c1(C(N2C(=O)CC(NC(N3C4(C)CC4CC3)=O)C2)C2CC2)cc2ccccn2n1 49954,c1(C(=O)NCC(COC)NC(=O)C(OC)OC)cccnc1-n1ccnc1 49955,C1(NC(C(C)(C)C(F)(F)F)=O)CC(C2CCN(C(=O)CNc3nccs3)C2)C1 49956,c1(C(=O)OC)[nH]c(=NCC23CCC(C)(CC2)CO3)sc1C 49957,C(C(F)(F)C(F)(F)F)OCC.C#CCCC(=O)NCC12CN(C1)C(=O)CCO2 49958,c1(C(=O)NCCCCCCNC(=O)CC2CC(=O)NC2=O)cnc2[nH]cncc1-2 49959,c1(NCC(CCCC)NC(C2(C)CCCCN2)=O)cnc(C#N)c(C#N)n1 49960,CCCC(CC)C(=O)NC(C)C(CO)NC(c1cc(F)ccc1NS(C)(=O)=O)=O 49961,C1(CNC(C2(C)C=CCCC2)=O)CCN(C(=O)CCCS(N)(=O)=O)CC1C1CC1 49962,c1(OC)ccc(-n2cc(C(=O)NNC(=O)c3nn(C)nc3Br)nn2)cc1C 49963,N1(CC)CCCC1CC(=O)NCC#CCNC(=O)CCOCC1CC1 49964,c1(CN(CC)CC)ccc(C(=O)NCCC(C)NC(c2occc2C2CC2)=O)o1 49965,C1(OC)(OC)C(C(=O)NCC2(C)CCC(C3CC3)O2)CC1(F)F 49966,c1(CCC)ccccc1NC(c1ccc(N(C(=O)CC2CCCC2)CC)cn1)=O 49967,Cc1cncc(C(=O)N(C2CCCN(C(=O)CC=Cc3ccccc3)C2)C)c1Cl 49968,S(=O)(=O)(c1c(Cl)ccc2c1OCCO2)Nc1ncnc2sc(C)c(C)c21 49969,c1(SC)ccc(N)cc1C(N1CCC(NC(=O)Cn2cnnc2O)C1)=O 49970,Cc1nc2c(C#N)cnn2c(C)c1CCC(=O)NC(C)COC(F)(F)F 49971,C1(NC(C2CCN(CC)C2)=O)CCC12CN(C(=O)Cn1cc(C(F)(F)F)nn1)C2 49972,C1(C(=O)NC2CC(N(C)C(c3ncccn3)=O)C2)CC(=O)N(c2nccs2)C1 49973,C(CC(C)C)(C(=O)NCCOC(C)(C)CNC(=O)Cc1cscn1)NC(C)=O 49974,CCCC(CCC)CC(=O)NC1CC2(C1)CC2Nc1cc(Cl)ncn1 49975,c1(C(=O)NC(CC=C)CNC(=O)Cc2ccsc2C)cc2c(O)ncnc2cn1 49976,c1(CCO)nc(C2CCCN2Cc2ccccn2)n(-c2ccc(Br)cc2)n1 49977,C1(NC(CCC)=O)CC1C1CCCN(C(c2c(OC(F)F)cccc2Cl)=O)C1 49978,c1(N2CC(C)S(=O)C(C)C2)nc(=N)[nH]c(=NCc2cn3ccccc3n2)[nH]1 49979,CC1(C)CCN(C(c2cc(C3CC3)no2)=O)C1CC(=O)NC1CC1C1CCC1 49980,CCCCC(O)C(=O)NCCCOCCOCCNC(=O)CSc1ccc(Cl)cc1 49981,Cc1cc(C(=O)NC2CC2CNC(c2cc(Cl)c(Cl)s2)=O)c2nccn2c1 49982,C1(NC(C(C(C)O)N(C)C)=O)CCN(C(=O)CC2CC(C(C)(C)C)C2)CC1O 49983,c1(OC)cc(Cl)ccc1C(=O)NC1CCCC1CNC(C1CC2CCC1CC2)=O 49984,CC1(C(N2CCC(COC3CCN(C(c4cscn4)=O)C3)CC2)=O)CCCCC1 49985,c1(NC(C2CC2c2ccc(F)cc2)=O)c(F)ccc(C2CC2)c1F 49986,c1(-c2nc(Cc3c(OC)cc(C#N)cc3)on2)cc(Cl)cc(Br)c1F 49987,C(=O)(C1=CCc2ccccc21)NCCC(CNC(=O)CC1CC2(CC2)C1)O 49988,CCC(C)(C)CNC(=O)C(C1CCCC1)NC(=O)C=CC(C)(C)SC 49989,c1(C(=O)NCCn2cc(C(=O)NCC(=O)NCC(C)C)nn2)ncccc1F 49990,C(=O)(C(O)CC(C)C)NC1CCCC(CNC(CC2(OC)CCC2)=O)C1 49991,C1(C(N2CC(CNC(c3c(COC)ncs3)=O)(OC)C2)=O)CC12CCOC2 49992,c1(OC)ccc2c(CCC(=O)NC3CC(CNC(=O)CCF)C3)c[nH]c2c1 49993,C(CC(=O)NOCC1CC2C=CC1C2)C1CCN(C(c2[nH]cc(C(C)=O)c2)=O)C1 49994,N1(C(c2nn(CC)c(O)c2)=O)CC2(CCCC2)C1C(=O)NCC1=CCN(C)CC1 49995,C1(OC)CC(NC(=O)CCC2CC2(F)F)CN(C(=O)COC2CCC2)C1 49996,N1(C(c2n[nH]c(CC)c2Cl)=O)CCC2(CCC2CNC(=O)C(C)C(C)C)CC1 49997,c1(CCC)sc(C(=O)N(C)CC2(CNC(=O)C(C)(C)O)CC2)cc1CC 49998,c1(-c2cc(NCc3c(C)ccc(C(=O)O)c3)ncc2)ccc(C2=COCC2)cc1 49999,c1(C(N(CC(C)NC(=O)C(F)n2ccnc2)C)=O)cccc(N2CCOC2=O)c1 50000,c1(C(=O)NC(C2(O)CCN(C(C(=O)NCC)=O)C2)C)ccc2ncn(C)c2n1 50001,N(C(=NCC1CCCSCC1)NC1CCN(CC(F)(F)F)C1)C(CC)CC 50002,CCC(C)CCC(=O)N1CC2(C(=O)NCC3CCCC3OC)CC1CO2 50003,C(=O)(CCS(C)=O)N1CC(C(C)NC(=O)CC(c2ccccc2)N(C)C)C1 50004,CCCC(CCCNC(C1(C)CCN(C)C1=O)=O)NC(c1c[nH]nc1OC)=O 50005,N1(C(c2c(C)nc(CCC)o2)=O)CC(NC(C2CCC(N=[N+]=[N-])C2)=O)CC(C)C1 50006,N1(C(C=C(C)Cl)=O)CC2CC(NC(C3(CCN(C)C)CCCC3)=O)CC2C1 50007,Cc1oc(C(=O)NC2CCN(C(=O)C(C)(C)OC(C)C)CC2F)cc1S(C)(=O)=O 50008,c1(C(=O)NCCCCC(C)NC(c2cnc(C3CC3)o2)=O)cccc2c1CCN2 50009,C(=O)(C(C)C(C)S(C)(=O)=O)NCC(CC)NC(=O)C=Cc1ccn(C)c1 50010,CC(C)C(C(=O)N1CCC(C)(C)CC1C(N1CCCC1CF)=O)C(C)C 50011,c1(CC)ccc(C(=O)NCC2CC(F)CN2C(=O)CSCc2ccccc2)cn1 50012,c1(C(=O)NCC2N(C(C3CC(=C)C3)=O)CCOC2)c[nH]c2cc(OC)ccc12 50013,C1(N(C(C(CC)n2cccn2)=O)CCF)CCCN(C(=O)C=CC(C)(C)SC)C1 50014,CC1(C(=O)NCC2CC3CCC2N3C(C2(CO)CCC2)=O)CCCNS1(=O)=O 50015,C1(NC(C(C)c2ccsc2)=O)CCN(c2cnc(F)cn2)CC1O 50016,N1(Cc2cnc(-c3sccc3)o2)CCC2CC2C1 50017,C1(C)(NC(c2c(COC)c(F)ccc2)=O)COCCN(C(=O)CNC(=O)OC)C1 50018,C1(OC)CC(C(N2CC=CC(O)C2)=O)N(C(c2sccc2Cl)=O)C1 50019,Cc1cccnc1CC(=O)NC1CC(C)N(C(=O)CN2CCOCC2)C1 50020,N1(C(C2N(C(C(N)=O)=O)CC2)=O)CCOC2CC12 50021,C1(CC)C(NC(=O)COc2cccc(F)c2)CCN1C(=O)C(C)SC 50022,c1(CC)ncc(C(N2CCN(C(=O)CCn3cccn3)C(CC)C2)=O)c(O)n1 50023,C(=O)(C1=NOC(CNC(=O)CC2NC(=O)NC2=O)C1)N1CC(C(=O)OCC)C1 50024,c1(C(N2CC(Cn3cc(CC4CCCCO4)nn3)C2)=O)ccnc2cc[nH]c12 50025,c1(C(N(CC(C)NC(C2CCCN2Cc2nnn(C)n2)=O)C)=O)ccc(Cl)cc1 50026,Cc1cc(C(=O)NC2CC(F)(F)CC2NC(=O)C2=CCOCC2)cc(Cl)c1 50027,N1(C(CC2(C=C)CN(C(=O)CP(C)(C)=O)C2)=O)CCN(CC)C(=O)C1 50028,c1(C(N2CCN(C(=O)OCC)CC2)=O)cc(OC)nc2cc(Br)ccc12 50029,N1(C(C(CC)=CCCC)=O)CCC2CN(C(c3sc(C)cc3Cl)=O)CCC12 50030,CCC(C)(C(=O)NCC1CCC1NC(c1nc(=O)n(C)[nH]1)=O)OC 50031,N1(CCC2N(C)CCC2)CC(=O)N(CC2(n3ccnn3)CC2)C1=O 50032,c1(C(N2CC(O)(CNC(C3C(OC)C3)=O)C2)=O)ccc(Br)cc1O 50033,Fc1cccc(CN=C(NCC2CCN2C2CCOCC2)NCC(F)F)c1F 50034,c1(C(N2CCC3CCN(C(CC(C)(C)O)=O)CC32)=O)c[nH]c2ccccc2c1=O 50035,Cc1ccc(CC(=O)NC2CCCCN(C(c3cc(=N)[nH]c(Cl)n3)=O)C2)cc1C 50036,c1(CC)nc(=NCC(C2CCCCC2)C(=O)NC2(C3CCC3)CC2)s[nH]1 50037,C1(C(N2CC(C)(NC(=O)CC3CCCCC3)C2)=O)CC2(CCCC2)CO1 50038,c1(OCC=C)ccc(Cl)nc1C(=O)NC1CCC1NC(=O)C(C)c1ccco1 50039,c1(C(N2CCCC(CN(C(=O)CC3CCC3)C)C2)=O)cc(F)ncc1Br 50040,N1(C(N2C(C(=O)OC)C(OC)C(OC)C2)=O)CCSC(C)(C)C1C(=O)NCC1CC1 50041,C1(C(=O)NCC(C2CCCO2)O)CCOC12CCC2 50042,C(C1CN(C(=O)CCC2CCOC2)CC1C(=O)NCC1CC(=C2CCC2)C1)=CC 50043,N1(C(C2N(C(C(C)C)=O)CCCC2)=O)CCC(NC(c2cnc(S)[nH]2)=O)C(F)C1 50044,C(CCN(C)C(c1ccc(CC)s1)=O)(C(C)C)NC(c1cc(CCC)[nH]n1)=O 50045,N1(C(C23CC(C#N)(C2)C3)=O)CCC2(CCN(C(=O)C=Cc3cncs3)CC2)C1 50046,CCCS(=O)(=O)C(C)C(=O)NC1CN(C(c2cc(C)ncc2C)=O)C2(CCC2)C1 50047,c1(CC)ccc(C(C)CC(=O)NCC(O)CN(C(=O)Cc2cc[nH]n2)C)cc1 50048,C1(C(=O)NCC2(C)N(C(c3ncc(NC)nc3)=O)CCC2)C2CCCCCC12 50049,C12(NC(C(C3CCCOC3)OC)=O)CC(C(=O)Nc3ccn(C)c3C)(C1)OC2C 50050,Cc1ccc(C(=O)NCC(C)(C2CC2)NC(=O)COCP(C)(C)=O)c(C)c1 50051,c1(-c2ccc(CN(C(c3c(CCC)nccc3)=O)C)cc2)cc(OC)cc(O)c1 50052,c1(NCC(C)(C)N(C)C)cc(Br)ccc1S(=O)(=O)NCC1CCOC(C(C)C)C1 50053,C1(C(CC)CC)CCN(C(=O)CC2C=CC(NC(=O)C(C)CC3CCCC3)C2)C1 50054,C(CCCC(=O)N1CC2CC2(CNC(=O)CNC(c2ccc(Cl)cc2)=O)C1)OC 50055,c1(C(N(C2C(N(C)C(C3CC3F)=O)CCCC2)C)=O)cnc2ccnn2c1 50056,N1(C(CSCCCC)=O)CCC12CN(C(=O)CCC(C)(C)F)C2 50057,C1(C(N(C(C(=O)NCCCOCC=C)C)CC)=O)C(C(C)=O)C1(C)C 50058,C(CCCCC(=O)NC1CCC1O)N(C(=O)Cc1cncnc1)C 50059,N1(C(CN(c2ccncc2)C)=O)CCCCCC1CNC(c1ccccc1F)=O 50060,CC1=C(C(=O)NC2COC3(C2)CN(C(c2scnc2C2CC2)=O)C3)CCS1(=O)=O 50061,c1(NC(CN(C(=O)C(F)OC(F)(F)F)C(CC)C)=O)cc(C)cc2c1NCCC2 50062,CC1CC(NC(c2c[nH]c(C(N)=O)c2)=O)CCN1C(=O)CC1(C)CC1 50063,C(=O)(CCCCCc1cn(CCCF)nn1)NC1C(C)(C)C1 50064,CC(C(=O)N=c1ccn(CCO)[nH]1)C1CCN(C(c2ccc3occc3c2)=O)C1 50065,Cc1nccc(C(=O)NC23CC2CN(C(=O)C#CC2CC2)C3)c1C 50066,CCCCCC(O)C(=O)N1CCCC(CCNC(C2(OC)CCSCC2)=O)C1 50067,C(C(CC(=O)N1CC(COC(C)C)C1)C1CCC1)N(C(CCOC)=O)C 50068,N1(CC)CCCC1N(C(=O)C(N1CCC(Oc2ccncc2)C1)=O)C 50069,C#Cc1ccc(CC(N2CCC(NC(=O)C(C)N3CCCC3)CC2C)=O)c(F)c1 50070,C#CC1CCC(C(N2CCC(NC(C3CCC(C4CC4)C3)=O)C2CC)=O)CC1 50071,CCCCC(C)CCC(=O)N1CCC(CNC(c2coc(Br)n2)=O)C12CC2 50072,c1(C(C)(C)C)cccc(COc2cnc(C3CN(C(=O)OC(C)(C)C)C3)o2)c1 50073,n1(CC)nnc(C(=O)NCCC2(C)CCN(C(C3CCS(=O)(=O)N3)=O)C2)c1C 50074,C1(C(=O)NCc2n(C)ccn2)CC2CCC1N2C(=O)C(O)C1CCC1 50075,n1(CC(=O)NCC2(NC(C(C)OCC3CCCO3)=O)CCOC2)ncccc1=O 50076,CON1CCC(C(=O)N(C2CCC(NC(c3cccs3)=O)CC2)C)CC1 50077,C(=O)(C1=CS(=O)CCC1)NC1(CNC(C2(C)CCN(C(C)=O)C2)=O)CCCCC1 50078,Cn1cnc2ncnc(Nc3cc(-c4ccc([N+](=O)[O-])nc4)ccn3)c12 50079,c1(C(=O)NC2CC(NC(C34C(C(=O)OC)(CCC3)C4)=O)C2)ccn2nnnc2c1 50080,c1(C(C(=O)N(C2(C(=O)OCC)CC2)C)NC(N)=O)ccccc1 50081,CC1CCC(NC(=O)CCC#N)CN1C(=O)C(CCO)N(C)C 50082,C1(C(COC(C(C2CCCO2)OC)=O)=O)CC=CCC1 50083,c1(-c2nc(CSC)nn2CC2CC(C)C2)ccc2c(c1)COCC2 50084,Cc1ccc(C(N2CC(F)(F)CC2C(=O)NCCC(C)C)=O)c(O)c1 50085,C1(C(C(c2n(C(CC)(C)C)nnn2)NCCc2ccncc2)C)CC2CCC1O2 50086,N1(CC)CCC1C(=O)NC(CN)C1CCC1.C1(C(=O)C2CC2)(C)CC1 50087,N1(C(c2nc(COC)sc2)=O)CC(NC(=O)C2=CCCO2)C(C)(C)C1 50088,CC1(C)CC(NC(c2ccc(Cl)cc2N)=O)CN1C(C1CS(=O)C1)=O 50089,Brc1cc(NC(c2csc3c2CCNC3)=O)c2c(c1)OCO2 50090,c1(OC)ccc(CC(N2CCNC(C(=O)Nc3c(C)ccnc3Br)C2)=O)cc1Cl 50091,N1(C(C2CC(=O)NC2)=O)CCCC(C2CCN(C(=O)CCn3ccnn3)C2)C1 50092,C1(C(=O)NC(C2CC3(CCC3)C2)C)CN(C(C2(C)CCOC2)=O)CCO1 50093,C1(CNC(C2(C)CC2)=O)CCN(C(=O)CCc2ccncn2)CC1 50094,c1(CC)cn2c(n1)CC(C(=O)NCC1C=CCN1C(=O)CNc1nccs1)CC2 50095,N#Cc1cc(C(N2CCOCC2CNC(c2cnc(C3CCCO3)s2)=O)=O)c[nH]1 50096,N1(C(C(C)N(C)C)=O)CCCCCC1C(=O)NCC1(N2CCOCC2)CCCC1 50097,CCCC(O)CC(=O)N(CCC(C)NC(c1occc1-c1ccc(F)cc1)=O)C 50098,N1(C(C2(CC#C)CCCCO2)=O)CCN(C(=O)Cc2cncnc2)CC(CO)C1 50099,N1(C(CCc2cncc(C)c2)=O)CCN(C(=O)Cc2ccc(C)nc2)CC(O)C1 50100,C1(CNC(C=Cc2ccc(C)o2)=O)CN(C(c2cnn(CCF)c2)=O)CCN1C 50101,N1(Cc2cccc(OC(F)F)n2)CC2CC3CCCN3C2C1 50102,C12(NC(C(N)=O)=O)CCCC1CN(C(=O)Cc1c(F)cncc1Cl)C2 50103,Cc1cn2ccnc(C(=O)NC(C3CCN(C(c4cccn4C)=O)CC3)C)c2n1 50104,c1(C(=O)NC(C(=O)OCC)C)ccc(CNC(C2CCCC2(OC)OC)=O)cc1 50105,C1(C(=O)NCCN(C(c2ccn(CCF)n2)=O)CC)CC(O)CN1C(C)=O 50106,C1(C)(C(=O)OC)CC(F)(F)CN1C(=O)CC1CNCC(C)(C)O1 50107,C1(C(C)(O)C(N2CCC(NC(C3CCCCC3)=O)CC2)=O)CCC(F)(F)CC1 50108,c1(NC(C2(F)CN(C(C3CC(O)C3)=O)C2)=O)c(Br)cccc1[N+](=O)[O-] 50109,c1(OCOC)ccc(C(=O)NC(C)(C)CNC(C2CCCC23CC3)=O)cc1 50110,Cc1nsc(C(=O)NC(C)CN(C(=O)C(C)Cc2ccccc2)C)c1N 50111,CC(C)(C#N)CCC(=O)NCC(C)(C)OCC(=O)NCCC1(CO)CCC1 50112,c1(CC)cnccc1C(=O)NCC1CCN(C(C2C=CCC2)=O)C1 50113,CC(C(=O)NC1CCCC1NC(=O)C=Cc1c(Cl)cccc1Cl)C(F)(F)C(F)F 50114,C(C(C)(C)SC)(c1nnnn1CCCC(=O)OC)NCC.C12CC(C1)OC2 50115,C1(NC(c2cccc(COC)c2)=O)CCN(C(=O)C(C)S(N)(=O)=O)CCC1(F)F 50116,c1(C(=O)NC(C(C)C)CNC(c2ncsc2C2CC2)=O)ccc(Br)cn1 50117,C(C(O)C(=O)NCC1(NC(C2CC(N3CCCC3)C2)=O)CCOC1)OC 50118,Cc1nn(CC(=O)N(CC(C)NC(c2n[nH]cc2C(F)(F)F)=O)C)cc1Cl 50119,C12(C(N(C3CCN(C(C(C(C)C)F)=O)C3)C)=O)C3CC(CC13)C2(F)F 50120,c1(CC(N2C(C)(C)CC(CNC(=O)CNS(C)(=O)=O)C2)=O)cnc2n1CCOC2 50121,CC1(C)OCC(CCN=C(NCC2CCCO2)NC2CC=CC2)CO1 50122,C(CS(=O)(=O)NC(=O)CC1CC1C1CCCC1)OC 50123,C(=O)(CCCS(N)(=O)=O)N1CC(N(C(=O)C(c2ccccc2)F)C)C(O)C1 50124,C1(C(=O)NC2CCCC(NC(c3c(C)cc(F)s3)=O)C2)CC2C(C1)C2(F)F 50125,N1(C(c2c(OC)cccn2)=O)CC2(NC(=O)Cc3ccc(F)cn3)CCC1CC2 50126,CCCC(C)(CCC)C(=O)NC(C)C(C)NC(=O)C=Cc1ccccc1 50127,N1(C(C(CC)OC)=O)CC2CCC1(CNC(=O)C(O)C(C)c1ccccc1)CC2 50128,c1(CCC(=O)N(CCN(C(COCCC#C)=O)CC)CC)ccccc1Cl 50129,C1(CN(C(=O)CN(C)C)C)CC(F)CN1C(=O)CNC(=O)CCn1ccnc1 50130,c1(OC)noc(C)c1C(=O)NC1COCCC1NC(C1CC12CCC2)=O 50131,CCC(C(=O)NC1CCCC1NC(C1(OC)CC1)=O)SC 50132,C1(C(N(CCCNC(C2(C)CCN(C)C2=O)=O)CC)=O)COCCN1C=O 50133,C(C(CC(=O)N1CC2=C(C1)CN(C(C1C3CCC1CC3)=O)C2)C(F)(F)F)N(C)C 50134,S(=O)(=O)(c1cccc(=NCC(O)c2ccccc2F)[nH]1)N1CC(CC)N(C)CC1 50135,C1(CNC(CSCCCC)=O)N(C(=O)C(C)C(=O)OC)CCCC1(C)C 50136,CC(CC(=O)NCC1CCC1NC(c1ccc2c(n1)CCO2)=O)CC(C)(C)C 50137,CC(C)CCC(C(=O)NCC(CO)C(C)C)NC(=O)CCN(C)CCO 50138,c1(C(=O)NC(CNC(c2c(C)ccnn2)=O)C)cn2cccc(F)c2n1 50139,CCCC(CC)CCC(=O)NC1CN(C(=O)CCc2ccc(N)c(F)c2)CC1F 50140,C(=O)(C(C)(C)Cc1ccccc1)N(CCN(c1nnc(C)s1)C)C 50141,c1(N(C(C2(CNC(=O)OC(C)(C)C)CCCC2)=O)CC)ccc(Br)cn1 50142,C(=O)(C(C)CC(F)F)N.c1(C(N2C(C(C)O)CCC2)=O)cc(OC(F)F)ccn1 50143,C(c1ccc(Br)cc1)=CCN(C(C(=O)NCCCOCCOCC)C1CC1)CC 50144,C#CCCC(C(=O)NCC(F)(F)C(N)=O)NC(c1cnc(O)cc1C)=O 50145,c1(OC)cccnc1C(=O)N(C1CCN(C(C2CCOC2C(C)C)=O)CC1)C 50146,c1(CN(C(=O)NCc2ccccc2)CC2N(C)CCOC2)c(Cl)cnc(F)c1F 50147,C1(C(N(CC(C)(C)O)C2CC2)=O)CC2(CC2)CN1C(=O)CSCCCF 50148,N1(C(CN(C(=O)CC(O)CN(C)C)CCC)=O)CCC(C)(C)C1C 50149,N1(C(C2C(C3C(C)C3)C2)=O)CC2(C1)CN(C(C1CCC(=O)N(C)C1)=O)CC2CO 50150,Cc1cnncc1C(=O)NCC(C1CCC1)NC(=O)C(C)Cc1cccc(Cl)c1 50151,C1(OC)CN(C(C)=O)CC1NC(=O)C(C(C)C)n1cnnc1 50152,C(=O)(C(C)C(C)NC(=O)CCN1CCCC1=O)N(C)CC1C(C)OCC1 50153,n1(CCC)nnnc1C(CCC)(C1CC1)NCc1cnc(CC)s1 50154,c1(C(=O)NCCN2CCN(C(CC(C(=C)C)OCC)=O)CC2)ccc2n[nH]cc2n1 50155,CCC(C)C(O)C(C)C(=O)NC1CC12CCN(C(C1OCCC1CC)=O)CC2 50156,C1(CCNC(C2CN(C(N)=O)C2)=O)CN(C(c2nnsc2C(F)F)=O)CCO1 50157,N1(C(=O)C(c2cccc(Cl)c2)O)CCCC(NC(C2CC(C(F)F)C2)=O)CC1 50158,c1(C(N(C(C)CNC(=O)CSc2nc[nH]n2)CC)=O)cnsc1 50159,CC1CC(NC(=O)C(C)(C)CC2CC2)CN(C(=O)Cc2cncn2C2CC2)C1 50160,C1(NC(C(c2cnn(C)c2)OC)=O)CC12CC(NC(=O)CCCC1CCCC1)C2 50161,CC1=C(C(=O)NC2C=CC(C(=O)NC34CCC(CO)(CC3)C4)C2)CCCO1 50162,C=CCC(C)(C)C(=O)NCC1(C)CCN(C(C2CCC(C(=O)N(C)C)CC2)=O)C1 50163,Cc1ccc2c(c1)C(C(=O)N1CCCC(CCNC(=O)CC(C)C)CC1)OCC2 50164,C1(NC(CCOCC)=O)COC2(CCN(C(c3ncsc3NCC)=O)C2)C1 50165,C1(N(C(C(CCCC)N(C)C)=O)C)CC2CCC(C1)N2C(c1ocnc1C)=O 50166,c1(C(=O)NCC2CCC2NC(C2CCC2(F)F)=O)cncc(N2CCCC2=O)c1 50167,Cc1c(C(=O)NC(CNC(C2CCS(=O)CC2)=O)C2CCC2)c[nH]c2nccc1-2 50168,N1(C(C2CN(C)C(=O)N2)=O)CCN(C(=O)CCCC2CCOCC2)CC(O)C1 50169,N1(CC(N2C(C(C)NC(c3c(Cl)nsc3Cl)=O)CCC2)=O)CCN(C)C(=O)C1 50170,[N-]=[N+]=NCC(C(=O)NCCN1CCC(CO)C1)NC(c1nnsc1N)=O 50171,C1(NC(C2(CC#C)CC2)=O)CCC2CCN(C(=O)C(c3ccc(C)cc3)C)C12 50172,C1(NC(Cc2n(CC)cnc2)=O)CCCC(N)CC1 50173,N1(C(c2c(C)occ2)=O)CC(NC(=O)C(c2cccc(F)c2)O)C(C)C1 50174,c1(OC)cc(C)cc(C(=O)NC2CCCCCC2NC(=O)CNC(N)=O)c1O 50175,C(CCC(C)(F)F)N(C)C(C1OCCC1NC(=O)CC1CCCOCC1)=O 50176,N1(C(C(CC)C2CCC2)=O)CC(CN(C)S(N)(=O)=O)C2CCCC12.CC(C)(C)O 50177,N1(C(CC(C)(C)O)=O)CCC2(CCN(c3nccc(-c4cnccn4)n3)C2)C1 50178,c1(OC)ccc2[nH]c(CN3CCC(O)CC3C(=O)Nc3csc(C)n3)cc2n1 50179,c1(C(N2C(C)C(NC(=O)CCCC(F)F)CCC2)=O)cnc([N+](=O)[O-])n1C 50180,CC1CN(C(=O)CO)CC(C)N(C(c2cc(Cl)cc(Br)c2F)=O)C1 50181,C=CCC(CC)C(=O)NC1C2CC1N(C(c1ccc(CC)c(Cl)c1)=O)C2C 50182,C1(C(N2CC(OC)C(NC(=O)CC34COCC(C3)C4)C2)=O)CC2(CCCO2)C1 50183,Cc1cc2ccccc2n1CC(=O)NC1(C)CCN(C(C2(C)CCN(C)C2)=O)C1 50184,Nc1cc(C(=O)NCC2CCCN2C(c2cnccc2C(F)F)=O)cc(F)c1O 50185,S(=O)(=O)(c1cccc(=NCc2cnc(NC)nc2)[nH]1)NC(C(CC)(C)C)C.C=O 50186,N1(C(CSC)=O)CCc2nc(CNC(C3(C)CC3(F)Cl)=O)sc2C1 50187,CC1CCN(C(c2ccc(CNC(=O)C=CC3CC3)nc2)=O)CCS1 50188,c1(OCC)c(C(N2CC(CNC(c3c(C)cccc3Br)=O)C2)=O)cccc1F 50189,S(=O)(=O)(c1ccccc1Cl)NCC(=O)N(C1CC(NC(c2occ(C)c2)=O)C1)C 50190,c1(NC(CCC)CC)[nH]c(=NC2CSCCC2C)nc2c1ncn2CC 50191,N1(C(C(CC)=CC)=O)CCC2(NC(c3nncn3CC)=O)CCCCC12 50192,C1(C(=O)NC(C(=O)NCC(C(C)O)O)(C)C2CCC2)C(C#N)C1(C)C 50193,c1(SC)cnn(C)c1Cl.C12CCN(C1=O)c1sccc1NC2=O.c12ccccc1N2 50194,C1(C(N(CCCN(C(C(CC)NC(C)=O)=O)C)C)=O)CC(F)CN1C 50195,C1(C(=O)NC(C2CCCC2O)C)CCCC1CNC(c1cc[nH]n1)=O 50196,c1(C(N2C(CC(=O)NCc3ccc(F)cc3F)CCC2)=O)ncnc2[nH]cnc12 50197,c1(CC)ccsc1C(=O)N(C)CC1CCN(C(C2CC3CC3C2)=O)C1 50198,Cc1nc2ccnn2cc1C(N1CC(O)(CNC(C2CC2(C)Br)=O)C1)=O 50199,N1(C(C(C)C2CCC2)=O)CCC(CO)(CNC(c2ccnc(Cl)c2N)=O)CC1 50200,C1(SC)CC12CC2(F)F.c12cnn(c1)C(=O)N(CC)CCNC(=O)c1ccoc1-2 50201,CCCC(C)C(=O)N1CCC(CC(=O)NOCC(O)CO)CC1 50202,N1(C(c2ccc(CO)o2)=O)CCC2(CC(C(N3CC(CO)C4(CCC4)C3)=O)C2)C1 50203,C1(C#N)(CNC(CC2(C)N(C(Cc3nc(C)[nH]n3)=O)CC2)=O)CCCC1 50204,CC1CCCCN1C(C1CC(NC(C2C=CCS2)=O)C1)=O 50205,CC1CC(=O)NCC1C(=O)NCC1CC(NC(c2cccc(Cl)n2)=O)C1 50206,c1(C(N(CC(C)(C)NC(=O)C2=NOCC2)C)=O)cc(F)cc2nc(S)[nH]c12 50207,C(C(CC)CCO)NC(CCN(CC#C)C(c1cnc(Cl)s1)=O)=O 50208,N1(C(C(C)(C)N=[N+]=[N-])=O)CC2(C1)CN(C(C1CCC(=O)N1)=O)CC2CO 50209,Cc1cc(C(c2nnnn2C2CC2)NCC(C)(C)C(N)=O)cc(C)n1 50210,C12(C(=O)NC(C(C)NC(=O)CCNC(=O)CO)(C)C)CC(C)(CCO1)C2 50211,C1(NC(c2ccc(C#N)o2)=O)CC(C(=O)NCC2CCCC2O)C12CCC2 50212,CCCCC(C(=O)NCC(C)N(C)C(c1nc(C(F)(F)F)cs1)=O)C(C)C 50213,N1(C(c2cc(Cl)c3n[nH]cc3c2)=O)CCC2(CCN(C(c3ccco3)=O)CC2)C1 50214,C(=O)(CC1=NNC(=O)C1)N1CCC(C)(CNC(C=Cc2n(C)ccc2)=O)C1 50215,CC#CCC(C(=O)NC1CCC12CCCC2)NC(c1ccc(OC)nn1)=O 50216,C(=O)(C(C)C(=O)NCCOCCCNC(C1CNC(=O)C1)=O)OC 50217,C1(NC(C23CCC(OC)C2C3)=O)CN(C(=O)CC2CC3(CCO2)CC3)CCC1O 50218,S(=O)(=O)(c1ccc(CNCc2cnn(Cc3ccccc3)c2)cc1)NCC(N)=O 50219,N1(C(C23CC(COC)(OC2)C3)=O)CCCC(NC(C2ON=C(C)C2C)=O)CC1 50220,C1(CC=C)(NC(=O)C2=CCC2)CCN(C(c2ccc(CCC)cc2)=O)CC1 50221,c12nc(cs1)CNC2=O.C1(CNC(CCNC(=O)OC)=O)(CO)CC1(F)F 50222,CC1(C)C(C(=O)NCC23CCCN(CC2)C3)CCN1C(c1ccsn1)=O 50223,N1(C(C(COCC)C)=O)CC2CCC(C1)N2C(c1cccc(F)c1O)=O 50224,Cc1nc(C(C)C)sc1C(N1CC(NC(=O)C2=CCC2)CC1CO)=O 50225,c1(C(N(CC(C)N(C(CN(CCC)C)=O)C)C)=O)sc(Cl)c(Cl)c1C 50226,c1(C(C)NC(CC2(N(C(c3cn(CC)nn3)=O)C)CC2)=O)ccc(F)cc1 50227,C1(C(C)NC(=O)CCSCC(N)=O)CCCN1C(=O)CC1(C)CCCO1 50228,N1(C(C2(C(C)(F)F)CCC2)=O)CC(NC(=O)CC2OCCC2(C)C)CC(F)C1 50229,C1(C(=O)N(C)Cc2cncnc2)(CC)CCN(C(=O)C(C)NC(=O)NC)C1 50230,CC1=C(C(=O)N2CCOCC2CNC(=O)CC2C=CCC2)CCC1 50231,C1(NC(=O)C(C)(C)C)CN(C(=O)CC(N(CC(C(C)C)C)C)=O)CC1C(C)C 50232,C(=O)(C(C)CCCOC)NCC1CN(C(C(c2cccc(Cl)c2)CC)=O)C1 50233,Cc1c(Cl)c(Cn2cc(CCC3CCCCC3)nn2)nc2ccccc12 50234,CCCC(C)CCCC(=O)N1CCCC1C1(O)CN(C(c2ccc(C)nc2)=O)C1 50235,c1(OC)c(C(N2CCC(N(C)C(c3csc(SC)n3)=O)C2)=O)cccc1F 50236,c1(OC)cccc(CNC2CC2C(=O)Nc2cc(C(C)(C)C)on2)c1C 50237,c1(C(=O)NCC2CC(C)N(C(c3cscc3C(F)(F)F)=O)C2)ccnc(C#N)c1 50238,C1(C(C)NC(=O)C(F)n2cccn2)CCCCN1C(c1ccc(CO)cc1)=O 50239,N1(C(C2CCC(C)(C)O2)=O)CCC2CN(C(=O)CCCC#N)CC2CC1 50240,N1(C(C2=CN=C2C(F)F)=O)CCN(C(c2cc(C3CC3)sn2)=O)C(C2CC2)C1 50241,C(=O)(C1(N(C)CP(C)(C)=O)CCc2c(OC)cccc21)OC 50242,C(CCC(C)C(C(=O)NC1CCC1)N(C)CCc1ccc(Cl)cc1)=C(C)C.C1(C)CC1 50243,CC(CNC(c1ccsc1Cl)=O)CC(F)F 50244,c1(NC(C(C)CSC(F)(F)F)=O)cccc(-c2cn(CCCN(C)C)nn2)c1 50245,c1(C(=O)OCC)ccc(CC(N2CCC2C(=O)Nc2cc[nH]c(=N)c2)=O)cc1 50246,N(C(=NCCN1CC2CCC1C2)NC1CCS(=O)(=O)C1)Cc1scc(C#N)n1 50247,O=C(C1=CCC(NC(c2n[nH]c(O)n2)=O)C1)NC(CC1CC1)C1CC1 50248,CCCC(F)(F)C(=O)NCC(CC(=O)Nc1ccc(C)c(C)c1)C1CCC1 50249,C(=O)(C(C)(C)C(=O)NC1CC(NC(=O)C(C(C)C)n2cc(Br)cn2)C1)OC 50250,N1(CCC(C)C2CCCO2)CC(=O)N(Cc2c(I)cnn2C)C1=O 50251,C12(NC(CCCOC(C)=O)=O)CCC(CC1)N(C(C)=O)C2 50252,c1(C(N(C2CCCN(C(=O)CCc3cocn3)C2)CC)=O)cc(F)cnc1O 50253,C1(CNC(CCC(C)OC)=O)(NC(C2CCC(F)(F)C2)=O)Cc2ccccc2C1 50254,c1(SCC(=O)NCCN(C2CCCC2)C(C=CC(CC)=CC)=O)n[nH]c(C)n1 50255,C12(NC(c3cc(CCC)[nH]n3)=O)CCC(CC1NC(=O)C(C)n1cncn1)C2 50256,c1(CSCC(=O)NCC(CN(C(C(F)OC)=O)C)C)nnnn1C1CCC1 50257,Cn1cc(C(N2CC(NC(C34CCOC3CCOC4)=O)C2)=O)c2cccnc12 50258,C1(NC(C2(C(O)C(F)(F)F)CC2)=O)CCC2CCN(C(c3coc4c3COC4)=O)C12 50259,CC(CN1CCC1)CN=c1[nH]c(=NCC2(Cl)CC23CCC3)[nH]c2c1CCCCC2 50260,c1(C(N2CCC(NC(C(C(CC)C)OC)=O)C(OC)C2)=O)c(F)ccc(F)c1N 50261,C(CCCCC(=O)NCC1CCN1C(=O)CCn1cnc([N+](=O)[O-])c1)NC(N)=O 50262,CC1CN(C(c2cnc(O)cc2O)=O)CC(CCNC(c2ccn(C)c2)=O)O1 50263,c1(C(N2CCC(COC)(NC(=O)C(O)C3CC3)CC2)=O)cc2cccnn2c1 50264,CC(C(=O)N1CCC(CO)(CNC(=O)C(C)NC(N)=O)C1)S(N)(=O)=O 50265,CC#CCCCC(=O)NNC(=O)c1cc2ccccc2[nH]1 50266,N1(C(C(=Cc2cn[nH]c2)C)=O)CCN(C(c2csc(C(F)(F)F)n2)=O)CCC1C 50267,N1(C(C(=CC2CCCC2)C)=O)CC2OCCN(C(=O)CCS(C)=O)C2C1 50268,CCCCC(C(=O)NC1CCCCCC1C)NC(=O)C=CCN1CCCC1 50269,C(=O)(CCC(C)S(C)(=O)=O)NCC1CC(NC(CC(C)C(F)(F)F)=O)C1 50270,Cc1cc(CC(=O)NC2CC(C)(CNC(c3c(C)cccc3F)=O)C2)cc(F)c1 50271,Cc1ncc(C(N2CCCC2(C(=O)Nc2ccc(O)nc2)C(C)C)=O)c(=N)[nH]1 50272,c1(CC(=O)NCC(C)NC(c2ccnn2CCC#N)=O)ccccc1CC1CC1 50273,C(=O)(CCCCNC(C)=O)N1CC(C(=O)NCC2(OC)CN(C)C2)(SC)C1 50274,Cc1ccc2[nH]c(C(N3CC4CCC4(NC(C4(F)CCOC4)=O)C3)=O)cc2c1C 50275,N1(C(=O)CN2CCCC2CO)CC2(NC(C3CC(n4cnnc4)C3)=O)CCC1C2 50276,C(CC(O)CNC(c1cnn(C2CC2)c1)=O)NC(C(N1CCCC1=O)C)=O 50277,C1(CN(C(Cc2cc(C)no2)=O)C)CCCN(C(c2occc2Cl)=O)C1 50278,C=Cn1nncc1C(=O)Nc1cccc(NC(=O)CC(O)c2ccccc2)c1 50279,C(C(N=[N+]=[N-])C(=O)N1CC(CNC(=O)CSSC)C1)OCC 50280,N1(C(c2nc(N(C(C)=O)C)sc2)C2CC2)CCC(=O)N(Cc2cccnc2Cl)C1=O 50281,N1(C(C2CCC(SCC)C2)=O)CCN(CCN(C)C(C2CCN2SCC)=O)CC1 50282,C1(CC)(NC(=O)CC2CCC(=O)O2)CCN(C(=O)CCCn2ccnn2)CC1 50283,C1(S(C)(=O)=O)(C(=O)NCC2C(CNC(CSC)=O)C2)CCCCC1 50284,c1(N(C)CC)ccc(C(=O)NC2(CO)CCN(C(C34COCC3C4)=O)C2)cc1 50285,C(CC1=CCN(C(C2CC23CC3)=O)CC1)NC(c1n[nH]c2c1CCCC2)=O 50286,Cc1cccc2c(C(N3CCCN(C(=O)COC(C)C)C(C)C3)=O)csc12 50287,N1(c2ccc(CC)cc2)Cc2ccc(NC(=O)NC(CNC)C(C)(C)C)cc2C1=O 50288,N1(C(c2ccc(C(=O)OC)cn2)C(=O)NCCCC)CCC2(CCCCN2C)C1 50289,Cn1nc(C(N2CC3CC3(CNC(c3ccncc3N(C)C)=O)C2)=O)cc1O 50290,C(=O)(C1c2c[nH]nc2CCC1C)N1CC2N(Cc3cc(C)on3)C(CC2)C1 50291,C(=O)(CCC(C)(C)N(C)C)N(CC(C)N(C(=O)COC1(C)CCCC1)C(C)=O)C 50292,c1(C(N2CC3C(NC(C(CCC)OC)=O)(C3)C2)=O)ccc(Br)cc1F 50293,C1(N(C(CCC(=C)Cl)=O)C)CN(C(=O)C(CC(=C)C)NC(C)=O)CC1(C)C 50294,S(=O)(=O)(c1cc(C(=O)NC(C)CCN(C(=O)C=C2CCCCC2)C)c(C)o1)NC 50295,C(=O)(CS(=O)(=O)N1CCN(CCCNC(C2(C)CC2F)=O)CC1)OCC 50296,N1(C(c2ccnc(C)n2)=O)CCC(C)CC1CNC(=O)COCCCC(C)C 50297,C1(C)(c2cn(CC(=O)OC)nn2)CCN(C(=O)CCC2COC(C)(C)O2)CC1 50298,CN1CC(C(N2CC(O)(C(F)C(=O)NCC3CC(O)C(O)C3)C2)=O)CCC1=O 50299,c1(C(=O)NCC(CC)NC(C(CCC)O)=O)cccc(S(=O)(=O)NCC(N)=O)c1 50300,c1(CC(n2cc(-c3c(C)noc3C)nn2)C)c(C)nn(C)c1C 50301,C(=O)(CC(O)CC(C)(C)C)N(C(CC(C)C)C(=O)NCC1(F)CCN(C)C1)C 50302,c1(C(=O)NCC(N2C(C)CC(NC(C3CC(C)(O)C3)=O)C2)=O)ccc(F)c(F)c1 50303,c1(CC(N2CC(NC(C3C(CC)C3)=O)C(C)C2)=O)cc(SC2CC2)cc(F)c1 50304,N1(C(C(C)O)=O)CCN(C(c2cc(C3CCCN3C)[nH]n2)=O)CC1 50305,c1(OC)cccc(C(=O)N(C)CC2CN(C(c3cnco3)=O)CCO2)c1OC 50306,CS(=O)(=O)c1ccccc1CN1CC2C(C1C(N1CCCC1CO)=O)C2(C)C 50307,C(=O)(C1CCc2cc(Cl)ccc21)N1CC(NC(c2nc(C)n(C)c2)=O)C(F)C1 50308,c1(C(=O)NCC(CC=C)NC(=O)C(C)OCCCC)cc2nc(OC)ccc2[nH]1 50309,C1(C(N(CCCNC(C2CCC2C(C)(C)C)=O)C)=O)CCS(=O)(=O)CC1 50310,C1(n2c(CN)nnn2)CCCCCC1.Clc1csc(C(C2CC2)C2CC2)n1 50311,c1(C(N2CCC(N(C)C(c3cnco3)=O)C2)=O)ccc2c(n1)CCCC2 50312,c1(CNC(=O)Cn2cnc(C(F)(F)F)c2)cc[nH]c1C(=O)NC1C(OC)C1 50313,c1(CNC(Cn2c(C)ccn2)=O)cccc(NC(C2CCCCC2C)=O)c1 50314,c1(C(=O)NC2(C)CCN(C(C(C)SCC)=O)C2)cc2c(Br)c(C)ccc2[nH]1 50315,C1(N(C)C)CN(C(C2CSCCS2)=O)CC1CNC(c1csc(CO)n1)=O 50316,N1(C(C(C)C)=O)CCC(C)CC1CNC(c1ccc(SCCCO)cc1)=O 50317,C1(C(=O)NC(CCC(=O)OC)C)CN(C(=O)CCCCSC)CCC1(C)C 50318,C1(C(N2CC3CC3(C(N3CCC(n4ccnn4)C3)=O)C2)=O)CC2CC1CC2O 50319,c1(CC)ccc(Br)cc1C(=O)NC1CC(N(C(=O)CC2CCOCC2)C)C1 50320,c1(C(N2CC3CC2CN3C(C2CC3(CCCO3)C2)=O)=O)ccc(Cl)cc1Cl 50321,C1(NC(C(C)C)=O)CCCN(C(=O)CNC(c2ccc3nn[nH]c3c2)=O)CC1F 50322,CCCCC(C)(F)C(=O)NCC1CC(NC(=O)CC2(N(C)C)CCCC2)CCO1 50323,Cc1onc(Cl)c1C(N1CC2C(CNC(c3snc(Cl)c3Cl)=O)C2C1)=O 50324,N1(C(C)C)CC(NC(=O)CN2CCN(C(=O)Cn3ncccc3=O)CC2)CC1=O 50325,C1(NC(C=C(C)C(C)C)=O)C2CC1N(C(=O)Cn1cc(C)cn1)C2 50326,C1(CNC(CCCN(C)C(C2(C3CC3)CC(=O)C2)=O)=O)CC2CCCC2C1 50327,c1(C(N2CCCC(CCNC(C(COCC)(C)C)=O)C2)=O)cnc2scc(C)n12 50328,N(S(=O)(=O)N1CCC2(CCCCC2)CC1)CC(CCCC)OC 50329,C1(C2CCN(C(=O)CCC3=CCCCC3)CC2)(NC(CC(=O)NCC#C)=O)CC1 50330,N1(C(C(C)N(C)C)=O)CCC(N(C)C(c2ncc(C(F)F)s2)=O)CC1 50331,N1(C(C(COC)(C)O)=O)CC2(CC(NC(c3cn4cc(C)ccc4n3)=O)CO2)C1 50332,C1(C(=O)NCC2N(C(c3n[nH]c(CC)c3Cl)=O)CC(O)C2)CCOC(C)(C)C1 50333,c1(COC)nc(C)c(C(=O)NCCCC2CCCN2C(=O)CN2CCC2)s1 50334,N1(C(c2c(C)c[nH]n2)=O)CC2CCC(Nc3ncc4c(n3)COC4)CC2C1 50335,C1(CC(=O)Nc2ccccc2)(N(C(=O)CSC(F)(F)F)CCF)CCOC1 50336,C1(CNC(CCC2C(C)(C)C2)=O)(NC(c2ccc(=N)[nH]n2)=O)CCCCC1 50337,C1(C(=O)NCC(C(C)(C)C)NC(c2c(CC)c[nH]c2)=O)CCCCC(=O)N1 50338,c1(OC)cc(-c2ccccc2)c(-c2ccc(C)c(F)c2)cc1C(N)=O 50339,CCCCC(C)(C)NC(C1(NC(=O)C(CC)NC(C)=O)CCSC1)=O 50340,N1(c2c(Cl)cnc(OC)n2)CCC(C2(NC(=O)CCN(S(C)(=O)=O)C)CC2)CC1 50341,c1(OC)ccc2c(c1)C(C(=O)Nc1ccc(C(=O)NCCC(C)(C)O)cc1)CC2 50342,n1(CC)cc(C(=O)NC2CN(C(=O)CN3CCN(C)CC3)C2)c(C(C)C)n1 50343,C1(OC)CCCC(C(=O)NCCCN(C2CCCC2)C(c2cn(C)c(C)n2)=O)C1 50344,C(N=c1[nH]cnc(Cl)c1C(C)C)C1C(NC(Cn2c(C)ncc2)=O)CCCC1 50345,CCC(CC)CCC(=O)NCC1(C)CCN(C(=O)C(C)CNC(=O)OC(C)(C)C)C1 50346,C(=O)(C(F)C(=O)NC(C)(C)CC=CC(=O)N(CCC#N)C)OCC 50347,C(=O)(C(C)(CCC)CCC)NCCC(=C)CNC(=O)COC(C)=O 50348,N1(C(c2n(CC)nc(C)c2)=O)CCC2(CC2NC(=O)C(C)N2CCCC2)C1 50349,c1(C(N(C(CNC(C=COCC)=O)C)CC)=O)ccnc2ncnn12 50350,c1(OC)ncc(C(=O)N(C2CC3CC2N(C(=O)CSCC(C)C)C3)C)cc1Cl 50351,Cn1nc(Br)c2c(NCCNC(c3ccc(Cl)cc3F)=O)ncnc12 50352,N1(C(CCCC#C)=O)CC2CCCC1C2CNC(=O)CC=C 50353,c1(CC)ncc(CNC(=O)C(C(C)C)NC(=O)OC(C)C)c(=N)[nH]1 50354,c1(SC)ccncc1OCCNC(c1nncn1C)=O 50355,N1(C(c2cc(C#C)c(Cl)cc2)=O)CCC2(C1)CN(C(=O)CCN(C)CC)CCO2 50356,N1(C(C(C)=CC2CC2)=O)CC(C(N2CCC(CCO)C2)=O)(SC)C1 50357,Cc1cnc(NCc2cscc2C)c(S(=O)(=O)NC2CC3CC(CO)CC23)c1 50358,c1(C(N(CCN(C(=O)CC(C)(C)CC)CC)CC)=O)cc([N+](=O)[O-])c(C)cc1C 50359,c1(C(=O)NC2CC(CNC(C(C(C)c3ccccc3)O)=O)C2)ccnc(F)c1O 50360,C1(C)(NC(CCCOCC)=O)CCCN(C(=O)CC(CC#N)c2ccccc2)C1 50361,CC(C)C(O)C(C)(C)C(=O)NC1COCC1C(N1CC(C)(CF)C1)=O 50362,c1(C(=O)OC)cccc(C(=O)NCCCC2N(C(C3(Cl)CC3)=O)CCOC2)c1 50363,C1(NC(CCC)=O)CC(CNC(=O)CCCOC(C)C)C1(C)C 50364,N1(C(C23CCC(CC2)C3)=O)C2CCC1CC(NC(CSCC(=O)NC(C)C)=O)C2 50365,N1(C(CCOC)=O)CCC(C(C)C)CC1CNC(c1cnn(CCO)c1)=O 50366,C1(C(=O)NC(C(C)C)CCN(C)C(C2CC2(F)F)=O)CC1C1CCCCC1 50367,C(=O)(CCCCCCN=[N+]=[N-])N1C(C)(C)CC(C)(CNC(C2CC2(C)C)=O)C1 50368,Cc1ccc(C(C)C(N2CCCC(NC(c3ccc(Cl)nc3)=O)C2)=O)cc1 50369,CC(CN(C)C)CC(=O)NCC1C2CC1N(C(C1COCCN1C)=O)C2 50370,N1(C(C(CC)(C)COC)=O)CCCCC(CNC(=O)Cc2ccc(C)cc2)CC1 50371,c1(NC2C(C(=O)OC)C2)cc(OC)c(OC)cc1OC.c12c[nH]c(c1)C(=O)NC2 50372,C1(CC#C)(C(=O)NCC(O)C(F)F)CCN(C(=O)CCCC#N)C1 50373,c1(C(C(=O)NCCCOC)N(CCC(N)=O)CC2CC2)nc(C#N)cs1 50374,Cc1cc(C(=O)NC2(CC(=O)Nc3nnc(C)o3)CCC2)nc(C)c1 50375,Cc1cnc2c(N(C)CC3(OCCO)CCCSC3)nccc2n1 50376,C(C)(C)(CC(F)C(=O)NC1(c2ncc(C)o2)CC1)NC(c1c(CC)nn(C)c1)=O 50377,c1(C(N2C(CNC(c3nccc(C)c3)=O)C(C)CC2)=O)cc2c(ncn2C)[nH]1 50378,c1(C(=O)NC2C3CN(C(c4ccn(C(C)(C)C)n4)=O)C2C3)n[nH]c2c1COCC2 50379,C1(NC(c2sc(C)c(O)n2)=O)CC2CC(C1)N(C(C1(C)CCCCC1)=O)C2 50380,c1(C(C)C)nc(C(=O)NCC2C(NC(=O)Cc3cnns3)CC2O)co1 50381,c1(CNc2cccc(NC(COC(C)(C)C)=O)n2)ccc2c(c1)CCO2 50382,C(=O)(C(C)(F)F)NCC(C)CN(C)C(c1ccc(CSC(F)F)o1)=O 50383,CC1CN(C(C2CC2c2cn[nH]c2)=O)CCCN1C(c1csc(C(F)(F)F)c1)=O 50384,CC(CCCNC(c1nc(Cl)cs1)=O)NC(=O)C(C)(C)c1cscn1 50385,C1(COC)(NC(=O)C(C)n2cnnn2)CN(C(=O)CCC2CCCCC2)C1 50386,C(C)(CNC(=O)C(c1ccnn1C)C)(C(C)C)NC(CN(C)CC)=O 50387,c1(OC)ccc(N)c(C(N2CCOCC2CNC(=O)Cc2cc(Cl)cs2)=O)c1 50388,C1(C(N2CCN(CC(=O)NC(c3cscn3)CO)CC2)=O)CC12CCCCC2 50389,CC1N(C(C2N(C(c3ccc[n+]([O-])c3)=O)CCC2(C)C)=O)CCOC1(C)C 50390,c1(C(N2CCC(N(C(C(CC(C)C)C)=O)CCO)C2)=O)nn2cccnc2c1Cl 50391,Cc1cnc(CC(=O)N(C)CC2CCCN2C(=O)C(C)CC2CCC2)o1 50392,c1(C(=O)NCC(CO)NC(=O)CCn2cccn2)ccc(F)c2ncccc12 50393,C1(CC)CNC(=O)CN1C(=O)CC1CN(C(=O)Cc2cccc(C)c2)CC1C 50394,CC1(C)CN(C(C2CCC(=O)NC2)=O)CC1CNC(=O)Cc1ccc(O)cc1 50395,Cc1ccc(Cl)cc1C(N1CC(CO)(NC(=O)C(C)C2(O)CCC2)C1)=O 50396,C(=O)(C1=C(C)OCCS1)NCc1nc(CNC(CC(CCC)C)=O)sc1 50397,CN1CCC(NCCNC(C2CCN(C(=O)C(F)=CCF)CC2)=O)C1=O 50398,C1(C)(CNC(CN2CCC(C)CC2)=O)COCCN(C(c2cnsn2)=O)C1 50399,C(=O)(CCC(=O)NCC(CC)NC(C1CCCN1c1ncccn1)=O)NCC 50400,C(=O)(C1=COc2ccccc2O1)NCCOC(N(C)CC12CCCCC1C2)=O 50401,CC1CN(C2CCOCC2)CCN1c1nnc(C(c2ccc(F)cc2)(C)C)n1C 50402,N1(C(C2(OC)CCN(C(C=CC)=O)C2)=O)CC(OC)C2(CC2)C1 50403,C#CC1(C(=O)NC2CC3CCCCN3C2)CCN(C(=O)CC2OCCCO2)CC1 50404,c1(CCC(=O)NC(CC2CN(C(C(CC)(C)F)=O)C2)C)c(C)nn(C)c1C 50405,C1(CC(=O)NC2CC(NC(Cc3cn(CC)nc3)=O)C2)CCC(=O)NC1=O 50406,Cc1cc(I)c(C(N2C3CCC2CC(NC(=O)C(C)(C)CN(C)C)C3)=O)cc1C 50407,C(=O)(C(C)(C)C(=O)N1CCOCC(C(N2CCN(C)C(CO)C2)=O)C1)N(C)C 50408,N1(C(COC(C)C)=O)CCN(C(=O)Cc2cncnc2)C(CS(C)(=O)=O)C1 50409,CCCC(CNC(=O)Cc1scnc1C)C(=O)NCCOCC1CCCC1 50410,C(CCCC(=O)NC1CCC(NC(C2(C)CSC2)=O)C1)SC 50411,C(=O)(CC(C(F)(F)F)OCC)N1CCC(CC=C)(NC(=O)COCCCOC)C1 50412,N1(C(CC(C)CNC(=O)CCc2ccc[nH]2)=O)CC2(CNC(=O)N2)C1 50413,C1(N(C(C(C)C(=O)OC(C)(C)C)=O)C)CN(C(=O)CCCCC2CC2)CC1(C)C 50414,CC1Cc2cc(OC(c3ccc(C(C)C(F)(F)F)cc3)=O)ccc2O1 50415,CN1C(=O)CSC1=CC(=O)NCC1CC2CCC1N2C(=O)CN1CCCCC1=O 50416,Cc1ncc(C=CC(N2CCC3CN(C(c4cc(C)nn4C)=O)CC23)=O)c(O)n1 50417,N1(C(CCc2cc(OC)no2)=O)C2CCC1CC(NC(C1CC(=O)N(C)C1)=O)C2 50418,Cc1ccc(C(=O)NCC(=O)NCCC(O)CNC(C23CC(CO2)C3)=O)s1 50419,c1(CC(=O)NCC(C)N(C(=O)Cc2nccn2C)CC)ncc(F)cn1 50420,C1(C(=O)NC2(CNC(C3(F)CCS(=O)(=O)C3)=O)CC2)CC(c2ccccn2)=NO1 50421,C1(CC(=O)OCC)CCN(C(c2cccc(Br)c2Cl)C(=O)NCCSC)C1(C)C 50422,c1(C(=O)NCC(CN(C(C=C(COC)C)=O)C)C)ccc2c(c1)SCC(=O)N2 50423,N1(C(C(C=CC)O)=O)CCN(C(=O)CSCCCc2ccccc2)C2CC12 50424,CC1CC(CNC(=O)C#CC(=O)NC2CC2)CN1C(C1CC(=C2CCC2)C1)=O 50425,N1(C(C(C)Oc2cccc(Cl)c2Cl)=O)CCC2(CC(NC(=O)C(F)Br)CO2)C1 50426,c1(OC)ccc2c(C(=O)NC(C)CNC(C3CC4(CSC4)C3)=O)coc2c1 50427,c1(NCC(C)(C)CC2CCC2)ccc2c(c1)OCC2 50428,C(=O)(CCC[N+](=O)[O-])N(C1CCN(C(C(C(C)C)F)=O)C1)CCO 50429,c1(C(N(CC(CC)NC(=O)CSC(F)F)C)=O)ccc2c(C)noc2c1 50430,CC1(NCC(C)(O)CN2CCOCC2)CS(=O)(=O)C1 50431,CS(=O)(=O)C1CCC(CNC(=O)C(=O)NC2CCC(O)C2)CC1 50432,C(CC(C)C)(C(=O)NC(C1CCCCC1)CNC(=O)CN1CCN(C)CC1)OC 50433,CC(C)CC(C)(O)C(=O)N1CCN(C)C(C(=O)NCc2cnn[nH]2)C1 50434,c1(C(=O)NC(CCNC(c2cc(C)n(C)n2)=O)C)c[nH]c2cccc([N+](=O)[O-])c12 50435,CCC(CC(=O)N1CCN(C(=O)C(=Cc2cccnc2)C)C2(CC2)C1)C(F)F 50436,c1(NC)c(OC)cc(OC)cc1N.C12(CCCC1)C(=O)NCC(CO)NC2=O.COC 50437,c1(OC)cc(C(=O)NC2CCCC2NC(=O)CC2CC2(Cl)Cl)cc2c1OCC2 50438,C(=O)(CC1OCCc2ccsc21)NCC1C(C)CCCN1C(=O)Cc1cccs1 50439,CC1CCN(CC(=O)Nc2ccnc(C(=O)NCc3cccnc3O)c2)CC1 50440,N1(C(C=C(C)C(C)(C)C)=O)CCOC(CCNC(=O)CN2CC(C)C2)C1 50441,Cc1cc(CCC(=O)NCC2CC(NC(=O)Cn3nccn3)C(O)C2)nn1C 50442,c1(C(=O)NCC2CCN(C(C3(CC)CCCO3)=O)C2)cncc([N+](=O)[O-])c1 50443,C12(NC(C=C(C)c3ccco3)=O)CCCCCC1N(C(c1n[nH]cc1F)=O)CC2 50444,c1(C(=O)NC(C(C)NC(=O)CSc2nnc(S)s2)C)cc2cccnc2[nH]1 50445,Cc1nc(O)sc1C(=O)NC1CCOCC1C(=O)NCCC1CC(F)(F)C1 50446,Cn1c(-c2noc(C34COCCN3CC4)n2)ccc1Cl 50447,c1(C(=O)NC2CN(C(C3(C=C)CCC3)=O)CC2C)ccc(NC(=O)OC)cc1Cl 50448,c1(CC)ncc(C(N2CC(NC(=O)C(C)CN(C)C)C(C(F)F)C2)=O)c(O)n1 50449,C1(CNC(C(CC#C)C2CC2)=O)CN(C(c2cccn2CCC)=O)CC12CCC2 50450,CCC(C(=O)NC(C)(C)C=CC(=O)N(C)CCn1cncn1)n1ccnc1 50451,c1(-n2c(C3C(CC)C3)nc(C3CC3(C)C)n2)ccc(C)cc1OC 50452,CCC(C)CC(=O)C(=O)N(C(C)C(=O)NCCc1cc(C)on1)C1CC1 50453,C1(CC(N2CC(COC)(NC(=O)CC3(F)CCOCC3)C2)=O)(OC)CCOCC1 50454,C1(NC(C2CC(=C)C2)=O)CC(CNC(c2ccc(NC3CC3)nc2)=O)C1(C)C 50455,c1(C(=O)NC(CNC(CN(C(C)C)C)=O)C(C)C)cn2c(n1)SCC2 50456,S(=O)(=O)(c1nc(N2CCC(C(C)(C)CO)CC2)ccc1Br)NC(CC)CO 50457,c1(C(=O)NCC2(C)CCN(C(C3CCCCO3)=O)C2)ccc2cnsc2c1 50458,N1(C(C2C(=C)C2)=O)CCCCCC1CNC(c1cc(C(C)C)nn1C)=O 50459,C1(CC(=O)N(CCO)Cc2cc(NCc3cccs3)no2)CCCCO1 50460,c1(CCC(=O)NCC(CC)OC)ccccc1CNC(=O)CN1C(=O)CCC1=O 50461,c1(C(=O)Nc2c(C(N(C)Cc3ccc(CC)cc3)=O)c[nH]n2)cc2occc2[nH]1 50462,c1(N(C)C)ccccc1N(C(=O)C(=O)NCC(=O)Cc1ccccc1)C 50463,C(=O)(C(C)C(O)CCCC)N(CC(N1CCCC(C)C1CCO)=O)CC#C 50464,Cc1ccc2nn[nH]c2c1NC(=O)N=c1cc(C(F)(F)F)[nH][nH]1 50465,CCCCCCC(CC)C(=O)N(CCCNC(c1cc(C(=O)OC)no1)=O)CC 50466,C1(C(=O)NC2CC(C(CC)CC)OCC2)CC2(CCOCC2)CCO1 50467,N1(C(c2ccccc2F)C)CCC(CN(C)C(C23CCC2C3)=O)CC1 50468,N1(C(CC(C)F)=O)CCN(C(c2csc(CO)n2)=O)CC1c1ccc(F)cc1 50469,N1(C(C(CCCC=C)NC(C2CSCC(=O)N2)=O)=O)CC(C)OC2(CCC2)C1 50470,C1(C(N2CCN(C)CC2)=O)CCCC(NC(=O)CCc2nc(=N)[nH][nH]2)CC1 50471,N1(C(c2cccc(COC)c2)=O)CC(NC(C2CCCCC2C#N)=O)CC(C)C1 50472,C1(C(N2C(C(N(CCn3c(C)ncc3)C)=O)C(C)C2)=O)CCCC(C)(C)C1 50473,C12(C(=O)NCC#CCNC(c3cc(C)nc(O)n3)=O)OCCCC1C2(F)F 50474,C1(C(=O)OC(C)(C)C)CCCCN1S(=O)(=O)NCC1(c2ccon2)CCC1 50475,c1(C(N2CCC(NC(c3c(C(C)C)[nH]cc3)=O)C(C)C2)=O)cccc2cnnn12 50476,c1(C(N2CCC(CC=C)(NC(C3CC34CC4)=O)C2)=O)cc2c(Br)cccn2n1 50477,N1(C(=O)C2=CS(=O)CCC2)CCOCC2(COCCN2c2nc(Cl)ncc2F)C1 50478,CCS(=O)(=O)CC(=O)N1CCCCC1C1CCN(C(C2CC2F)=O)C1 50479,c1(NC(c2c(C(C)C)scn2)=O)cc2c(cc1Br)CCC(=O)N2 50480,N1(C(C2C(CC)C2)=O)CCC(O)(CCNC(c2ccc(CC3CCC3)cc2)=O)C1 50481,CC1CN(C(=O)CC2C(C)(C)C2(C)C)CC1NC(c1ccc(C2CC2)o1)=O 50482,c1(CC)cnccc1C(N1CCOC(CNC(c2c[nH]c(=NC)s2)=O)C1)=O 50483,N1(C(C(C)OCCC(C)C)=O)CCNCC(O)C1 50484,c1(C(=O)NCC2CC(OC)CN2C(c2cncc(Br)c2)=O)cn2c(n1)CCC2 50485,CC1(C)CCCCC1(C)NC(c1cccc(CNC(c2cscn2)=O)n1)=O 50486,N1(C(C(CC)O)=O)CC2CCC(NC(c3ccc(C(F)(F)F)cc3)=O)C2C1 50487,c1(C(=O)NC2(C(=O)NCCC(COC)OC)CCCC2)nc(C)cc(O)n1 50488,CCN(Cc1ncc[nH]1)N1CC(C(F)(F)F)C(S(C)(=O)=O)C1.C1CCCO1 50489,c1(C(=O)NCC=C2CCN(C(CC(C)C3CC3)=O)CC2)cc(Cl)cc([N+](=O)[O-])c1 50490,C1(NC(=O)CCCC2CCCC2)CC2(C1)CC2C(=O)NOC1CCOC1 50491,c1(C(N2OCC(C)C2)=O)cc2cc(-c3cn(C)c4ncccc34)ccn2n1 50492,N1(C(CCCCC#C)=O)CCC2(CC1)CC2CNC(c1c[nH]ccc1=O)=O 50493,C1(N(c2cncc(Cl)n2)C)CCCN(C(=O)OC(C)(C)C)C1=O 50494,N1(Cc2cccc(C(N)=O)c2)C(=O)CN(CC2CC(F)C(=O)N2)C1=O 50495,CC1CN(C(=O)CCP(C)(C)=O)CC1(C)C(N1CCCC(CN=[N+]=[N-])C1)=O 50496,c1(C(C)NCc2noc(C(C)(C)C)n2)ccoc1CNC(C1(CCC)CCC1)=O 50497,C(C)(CN=c1[nH]c2ccccc2cc1C#N)NC(C1CCC(C)CC1)=O 50498,c1(NC(C2CCN(C(=O)CCC3CCC3)CC2O)=O)cncc(Cl)c1Br 50499,C(=O)(C1=NOC2(CCC2)C1)NCC(CN(C(=O)CCSc1cccs1)C)(C)C 50500,c1(CC)cccnc1C(N1CCC(C(C)NC(=O)CNC(C2CCC2)=O)CC1)=O 50501,C1(NC(C(C(C)C)SC)=O)CC2CCC1N2C(c1c(C)noc1C1CC1)=O 50502,N1(C(CCCCOC)=O)CCC(C2CCN(C(=O)Cc3c[nH]ccc3=O)C2)CC1 50503,c1(C(=O)NC23CC(NC(C45CCCC4CC5)=O)(C2)C3)cc2ncccc2s1 50504,Cc1ccncc1C(=O)N(C)CCOCCN(C(=O)Cc1cscc1F)C 50505,CCC(CC)C(F)C(=O)NCCN(C(=O)Cn1cnnn1)C 50506,Cc1ccc([N+](=O)[O-])c(C(=O)NCC2CCN(C(=O)CCC(C)(C)C#N)CC2)c1 50507,N1(C(C2OCC(=O)C2)=O)CC2CC(N=c3cnc(F)c[nH]3)C2C1 50508,c1(C(=O)NC2C(C)CN(C(=O)C=CC(C)(C)C)C2)nn(C)cc1S(C)(=O)=O 50509,N#CC1(CC(=O)NC2CCOC(CNC(=O)C=CC3CC3)C2)CCCCC1 50510,c1(CNC(c2nnnn2C(C)(C)C)(COC)C)nc(O)c2cnn(C)c2n1 50511,c1(C(=O)NCC2(OC)CN(C(=O)CN3C(=O)CCC3=O)C2)ccc2cc[nH]c2n1 50512,C1(C(=O)NCC(C)NC(=O)CCCC(N)=O)CC12CCC1(CC2)OCCO1 50513,c1(C(N(C2C3CN(C(c4cnc(C5CC5)[nH]4)=O)CC23)C)=O)ccc(O)nc1Cl 50514,C1(C(C)(C)NC(C2CN(C(C)C)C2)=O)CCN(C(=O)Cc2nncn2C)CC1 50515,c1(CNC(N2C(CC)C(=O)NCC2)=O)ccc2c(c1)cc(C)n2C 50516,C(C1CN(C(=O)CC2CCN(C)C2=O)CC1C(=O)NCC(F)C1CCC1)=CC 50517,c1(NC(C2N(C(C3(COC)CCC3)=O)CCC2)=O)nnc2ccc(Cl)nn12 50518,O=C(NN1CC(C(=O)O)C1)C1CC=CCC1OCc1ccccc1 50519,CCC(C)C(CC(=O)N1CC(O)C1)NC(C1CCCS1)=O 50520,c1(C(=O)NCC(C)(C)NC(C2CC3(CCC3O)C2)=O)cc(F)cc(F)c1O 50521,C(=O)(CCCC(=O)N1CC2(CNC(=O)CC3(C)CC(F)(F)C3)CC1CO2)N(C)C 50522,c1(NC(C2(C)CCCN2Cc2ccc(O)cc2O)=O)ncnc2sc(Br)cc12 50523,c1(C(N(CC(CNC(CSCC(C)C)=O)C)C)=O)cc([N+](=O)[O-])c[nH]1 50524,c1(C(=O)NC2CN(C(c3c(C)nns3)=O)C(C)CC2)cccc2nc(Cl)cn12 50525,c1(NC(C2CCCN(C(=O)CSc3cccc[n+]3[O-])C2)C)ncc(C#N)cc1Cl 50526,N1(C(COCC#C)=O)CC2CC2(C(=O)NC(COC(C)C)CC)C1 50527,Cc1cnc(C(=O)NCCNC(C23CC(F)(CO2)C3)=O)cc1Br 50528,C1(C(N2CCC(Cc3cn(CC4CC5CCC4C5)nn3)C2)=O)CCC(C2CC2)C1 50529,C1(O)(C(C(=O)N(CC(=O)NC2(c3cc[nH]n3)CC2)C2CC2)F)CCCC1 50530,C1(NC(c2cnc(CC3CC3)nc2O)=O)CCCC2CN(c3ncccn3)CC12 50531,C1(C(=O)NC2(CO)CN(C(C(C)(C)C3CCCC3)=O)C2)CCCCC1F 50532,N1(C(C2C(C)CCO2)=O)CCC(CCN(C)C(c2ccnc(CO)c2)=O)CC1 50533,C1(CC#C)(C(=O)NCC2CCN(C(=O)C(c3ccccc3)C)C2)CCCC1 50534,n1(CC(=O)NC2(C3N(C(CC(C)F)=O)CCC3)CC2)cc2ncccc2n1 50535,N1(C(c2ccc(=NC)[nH]c2)=O)CCCC2(NC(c3nc(F)ccc3Cl)=O)CC2C1 50536,C#CC(CC(C)C)NC(=O)C(C)CN(C(=O)C(C)(C)CC)C 50537,CN1CCCC12CN(C(C1(C(=O)O)CCN(C(=O)OC(C)(C)C)CC1)=O)C2 50538,c1(OC)ccc(C(N2CCN(C(C3CC(O)C3)=O)C3CC23)=O)c(OC)c1C 50539,C(CC(C(C)C)NC(c1cccc(-n2cncn2)n1)=O)N(C(C(C=CC)O)=O)C 50540,C1CN=C2N=C(C=C(C)N2)NC2CC(COC)CN(C2)C1.C(C)(C)(C)OC1CC1 50541,C(CCC1CCC1)(C(=O)N(C1(CO)CC1)C)NC(COC(CC)CC)=O 50542,c1(CC)cccc(C(N2CCC(C(N)=O)(CO)C2)c2ccccc2)c1F 50543,c1(C(N2CC3CC3(C(=O)NCCc3cc[nH]n3)C2)=O)c(F)ccc(F)c1Cl 50544,N1(C(C(n2ccc(C)n2)C)=O)CC2(CC2)CC1C(=O)NCC1CCOC1C 50545,c1(C(=O)NC(CC2CN(C(C3CC(CCC)C3)=O)C2)C)cc(C)nn1C 50546,C12(NC(C3(S(C)(=O)=O)CC3)=O)CCOC(CNC(C3(C(F)(F)F)CC3)=O)(C1)C2 50547,c1(C(=O)NCC2(O)CN(C(C(C)NC(=O)NC)=O)C2)ccc2cc[nH]c2c1 50548,Cc1cccc(C(=O)NC2CCCCC2CC(=O)NC(c2cccnc2)C)c1N 50549,C1(CNC(=O)Cc2ncccc2F)COCCN(C(c2n[nH]c3c2COC3)=O)C1 50550,c1(CNC(=O)NC2(C)C(C)OCC2)ccc(S(N)(=O)=O)cc1 50551,c1(C(N2CC(C(=O)Nc3ncc(SC)s3)NCC2)=O)cc(O)c(O)c(Cl)c1 50552,c1(C(=O)NC(C2CN(C(=O)C=CCN(C)C)C2)C)ccnn1C1CC1 50553,C1(CC)CCCCC1C(N1CC2C(CNC(=O)CCc3ccncc3)C2C1)=O 50554,n1(CC)cc(C(=O)N(C2CCN(C(=O)C(O)COCc3ccccc3)C2)C)nn1 50555,N1(C(C2(CCCC)CC2)=O)CC(NC(=O)CNS(=O)(=O)C2CC2)CC(O)C1 50556,N1(C(C(C)CO)=O)CCCCC(N(C)C(c2cnnc(-c3ccccc3)c2)=O)C1 50557,N1(C(Cc2c(C)cco2)=O)C2CCC1CN(C(C1CCC(C)(F)CC1)=O)C2 50558,N1(C(c2cc(C)nnc2)=O)CC(=O)NCC1C(=O)NCCCSC(F)F 50559,C1(C(=O)NC(CC2CN(C(C3CCC(C(=O)OC)C3)=O)C2)C)CC12CCOC2 50560,N(C(=NCCc1ccccn1)N1CCCC(O)CC1)CC(C(=O)OC)C 50561,C(C(C)C(C)C(=O)N1CC(C(C)NC(c2ccc(F)cc2F)=O)C1)OC 50562,CCC(C)CCC(=O)NCC12CC1CN(C(=O)C=CSCc1ccco1)C2 50563,N1(C(c2c(C(C)(C)C)ncnc2)=O)CC2(C1)CN(C(=O)CC1CCC(C#N)C1)C2 50564,N1(C(C2C(NC(c3c(C)n[nH]c3)=O)CCC2)=O)CCN2CCOCC2C1 50565,C1(CC(N2CCC(COC)(NC(=O)CCCF)C2)=O)CN2CCN1CC2 50566,N1(C(c2c(OC)c[nH]n2)=O)CCN(C(=O)Cc2cnccc2Cl)CC1C 50567,C1(CNC(CC2ON=C(C)C2)=O)(CNC(c2cncc(Cl)c2)=O)CC12CCC2 50568,c1(C(N2CC(COC)(NC(=O)CN(C(=O)C(C)C)C)C2)=O)ccc2c(n1)CCOC2 50569,C1(NC(C(C)(C)C2CCOCC2)=O)CC(F)CN(C(C2C3COCC23)=O)C1 50570,Cc1c[nH]cc1C(N1CCC(NC(c2ccsc2-n2cnnn2)=O)C1)=O 50571,Cc1cnn2ccc(C(=O)NC(C)C(CO)NC(=O)C(n3nccc3C)C)nc12 50572,N1(C(C2=C(C)CCC2)=O)CC2CCCC(CNC(c3cc(C)cs3)=O)C2C1 50573,C(N(O)C(=O)C(O)Cc1ncccn1)c1cn(C(C2CCCCC2O)C)nn1 50574,C=C(C)CCC(=O)NC1CCC(CCNC(c2nccnc2C)=O)C1 50575,N1(C(CCOC)=O)CC2CCC1C(CNC(c1cc(Cl)ccc1O)=O)C2 50576,n1(CC(N2C(C(CNC(C)=O)Cc3ccccc3)CCC2)=O)cc(F)ccc1=O 50577,c1(C(=O)NCC(=O)Nc2ccc(C(C)=O)cc2)c(N)cc(F)cc1Cl 50578,C=C(Cl)C(C)(C)C(=O)N1CC2(CC)CC1(CNC(=O)C(C)NC(=O)C(C)(C)C)C2 50579,c1(C(N2CCCCC(NC(C(COC)OC)=O)CC2)=O)nc2n(c1Cl)CCCC2 50580,O=C1CC2(C1)CC(CNC(=O)CCn1cc(-c3ccc(C(F)F)cc3)nn1)C2 50581,N1(C(C=C(C)Cl)=O)CC2CCCC1C2CNC(=O)CSCCN(C)C 50582,Cc1occc1CC(=O)NC1CC1CNC(c1nocc1-c1ccccc1)=O 50583,C1(CC)CCCN(C(c2cc(CNC(=O)CCc3ccn(C)n3)nn2C)=O)CC1 50584,c1(C(=O)NC(C2CCCCC2)C(N2CC(O)C(O)C2)=O)ccn2nccc2c1 50585,C(=O)(C(C)(CO)NC(=O)C(C1CCN(C(=O)CC2CCOCC2)C1)C)OC 50586,N1(C(c2ccc(CN(C)C)nc2)=O)CC2CC(C1)C2NC(c1ccccc1F)=O 50587,N1(C(CC2(COC)CCCCO2)=O)CCC2(CCC(NC(=O)C3CC3)C2)CC1 50588,N1(C(Cc2ccc(C#C)cc2)=O)CC2CCC(C1)N2C(C1CC1C(=O)OC)=O 50589,c1(C(c2n(CC)nnn2)NCC(C)(C)COC)ccc(Br)c(F)c1F 50590,N1(C(CC)=O)CCOCC(C(=O)Nc2cccc(CC(F)(F)F)c2)C1 50591,c1(C(=O)NCC2(NC(C3CN(C)C3)=O)CCCCC2)cc2c(cc1N)CCC2 50592,C1(C(=O)NC(COC)CO)N(C(=O)CCNC2CC2)CCCC1(C)C 50593,c1(C(N(CCN(C(=O)C(O)C(F)F)C(C)C)C)=O)cc(Cl)ccc1C(F)(F)F 50594,Cc1ccc(C(N2CC(c3ccccc3)(NC(c3cnc(S)[nH]3)=O)C2)=O)cc1 50595,N1(C(C(C(C)O)(F)F)=O)CCC2(CC1)CCN(C(C1(CCN(C)C)CC1)=O)CC2 50596,C1(CNC(C2(C)CC3CC3C2)=O)CCN(C(=O)C(O)C2CCC2)CC1(F)F 50597,c1(N(C)C)ccc([N+](=O)[O-])c(C(=O)NC2CN(C(C3CCC3(F)F)=O)CC2O)c1 50598,C1(C(=O)NCC(C#C)OC)(COC)C=CCN1C(=O)CCOCCN(C)C 50599,CC1(C)CC(CNc2cc(N3CCOC(c4ccc(F)cc4)C3)ncn2)CO1 50600,c1(C(CNC(C(=O)Nc2cn(CCC#C)nc2)=O)F)ccc(Br)cc1Cl 50601,C1(CNC(c2c(CC)noc2C)=O)CCN(C(c2c[nH]c(C)c2)=O)CCC1(F)F 50602,N1(C(CC(C)F)=O)CCCC(CNC(C2(F)CCCCC2)=O)CC1 50603,CC(CF)CC(=O)N(C(C)CNC(=O)C(c1ccc(Cl)cc1)(F)F)C 50604,c1(C(=O)NCC(C)NC(c2c(F)ncc(OC)c2)=O)ccc(F)c(C)c1N 50605,C1(COCC)CCCN(C(CC2CCC3CC23)C(=O)N(C)C(C)C)C1 50606,CCC(C)(C(=O)NC1CN(C(c2ccccc2C)=O)C(CC)(CC)C1)OC 50607,c1(C(=O)NC2(CC(=O)OC)CCCOC2)sc2ccsc2c1C 50608,c1(CCC(=O)NCc2c(C)ocn2)ccnc(Cl)c1F 50609,C(=O)(C(CC(C)C)NC(C)=O)N(C1C2CN(C(C3(CO)CCCO3)=O)CC12)CC 50610,c1(C(=O)NC(CN(C(c2c(COC)nn(C)c2)=O)C)C)cc2cc(Cl)ccc2s1 50611,c1(C(=O)NC2(CN(C(C3CC(C)NC(=O)C3)=O)C)CC2)ccc(Cl)c(F)c1N 50612,c1(CC)ccc(C=CC(=O)NC2CN(C(=O)CCN3CCCC3)CC2SC)o1 50613,CC(CS(C)(=O)=O)C(=O)NC(C)(CNC(c1cc2c(ccn2C)[nH]1)=O)CO 50614,C1(OC)CC(N(CC(=O)OCCOc2ccc(C)cn2)C)C12CCOCC2 50615,c1(CCC(N2CC(NC(CSCCCC)=O)C2)=O)cc2ccccc2o1 50616,C1(C(=O)NCC(CCC)C)(C(C)C)CCN(C(=O)C(CO)NC(N)=O)C1 50617,Cc1cc(C)n(CC(N2CC(N(C(=O)Cc3c(C)noc3Cl)C)C2)=O)c(=O)n1 50618,c1(C(=O)NC2CN(C(C3(c4ccncc4)CC3)=O)CC2F)cc2cccnn2n1 50619,C1(CNC(CCC(=O)NCC)=O)CCCN(C(=O)C2=CCCSC2)CC1 50620,c1(OC)ccc2c(CN3CCNCC3C(=O)Nc3ncc(Cl)cc3Cl)c[nH]c2c1 50621,c1(-n2cc(C3(F)CCN(C(C(C)OCCOC)=O)C3)nn2)cccc(F)c1Br 50622,C1(C(C)=O)CC(C)(NC(n2cc(C(N3CCCC3)(C)C)nn2)C2(O)CCOC2)C1 50623,c1(COC)ocnc1C(c1nnnn1C(C)C)NC(CF)CF 50624,c1(CC(N2C(CNC(c3c(CC)nco3)=O)C=CC2)=O)ccc(CSC)c(C)c1 50625,C1(NC(c2cnc(C3CC3)[nH]2)=O)CC2CC1N(C(c1csc(Cl)c1Cl)=O)C2 50626,c1(C(N2CC=CC(O)C2)=O)cnc2[nH]ccc2n1.C1(N)CCCO1 50627,N1(C(Cc2cc(C)ncc2)=O)CCC(C)N(C(c2cccc3nsnc23)=O)CC1 50628,N1(C(c2n(C)c(=O)ccc2)=O)C2CCCC1CN(C(C1CCC13CCC3)=O)CC2 50629,Cc1cccc(C)c1CS(=O)(=O)NC(C1CCC(F)(F)C1)C 50630,C1(CC)(CC)CC(NC(c2cnn(C)c2C(F)F)=O)CN1C(=O)CC1CCOC1 50631,C1(NC(Cc2c(C)ocn2)=O)CN(C(C2CN(C3CCCCC3)C2)=O)CC12CC2 50632,Cc1nc(-c2c[nH]c(C(N3CCC3CNC(=O)CC3CC4(CC4)C3)=O)c2)cs1 50633,N1(C(c2cc(C(C)C)on2)=O)CCC2(CCN(C(c3ccc(F)cc3Cl)=O)C2)C1 50634,C1(CC(=O)N(CC(=O)NCCOC(CC)CC)C2CC2)CC2C=CC1C2 50635,n1(CCNC(=O)Nc2cnns2)ccc(=O)cc1.c12nnnn1C2C1CC1 50636,CC1CCC(C2CCCC2)CN1C(=O)Nc1cnc(Br)c(F)c1 50637,c1(OC)ccc(Cl)cc1C(N1CCC(NC(=O)CC2(C(F)(F)F)CC2)C(O)C1)=O 50638,N1(C(CC2(C=C)CCC2)=O)CC2CC2(CNC(=O)CC2CCC(=O)N2C)C1 50639,c1(C(N(C2CCN(C(=O)C=Cc3cn[nH]c3)CC2)C)=O)cc(O)cc(C#N)c1 50640,COn1cnc(C)c1C(=O)NCC(c1ccccc1F)NC(=O)Cc1ccns1 50641,C(=O)(CC(C)CC(C)C)NCCCCN(C(c1cccc(NC(=O)OC)c1)=O)C 50642,C(=O)(C1CCc2ccccc21)N1CC(COC)(NC(=O)C(C2CCCC2)OC)C1 50643,N1(C(C(CC)(C)C)=O)CC2CCC2(NC(=O)CCOc2cccc(F)c2)C1 50644,C(=O)(C1CCCc2scnc21)NC1CN(C(COCCOCC#C)=O)C1 50645,Cn1nc(C(=O)NC2CCN(c3nc(C4CC4)ns3)CC2O)c2c1CCCC2 50646,C1(CNC(c2cc(C(C)C)n(C)n2)=O)C(C)CCCN1C(c1cnn(C)c1)=O 50647,C1(CNC(CCC2N(C)CCCC2)=O)CCN(C(c2ccc[nH]2)=O)CC1O 50648,CC1(NC(=O)C(O)C(C)(C)C)CCN(C(=O)Cn2cnnc2)CC1 50649,C(=O)(C(C(C)O)NC(=O)CC1CCCN(C)C1)N(C1CC(C)C1)C 50650,C1(C(N(CCCNC(=O)COC2CCOC2)C2CC2)=O)CC=CCC1 50651,Cc1noc2nc(C(=O)N(C3CCCN(C(=O)CC4CNC(=O)C4)C3)C)ccc12 50652,CC(c1ccccc1)=CC(=O)NC1CC1NC(=O)C(C)n1ccnn1 50653,C1(NC(C2CCCN(CC)C2)=O)CC2CN(C(=O)Cc3nccs3)CC2C1 50654,C1(COC)CN(C(C2(C)CCCCO2)=O)CCN1C(=O)CN1CCC(O)CC1 50655,N1(C(CC2OCC(C)(C)C2)=O)CC(C(N2CC(N3CC(F)C3)C2)=O)C(F)(F)C1 50656,c1(C(=O)NC2CCCN(c3ccc(C#N)cc3)C2)cc(Cl)sc1S(N)(=O)=O 50657,c1(CN2CCC(C)(CNc3ncn(C)c3C(F)(F)F)CC2)ccc(C#N)c(F)c1 50658,c1(N(C(CCSCC)C)C)nnc(-c2nc(C)no2)n1CC(C)C 50659,c1(N2CCN(C)C(CNC(c3cn4c(n3)CCC4)=O)C2)ncnc2[nH]ccc12 50660,c1(C(C(=O)NCC(C)(C)F)NC(C(C2CCC2)OCC)=O)ccccc1 50661,C1(C)(C(=O)OC)CNCCN1Cc1ccncc1 50662,c1(N(C(c2ccc(Cl)o2)C(=O)Nc2ccccc2)C)ccc(NC2CCC2)cc1 50663,CN(CCOCc1ccccc1)N1CC(CO)OC2(CCC2)C1 50664,n1(CC2CC(C)C2)nc(COc2cnn(C)c2)nc1-c1cc(C2CC2)[nH]n1 50665,C1(NC(C=C(C)Cl)=O)CCCCC12CCN(C(=O)C=Cc1ccoc1)CC2 50666,N1(C(C(CCC#C)NC(c2cnc(N)cn2)=O)=O)CC(O)C2(CCCC2)C1 50667,c1(CC)cc(C(N2CCCC2CCC(C)C)C(=O)NCCC#N)ccc1Cl 50668,Cc1nc2cccc(C(=O)NCC(O)CNC(=O)Cc3cncc(O)c3)c2[nH]1 50669,C12(CNC(c3ccn(CCF)n3)=O)CC1CN(C(C1C=CCC1)=O)C2 50670,CCC(O)C(C)(C)C(=O)NCC(=O)NC1C2CCCC1CCC2 50671,c1(OC(C(=O)NCCC(C)N(C(c2n(CC)ncc2)=O)C)C)cccc(CO)c1 50672,c1(C(=O)NCC2CC(C)N(C(=O)CC3CCCO3)CC2)ccc2c(n1)CCC2 50673,CCN=c1[nH]c(C(N2CC(CNC(=O)CC3CC4CC4C3)C3(CC3)C2)=O)cs1 50674,C1(C(N2CC(c3onc(C)n3)C2)=O)CCOCC1NC(C12CC(C#N)(C1)C2)=O 50675,N1(CC(=O)Nc2c(C)ccc(NC(=O)CC(C)C)c2)CC2CS(=O)(=O)CC(C1)O2 50676,CCCC(CC)CC(=O)N1CCCCC(NC(c2cc(C3(Cl)CC3)n(C)n2)=O)C1 50677,C(=O)(CC(P(C)(C)=O)c1ccccc1)N(CC(O)CNC(C1(C)CCC1)=O)C 50678,C1(CCOC)CN(C(C2(CC(F)(F)F)CC2)=O)CCN1C(=O)CCS(C)=O 50679,N1(C(c2c(C)n(C)nc2)C(=O)O)CCN(S(=O)(=O)N2CCN(C)CC2)CC1 50680,CC(C)(C)S(=O)(=O)CC(=O)NCC1CCCN1C(C1CCC(C(F)(F)F)CC1)=O 50681,C1(C(=O)NC2(c3onc(C)n3)CC2)CCCCCCN1C(=O)C(C)CC#N 50682,CCCC(CCNC(=O)CCC1(C)CN(C(C2CCC(O)CN2C)=O)C1)CCC 50683,C12(C(=O)NCC(C(=O)NCCN3CC=CCC3)OC)C(=O)C3CC1C2C3 50684,c1(OCC(N2CC(NC(=O)C=Cc3ccccc3)C(O)C2)=O)ccc(F)c(Cl)c1 50685,C(c1ccccc1)=CCCN1CC(CNC(C2N(C(C)=O)CCC2)=O)C1 50686,C1(CNC(Cc2ccc(C)s2)=O)CCC2(CN(C(c3ccccc3O)=O)C2)O1 50687,CCC(CC(=O)N1CC2C(NC(c3ccc(F)c(C(F)(F)F)n3)=O)C2C1)C(F)F 50688,N1(C(C2C(C=C)C2)=O)CC(O)(CN(C(=O)CC2COCC2O)C)C1 50689,Nc1cnc(C(=O)NC2CCC2NC(=O)CC=Cc2ccccc2)c(Cl)c1 50690,C=CC(C)(O)C(=O)NCCC1CCC(NC(=O)CC(CC)OC)C1 50691,CC#CCC(C(=O)NCCC(O)CCC)NC(=O)COc1ccccc1 50692,c1(C(C)(C#N)NC(C(C)Sc2nn[nH]n2)=O)ccccc1Br 50693,N1(C(CCCOCC=C)=O)CCN(C(CNC(c2cc(C)cs2)=O)C(F)F)CC1 50694,C(=O)(CC(CC)C(C)(C)C)N(CC=CC(=O)NCc1snc(CC)n1)C 50695,c1(C(N2CC(C)(NC(CC(CCC)C)=O)C2)=O)cc2c(nc1O)CCC(CC)C2 50696,n1(C(CC)C)cc(-c2nc(COc3ccccc3)no2)c2ccccc12 50697,Cc1c(C(C)NC(c2ccc(O)nc2)C)cccc1Cl 50698,N1(C(C(=O)NC(CN(C(C(C)SCC)=O)CC)CO)C2CCCC2)CCOCC1 50699,C(=O)(C(F)C(F)(F)F)NC(C)CCNC(C1(CNC(N)=O)CC=CC1)=O 50700,C=CCCCCCC(=O)N1CC2CC(NC(c3cc(C)oc3CC)=O)CC2C1 50701,C=CCCCCC(=O)NC(C1CCN(C(=O)C=C(Cl)Cl)C1)C 50702,c1(C(=O)NC2(CC=C)CN(C(=O)CS(=O)CC)C2)cnc(F)c(C)c1 50703,C1(C(CNC(C2(C)CCCC2)=O)O)CCN(C(c2ccc(O)nc2)=O)CC1 50704,C(CNC(c1cccc(CCCCO)c1)=O)(CC(F)(F)F)NC(C(C)OCC)=O 50705,S(=O)(=O)(c1ccc(-c2ccc(C(C)NC)cc2)s1)N(CC=C)C(C)C 50706,c1(C(=O)NCC2CCCN(C(c3c(CC)n(C)nc3)=O)C2)c(C)cc(O)cc1C 50707,C1(NC(C=C(COC)C)=O)CC(CNC(=O)CCc2cccnc2)C1(C)C 50708,c1(CCC(N2CCC(N(C(=O)C(C)n3cnnn3)CCC)C2)=O)ccnc(Cl)c1 50709,C=C(C)CCCC(=O)N1CCC(C)C(CC(N2CC(CO)CC2CO)=O)C1 50710,c1(C(N2CC(C)C(NC(=O)CCCCC3CC3)C2)=O)ncc(C(F)(F)F)cc1Cl 50711,c1(N(CCc2ccc(C)cc2)C)nc2c(c(=NC3CCCSC3)[nH]1)CC(C)CC2 50712,C(=O)(CCCCCNC(N)=O)NC1(F)CN(C(CN2CC(C)(OC)C2)=O)C1 50713,C1(CCOC)CCN(C(=NCCc2ccnc(OC)n2)NCC2CCCCO2)C1 50714,N1(C(CC)=O)CC(=O)N2CCOCC2(CNC(=O)CC2CCCCC2(F)F)C1 50715,c1(CC)cccc(C(=O)NC(C(=O)NC2CN(C)NC2=O)C2CCCC2)c1 50716,C1(COC)(NC(=O)CCSC(F)(F)F)CCN(C(c2c[nH]nc2C(C)(C)C)=O)C1 50717,c1(C(=O)NCCCN(C(C(C)C(C)(C)O)=O)C2CC2)csc2ccccc12 50718,C1(C)(C(N2C(C(C)=O)CCCC2)=O)CC12CCN(Cc1ncccc1Cl)CC2 50719,c1(C(=O)NCCC(CNC(C2(C)CC2)=O)O)ccc(C(N2CCCCC2)(CC)N)cc1 50720,N1(C(CNC(CCC)=O)=O)CCN(C(=O)C(C)NC(C)(C)C)C(CC(C)(C)C)C1 50721,CCCCCC(F)C(=O)N1CCCC1(C(=O)NCC(C)C(=O)OC)CC 50722,Oc1nc(CCNCc2cc3c(O)ncnc3cn2)nc2ccccc12 50723,c1(OC)cc2c(cc1OC)C(NC(c1occ3c1CCC3)=O)CCCC2 50724,c1(OC)c(Cl)cc(C(N2CCC(NC(=O)CCC3CCC(=O)N3)C2)=O)cc1Cl 50725,N1(C(c2c(CCC)occ2)=O)CC2(CC(NC(=O)C=CCN3CCCCC3)C2)C1 50726,c1(N2CCC(CC)C2)nc(=NCc2nc(C(F)(F)F)n[nH]2)[nH]c2c1CCCC2 50727,c1(NC(C(C)N(CC(F)C(=O)N(CCCCSC)C)CC)=O)c(F)cccc1F 50728,CC(C)CC(C)(C)C(=O)NC1COCC1NC(c1ccccc1OCCF)=O 50729,c1(C(=O)NC2CCN(C(c3c(C)onc3)=O)CC2C)cnc2cc(O)ccc2c1 50730,C(=O)(C#CC1CCCCO1)N(C(CNC(C1C(C=C(C)C)C1(C)C)=O)C1CC1)C 50731,c1(CCC)cc(C(=O)N(CCC(C)NC(=O)C(=C2CCCCC2)F)C)ccn1 50732,Cc1cccc(C(C)NC(=O)CCC2(C)CN(C(=O)CCC3(C)N=N3)C2)n1 50733,C(C(CO)C(C)(C)C)c1onc(-c2ncc(C)o2)n1 50734,C1(C(N(C)CC2CCCN(C(c3cn(C)nn3)=O)C2)=O)CCCC(F)(F)CC1 50735,C1(C)(C(N2CC(CC)(NC(c3ccc(C(F)(F)F)cn3)=O)C2)=O)COCC1(F)F 50736,S(=O)(=O)(c1nc(N2CCCC(F)C2)ccc1Br)N(C)CCOC(C)(C)C 50737,C1(C(=O)NCCCN(C(c2cscn2)=O)C2CC2)CC2CC(=O)C1O2 50738,N1(C(C(CC)(F)F)=O)CCC(F)(CNC(=O)CC2CCCC(C3CC3)O2)CC1 50739,C12(CN3CCC(c4cn(-c5cncc(C)n5)nn4)C3)CCCC(CC1c1nn[nH]n1)C2 50740,C(=O)(C(F)CC(CC)CC)NC(CC#C)(C)C(=O)NC1CC(C#N)C1 50741,O=C1CCC(C(=O)NC(Cn2cccn2)C(=O)N(CC(F)F)C2CC2)O1 50742,c1(OC)c(F)ccc(F)c1C(=O)NC1CCN(C(c2cc(C)ccn2)=O)CC1F 50743,C1(C(N2CCN(CC(C)NC(C3(C)CC3(C)C)=O)CC2)=O)Cc2cscc2C1 50744,N#CC1CN(Cc2ccc(O)c(O)c2)CC1NC(=O)Cc1cccc(C(N)=O)c1 50745,N1(C(c2ncn(C)n2)C(=O)N2CC(NC(N)=O)C2)CCC(O)C(F)C1 50746,Cc1ccccc1C(C)CC(=O)NC1CCN(C(=O)CCCF)C1 50747,N1(C(C2C(CNC(CN(CCOC)C)=O)CCO2)=O)CC(CO)C1(C)C 50748,C1(NC(C=Cc2scc(C)n2)=O)CC2CC(C1)N(C(=O)CC(C)C(F)(F)F)C2 50749,c1(SC)c(C(=O)OC(=O)CC(c2ccccc2)N(C)C)ncnc1C 50750,CCC(C)(C(=O)NCC(C)C(=O)Nc1conc1C)OC 50751,CC(C)CC(C(=O)NCC1COCCN(C(=O)C(O)Cc2cnc[nH]2)C1)N(C)C 50752,Cc1cn(C)cc1C(=O)N(CC(C)NC(c1cc[nH]c1C)=O)C 50753,c1(C(=O)NC(C2CN(C(c3ccn(CC4CC4)n3)=O)C2)C)cn(C(C)(C)C)nn1 50754,CCC(C)(C(=O)N1CC(NC(=O)C(F)(F)c2cnn(C)c2)C(SC)C1)OC 50755,C1(NC(c2c(CC)scc2)=O)CC(NC(=O)C(C)C)C12CCOCC2 50756,N1(C(CCCOC)=O)CC(N=[N+]=[N-])CC1C(N1CCC(CF)C1)=O 50757,c1(OC)nc(Cl)ccc1CN1CCOC(C(=O)NCc2ccc(Cl)cc2F)C1 50758,c1(C(C(F)(F)F)NC(N(C)Cc2ncc(Br)s2)=O)cccc(F)c1 50759,N1(C(CCOc2ccc(OC)cc2)=O)CC(NC(C2(C)CC2)=O)CC(O)C1 50760,CC(C)CC(F)C(=O)NCC1(C)CCCN(C(c2c(Br)cnn2C)=O)C1 50761,N1(C(c2ncc(F)cn2)=O)CCCC2(CCO2)C1 50762,CC(CC(=O)NCC(C)NC(c1cnc(C(F)(F)F)s1)=O)C1CC1 50763,CCC(C)(COC)C(=O)NCC(C)N(C(=O)CC1CCC=CCC1)C 50764,N1(c2n(CCC#C)c(-c3ccccc3Cl)nn2)CCc2cc(Cl)c(Cl)cc2C1C 50765,N1(C(c2cncc(N=[N+]=[N-])c2)=O)C2CCCC1CN(C(c1coc(CO)c1)=O)C2 50766,CCCCC(CNC(=O)CC1(OCC)CCC1)NC(=O)Cc1cccc(OC)c1 50767,CC1CCN(C(C2(C)SCCCS2)=O)C1c1cn(-c2ccc(Cl)nc2)nn1 50768,CC1CN(C(=O)CCN(CCCO)C(C23CC(C#N)(C2)C3)=O)CC(=O)N1 50769,N1(C(Cc2ncc(C)s2)=O)CC2CC(NC(C3CC4CCC3CC4)=O)CC1C2 50770,N1(C(C(COC)O)=O)CC2CCCC(CNC(=O)CC3CCCC3)C2C1 50771,N1(C(C2CCCN(CC)C2)=O)CCN(C(c2csnc2OC)=O)CC1CN(C)C 50772,N1(CC(=O)NCCC2(C)CC2)CCN(C(=O)Cc2cnoc2)CC1 50773,C(C)(CNC(C1CCCS1)=O)(CC(C)C)NC(CCOc1c(C)cccc1)=O 50774,C1(NC(CCCC#CC)=O)CCC(C)(C)CC1CNC(c1cnc(N)c(N)c1)=O 50775,C(C(=O)NCC1(C)CC1)(C1=CCCCC1)N(C(CS(CC)(=O)=O)C)C 50776,C1(O)(Cc2scc(C)n2)CCN(C(=O)CCn2cccnc2=O)CC1 50777,C1(C(=O)NC(C)Cc2cccnc2)CC2CCC1N2C(C1(C#N)CCCC1)=O 50778,N1(C(C(C)OC(C)=O)=O)CCC(NC(C2CC(O)CN2C(N)=O)=O)C(C)C1 50779,S(=O)(=O)(c1ccc(N)c(NC(C2CCCC(COC)O2)=O)c1)NCC 50780,C1(CC(C)NC(C(COC)O)=O)CCN(C(c2cncc(F)c2)=O)CC1 50781,C=Cc1ccc(C(N2CCC(C)C(NC(=O)CCC(C)(C)F)C2)=O)cc1 50782,c1(C(=O)NC2C(C#N)CN(Cc3nccnc3Cl)C2)c[nH]c2ncccc12 50783,N1(C(c2cc(CC)n(C)n2)=O)CC2(CCNC(=O)C(C)=C(C)C)CCC1C2 50784,C1(CC)CN(C(=O)C(F)=CCCF)CC1NC(c1cc(Cl)ccn1)=O 50785,C1(C(=O)NCCNC(CC(C)F)=O)CC(c2cccc(Br)c2)=NO1 50786,c1(C(N(C(CCNC(C2N(C(C)=O)CCOC2)=O)C)C)=O)nccc2n[nH]cc12 50787,c1(C(=O)NC2CC(C)(COC)N(C(=O)CCSC)C2)cnc(O)c2ccsc12 50788,n1(CCC)nnnc1C(c1cnc(C(=O)OCC)s1)NCCC(C)OC(C)(C)C 50789,Cc1c(C(C)NC2(C)CC2(C)C)cnn1-c1ccc(F)cc1 50790,c1(C(N2CC(C(=O)NCCOCC(F)(F)F)(CC)C2)=O)cc(C)oc1C 50791,C1(C(C)C)N(C(=O)CN2CCOCC2)CC12CC(N)C(O)C2 50792,CC1(C)CN(C(=O)CCCCCC#N)CCN(C(c2cc(C#N)c[nH]2)=O)C1 50793,N1(C(C2(C)COC2)=O)CCC2C1CCCN2C(=O)C(F)(F)c1ccccc1 50794,C1(F)(C(=O)NCC2CC(C#N)C2)CCN(C(=O)Cn2cncn2)C1 50795,CC1COC2(C1)CN(C(C1C3CCCC3CN1C(C1CC(=O)CCO1)=O)=O)C2 50796,C1(C)(NC(C(C)Cc2cnn(C)c2)=O)CCN(C(=O)CC2CCCO2)CC1 50797,Cc1sc(Cl)nc1C(N1CCN(C(C2CCCSC2)=O)CC1)=O 50798,N1(C(C(C)NS(C)(=O)=O)=O)CCC2(NC(c3nc(=O)n(C)[nH]3)=O)CCCCCC12 50799,C1(N(C(CCc2ncc(C)[nH]2)=O)C)CN(C(c2cc3occc3[nH]2)=O)CCC1C 50800,C(C(C)C(F)C(=O)NCCc1cccnc1O)NC(C1(CC#C)CC1)=O 50801,c1(C(=O)NON2CCC(O)CC2)cc(Br)cnc1O.c12cccc(c1)C2=O 50802,c1(C(N2C(C)CN(C(C3CC34CCC4)=O)CCC2)=O)noc2cc(F)ccc12 50803,N1(C(C(C)C)C)CCC(C)(C)C1.C1(=O)CCCn2cc(nn2)C(C)(C)N1 50804,N1(Cc2c(C)noc2)CCC2(NC(c3ccnn3CC3CCC3)=O)CCCC12 50805,C1(C)(OC)CCN(C(C2C=CC(NC(c3cccc(Br)c3F)=O)C2)=O)CC1 50806,N1(C(CC(C)N(C)C)=O)CCCC12CCCN(C(=O)CC1(O)COC(C)(C)C1)C2 50807,c1(OC)ccc(C(=O)N(CCCCNC(=O)C(=O)N(C)C)C)nc1N 50808,c1(C(=O)NC2CN(C(c3cn(CC=C)nc3)=O)CC(C)C2)cc(C)c(=O)n(C)c1 50809,N1(CCC=CCC)CCC(C2CCN(C(C3(C)CCS(=O)(=O)CC3)=O)CC2)C1 50810,N1(C(Cc2cccc(C)c2C)=O)CC2CCN(C(c3cn[nH]c3)=O)C2C1 50811,c1(C(=O)NCCC(C)N(C)C(c2ccnn2C(F)F)=O)cc(C(F)F)ccn1 50812,c1(OC)cscc1C(=O)NCC1CCC1C(N1CCCC1C(C)(C)C)=O 50813,c1(OC)ccc(CC(=O)NC2(C)CCCN(C(c3ccc(F)c(O)c3)=O)C2)cc1C 50814,C(=O)(CCC(CC)CCC)N1CC(NC(CC(=O)NCC)=O)C1 50815,C1(NC(c2cc(C)ncc2)=O)COCCN(C(=O)CNC(=O)NC2CC2)C1 50816,c1(CC(=O)N(C2CC(NC(=O)C=CCO)C2)C)ccc2c(c1)OCO2 50817,C(=O)(C1CCCc2n[nH]cc21)N1CC(CCCNC(CC=CCC)=O)OCC1 50818,CC(C)(CCC(=O)NC1CCN(C(c2ccc(Cl)cc2)=O)C12CCC2)[N+](=O)[O-] 50819,C(=O)(C1=C(Cl)CCC1)N1C(CNC(c2ncccc2Br)=O)CCCC1 50820,c1(CCC)cc(C(N2CCC(N(C(=O)C=CSCc3ccco3)C)C2)=O)ccn1 50821,CC(C)(CC(=O)N1CCC(NC(c2conc2C2CCC2)=O)C1)c1cccs1 50822,C1(O)(CC=C)CCN(C(=O)NCC2CCC2NC(=O)OC(C)(C)C)CC1 50823,c1(CC)cc(C(=O)NC2(CC)CCN(C(C3(C)CC3Br)=O)CC2)ccc1C 50824,Cc1c([N+](=O)[O-])c(C(=O)NCC(C)(CO)NC(=O)CCC(C)(C)C)nn1C 50825,Cc1cc(C(=O)NC2CCCC(CNC(C3COC(=O)O3)=O)C2)n(C2CCC2)n1 50826,CC(O)CCCC(=O)NCC1CCN(C(c2cc(C3CC3)cnc2Cl)=O)C1(C)C 50827,N1(C(c2coc(C(F)F)n2)=O)CCOCC(F)(CNC(C2C3CC4C(C3)C24)=O)C1 50828,CC(C)CCCCC(=O)NCC1CN(C(C2OCCC2C(F)(F)F)=O)CC1C 50829,N1(C(CN(CC(C)(C)C)C)=O)CCC(C(=O)NOC2CCC(F)(F)C2)CC1 50830,N1(C(C(CC)C2CCCCC2)=O)CCC12CCCN(C(=O)CSc1cccs1)C2 50831,C=C(C)c1cccc(NC(C2CCN(C(c3cscn3)=O)C23CCC3)=O)c1 50832,C(=O)(CCCCC(N)=O)NCC1(C)C(C)CN(C(C(C)OCC(C)C)=O)C1 50833,C1(CC)CCCCN1C(=O)C(CCN(C)C)NC(=O)C(CN(C)C)CC 50834,N1(C(C(C2CC2)OC)=O)CCN(C(c2cnc[nH]2)=O)C(C2CCCC2)C1 50835,c1(C(=O)NCCN(C(c2cnn(CCF)c2)=O)CC)cc2cccc(C)c2nn1 50836,C(C(C)C(C)C(=O)N(C)CC1(O)CCN(C(c2cn(C)cn2)=O)CC1)OC 50837,C(=O)(C1=CCC(F)(F)CC1)NC12CCN(C(c3ccc(C=C)cc3)=O)CC1C2 50838,C1(NC(COC2CN(C(CC3C(CN(C)C)C3)=O)C2)=O)CC2(CCC2)C1O 50839,C(=O)(CCCC(C)(C)C)N1CCC(C)CC1CNC(=O)CCc1cccnc1Cl 50840,C1(NC(C(c2ccccc2)N(C)CC)=O)CN(C(=O)CNC(=O)OC)CCC1O 50841,N1(C(C2CC(CC)C2)C(=O)NCC2CCOC2)CC(OC)C2(CCCC2)C1 50842,CC(C)C(O)C(C)C(=O)NCC1CN(C(c2ccn(CCO)c(=O)c2)=O)C1 50843,CC1CN(C(C2(O)CCCC2)=O)CCC1CNC(c1cc(N(C)C)ccn1)=O 50844,n1(CC(=O)OC(C)(C)C)nccc1-c1cn(CCNC(c2cnc(Cl)[nH]2)=O)nn1 50845,C(=O)(CS(=O)(=O)C1CC1)NC1C2(CN(C(c3c(C)cc(O)nc3)=O)C2)CC1 50846,c1(C(N2CCN(C(c3occ(OC)c(=O)c3)=O)C(C)C2)=O)c(C)ccc(F)c1N 50847,C1(CCOC)(NC(=O)CC2(O)CCCCC2)CCN(C(C2CCCC2(C)C)=O)C1 50848,C=C1CCN(C(C2CCN2C(C)(C)C)=O)C(C(=O)N(C(CCO)C(F)F)C)C1 50849,N1(C(=O)Cn2cc(C3CCOCC3)nn2)CCCC2(C1)C(O)CC2O 50850,N1(C(c2c(CC)ncc(Br)c2)=O)CC2CCC(C1)N(C(=O)C1=CCC1)C2 50851,Cc1cc(F)c(N)cc1C(N1CCCN(C(c2cscc2C(F)F)=O)CC1C)=O 50852,N1(C(CNC(C)=O)=O)C(CC(N2CCC2C2CCCCC2)=O)C2CCCC12 50853,C1(NC(C2(OC)CCN(C(C3CC(CC)(CC)C3)=O)C2)=O)CCC(C)(C)CC1 50854,N1(C(CCC=CC(C)C)=O)CC(CNC(C2CCC(CO)CC2)=O)C(C)C1 50855,CC(C(=O)NC1C2CN(C(=O)CCc3cccc(C(F)(F)F)c3)CC12)C(C)(F)F 50856,c1(C(=O)NCC2CC(NC(=O)C(=Cc3cccnc3)F)C2)ccc2nsnc2c1 50857,CCC(C)C(O)CC(=O)NC1C2CC3C1C3C2C(N1CCC(C)(O)CC1)=O 50858,C1(CC)CN(C(=O)CN2CCC(=O)NC2=O)CCN1C(c1cnn(C)c1Cl)=O 50859,c1(NC(c2cc(CNC(C(CC)C)=O)ncc2)=O)cnc2cc(Br)ccc2c1 50860,c1(OC)ncccc1C(N1CCCC(CC(=O)NC(C)(C)CN2CCCC2)C1)=O 50861,CCC(CC)C(=O)NC(C)CN(C)C(C1CC(=O)N(C2CC2)C1)=O 50862,C(CC(=O)N1CCn2ccnc21)(C(F)(F)F)NC(C=CC(CC)C)=O 50863,N1(C(CCN(C)CCO)=O)CC2C(CC(=O)NCC3(C)CC=CCC3)C2C1 50864,c1(C(N2CC(CNC(C3CC(OC)C3)=O)C(O)C2)=O)cc2cccnn2n1 50865,CCCCC(O)CC(=O)N1CC(CC(=O)NC23CCC(CC2O)C3)C(C)C1 50866,CCCC(CCCNC(c1cnc(OC)cn1)=O)NC(c1cnc(C)o1)=O 50867,Cc1ccc(C(N2CC(C(N3CCCC3C(F)(F)F)=O)C2)=O)c(O)c1 50868,C1(C(N2CC(N(C)C3CC3)C2)=O)CC(=O)N(C2CCNCC2)C1 50869,C1(NC(C(CC)N(CC)CC)=O)CCN(C(c2cc(C)cs2)=O)C(C)C1 50870,c1(C(=O)NC2CCN(C3CN(C(C(CC)OC)=O)C3)CC2)cc(N)c(O)c(F)c1 50871,CC1CCC(CO)CN1C(C1(NC(c2cnn(C)n2)=O)CC1)=O 50872,C(=O)(C(O)CCCNC(c1ccccc1)=O)N(CC)Cc1ccoc1 50873,CC1(C)CCCC(C(=O)NC(CNC(=O)CCc2ncco2)C2CC2)C1 50874,c1(C(=O)NC2(CC=C)CC=CC2)ccc(CNC(=O)C(CC)N(C)C)nc1 50875,C=CCC(C(=O)NCCCN(C(C1CCC(C)(C)O1)=O)C(C)C)NC(C)=O 50876,C1(C(=O)NC(C)CCN(C(=O)Cc2ccsc2Cl)C)CCC(C)(C)OC1 50877,CCCC(CCC)C(=O)NCC1CC2(CC2)CN1C(c1[nH]nc(OC)c1Cl)=O 50878,Cc1c(C(=O)NC2(C#N)CCN(C(c3ccon3)=O)C2)cncc1Br 50879,Cc1c(C(N2CCC(NC(=O)C=CC3CC3)C23CC3)=O)sc(Cl)c1Cl 50880,C1(C(=O)NCC(C(C)C)(C)F)CCCC(NC(C2CCCSC2C)=O)CC1 50881,N1(C(CCc2cc(C)on2)=O)CC(N(C(=O)Cc2nn(C)cc2Cl)C)C(F)C1 50882,C(=O)(C(CCF)NC(=O)CC#N)N(CC(O)CO)C 50883,N1(C(C(C)OCCC(C)C)=O)CC(CO)C2(C1)CN(c1cc(C3CC3)ncn1)C2 50884,N1(C(CCCSC)=O)CC(NC(=O)C(C)(O)C2CCC2)CC1C 50885,C1(C(N(C(C)C)CCNC(C2(CO)CC(F)(F)C2)=O)=O)CCCCCN1C 50886,C(=O)(C(O)C1=CCCCC1)N(CCCNC(=O)Cc1csnn1)CC 50887,Cc1cc(Cl)nc(Cl)c1NC(C1CC(O)CCN1Cc1cc(F)c(Cl)cc1Cl)=O 50888,C1(C(N2CC(NC(CSc3ccc(C)cc3)=O)C2)=O)CC2CCC(C1)C2(F)F 50889,Cc1cc(C)c(C(N2CC=C(CNC(=O)CC3CCOC3(C)C)CC2)=O)cc1N 50890,N1(C(C2(C)C=CCC2)=O)CCN(C(c2onc3ccccc23)=O)CC(O)C1 50891,C(=O)(CC1CCCc2ccccc21)N(CCNC(C(CC#C)C)=O)C1CC1 50892,c1(C(N2CCC(NC(CC(CC)C3CC3)=O)C2C)=O)cc2n(n1)CCNS2(=O)=O 50893,CC(C)CC(CN(C)C)N=c1nc2c(ncn2C)c(NCc2c[nH]c(=N)s2)[nH]1 50894,c1(CC(=O)NCC(C(=O)NC(CCC)C)N(C)C)ncccc1C 50895,c1(SCC)nc(C(=O)NC2CC(C)N(C(=O)CCSC3CCCC3)C2)cc(=N)[nH]1 50896,CS(=O)(=O)CCC(=O)NCCCC1CCCN1C(=O)CCc1cncc(F)c1 50897,N1(C(C(C)N(CC)CC)=O)CC(NC(C2CN(C(=O)N(C)C)C2)=O)C2(CCC2)C1 50898,c1(C(C)O)ccc(C(=O)N(C2CCC(NC(=O)CC3CCCCO3)CC2)C)cc1 50899,C1(C(=O)NC2(CC=C)CN(c3nc4ccccc4o3)C2)CCc2nncn2C1 50900,c1(OC)ccc(CNC(n2cc(CNc3nc(C(C)(C)C)c(Br)s3)nn2)C)cc1 50901,Cc1c(CN(C(=O)CCCCNC(c2ccncc2)=O)C)cnn1C 50902,C#CCCC(=O)N(CCC(=O)NC1CCOC1=O)CCCO 50903,Cc1ccc(NC(C2CCCC2CNC(c2ccc(CO)s2)=O)=O)c(C)n1 50904,C1(CCOC)(C(=O)NC2CC(O)(CNC(=O)C(C)C3CCC3)C2)CCCC1 50905,C12(C(=O)N(CCC3(NC(c4cc(CCC)on4)=O)CCC3)CC)CCCN1CCC2 50906,C(CCC(C)C(=O)N(CCCCC(=O)N(C)Cc1ocnc1C)C)OC 50907,Cc1c(Cl)sc(Cl)c1C(=O)N(CC(C)NC(c1cc(C(N)=O)c[nH]1)=O)C 50908,Cc1cc(C(=O)NC2(C)CC(C(=O)NCC3CC(O)CN3C)C2)cnc1O 50909,N1(C(C(C)(C)CCl)=O)CCOC2(CCN(C(=O)C(O)O)C2)C1 50910,Cc1cc(C(F)(F)F)nn1CC(=O)NCCC1CCN(C(c2cncs2)=O)C1 50911,N1(C(C(C)NC(C2CCCC2)=O)=O)CC(C)(C)CC1C(=O)NCC1(C)CC1(F)Cl 50912,C1(CC)C(C(N2CCC2(C)CCO)=O)CCN1C(=O)Cc1ccc(C)o1 50913,C1(CNC(C2(CC=C)CCCC2)=O)CN(C(=O)Cc2ccnc(O)c2)CCN1C 50914,C1(C2CCCO2)(C(=O)NCC2CC(C)N(C(c3ccncc3F)=O)C2)CCCO1 50915,C1(NCc2c(C)ncs2)CCN(C(=O)CC2(O)CCCC2)CC1C 50916,C(=O)(CC(=O)NCCC1(C(=O)NCCC(O)CO)CCCC1)N(C)C 50917,C(=O)(CC(O)C(=O)N1CC2CC2(CNC(c2coc(Cl)c2)=O)C1)OC(C)(C)C 50918,Cc1cnc(C(=O)NC2CC(F)CN(C(=O)C3=CCCCC3)C2)cc1C 50919,N1(C(CCC(C)(C)NC(=O)C=Cc2ccco2)=O)Cc2ccccc2C1 50920,C1(CNC(CN(C)C(N)=O)=O)CC(F)(F)CN1C(c1cccnn1)=O 50921,c1(N(C(C)=O)C)ccc2c(c1)CN(C(=O)C(=O)N(CCCN(CC(C)C)C)C)C2 50922,C1(NC(C(C)=C2CCC2)=O)CN(C(c2nn(C)nc2C(F)(F)F)=O)CCC1CO 50923,C(=O)(CCCCCC(C)O)N1CCC(OCCNC(C(CC(C)C)O)=O)CC1 50924,C1(C(=O)NCCCCNC(c2cn(C)nc2O)=O)CS(=O)(=O)CC1C(F)(F)F 50925,C1(C#N)(CNC(C2N(C(COC3CN(C(C)=O)C3)=O)CCCC2)=O)CCCOC1 50926,CN1CC(C(N2CCC(F)(C(=O)NCCC(F)=C(F)F)C2)=O)CC1=O 50927,C1(NC(c2nc(C)n(C)c2)=O)CCCC(C(=O)N(CC(Cl)Cl)C)CC1 50928,CC1CN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CCC1NC(=O)CC12CCC(CC1)CC2 50929,c1(CC(=O)NC2CCC2CNC(c2ccncc2)=O)ccc(F)cc1C(F)(F)F 50930,c1(CC)conc1CC(=O)NC(C(=O)NC1CN(CC2CC2)C1)c1cccs1 50931,CCC(CC)CC(F)C(=O)NCc1cc(C(=O)N(CC(O)C(F)(F)F)C)cs1 50932,c1(C(=O)NC(c2ccc(Br)s2)n2cncn2)cnc(O)c2ccsc12 50933,C12CCC(CC1)NC2=O.C(=O)(C(C)=O)N(C1CCCC1)CC 50934,N1(C(CCc2c(C)noc2Cl)=O)CCN(C(c2nnc(O)nc2O)=O)C(C)C1C 50935,C1(NC(CC(C2CC2)NC(C)=O)=O)CCCC(CNC(=O)C=C(C)C(C)(C)C)C1 50936,C(CC(C)C(=O)N(CCNC(c1cnc(O)o1)=O)C1CC1)=CCC 50937,C1(CCCC)CN(C(=O)C(CC(C)C)NC(N)=O)CCN1C(=O)C=CC(F)(F)F 50938,CC(CCNC(=O)C(C)Cc1ccco1)CCNC(=O)CCc1cn[nH]c1 50939,N1(C(c2ccc(CSCCC)o2)=O)CC2=C(C1)CN(C(=O)C=C1CCOCC1)C2 50940,C1(C(=O)OC(C(C)C)c2cccs2)CCCCCN1C(=O)Oc1ccccc1 50941,C(C)(CN=c1ccn2ncc(S(=O)(=O)NCc3cc4ncccc4o3)c2[nH]1)OC 50942,c1(OC)cnc(C(N2CCCC(NC(=O)CC3CN(C)C3)CC2)=O)c(OC)n1 50943,C1(NC(COCCC)=O)CC2(N(C)C(C3CCN3CC)=O)COC1C2 50944,C(C)(C(=O)N(CCCCC(=O)NC1CC(=O)N(C2CC2)C1)C)(C(C)C)OC 50945,C#Cc1cc(C(=O)NC2CC(NC(=O)CCc3ccccc3C#N)C2)cc(F)c1 50946,CCC1=NOC(CC(=O)NC(c2cc(C(=O)NC3CCC3CN(C)C)no2)C)C1 50947,c1(C(N2CC(CCCCNC(C3(O)CC4CCC3C4)=O)C2)=O)cc2sccc2s1 50948,C1(OC)CC(OC)C12CCN(C(c1ccc(-n3cnc([N+](=O)[O-])n3)cc1)=O)CC2 50949,c1(OC)cc(C(=O)Nc2ncc(-c3cccc(C)n3)cc2C)cc(Cl)n1 50950,CC1(NC(=O)CC2CC(F)C2)CCC(NC(c2ncoc2C(C)(C)C)=O)CC1 50951,CC1CC(CNC(=O)CCCc2cnn[nH]2)CCN1C(=O)CC1CCCO1 50952,c1(C(=O)NOCC2CC=CCC2)coc2c1CN(C(C1CC=CC1)=O)C2 50953,c1(C(=O)NCC2CC2NC(C2CCC2)=O)ccc2nc(O)nc(O)c2c1 50954,N1(C(C(COC)OC)=O)CCC(CCC(C)(C)NC(c2cnc(S)[nH]2)=O)CC1 50955,C1(NC(NC(COC)C)=NCCCNS(C)(=O)=O)CCS(=O)(=O)C(C)(C)C1 50956,N1(C(CCOC)=O)CCCCC(N(C(=O)CC(C(C)C)c2ccccc2)C)C1 50957,Cc1cc(C(=O)NCC(C)CNC(=O)CCc2cccc(O)n2)c2n[nH]cc2c1 50958,Cc1c(O)ccc(CNC(C2(Cc3coc(C#N)c3)CCC2)=O)c1O 50959,O=C(CC(C(F)(F)F)NC(=O)C(c1ccccc1)OCC1(C2CCC2)CC1)OC 50960,N1(C(CC(C=C)(C)C)=O)CCN(C(=O)CCCN(C)C)C(C)C1C 50961,C(=O)(C(C(C)CC)NC(c1ccc(SC)o1)=O)NCCSCCC=C 50962,c1(CC)c(C(=O)NC(CNC(=O)COCC2CCCO2)CC2CC2)cccc1F 50963,CN1CCC(C(=O)NCc2nc(CNC(=O)C3=CCCC3)cs2)S1(=O)=O 50964,Cc1cnc(NCC2CCCCC2NC(C2(O)CCOCC2)=O)nc1O 50965,Cc1cc2ccccc2cc1C(=O)NCC(CNC(c1cccnc1)=O)CO 50966,N1(C(COCc2cccc(C)c2)=O)CCC(NC(=O)CCOC2CC2)C(O)C1 50967,N1(C(c2n[nH]c(C)c2Cl)=O)CCC(O)(CN(C)C(C2CCC(C(N)=O)C2)=O)CC1 50968,CC(C)C(C)C(CNC(=O)C=Cc1ccoc1)NC(=O)CCCCCN(C)C 50969,c1(C(=O)NCC2CC(F)(CNC(CCC#C)=O)C2)cc([N+](=O)[O-])n[nH]1 50970,CC(C)C(C(=O)NC1CCN(c2ccnc(Cl)n2)CC1)c1ccc(-c2nn[nH]n2)cc1 50971,C1(NC(COc2cc(C)on2)=O)CC2CN(C(=O)C3=CCCO3)CC12 50972,C1(C(N2C(CNC(CC3CC(=C)C3)=O)CC(C(F)(F)F)C2)=O)CCCCC(=O)N1 50973,C12(COC)CC(CNC(c3cnn(C)c3)=O)(CN1C(=O)CSC1CCCO1)C2 50974,C1(C2CCOCC2)(C(=O)NC2CC(NC(C(C(C)C)OCC(C)C)=O)CC2O)CC1 50975,C(=O)(C(O)CC(C)(C)C)NC1CCC(CNC(c2cc(C)[nH]c2)=O)C1 50976,C=C1CCN(C(c2nonc2N)=O)C(C(=O)Nc2cnc(F)nc2)C1 50977,C(=O)(CC1=CCCC1)OC(C(C(=O)OCC)=O)C 50978,c1(C(N2CCC(N(C(c3cscc3OC)=O)CC)C2)=O)oc(C)nc1C 50979,CS(=O)(=O)C(CNC(=O)Cc1cccc(Cl)c1)CNC(c1cc(C#N)cs1)=O 50980,c1(OC)cccc(NC(c2sccc2CNC(=O)N(C(C)C(=O)OC)C)=O)c1 50981,N1(C(C(C)=C2CCC2)=O)CCC(NC(c2cc(C(C)(F)F)ccn2)=O)CC1C 50982,C(C(=O)N1CCCN1)NC(C1CC2CCC1C2)=O 50983,CC1CCN(C(=O)CCc2cncnc2)CCN1C(c1cccc(N(C)C)n1)=O 50984,N1(C(c2ccc(CC)o2)=O)CCC(O)(C2CCN(C(c3cnns3)=O)CC2)C1 50985,N1(C(C2CN(C(CCNC(=O)CO)=O)CC23CCC3)=O)CC2CCC(O)C(O)C12 50986,C(C(C)(CC(C)C)NC(c1csnn1)=O)NC(c1c(C)cc(C(F)(F)F)s1)=O 50987,C1(CNC(C2(C)CCCC2)=O)CCN(C(=O)Cc2ccc(O)c(Cl)c2)CC1(F)F 50988,C1(CNC(c2ccc(C(C)C)cn2)=O)CCC2(CCC2)C1NC(=O)C=C1CCC1 50989,CC(C)CC(CNC=O)CC(=O)NC1CCCN(C(=O)C=CCN2CCCC2)C1 50990,N1(C(c2c(C)nc[nH]2)=O)CC(C)C(NC(=O)C=CCO)C(C)C1 50991,c1(CC)ccc(NC(=O)COCC(C)(C)C)cc1F.N12CCCC1C1(CC1)C2=O 50992,C(=O)(C1COc2ccc(Cl)cc21)N1CCC(CN(C)C(C2CC3CC3C2)=O)C1 50993,c1(C(N2C(C)(CNC(c3cnc(SC)[nH]3)=O)CCC2)=O)cccc(N)c1O 50994,c1(C(N2CC3(CCN3C(=O)C=CCF)C2)=O)cc(N2CCC2)cc(Br)c1 50995,CC(C)C(F)C(=O)NCCC1CCC(NC(=O)CC2CC=CC2)C1 50996,N1(C(c2cn(C)c(=O)cn2)=O)CCC(NC(=O)CNS(N)(=O)=O)CC(O)C1 50997,C1(N(C(=O)CSc2cccs2)C)CCCC(NC(c2c[nH]cc2Br)=O)C1 50998,C1(NC(C=C(COC)C)=O)CN(C(c2cc(CC(C)C)c[nH]2)=O)CC1N=[N+]=[N-] 50999,c1(C(=O)NCC(C(C)C)NC(C2COCCO2)=O)sc(N2CCOCC2)nc1Cl 51000,c1(OCC(=O)N(C2CCN(C(C34CC(O)C3C4)=O)C2)CC)cc(Cl)ccc1Cl 51001,C=Cc1ccc(C(=O)NCC2(O)CCN(C(=O)CSc3nncs3)C2)cc1 51002,c1(C(=O)NC23CCN(C(=O)CN4CCOCC4)CC2C3)ccc(Cl)cc1Cl 51003,N1(Cc2cnc(OCC)nc2)CC2(CCN(S(=O)(=O)c3cnn(C)c3)C2)C1 51004,c1(OC)cc(CN2CCNCC2)ccc1I.c12ccc(nc1)[nH]2 51005,c1(C(=O)NC2(C)CN(C(C3(CC(C)C)CCC3)=O)C2)nn(C)c2ccccc12 51006,c1(C(N(CCCN(C(c2scc(OC)c2OC)=O)C)C)=O)cnc2c[nH]nc2c1 51007,Cc1ccc(-c2cn(C3CCN(C(=O)CC(=O)N(C)C)CC3)nn2)cc1N 51008,NS(=O)(=O)c1ccc(SCCN(C2CC2(F)F)CCCCC(F)(F)F)o1 51009,C1(C(=O)NC2CN(C(=O)CCCc3cccc(F)c3)C2)(COC)CCCCC1 51010,c1(C(=O)NCCc2ccc3c(c2)COCC3)nc(Br)c2c(F)cccn12 51011,C1(C(=O)NCCC(=O)NCC)CC2(CCN1C(c1cn(C)nn1)=O)CC2 51012,C1(CC(=O)NC(C=CC(=O)NCCOCCOCC)C)CCCCCC1 51013,c1(-c2cn(C3CC(NC(c4cc(CC)[nH]n4)=O)C3)nn2)cc([N+](=O)[O-])ccc1OC 51014,O=C1CN(C(c2ccc(Cl)cc2C(F)(F)F)=O)CCN1Cc1ccco1 51015,N1(C(COC(C)=O)=O)CCOCCC1C(=O)N(C)CC1CCN(C)CC1 51016,CCCC(C(=O)OC)C(=O)NC1COCCC1NC(c1ccc2n[nH]cc2n1)=O 51017,c1(C(N2CCCC(NC(CCOCCOC)=O)C2C)=O)cc2c(s1)CCC(C)C2 51018,CCCCC(O)CC(=O)NC(CC(F)F)C(=O)N1CCOC2CC12 51019,N1(C(c2c(CC)csc2)=O)C(C(=O)NCCOC(C)=O)CCC12CC2 51020,C1(CNC(c2cc(C3CCC3)no2)=O)CN(C(C2(CO)CCCC2)=O)CC1(F)F 51021,c1(OCCC)ccc(Cl)cc1NC(N1CCC(C)C1(C)C)=O 51022,CC1CN(C(CC(C)(C)C)C(=O)NCC2CCOCC2)CC(C)(C)C1 51023,c12ccccc1NC(=O)CO2.c1(CC)n[nH]cc1C(C)C.N12CCC(C1)C2 51024,C1(NC(CCc2cc(C)no2)=O)(CO)CCCN(C(C2CC23CC(C)(C)C3)=O)C1 51025,N#CC1(C(=O)NCCc2ccc(Br)cn2)CC12CCCC2 51026,N1(C(=O)OCCCC)CCN(C(C)C(=O)NC2CC(n3cccn3)C2)CC1 51027,c1(C(C(=O)NCCCF)N(CCC#N)CC)ncc(Cl)cc1Cl 51028,N1(C(c2ncn(CC)c2)=O)CCN(C(=O)C(F)(F)C(F)F)CC1CO 51029,N1(C(c2n(C)cnc2)=O)CCCC2(CCC(NC(c3coc(Cl)n3)=O)C2)C1 51030,C=C(C)CC(C(=O)NC(CNC(=O)CN1CCOCC1=O)CCC)NC(C)=O 51031,CC1CN(C(=O)C(C)Cn2cccn2)CC(C(=O)NC(C2CCCO2)(C)C)O1 51032,C1(CC#C)CN(C(C2(N(C)C(=O)OC(C)(C)C)CCOCC2)=O)CCO1 51033,C(CC(=O)N1CC(F)(F)C1C1CC1)(C(F)F)NC(c1n(C)c(S)nn1)=O 51034,CCCS(=O)(=O)CC(=O)NC1CN(C(c2ccc(O)nc2)=O)CC1CO 51035,c1(OC)ccc(C(N2CC(NC(C3CC(OC(F)F)C3)=O)C(O)C2)=O)cc1 51036,c1(C(=O)NCC(F)CNC(C2CC(F)C(=O)N2)=O)cc2cccc(O)c2[nH]1 51037,c1(N2CC3C(NC(c4ccc(S)cc4)=O)C3C2)ncnn2cccc12 51038,N1(C(c2c(CC)con2)=O)CCOCC1CC(=O)NC1CCOC(C)C1 51039,C=C1CC(C)C1.C(C(=O)NCC(C)(C)O)(c1cccs1)N(CCCO)C(C)C 51040,CCCS(=N)(=O)c1cccc(CNc2cccc(C#N)c2F)c1 51041,C=CC(CC)CC(=O)NCCCOCCC(=O)NC12CCN(CC1)C2 51042,C=C(C)CCCC(=O)N1CC=CC(NC(C2(Cc3cccc(F)c3)CC2)=O)C1 51043,C1(C(N2C(C)CCC(NC(CN(CCOC)C)=O)C2)=O)CC2(C1)CC1(CCC1)C2 51044,CC1(C)CN(C(C2(S(C)(=O)=O)CC2)=O)CC(C)(C)C1NC(=O)C(F)CC1CCC1 51045,c1(C(N(CC(CNC(CCNS(CC)(=O)=O)=O)C)C)=O)[nH]c(C)cc1C 51046,N1(C(C(C#C)(C)C)=O)CCN(C(=O)CC2CCN(C)C2)C(CC(C)(C)C)C1 51047,C(C(COC)C(=O)N1CC(C)(CCC(=O)NC2CC(OC)C2(C)C)C1)OC 51048,C(C(=O)NCCCCC(=O)NC(C12CC(CO1)C2)C)(C(C)C)OC 51049,Cc1cc(C(N2CCC(NC(=O)CSc3n[nH]c(O)n3)C23CC3)=O)c(N)c(Cl)n1 51050,CC1CC(NC(=O)CC(C)(C)C2CC2)CN1c1nnc(C2CC2)s1 51051,c1(CC)ccc(C(=O)N(CC(C)NC(=O)Cc2ccsn2)CC)cc1 51052,C1(O)(CC(=O)NC2C(C(=O)NCC(C(=O)NC)O)CCC2)CCCCC1 51053,CC1(C)C(NC(=O)C(CC2CCCC2)CN)C(C)(C)C1O 51054,C=CC(CC(=O)N(c1ccccn1)CCNC(=O)COCC)c1ccccc1 51055,Cc1ccnn1C(C)C(=O)NC1CCCCC1.C12CC(C1)CNC2=O 51056,c1cn2c(n1)C(Nc1cc(NCC3=CCCC3)ncn1)CCC2 51057,N1(C(c2cn(C3CC3)nn2)=O)CCN(C(=O)CN2CCCS2(=O)=O)C2CCC12 51058,C(CC)(C(=O)NC(C1CN(C(=O)CC2CC2C)C1)C)=CC 51059,N1(C(C=CC(C)=O)=O)CCN(C(C2(CO)CCOCC2)=O)C(C)C1 51060,c1(OC)cccc2c1CCCC2NC(=O)C(=O)NCC(c1ccc(F)cc1)(F)F 51061,c1(NC2CC(NC(C3C(OCC)C3C)=O)C2)ncc(C(N)=O)cc1Cl 51062,c1(C(=O)NCC(CC(C)C)NC(CC2CC(CC)C2)=O)c(F)cncc1Br 51063,c1(C(=O)NCC2CCN(C(C(CC=CC)C)=O)C(C)C2)cn2ccccc2n1 51064,c1(C(c2ccccc2)NC(CC)C2CC2)ccccc1Br 51065,C1(C(C)C)CN(C(C2CNC(=O)C2)=O)CCN1C(=O)CCc1cnc[nH]1 51066,c1(CCCC(=O)NCC2CC(OC)CN2C(=O)C(F)F)c(F)cccc1F 51067,N1(C(COCCC)=O)CCN(C(=O)CCc2cc(C)n(C)n2)CC2(CC2)C1 51068,CCCCCCC(CC)(c1nnnn1CCOC)NCc1ccc([N+](=O)[O-])o1 51069,N1(C(CSCC)=O)CCC(N(C(c2cocc2C)=O)Cc2cccnc2)CC1 51070,C(Nn1cnc2ccccc12)c1onc(-c2cccc(C(N)=O)c2)n1 51071,c1(C(N2C(C(=O)Nc3nccs3)CC(F)C2)=O)c(F)cccc1F 51072,C1(C(=O)NCC2(C)CCN(C(c3cnco3)=O)C2)(CC)CNC(=O)C1 51073,c1(C(=O)NC2CN(C(c3nc(C)nn3C)=O)CC2C)cnn2ccn(C)c12 51074,Cc1cccc(CC(=O)NCCCCNC(=O)C(N2CCC(C)C2)=O)c1F 51075,C#CC(CCC)NC(C1CCC1CNC(=O)C=Cc1cocn1)=O 51076,Cn1cc(S(N)(=O)=O)c(C(=O)NCC(C)(CO)NC(C2CCS(=O)(=O)N2)=O)n1 51077,CC(C)(C)C(CO)C(=O)N1CC2CC1CN2C(=O)CCCC1CCCO1 51078,CCCC(C)(CC)C(=O)NCC(C1CCC1)NC(c1cnc(OCC)c(Cl)c1)=O 51079,N1(Cc2nnc(CC)s2)C2CCC1CN(C(c1cc(C)[nH]n1)=O)CC2 51080,Cc1c(C2(C(=O)NCCC(C)NC(C3(O)CC(F)(F)C3)=O)CC2)cccc1F 51081,N1(C(CN(C(=O)CSCCN(C)C)CC)=O)CC(=O)NCC1C 51082,N1(C(CC(=C)C)=O)CCN(C(=O)COc2ccccc2C#N)CC1C1CC1 51083,C1(C(N2CCN(CCN(C(C(CC)=CC)=O)C)CC2)=O)CCC(C)(C)CC1 51084,c1(OCC)ccc2c(c1)CCN(C(c1cccc(O)c1)C(=O)NCCC1CC1)C2 51085,C=CCC(C)(O)C(=O)NC1CCC1C(=O)N(C1CC(C)(C)C1)C 51086,CCCC(CCC)C(=O)NC(C)C(N1CCC(C)(F)C1)=O 51087,c1(CC(CNC(=O)NCc2ccc(OC)cc2)CO)c(OC)cccc1C 51088,c1(CC)oc(C(=O)NC2CC(CNC(C3CC34CCC4)=O)C2)cc1C 51089,C(C)(C)(CCCF)NC(C(C1(C)CC1)NC(C1CC(=C2CCC2)C1)=O)=O 51090,C1(CC)CC(C(=O)N(C2CCC2C)C)CCN1C(c1nn(C)cc1Cl)=O 51091,N1(C(C2=NOC(C)C2)=O)CCC(C2(NC(=O)C=Cc3ncc[nH]3)CC2)C1 51092,C1(OC)CN(C)CC1NC(=O)C(C1CCCC1)NC(C1CC1(C)C(F)F)=O 51093,c1(C(C(=O)NCCOCC)N(CC(C2CCCO2)OC)C)ccc(F)c(Br)n1 51094,C(=O)(CCCC(C)=O)NCC(CC=C)NC(=O)C=Cc1ccco1 51095,CC1(C)CCCC(C(=O)NCC2(O)CN(C(C3C4CCCCC34)=O)C2)C1 51096,C1(C(N2CC(N(C)C3CC3)C2)=O)(COC)C=CCN1C(C1C2CCCOC12)=O 51097,C(=O)(C(CC)C(C)C)N1CC(C=C)(C(=O)NC(CO)CC=CC)C1 51098,N1(C(C(COC(C)=O)C)=O)CCC(C(=O)NCCNC(=O)C(C)C)CC1(C)C 51099,N1(C(C(C)(C)OC)=O)CCN(C(=O)CCCNC(C2CCCO2)=O)C(CCO)C1 51100,CCCC(C(=O)N(CCCN(C(=O)CCc1cc(C)sc1C)C)C)NC(N)=O 51101,Cc1nn(C)c2[nH]c(=NCC=CCNC(C3CCSC3)=O)c(C#N)cc12 51102,CC1COCCC1NC(=O)C(=O)N(CCCC1CC2CCC1C2)C 51103,CN1CCC(CCNC(=O)CC2C=CC(NC(c3cncn3C)=O)C2)C1 51104,Cc1cc(CC(N2CC(NC(=O)C=Cc3cc[nH]c3)C(C(F)F)C2)=O)ccn1 51105,C12(C(=O)NCC3C(C)(C)N(C(C4CCCOCC4)=O)CC3)CCC(N=[N+]=[N-])C1C2 51106,Cn1nnc2cc(C(N3CCC(CCNC(C4CCCC(F)(F)C4)=O)C3)=O)sc12 51107,C1(NC(c2c(COC)noc2)=O)C2CCN(C(C3CC4(CC4)C3)=O)CC12 51108,c1(SCC)ccc(C(=O)NCC(CCCC)NC(C2CSCCS2)=O)cn1 51109,C1(C(N(CCCNC(C(n2ccc(C)n2)(C)C)=O)C2CC2)=O)C(Cl)(Cl)C12CC2 51110,N1(C(C=COCC)=O)CC(NC(=O)CCC2CCCCN2C)CC(C)(C)C1 51111,C(=O)(CCCCCCC(=O)OC)NC1CN(C(CC=CC)=O)CC(F)C1 51112,Cc1ncc(C(N2CCN(C(C3(C(F)(F)F)CC4(CCC4)C3)=O)CC2)=O)c(=N)[nH]1 51113,Cc1cccc2c1OC(C(=O)NC1CN(C(c3ccon3)=O)CC1C)C2 51114,C1(C(N(CCNC(c2ccc(OC(C)C)nc2)=O)CC)=O)CCC(F)(F)C1O 51115,C(CN=C(NCC(F)F)NCC1CCC(=O)N1)c1cccc(C(=O)NC)c1 51116,C1(NC(Cc2c(C)ccc(F)c2)=O)CCCC12CN(C(C1NC(=O)C3CC13)=O)C2 51117,CC(CC(=O)N1CCN(C(=O)C=C2CCOCC2)CC1)C(C)(C)C 51118,c1(C(=O)NC2C3(CC(NC(C(c4cnccn4)C)=O)C3)C2)cccn2nncc12 51119,NS(=O)(=O)c1n[nH]cc1C(N1CC2CCC1C2NC(=O)Cn1cnccc1=O)=O 51120,CCCC(CCC)C(=O)NC(C)CN(C)C(c1onc(OC)c1Br)=O 51121,c1(C(=O)NC2CN(C(c3ccc(C(C)C)o3)=O)C3C2C3)cc(F)cc(F)c1 51122,c1(OC)ccncc1C(=O)NCC1(NC(=O)CCc2cscn2)CCOC1 51123,c1(C(=O)NC(CNC(C2C(C)CC2)=O)(C)C)ccc(C(F)F)cc1Cl 51124,C(CN=c1ccc(Br)c(S(=O)(=O)N(CC(C)(C)C)C)[nH]1)c1cc(SCC)ncc1 51125,Cc1ccc(C(C)NC(C2CC(O)(CNC(=O)OC(C)(C)C)C2)=O)c(Cl)c1.C 51126,CC1CN(C(C2C(F)(F)C23CCC3)=O)CCC1CNC(=O)CC1OCCC1(C)C 51127,C1(OC)CCC(C(=O)NC(C)CNC(c2sccc2C(C)(C)C)=O)CC1 51128,C(C)(C)(C(=O)NCCCC1(NC(=O)CC2CC(F)C2)CC1)OCC 51129,C1(C(=O)NC(c2n(C)ncc2)C(=O)NC2CC(O)C2)C2CC3C(C2=O)C13 51130,CC1OCCC1C(=O)NCCC1(NC(=O)COCC2CCC2)CCC1 51131,N1(C(CN2CCC(C)C2)=O)CC2CCC1CN2C(=O)C(C1CCCCC1)O 51132,CCCCCC(=O)NC1CN(C(c2cnn(C(C)C)n2)=O)C2CC12 51133,CC1CN(C(=O)C(C)(F)c2ccon2)CC1CNC(c1ccn(C)n1)=O 51134,c1(C(C(=O)NCC=C)N(C2CCN(CC)C2)CC)cnn(C)c1Br 51135,C(=O)(C1CCc2c[nH]nc21)N1CCC(C(C)NC(c2cnsc2)=O)CC1 51136,C1(CC(=O)NCCc2nc(=N)[nH][nH]2)NC2CCCC12 51137,C#CCC(CC#C)C(=O)NCC(C1CCC1)NC(=O)COCc1ccccc1C 51138,CC(C(=O)N1CC(NC(C2CNC(=O)N2)=O)C(C)C1)C(C)c1ccccc1 51139,c1(CCCC)ccc(C(c2nnnn2C)NCCc2csc(C)n2)cc1 51140,C(C(=O)NCC(C1CC1)NC(=O)Cc1c(Cl)cnn1C)(C(C)C)n1cc(C)nc1 51141,C1(C)(NC(C(=Cc2cnc[nH]2)C)=O)CCN(C(c2cc(C3CCOCC3)on2)=O)C1 51142,N1(C(=O)NCCOC(=O)OC2CCCC2)CCN(c2ccccc2)C(=O)C1 51143,c1(C(N2CC(CNC(c3ccc(SC)cc3)=O)C3C2C3)=O)cncc(Cl)c1C 51144,Cc1ccc2c(c1)C(C(=O)NC(C)CCNC(=O)C(=O)NC1CC1)CC2 51145,CC1CN(C(c2ccns2)=O)CCCN1C(=O)CCc1cccc(OC(F)F)c1 51146,N1(C(CC(C)C(F)F)=O)CCC2CCCC12C(=O)NC(C1CCC1)C1CC1 51147,CCC(F)(F)C(C)(C)C(=O)N1CCC(C(C)(C)NC(c2cccnc2S)=O)C1 51148,c1(C(N2CCN(C(=O)CCn3cnnn3)C(CO)C2)=O)ccc(O)cc1Cl 51149,C12(C(N3CC(C)(NC(c4ncc(OCC)nc4)=O)C3)=O)CCCCC1OCC2 51150,C#CC1CC2CCC1N(C(C1CCN(C(=O)CCC3CCCN3C)C13CC3)=O)C2 51151,c1(C2C(C(=O)NCCN(C(C34CCC(C3)C4)=O)CC)C2)ccc(CO)c(Cl)c1 51152,c1(C(N2CC(OC)(CNC(c3cnnn3C)=O)C2)=O)cc2ccccc2[nH]1 51153,c1(C(N(CC)CC2CCCN2C(C2OCCC2C(C)C)=O)=O)cccc(=S)n1O 51154,CC(C)(C(=O)NCCN(C1CCCC1)C(C1OCCOC1C(F)(F)F)=O)C(N)=O 51155,N1(C(CCC=C)=O)CCN(C(=O)C(c2ccccc2F)C)CC1CCO 51156,CCC(C)(COC)C(=O)N1CC(C2CC2C(N2CCOC(CCO)C2)=O)C1 51157,N1(C(CCP(C)(C)=O)=O)CC(CNC(=O)Cc2cccc(C#N)c2)CC12CCC2 51158,c1(OC)ccc(Cl)cc1CC(=O)NC1CC(NC(C2(O)CCCC2)=O)C1 51159,c1(C(N2CC(CC(=O)NC3CC4C=CC3C4)OCC2)=O)cc2n(n1)CCC2 51160,C1(CCC)CN(C(c2oc(C)cc2C)=O)CC1NC(c1ncccc1C1CC1)=O 51161,N1(C(CCC)=O)CCN(C(c2cc(C)nn2C)=O)C(CCO)C1 51162,C1(C(=O)NCC(CNC(=O)CN2CCS(=O)(=O)CC2)O)CC2C=CC1C21CC1 51163,c1(C(N2CCC(CNC(C(CC)(C)O)=O)C2)=O)cc2ccccc2cn1 51164,CC1CCN(C(C2CNC(=O)O2)=O)CCN1C(c1ccnn1CCF)=O 51165,N1(C(c2ccc(C(C)=O)cc2)=O)CCN(C(c2coc(C)n2)=O)CC1C(F)F 51166,Cc1ccc(C(=O)NCCSCC(=O)NCC(C)(C)O)c(F)c1 51167,c1(C(N2C(CN(C(=O)Cn3nnc(C)n3)CC)CCC2)=O)cc(C)nc(O)n1 51168,N1(C(CC=CC=C)=O)CCCC(N(C(=O)CCOc2cccc(C)c2)C)C1 51169,C1(C#N)(C(N(CCCC(=O)NC(CCOC)CO)C)=O)CCCOC1 51170,N1(C(C(C)(C)C)=O)CCC2CCCC12C1(N(C(=O)CCF)CCl)CC1.C1C(=O)N1 51171,CCC(C)(C)CC(=O)N1CC(N(C(=O)C(C)OC)C)C(O)C1 51172,C1(CNC(C=CC=CCC)=O)CN(C(=O)C(=O)NC(C)C)CCC1C 51173,N1(C(C2C(CCOC)C2)=O)CCCN(C(=O)Cc2sc(S)nc2C)CC1C 51174,N1(C(C2C(NC(c3c(COC)noc3)=O)CC=CC2)=O)CC(C)N(C)C(C)C1 51175,N1(C(CNS(CCCC)(=O)=O)=O)CCc2nc[nH]c2C12CCN(C(=O)C(N)=O)C2 51176,c1(C(=O)NCCC(C)NC(CC=CC)=O)cnc2ccccn2c1=O 51177,Cc1ccc(C)c(C(=O)NC(c2ccccc2)C(C)NC(c2ccncc2)=O)n1 51178,c1(SC(C)C(=O)NCCCCCn2cc(C3CC34CC4)nn2)ccc(F)cc1 51179,C1(C(=O)NC(C)Cn2cc(C3(N(C)C)CCC3)nn2)CCC(N(C)C)CC1 51180,c1(NC2CC(C)N(C(c3cc([N+](=O)[O-])c[nH]3)=O)CC2)ncc2c(c1C#N)CCC2 51181,C1(C)(C(=O)NC)C=CCN1C(C1CS(=O)(=O)C1)=O 51182,c1(C(N2CC(CNC(C(C)c3ccsc3)=O)C2)=O)ccc(-c2ccco2)o1 51183,N1(C(C2ON=C(C(C)C)C2)=O)CCC(N=[N+]=[N-])(C(=O)N(C)Cc2ccncc2)C1 51184,Cc1cc(O)ncc1C(=O)NC(C)CCCCNC(=O)CC1CCC(=O)NC1=O 51185,N1(C(C(C)C(C)(F)F)=O)CC2(COC(CNC(=O)C(C)N(C)C)C2)C1 51186,Cc1ccc(C(N2CCC(C)(C(N3CC(c4ncc[nH]4)C3)=O)CC2)=O)nc1C 51187,N1(CC)Cc2ccccc2OC(C)C1.C1(=O)N2CCC(CO2)CN1 51188,C1(C(=O)OCC)CCCN(C(C2(C)CCN(C(C3CC3(C)C(F)F)=O)C2)=O)C1 51189,Cc1ccc(C(=O)NC(C)CN(C(=O)C(C(C)O)N(C)C)C)cc1I 51190,c1(C(C)C)cc(C(=O)NCCN(C)C(c2ccc(=N)[nH]n2)=O)cc(Br)c1 51191,C1(NC(=O)C=CBr)CN(C(=O)COc2ccsn2)CC(F)(F)C1 51192,CC(C)(CCNC(C1OCC1(C)C)=O)NC(=O)CNC(c1ccccc1)=O 51193,C1(C2(O)CCC2)(C(N(CC(C)N(C)C(C2CC3CC2CC3O)=O)C)=O)CC1 51194,c1(CC)cnc(C(=O)NCC2(NC(C3CCC34CCC4)=O)CCCC2)cn1 51195,N1(C(CCCCC)=O)CC2CC(C(N3CCCC4(C3)N=N4)=O)(C2)C1 51196,c1(C(N2CC3C(NC(C(C(CC)CC)C)=O)(C3)C2)=O)nc(N)cc2ccccc12 51197,N1(C(C(CC)(F)F)=O)CCC(C)C(NC(c2ccc(CNC(C)=O)o2)=O)C1 51198,C1(C(N2CCN(C(C3C(c4c(C)cccc4)C3)=O)CC2)=O)CCC2CC2CC1 51199,C1(CSC)(NC(c2cc(Br)ccn2)c2nnnn2C)CCOCC1 51200,C1(NC(C(CC#C)O)=O)C2CCN(C(C3(C4CC4)CCCO3)=O)CC12 51201,c1(NC(C2C(C)C2c2ccccc2)=O)ccc(CCC(=O)O)cn1 51202,CC1(C)CN=C(N2CCN(Cc3ccccc3S(C)(=O)=O)CC2)S1 51203,c1(C(=O)NC(CC=C)CNC(c2cnc(C)n2C(F)F)=O)cnc(CO)nc1C 51204,CCC(C)C(C(=O)NCCn1ncnn1)NC(c1ncnc(O)c1F)=O 51205,N1(C(c2ccc(NCC)cc2)=O)CCCC(C)C1CNC(c1ccccc1)=O 51206,c1(-c2ccc(C(=O)NC(CNC(C3CCSC3)=O)CO)s2)cccc(F)c1 51207,C1(C(=O)NCC(CN(C(COCC(C)C)=O)C)C)CCC(N(C)C)CC1 51208,C1(NC(CCN(C(=O)C(c2ccn(C)n2)C)CC=C)=O)CCCC1C(C)C 51209,C1(CC(=O)NCC(C2(O)CN(C(c3cnn(C)n3)=O)C2)(C)C)CC2C=CC1CC2 51210,C1(CC(=O)NC2CC(N(C(CSCC(C)C)=O)C)C2)CN(C)CC1O 51211,O=C1NC(=O)C2CN(c3ccncc3S(=O)(=O)NCCCN3CCC3)CC12 51212,C1(OCC)CC2CCC1C2.n1(CC(=O)OCC2CC2)cccn1 51213,CC(=O)N=c1nc(C2CCN(C(C3CCN(C(=O)C(C)C)CC3)=O)CC2)[nH]n1C 51214,N1(C(c2ccc(OC)cc2C)=O)CCN(C(=O)C=CC=C(Cl)Cl)C(C)C1C 51215,C(C)(CCC(=O)NCCCCCO)NC(C1ON=C(C)C1)=O 51216,N1(C(C2CC2F)=O)CCC2(CCN(S(=O)(=O)c3ccc(O)cc3)CC2)C1 51217,c1(NC2C(NC(=O)OC(C)(C)C)CCOC2)ccc(C#N)c(Cl)c1 51218,Cc1cccnc1C(=O)NC1CC1CNC(c1c[nH]nc1C1CCC1)=O 51219,C1(C(N(CC(C)NC(=O)C(C)(C)N(C)C)CC)=O)CCC(O)CN1C 51220,Cc1ccc(C(C)C(=O)NCc2nc(CNC(=O)CC3C=CCC3)cs2)cc1 51221,C1(C(C)NC(c2ccc(C)o2)=O)CN(C(=O)CC23COCC(C2)C3)CCO1 51222,c1(OCC)cc(NC(C2CCCC(CNCC3(C)CNC3)C2)=O)ncn1 51223,C1(N(C(CCSCCCC)=O)C)CN(C(c2cc(O)n(CC)n2)=O)CCC1C 51224,C1(NC(CC(C)C2CCCO2)=O)CCC(C)N(C(=O)Cc2cnn(C)n2)C1 51225,N1(C(CCCc2onc(C)n2)=O)Cc2nccn2CC(NC(=O)C(C)(F)F)C1 51226,O=C(C=C(Cl)Cl)NCC1CC1CNC(c1sccc1-n1cccc1)=O 51227,Cc1nccn2c(C(N3CCNC(=O)C3c3ccccc3Cl)=O)cnc12 51228,c1(C(=O)NC(CNC(C(CC=C)C)=O)CO)cccc2[nH]c(C)cc12 51229,c1(N(CC(CN(C)C)O)C)ccc(Br)c(S(=O)(=O)NC2CN(C)C3(CCC3)C2)n1 51230,c1(C2(NC(=O)NCc3cc(Cl)cs3)CC2)ccc(F)c(F)c1 51231,N1(C(C2CCN(CC)CC2)=O)CCCC(O)(Cc2nc(C3CC3)no2)C1 51232,N1(C(C(C=CC)O)=O)CCOC(CCC)C1.C12(CCC1)C(=O)NC2 51233,C1(CC)COC(C)(C)CN1C(=O)C1=CCN(C(=O)CCC2CCCCO2)C1 51234,C1(CNC(COCCC)=O)CCCCC1NC(=O)Cc1ccc(Cl)s1 51235,C(=O)(C1=NOC2(CCC2)C1)N1CC(C)C(C(=O)NC2(c3nn[nH]n3)CC2)CC1 51236,N1(C(C(CC)F)=O)CC(C2CCCCN(C(C3CCc4n[nH]c(C)c4C3)=O)C2)C1 51237,c1(CC)cc(C(N2CC(Cc3ccoc3)C2)=O)nn1C.C12(CC1)CC(=O)N2 51238,C1(C(N2CCC(SC)CC2)=O)CCN(C(=O)Cc2nc(C3CC3)n[nH]2)C1(C)C 51239,C(=O)(C1=CCOC1)N1CCC1.CC(Cn1cccn1)C(=O)N(C1CCC1)C 51240,c1(C2C(NC(C3C(C(=O)O)NCC3)=O)C2)ccc(Cl)cc1 51241,c1(C(N2CC(CC(=O)NC(C(=O)NCC)(C)C)C2)=O)cnc(N(C)C)nc1 51242,C1(C(=O)NC(C2(O)CCN(C(=O)C(C)c3cccs3)C2)C)CCS(=O)(=O)CC1 51243,c1(C(=O)NC2(COC)CCCN(C(=O)CC(C)F)C2)ccc(C)c([N+](=O)[O-])c1 51244,C(CCC(C)(C)NC(=O)C(=Cc1cn[nH]c1)C)NC(CC(=C)C)=O 51245,c1(C(=O)NC2(CO)CN(Cc3ncsc3Br)C2)cccc(C(F)(F)F)n1 51246,C1(NC(c2c(C)ccc(Cl)c2)=O)COC2(C1)CN(C(c1ccnc(Cl)c1N)=O)C2 51247,Cc1cccc(C(C)C)c1-n1nc(CC2CC2)nc1C(c1cnn(C)c1)C 51248,C1(N(C(=O)CN(C(=O)COC)C)CC#C)CCN(C(c2n[nH]c(CO)n2)=O)C1 51249,c1(C(N2CC(C)C(NC(=O)Cc3cnn(C)c3)CC2)=O)ccn2nccc2n1 51250,C(C)(C)(CC(F)C(=O)NCCC1CCOC(C)C1)NC(C(=O)NCC)=O 51251,CN1CCN(C(=O)CN2CCCC2=O)CC1C(=O)NOCc1ccncc1 51252,C1(C(N2CC(O)(CNC(c3cnc(C4CCOC4)s3)=O)C2)=O)CC2(C1)CC2(F)F 51253,CCCC(C)(O)C(=O)NCC1CCC1NC(c1ccc(N)c(CC(C)C)c1)=O 51254,CC1CC(NC(=O)CC2CCN(C(C3CC(F)CN3)=O)C2)C(=O)O1 51255,N1(C(C(=O)NCC2CC(SCC)C2)=O)CCC(CNC)C(F)(F)C1 51256,CN1CCC(C)(C(=O)NCCOC2CCN(C(=O)CSCCC(F)(F)F)CC2)CC1 51257,C=CC(CC)CC(=O)NCC1CCN(C(c2cc(C(F)(F)F)ccc2O)=O)C1 51258,c1(OC)c(C(=O)NCC(C2CCCC2)NC(c2c(Cl)cnn2C)=O)ccnc1Cl 51259,Cc1ccnc(O)c1C(N1CC(NC(C23CC4CC2C3C4O)=O)C(C)C1)=O 51260,Cc1c(C(N2CC(F)(C(=O)NC3(C)CCCC3(F)F)C2)=O)cccc1O 51261,C=CC(C)(O)C(=O)N1CCCC(CN(C)C(c2ccnn2C(CC)CC)=O)C1 51262,[N-]=[N+]=NC1CC(C(=O)NOCC(=O)NCC2(C(N)=O)CCCC2)C1 51263,C(CCCCC(=O)NCCC1(O)CCN(C(=O)CCn2ccnc2)C1)NC(N)=O 51264,C1(C(=O)NC(C2CN(C(c3ncoc3-c3ccon3)=O)C2)C)C(C)(C)C1(C)C 51265,c1(OC)ccccc1C(CNC(C1CCC2CC12)=O)NC(C12CC(CO1)C2)=O 51266,C=CC1(CC(N2CCC(C)C2CO)=O)CN(C(c2nnsc2C)=O)C1 51267,C(=O)(CC(C)CNC(C1CC(NC(=O)C(CC2CC2)OC)CCO1)=O)NC 51268,CCCS(=O)(=O)CC(=O)NCC(C)(O)CNC(C1CC2(CCC2)CO1)=O 51269,N1(C(c2c(C)nc(N)cn2)=O)CCC2(CCC(NC(=O)C#CC3CCOC3)C2)C1 51270,c1(CC)ccc(CC(=O)NCC2CC2NC(c2cc(=O)n(C)cn2)=O)cc1F 51271,C1(C(=O)NC2C(NC(c3cc(F)cs3)=O)CCC2)CC2CCCC(C1)C2 51272,c1(C(N2CC(CNC(C(C=C)O)=O)OCC2)=O)ccc(C)c(S(=O)(=O)CCO)c1 51273,Cc1ccc2c(C(=O)N(C)CCN(C(=O)CC3CC(=O)C3)C)coc2c1 51274,N1(C(C(CC=C)CC=C)=O)CC2COCCC2(NC(c2ccc(Cl)nc2N)=O)C1 51275,c1(CNC(C(C2CC2)NC(C2N(C(C)(C)C)CC2)=O)=O)ccc(F)c(O)c1 51276,N1(C(c2cc(CNC(=O)CCc3cncnc3)no2)=O)CCC(C2CCCC2)C1 51277,C(C(CC)CO)NC(C1(N(C(COCCC=C)=O)C)CC1)=O 51278,c1(C(=O)NCC(C(=O)N(N2CCC(OC)C2)C)C)sc(C)nc1C 51279,CCCCC(O)CC(=O)NCC1(Cc2ccc(F)c(O)c2)CCCN1C(=O)C1CC1 51280,c1(-c2scc(CC(=O)NCC3(F)CCS(=O)(=O)C3)n2)ccc2c(c1)OCO2 51281,C1(C)(C(=O)NCC(CNC(C2(CC#C)CCCC2)=O)O)Cc2ccccc2N1 51282,C1(C(N2C(C)COC(C)C2)=O)CCCC2(CCCC2)O1 51283,CC1CN(C(c2nn(C(C)(C)C)cc2Cl)=O)CCN1C(C1CC(=O)NC1(C)C)=O 51284,c1(OC)c(F)cc(Br)c(C(=O)NNC(=O)Cn2nc(C)cc2C)c1F 51285,c1(C(=O)NC2CC2NC(c2cnns2)=O)cc([N+](=O)[O-])c2nsnc2c1 51286,c1(OC)nccc(C(N2CC(OC)CC(NC(=O)CSS(C)(=O)=O)C2)=O)n1 51287,Cc1nn(C)cc1C(=O)NC1(C)CC(NC(=O)C(C2CCCCCC2)O)C1 51288,c1(NC)cncc(C(N2CC3C(CNC(C4(C(C)(F)F)CC4)=O)C3C2)=O)c1 51289,c1(NCC2CCOCC2)cc(Br)ccc1S(=O)(=O)NC1C(CC(C)C)C1 51290,Cc1cccc(CN2CCC(C)(CN)C2)c1Br 51291,N1(C(C=NOC)=O)CCCCC1CC(=O)NC1C(C)C1C 51292,C(C(CC(=O)NC(CC1CC1)CO)NC(C1(C)COC1)=O)OC 51293,C1(CNC(c2ccns2)=O)COC(CNC(c2ccc(-c3ccccc3)o2)=O)C1 51294,c1(C(N(CCCCNC(C(C(CC)C)O)=O)C)=O)cc2ncn(C)c2cn1 51295,CCC(COC)C(=O)NC1CN(C(c2ccc(-c3csnn3)cc2)=O)CC1C 51296,C(=O)(C(F)C(C)(C)O)NCC1C(C)CN(C(=O)C=CCN2CCCC2)C1 51297,C1(C(NOC(C=C)C)=O)N(C(c2csnn2)=O)CCCC1(C)C 51298,N1(C(=O)CCc2ccccc2)CCC(C2CCCN(C(c3ccco3)=O)C2)C1 51299,Cc1sc(-c2ccccc2N2CCOCC2)nc1C(N1CC(OC)C2(CC2)C1)=O 51300,c1(C(=O)NC2CC(CNC(C3(C)N(C)CC(O)C3)=O)C2)ccc2nc(=N)[nH]n2c1 51301,C1(NC(c2n(C)ncn2)=O)CC2CN(C(=O)Cc3c(Cl)cnn3C)CC12 51302,C#CC1CN(C(c2cc(F)n(C)n2)=O)CCN1C(C1CCN(C)C1=O)=O 51303,C1(C(N(C)CC2C(NC(C3CC(C(C)C)C3)=O)CCC2)=O)CCc2nc[nH]c2C1 51304,CCCCCCCCCCC(=O)N1CCCC(N(C(=O)C2=CSCS2)CCO)C1 51305,N1(C(c2cc(C(N)=O)oc2)=O)CCC(NC(c2ccc(F)c(CO)c2)=O)C(F)C1 51306,Cn1cc(C(C(=O)NCC2(F)CCC2)NC(=O)CC2(O)CCC2)nn1 51307,N1(C(CCOCC#C)=O)CC(CNC(c2c(NC(C)=O)c[nH]c2C)=O)CC1C 51308,c1(C(=O)NC(CC(=O)N2C(C)(C(=O)NC)CC2)COC)coc2c1COC2 51309,c1(C(=O)NC23CC(NC(C45CC(CCO4)C5)=O)(C2)C3)ccc(F)cc1C(F)(F)F 51310,N1(C(CC(=O)OCC)=O)CCC(O)C(C(N2CCCCC2C(N)=O)=O)C1 51311,C1(O)(CCNC(c2c(C)coc2)=O)CCN(C(c2cc(Br)c[nH]2)=O)C1 51312,N1(C(c2ccc(OC)cc2)=O)CC(C)C(C)(CNC(=O)CCCCSC)C1 51313,CCCC(O)C(=O)NCC1(CNC(=O)C(C)SC)CCOCC1 51314,CCC(C)(CCC(C)C)C(=O)N1CCOC(C(N2CCC(F)(F)C2)=O)C1 51315,c1(C(=O)NC2C(C#N)CN(C(c3ccno3)=O)C2)ccc2ccccc2n1 51316,CCC(CC(=O)NC(C(=O)NC(C)COC)c1cccs1)C(F)F 51317,C1(CNC(CN(CCC#C)C)=O)CN(C(=O)CC2CN3CCC2CC3)CC1(C)C 51318,N1(C(C(C)C2CCC2)=O)CCCC(C2CN(C(c3cccc(C4CC4)n3)=O)C2)C1 51319,N1(C(C2COCCN(C(c3c(CC)ncs3)=O)C2)=O)CCCc2ccccc21 51320,c1(C(N2CCC(NC(c3n(C)ccn3)=O)C(F)C2)=O)cncc2[nH]ccc12 51321,C1(NC(C)=O)CCN(C(C2CCN(C(C3CCCC3C)=O)CC2)=O)CC1 51322,C1(C(C)(C)C)CC(C(=O)N2CC(CNC(=O)CCc3cn[nH]c3)C(C)C2)=NO1 51323,c1(C(=O)NC2(CO)CCN(C(C3C(c4c(C)ncs4)C3)=O)C2)ccc(N)cc1Cl 51324,c1(C(N2CC=CC(NC(=O)C3=CCC3)C2)=O)ccc2c(=O)ccoc2c1 51325,C(=O)(C#CC1(C)CCCO1)NC1CC2CN(C(c3nn(CC)c(O)c3)=O)CC21 51326,c1(C2C(C(N(C(C3CCOCC3)C)C)=O)C2)ccc2nsnc2c1 51327,c1(OC)cc(CN2CCCC2CC(N2CCC(CO)CC2)=O)ccc1O 51328,N1(C(C2(NC(CNC(CC)=O)=O)CCN(C)C2)=O)CCCN(C=O)CC1 51329,c1(CC)noc2ncc(C(N3CCN(C(C4CCCSC4)=O)C(C)C3)=O)cc12 51330,c1(C(N2CC3CC(NC(c4ncc(Cl)s4)=O)CC3C2)=O)ccc2c(n1)CCCC2 51331,S(=O)(=O)(C1CN(C(=O)NCC2CCOC2(C)C)CC1)NC 51332,C(=O)(C(C#N)C(C)C)N1CCC(C(C(=O)NC(c2nccn2C)CC)F)C1 51333,C(=O)(CCCCCNC(=O)C(C)C)OCC.C12CC1CNC(=O)CNC(=O)N2 51334,c1(NCC(=CCC(=O)NC)C=C)cc(N(C)C)ccc1C 51335,N1(C(c2c(CC)nco2)=O)CCOC(CCNC(=O)C(C)CF)C1 51336,c1(OC)cccc(C(=O)NC(C2CCN(Cc3cnc(C)s3)CC2)C)c1O 51337,C1(C(=O)NC(CCCNC(C(CC=C)(F)F)=O)CCCO)CN2CCN1CC2C 51338,Cc1nc(N(CCCO)C(C)C)ncc1-c1ccc(COCC(F)(F)F)cc1 51339,C=CC(CCC)CC(=O)N1CCOC(C)C1C(N1CCC(OCC)C1)=O 51340,S(=O)(=O)(c1ccc(OC)cc1C)NC(c1cccc(-c2ccsc2)c1)C(=O)OC 51341,N1(C(c2c(C)nns2)=O)CCCN(C(c2nc(Cl)sc2Cl)=O)CC1C 51342,N1(C(c2cc(CC)[nH]n2)=O)CC(CNC(=O)C(N2CCOCC2)C)CC(C)C1 51343,c1(OC)cc(N)c(F)cc1C(=O)N(C)CC1CCCN1C(C1C(C)C1C)=O 51344,Cc1ccc(Cl)cc1CN1CCC(n2cc(CC3CCCCO3)nn2)CC1 51345,C1(CC(=O)NCC=CCl)CCCCN1C(c1ccc(Cl)o1)=O 51346,C1(NC(CCc2c(C)cccn2)=O)CCN(C(C2(C)CCCC2)=O)CC1(C)C 51347,C(N=c1[nH]c(=N)[nH]c(=NC2CCN(CCF)C2)[nH]1)C1CC(CC)C1 51348,CC1C(NC(c2cncc(Cl)n2)=O)C(C)CCN1C(c1cc(Cl)cs1)=O 51349,C1(C(=O)OC)CC(CN)CN(C(=O)C(CC)(CC)OC)C1 51350,C=CC(C)(CC)C(=O)NCCCc1ccc(OC)cc1 51351,C1(F)(CNC(C)CC2CCC2)CCN(C(=O)OC2CCN(c3ccccc3)C2)C1 51352,N1(C(C(C)C)=O)CCN(C(=O)Cn2[nH]cnc2=N)C(C)C1 51353,C1(O)(CN(C)C(c2occc2Cl)=O)CCN(C(=O)CCC(N)=O)C1 51354,c1(NCC)cncc(C(=O)N(C)CCOCCNC(=O)CCc2cn(C)nn2)c1 51355,c1(OC)ccc2cc(C(=O)NC(CNC(=O)CC(C)C3CC3)C3CC3)[nH]c2n1 51356,c1(NCC2(CCOC)CC2)nc(N2CCC3(CC(=O)NC3=O)C2)nc2scnc12 51357,N1(C(CC)=O)CC2(C(N3CCN(ON=C(C)C)CC3=O)=O)CC1CO2.C(CO)SCC 51358,c1(C(N(CCCNC(=O)CC2CC3(CC3)C2)C)=O)sccc1C#N 51359,C1(F)(CNC(COCCCN(C)C)=O)CCN(C(c2cc(F)ncc2OC)=O)CC1 51360,C=Cn1nncc1C(=O)NC1CCC(NC(C2(CCC)CCC2)=O)C1 51361,c1(OC)cc(C)c(C(=O)NC2CN(C(=O)CCc3cnc(O)[nH]3)CC2O)c(C)c1 51362,n1(CC)nc(C)cc1C(N1CC(F)CC1C(N1CCC(O)(CC)C1)=O)=O 51363,C1(CN(C(=O)CCc2nccs2)C)CCCN(C(c2cnsn2)=O)C1 51364,N1(C(C(C(C)NC(c2cc(=N)[nH][nH]2)=O)(C)C)=O)CC(O)C2(CCCC2)C1 51365,c1(C(N2C(C3CCN(C(C=CC(C)(C)SC)=O)C3)CCC2)=O)cc(C)c(C)o1 51366,CCC(C)(C)C(C(=O)NCCn1cc(C(=O)NC2(CO)CCC(C)C2)nn1)OC 51367,N1(C(CC(C)P(C)(C)=O)=O)C(C)CC2CN(C(c3cccc4ncsc34)=O)CC12 51368,Cc1sc(C(=O)NCC2CCN(C(=O)C(C#N)C3CC3)CC2)cc1CS(C)(=O)=O 51369,C1(OC)CN(C)C(C)(C(=O)NCC(CO)NC(c2ccsc2SC)=O)C1 51370,N1(C(C(C)(F)F)=O)CCN(C(=O)CN2CC=CC2)CC(O)C1 51371,N1(C(c2cc(SC)oc2)=O)CCN(C(=O)CNS(=O)(=O)N(C)C)C(CC2CC2)C1 51372,C1(C(=O)OC)CC2CC2N1C(=O)C(N1CC2CC2C1)C 51373,CCC(C)(C)C(=O)C(=O)N(CCOC)CCOC(C)=O.C1C(=O)NOCCCO1 51374,c1(-c2ccc(C(=O)NCCN(C(=O)CCCc3ncco3)C)[nH]2)ccccc1F 51375,c1(C(N(CC(C)NC(=O)C(C)(O)c2ccccc2)CC)=O)ccc(C)nc1OC 51376,Cc1ccc(C)c(CN(C(c2cccc(Br)c2)C(=O)O)C)c1 51377,c1(C(=O)OC)cc(C#N)cnc1NC1CC2CN(C(C3C=CC=CC=C3)=O)CC12 51378,c1(C(=O)NC2(C)CN(C(C3CC(C#N)C3)=O)C2)nnn2c1CSCC2 51379,c1(CC)ccc(NC(C2(COC)CN(C(c3cccc(OC)c3)=O)C2)=O)c(C)n1 51380,Cn1ncc2c(N3CCC4(NC(=O)Cn5cnnc5)CCCC34)ncnc12 51381,C1(NC(=O)C(F)CC2CC2)CN(C(c2cccc(Br)c2)=O)CC2(CCC2)C1 51382,c1(C(=O)NC2CN(C(CC(CCC)O)=O)CC(C)C2)cc2ccc(F)cc2[nH]1 51383,C1(CC)(NC(=O)CN(C)C)CCCN(C(=O)CN2CCC(OC)CC2)C1 51384,C[Si](C)(C)CC(C(=O)O)NCc1ccc2c(c1)COC2 51385,CCCC(CCC)CC(=O)NCC1CCC(C)(C)CN1C(c1sncc1CC)=O 51386,CN1CCC(CC(=O)NCCNC(c2ccc(F)cn2)=O)CC1 51387,c1(N(C(CCN(C(C(OCC)OCC)=O)C)=O)C)cnccn1.C1CO1 51388,c1(C(=O)NCC(C2CCN(C(C(C(CC)O)C)=O)CC2)C)cc2cccnc2o1 51389,CCCCCC(O)CC(=O)N1CCCC(C2CCCCN2C(c2cnsc2)=O)C1 51390,CC(C)CC(O)C(=O)ONC(=O)CC1(CO)CC1.CC(CO)C(C)C 51391,C1(NC(C(COC)OC)=O)CC(N=c2[nH]c3c(C)c(C)ccc3s2)C12CCC2 51392,c1(CNC(C2(C)CN(C)C(=O)C2)=O)ccc2c(c1)CN(C(=O)CS(C)(=O)=O)C2 51393,c1(C(=O)NC2C(NC(C(CC)C)=O)C2)c(OC)cc(OC)cc1OC 51394,C1(C(N2C(CN(C)C(c3cnc(Cl)cc3I)=O)COCC2)=O)CCC(C#N)CC1 51395,c1(C(=O)NC2C(CNC(c3c(COC)nn(C)c3)=O)C2)cc2occc2n1C 51396,N1(C(N2C3(C)CC(C(F)F)(C2)C3)=O)CCCN2CCCC12 51397,CC(C)CC(C)N(C(=O)CCN(C(=O)CC1OCCO1)C(C)C)C 51398,CCC(C)(CCNC(=O)C(C)SC)NC(=O)Cc1ccn(C(C)C)n1 51399,C1(N(C(=O)C(C)Cc2ccco2)CC(C)C)CCN(C(C2COCCO2)=O)CC1 51400,C1(C(=O)NC(C2CC(NC(C3CC3C3(C)COC3)=O)C2)C)CCC(O)CN1C 51401,c1(C(=O)NCC2C(CNC(C3(CC=C)CC3)=O)C2)cnc2[nH]ncc2c1 51402,N1(C(Cc2cc(=N)[nH]cc2)=O)CCCC(NC(c2cccc(CO)c2)=O)CC1 51403,c1(NC(Cc2nc(CC)sc2)=O)ccc2[nH]c(C)cc2c1 51404,CCC(Cc1ccccc1)C(=O)NC1CCCC1CNC(c1ccc(SC)o1)=O 51405,c1(N2CC(C(C)N)OCC2)cc2nncn2cn1.C1(=O)CN1C.N(C)C 51406,C#CCC(O)C(=O)N1CCOC(CNC(C2C3CC(=O)CC23)=O)C1 51407,N1(C(c2cc(OCC)n[nH]2)=O)CCC2(CC1)CN(C(C1SCCS1)=O)CC(C)O2 51408,c1(CCNC(=O)NC(CSC)(C)CO)cc(C)ccc1Cl 51409,C=C1COc2c(C(=O)NC3CC(CO)N(C(C4(N(C)C)CCC4)=O)C3)cnn2C1 51410,Cc1nc(Cl)ccc1S(=O)(=O)N1CCC(F)(C(=O)NCC(F)F)C1 51411,c1(OCCCOC)ncccc1CNC(c1nnc(C2CCNCC2)s1)=O 51412,C1(C(=O)NC(COC)C(=O)N2CC(N3CCC3)C2)CCC2(CC2)C1 51413,Cc1cccc(Br)c1C(C(=O)NC1(C)CC1C)NC(C1(C)CCCCO1)=O 51414,c1(C(N2CCCC(NC(C(C=C=C)C)=O)C2)=O)ccc(S(N)(=O)=O)c(F)c1 51415,C1(NC(CSC)=O)CC12CCN(C(c1n[nH]cc1C1CCC1)=O)CC2 51416,CN1C(=O)CCC1CNC(c1occc1CNC(c1csc(F)c1)=O)=O 51417,N1(C(c2cccc(OCC)c2)=O)CCN(C(=O)CSC)C(c2ccnn2C)C1 51418,c1(C(N2CCCC(N(C(=O)C3=CCCO3)C)CC2)=O)ccc2cncn2c1 51419,C=CCC(F)(F)CN(C(=O)CN(C)C(C1CCN1C(C)(C)C)=O)C 51420,C1(C(N(C(C)CC(=O)N(C)CCC2CCCO2)C)=O)C2CN(C)CC12 51421,c1(NC(C)=O)ccc(Cl)c(C(N2CCOCC2CNC(=O)CNS(N)(=O)=O)=O)c1 51422,c1(-c2ccc(CN3CC(C(=O)OC)C(C)CC3)s2)cccc(F)c1C#N 51423,C=C(C)CC(=O)NCC(=C)CCNC(c1cncn1-c1ccccc1)=O 51424,C(=O)(CC(C)CC(=O)N1CCC(C)(C)C1C(=O)NCCCc1cc(C)no1)OC 51425,c1(CC=C)ccccc1C(=O)NC(C)C=CC(=O)NCc1c(C)noc1C 51426,C1(NC(C=Cc2c(C)ccs2)=O)CN(C(=O)C(=C2CCCCC2)F)CC12CCC2 51427,C1(C)(NC(C=CC(CC)C)=O)CC(NC(C2CCC(C(F)(F)F)O2)C2CCC2)C1 51428,c1(C(N2CCC(NC(C3(C)CCC(=O)N3)=O)C(O)C2)=O)cc2ccc(F)cc2s1 51429,c1(C(=O)NC2CC(CNC(C3CC(F)(F)C3)=O)C2)nccc(Br)c1O 51430,CC(F)(C(=O)N1CCC(CCOCCc2ccccc2F)CC1)C(F)(F)F 51431,CCCC(C(=O)NCC)NC(=O)C(c1cn(C)nn1)NC(=O)CC1CCN(C)C1 51432,C1(NC(c2nc(C#C)sc2)=O)CS(=O)(=O)CC1NC(=O)CN(CC)CC 51433,c1(C(N(C2CCCN(C(C(C)N(C(C)=O)C)=O)C2)CC)=O)ccc(F)c(C)c1N 51434,c1(C(c2onc(Cc3cn(C)nc3-c3ccnn3C)n2)=O)ccc(F)c(F)c1 51435,CC1CN(C(C2CCN2CC(F)(F)F)=O)CC1(C)CNC(=O)CCOCC(F)F 51436,Cc1cnc2c(C(=O)NC3CN(C(=O)CO)CC34CC4)cccn12 51437,C1(CC(=O)Nc2c(CC)ncs2)CCN(C(=O)CNC(N)=O)C1(C)C 51438,c1(C(=O)NC2(C)CCN(C(C3CCC3)=O)C2)nc(Cl)ccc1N 51439,N1(C(CNC(C=C(CC)C)=O)=O)CCC(N(C)C(c2[nH]c(C)nc2C)=O)CC1 51440,N1(C(CCc2cc(C)sc2C)C)CCN(C(N)=O)CC1C 51441,c1(C(C)C)cccc(OCC(N2CCC(C)(NC(=O)CCS(C)=O)C2)=O)c1 51442,N1(C(C2CN(C(C)=O)C2)=O)CC(C(=O)NCC(C)(F)C(C)C)C(F)(F)C1 51443,c1(C2C(C(=O)NCC3CC(NC(=O)C(F)=CC4CC4)C3)C2)ccc(F)cc1F 51444,C(c1ccccn1)=C(C)C(=O)NC(C)C(C)NC(=O)CN(CC(C)(C)C)C 51445,CC(c1cccs1)=CC(=O)NCC1(C)CCCN1C(=O)C=Cc1cocn1 51446,N1(C(CC2(N(C)C)CCC2)=O)CCC2CC12C(=O)NC(CO)CCCO 51447,C#CCC(CC(=O)NCC#CC1CC1)NC(=O)CN1CCC(C)C1 51448,C(C)(c1cnccn1)=CC(c1n(CC=C)nnn1)(C)NC1CCCCC12CC2 51449,C(=O)(CC(CN(C)C)C(F)(F)F)NCCN(C(CCC1C(C)=NOC1=O)=O)C 51450,c1(C(N2C3(CNC(CCCOCC)=O)CCC2CC3)=O)c(C)cc(C)cc1O 51451,C1(F)(C(N2CCC(OCC(C)C)C2)=O)CCCN(C(c2c[nH]nc2Cl)=O)C1 51452,c1(C(=O)NCCN(CC(C)O)C(=O)Cn2ncnn2)cc(F)cc(S(N)(=O)=O)c1 51453,c1(C(=O)NC2CN(C(c3cc(CC)[nH]n3)=O)C(C)C2)ccc(=O)n2c1COCC2 51454,C1(C(=O)NC(C23CCC(CC2)C3)CNC(COC(CC)C)=O)CCOC(=O)CC1 51455,c1(OCCN(C)C)ccc(C(N2CC(NC(=O)Cc3ccsn3)C(O)C2)=O)cc1N 51456,c1(C(=O)NC2CN(C(C3(F)CC=CCC3)=O)C2)cc(O)nc(O)n1 51457,C1(N(C(C2C(C)(C(C)C)C2)=O)C)CC2CCC(C1)N2C(C1CC(N(C)C)C1)=O 51458,c1(C(=O)NCC(CC=C)NC(C2CCCC(O)C2)=O)cccc2c1CCCN2 51459,C1(C(=O)NC2CC(NC(C(C)OCC)=O)C2)CCC2(CC1)CC2(F)F 51460,Cc1cc(C(=O)NCCC(O)CNC(=O)CCC2CC2)n(CCO)n1 51461,CCCC(C)(O)C(=O)NCCN(C(c1nc(C)nn1C)=O)Cc1ccc(Cl)nc1 51462,C1(NC(=O)NC(c2ccc(OC)nc2)C)(CO)CCCCC1C 51463,N1(C(C2C(C)CCO2)=O)CC=CC(C(=O)N(C)CC2CC2)C1 51464,CC1CN(C(=O)COC2CC2)CC(C(=O)NC2CC(C(F)F)C2)O1 51465,C(c1cccc(Br)c1)=CC(=O)NC(CC)CNC(=O)Cc1ncn(C)c1C 51466,C(CC(C)C)(C(=O)Nc1cncnc1C(C)C)ONC(C(C)NC(C)=O)=O 51467,c1(CNC(c2cccc(C)n2)CC)nn(C)c(Cl)c1I 51468,C(=O)(C(O)CC[S+](C)C)NCc1cn(CC(C)NC(c2cc[nH]n2)=O)nn1 51469,n1(CCN(CCCCCCCN)C)nc2ccccn2c1=O 51470,Cc1nnccc1C(N1CC(N2CCN(C(=O)Cc3cc[nH]c3)CC2)C1)=O 51471,c1(OC)c(C)cc(C(N2CCCC2CNC(=O)C=C2CCC(C)C2)=O)cc1C 51472,Cc1cc2c(CC(=O)N(C3CC(NC(c4ccc(=O)n(C)n4)=O)C3)C)csc2s1 51473,C1(C(=O)Nc2ccc(-n3cncn3)cc2)CC(F)CN(Cc2cc(Cl)ccn2)C1 51474,C1(NC(C2CCC(=C)CC2)=O)CCN(C(=O)Cn2cc(C(F)(F)F)nn2)C(C)C1 51475,C1(C(=O)NCC(C)C(=O)NC(c2ccncn2)C)C(C)(C)C1(F)F 51476,C1(F)(C(=O)NC2C(C(C)C)CCCC2)CCN(C(c2ccccc2)=O)CC1 51477,C1(CNC(=O)CSC(F)F)CN(C(C23CC4CC2C3C4O)=O)CCC1(F)F 51478,N1(C(c2cnc(CC)s2)=O)CC2(CC(CC(=O)N(CC)CC3CCC3)C2)C1 51479,c1(C(N2C(CNC(C=C(C)CCc3ccccc3)=O)CC2)=O)ccc(F)cc1O 51480,N1(C(C(C)n2cncn2)=O)CC2(C1)CN(C(=O)CC1(C#N)CCOCC1)C2 51481,CC1(CNC(C2CN(CC(F)F)C2)=O)CCCN1C(=O)CSCc1ncc[nH]1 51482,N1(C(c2c(C(=O)OCC)c[nH]c2)=O)CC2C(CNC(c3cnccn3)=O)C2C1 51483,C1(NC(C2N(C(C(CN(C)C)O)=O)CCN(C)C2)=O)CCCC(C2CC2)C1 51484,c1(C(N(C(C(=O)NCCC#N)C2CC2)C)C2CC2)ccc(F)c(F)c1 51485,C(CCCC(=O)N(C)CC1CCCN1C(=O)CNc1ccccc1)OCCC=C 51486,c1(C(N(C2CCN(C(CN(CCOC)C)=O)CC2C)C)=O)cc2cccnc2o1 51487,CC1C(NC(c2ccnn2CCF)=O)CCCN1C(C1(C#N)CCCCC1)=O 51488,Cc1nnc2n1CCCC2C(=O)c1noc(-c2cc(F)ccc2F)n1 51489,N1(C(C(NOC)=O)=O)CCC(C=CC(=O)N(C)C(C)C)CC1 51490,C1(CC(=O)O)CCCN(C(C2CCCN(C(=O)C(c3cccc(Cl)c3)O)C2)=O)C1 51491,C1(NC(C(=O)NCCOC)=O)CCCCN(C(=O)Cn2cccn2)C1 51492,CC(C)(CC(F)(F)F)C(=O)NCC1(F)CC(CNC(C2CN3CCN2CC3)=O)C1 51493,C1(O)(CN(C)C(c2ccnn2C(F)F)=O)CCN(C(=O)COC2CCOC2)C1 51494,C1(C)(CNC(C(C)(N(C)C(c2cn(C3CC3)cn2)=O)C2CC2)=O)CSCCO1 51495,CC1CN(C(c2cscc2Cl)=O)CC1NC(c1cccc(OC(F)(F)F)n1)=O 51496,c1(OC(C)C)c(F)cc(C(N2CC3CCC2CN3c2ncncc2Br)=O)cc1F 51497,C1(N(C(COCC(C)C)=O)C)CCN(C(=O)Cc2cncn2C2CC2)CC1 51498,N1(CC(=O)NCC2(NC(c3c(C(C)(C)C)cco3)=O)CCOC2)CCCNC1=O 51499,C(=O)(C(C)CC(C)C(C)=O)NC1C2OCC(NC(c3c(CC)n(C)nc3)=O)(C2)C1 51500,c1(CC)cncc(CNC(C2(CC)CN(C(C3CCCC(O)C3)=O)C2)=O)c1 51501,C1(CNC(c2c(C)coc2)=O)CN(C(=O)C(O)C2CCCC2)CC1(F)F 51502,C(CO)(CCCCNC(c1ccnn1C(F)F)=O)NC(c1c(C(C)C)ncs1)=O 51503,N1(C(CN(C(C(C)C)=O)C)=O)CCCC(C)(NC(=O)C(O)C(F)F)C1 51504,c1(OCCOCCNC(CC=CC=C)=O)nnc2n1CCC2.C1CO1 51505,C1(NC(Cc2c(C)con2)=O)CC=C(C(=O)N2CC(C)C(C)C2C)C1 51506,N1(C(CCC#CC)=O)CCC2(CC(NC(=O)Cc3nc([N+](=O)[O-])n[nH]3)CO2)C1 51507,c1(C(=O)NC(C2CCN(C(c3c(SC)csc3)=O)C2)C)n[nH]cc1[N+](=O)[O-] 51508,Cc1cc(Cl)cc(C(N2CC(NC(=O)CSc3ccncc3)CC(C)C2)=O)c1N 51509,C(=O)(CP(=O)(C(C)C)C(C)C)NC1CCN(C(C(CC2CC2)OC)=O)CC1F 51510,c1(OC)cccn2ncc(C(=O)N(CCO)Cc3cc(F)ccc3Br)c12 51511,c1(CC)cc(CNC(=O)NCC2(C)CSC(C)=N2)cc(C)c1 51512,C(=O)(C(C)S(N)(=O)=O)NCC1(O)CC(C(=O)NCCc2cc(C)no2)C1 51513,N1(C(C2(C)CCCN(S(=O)(=O)CCBr)C2)=O)C2CCCC1COC2 51514,CCCCCC(CC)C(=O)NC1CN(C(c2nccnc2CC)=O)CC1N=[N+]=[N-] 51515,C1(C(=O)O)(COC)CCCN(C(c2ccc(OCC(F)F)nc2)=O)C1 51516,C1(C(=O)NCCC2CCN(C(C=Cc3nc(C)sc3)=O)C2)Cc2ccccc2O1 51517,c1(C(N(CC(=O)NC2CCC2NC(C2CC23CC3)=O)C)=O)ccccc1Cl 51518,c1(-n2cc(C(C)NC(c3ccoc3)=O)nn2)cccc(Br)c1 51519,CN1CCC(N(C(=O)C(O)C2CN(C(=O)CN3CCC(O)CC3)C2)C)CC1 51520,CC(C)(CC(F)(F)F)C(=O)N1CCN(C(=O)CCCCC(N)=O)C(C(F)F)C1 51521,c1(NS(C)(=O)=O)ccc(F)c(F)c1.c12cncc(c1)C(=O)N(N(C)CCO)C2 51522,N1(C(c2c(CCC)occ2)=O)CC(OC)C(OC)C1CNC(=O)CC(C)F 51523,c1(OC)cc(NC(=O)CCC2CCC(NCc3cnn(C)c3)C2)[nH]n1 51524,c1(CC(=O)N(C(C)C)CCN(C)C(C2CCOC2C)=O)cnc2n1CCCC2C 51525,N1(C(C23N(C(CCSCCCC)=O)CC(CO)(C2)C3)=O)C2CCC1CC(C)C2 51526,Cc1cc(=NCCCN(c2ccccc2)C)[nH]c(NC2CCCn3nccc32)n1 51527,N1(C(C(CC(=C)Cl)NC(=O)Cc2ccn(C)n2)=O)CC(=O)NC(C)(C)C1 51528,c1(C2C(C(=O)NCC(CNC(c3cc(OC)ns3)=O)(C)C)C2)cccc(C#N)c1 51529,C1(C(=O)NC2C(OC)CN(C(=O)CC3(C#N)CCC3)C2)CCCCNC1=O 51530,c1(N(C)Cc2cccc(OC)c2OC)nccc(=NC2CCCC2S(C)(=O)=O)[nH]1 51531,C1(C(N(CCC(=O)NC(C2CC(F)C2)C)CC2CC2)=O)CCOCC1 51532,N1(C(CCCSC)=O)CCC2(C1)c1[nH]cnc1CCN2C(=O)CCc1nccs1 51533,N1(C(COCC)=O)C(C(N2CSCC2C(N)=O)=O)CCC12CC2 51534,C1(C(N(C(C#C)C)C)=O)C2CCC(C2)C1NC(C1CCC1C#N)=O 51535,C=CCC(C(=O)NC1C=CCC(C(=O)NCc2ccc(C)cc2)C1)C(C)C 51536,N1(C(C2C(C)C2)=O)CCC2(CC(C(=O)Nc3cncc(Br)n3)=NO2)C1 51537,c1(C(C(=O)NC2CCN(C(c3cnc(CC)[nH]3)=O)C2)C)c(C)n[nH]c1C 51538,N1(C(CC=CCNC(C(C(C)C)CN(C)C)=O)=O)CCC2(CC(F)C2)C1 51539,C1(CCC(=O)NCC(C2CCCC2)NC(C(C)N(C)C)=O)CCN(C)CC1 51540,C12(C(=O)NC(CCCC)CNC(=O)C(F)n3ccnc3)C3CC(CC13)C2(F)F 51541,N1(C(c2c(OC)cncc2)C(=O)NCC2CCOC2)CC(CO)C(C2CC2)C1 51542,c1(CC(OCC)OCC)cn(Cc2ccc(C(=O)N(C(C)C(F)F)C)o2)nn1 51543,C1(C(=O)NCC(CC=C)NC(c2cnc(C)[nH]2)=O)CCC(C(=O)OC)CC1 51544,c1(C(N(C2C(NC(CC(CC)C3CCC3)=O)CCCC2)C)=O)ncnc(C)c1C 51545,C(CC(C)(C)NC(=O)C(C)N1CCC1)NC(C(c1ccccc1)OC)=O 51546,C1(NC(C)=O)CCCCN(C(c2cc(C)n(CC3CC3)c2C)=O)C1 51547,N1(C(c2c(C)nn(C)c2)=O)CCc2c(C(N3CCCCC(O)C3)=O)csc2C1 51548,CCCCCC(O)CC(=O)N1CC2CCCC2(C(=O)NCC(C)C(C)(F)F)C1 51549,c1(C(=O)NC2C(C)N(C(=O)CCc3ccc(Cl)nc3)CC2)ccc2c(c1)COC2 51550,c1(OC)cncc(C(N2CCOC(CNC(C3CC(=O)N(O)C3)=O)C2)=O)n1 51551,Cc1ccc([N+](=O)[O-])cc1C(=O)NC(C)C(C)NC(=O)C(CO)C(F)(F)F 51552,C(CNC(C1CCCCCC1)=O)(CC(C)C)NC(C1(C(=O)OC)C(=C)CC1)=O 51553,C1(C(=O)NCC(COC)O)CCCN(Cc2ccc(CN(C)C)cc2)C1 51554,C12(C(N(CCN(C(=O)CCc3ccnn3C)CC)CC)=O)CC(CO1)C2(C)C 51555,c1(C(C)N(C(c2cnc(N(C)C)nc2)C(=O)NC2CC2)C2CC2)ncc(Cl)n1C 51556,c1(CCCCC)nc(C(=O)N(CC(CC)NC(=O)CCc2nc(=N)[nH][nH]2)C)cs1 51557,c1(CC(=O)NC(CCNC(CC(CC)SC)=O)C)ncn2c1CCCC2 51558,CC1CCC(C(=O)NCCn2ccc(C(=O)NCC(F)(F)C(N)=O)c2)CC1 51559,c1(C(=O)NCCN(C(Cc2c(C)ccs2)=O)C)ccc2[nH]ccc(=O)c2c1 51560,C1(C(=O)NC(CNC(C2(COC)CCCO2)=O)C2CCC2)CC2CCC(C1)C2 51561,C12(C)NC(=O)N(C1=O)CCC1(C)CN(C1)C2.c1(CNC(C)=O)sccc1C(=O)O 51562,c1(C(C(N2CCC(CNC(CNC(=O)OCC)=O)CC2)=O)O)c(C)cccc1C 51563,Nc1cccc(C(=O)NCCCCCNC(=O)CCn2cccnc2=O)c1 51564,c1(OC)noc(C)c1C(=O)NC1CCC(CC(=O)NC2CC2c2cncs2)CC1 51565,c1(OCCN(CC)Cc2ncc(OC(F)(F)F)cn2)ccccc1NC(C)=O 51566,Nc1ccc(F)c(C(N2CCC(NC(=O)Cn3cc([N+](=O)[O-])cn3)C(F)C2)=O)c1 51567,C(CC(C)C)(C(C(=O)NCC(F)F)N1CCSCC(C)C1)OC 51568,c1(CN(C)C(C2COCCN2C(=O)CC2CC2)=O)ccc([N+](=O)[O-])cc1 51569,c1(OC)cc(C)c(NC(=O)NC(c2ccc3c(c2)OCO3)CCO)c(C)c1C 51570,n1(CC)nc(C)c([N+](=O)[O-])c1NC1CN(C(=O)C(CC)OCCNC)C1 51571,c1(C(=O)NCC(F)CNC(C2(C(F)F)CC2)=O)cccc2ccnn12 51572,c1(C(=O)NCC2C(C)CN(C(C3CC(O)C3)=O)CC2)nc(Cl)c(=O)[nH]c1N 51573,C1(C(N(C(CCNC(Cn2ccc(C)n2)=O)C)C)=O)CC(=O)N(C2CC2)C1 51574,c1(C(=O)NC(CN(C(c2cnc(OCC)nc2)=O)C)CC)ccc(F)cc1C 51575,c1(C(N2CCCC(NC(c3cncc(F)c3Cl)=O)C2)=O)nc2cc(O)ccc2[nH]1 51576,N1(C(CCCCC#C)=O)CCS(=O)(=O)C(CCNC(=O)C(O)P(C)(C)=O)C1 51577,N1(C(C2C(OC)CC2)=O)CCC(NC(=O)CNC(c2cccc(C)c2)=O)C(C)C1 51578,C1(O)(C(=O)NCCCCC(C)NC(=O)CN2CC3C=CC2C3)CCCC(C)(C)C1 51579,c1(C(=O)OC)ccnc(C(N2CCNCC2C)=O)c1F 51580,S(=O)(=O)(c1cc(Br)c(Br)s1)N1CC2(CCN(Cc3cncc([N+](=O)[O-])c3)C2)C1 51581,C(=O)(C(CC1CC1)NC(c1cocn1)=O)N(CCOC)C(C)C1CC1 51582,C1(NC(c2cc(N)c(Cl)nc2)=O)CCCC12CCN(C(c1ccnnc1O)=O)C2 51583,c1(C(N(CC(O)CNC(C2(n3cccn3)CCC2)=O)C)=O)csc(Cl)c1 51584,C(C(=O)N=c1cc(C(N)=O)n(C)[nH]1)C1N(C(C(C=C)O)=O)CC(O)C1 51585,C(C(CNC(=O)C(CO)N(C)C)C(F)(F)F)NC(C1CCN(C)C1)=O 51586,c1(C(N(C)CC2N(C(CC(C=C)C)=O)CCCC2)=O)cc(C)cc2cccnc12 51587,C1(NC(c2n(C)ccc2)=O)C=CCCC1C(N1CCC2CCC12)=O 51588,c1(OCC(=O)N(C(CNC(c2c(C)c[nH]n2)=O)C)C)ccccc1C(C)(C)C 51589,c1(C(N2CC(CCNC(C(CC)c3cccnc3)=O)C2)=O)ccc2c(c1)COC2 51590,C(Cc1ccccc1)(CCCO)NC(=O)Nc1n(CC)nnc1 51591,c1(SC)ncc(C(=O)NCC(O)CNC(C2CCCN2C(=O)NC(C)C)=O)s1 51592,c1(SCC(N2CCN(C(C3CC(C)(C)C3)=O)CC2)=O)ccc(F)c(F)c1 51593,N1(C(C(c2ccc(C)cc2)CC)=O)CC2(CCC(CNC(=O)CC(C)F)O2)C1 51594,N1(C(C(C)NC(=O)NC)=O)CCN2CCN(C(=O)C(O)CC(C)C)CC2C1 51595,N1(C(c2c(COC)cccn2)=O)CCC(NC(=O)C(F)CC(C)(C)C)C(C)(C)C1 51596,c1(NC2CC(OC)C23CCNCC3)nc2c(cc1C#N)CCOC2 51597,CCS(=O)(=O)CCN(C(c1cccc(Oc2ccc(F)cc2)c1)C(=O)NC1CC1)C 51598,C1(NC(=O)OC(C)(C)C)CN(C(=O)CC(F)F)CC1C(=O)NC1CCCC1 51599,C(=O)(CCCCCNC(C)=O)N1CC(OC)C(NC(=O)C(O)C2CCCC2)C1 51600,N1(C(C2(CC)CC2)=O)CC2CCN(C(=O)C=C(C)I)C2C1 51601,N1(C(c2c(CNC(C(CCCC)=O)=O)occ2)=O)CC(C)OC2(CCC2)C1 51602,C#Cc1ccc(C(N2CCC(CCNC(c3cnc(C)s3)=O)CC2C)=O)c(F)c1 51603,CCC(C(=O)N1CC=CC1CNC(c1ncccn1)=O)NC(N)=O 51604,c1(C(=O)NC2C(NC(C(CC)n3cccn3)=O)C2)cc(OC)c(Cl)cc1OC 51605,c1(C(N2CC(CCNC(Cc3n(C)ccc3)=O)OCC2)=O)cnc2[nH]ccc2n1 51606,Cc1oc(C(=O)NC2CC3CCC2N3C(=O)C(O)C(C)C)cc1S(N)(=O)=O 51607,C1(NC(C2(C(N)=O)CC2)=O)CCCC(NC(=O)C(c2ccc(O)cc2)=O)C1 51608,N1(C(C(C)OCC)=O)CCC(F)(CNC(c2ccc(N)cc2Br)=O)CC1 51609,c1(SC(CNC(=O)Cc2ccno2)C2CN(C(=O)COC3CCC3)C2)nc[nH]n1 51610,Cc1c(CN2CCC(C(=O)C3CC3)C2)cc(F)cc1Br 51611,c1(CN(C(C)C)C(c2ccc(-c3cc(O)n[nH]3)cc2)=O)nc(O)c2ccccc2n1 51612,C1(C(=O)NC(c2ncc[nH]2)(C)C)CN(C(=O)CN2CCC(=O)CC2)CC1(F)F 51613,N1(C(C2N(CC#C)CCC2)=O)CCCC2(CC(NC(C3CC(F)(CO)C3)=O)C2)C1 51614,N1(C(C(CO)NC(c2ccc(F)cn2)=O)=O)CC2CC1CO2 51615,C(CN=c1[nH]c(=NC2COCC2CO)[nH]c2c1COC2)N1CCC(OCC)C1 51616,c1(CCC)c(C(=O)NCC(CC)NC(=O)CC2CC=CCN2C)cnn1C 51617,C1(NC(C=C(CCC)C)=O)CC2CC1N(C(=O)CC(CC)C1CCC1)C2 51618,c1(C(N2CCC(C)C(NC(C3C(=C)CC3)=O)C2C)=O)ccc2c(c1)COCCN2 51619,C1(C2CC2)(NC(C2C(OCC)C2)=O)CCN(C(=O)C(Cc2ccccc2)SC)C1 51620,C(=O)(CCCC(F)F)N1CCC(NC(C(C(C)C)C)=O)CC1 51621,C1(OC)CCCC(C(N2CCCC2CCCNC(=O)Cc2c(Cl)cnn2C)=O)C1 51622,N1(C(CCOCCOCC)=O)CC(C)N(C(C2CCC(C)(C)OC2)=O)CC1C 51623,C=CC(C)(CCOC)C(=O)N1CC2CC1C2CNC(C1(CC(C)C)CC1)=O 51624,c1(CC)ccccc1C(=O)NC1CCOC(C(=O)NOCCCN(C)C)C1 51625,c1(N2CCC(N3C(=O)CC(OC)C3)CC2)ccnc(-c2ccccc2)c1O 51626,C(N=c1[nH]c(=N)[nH]c(=NCc2ccc(Br)o2)[nH]1)C1(OC)CCS(=O)(=O)C1 51627,C1(C(C)=O)CC1(Cl)C(=O)NC1CC1NC(=O)COc1cn[nH]c1 51628,CCC(C)CC(C)C(=O)N1CC(CC(N2CC(O)C(N=[N+]=[N-])C2)=O)(OC)C1 51629,c1(OC(C)C)ccc(-c2cn(C(C)C(=O)NC3CCC3S(C)(=O)=O)nn2)c(Cl)c1 51630,N1(C(CC2CC(OC)C2)=O)CCN(C(=O)C(CN(C)C)OC)CC1CS(C)(=O)=O 51631,N1(C(CCc2ncc(C)[nH]2)=O)CCCCC(CNC(C2CCCN2C(C)C)=O)C1 51632,C1(NC(C(CC#C)NC(=O)C(C)CC2CC2)=O)CCCOC12CCC2 51633,N1(C(CCSCCC)=O)CCN(C(c2cn(C3CC3)cn2)=O)CCC1C 51634,C(C)(CC(C)C(F)F)NC(C(C)N(C(c1cc(CC)[nH]n1)=O)C)=O 51635,C1(O)(C(C)C)CCN(C(C2(NC(=O)C(C)C3CC3)CCOCC2)=O)C1 51636,CC1=C(C(=O)N2CC(CNC(c3ccccc3C(N)=O)=O)CC(C)C2)CCO1 51637,Cc1ccc2cc(C(=O)NC3CN(C(=O)COCCCF)C(C)(C)C3)[nH]c2c1 51638,C1(C(C)C)CCCC1C(=O)NCC12CC(NC(=O)CN3CCSCC3)(C1)C2 51639,N1(C(c2cnns2)=O)CCC2CN(C(C3CN4CCN3CC4)=O)C2C1 51640,C(C(C)(C)C#CC(=O)NCC(O)CCO)NC(C(CC)N(CC)CC)=O 51641,C1(C)(C(N(C2(C=C)CCOCC2)CC#CC)=O)CCN(CCN2CCCC2=O)CC1 51642,C1(C(=O)NCC2(C)CC3CC3C2)CN(C(=O)Cc2cscn2)CC1(F)F 51643,N1(C(CCc2n(C)ccn2)=O)CC2(CC(CC(=O)NCC(c3cccs3)O)C2)C1 51644,c1(OC)ccc(F)c(C(=O)NC2CC(CNC(c3cc(F)c[nH]3)=O)C2)c1OC 51645,c1(C(N(C(C)C(=O)NC(C)C(C2CCCCC2)O)CCC)=O)ccc(=NC)[nH]c1 51646,C1(C(=O)NC(CC)CCOC)CC(NC(=O)Cc2cscn2)CCO1 51647,N1(C(C2(C)COCCO2)=O)CCC2(CC(NC(c3cccc4c3CCO4)=O)C2)C1 51648,N1(CC(=O)NC2C=CCN(C(c3c(C(C)C)[nH]cc3)=O)C2)CCCCS1(=O)=O 51649,N1(C(C(C)SC)=O)CCC(C2CCCN(C(c3c(Cl)nn(C)c3Cl)=O)C2)C1 51650,C1(C)(C(=O)NCC2CN(C(c3sc(CC)c(C)c3)=O)CC2C)CCC(C)CC1 51651,C12(NC(N(OC)C)=NCC3CC3)CC3CC(C1)C(N1CCOCC(F)(F)C1)C(C3)C2 51652,N1(C(CSC2C(=O)OCC2)=O)CCC(NC(=O)Cn2cncn2)CC1 51653,CC(C)S(=O)(=O)C(C)C(=O)NCC1(O)CCCN(C(=O)CC2CC2)CC1 51654,N1(C(CCOC)=O)CCN(CC(C)(C)NC(C2CCCC(CF)C2)=O)CC1 51655,c1(C(N2C(C)CC(NC(CC(C)(C)OC)=O)C2)=O)cccc2[nH]cc(Cl)c12 51656,C(=O)(CC(O)CN(C)C)NC1(C(=O)NCc2ncn(C(C)C)n2)CC1(C)C 51657,CON1CC(C(=O)NCC2CCCC2C(=O)NCC2(C)CC2)CC1=O 51658,C(C)(CCC(=O)N(C)OC)(c1n(CCOCC)nnn1)NCCC1CC(C)(C)C1 51659,c1(N(CCNC(c2csc(C(F)(F)F)c2)=O)CC)nc(O)c2ccc(Cl)cc2n1 51660,N1(C(c2c(SC)cnn2C)=O)CC2CC(C)N(C(c3cccc(F)c3C)=O)C2C1 51661,c1(OC)ccc(NC(C2CC(NC(=O)C3=CCCOC3)C2(C)C)=O)cc1C 51662,N1(C(CC(CC)OC)=O)CC(N(C(=O)CCOC)CC)C2(CC2)C1 51663,c1(C(N2C(CNC(c3c(F)ccc(C)c3)=O)COCC2)=O)cc(C)c(C)cc1I 51664,O=C(CCCn1cc(-c2ccccc2F)nn1)NNC(=O)C1CCCS1 51665,C1(CC(=O)NCCN(C(c2n[nH]cc2OC)=O)CC)CCCC(=O)N1 51666,Cc1cc(N2CC3CC3C2)nc(=NCCc2ccc(C(F)(F)F)cn2)[nH]1 51667,C1(CC(=O)OC)(NC(=O)NC(C)CC2CCCO2)CCC1 51668,c1(CN2C(C)(COC)CCC2)cc(-c2cc(F)cc(F)c2OC)c(OC)c(Cl)c1 51669,C(CC(C(C)(C)C)NC(c1cc(OC)cs1)=O)N(C(c1cn(CC)nn1)=O)C 51670,N#CC1(C(N2CCOC(CNC(=O)CCC(N)=O)C2)=O)CC(F)(F)C1 51671,c1(C(=O)NC(C)CC(C)NC(C2CCCC2c2ccccc2)=O)ccc(O)nc1 51672,C1(C(=O)NC(CN(C(c2c(C)nc(C)[nH]2)=O)C)(C)C)CC2COCC2C1 51673,C(CC(C)CC)(C(=O)N(CC(C)(C)CO)C)NC(CC1CC(=C)C1)=O 51674,Cc1ccc(C(=O)NC2CC3C(NC(c4ccc(C5CC5)cc4)=O)C3C2)cn1 51675,C1(CN(C(=O)C(N2CC(F)(CO)C2)=O)C)CCCCC1O 51676,C1(C(C(C)OC(=O)NCc2ccccc2)C)CCCN1C(=O)CC1CC(F)(F)C1 51677,c1(CC)c(Cl)nc[nH]c1=NCC1CN(C(C2CC(=O)N2)=O)CC1C 51678,N1(C(CCCOCC)=O)CCN(C(c2cc(OC)ns2)=O)CC1C1CC1 51679,N1(C(C(C=C)(C)C)=O)CCC2(CC1)CC(NC(=O)C(CC)n1nccc1C)CO2 51680,N1(C(COCCC#C)=O)CC(C)N(C(c2cc(OC)c(C)c(OC)c2)=O)CC1C 51681,c1(CN2CCN(C(c3ccc(C)[nH]3)=O)C3C2C3)cc([N+](=O)[O-])ccc1O 51682,Cc1cccc(CC(=O)NC23CCC2CN(C(c2cnc(C(C)C)[nH]2)=O)C3)c1Cl 51683,N1(C(c2ccccc2)CCOC)CCC(S(=O)(=O)N(C)C)C1 51684,N1(C(CCC(=O)NC)=O)CC(CO)C2(C1)CN(C(c1n[nH]cc1Cl)=O)C2 51685,c1(C(=O)NC2CC2)cc2n(n1)CCCN(C(c1ccc3nc(O)oc3c1)=O)C2 51686,c1(CC(N2C(CC)C(NC(=O)CC#N)CCC2)=O)c[nH]c2cc(C)ccc12 51687,C12(CNC(C3CC(O)(CC#C)C3)=O)CCCC1N(C(=O)C(C)CSC)CCC2 51688,N1(C(c2cc(Br)cc(F)c2F)=O)CCOC2(C1)CN(C(C13CNCC1C3)=O)C2 51689,N1(C(Cc2cc(C)on2)=O)CCC(NC(c2sc(C(F)(F)F)nc2C)=O)C(F)C1 51690,C12(C(=O)NC3(C(=O)NC(C(C4CC4)OC)C)CC3)CC(C#N)(C1)C2 51691,N1(C(C(C=C)(C)O)=O)CCCC(C)(C(=O)NC2CCOC2=O)C1 51692,CCC(C(=O)NCC(C)N(C)C(C1(C#N)CC1(C)C)=O)C(C)C 51693,c1(NC(=O)CC2CN(Cc3nccc(N4CCCC4)n3)C2)cc(O)cc(O)c1 51694,c1(C(=O)NC2C(CNC(c3c(C)ncn3C)=O)C2)cc(Br)cc2c1OCC2 51695,N1(C(CCC(=C)C)=O)CCC2(CC1)CC(N=c1[nH]nc(CC)s1)CCO2 51696,Cc1ccc(NC(c2nccn2C)c2nnnn2CCN2CCOCC2)c(C)c1Br 51697,c1(C(=O)NC(CCNC(c2c(C)snc2)=O)C)nn(-c2ccccc2)cc1Br 51698,c1(C(N2CCC(CC(N)=O)C2)=O)ccc(NCCc2nc[nH]n2)cc1.CN1CC1 51699,C1(CNC(C(CC(C)C)O)=O)CN(C(c2ccccc2O)=O)CCC12CCC2 51700,c1(SC)ccc(C=CC(=O)NC2CCCCC2CNC(=O)C(C(C)O)N(C)C)s1 51701,C1(C(=O)NC2(C=C)CCC2)CCN(C(C2CCCN2CCC)=O)C1(C)C 51702,c1(CC)ccc(C(N2CCC2CNC(=O)C(C#N)=CC2CC2)=O)c(F)c1 51703,Cc1ccc(Cl)c(C(=O)NCC2CC2CNC(C2(n3ccnn3)CC2)=O)c1O 51704,CC(C)CC(C)(O)C(=O)N1CC(O)(C(C)NC(c2cc3c(s2)CCCC3)=O)C1 51705,C1(OCCNC(=O)NC(C)CC2(O)CCC2)CCCCC1 51706,c1(C(=O)NCC2CC(OC)CN2C(=O)COCC(F)(F)F)c(F)ccc(F)c1Cl 51707,C12(CNC(C3(C(=O)NC4CC4)CC3)=O)CCC(C1)N(C(=O)C(C)n1cccc1)C2 51708,C1(CC)(CC)CC(C(=O)NCC2(C(=O)NC3CCCC3C)CCCO2)C1 51709,c1(C(=O)NC(c2cn(C)nn2)C(=O)NCC(CC)N(C)C)cncc(C)n1 51710,Cc1cc(C(=O)NCC(CNC(=O)C(C)C(F)F)CO)c(Br)s1 51711,S(=O)(=O)(c1cccnc1N1CCn2cnnc2C1)N(CC(C)(C)N(C)C)C 51712,C(=O)(C1CCOc2ccccc21)N1CC(NC(=O)Cn2cccn2)CC(OC)C1 51713,C=C1CC2CCCC(C1)N2C(C1CCCN(C(c2csc(=N)[nH]2)=O)C1)=O 51714,C(=O)(C#CC1(C)CCCO1)NCC(CNC(c1cc(Cl)ns1)=O)OC 51715,c1(Sc2n(CCC)ncc2)c(Br)ccc2c1OCCO2 51716,CCCCC(O)C(=O)N1CC(CN(C)Cc2ccc(C(C)=O)s2)C2(CC2)C1 51717,C1(C(=O)NC2(CF)CCN(C(C3CCC(C)(C)C3)=O)C2)CC2(CC(=O)N2)C1 51718,N1(C(c2ncc(CC)cn2)=O)CCC2CCCC12C(N1CC2C(C1)C2(F)F)=O 51719,c1(C(=O)NC(C2CCCCN2C(=O)CC2CSC2)C)ccc(S(=O)(=O)N(C)C)cn1 51720,C1(C2CC2)(NC(c2cc(CNC(C3CCCC3)=O)[nH]n2)=O)CCCC1 51721,C(=O)(C1CC(=O)Nc2ncn(C)c21)NC1C(C)N(C(=O)C=Cc2ccsc2)CC1 51722,Cc1nn(C)c(F)c1C(N1CCC(CNC(c2ccnc(OCF)c2)=O)C1)=O 51723,CCC(CC(=O)N1CC(C)(C)CC1CC(=O)N(C)Cc1cnnn1C)CC(C)C 51724,CC(CC(=O)NCSc1ccccc1)SCCCNC1CCCC1 51725,C(CC(C)C)(C(=O)NCC1CN(C(=O)COc2cccc(C(C)C)c2)C1)OC 51726,CCCCS(=O)(=O)N1CCCC(C(=O)NCCSC2CCCCO2)C1 51727,C(=O)(C#CC1(C(F)(F)F)CC1)NCC(=O)NCC(CC)NC(c1ccncc1)=O 51728,CC1CN(C(=O)Cn2ccnn2)CCN1C(C1(C(F)(F)F)CCOCC1)=O 51729,N1(C(CC(=O)OCC)=O)CCC(CNC(C2CC(C(C)C)=NO2)=O)C1(C)C 51730,c1(C(N2CCC(NC(c3cc(C(C)C)no3)=O)C(O)C2)=O)ccc2snnc2c1 51731,N1(C(C(CCC)N(C)C)=O)CC(N(C(=O)C=Cc2cccnc2)C)C2(CC2)C1 51732,CC1(C)CC(NC(c2cnc[nH]2)=O)CN(C(=O)Cc2csc(C3CCCC3)n2)C1 51733,C12(C(N3CC(c4c(CNC(c5c(C)occ5)=O)nco4)C3)=O)COCC(C1)C2 51734,C(C(CC(C)C)C(=O)N1CCC(C)(C)C(O)C1)NC(COCCC=C)=O 51735,CCC(CCC(=O)N(C)CC1(CO)CC1)NC(=O)CC1(C)CCCCC1 51736,C(=O)(C(C)CC(F)(F)F)NCCN(C(C(CSC)(C)C)=O)C1CC1 51737,C12(NC(CCCC#N)=O)CCC(CC1)N(C(=O)CCN1CCC1)C2 51738,NS(=O)(=O)c1cc(C(=O)OCC2C3CCCCCC23)c(F)c(Br)c1 51739,c1(C(=O)NCCCOCCC(=O)NC2CCC(N(C)C)C2)cnc(N(C)C)cn1 51740,c1(C(=O)NCC(C2(NC(=O)OC)CC(O)C2)=O)cnnc(OC)c1 51741,N1(C(CCSCCC)=O)CCN(C2CCCN(C(=O)CSCCC#N)C2)C(=O)C1 51742,c1(OC)cc(C(=O)NCC(C)CNC(=O)C(=O)NCCC(N)=O)ncn1 51743,c1(C(=O)NC2CC(NC(C34CCC(F)(CC3)C4)=O)C2)c[nH]c2ncc(Br)cc12 51744,C(c1ncc(C)[nH]1)=CC(N1C(CN(C(C2CCC2(OC)OC)=O)CC)CCC1)=O 51745,Cc1cc(=O)c(C(=O)NCc2ncsn2)nn1-c1cccc(Cl)c1 51746,C1(NC(C(C)(C)OC)=O)CN(C(c2cn(C)nc2C2CC2)=O)CC1C 51747,C(CCO)(C(F)(F)F)NC(C(CC1CCC1)NC(=O)COCC1CC1)=O 51748,CCCCC(C(=O)N1CCN(C(=O)CSC)CC1c1ccccc1)NC(N)=O 51749,c1(C(N(CCN(C(=O)CSCC(F)F)C(C)C)C)=O)cnn2cccc(Cl)c12 51750,N1(C(C2=C(C)CC2)=O)C(CC(N2CC3CCCCC23)=O)C2CCCC12 51751,c1(NS(=O)(=O)c2sccc2C2OCCO2)nc(C)cc(C)c1CN(C)CC 51752,c1(CC(=O)NCCC2CC(NC(CCc3ccc(C)s3)=O)C2)cn(C)nc1C 51753,c1(C(N2CCCC2CC(=O)OC)C(=O)NCCC)csc(C)n1.c1(CN)ccco1 51754,N1(c2n(CC3(CC)CC3)c(C3CCCC3)nn2)CCN(C)C2(CCOC2)C1 51755,C=CCC(Cc1ccccc1)C(=O)NC1CCCC1NC(=O)CC(F)F 51756,c1(C(N(C)CC2CN(C(c3c(C)csc3)=O)CC23CC3)=O)ccc(S(C)(=O)=O)o1 51757,N1(C(C(C)OCCOC)=O)CCN(C(c2ccon2)=O)C(C(F)F)C1 51758,c1(C(N2CC3C(CNC(C4(C)CCN(C)C4)=O)(C3)C2)=O)cc(F)ccc1C1CC1 51759,S(=O)(=O)(c1ccc(F)cc1O)NC(c1cnn(C)c1C1CC1)=O 51760,C1(NC(c2cc(F)n[nH]2)=O)CC(NC(C2CC(CF)C2)=O)C12CCC2 51761,C(C(=O)NC(C)CCNC(=O)C(C)Sc1ccccc1)(C(C)C)NC(C)=O 51762,CC1C(=O)N(CC(=O)NC2(CNC(=O)Cc3nncs3)CCC2)C(=O)C1C 51763,C#CCCCCC(=O)NC1CCC(N(C)C(c2ccnnc2NC)=O)CC1 51764,N1(CC)CC(C(=O)NC2CCCN(C(C34COC(CCO3)C4)=O)CC2)CCC1=O 51765,n1(CC(=O)NC(C)CC(C)NC(C2CCC(=O)C2)=O)ncccc1=O 51766,C(C(C)(C)C(F)F)NC(C(C1CCN(C(=O)C=Cc2ccccc2)C1)C)=O 51767,c1(C(=O)NCC(CNC(Cn2c(C)ncc2)=O)CO)cc(C(F)(F)F)cc(N)c1 51768,c1(CCC(=O)NCC(=O)N(CC(=O)NC)C)nc2ccccc2o1 51769,N1(C(C(C)N(C)C)=O)CCC(CNC(=O)C(C)CC(N)=O)C12CCC2 51770,c1(OC)ncccc1C(=O)NC(C)(C)CN(C(=O)Cn1ccc(C)n1)C 51771,c1(C(=O)NCC(C2CCCCC2)NC(CC(C)SC)=O)cc2n(n1)CCCN2 51772,c1(C(=O)NCCNC(COC2(C)CCOCC2)=O)ccc2sc(O)nc2c1 51773,C1(NC(C(C)NC(c2ccco2)=O)=O)(CNC(=O)C(C)O)CC2CCC1CC2 51774,Cc1cc(C(C)C(=O)N2CC(CNC(c3nc(C(C)(F)F)cs3)=O)C2)c(C)o1 51775,C1(NC(=O)Cc2ccc(Cl)cc2F)CN(C(=O)CC2CCOC2=O)CC1C1CC1 51776,c1(CC)nc(C)[nH]c1C(=O)NC(CNC(=O)C(C(C)C)SC)CC(C)C 51777,CC(C)(C(=O)NCC1CCCN(C(=O)CCOCC(F)(F)C(F)F)C1)C(F)(F)F 51778,C(N=c1ncc(CCOC)c[nH]1)C1CCC(C(C)OC)CC1 51779,N1(C(C(CC)CC)=O)CC2CCCC(N(C(=O)C(COC)N(C)C)C)C2C1 51780,c1(C(N2CC(NC(C(C(C)O)C)=O)C(C)CC2)=O)ccc2ncccc2n1 51781,c1(OC)ncnc(OC)c1CN1CCCC1CC(=O)Nc1sccc1CO 51782,CN1CCN(C(=O)C(N2CCOC(c3ccc(F)cc3F)C2)=O)CC1C(C)(C)C 51783,CCCCCC(=O)NN(CCNC(=O)C(C(C)C)Oc1ccc(Cl)cc1)C(C)=O 51784,C1(NC(COCC)=O)CCCN(C(C2C(c3cccc(Br)c3)C2(C)C)=O)C1 51785,CC(CC(=O)N1CCCC1C(=O)N=c1cc[nH]cc1C(=O)O)CC(C)(C)C 51786,C1(NC(c2c(C)nn[nH]2)=O)CCC2CC1CN2C(=O)CCCCCC#N 51787,c1(OC)cccc2c(C(N3CC(NC(c4[nH]nnc4C)=O)C(C)C3)=O)coc12 51788,C1(C(=O)NCc2ccc(C(N(CCC(N)=O)CC)=O)s2)CCCCCN1C 51789,C1(NC(c2c(C)ccs2)=O)CCCCN(C(c2cnc(C(C)(F)F)s2)=O)C1 51790,C1(NC(c2c(CC)n[nH]c2)=O)CC2(CNC(=O)CCC3CCOCC3)CC1CO2 51791,N#Cc1cc(C(=O)NC2(CNC(c3scnc3Br)=O)CCC2)co1 51792,c1(CNC(=O)NC2CCC3CCCC23)cccc(Br)c1F 51793,C(=O)(C1=CCC(F)(F)CC1)N1CCC(C2(NC(c3cc(C)no3)=O)CC2)C1 51794,C#CCCC(=O)NCCn1ccc(C(=O)NCC2(SC)CC2)c1 51795,C1(CCNC(C=CCOCCOC)=O)CC(NC(=O)COCCCC)C1(C)C 51796,c1(NC(C2C(C=C)OCC2)=O)c(OC(c2nc(OC)cn2C)=O)cccc1C 51797,c1(C(CNC(CCC)=O)=O)c(O)nc(=O)n(CC2CCCN(CCNC)C2)c1N 51798,C(=O)(CS(=O)c1ccc(Cl)cc1)N1CCC(N(C(C=CC(C)(C)SC)=O)C)C1 51799,C1(C(N(C)CCN(C)C(C2CC3(CCOC3)C2)=O)=O)CCS(=O)(=O)C1(C)C 51800,N1(C(C(=O)NCC=C)C(C)C)CCOC(C)(C(F)(F)F)C1 51801,C(C(F)(C(=O)NCC1CCCCO1)C(C)C)NC(c1c(C)nsc1C)=O 51802,CCC(CCC(=O)NC1CC2(C1)CC2NC(=O)CCCNC(N)=O)OC 51803,N1(C(C=Cc2n(C)cnc2)=O)CCC2CCC(C1)N2C(=O)CC1(C)CC1 51804,C12(C(=O)NCCC(C)S(N)(=O)=O)CCC(CC1=O)C2(C)C 51805,C1(n2cc(C(=O)NCC3(O)CC(CO)C3)nn2)CCCN(C(=O)C(F)(F)CO)C1 51806,CCC(CC(=O)NC(C)CCCn1ccnc1)NC(=O)COc1ccc(O)cc1 51807,C12(CNC(CCc3onc(CSC)n3)=O)CCCN(C(=O)COC(C)C)C1C2 51808,c1(C(N(CC)CC2CCCN2C(=O)COc2ccc(OC)cc2)=O)cnc(Cl)c(N)c1 51809,C1(NC(C)=O)CN(C(=O)CCc2cc(Cl)cc(Cl)c2)CC12CC2 51810,c1(C(N2CCC(C)C2C)C(=O)NC(CC)(C)C)nn(C)cc1Cl 51811,c1(NC(C2(C)CCN(C(c3n[nH]c(CC)c3F)=O)C2)=O)ncc(C)cc1Br 51812,CCCCCC(O)C(C)C(=O)N1CCCC(CCNC(c2ccoc2Cl)=O)C1 51813,c1(C(=O)NCCC23C(CN(C(C4C(C)C4)=O)C2)CC3)cc2c(Cl)c(Cl)ccc2[nH]1 51814,CCCC(CC)C(=O)NC(CC(=O)NCC1(C#N)CCC1)C(C)OC 51815,n1(CC(=C)C)nc(-c2ccc(Cl)s2)nc1CC1CCC(F)(F)C1 51816,c1(C(N2CCC(C(CC)CC)C2)C(=O)NCC)cc(F)cc([N+](=O)[O-])c1 51817,Cc1cnn(CCC(=O)NCC(O)CNC(c2csc(Cl)c2)=O)c1 51818,C12(C(=O)NCC(C)NC(c3cncn3C)=O)CC(CCO1)C2 51819,C1(CNC(C(c2cnn(C)c2)C)=O)COC(C)(C)CN1C(c1ccoc1C)=O 51820,c1(OC)cc(-c2nc(-c3cccc(C)c3)nn2CC(C)(C)C)ncn1 51821,C12(CC(N3CC(C)C(C)(C(=O)NOCC(C)(C)O)C3)=O)CC3CC(CC(C3)C1)C2 51822,c1(C(=O)NCC(CNC(CC(CC)OC)=O)CO)ccc2c(c1)nc(O)n2C 51823,c1(CC(N2CC3CC(CNC(C4(CC5CC5)CC4)=O)C2C3)=O)c(Cl)cccc1Cl 51824,Cc1cc(CNC(=O)CC(C)NC(c2ccccn2)=O)cc(C#N)c1 51825,c1(CN(C(=O)C(C)OC2COC2)CCNC(CC=CC)=O)ccccc1 51826,N1(C(c2nc(C)nn2C)=O)CCC2(CC1)CC2CNC(=O)CC(C)C1CC1 51827,C=C=CC(C)C(=O)NCC(C)C(=O)NCCCN(CC(C)C)C 51828,c1(-c2c(F)ccc(-c3n(CCCC(C)C)ccn3)c2)cccc([N+](=O)[O-])c1 51829,CC(CCCNC(=O)CCc1cnoc1)NC(=O)CSc1nncs1 51830,C1(NC(C2C(CC)C2)=O)CC2CC(NC(c3cc(COC)on3)=O)CC12.[nH]1cccn1 51831,c1(CCC(=O)NC23CC2CN(C(c2ccoc2Cl)=O)C3)nnc(O)nc1O 51832,Cc1ccc(O)cc1C(N1CCC(NC(=O)C=C2CCN(C)C2)C(F)C1)=O 51833,C#CC1(C(=O)NCC2CC(n3cccn3)C2)CCN(C(=O)C(CSC)OC)C1 51834,c1(C(N2CC(CC(=O)NCc3n(CC)ncn3)C2)=O)cc2cccnc2[nH]1 51835,N1(C(c2ccc(C)nc2)=O)CCC2C(CCCN2C(c2c[nH]cc2C2CC2)=O)C1 51836,CC(C)(C)C(O)C(=O)NC1CCN(C(=O)CCc2cccs2)CC1O 51837,c1(OCC)c(C)[nH]c2ccc(OCC3CC3)cc12.C12C(C1C1CNC1)C(=O)N2 51838,CCC(CC(=O)NCCOCCNC(C1CC2(CCC2)CO1)=O)CC(C)C 51839,N1(C(C2(C(N(C)C)=O)CC2)=O)CC(NC(c2ccn(C(F)(F)F)n2)=O)CC(F)C1 51840,Cc1cnccc1-c1cn(CCCN(C(=O)CC2CC3C=CC2C3)C2CC2)nn1 51841,C#Cc1cccc(OCC(=O)NC2CCOCC2NC(=O)CC(=O)N(C)C)c1 51842,c1(C(N2CC(CN(C)C(C3CCCS3)=O)C2)=O)csc2nccn12 51843,C(C1=CCN(C(c2cc(CCCO)on2)=O)CC1)NC(=O)C(F)=CC1CC1 51844,C1(CC=C)(C(=O)NC(CSC)CCOC)CCCN1C(c1cccs1)=O 51845,C1(NC(c2cc(C)nc(C)c2)=O)CN(C(c2cnn(C)c2)=O)CC(C)(C)C1 51846,C(C(C)(C(=O)N1CC2C(C)C2C1)NC(c1cccc(CC#N)c1)=O)SC 51847,c1(C(=O)NCCc2c(C)cc(Cl)cc2)nc2ccc(Br)cn2c1F 51848,C(CC(C)C)(C(=O)NCC1CCCN(C(=O)Cc2cocn2)CC1)OC 51849,C1(CC)CN(C(C2(C)C=CCC2)=O)CCN1C(=O)COc1cc(C)on1 51850,C12(C(N(C3CCCCC3)C(CC)C)=O)CC(CN(C(c3cnccc3C)=O)C1)C2 51851,N1(C(C2C(CNC(C3CC4(CCC4)C3)=O)CCO2)=O)CCC(=C(F)F)CC1 51852,C=CCCC(C(=O)Nc1cn(C)nc1OCC)NC(=O)Cc1ccccc1F 51853,Nc1ccc(O)c(C(=O)NCC(c2ccccc2OC(F)(F)F)n2ccnc2)c1 51854,Cc1ncnc(N2CCC(CNC(=O)COC(F)(F)F)C2)c1Br 51855,c1(C(=O)NC(CC)(C)CNC(=O)COCP(C)(C)=O)ccc(Br)cc1 51856,N(C(=NCC(C)C)N1CCC(CC(C)C)C1)CC(c1ccc(F)cc1)OC 51857,c1(C(N2CC(OC)(CNC(=O)C3=C(Cl)CC3)C2)=O)c(C)nc2cccnn12 51858,c1(OC)cncc(C(=O)NC2CN(C(=O)CC(C)SC)CC2SC)n1 51859,C(=O)(CC(C)CNC(=O)CC1CCOC1=O)N(C(C)C(=O)NC)CC 51860,N1(CC(N2CC(c3n(C)ccn3)C(NC(=O)CNC=O)C2)=O)CCC(=O)NC1=O 51861,N1(C(c2ncc(N(C)C)nc2)=O)CCN(C(C2(F)CC2)=O)C2CS(=O)(=O)CC12 51862,C(C(C(C)C(C)C)NC(=O)Cn1ccc(C)cc1=O)NC(C)=O 51863,C1(C(=O)NC(C)CN(C)C(c2cn(C)nc2C2CCCO2)=O)CN2CCC1CC2 51864,n1(CC(=O)NCCN(CCC)C(C2CCC(=O)C2)=O)c(C)c(C)sc1=O 51865,C1(CNC(CNC(=O)OC)=O)CCCN(C(C2CCC(C)(C)C2)=O)C1 51866,C12(CNC(c3cc(C)sn3)=O)CC3CC(CC(C3)C1NC(C1CNC(=O)C1)=O)C2 51867,CC(CN=c1[nH]nco1)(C1CC1)NC(c1cc(S(N)(=O)=O)co1)=O 51868,CCC(CC)C(=O)NCc1nnn(C)c1C(N1CCCCC1C1CC1)=O 51869,C1(C(=O)NC(C2N(C(CCC(=O)NC)=O)CCCC2)C)C2(CCC2)C12CCC2 51870,C(=O)(C(C)N(CC(C)NC(=O)C(C)C1CC1)C)N(C1CC1)CC 51871,n1(CCC)nc(C)cc1C(=O)N(C)CCN(C(=O)C(C1CC1)OC)C 51872,C1(NC(Cn2c(C)ccc2C)=O)CCN(C(C2CC(=C(F)F)C2)=O)CC1C 51873,N(C1CCCn2ncnc21)C(C(C)(N(C(COC)=O)C)C1CC1)=O 51874,c1(C(=O)NCC(CNC(C(C)OCC)=O)OC)cc(Cl)c(Br)cc1C 51875,C(=O)(CC1=CCOCC1)NCC(CC)NC(C1CC(C)(C)OC1(C)C)=O 51876,N1(C(C(CC(C)=O)(C)C)=O)CCC2(CCCN2C(=O)CC2CCCC2C)C1 51877,N1(C(C=CC(=O)OCC)=O)CCCC2CCN(C(c3n[nH]c(C4CC4)n3)=O)CC12 51878,N1(C(=O)Cc2ccccc2)CC2CC(C1)N2C(=O)C(F)C1CCOC1 51879,C(C(C)(C)CC(=O)NC1CCOCC1NC(=O)CSCC(F)(F)F)OC 51880,C(C(C(=O)Nc1cnn(CCF)c1)C(C)(C)C)NC(c1c(C)n[nH]c1C)=O 51881,c1(NC(C)C)ncc(Br)c(C(=O)NCCOCc2ccccc2F)n1 51882,N1(C(C(N2C(=O)CCC2=O)C)=O)CC2CN(C(C3C(C)(C)C3(C)C)=O)CC2C1 51883,c1(C(N2C(C(=O)NCC(CCC)C)CCCC2)=O)cc(C)cc(F)c1 51884,Cc1nc(CC(=O)NC2C=CCC(C(=O)NC(CC3CC3)CO)C2)[nH]c1C 51885,CC1(C)CCC(C(=O)NCC2CN(C3CC3)C2)(NC(c2cc([N+](=O)[O-])n[nH]2)=O)C1 51886,N1(C(C(C)(C)C2CCCCO2)=O)CCC12CN(C(=O)CCSc1ccccn1)C2 51887,C1(C(=O)NCCOCCCNC(c2ncsc2C2CC2)=O)CCC(C2CC2)C1 51888,C1(C(=O)NCC(CC)NC(=O)CCCCOC(C)C)COC2CCCCC12 51889,N1(C(c2c(OCC(=O)OC)cccc2)=O)CC2CC1CN2C(C1CCOC1=O)=O 51890,c1(C(=O)NC(C)CNC(=O)CN2CCSCC2)ccc(SCc2cnc[nH]2)cc1 51891,N1(C(C2N(C(c3c(CC)cno3)=O)CC=CC2)=O)CCCC(O)(C(N)=O)C1 51892,c1(OC)c(C)ccc(C(=O)NC2COCCC2NC(=O)CCc2cnoc2)c1F 51893,CC1CCCc2ncc(C(=O)NC3CC34CCN(C(=O)Cc3cnoc3)CC4)n21 51894,C1(CC)(NC(c2ccn(C)c2)=O)CCCN(C(C2CCCN(CC(C)C)C2)=O)C1 51895,C12(CNC(C3(C#C)CCC3)=O)CCC(CC1)N(C(c1ccoc1)=O)C2 51896,c1(C(C)NC(c2n(CC)nnn2)c2conc2COC2CC2)ccccc1OC 51897,C1(C(N(CCN(C(c2cnn(CCF)c2)=O)CC)CC)=O)CC(NC)CCO1 51898,S(=O)(=O)(c1ccc2ccccc2c1)N1CCN(C(C(C(CC)C)O)=O)C(C)C1 51899,c1(C(=O)NC2CN(C(C(c3ccccc3)OC)=O)CC2C)nccc2cc[nH]c12 51900,C1(CC(=O)NCCc2ccccc2O)CN(C(c2cccnc2)=O)CC12CC2 51901,c1(-n2cc(C3N(C(C4(C5CCCO5)CC4)=O)CCC3)nn2)cccc(Br)c1 51902,N1(C(CC2(COC)CCCC2)=O)CC2CCN(C(=O)Cc3csc(C)n3)CC12 51903,Cc1ccc(C(N2CCC(CN(C)C(C3COCCO3)=O)C2)=O)cc1CO 51904,N1(C(CCCCCCC)=O)CCN(C(C2CCc3cncn3C2)=O)CC2(CC2)C1 51905,CCC(CCC(=O)OCCOC)N(C)OC 51906,C1(NC(c2ncn(CC)c2)=O)CCC(N(C(=O)COc2cn[nH]c2)C)CC1 51907,C1(C(=O)NCCN(C(=O)C(F)C2CCOC2)CCOC)CCC=CCCC1 51908,Cc1cccc(C(=O)NC(CNC(=O)CN2CCOCC2=O)C(C)C)c1F 51909,c1(NC(CC2OCCN(C(C3C(C(=O)OCC)C3)=O)C2)=O)ccc(C)nc1C 51910,c1(C(=O)OC)cc(N2CCC(C(C)O)C2)c2cccc(Br)c2n1 51911,Cc1csc(C(N2CCCCC2C(C)(C)CNC(c2ccnnc2C)=O)=O)c1C 51912,CC(N=c1nn[nH]n1C)C1CCCCN1C(c1c(Cl)cnn1C)=O 51913,N1(C(CC(C=C)C)=O)CC2CC(C1)C(CO)C2NC(=O)CCSc1nccn1C 51914,N1(C(C(C=C=C)C)=O)CCC(CC(=O)NCC(C2CCCC2)C)C1(C)C 51915,CCC(CC(=O)N(CCCN(C)C(C1CCC(C(=O)OCC)CC1)=O)C)OC 51916,CN1CCC(N(C(c2cc(Br)cs2)C(=O)NC2CCOCC2)C)C1 51917,N1(CC(c2nccs2)=O)CC(n2cc(C(c3ccccc3)O)nn2)C(O)C1 51918,C1(C(=O)NC2CC(CCNC(c3ncncc3Cl)=O)C2)CC2(CCCCC2)CO1 51919,c1(OC)ccsc1C(=O)NCC1CCCC1C(=O)NOCc1nc[nH]n1 51920,c1(C(N2CC(CNC(C3CCC34CCC4)=O)C2)=O)cccc(C#CCO)c1 51921,c1(C(=O)NCC2C(C)CCN(C(=O)CSC(C)(C)C)C2)cc2ccccn2n1 51922,C1(NC(c2cc(CCC)[nH]n2)=O)CCN(C(C2OC3CCC2CC3)=O)CC(O)C1 51923,C1(CNC(C=CSC)=O)CCN(C(=O)CCc2ccccn2)CC1(F)F 51924,c1(C(=O)NC(c2ccccc2F)CNC(CC2CC(C)(C)C2)=O)nccnc1O 51925,CC1CC(C(N2CCN(C(=O)CCNc3ncccn3)CC2)=O)CC(=O)N1 51926,N1(C(CC(C)(C)OC)=O)CCC2CCCC12C(N1CC2C=CC1CC2)=O 51927,C1(NC(=O)CC2CC=CCC2)CCC2(CC1)CCN(c1nc3ccccc3o1)C2 51928,c1(C(N2CCOCC(CNC(COCC=C)=O)C2)=O)ncc2ccccn12 51929,CC1(C(N2CC3(CCC3NC(c3ccccc3F)=O)C2)=O)CCCCCC1 51930,CC(C)C(N=c1[nH]nc(CC(F)(F)F)s1)C(C)NC(C1CCS(=O)(=O)C1)=O 51931,C1(CNC(Cc2c(C)nc(C)s2)=O)CC2(CO1)CN(C(=O)C(C)CS(C)(=O)=O)C2 51932,N1(C(C=Cc2ccc(C)s2)=O)CCCCCC1CNC(=O)CC1CC=CCN1C 51933,CCCC(O)CC(=O)N(CCNC(=O)C(F)C(C)(C)O)CCOC 51934,C=CCN=c1ccc(S(=O)(=O)N2CCCCC2c2ncc(Br)cn2)c[nH]1 51935,N1(C(c2cc(OC)ncn2)=O)CC(NC(=O)COC(F)(F)F)CC1(C)C 51936,C1(CC(=O)OCC2(C)CCCC2O)(NC(=O)OC(C)(C)C)CCCCC1 51937,CCC(CNC(c1cc(C#N)oc1C)=O)(CC)C(=O)NC12CCCCC1C2 51938,CCCCCCC(F)C(=O)N1CCCC(NC(c2ccc(Cl)nc2O)=O)C1 51939,Cc1ccc(C)c(C(=O)NC2CCCC2(C)NC(=O)CC2CCCO2)n1 51940,C(=O)(C1=CS(=O)(=O)CCC1)NC1CN(C(Cc2n[nH]c(=NC)s2)=O)C(C)C1 51941,N1(C(CSc2ccc(C)cc2C)=O)CC(CNC(=O)CC#N)C2(CCC2)C1 51942,C1(NC(c2nccc(C)c2)=O)CCN(C(c2cc(CO)c(C)o2)=O)CC1O 51943,C(C(=O)NC(C(=O)N(C)CC1CCOC1C)C1CCOC1)(C(C)(C)C)OC 51944,N1(C(C(C)=CC=C)=O)CCC(C(=O)NCc2ncsn2)=C(F)C1 51945,c1(C(N(C(C)C(=O)N(CCC(=O)NC2CC2)C)CCC)=O)cnc(C)o1 51946,C(C(C)(C1CC1)NC(=O)CNS(C)(=O)=O)NC(COC(CC)C)=O 51947,c1(COC)csc(C(C(=O)NC(C)(C)C)N(C2(c3cc[nH]n3)CC2)C)c1 51948,Cc1cc(C)n(CCC(N2CC3CC2C3NC(c2ccc(C(F)F)cn2)=O)=O)n1 51949,c1(N(C2C(C(C)C)CCC2)C(N2CCCC2C2CCCOC2)=O)ncccc1O 51950,C1(NC(N(c2ccsn2)C)=O)CC(F)(F)CC1NC(c1cocn1)=O 51951,Cc1cc(C(=O)NCCNC(c2ccccc2Cl)=O)ccc1-c1ccncc1 51952,C#CC1CC2CCC1N(C(=O)C=CC(C1CC1)NC(=O)CSCCOC)C2 51953,Cc1nsc(CNC(c2nnnn2CCN2CCOCC2)C2CC=CC2)n1 51954,C1(CC)(CO)CCCN(C(=O)C(=O)NCCOCCS)C1.c1(O)ccccc1 51955,C1(CN(C(c2c(C(C)C)noc2)=O)C)COCCN1C(=O)C=Cc1ccncc1 51956,c1(CC)nc(C)c(C(=O)NC(C)CCN(C(=O)COCC2CCCO2)C)s1 51957,C(C1COc2ccccc21)NC(NC(c1cccs1)C)=NCCF 51958,C(=O)(CCS(=O)(=O)N(C)C)N1C(C)(CNC(Cc2nnc(C)s2)=O)CCC1 51959,c1(OC)ccc2c(c1)CC(C(=O)NC1CCCC13CCC3)O2 51960,CCCC(C)(O)C(=O)N1CC(NC(c2ccc(CC)c(F)c2)=O)C1 51961,C1(C(=O)NC2CC(CCNC(c3cc(C4CCC4)no3)=O)C2)CC2(C1)OCCO2 51962,C12(C(N(CCNC(c3nn(CC)nc3C)=O)C)=O)CCC(C(F)F)(CC1)C2 51963,c1(C(=O)NCC=CCNC(c2occ(C)c2C)=O)c(O)cc(=O)n2c1CCCC2 51964,N1(C(C(C)SCC)=O)CCC(C(=O)NOCCCCC2CC2)C(C)C1 51965,c1(C(N2CC(F)(C(=O)NCC3(CCO)CCC3)C2)=O)ncccc1Cl 51966,CC1COc2c(C(=O)NCCn3cc(CCO)nn3)cnn2C1 51967,C1(CNC(c2cnc(COC)s2)=O)CN(C(=O)CC2C=CCC2)CC1O 51968,c1(C(=O)NC2CC(CCNC(=O)C(Cl)=CCl)C2)cccc(C(F)(F)F)n1 51969,C(=O)(CCCCCC(C)C)N(C)CC1N(C(c2c(C)ccc(Cl)c2)=O)CC(F)C1 51970,c1(CNC(=O)NCc2cc(-c3cccc(Br)c3)no2)ccc2c(c1)OCCO2 51971,C1(CN(C(C2CCOC2)=O)CC)CCCN1C(C1C=CCS1)=O 51972,N1(C(C(c2cccc(O)c2)C)=O)CCC(F)(F)C(CNC(=O)CCF)C1 51973,N1(C(C=NOC)=O)CCC(N(C(C2CC2OC(C)(C)C)=O)CC2CC2)CC1 51974,CCC(C(=O)N1CCN(C(c2ccnnc2O)=O)C(CO)C1)C(C)(C)CC 51975,CC1(C=CC(=O)N(C2CCCN(C(=O)CC3CC34CC4)C2)CCO)CCOCC1 51976,S(=O)(=O)(CCCCS(N)(=O)=O)N1CCCC(C(C)(O)CN)C1 51977,C(=O)(C(C)C(O)CC)N(C1CCN(C(N2CCC(N)C2)=O)CC1)CC(C)C.CCO 51978,C(=O)(C(F)(CNC(c1ccccc1C1CC1)=O)C(C)C)N(CC=C)CC 51979,C1(C(=O)NC(CC)CC(F)(F)F)CCC2(CN(C(=O)CCc3sc(O)nc3O)C2)O1 51980,c1(-n2c(COCC(C)C)nc(-c3cnccn3)n2)ccc(Cl)c(Cl)c1 51981,CCC(CC)C(C(=O)NC1(C(=O)NCC(C)CC2CC2)CSC1)OC 51982,C(N=c1[nH]cnc(NCc2ccc(Cl)c(F)c2F)c1C)c1cc(CC)no1 51983,c1(CC)nc2c(C(=O)NCC(C)(CO)NC(=O)C(C)C3CC3)ccnc2[nH]1 51984,CC1(C)CC(c2nn[nH]n2)CN(C(C2CC(F)CN2)=O)C1 51985,CCC(CC)CCC(=O)N(C1CCCN(C(=O)CCCN2CCOCC2)C1)CC 51986,Cc1nnc2c(C(N3CCCOC(CNC(=O)C(C)(C)C)C3)=O)cccn12 51987,C1(C(C(=O)NC(c2cccnc2)C(=O)N(C2(CC)CC2)C)C)CCOCC1 51988,c1(OC(C)C)cncc(C(=O)NCCCC(C)(C)NC(c2ccco2)=O)c1 51989,c1(OC)cc(Cl)c(Br)cc1CN=c1[nH]c(-c2cccnc2C)cs1 51990,c1(C(=O)NCCC2N(C(C3C(CC)C3)=O)CCC2)cc2c(nc1O)CCOC2 51991,N1(C(C=CC=CC)=O)CCC2(C(=O)NCc3cnccc3C)CCCC12 51992,C(c1ccnn1C)=CC(=O)NC(C(=O)NC(c1n(CC)ncc1)C)c1ccoc1 51993,CCCC(C(=O)NCC(CNC(=O)Cn1cnccc1=O)OC)c1ccccc1 51994,C1(C(=O)NCC(CSC)OC)CCC(O)CN1C(=O)Cc1nocc1C 51995,N1(C(C2N(CC)CCC2)=O)CC2CC(C(=O)NCc3cc(C)sc3C)(C2)C1 51996,C1(NC(c2cc(OC)n(C)n2)=O)CN(C(=O)CC2CCCS2(=O)=O)CCC1CO 51997,CC1CCN(C(c2ccccc2C2CC2(F)F)=O)CC1NC(C1CCCS1)=O 51998,c1(CN(C)C(=O)NCc2cncc(Cl)c2)nc2c(s1)CCCC2 51999,c1(COC)ccc(C(N2CC(NC(=O)CC3COC(=O)C3)CC2C)=O)cc1 52000,c1(C(N2CCSC2c2ccco2)=O)cccnc1NC(=O)C1CC1 52001,CC(CC(F)F)C(=O)NC1COCC1CNC(c1ccc(C(=O)CF)cc1)=O 52002,C12(C(N3CCCC(CCC(=O)N(C)CCC4CCCC4)C3)=O)CCCC1C2(F)F 52003,n1(CC(=O)NC(c2ccccn2)(C)C)cc(C#N)c(O)nc1=O 52004,C(=O)(C(C)(C)C(c1ccccc1)NC(C1CC(=O)N(O)C1)=O)OC 52005,Cc1c(C(=O)N(CCNC(C2CC(C(C)C)C2)=O)C(C)C)sc2ccc(F)cc12 52006,C(=O)(C(C)(C)C(=O)NCC(O)CN(C(=O)CCn1cc[nH]c(=O)c1=O)C)OC 52007,C1(CC=C)(NC(C2CC2(C)C)=O)CCN(C(=O)Cc2c[nH]ccc2=O)C1 52008,C1(F)(C(=O)NCCC2CN(C(C3N(CC)C(=O)CC3)=O)CC2C)CC2(CCC2)C1 52009,c1(CC(=O)NCC2CC(NC(CCP(C)(C)=O)=O)C2)ccc2nsnc2c1 52010,c1(C(N2CC3C(NC(C(C)S(N)(=O)=O)=O)(C3)C2)=O)cccc2cc(O)ccc12 52011,N1(C(CCCCC)=O)CCN(C(=O)COC2CCCCC2)CC1CC(F)F 52012,CC1(C)CCC=C1C(=O)OCn1ccc(=O)n(Cc2ccccc2)c1=O.C1CO1 52013,C(=O)(CCCCCCCCCO)NCC1C(C)(C)CN(C(C2C=CCCC2)=O)C1 52014,Cc1nc(N2CCC(NC(=O)C(C3CC3)C3CC3)CC2C)cc(C#N)n1 52015,c1(SCC(N2CC3C(CN(C(=O)COCCF)C)C3C2)=O)ccc2c(c1)OCCO2 52016,C1(O)(CNC(C(CCOC)OC)=O)CCCN(C(=O)Cc2cnc(C)s2)CC1 52017,c1(CCC(=O)NCC=CCNC(=O)CCCCC2CC2)c[nH]c2ncccc12 52018,c1(C(=O)NCC2C(NC(COCC)=O)C2)cc(OC)c(OC)cc1N 52019,N1(C(c2cc(C)cc(OC)c2N)=O)CC2CC(C1)CN(C(C1CC1OC)=O)C2 52020,CCCCCC(O)C(=O)N1CCCC1Cn1cc(CNC(C2(F)CC2)=O)nn1 52021,N1(C(CC=CCC)=O)CCOC2(CCN(Cc3ccc(F)c(O)c3F)CC2)C1 52022,c1(CN2CCC3(C(NC(Cc4cn(CC)nc4)=O)C3)C2)cn2ccccc2n1 52023,N1(C(CC2C(CC)C2(F)F)=O)CCC(NC(C2(C)CC2(F)F)=O)CC(O)C1 52024,CCC(O)CC(=O)NCC1CCC(NC(=O)CC2CSC2)CC1 52025,CCCC(CCCNC(c1ccc(=O)n(C)c1)=O)NC(c1sc(C)cc1C)=O 52026,c1(C(N(CC(C)NC(c2cc(CC)[nH]n2)=O)C)=O)ccc2cnsc2c1 52027,N1(CCN(C(=O)CCc2ccc(CO)cc2)C)CCN(C(=O)CC2(C)CC2)CC1 52028,c1(C(=O)NC(CC)(CNC(C2CCC(=O)O2)=O)CC)cc2ccc(Cl)cc2o1 52029,C(=O)(C1CCCn2ncnc21)NC(C(C)C)CNC(=O)CCC(N)=O 52030,CC(C)(CO)C(=O)NC1(C)CCN(C(=O)COc2cccc(Br)c2)C1 52031,N1(C(C(C)Cc2ccc(Cl)cc2)=O)CC(NC(C2(O)CC2)=O)Cc2ccccc21 52032,C1(C(N(C2CC(NC(Cn3c(C)cc(C)n3)=O)C2)C)=O)CCn2ncnc2C1 52033,C1(COC)(CNC(=O)C(C)n2cccn2)CCCN1C(C1CC(CCO)C1)=O 52034,N1(C(Cc2c(Br)cn(CC)n2)=O)CC(C2(NC(=O)C3=CCCS3)CC2)C1 52035,CC1CCOCC1C(=O)NCC1(NC(c2cccc(N(C)C)n2)=O)CCC1C 52036,C=CC1(CNC(C2(C)CC(O)CN2C(=O)C(C)c2cccs2)=O)CCOCC1 52037,C1(C(N2CCC(NC(=O)CCCCCF)C2)=O)(COC)CCCNS1(=O)=O 52038,C1(C2(O)CCC2)(C(=O)NCCCCNC(c2cnc(CCCC)s2)=O)CC1 52039,n1(CC(=O)NCCc2ncc(C(=O)O)s2)cc(C(O)C2CC2)nn1 52040,C1(COC)CC(O)CN1C(C1COCCC1NC(c1cc(Cl)n[nH]1)=O)=O 52041,C1(C(N2CC(NC(C=C(C)C(F)F)=O)C3(C2)CC3)=O)CCOCC12CCCCC2 52042,N1(C(c2c(C)nc(C3CC3)s2)=O)CCC(CNC(c2ccc(Cl)nn2)=O)C(C)C1 52043,C(=O)(C1CCCc2ncnn21)N1CCN(C(c2[nH]nnc2C2CC2)=O)CC(C)C1 52044,N1(C(c2c(C)c[nH]n2)=O)CCC(O)C(C(=O)NCc2ccccn2)C1 52045,c1(OC)ncc(CNC(=O)C(C2CCC(=O)N2)C)s1 52046,Cc1cc(C(=O)NC23CCCN(C(c4ccsn4)=O)C2C3)ccc1Br 52047,c1(COc2ccc(CNC)cc2)ccc2c(c1)OCO2.N12CCC(CC1)C2 52048,N1(C(CCC(=O)OC(C)(C)C)=O)CCC(O)(C(=O)Nc2ncc(C3CC3)s2)CC1 52049,c1(C(=O)NC2CCCC(N(C(=O)Cc3ccoc3)C)C2)ccc2ccn(C)c2c1 52050,N1(C(CC)CSC)CCc2c[nH]c(=N)nc2C1 52051,c1(C(N2C(CNC(C3OCCC(C)C3)=O)CCC2)=O)cc2ccccc2cc1O 52052,N1(C(COC(C)C)=O)CCCC2(CC(C(=O)N3CCCCC(C)C3)=NO2)C1 52053,C1(CNC(c2n(C=C)ncc2)=O)CC2CCC1N2C(C1SCCCS1)=O 52054,C1(NC(=O)CCc2cncnc2)CC2CC(C1)N(C(=O)CN1C(=O)CNC1=O)C2 52055,C(C(O)CCNC(C1(n2nccn2)CC1)=O)NC(COCCSC)=O 52056,c1(C(=O)NC(CNC(C(c2ccc(CC)cc2)C)=O)C2CC2)cc(C)cc(N)c1 52057,N1(C(C(CC)CC)=O)CCC(NC(=O)C(CC)n2ccc(C3CC3)n2)C2(CCC2)C1 52058,CC1CN(C(C2(N=[N+]=[N-])CC2)=O)CCC1CNC(c1ccc(N)cc1F)=O 52059,C1(CNC(C(C)NC(N)=O)=O)CN(C(=O)CC2CC(F)(F)C2)CCC1(C)C 52060,N1(C(C2CC(C#N)(OC)C2)=O)CC(NC(c2cnc(N(C)C)s2)=O)C2(CCC2)C1 52061,C=C(C)C(O)CC(=O)NC1CN(C(c2cc(N(C)C)ccc2F)=O)CC1C 52062,CN1CC(C(=O)Nc2occc2CNC(=O)C(C2CCCCC2)F)CC1=O 52063,Cc1ncc(C(=O)NC2CC(CNC(c3ccc(F)cc3)=O)CC2O)n1C 52064,Cc1cc(Cl)ncc1CC(=O)NC1CCC(CNC(=O)CC2CCC3CC23)CC1 52065,C1(NC(c2ccc(Cl)o2)=O)C2CC3CN(C(c4ccc(O)c(F)c4)=O)C1C3C2 52066,c1(-n2c(C(CC=C)CC)nc(-c3occc3C)n2)ccc(C)c(F)c1 52067,C=C=CCCC(=O)N1CC(CNC(C2CN(C)C(=O)N2)=O)C1 52068,c1(C(=O)NCC(C)CNC(c2nnn3c2CCC3)=O)nccc2ccncc12 52069,c1(C(N2C(CCNC(C(CC#C)O)=O)CSCC2)=O)cccc(F)c1C 52070,Cc1nc(CC(=O)NCC(O)CN(C)C(c2cc(F)n(C)n2)=O)[nH]c1C 52071,CCC(F)(F)C(=O)NCC1CC(NC(c2cnc(C)nc2)=O)C1 52072,c1(C(N2CC3C(CNC(=O)C4=CC5CCC4C5)(C3)C2)=O)cc(Cl)cc([N+](=O)[O-])c1 52073,CC(C)(C)C(C#N)C(=O)N1CC=CC(C(=O)Nc2cccc(F)c2)C1 52074,C1(NC(CC2CCN(C(c3c(COC)cco3)=O)C2)=O)CCn2nccc2C1 52075,C(=O)(C1=NOC2COCC12)NC.CC(C)C(CCN1C(=O)CC1C1CC1)C1CC1 52076,C1(NC(C2CCCCO2)=O)(CO)CN(C(C2(CO)CCC2)=O)C1 52077,N1(C(CC(C)O)=O)CCCCC(N(C)C(c2cc(C(F)(F)F)ccn2)=O)C1 52078,C1(CC(=O)NC(C#C)C(C)C)CC2(CC2)CN1C(c1cc(CO)n(C)n1)=O 52079,C(=O)(C(C)(C)CC(C)(C)C)NC1CN(C(C(C(CC)CC)C)=O)CC2(C1)CC2 52080,c1(N2CCC(CCNC(C(C)c3ccsc3)=O)C2)cc(=O)n(C)cn1 52081,C1(C(=O)NCCC2(OCC)CCC2)CCN(C(=O)C(CCO)N(C)C)CC1(C)C 52082,C1(NC(Cc2nc(C(C)(C)C)sc2)=O)CC2CCC1(CNC(C1(F)CCC1)=O)C2 52083,Cc1nc(NCCN2CC3CCC3(CO)C2)cc(N2CCC(CCO)C2)n1 52084,CC(C)(COc1ccccc1)C(=O)NC1CC(CNC(c2cccc(Cl)c2)=O)C1 52085,c1(CC(=O)NC(C)C(C)(C)NC(=O)CCCN2CCCC2)ccc2c[nH]nc2c1 52086,c1(C(=O)NC(C(N2CCCC(C=C)C2)=O)C2CCOC2)coc2ccccc12 52087,C12CCOC(C)(C1)CC1(O)CC(C1)NC2=O.n1(CCO)cc(C(C)OC)nn1 52088,N1(C(c2ccc(CNC(c3cncc(C)c3)=O)cn2)=O)CCC(C)(N(C)C)CC1 52089,CC1CN(C(=O)CC2CC2CNC(=O)C=Cc2cccnc2)CCS1=O 52090,c1(OCCC)ccc(C(=O)NC2(CO)CCOC2)cc1OC 52091,c1(C(N2CCCC(O)(CNC(C(=O)NCC)=O)C2)=O)cnc2cc(OC)ccn12 52092,C1(C(N(CC(C)NC(=O)CCc2ccc(N)cn2)CC)=O)CCc2nn[nH]c2C1 52093,c1(C(=O)NC2C(C)(CNC(COCCC)=O)CCC2)sc2nccnc2c1NC 52094,C(=O)(C1=CCCOCC1)N1C(C)CC(NC(=O)CSC(F)(F)F)CC1 52095,C1(NC(C2CN(CC)C(=O)N2)=O)CN(C(c2cocn2)=O)CCC1F 52096,C(=O)(C1CCc2ccccc21)N1CCC(N=[N+]=[N-])(C(=O)NC(CCCC)C)C1 52097,N1(CC)CCOCC1C(=O)NCCCCC(=O)NCCC1CCCN(C)C1 52098,C1(C(N(C(C)C2CC2)C)=O)CCN(C(=O)C(CO)NC(N)=O)C(C)(C)C1 52099,CC1OCCCC1C(=O)NC1CCC(NCC(O)CNC(N)=O)CC1 52100,C(c1ccccc1)=CC(=O)NC(C)C(C)NC(C1C(c2ccccc2)C1(C)C)=O 52101,C(=O)(C(O)C(C)(C)C)NCCCN(C(CC1(CC)OCCO1)=O)CC 52102,Cn1cc2c(n1)CCCC2C(=O)NC1CC(F)CN(C(=O)CC(C2CC2)C2CC2)C1 52103,C(=O)(C1=CCCOCC1)N1CC(COC)N(C(=O)C(n2cc(C)cn2)C)CC1 52104,CC1(C)CCC=C1C(=O)NC1CCN(C(=O)Cc2ccccc2Br)C1 52105,C(CC(F)(F)F)N(C)C(C1(CNC(=O)CC2CCOCC2)CC1)=O 52106,Cc1cccc(C(C2CC2)NCC(N2CCC(c3cn(CC(=O)O)nn3)CC2)=O)c1 52107,c1(N2CC(C(C)NC(c3csnn3)=O)C2)c(F)cc([N+](=O)[O-])cc1F 52108,c1(N2CCC(C=C)C2)ncnc(Nc2ccccc2NCCN(C)C)c1C 52109,c1(C2(CNC(c3n(CCCC)nnn3)(C)CCOCC)CC2)cc(C)cc(F)c1 52110,C1(NC(=O)COC(F)(F)F)CN(C(c2cnn[nH]2)=O)C2CCCCC12 52111,c1(C(=O)NC2(CNC(C(CSC)C)=O)CCCCC2)[nH]cc2c1CCS2(=O)=O 52112,c1(CC(=O)NC2CN(C(C(C)=C3CCC3)=O)CC(C)C2)ccc(S(N)(=O)=O)cc1 52113,CC1CN(C(=O)CCc2ccc(N)cc2)CC1CNC(=O)C(C)(C)C1CCC1 52114,C1(CNC(C2(CC(C)C)CC2)=O)CN(C(c2csnc2Cl)=O)CC1C 52115,CC(CCN(C)C)C(=O)NCC1C2CN(C(=O)C(C)(C)N(C)C)CC12 52116,c1(C(=O)NCC(C)N(C(=O)C(C2CCCCC2)F)C)cscc1C(N)=O 52117,c1(C(N(CCC)CCNC(C2(CC)CNC(=O)C2)=O)=O)cc2cscc2s1 52118,CC1CN(C(c2ncncc2Cl)=O)CC(C)N1C(=O)CCC1CCOCC1 52119,c1(C(N2CC3CN(c4ncc(OC)cn4)CC32)=O)cncc(S(C)(=O)=O)c1 52120,C1(C(=O)NC2(CNC(C3(CN(C)C)CC3)=O)CCOCC2)Cc2nncn2C1 52121,C1(NC(c2cccc(-n3cccn3)c2)=O)CC(F)CN(C(c2n[nH]cc2Cl)=O)C1 52122,c1(CC(N2CC(CNC(C3C(C)C3)=O)OCCC2)=O)c(C)[nH]c2ccnn2c1=O 52123,CCC(C)(CNC(C1(NC(=O)CC2CCCCO2)CC1)=O)OC 52124,C=CCCC(CC(C)C)C(=O)NCCN(C(=O)CCC1(C)CC1)C(C)C 52125,c1(C(N2CCN(C(COCCC#C)=O)C(C(C)C)C2)=O)cc(Cl)cc2c1CCC2 52126,c1(C(N(CCCCCNC(C(CC=C)CC)=O)C)=O)ccc2c(c1)nc(C)n2C 52127,C(C1CN(C(=O)C(C)(F)c2ccon2)CC1C(=O)NC12CC(C)(C1)C2)=CC 52128,C1(c2cn(CCF)nn2)(C(=O)OC)CCN(C(c2ccc(Br)s2)=O)C1 52129,c1(C(=O)NCCOC2CCN(C(C3(CCCC)CCCC3)=O)C2)nccnc1C 52130,C1(CCNC(C2=CC(C)(C)C2)=O)CCN(C(C2CCCO2)=O)CCC1(F)F 52131,CCC(C(=O)OCC)C(=O)N(CCC(=O)NCc1nc(C(N)=O)co1)OC 52132,C(C1CCN(C(c2nccn2C)=O)CC1)=CC(=O)NCc1c(C)cnn1C 52133,c1(CN(C(CC)CC)Cc2nc(C)c(C)s2)nc(C)c(C)nc1C 52134,CN1CCN(C(C2CCSC2)=O)CC1CNC(C1CC(F)(CO)C1)=O 52135,C1(NC(C(C)Cc2ccco2)=O)(CO)CCCN(C(c2cnc(Cl)cc2Cl)=O)C1 52136,c1(CCNC(=O)NCC2CCCCS2)ccc(Cl)cc1 52137,N1(C(c2nc(C(=O)NCc3ccc(Br)cc3)sc2)=O)CC2CCC1CO2 52138,c1(CNC(=O)CCOC2CC2)cnn2c1CN(C(=O)CC13CC(C1)C3)CC2 52139,C(=O)(C(C)(C)CS(C)(=O)=O)N1CC(NC(=O)C(C)(C)N2CCCCC2)CC(C)C1 52140,N1(C(C2(COC)COC2)=O)CCCC(NC(=O)Cc2noc(C)n2)CC1 52141,CN1CCN(C(c2cc(C3CC3)no2)=O)C(C(=O)N(C)Cc2ncnn2C)C1 52142,N1(C(C(Cn2ccc(C)n2)C)=O)CC2(CC(NC(=O)CCCC(N)=O)CO2)C1 52143,Cc1cc(C(=O)NCC(O)CN(C(=O)Cc2c(C)noc2C)C)sc1Br 52144,C(C)(C(C)C(=O)NCCSCC1CCC1)NC(C1(C(C)C)CCC1)=O 52145,C(CC(C(C)(C)C)NC(c1ncccc1Cl)=O)N(C)C(c1cc(F)ccc1F)=O 52146,C1(CC(=O)NC2CCCOC2)(NC(=O)COC(F)F)CCCCC1 52147,C=CC1(C(N2CCCC(C)C2CO)=O)CCN(C(c2ccc(C)c(F)c2)=O)C1 52148,C1(CC=C)(NC(=O)CSCCCC)CCN(C(c2cc(Cl)c(Cl)[nH]2)=O)C1 52149,N1(C(c2[nH]cc(C#N)c2)=O)CCOC2CN(C(c3cccc(F)n3)=O)CC12 52150,O=C1COc2nc(C(=O)NCC(CO)NC(=O)CN3C(=O)CNC3=O)ccc2N1 52151,CC(C)(C)C(CO)C(=O)NC1CCOCC1.C(=O)(CCCCCO)NCC=C(C)C 52152,c1(C(=O)NCCC2CCN(C(C3CC3F)=O)C2)csc2cccc(F)c12 52153,C1(C(=O)NCCCC(C)(C)NC(=O)CN2CC3CC3C2)CCc2nnc(O)n2C1 52154,CC(O)C(C(=O)NCC1(NC(c2csc(C3CC3)n2)=O)CCCCC1)N(C)C 52155,c1(C(N2CC3(CN(C(C)=O)C3)C2)=O)cc2cc[nH]c(=O)c2s1 52156,N1(C(c2cnc(COC)s2)=O)CCCN(C(C2CCNC(=O)C2)=O)C(C)C1 52157,c1(OC(=O)NCC2CCC23CC3)c(Cl)cc(Cc2nn[nH]n2)cc1Cl 52158,CC1CN(C(=O)C=CC2COC(C)(C)O2)CCN1C(c1cncs1)=O 52159,C(=O)(CC(F)(F)C(F)F)N(C1CCCCC1)CCNC(=O)CN1CCC(F)(F)C1 52160,C12CC(C)N1C2=O.n1(C2(CNC(COCCC)=O)CC2)cccn1 52161,C1(C(N2CC(SC)C(NC(c3cnc(S)nc3)=O)C2)=O)CN2CCCN1CC2 52162,C(N=c1cc[nH]cc1S(=O)(=O)N1CCC(CN(C)C)C1)c1nnc(COC)s1 52163,c1(C(N2CC(C3CN(C(c4cnn5ccsc45)=O)C3)C2)=O)ccc2c[nH]nc2c1 52164,CCS(=O)(=O)CC(C)NC(c1cc(N(C)C)ccc1C)c1nnnn1CC(F)F 52165,C(=O)(C1CCc2cccnc21)N1CC(CNC(=O)Cn2ccnn2)OCCC1 52166,c1(C(=O)NCC(CO)NC(=O)Cn2cc(C3CC3)nn2)cc(C(F)F)ccc1F 52167,Cc1nc(C(=O)Nc2ccnc(-c3ccnc(F)c3Cl)c2)ccc1F 52168,c1(CC)ccc(C(=O)N(CCC(C)NC(=O)CCC2CCC(=O)NC2)C)cc1 52169,C1(NC(c2c(C)nc(COC)s2)=O)CCN(C(=O)C=C(C)C(C)C)CC1C 52170,c1(CC)cccc(C(N2CCOCC2CCNC(c2ncccc2F)=O)=O)c1N 52171,C1(C(N(CCC(C)NC(C=Cc2scc(C)n2)=O)C)=O)CCCCN1N=O 52172,C12(C(N3C(C)(CC(=O)NCC4(SC)CC4)CC3)=O)CCCC1OCC2 52173,C12(NC(c3cnco3)=O)CC(CNC(c3cnn[nH]3)=O)(C1)C2 52174,O=S(=O)(c1ccc(Br)cc1N1CCC(NC2CCOC2)CC1)N1CC2CC1C2 52175,C(=O)(C1=C(C)CCCC1(C)C)NCCC(CNC(c1cc(C)oc1)=O)O 52176,c1(C(=O)NCCN(C(COCC)=O)CC(C)O)sc2c(Br)csc2c1C 52177,c1(CCNC(C(C)N(C(C(n2ncc(C)c2)C)=O)C2CC2)=O)ccc(C)nc1 52178,CC1=NOC(C)(CNC(=O)CCc2ccncc2Br)C1.n12cc(nn1)C2(C)C 52179,c1(SC)ncc(CN2CCC(NC(c3ccc(-c4ccccc4)s3)=O)C2)c(Cl)n1 52180,C1(C(N(CCC(F)(F)F)CC)=O)CC2(CCC2)CN1C(=O)Cc1cnnn1C 52181,c1(C(=O)NCC(C)(C)OCCNC(C2C(C)CCOC2)=O)cnn2c1CCC2 52182,Cc1cc(C(=O)NC2CC(NCc3cc(Cl)ncc3Cl)C2)cc(C)c1Br 52183,C1(C(N(C2CSC2)CC#C)=O)CCN(C(=O)C2(C)CC(=C)C2)O1 52184,N1(C(C2CC(SC)C2)=O)CCCC2(C1)CN(C(=O)Cc1cccc3nsnc13)C2 52185,C1(c2n(C)cnn2)CCCN(CCN2CCCCC2)C1 52186,CC1(C)CCC(CNC(=O)C(C)(C)C(N)=O)C(CN=c2[nH]nco2)C1 52187,Cc1cc(C(N2CC3CC3(C(=O)NCC3CC3CO)C2)=O)ncn1 52188,c1(C(C)C)cccc(C(N2CC(NC(C3CC4CCC4C3)=O)C(C)C2)=O)n1 52189,n1(C(C)C)cnc2ccc(CN3CCC(C(=O)NC)CC3)cc12 52190,c1(NC(=O)C(=O)NCCc2cccc(C(F)F)n2)ccc(I)c(Br)c1 52191,C1(NC(C(C)=C(CC)C)=O)CCCN(C(C2(CCOC)CC2)=O)CC1 52192,Cc1sc(O)nc1C(=O)NC1CCCCC1N(C)C(c1cc(C(F)F)ncn1)=O 52193,C(=O)(C1=CCC(C)(C)CC1)NCC(C)NC(=O)CCCOc1cccc(F)c1 52194,N1(C(=O)OC(C)(C)C)CCC2(CCC2)C(NC(C2(S(N)(=O)=O)CCCC2)=O)C1 52195,c1(CNC(C2CCC(CNC(C3CC34CCOC4)=O)O2)=O)cnccc1Cl 52196,Cc1ccnnc1C(N1CCCC1C(C)(C)C(=O)N(C)Cc1ncco1)=O 52197,c1(OC)nc(N2CCC2(C)C(=O)NCCN2CCCCCC2)ncc1Br 52198,N1(C(C2=CCCC2C)=O)CC(CO)C2(C1)CN(C(c1sccc1Cl)=O)C2 52199,C1(C(=O)NCC(C)CN(C)C(c2cccc(N)c2N)=O)CC2CCC(C1)C2 52200,c1(CNC(CC2(C)CN(C(c3cnc(Cl)s3)=O)C2)=O)cccc(S(C)(=O)=O)c1 52201,CCC(CN=c1cccc(S(=O)(=O)NCCN(C2CC2)CC)[nH]1)N(C)C 52202,N1(C(c2cc(C)ns2)=O)CCC(C)(CC(N2CCC(F)CC2)=O)C1 52203,n1(CC)nc(C(=O)NC2CN(C(C3(Br)CC34CCC4)=O)C2)cc1C 52204,c1(OC)nc(C(=O)NC(C)(CNC(=O)CCc2nccs2)C2CC2)sc1C 52205,c1(CNC(C(CC)SC)=O)nnn(C)c1C(=O)NC(C(N)=O)C(C)OC 52206,c1(C(=O)NCC(C)(C)NC(=O)Cc2sc(O)nc2O)ccc(O)c([N+](=O)[O-])c1 52207,C1(CC(N2CCC(NC(CCOC)=O)C2)=O)CCCC(C)C1 52208,N1(C(=O)Cc2cnsc2)CCC2CN(C(=O)Cc3cccc(F)c3F)CCC2C1 52209,c1(CC)ccc(C(=O)NCC(C)N(C(=O)COCc2ccccc2)C)o1 52210,N1(C(c2ccc(CSCC)cc2)=O)CCC(O)C(NC(=O)CC(C)C(F)F)C1 52211,N1(C(C2C(CC)C2)=O)CCC2(CC1)CC(NC(c1cnc(C(C)(C)C)s1)=O)CO2 52212,C12(C(N(CCCNC(=O)CC(F)(F)F)CC)=O)CCCC(CCC1)C2 52213,C1(C(=O)NCC(=O)OCC)(CC)CCCN(C(C2CC3CCCC3C2)=O)C1 52214,C(=O)(CCCCC(N)=O)Nc1ccc(OCC)cc1.C12CCCCN1C2 52215,n1(CCO)ccc(=NC(c2nc(CO)cs2)c2nnnn2CC(F)F)[nH]1 52216,C1(C(=O)NC2(CC)CN(C(C3C4(CC4)C34CC4)=O)C2)CCC2CC1C2(C)C 52217,CC1(C)COC(CCC(=O)NCCC2(O)CN(C(c3cc(O)cs3)=O)C2)C1 52218,c1(C(=O)NC)cccc(OCC(=O)NC2CCCC2NC(C2(C)CC2C)=O)c1 52219,CC1(C)COc2cc(CC3CC4(c5ccc(F)cc5)CC3C4)ccc21 52220,N1(C(C)=O)CCOCC1CC1CCN(C(=O)C(C)NC(=O)NC2CCC2)CC1 52221,N1(CC(=O)NC2CN(C(CCCCC#C)=O)CC2O)C(=O)NC(C)(CC)C1=O 52222,c1(OCC)ncccc1C(=O)NC1CCCCC1NC(C12CCCC1(C(N)=O)C2)=O 52223,N1(C(C)=O)CC(O)CC1C(=O)NCC(C1CCCC1)NC(c1nnsc1C)=O 52224,C1(C(=O)NC(C)CN2CCOCC2)CCOCCN1C(C1CC1(C)C(=O)OC)=O 52225,Cc1cc(CCC(=O)NCC(C)NC(C2CCCC2C2CC2)=O)cc(C)n1 52226,N1(N(CCS(CC)(=O)=O)C)CC(=O)N(CC(c2csc(C)n2)(C)C)C1=O 52227,CCCC(O)C(=O)NC1CN(C(c2ncncc2Br)=O)CC1C 52228,N1(C(CN(C(Cn2c(C)ccn2)=O)C(C)C)=O)CCC2CCN(C)C2C1 52229,N1(C(CCCCCC)=O)CCC(CCNC(c2cccc(C)c2F)=O)C(F)(F)C1 52230,Cc1cc(CCC(=O)NC2CCN(CCNC(=O)C(C)C)CC2F)ccc1O 52231,C(=O)(C(C)(C)C(=O)NCc1c(Br)nnn1C)N(C)C 52232,CCCCC(CN=c1[nH]cnc(Cl)c1Br)NC(=O)C1CCc2ccccc21 52233,C(=O)(C(C)(O)CC(C)C)NCC(CO)NC(c1ccc(OCCC)cc1C)=O 52234,CCCCCCC(=O)NC1CC2(C1)CC(CNC(C1CC3C(C1)C3(C)C)=O)C2 52235,C1(C(NOC(C)C)=O)CN(C(C2CC(C)(C)CN2C)=O)CCN1C 52236,C(=O)(CC(C)CC(F)(F)F)NCCC1N(C(c2nc(C)[nH]n2)=O)CCOC1 52237,c1(C(=O)NCC2CCN(C(C(C)CF)=O)C2)cnnc2ccccc12 52238,N1(C(C2CC(C#C)(O)C2)=O)CC2CC(NC(=O)C(C)OCC(C)C)CC1C2 52239,Cc1ccc(N)c(C(N2CC(NC(c3cnn(CCO)c3C)=O)C3(CC3)C2)=O)c1 52240,N1(C(C(C2CCC2)OCC)=O)CCN(C(c2cccc(N)c2F)=O)CCC1C 52241,CCC(C)CC(C(=O)N1CC=CC1CN(C)C)NC(=O)CCc1cccn1C 52242,C(CC(C(=O)NC(C)(C)C)N1CCCC1CNC(=O)Nc1ccccc1)SC 52243,Cc1cccc2oc(C(=O)NC3CC(O)CN(C(c4ncc[nH]c4=O)=O)C3)cc12 52244,CC1(C(=O)NC2CCCN(Cc3ccccn3)C2)CCCN(CCCl)C1 52245,c1(C(=O)NCc2occ(C(N(C)CC3C(C)OCC3)=O)n2)cc2ccccn2c1 52246,c1(C(C(=O)NCc2nncs2)NC(CSC(C)C)=O)cnn(C)c1 52247,CN1CC2CC1CN2C(C1CC(NC(c2ncn3c2CCC3)=O)C1(C)C)=O 52248,c1(-c2cn(CCCc3cccc(OC)c3)nn2)ccc2c[nH]nc2c1 52249,C(=O)(C(O)CC(=O)OC(C)(C)C)N1CC(C)C(CCNC(c2csnc2Cl)=O)C1 52250,C(c1cnccn1)=CC(=O)NC1CCCC1CNC(C1CCCCC1O)=O 52251,N1(C(C2CCC(C)(CC)O2)=O)CCN(C(C2CC(C)=NO2)=O)C2COCC12 52252,N1(C(C=C(C)c2ccccc2)=O)CCNCCC12CC2 52253,N1(C(C=CCN(C)C)=O)CCCCC(C2CN(C(=O)CCC(C)(C)C#N)C2)C1 52254,C1(NC(c2c(N(C)C)cccn2)=O)CCN(C(=O)C(O)CC2CC2)CC1F 52255,Cc1cc2nc(N3CCC(NC(=O)C(F)(F)c4cscn4)CC3C)cc(=O)n2o1 52256,c1(C(C(=O)NCC2C(NC(CC(=C)Br)=O)CCC2)C)ccc(CC)cc1 52257,C1(NC(CCOCC(C)C)=O)CCCC1C(=O)NOCC(C)(C)O 52258,N1(C(C2CC(CC)(CC)C2)=O)CCC(NC(=O)CC2CCC(=O)N2)C(F)(F)CC1 52259,Cn1c(I)cc2c(N(C(=O)CC(F)(F)F)C3CCNC3)ncnc12 52260,N1(C(C(CC)Br)=O)CCC2C(C1)OCCN2C(C1=NC(=O)N1C)=O 52261,C=CC1CN(C(=O)CCN(C)CC)CC1NC(C1CCN(C2CCCCC2)C1)=O 52262,c1(C(=O)NC2C(NC(c3cn(CC)nc3C(C)C)=O)CC2)coc2ccccc12 52263,c1(C(=O)NCCCN(C(C(CC=CC)C)=O)C)cc(OC)cc2ccoc12 52264,CC(C)(CC(F)C(=O)NCCCc1nncs1)NC(C1CC2C(C1)C2(C)C)=O 52265,C1(N(C(C)C)CCN(C)C)COc2cc(Br)ccc2C1 52266,N1(C(C(C)OCCOC)=O)CCC(NC(=O)Cc2[nH]cnc2C)C(CO)C1 52267,C(=O)(C(CC)CC(F)(F)F)NCC(CC=C)NC(C1(CC#C)CCC1)=O 52268,CC(C)(CNC(C1CCC1C#N)=O)CC(=O)N1CCCCC1C1(O)CC1 52269,N1(C(C2(CC)CCN(C(C3CCCN3C=O)=O)C2)=O)CCCCC(CO)C1 52270,C=C1CC2(C1)CC(C(=O)N(C(CNC(c1ncccc1F)=O)C1CC1)C)C2 52271,N1(C(C2C(C)(CC)C2)=O)CC2(CCN2C(=O)CCN(S(C)(=O)=O)C)C1 52272,C1(NC(C(CC=C)CNC(C2(O)CCC(C)CC2)=O)=O)C2CCN(CC2)C1C 52273,C1(NC(C(n2cc(CNC(COCCCC)=O)nn2)C)=O)CN(CC)C(=O)O1 52274,N1(C(C(c2n(C)cnc2)O)=O)CC=C(C(=O)NCc2ccc(F)c(F)c2)CC1 52275,CN1CCC(C(=O)NC2CS(=O)(=O)C23CCN(C(=O)CO)CC3)c2ccccc21 52276,c1(C(=O)NCC2C(NC(c3c(N)c(F)ccc3)=O)C2)cccc2c1OC(F)(F)O2 52277,C(=O)(CC1=NNC(=O)C1)NCCOCCCNC(C1C(C(C)C)CCC1)=O 52278,C1(C(NOC)=O)CCCN(c2ccc(C)nn2)C1 52279,C1(c2onc(C)n2)CCCCN1C(c1cnc(C)s1)C(=O)NCCC#N 52280,c1(C(N2CC3C(NC(C4N(CC)CCC4)=O)C3C2)=O)cc(OC)cc2c1CCC2 52281,c1(C(=O)NC(C(C)C)CNC(c2coc(CO)c2)=O)cc(Cl)cn1C 52282,Cc1cccc(C(N2CCCC(CNc3nccnc3C#N)C2)=O)c1Cl 52283,C1(CCCNC(CCCOC(C)C)=O)CCN(C(=O)CC2CCOC2)CC1 52284,CCC(C)CC(C)N(C(=O)CN(C(=O)CNC(C)=O)CC1(OC)CC1)C 52285,c1(OC)ccc(C)c(CN2CCC3(CC3C(=O)N(CC#N)CC#N)C2)c1 52286,N1(C(CC=C)=O)CC2CC(C)N(C(=O)CCOc3ccc(Cl)cc3)C2C1 52287,c1(OC(C)C(=O)N(CC(C)NC(C2(CN(C)C(C)C)CC2)=O)C)cccnc1 52288,c1(C(=O)NC2C(NC(C3(CC)CCNC3=O)=O)CCCC2)cnc(Cl)cc1N 52289,C12(CNC(Cc3ncc(C)o3)=O)CC1CN(C(=O)C=Cc1cnc[nH]1)C2 52290,CCCCC(C)CCC(=O)NC(Cc1cnn(C)c1O)C(=O)NCC[Si](C)(C)C 52291,c1(OC)nc(C(=O)N(C2CCN(C(=O)C(C)(C)C(F)F)C2)CCO)ncc1F 52292,c1(SC)c(C(=O)NC2CC2NC(c2cnc(OC(C)C)nc2)=O)cnn1C 52293,C1(C)(NC(C(CNC(CN(C)CC)=O)C)=O)CN2CCC1CC2 52294,N1(C(C(=Cc2cn[nH]c2)C)=O)CC2CCN(C(C3CCCCO3)=O)C2C1 52295,C(=O)(NNC(=O)N=c1nnn(CC(=O)O)[nH]1)c1cc(CN=[N+]=[N-])cc(Br)c1 52296,N(C1COc2c[nH]nc21)C(CCC(CC)NC(c1cccc(F)c1N)=O)=O 52297,CCC(C)C(O)CC(=O)NCC(C)(F)CNC(c1ccnc2cc[nH]c12)=O 52298,O=C(CCCCCCBr)N1CCN(Cc2c(Br)cc(F)cc2Br)CC1C(F)(F)F 52299,C(CCO)(C(=O)N1CC(NC(C2CCN(C)C2=O)=O)C1)N(C)C 52300,C(CCC(C)C)(C(=O)NC1CN(C)CC1C)NC(COCCCOC)=O 52301,N1(C(C2(CC#C)CC=CCC2)=O)CCC2(CC1)CN(C(c1nccnc1C)=O)C2 52302,CC(CCC(=O)NCC1COC(C)(C)C1)NC(=O)C(F)C1CCC1 52303,c1(C(C2CCCCC2)NC(c2cn(C)cn2)C)cccc(C(F)(F)F)c1 52304,Cc1ncc(C#N)c(N(C)CC2CN(C(c3c(C)cc(O)cc3O)=O)C2)n1 52305,C(CC(F)F)(C(=O)NC1CN(C)CC1C)NC(C1CCC(=C)CC1)=O 52306,C1(CCNC(C2(CNC(C(C)C3CC3)=O)CC2)=O)CSCN1C(=O)C(C)(C)C 52307,N1(CC)C2CCC(C2)C1Cc1cc(NCc2cc(C(=O)C#N)ccc2F)no1 52308,C(c1cncn1C)=CC(=O)NC1CC(CNC(CSCCC)=O)C1 52309,Cc1ccc(C(F)(F)C(=O)NC2CN(C(C3CCC(C(CC)OC(C)C)O3)=O)C2)nc1 52310,n1(CC(=O)NCC2N(C(COCC(=C)C)=O)CCC2C)cccc(C)c1=O 52311,CCC(CN(C)C)CC(=O)NC(C)(CSC)C(=O)N(C)CCSC 52312,CC1C2CC(C2NC(=O)CSc2cccc[n+]2[O-])N1C(=O)CSC1CCCCO1 52313,C1(CC)CCN(C(C2CN(C(=O)C=C3CCOCC3)CCO2)=O)CCO1 52314,C1(C(N2CC(COC)(NC(C3CCCC3F)=O)C2)=O)CC(O)C(F)C1 52315,N1(C(C(F)=C(C)C)=O)CCN(C(c2cccc(Cn3cccn3)c2)=O)CC1C 52316,N1(C(c2ccc(OCC=C)cc2)C(=O)NC)CCCC(C)(OC)C1 52317,C1(C(=O)NC2CCCC(N(C(=O)C=CBr)C)C2)CC2(CCC2=O)C1 52318,C(=O)(C#CC1CCCCO1)NC1CCCN(C(C)=O)C1C 52319,Cc1[nH]c(C#N)cc1C(=O)NC(C)(CNC(C1CC2CC2C1)=O)Cn1cccn1 52320,c1(NC(CC2(NC(CCN(C)C)=O)CCC2)=O)cnn(CC(=O)NC(C)(C)C)c1 52321,Cc1ccc(C(CNC(c2[nH]c(O)nc2C)=O)NC(C2CCCSC2)=O)cc1 52322,CCC(CC)C(C)C(=O)N(CC(O)CN(C)C(c1cccc(COC)c1)=O)C 52323,CC(C)(CCC(=O)N1CCC(=CCNC(=O)CCC2CC2(C)C)CC1)[N+](=O)[O-] 52324,C1(CNC2(C(C)C)CCC2)CCC2(CCC3(CC2)OCCO3)O1 52325,C=CC1(C(=O)N(C)Cc2cscn2)CCN(C(c2cc(CCC)on2)=O)C1 52326,N=c1cc(C(=O)NCC2CCCC(NC(=O)C=Cc3cccs3)C2)cc[nH]1 52327,C1(CNC(c2c(CC)c[nH]c2)=O)CCCC(CNC(=O)CCC2CCCCO2)C1 52328,CC(CC(=O)c1cccc(F)c1)C(=O)NCC1CCN1C(c1ccc(CO)s1)=O 52329,c1(CC)nc(C(=O)N(CC)CC2CCCCN2C(=O)CC2CCOC2)c(N)s1 52330,c1(SC)cc(C)ccc1C(=O)NCC(C(C)C)NC(=O)C(C)(O)C1CC1 52331,N1(C(C=CCC)=O)CCOCC(CNC(C2CCC(=O)N(C(C)C)C2)=O)C1 52332,c1(NC)ccc(C(=O)NC2CC2CNC(c2sc(F)cc2C)=O)c(Cl)c1 52333,C1(NC(C2(NC(CN(C3CCCC3)C)=O)CC2(C)C)=O)CCn2ccnc2C1 52334,C1(F)(C(=O)NC2CCCCN(c3c(C(=O)O)cncn3)C2)CCCCC1(F)F 52335,N1(C(CCC=CCC=C)=O)CC(C)CCC1CNC(=O)Cc1cnsc1 52336,C1(NC(=O)CCc2ccncn2)CCCC12CN(C(c1sccc1F)=O)C2 52337,CC1CCN(C(C2(O)CC2)=O)C1CNC(c1cnn(C2CC2)c1)=O 52338,N1(C(c2cnc(OC)s2)=O)CC2CC(C)N(C(C3(F)CCCCC3)=O)C2C1 52339,CC1(C(N2CCOC(CNC(=O)CSCc3ccncc3)C2)=O)CC(C#N)C1 52340,C(=O)(C(C)(C)S(C)(=O)=O)N1CC(CNC(CCc2c(OC)ccc(F)c2)=O)C1 52341,C1(C)(CNC(c2cc(NC)ncc2)=O)CCCN(C(C2CCCC2C(C)C)=O)C1 52342,C(C(C)(C)CC(=O)NCC1(C)CCN(C(c2ccc(C3CC3)c(F)c2)=O)C1)OC 52343,c1(N2CCC(N(C(=O)C(n3cc(C)cc3C)C)CC#C)CC2)ncccc1C#N 52344,CC(C)CC(CNC(C1(P(C)(C)=O)CC1)=O)NC(C1CCCC(CF)C1)=O 52345,N1(C(c2cc(C)ns2)=O)CC2CC(C1)CN(C(c1ccc(C(O)CF)cc1)=O)C2 52346,c1(C(=O)NC2C=CC(CNC(c3cnns3)=O)C2)ccc(OCCO)cc1 52347,O=C(C(=O)N=c1nc[nH]n1-c1ccccn1)N1CCC(C(O)CO)CC1 52348,n1(CC)nc(C)c(C(c2nnnn2C2CCCC2)Nc2cccc(CO)c2)c1Cl 52349,c1(CNCC(C)CC2CCCNC2)ccccc1O 52350,c1(C(=O)NC(CNC(C(CCCC#C)C)=O)C)cc(C)c2occc2c1 52351,CC1CC(C)N(C(c2nccc(N)c2Cl)=O)CCN1C(c1cnns1)=O 52352,n1(CC(=O)NC2CC(C)(NC(C(C3CCC3)OCC)=O)C2)nnc2c1CCCC2 52353,N1(C(C2ON=C(C)C2)=O)CC(NC(=O)C(C)N2CCC2)C(CO)C1 52354,C12(C(N3CCC(CNC(CCCC=C)=O)CC3)=O)CC3CC(CC(C3)O1)C2 52355,O=C(C#CC1CCC1)NC1CC(NC(=O)C=CCN2CCCCC2)C12CCC2 52356,C1(CNC(Cc2c(C)nc[nH]2)=O)CCCCCN1C(c1cnn(CC2CC2)c1)=O 52357,c1(CN2C3CN(C(C4C5COCC45)=O)C(C3)C2)cc(F)c(F)c(Cl)c1F 52358,N1(C(c2cc(CC)[nH]n2)=O)CC2(CCN(Cc3ccc(Cl)nc3Cl)C2)C1 52359,C1(C(C)(C)C)CCCC1(C)OC(C1CCC(SCc2cnnc(Cl)c2)O1)=O 52360,C1(CCC(=O)NCC2CCCC2NC(=O)Cn2nnc(C3CC3)n2)CC(F)(F)C1 52361,c1(C2OCCN(C(c3cc(Br)cc(Br)c3)=O)C2)cc(F)c(Cl)cc1Cl 52362,CC(C)C(C(=O)NCCCS(N)(=O)=O)NC(=O)Cn1cnnn1 52363,c1(C(N2C(CNC(c3coc(Cl)c3)=O)CC(F)(F)C2)=O)cn2c(n1)CCCC2 52364,C1(CN(C)CP(C)(C)=O)CCS(=O)(=O)CC1 52365,c1(OC)cc(C2CC2)ccc1C(=O)NC1CN(C(C23CC(F)(C2)C3)=O)CC12CC2 52366,N1(C(CC(=O)OCC)=O)CC2(CCC2NC(=O)C(O)CCSC)C1 52367,CC(CO)C(=O)NCC(C)(F)CNC(c1n[nH]cc1C1CC1)=O 52368,C1(C(F)(F)F)CCOCCN1CCCc1cccnc1Br 52369,c1(N(CC(C)NC(C2(C3CCCCO3)CC2)=O)C)ncnc(Cl)c1C(C)(C)O 52370,C(CCC(C)C)=CC(=O)N(CCOCCC(=O)NC(CCC)c1ccco1)C 52371,c1(OC)ncc(-c2cc(F)ncc2F)cc1C(=O)NC(c1ccccc1)CO 52372,CCC(C)(C)CCCC(=O)N(CC(C)NC(c1cc(O)ncc1F)=O)CC 52373,N1(C(c2cn(C3CC3)nn2)=O)CCCC(C2CCN(CC3CC3)C2)C1 52374,C(=O)(C1=CCC(C)CC1)NCC1(F)CCC(CNC(c2cncc(C)n2)=O)CC1 52375,n1(CC(N2CCC(C(CNC(CCSC)=O)F)CC2)=O)nc([N+](=O)[O-])cc1C 52376,c1(OC(C)C(N2CCN(C(C3C=CS(=O)(=O)C3)=O)CC2)=O)cccc(F)c1 52377,c1(C(N2C(CNC(CC(C)SC)=O)CCC(C)(C)C2)=O)cnc2sc(C)c(C)n12 52378,C(=O)(C(C)(C)CCC#N)N(CC(CN(C(c1nn(C(CC)C)c(C)c1)=O)C)O)C 52379,c1(C(N2CC(NC(C3CC4(C3)CC4F)=O)CC(C)C2)=O)cccc2cccnc12 52380,c1(C(=O)NC2C(NC(c3c(CC)n[nH]c3)=O)COCC2)n[nH]c2c1CCC2 52381,S(=O)(=O)(c1ccc(N2CCN(C(C3CC3C)=O)CC2)nc1)NCCCCC 52382,c1(NC(C2(C)CCN(Cc3c(C)c(F)c(F)cc3)C2)=O)cc2[nH]ccc2cc1Cl 52383,C=CC1CN(C(c2c(C)nn(C)c2C)C(=O)NC2CCC2)CC1O 52384,C#CCCC(O)C(=O)NC1(CO)CCCN(C(c2c[nH]nc2CC)=O)C1 52385,C1(CCOC)CN(C(C2CC(C)(C)O2)=O)CCN1C(=O)C=C1CCCC1 52386,c1(C(N2CC(NC(Cc3c(C)non3)=O)C(C)C2)=O)cnc2sccc2c1 52387,N1(C(c2c(C)nn(C)c2C)=O)CCN(C(c2cccc3c2CCC3)=O)CC(O)C1 52388,C1(NC(c2c(C)cns2)=O)CN(C(C2CC(F)C(=O)N2)=O)CC2(CCC2)C1 52389,C(=O)(CCCC(=O)N1CC=CC(NC(=O)C(C)C(C)O)C1)NC 52390,c1(OC)ccnc(NCC(=O)NC2CC2CNC(c2cc(Cl)cs2)=O)n1 52391,N1(Cc2nc(C(C)OCC)sc2)CCN(C(c2ccnc(CC)c2)=O)CC1 52392,C1(C)(C(=O)NCC(C2(O)CCN(C(C(C)OC(C)=O)=O)C2)C)CCCN(C)C1 52393,N1(C(CC(CN(C)C)O)=O)CC=C(CC(=O)N2CCCC(CCO)CC2)CC1 52394,N1(C(c2ccc(NC)cc2)=O)CC2CCCC2C1C(=O)NCc1ccco1 52395,c1(NC(C)=O)ccc(NC(C2CCCN(Cc3ccncc3O)C2)=O)cc1 52396,c1(C(=O)NCCCOCCC(=O)N(C(C)CCO)C)cnn(C)c1 52397,C1(C(=O)NCc2c(C(=O)NC(Cn3ncc(C)c3)C)scc2)CC2CCCC2C1 52398,CCC(C)C(O)C(C)C(=O)N1CCOC(CN(C(=O)CCC(C)C)C)C1 52399,C(=O)(C1Cc2c(Cl)cccc21)N1CC(CNC(c2cc(F)ccc2O)=O)OCC1 52400,c1(OCC)ccc(C(=O)NCCC(C)N(C)C(c2ncnn2C)=O)cc1OC 52401,N1(C(c2cc(CNC(COCCCC#C)=O)sc2)=O)CCCC2(C)CCCC12 52402,c1(C(=O)NCC(CNC(=O)COC(F)F)CO)c(Cl)ccc(Br)c1F 52403,c1(C(=O)NCCC2N(C(C#CC(C)C)=O)CCCC2C)ccn2ccnc2n1 52404,Cc1ccc(C(N2CCCC2CN(C(=O)CNC(c2cccs2)=O)C)=O)nn1 52405,C(=O)(CCCCCC(C)(C)C)NC1CN(C(c2c(C)oc(Cl)n2)=O)CC1F 52406,C1(CNC(c2nc(C(=O)NCC=C)sc2)=O)CC(F)CN1C(c1cocc1C)=O 52407,C1(C(N2CCC(CC)C2)=O)COCCN(C(C2CC(N=[N+]=[N-])C2)=O)C1 52408,CC1(C)CN(C(C2CC(F)C(=O)N2)=O)CC(C)(C)C1 52409,C#CC1CCCC(NC(C2CCOC2CNC(=O)Cc2c(C)cnn2C)=O)C1 52410,C(=O)(CC1=CCOCC1)NC(CC(=O)NCC1(CCO)CCC1)C(F)F 52411,N1(C(C2(CC)CC(OC)C2)=O)CCC(O)(CC(=O)NC2CCCC(O)C2)CC1 52412,N1(C(c2cc(O)ncc2Br)=O)CCC(NC(C2(C3CC3)CCC2)=O)C(O)C1 52413,C(c1ccccn1)=C(C)C(=O)NCC1(C(C)NC(c2ccnc(C)n2)=O)CC1 52414,C1(C)(NC(c2nc(C)ccc2F)c2n(CCCOC)nnn2)CC2CCC1C2 52415,C(=O)(C(C)=Cn1ccnn1)NC(c1ccc(CNC(CC(=O)OCC)=O)cc1)C 52416,C(=O)(C1CCCc2ncc(C)n21)N1CCN(C(C(CCCC=C)(C)C)=O)CC1C 52417,C1(CCNC(CNC(C)=O)=O)CCN(C(c2c[nH]c(=N)nc2C)=O)CCC1(F)F 52418,C(=O)(CC(O)CC(C)(C)C)N(C)Cc1c(F)cc(C#N)cc1Cl 52419,N1(C(C(CC)C)=O)CCC2(CCCC2CNC(=O)CCOC2CCCC2)CC1 52420,C1(C(=O)NCC(O)Cc2ccccc2)C2CCC(C2)N1C(c1cccc(F)n1)=O 52421,C(=O)(CCC(O)C(C)(C)C)N1CC(CNC(C2(CC#C)CCCO2)=O)C(C)C1 52422,C(=O)(C(O)CCc1ccco1)NC1C(CNC(=O)C(c2ccccc2)O)COC1 52423,n1(C(C)C(=O)O)cc(C2(O)CN(C(=O)Cc3ccccn3)C2)nn1.C1(=O)C(C)N1 52424,CC1(C)CC(NC(=O)CCc2ccc(F)cc2Cl)CN(C(=O)Cc2nc[nH]n2)C1 52425,c1(C(N2CCC(NC(c3c(C)[nH][nH]c3=N)=O)C2)=O)ccc(C)c2ccccc12 52426,Cc1nc(NCC(C)(C2CC2)NC(c2ccsc2C)=O)c(C)c(O)n1 52427,C1(NC(CNC(C(CC)C)=O)=O)CCN(C(c2c[nH]c(=N)nc2C)=O)C12CC2 52428,n1(CC)ncc(C(=O)NCc2ocnc2C(=O)NC2(C)CCOC2C)c1C 52429,N1(C(C(C)O)=O)CCN(C(C(=O)NCC2CCCO2)c2ccon2)CC1 52430,CCC(C)(C)C(O)C(=O)N1CC(N(C)C(c2ccc(OC)c(F)c2)=O)C(C)(C)C1 52431,c1(C(=O)NCC2CC(NC(c3n[nH]cc3Br)=O)C2)ccc(CO)cc1 52432,C1(NC(C=CSC)=O)C(C)CCN(C(c2cnc(C3CC3)o2)=O)C1C 52433,CC1CCCCC1(C)C(=O)NC1CCC(N(C)C(c2csc(C#N)c2)=O)CC1 52434,N1(C(c2c(C)ccc(C)c2)=O)CCCCC2(CCN(CCC3CCOC3)C2)C1 52435,N1(C(C(CC(=O)OC)N(C)C)=O)CC2CCC1CN2C(c1coc(N(C)C)n1)=O 52436,N1(C(c2c(CC)ncs2)=O)CCCN(C(c2ccc(O)c(O)c2)=O)CC1C 52437,C1(CNC(CC(C)OC)=O)CC2(CCC2)CN1C(=O)C=CC1CCCCC1 52438,N1(C(C=CC=CC)=O)CCCCC2(C1)CN(C(c1ccc(OCOC)cc1)=O)C2 52439,c1(C(=O)NCc2c(C(N3CC(C#CC)C3)=O)nn(C)c2)cc2ccccn2c1 52440,C1(C)(CNC(CCCc2nc(C)sc2)=O)CCCN(C(C2CC23CCCC3)=O)C1 52441,C1(C(N2CCC(NC(c3c(C)[nH][nH]c3=N)=O)C2C)=O)CCC2(CCC2)O1 52442,C(=O)(C(C(C)(C)C)N1CCNC1=O)NCC(C1CC1)NC(c1cc(C)on1)=O 52443,c1(C(=O)OCC(c2scc(C)c2)=O)ccc2cc(I)ccc2n1 52444,Cc1cc(C(=O)NC(C(=O)N(C)Cc2nc[nH]n2)C2CCCC2)ncc1N 52445,N1(C(C2(C)CCCN2C(c2cnn3ccncc23)=O)=O)CCn2cccc2C1 52446,CCCCC(CC(=O)NCC(F)(F)C(C)C)NC(c1cc(C)ncn1)=O 52447,C=CCCCCCCc1nc(C2CSC2)nn1-c1ncccc1Cl 52448,CCCC(C(=O)NCC(F)CNC(c1ccccc1Cl)=O)NC(N)=O 52449,Cc1ncnc(C)c1CC(=O)NC1CC2CN(C(=O)C(C)n3ccnc3)CC12 52450,C=CC(CC)CC(=O)N1CCN(C(=O)C2=CCSC2)C(CCO)C1 52451,CC1(C)NC(=O)CCC1NC(C1CC(NC(=O)C=Cc2ccco2)C1)=O 52452,CCCC(CC)CCC(=O)NCc1cc(C(=O)NC2(c3noc(C)n3)CC2)cs1 52453,CC1CN(C)CC(C(=O)NC2CCC(CCC(=O)NCC(C)(F)F)C2)O1 52454,n1(CC(=O)NC(C)C(C)NC(=O)Cc2cccc(F)c2)nnc2c1CCCC2 52455,O=C(C1=CCSC1)NC1CN(C(c2ccccc2)=O)CC1CO 52456,C12(C(N(CCNC(C3N(C(CC)=O)CCC3)=O)C)=O)CCC(CC1)CO2 52457,C(C1CCc2nccn21)NC(C1=NOC(CNC(C(CC)OC)=O)C1)=O 52458,c1(SC)ccccc1C(=O)NC1CN(C(=O)COc2ccsc2Cl)CC1F 52459,C1(CNC(C(C)c2ccco2)=O)CCC(NC(=O)CC2(CO)CCC2)CC1 52460,C1(NC(CC2C(C)OCC2)=O)CC(C(=O)NCC2CC2CC(C)(C)C)C1(C)C 52461,Cn1ncc2cccc(-c3nc(C4CCOC4)nn3-c3ccnc(O)c3)c12 52462,N1(C(C(=O)NCC(F)F)=O)C(CO)CCC1CO.N12CC(C(O)C1)CCC2=O 52463,N1(CC(=O)NCC(CN(C(=O)C(C)C2CCCC2)CC)(C)C)CC(=O)N(C)C1=O 52464,c1(C(N(CC(C)N(C(=O)COc2cn[nH]c2)C)C)=O)c[nH]c2nccc(Cl)c12 52465,C1(CC(=O)NCc2nccc(CC)c2)CCCN(C(c2coc(C#N)c2)=O)CC1 52466,c1(CC(N2CCCC(NC(C(CC)(C)C)=O)C2)=O)ccc2c(c1)CCCC2 52467,CCCCC(O)C(=O)NC(C1CCCC1)CNC(c1ncc(F)cn1)=O 52468,Cc1cnc2cccc(C(N3CCN(C(=O)Cn4cnnc4)CCC3C)=O)n12 52469,CCC(CC1CCCCC1)C(=O)NC1CCOC(CNC(C2CC(C#N)C2)=O)C1 52470,N1(C(C2CCC(C)NC2=O)=O)CCC2(CCN(C(=O)C=Cc3ccsc3)CC2)C1 52471,C(CCCC(=O)NCC(C)N(C(=O)Cn1nnc(-c2cccs2)n1)C)OCC 52472,N12CCC(C1)CN(C(C)(C)C1CC1)C2=O.C1(C(C)(C)C)CCCC1 52473,c1(C(C(=O)NCCOCC)N(n2cccn2)CCOC)ccc(S(C)(=O)=O)cc1 52474,N1(C(CN(C(=O)Cc2ccc(C#N)cc2)C(C)C)=O)CCS(=O)C(C)C1 52475,c1(OCC)ccc(C(=O)NC2(Cc3nc(C(C)(C)C)co3)CNC2)cc1 52476,C1(NC(Cc2ccc(C(=O)NC)cc2)=O)CCN(C(=O)CCNC(C)=O)C(C)C1 52477,c1(NCC(C(F)(F)F)OC)nccc(=NC2CCN(c3ccncc3)CC2)[nH]1 52478,C1(CC(=O)N(C2C(C)CC2)C)CN(C(=O)C(C2CCOCC2)O)CCO1 52479,N1(C(=O)NCC2CC(OCC)C2)CCCCCC1c1ccccc1C(F)(F)F 52480,c1(C(C)C)ccc(C#N)c(NCC2CCCN2C(C2CCCC3CCCN23)=O)n1 52481,c1(C(N2CC(CCNC(C3C(OCC)C3)=O)OCC2)=O)cnc2c(n1)CCCC2 52482,c1(C(=O)NCC2(CNC(Cn3ccc(C)n3)=O)CC2)c(C)cc(Cl)cc1C 52483,Cc1ccccc1C(C)C(=O)NCCCCCNC(C1CCC(F)C1)=O 52484,c1(C(=O)NC(CC2CCC2)C(=O)NCc2cncs2)cccc[n+]1[O-] 52485,N1(C(c2nc(CC)[nH]n2)=O)CC(NC(=O)C(C)CCN(C)C)C(C)(C)C1 52486,c1(SC)ccc(C(=O)NC2CCC2NC(=O)CCc2cnc(C)o2)cc1[N+](=O)[O-] 52487,c1(C(N2C(C)(CC)CC(NC(C3(NC(C)=O)CC3)=O)C2)=O)c(C)nc2sccn12 52488,c1(C(=O)NCC(CN(C(C2(CCC=C)CC2)=O)C)C)cnc(Cl)s1 52489,c1(C(N2CC(NC(Cc3c(C)cco3)=O)C(O)C2)=O)ccc(Cl)c2ccccc12 52490,C(=O)(CCCC(C)NC(=O)CC(C)(C)OC)N1CC(CC)SCC1 52491,C(=O)(C(O)CCCNC(=O)CCCC1CC1C)N(CCC(=O)NC)CC 52492,C(=O)(C(O)CC(C)C)N(C(C)CNC(c1nn(C)cc1Br)=O)CC 52493,CC1(C)CCCN(C(=O)C=Cc2cnc(O)nc2O)C1CNC(C1OCCO1)=O 52494,c1(N(CC(CC)CCCC)CCCCCCC)cc(OC)c(OC)c(Cl)c1 52495,n1(CC)nc(C)cc1C(=O)NC(C(=O)NCC(F)C1CCC1)C1(O)CCC1 52496,c1(C(N2CC3C(NC(C4CN(C)C(=O)C4)=O)C3C2)=O)cc2c([nH]1)CCCC2 52497,C12(C(=O)NCC3(NC(CNC(N)=O)=O)CCCCCC3)CCCCC1C2(F)F 52498,c1(C(CN2CCC(NC(=O)NCc3n(C)ccn3)CC2)=O)c(Cl)cccc1Cl 52499,CN1CC(C)(C(N2CC(N(C(=O)CSc3nncn3C)C)C2)=O)CCC1=O 52500,C1(NC(CCC2CC(OC)C2)=O)CC2CCC1(C(N1CC(C3CCCO3)C1)=O)C2 52501,C1(CC(N2CC(N(C)C(c3ccncn3)=O)C2)=O)NC(=O)CN(C)C1=O 52502,N1(C(=O)Nc2cn(C(C(=O)OC)(C)C)nc2)CCC(=O)N2CCCCCC12 52503,C1(CC)CN(C(=O)CC(F)(F)CC)CCN1C(=O)COc1cc(F)ccc1F 52504,C1(CC)CC(O)CCN1C(C1CCOC1CNC(c1cnnn1C)=O)=O 52505,CCC(CC)C(=O)NCc1csc(C(=O)NC(C)CS(C)=O)c1 52506,c1(SCC(=O)NCC(F)CNC(=O)CCN2CCOC2=O)ccccn1 52507,C1(NC(C=C(C)C)=O)CCC(C)N(C(C2C3COCC23)=O)C1 52508,C=C(C)C1OCCC1CNC(=O)CC1CC(C(=O)OCC)C1 52509,C1(C(CNC(C2C(CC)C2)=O)(C)O)CCN(C(C2(C(N)=O)CC2)=O)CC1 52510,Cc1ccn2c(C(N3CCOC(CCNC(c4ccccn4)=O)C3)=O)cnc2c1 52511,C1(C(=O)NC2CCCN(C(C3(CC)CC(F)(F)C3)=O)CC2)CC2CCC1C21CC1 52512,C1(CNC(C2CCS2(=O)=O)=O)CCN(C(c2csc(C(F)(F)F)c2)=O)C1 52513,c1(C(N2CC(C)C(CNC(c3cc4c[nH]nc4s3)=O)C2)=O)cc(N)c(Cl)c(O)n1 52514,C(=O)(C1=NOC(C)(C)C1)N(C1CCCC(NC(c2c(CC)[nH]cc2)=O)C1)C 52515,c1(CNC(c2c(C)c[nH]n2)=O)cccc(C(=O)NC(C)CN2CCCC2=O)n1 52516,C#Cc1cccc(CC(=O)NCC2(NC(c3[nH]c(C)nc3C)=O)CCOCC2)c1 52517,c1(C(=O)NCC(CC)NC(=O)C(F)(F)c2csc(Cl)c2)n[nH]c2c1CC(C)CC2 52518,S(=O)(=O)(c1cccc(NC(=O)COCCOCCN)c1)NC 52519,C#CCCCC(C)C(=O)NC1CC(C(=O)NCCCN2CCCC2)C1 52520,Cc1cc(C(N2CC(O)(CCNC(C34CCCCC3C4)=O)C2)=O)cc2nc[nH]c12 52521,C1(C(=O)NCC2COC3CC2C3)CCC2(CCOCC2)C1 52522,c1(C(=O)NC2(CCNC(C3CCC(C)C3)=O)CCC2)nc(N(C)C)nc(=N)[nH]1 52523,C(=O)(C(C1CCCC1)SC)N(C(C)CNC(=O)CNC(C)=O)CC 52524,N1(CC(=O)NC(C(C)C)CNC(c2cc(Cl)n[nH]2)=O)CCC(=O)NC1=O 52525,C1(N(C(C(c2ccnn2C)C)=O)C)CCCN(C(=O)CCN2CCC2)C1 52526,n1(C(C)(C)C)ncc(C(N(C2CC2)CCc2ccc(CCC3CCC3)cn2)=O)c1Cl 52527,O=S(=O)(c1ccc(Cl)cn1)NC1CCN(Cc2cccc(Br)c2O)C1 52528,C(=O)(CC(CNC(=O)CN(C1CCCCC1)C)C1CCC1)N(C(C)C1CC1)CC 52529,CC1CC(NC(=O)C(C)(F)F)CCN1C(C1(c2ncccn2)CC1)=O 52530,c1(CC(N2CCC(O)(CNC(C)=O)C2)=O)ccc2nc(Cl)sc2c1 52531,c1(CN2CC(CNC(C(CC)C)=O)OCC2)nc2ccccc2[nH]1 52532,N1(C(c2cc(C(OC)OC)on2)=O)CCCCC1CNC(=O)C(C)(C)C1CC1 52533,c1(C(N2C(CN(C(=O)C=CC3CC3)C)CCC2)=O)c(O)nc(=O)n2c1CCC2 52534,n1(CC(=O)OC)cnc(C)c1C(=O)NC1CC(C)(NC(c2cccnc2C)=O)C1 52535,c1(C(c2n(CC(=C)C)nnn2)NCC2CCO2)c(Cl)ncn1C 52536,O=S(=O)(c1[nH]cc2c1CCS2(=O)=O)Nc1ccncc1C(F)(F)F 52537,Cc1ccnc(NCC2CCCN2C(=O)C(C)Oc2ccccn2)c1[N+](=O)[O-] 52538,C12(NC(C(C3CCCCCC3)C)=O)CCC(CC1)N(C(C1CCCCC1(C)C)=O)C2 52539,c1(OCC)ncc(NC(=O)CCCN(c2ccccc2)C(C)=O)cn1 52540,C1(F)(C(=O)NCC2C3CN(C(C4(CC)CCOC4)=O)CC32)CC2(CCC2)C1 52541,C(=O)(C(CCOC)NC(=O)CCc1nc(C)no1)NC(C=C)C1CCC1 52542,N1(C(COCCOCCOC)=O)CC2CC(NC(c3ccc(CO)cn3)=O)C1C2 52543,CC1CC(C(=O)Nc2nnc(-c3ccco3)o2)N(C(C2CCCO2)=O)C1 52544,N1(C(C2=CCN(C(c3cnc(C)[nH]c3=N)=O)CC2)=O)CCC2CCC(O)C1C2 52545,c1(C(=O)NCCOCCCNC(C(C)OCCC=C)=O)cc(Cl)c(Cl)[nH]1 52546,C(=O)(C(F)(F)C(F)(F)F)NC1CCCN(C(c2ccc(OC)s2)=O)CC1 52547,C(=O)(CCCCCCS(N)(=O)=O)N1CCCC(C(N2CC(C)NC(=O)C2)=O)C1 52548,c1(N2CC3(C(NC(C4CC5C=CC4C5)=O)CCC3)C2)c(Cl)cc([N+](=O)[O-])cc1Cl 52549,Cc1cc(C(=O)NCCCOCCNC(=O)C(O)CC(F)F)nc(O)c1 52550,C#CC1(C(=O)NCc2cc(C)c(C(=O)NC(C)C(C)C)o2)CCCC1 52551,C1(C(=O)OC)(COC(c2cc(C)cc(C)c2)=O)COS(=O)(=O)C1 52552,C=CCCC(C(=O)N1CCC(C(F)F)C1)NC(c1ccc(C)cc1)=O 52553,CN1CC=C(c2ccc(C3(CNc4ncc5cccc(O)c5n4)CC3)cn2)CC1 52554,C1(CNC(C2(CC=C)CC=CC2)=O)CC(OC)CN1C(C1CCC1COC)=O 52555,c1(C(=O)NCC(CN(C)C(c2ccncc2)=O)O)cncc(N(C)C)c1 52556,c1(CC(=O)NCC2C=CC(NC(C3CNC(=O)N3)=O)C2)cccc(C(F)(F)F)n1 52557,C1(C(=O)NCC(C)NC(=O)C(C2CC(F)(F)C2)O)CCCN(C)C1 52558,CN1C(=O)COC12CCN(C(c1cc(-c3csc(Cl)n3)on1)=O)CC2 52559,N1(C(CCC=CC(C)C)=O)CCC(C2CCN(C(c3c[nH]nc3C3CC3)=O)C2)C1 52560,C(=O)(C(F)(F)CN1CCCC1)NCCCN(C)C(C1(F)CCCCC1)=O 52561,c1(C(=O)NC2CCC(C)N(C(=O)CN(C3CCSC3)C)C2)ccc2cnoc2c1 52562,N1(C(C=CSC)=O)CCC2CCC(C1)N2C(c1cccc(N2CCOCC2)c1)=O 52563,Cc1c(C(N2CCC(C(N3CC(C)C(O)C3)=O)C2C)=O)c[nH]c1C#N 52564,C1(C(C)(C)NC(c2nc(Cl)cs2)=O)CCN(C(C2CCCCS2)=O)CC1 52565,C1(C(=O)NC(c2ncc[nH]2)CC)(NC(=O)CC2(C)CCCC2)CC(CO)C1 52566,c1(NC(=O)NC(c2ccc(Cl)cc2)CC(=O)OC)ccc2c(c1)OCC2 52567,C(=O)(C(CCF)NC(=O)CC(=O)NC1CC1)NC(C)CCCO 52568,C(=O)(C(O)CCCNC(=O)CC1CCCN(C)C1)NC(C)C(C)n1cccn1 52569,N1(C(C2CC(CC)C2)=O)CC2(C(=O)NCC3CC(C(C)(C)C)C3)CC1CCO2 52570,C(=O)(C1=CCCCCC1)NCC(CC=C)NC(C1CC(Cl)(Cl)C1)=O 52571,C1(O)(CNC(c2cc(C)c(F)cc2)=O)CCCN(C(C2C=CCS2)=O)CC1 52572,C1(NC(C=CCCC)=O)CC2(CNC(=O)CC(C)c3cccnc3)CC1CO2 52573,n1(CC)cnc(C(=O)NC2CC(C(=O)NCCCCO)C2)n1 52574,N1(C(C2CC(=C3CC3)C2)=O)CCN(C(C2(C3CCC3)CC2)=O)C2COCC12 52575,c1(C(=O)OC)c[nH][nH]c1=NC(=O)C1CN(C(c2cccc(O)c2F)=O)CCC1O 52576,N1(C(CC2(C=C)CC2)=O)CCC2(CCCN2C(=O)Cc2cnn3ccccc23)C1 52577,Cc1cccc2[nH]cc(CCC(N3CCC(CCNC(=O)CSC(C)C)C3)=O)c12 52578,c1(C(N2C(CNC(C3CCN(C)CC3)=O)COCC2)=O)cnc2c(n1)CCCC2 52579,N1(C(Cc2c(C)n[nH]c2)=O)CC(NC(=O)C(C)(C)C#N)C(c2ccc(F)cc2)C1 52580,CCCCC(=O)C(=O)NC(CN(C)C)C(=O)N(CC)Cc1ccoc1 52581,C1(C(NC(C)C)=O)CCCN(CCCC)C1.N1(C(CC2CC(=C)C2)=O)CCC(CN)C1 52582,N1(C(c2cc(N)c(F)c(F)c2Cl)=O)C2CCCC1CN(C(c1ccsc1)=O)C2 52583,C1(C(=O)NC(C)C2CC2)CC(F)CN(Cc2ncc[nH]2)C1 52584,CCC1(CNC(CCCC2CC2)c2nnnn2C2CC2)OCCc2ccccc21 52585,N1(C(C(C2CC(F)(F)C2)OC)=O)CC(C)(C)CC1CNC(C1CC(SC)C1)=O 52586,c1(-c2onc(CCCC(C)=O)n2)n[nH]c2c1CC(C)CC2 52587,CCC(O)C(C)C(=O)N1CCCC(CCNC(c2cc(C3CC3)n(C)n2)=O)C1 52588,c1(C(N2CCCCC(CNC(C3C(CC(C)C)C3)=O)C2)=O)cnn2c(=N)[nH]cnc12 52589,N1(C(C(CC)C(C)C)=O)CC2(C1)SCCC2NC(c1cccn2cncc12)=O 52590,C1(C(=O)NCC(c2ccccc2)C)CC(O)CN1C(=O)CC1CC(=O)NC1=O 52591,C#Cc1cc(C(=O)NCCC(O)C(=O)NC(C)CC(=O)NC(C)C)ccc1C 52592,C1(C2CCCCO2)(C(=O)NCC(C)CN(C)C(c2ccc(CO)o2)=O)CCCO1 52593,n1(CC(=O)NCC2(CNC(CCSC)=O)CCC2)cc2ccccc2n1 52594,N1(C(COCCSC)=O)CCC(NC(C2Cc3nccn3C2)=O)C(C(N)=O)C1 52595,C1(C(N2CCCC(N(C(CCN3CCN(C)CC3)=O)C)C2)=O)CC(C2CC2)=NO1 52596,CC1CN(Cc2ccccc2)C(C)CN1C(=O)CC1CCCNC1 52597,C1(NC(C2CC(C)C2)=O)CN(C(=O)CC2CCCS2(=O)=O)CCC12CCC2 52598,c12ccc(nc1)C(=O)NC1CCC(C1)N(C)C2.c1(OCC)ccc(C(=O)OC)o1 52599,c1(C(=O)NCC2CCN(C(CCOCCOC)=O)C2)nc(C)c(C)nc1C 52600,N1(C(=O)C=CC2CCCC2)CCC2OCCN(C(C3CCCS3(=O)=O)=O)C2C1 52601,c1(C(N2CC(O)CC(NC(C3CC(CC)C3)=O)C2)=O)n[nH]c2c(C)cccc12 52602,C1(CNC(C2C(C)OC(=O)N2)=O)CCN(C(C2CC(=O)NC(=O)N2)=O)C1(C)C 52603,c1(C(C)NC(CC2CC(NC(CC=CC=C)=O)C2)=O)nc(C)cs1 52604,CCC(C)C(C(=O)NC1C2CC3C1C3C2C(=O)NCCCO)OC 52605,C1(CN(C(COCC=C)=O)C)C2CN(C(=O)CCCc3nc(C)no3)CC12 52606,c1(NC(=O)Cc2cc(=O)n(-c3ccccn3)[nH]2)ccc(F)cc1C(N1CCCC1)=O 52607,N1(CC)CCC(C(=O)NC23CC(C(=O)NCC(O)C(F)F)(C2)C3)C1 52608,CCC(C)C(C)C(=O)N(C1CN(C(=O)C(N)=O)C1)C 52609,C(=O)(C(Cc1ccco1)NC(c1cc(O)cs1)=O)NC1CC(C(=O)OC)C1 52610,N1(C(c2cc(C)sc2C)=O)CC(CNC(=O)C(O)C2CC2)CC(C)(C)C1 52611,N1(C(C2C(C)CC=CC2)=O)CCOCCC1C(=O)N(C1CCC(F)(F)C1)C 52612,N1(C(C(C)N(C(c2cnnn2C)=O)CC)=O)CCN2C(=O)NCC2C1 52613,N1(CC)C(=O)CCC1CC(=O)NC(C)(C)CCNC(=O)C(C1CCC1)OC 52614,CC(=O)C(C)(C)CC(=O)NC(CNC(C1CC12CCCCC2)=O)CCO 52615,N1(C(=O)NCCN(C2N(CCC=C)CCCC2)C)CCC2(CCCCC2)CC1 52616,N1(C(C(C#C)(C)C)=O)CC2CC(NC(=O)C(=Cc3cccs3)C)C2C1 52617,CC1(CC(=O)NC(CO)C(F)(F)F)CCN(C(c2nccnc2N)=O)C1 52618,CCC(C)CC(C(=O)NCC(C)(C)C(F)(F)F)NC(=O)CN(C)CC 52619,C1(C(=O)NCCC2(OC)CN(C(c3ccnnc3O)=O)C2)CCC(C)NC1=O 52620,C1(=CCNC(C(C)(O)C2CCOCC2)=O)CCN(C(=O)C(F)OC(F)(F)F)CC1 52621,C1(NC(=O)CCc2cc(Cl)no2)CC2CC(C1)N(C(C1SCCCS1)=O)C2 52622,CCC(F)(F)CC(=O)NC(CC1CC1)CC(=O)N(c1cnn(C(C)C)c1)C 52623,C1(C(N2CCC(C(C)OC)CC2)=O)CN(C(C2CC2(F)Cl)=O)CC1C1CC1 52624,c1(CC(=O)NCC(=C)CCNC(c2cc[nH]n2)=O)nc(C2CC2)nn1C 52625,c1(-n2cc(CC(C3CCCS3(=O)=O)C(=O)OC(C)(C)C)nn2)cccc(Br)c1Br 52626,c1(C(N(CC(CN(C(CSCC=C)=O)C)O)C)=O)cc2cc(Cl)ccc2s1 52627,C(=O)(C1=COc2ccccc2O1)N(CC(C)NC(C1(CCOC)CCC1)=O)C 52628,C(=O)(CCS(=O)(=O)CC(C)C)c1nc(-c2ccc(C(C=C)C(C)(C)C)cc2)on1 52629,C1(CN(C(=O)Cn2cnnn2)CC)CCCN(C(=O)CCOCCCOC)C1 52630,C1(OC)CCCC(C(=O)NC2(C)CC(NC(c3cc(Br)n(C)n3)=O)C2)C1 52631,c1(C(N2CCCC(C(N3C(CC)COCC3)=O)CC2)=O)cc2ccccn2n1 52632,C(=O)(C(F)C(C)(C)O)NC(C(C)C)CNC(=O)C=Cc1ccccn1 52633,c1(CC(N2CC3CC3(CNC(C3(F)CCOCC3)=O)C2)=O)ccc(CO)cc1 52634,Cc1cc(F)ccc1Oc1ccc(C(=O)N(C)CC2CCN(C)C2)cc1 52635,N1(C(c2n[nH]c(C)c2O)=O)CCC(CNC(=O)Cn2cc(Br)cn2)C1(C)C 52636,C(=O)(C=CSc1ccccc1)NCCN(C(c1nscc1N)=O)CC 52637,Nc1ccc(C(N2CCCCC(CNC(=O)COCC(F)(F)F)C2)=O)nc1F 52638,N1(C(C2C(CC)CCN2C(C2CC3CC(C2)C3)=O)=O)CCSC2(CCC2)C1 52639,N1(C(COCCCC)=O)CC2CCN(C(C3CCCCS3)=O)CC12 52640,N1(C(C(F)OC)=O)CC(C2CCCCN(C(c3ncc(C)cc3F)=O)C2)C1 52641,C1(CC(=O)N(CC(C)(C)CNC(c2ccc(Cl)s2)=O)CC)C(=O)N(C)N=C1C 52642,N1(C(CS(=O)(=O)NC)=O)CCCC(C)(C)C1C(=O)NC1CN(C)C(C)(C)C1 52643,C1(NC(C2CC(C)SCC2)=O)COCCN(C(c2ccc(=O)n(C)n2)=O)C1 52644,c1(C(=O)NC2CCC(CNC(c3nocc3Cl)=O)C2)ccc(F)c2occc12 52645,c1(CC(=O)NC2(C)CN(C(C3C4CCC(=O)C34)=O)C2)ccc(F)cc1Br 52646,N1(C(CNC(=O)OCC=C)=O)CCCC1C(C)NC(C1(C(F)F)CC1)=O 52647,C1(NC(c2cnc(C)[nH]2)=O)C2CCC(C2)C1C(N1CCC(O)C(F)C1)=O 52648,C(CNC(c1ccc(C(C)=O)cn1)=O)(C(C)(C)C)NC(CC1(OC)CC1)=O 52649,c1(OC)cc2ncn(CC(=O)C(C)C)c(=O)c2cc1OC 52650,C(=O)(C(C)Cc1cnc[nH]1)N(C(CCNC(CCNC(=O)OC)=O)C)C 52651,C(c1ccc(OC)cn1)=CC(=O)NC(CC)(CNC(=O)COCCCF)CC 52652,c1(C(=O)OC)cc(C(=O)Nc2cccc(CNC(c3coc(C)c3)=O)c2)ccn1 52653,Cn1nc(Cl)c(C(=O)NCC2CCCC2NC(c2cncc(F)c2)=O)c1Cl 52654,C1(CCC=C)(C(=O)N(CC)Cc2ccncc2)CN(C(=O)CCC2CC2(C)C)C1 52655,C1(C(N(CCCCN(C(C(CCN(C)C)N(C)C)=O)C)C)=O)CCCC(=O)CC1 52656,C1(CNC(CCC)=O)(CNC(=O)C(c2ccc(Cl)cc2)(C)C)CC12CCC2 52657,C(=O)(C(C)(C)NC(=O)OC(C)(C)C)N1CC(C(C(=O)NCC2C(C)C2)O)C1 52658,C1(C)(CC(=O)N(C)CC2CCCN2C(C2(C)COC2)=O)CCCCC1 52659,CC(C(=O)N1CCC(C)(C(=O)NCCOC2CCCC2)CC1)S(C)(=O)=O 52660,S(=O)(=O)(CCC(=O)N1CCC(NC(c2ccnc(C)n2)=O)C1C)NC 52661,CS(=O)(=O)c1ccc(C(=O)NCC(C2CC2)NC(C2(CO)CC2)=O)o1 52662,C#CCC(C)(C(=O)NC1CC1C(C)C)NC(c1cnc(NC)cn1)=O 52663,C1(NC(c2c(C)cccc2)=O)CN(C(=O)C=C2CCOCC2)CC(C)(C)C1 52664,C1(NC(C=CC=CC)=O)CC2CCC1CC2NC(c1ccncc1O)=O 52665,N1(C(C2C(C)C2)=O)CCN(C(C2CC3CC2C3)=O)C(CS(C)(=O)=O)C1 52666,CCS(=O)(=O)c1ccc(CC(=O)NCC2CN(C(=O)C(C)N(C)C)C2)cc1 52667,C=CCCC(F)(F)C(=O)N1CCC(N(C(=O)CCN(C)CCO)C)C1 52668,C(=O)(C(O)CCNCCC1CCC(=O)N1)NC(C1CCCC(=O)N1)=O 52669,c1(C(=O)NCCCNC(C2C(C)(C)OC(=O)N2)=O)cnn2c(Cl)cccc12 52670,N1(C(C2CCC(C)CC2)=O)CC2(CO)CC1(C(=O)NC1CCN(C(C)(C)C)C1)C2 52671,N1(C(c2c(C)nsc2C)=O)CC(CC(N2CC(N(C)C)C(C)C2)=O)C2(CC2)C1 52672,Cc1ccc2c(C(=O)NC(C3CCCN3C(c3c[nH]c(=N)s3)=O)C)c[nH]c2c1 52673,C(C)(C(CC(=O)NCc1noc(C)n1)NC(c1[nH]cc(C)c1C)=O)OC 52674,C(=O)(C(C(C)C)C(C)C)N1C(CNC(C2CCCC(=O)N2)=O)CC(OC)C1 52675,CCCC(CCO)ONC(C1CCCN(c2ccc(NC)cc2)C1)=O 52676,N1(C(c2c(CC)scc2)=O)CCOC(CCNC(=O)CCCn2cccc2)C1 52677,C12(NC(c3cccc(Br)c3)=O)CCC(C(N3CC4(CCC4)C3)=O)(CC1)CC2 52678,C(C)(C)(CCC(=O)N(C1CCN(C(=O)C=C(C2CC2)C2CC2)CC1C)C)OC 52679,Cc1cc(NC(C)C)ncc1S(=O)(=O)N(C)C(c1ccc(S(N)(=O)=O)cc1)C 52680,c1(C(N2CCC(O)(C(CNC(C(C)=C3CCC3)=O)C)C2)=O)cnc2scc(C)n12 52681,CS(=O)(=O)C=CC(=O)NCC1(O)CCN(C(C2CC3(CCC3)C2)=O)C1 52682,c1(C(=O)NC2C(C)N(C(c3cn4c(n3)SCC4)=O)CC2)cc(F)c(Cl)cc1Cl 52683,CC(C(C)C(=O)NC1(C2CCCCO2)CC1)NC(c1ncccn1)=O 52684,c1(CC(N2C(C)(C(=O)Nc3cncc(OCC)c3)CC2)=O)ccc(F)c(F)c1 52685,C1(SCC)CC(CC(=O)NC2CC(NC(=O)C(Br)=C(C)C)C2)C1 52686,Cc1ncc(C=CC(=O)NC2CCC(CCNC(=O)CCS(N)(=O)=O)C2)c(O)n1 52687,C(CCCC(CO)NC(C1ON=C(C)C1C)=O)NC(c1c(C)nc(CCC)o1)=O 52688,Cn1ncc2c(NCCCCCO)[nH]c(=NCC3CCc4ccccc43)nc12 52689,c1(C(=O)NC2C(NC(Cc3c(C)scc3)=O)CCOC2)ccc(N)c(Cl)n1 52690,c1(OC)cccc(N(C)C)c1C(N1CC2C(C1)N2c1ncc(C)cn1)=O 52691,Cc1ncc([N+](=O)[O-])cc1C(=O)NCCCCN(C)C(C1(C(C)(C)O)CC1)=O 52692,C1(C(=O)O)CC(F)(CNC(C2C=CCCN2)=O)C1 52693,CC1C(C(=O)NC(CCO)C2CCCC2)CCN1C(c1ccco1)=O 52694,N1(C(COCc2cc(C)on2)=O)CCCC(NC(c2cncc(Cl)c2C)=O)CC1 52695,C1(NC(c2cc(C)[nH]n2)=O)COC2(CCN(C(C3(CO)CCOCC3)=O)C2)C1 52696,CCCS(=O)(=O)CC(=O)NCC1CC2(CO1)CN(C(c1c(C)csc1Cl)=O)C2 52697,c1(-c2n(-c3cccc(C)c3)nc(C3CCOC3)n2)cn(C)cc(Br)c1=O 52698,c1(OC)ccc(N(C)C(C)=O)cc1.c12cc(n[nH]1)C(=O)COCC(=O)N2 52699,C(=O)(C1=CCCN(C(C2CCCC(O)C2)=O)C1)NC1(C)CCCC1O 52700,N1(C(CCNC(C(C)(C)C)=O)=O)CC(O)(C2(CNC(=O)CC(C)(C)O)CC2)C1 52701,c1(OCC(=O)NC)ccc(C(=O)NCCC2(O)CN(C(=O)CCOC)C2)cn1 52702,c1(C(=O)NC(CC(=O)NC(C)C)C)ccc(N(C)C)c(C#N)c1F 52703,c1(NC(CNC(c2ccn(C(CC)CC)n2)=O)C2CC2)cc(O)nc(O)n1 52704,C1(C(=O)NC(CCC=C)CO)CC12CCN(Cc1cc(C(=O)O)cc(C)c1)C2 52705,N1(C(C2(C3N(C(c4ccc(OC)o4)=O)CCC3)CC2)=O)CC(=O)NCC1C 52706,N1(C(c2cc(C)oc2)=O)CC(NC(=O)C(C)Cc2cnc[nH]2)C(N=[N+]=[N-])C1 52707,C(C(F)(C(=O)NC(CC)C(N)=O)C(C)C)NC(c1ccn(CCC)n1)=O 52708,c1(NCCCCCCN(C)C(C2CC=CCO2)=O)cc2nncn2cn1 52709,n1(CCC(=O)N(S(C)(=O)=O)C)cc(CNC(=O)C(C)(C)O)nn1 52710,c1(-c2n(-c3c(CC)cccc3)nc(C(O)CC)n2)ccc(F)c(Cl)c1F 52711,c1(C(N(C)CC2CCN(C(=O)C=CC3CCOCC3)C2)=O)cn2c(n1)CCCC2 52712,N1(C(C=NOC)=O)Cc2nccn2CC(NC(c2cccc(C(F)(F)F)n2)=O)C1 52713,c1(C(N2CCCC(n3cc(C(C(C)C)O)nn3)C2)=O)ccc2ncn(C)c2c1 52714,C1(C)(CC(=O)NC(c2ccccn2)CC)CCN(C(=O)CCN2CCOC2=O)C1 52715,Cc1cc(C(=O)NCCN(CC(C)O)C(=O)CSS(C)(=O)=O)c(O)c(C)c1 52716,N1(Cc2cccc(N3CCC(COCCOC)C3)n2)CCNC(=O)C1 52717,c1(OC)cc(Br)c(CNC(=O)C(C2CCS(=O)(=O)CC2)F)cc1C 52718,c1(OC)ccc2cc(C(N3CCC4(CCN(C(=O)C5CC5)CC4)C3)=O)n(C)c2c1 52719,N1(C(c2c(C)nc(CO)nc2)=O)CCN(C(c2ccccc2O)=O)CC12CCC2 52720,C1(CC(N2CCCC(CNC(c3[nH]cc(C(N)=O)c3)=O)C2)=O)CN2CCN1CC2 52721,C(=O)(CCCCC(F)F)NC(C)CCNC(C1(CF)CCOCC1)=O 52722,N1(C(C(c2ccccn2)C)=O)CCCC(C)(CN=c2[nH]nc(CC(F)(F)F)s2)C1 52723,CC1CC(NC(=O)Cc2ccnn2C)CN1C(=O)Cc1coc(-c2cccs2)n1 52724,N1(CCCNC(CC=CC)=O)CCN(C(c2cccc(C3CCC3)c2)=O)CC1 52725,C(F)(F)(C(F)(F)F)OC.c12ccc(cc1)C(=O)OC2C(=O)OC 52726,c1(C(=O)NC(CNC(c2nc(OCC)sn2)=O)(C)C(C)C)ccc(N)c(C)c1F 52727,n1(CC)nc(C(=O)NCC(C)C(=O)NCCC2COC(C)(C)C2)cc1C 52728,Cc1[nH]nc(C(F)(F)Cl)c1C(=O)NC1CC(C)N(C(=O)CC(=O)NC2CC2)C1 52729,C1(C(N2CCC(OCCNC(CC3CCC(=O)NC3)=O)C2)=O)Cc2cscc2C1 52730,C1(NC(c2ccc(F)c(Cl)c2F)=O)CCC12CCN(C(C1CCC(O)C1)=O)CC2 52731,c1(C(C)(C)CN2CCC(n3ccc(C(F)(F)F)n3)CC2)ccc([N+](=O)[O-])[nH]1 52732,CC(CN(C)C)CC(=O)NCCCCCNC(=O)CCc1nncnc1O 52733,C1(C(=O)NCC(C)OCC#C)CCOCCN1C(c1nc(C)ccc1F)=O 52734,N=c1cc(C(N2CCN(CC3CN(C(=O)C=CI)C3)CC2)=O)cc[nH]1 52735,C1(C)(C(=O)NC(C)C(C)NC(C2(CO)CCCC2)=O)SCCCS1 52736,C#CC1C(C(N2CCC2CNC(=O)CN2CCC(O)CC2)=O)C1(C)C 52737,C(=O)(CC(O)CC(C)C)N(CCOC)CCNC(=O)Cn1nc(C)nc1C 52738,Cc1c(C(=O)NC23CCC2CN(C(c2cc(Br)n(C)n2)=O)C3)nn(C)c1N 52739,Cc1c(Br)csc1C(N1CCCC1Cn1cc(C2OCCO2)nn1)=O 52740,n1(CC(=O)NCC2C(NC(C=C(C)C3CC3)=O)COC2)ncn2nccc2c1=O 52741,c1(C(=O)NCCC(C)(C)NC(C2CCC(C)S2)=O)ccccc1-c1ncnn1C 52742,N(C(=NCCC1CCC2(CCC2)O1)NCC(F)(F)Cl)C1CCS(=O)(=O)C1 52743,C1(NC(=O)Cc2cncnc2)CC12CCC(NC(c1cc(Cl)cs1)=O)CC2 52744,c1(N2CC(C)(CC(=O)Nc3cccc(C(F)(F)F)c3Br)C2)ccn2nccc2n1 52745,CC1(NC(=O)C(=O)NC(C)(CC(F)(F)F)CO)CCOC1 52746,N1(C(c2sccc2I)=O)CC2CC2(C(=O)NC(CO)C2CC2)C1 52747,c1(C(C(=O)NCCCCCNC(=O)CC(C)c2ccco2)OC)ccc(Cl)cc1 52748,c1(SC)cc(OCC2CCCN2C(c2cn(C3CCCCC3)nc2C)=O)ccn1 52749,C12(C(=O)NCCn3ncc(C(=O)NC(COCC)C)c3)C=CC(CC1)C2 52750,Cc1ccc(C(N2C3CN(C(c4cnn(C)c4C(F)(F)F)=O)CC23)=O)c(F)c1 52751,CCCC(C(=O)N1CC(NC(c2cc[nH]n2)=O)CC(O)C1)S(N)(=O)=O 52752,C1(NC(=O)Cn2cccn2)CN(C(C2CC3(C2)CC3F)=O)CC12CCC2 52753,C(=O)(CC(C)(C(F)F)N(C)C)NCCN(C(C1(C)CCC(=O)N1)=O)CC 52754,CC12CCC(C(=O)NCC3(O)CN(C(=O)Cc4ccc(Cl)c(Cl)c4)C3)(CC1)CO2 52755,CC1CC(C)C(CNC(C23CC(CF)(CO2)C3)=O)CN1C(=O)C1=CCCCC1 52756,c1(C(=O)NC2CN(C(C(CC)C(C)C)=O)CC2O)cc(F)c(F)c(Cl)c1F 52757,c1(NC(CNc2c(CCC)n[nH]c2)=O)cn(CC(C)C)nc1C1CC1 52758,C(CC(=O)N(C)CC1(CO)CC1)(C(C)(C)C)NC(c1cc(C)c(=N)[nH]c1)=O 52759,c1(C(=O)NCC(C)N(C(C(CC)CCOC)=O)C)cc2c(OC)ccc(C)c2[nH]1 52760,C(=O)(CC(C)N(C(=O)COC1CC1)C)NC(CC#C)C 52761,CN1CCC2C(CCCN2C(COC(C)(C)C)C(=O)NC2(C)CC2)C1 52762,C1(C(=O)OC)CCCN(C(=O)C(C)C)C1.C1(OC)C(=O)N2CC1C2 52763,O=[N+]([O-])c1cc(S(=O)(=O)N2C(C(=O)N=c3cc[nH]cc3O)CSC2)ccc1Cl 52764,c1(C(=O)NCC(CC)(CC)NC(C2CC(C)(C)C2)=O)ccc(C)c(OCCF)c1 52765,c1(OC)cnc(C(=O)NCC2CCC2NC(c2cccc(C(C)C)c2)=O)c(C)c1 52766,c1(SC)cn(C)nc1C(=O)NC1CC1CNC(c1ccc(CN(C)C)cc1)=O 52767,c1(C(N2CCCC(C(C)NC(CCOCCC)=O)C2)=O)nnc(O)cc1O 52768,c1(COC)ccccc1COCC(=O)NC(C)CNC(C1CCC1)=O 52769,C1(C(=O)NCC(CN(C(c2c(OC)noc2C)=O)C)C)CCCCCC1(F)F 52770,N1(C(C=Cc2ncn(C)c2)=O)CC(C2CC2C(=O)NCC2(C3CC3)CC2)C1 52771,c1(CNC(N(C(CCC)C)CC)=O)ccc2ocnc2c1 52772,c1(C(=O)NCC2(NC(C(C)NC(C)=O)=O)CCCCC2)cc2c([nH]1)CCOC2 52773,C(=O)(C1=CCCCC1C)NCC1CN(C(C2(C(=O)OCC)CCC2)=O)CC1O 52774,n1(CCC=C)c(CCCSC2CCCCC2)nnc1-c1nc(C2(C)CC2)no1 52775,C1(CNC(C2CCC(CC)O2)=O)(NC(=O)CC(C)(C)C(C)=O)CCC(C)(C)CC1 52776,CC1(C)CCN(C(C2(C#N)CC2)=O)CC1NC(=O)CCCOCc1ccccc1 52777,O=C1CC(C(=O)OC(c2cccc(F)c2)c2ccccc2)=NN1 52778,N1(C(c2ccc(C#C)nc2)=O)CCN(C(C2CC2(F)F)=O)CC(O)C1 52779,C1(NC(Cc2nc(C)[nH]n2)=O)CC(=O)N(C2CN(CCC(=O)NC3CC3)C2)C1 52780,CN1CC2(C1)N=C1C=CC(Br)=C(N1)C(CC)c1c2cccc1 52781,CC(C)C(C(=O)N1CCCC1CCNC(=O)C(F)OC(F)(F)F)NC(N)=O 52782,Cc1ccc(C(CNC(c2cnc(S)n2C2CC2)=O)NC(=O)CC(C)F)cc1 52783,C1(C(N(C(CC(=O)OC)C)C)=O)(NC(=O)CCn2ccnc2C)CC(F)(F)C1 52784,C12(C(N3C(CO)CC(NC(Cc4n(C)nnc4)=O)C3)=O)CC=CCN1CCC2 52785,CCCCCCCCC(CCCCCC)C(=O)NCC1CCN(C(=O)CC)C1 52786,c1(CCC(=O)NC(CNC(c2ncccc2F)=O)CO)ccc2cccnc2c1 52787,C=O.N(CCCCOC)(N(C(=O)C1CC1)CC)C(=O)C1CC1 52788,N1(C(C(C)n2cnnn2)=O)CCC2CN(C(C3(c4cccc(F)c4)CC3)=O)CC12 52789,c1(O)ccc(S(N)(=O)=O)cc1.c1(N(C(=O)CN(C)C)CC)ncc(CCCOC)cn1 52790,Cc1ccc(C2CC2NC(=O)Cc2nc(C(C)(C)C)ns2)cc1C 52791,N1(C(C2(OC)CC2)=O)CC(CNC(C2(C)CC(F)(F)C2)=O)OC(C)(C)C1 52792,c1(C(=O)NCCN(C(CS(CC)=O)=O)Cc2ccccc2)cc(C#N)cc(C)n1 52793,C(c1ccc(Br)s1)=C(C(c1nnnn1CCC1CC1)NCC(CC)(C)C)C 52794,C1(CNC(=O)NC2N(C(CCC)=O)CCCC2)(CO)CC2CCC1C2 52795,CN1CCn2nc(C(=O)NCC3CCN3C(c3cccc([N+](=O)[O-])c3)=O)cc2C1 52796,Cn1cc(CC(N2CCCC2CCC(=O)NC2C=CCC2)=O)nn1 52797,CCC(C)(C(=O)NC1CCC(NC(c2ccnc(C)n2)=O)CC1)C(N)=O 52798,c1(C(N(CC(=O)NCc2c(CC)nns2)CC)=O)ccc(C)n1C 52799,N1(C(C2C(CC)CCC2)=O)CCN(C(c2ccc(C)c(O)c2)=O)CC1C 52800,N(C1CCC=Cc2ccccc21)c1cc(NC(c2ccc(Br)cn2)C)ncn1 52801,C1(N(C)C)CCCN(C(C2CN(C(=O)CC3CCCC4CC34)CCO2)=O)C1 52802,CC1(C)CC(CC(=O)N(CCCNC(c2cscn2)=O)C2CC2)C1 52803,Cc1c(CN2CCN(C(C3(F)CNCC34CCC4)=O)CC2)oc2ccc(Cl)cc12 52804,C(C)(C(CCc1ccccc1)NC(=O)CCF)NC(c1ccc(C)s1)=O 52805,c1(C(N2CCC(C(NOCC)=O)C2C(C)C)=O)cnn2cccc2c1 52806,Cc1c(C(=O)NCC(F)CNC(=O)C(C)(Cl)Cl)oc2cc(Cl)ccc12 52807,C(=O)(C1=CCCCC1C)NCC(C(=O)NCC1CC(SC)C1)C 52808,N1(C(CCN(CCC)C)=O)CC2CCCC2(C(=O)NCC(C)C(C)(C)C)C1 52809,C1(NC(Cc2nc(C)oc2)=O)C2CC3C1C3C2C(=O)NC(CF)C(F)(F)F 52810,c1(OC)ccc(C(=O)NCCCCCN(C(=O)C2=CCC(C)CC2)C)c(O)c1F 52811,C1(NC(C(=O)NCCOC)=O)(CO)CCCN(C(=O)C(C)(C)CCSC)C1 52812,N1(C(CSCC(C)C)=O)CCOC2(CCN(C(=O)CC3CN4CCN3CC4)C2)C1 52813,c1(C(=O)NC(CCN(C(Cc2cc(CC)no2)=O)C)C)c(C)noc1C 52814,S(=O)(=O)(c1ccc(NCCC2(C)OCCO2)cc1Cl)NCCCC 52815,c1(OC(C)C(=O)NC2CCCN(C(=O)CCCF)C2)ccccc1Br 52816,C1(NC(c2cccc(CO)c2)=O)CC2(CCN(C(=O)C=Cc3cccs3)CC2)C1 52817,N1(c2nc(C)c(Br)cn2)CC(C)CN(C(C2C3CCCC23)=O)CC1C 52818,N1(C(C2C(C)(C(=O)O)C2)=O)CCOCC1Cc1cn(C2CCCC2)nn1 52819,N1(C(C2CCN(C(C=CCC)=O)C(C)C2)=O)CCCN(C=O)CC1 52820,c1(C(=O)NC(CC=C)CNC(=O)C(C)OCCN(C)C)ccc(O)nc1Cl 52821,N1(C(CCCn2cc(-c3cn(CC)nc3)nn2)=O)CCCC(CC(N)=O)CC1 52822,N1(Cc2c(C)nn(C3CCOCC3)c2Cl)CC=C(c2ccnn2C)C1 52823,c1(N2C3CN(C(C(CC)(C)CC)=O)C(CC3)C2)ccc([N+](=O)[O-])c(O)n1 52824,c1(NC)snc(C)c1C(=O)NC1CCC(NC(=O)CCc2ccc(O)nc2)CC1 52825,N1(C(C(C)=C(CC)C)=O)CC(OC)CC1(C)CNC(c1ccc(C)cc1N)=O 52826,N1(C(c2c(N(CCC)C)cccc2)=O)CCC(NC(c2cnsc2C)=O)C(C)C1 52827,N1(C(c2c(Cl)ccc(C)c2)=O)CCC2CN(C(C3(C(C)C)COC3)=O)CCC2C1 52828,c1(CN2CCCC(NC(=O)COC(F)(F)C(F)(F)F)CC2)cc2ccccc2o1 52829,Cc1cc(C)c(C(N2CC=CC(NC(c3ccsc3)=O)C2)=O)c(Cl)n1 52830,C(=O)(C1=CC2(CCOC2)C1)NCCC1(NC(c2c(C)c(Br)no2)=O)CCC1 52831,CC(C)C(F)(F)CC(=O)N1CC(CNC(c2c[nH]c(C(N)=O)c2)=O)CC1C 52832,c1(SCC(=O)NCC(C)CN(C)C(c2c[nH]ccc2=N)=O)ccsc1[N+](=O)[O-] 52833,N1(CC(=O)N(C2CC(NC(=O)CCC3CCCO3)C2)C)C(=O)C(=O)N(C)C1=O 52834,CC(C)CCCCC(=O)N1CCC2CN(C(=O)CS(=O)(=O)Cc3cccs3)C2C1 52835,CCCCC(O)CCC(=O)NC(C1CCN(C(=O)CN2CCC(C)CC2)CC1)C 52836,CCCC(O)CC(=O)NCCN(C(=O)C(c1ccc(CC(C)C)cc1)C)C 52837,N1(C(CCOCC(C)C)=O)CCC(NC(C2CC(n3cnnc3)C2)=O)CC1 52838,CC1(NC(c2ncc(Cl)nc2Cl)=O)CCCN(C(c2cscn2)=O)C1 52839,N1(C(c2c(C)cn(C)n2)C(=O)NCC(C)C)CCC(O)C(CC(C)C)C1 52840,C1(C(=O)NC2C(C)CN(C(C3(O)CCOC3)=O)C2)CCC2(CCC2)CO1 52841,C(=O)(C(CCNC1CC1)NC(=O)COc1cnn(C)c1)NC(C#C)CC1CC1 52842,N1(C(C(C)SC(F)(F)F)=O)CCOCC(NC(C2(c3ccno3)CCC2)=O)C1 52843,c1(C(=O)NC(c2ccc(CNC(=O)C(O)CN(C)C)cc2)C)cnc(O)n(C)c1=O 52844,N1(C(C(C)CC2CCCC2)=O)CCC(C2CC2)(CNC(=O)COCCF)C1 52845,Cc1c(C(=O)NC2(CCNC(=O)C=Cc3ccoc3)CC2)cc(F)cc1Br 52846,c1(NC(CNC(Cc2cc(C)on2)=O)C(C)C)ncnc2sccc12 52847,C1(C(=O)NCCN(C(C2CC2F)=O)CC)(CO)CCCC1 52848,Cc1nnc2cc(NCCN(C(=O)Cc3cccc(Cl)c3F)C)ncn12 52849,C1(N(C(CC2CC(=C)C2)=O)C)CN(C(=O)C(C(=O)ON)OC)CC1(C)C.CC 52850,C1(NC(CS(C)(=O)=O)=O)CN(C(=O)C=Cc2cccc(F)c2)CCC1O 52851,C1(NC(c2nc(CCC)oc2)=O)C2CC3CN(C(=O)CC4=NNC(=O)C4)C1C3C2 52852,CC(CC(=O)N(CCCNC(=O)CCC1CC(F)(F)C1)CCO)C1CCCO1 52853,c1(CC(=O)NCC(CO)NC(=O)CCc2nncs2)c[nH]c2cnc(Cl)cc12 52854,Cc1ccc([N+](=O)[O-])c(OCC(=O)NC2CC(CNC(=O)C(F)=CC3CC3)C2)c1 52855,C(=O)(C1=CCCCC1P(C)(C)=O)N1CC2(OCCN(C(C(C=C=C)C)=O)C2)C1 52856,c1(C(=O)NC(c2cn(Cc3ccc(Cl)nc3)nn2)C)cn2ccccc2n1 52857,c1(NCc2cn(-c3ccc(C(C)(C)C)c(Br)c3)nn2)ccc(C#N)c(F)c1 52858,C1(C(=O)NCCCNC(=O)CC2CCCO2)(Cc2cccs2)CCCCC1 52859,C(CNC(C1C(CNC(C2(N3CCCC3)CC2)=O)C1(C)C)=O)(C(F)(F)F)OC 52860,c1(C(N2CC(C(C(=O)NC(C(C)C)C3CC3)OC)C2)=O)cc(O)cc(=O)o1 52861,C1(C(N2C(C(C)NC(=O)CN3CCCNC3=O)CCC2)=O)COC2CCCCC12 52862,N1(C(c2c(C)nc(CSC)s2)=O)CCC(NC(=O)C(C(C)C)NC(C)=O)C(O)C1 52863,CC1(C)CCC(CNC(C23CC=CCN2CCC3)=O)N(c2nnccc2C#N)C1 52864,C1(C(=O)NC(C2(O)CN(C(C3(CC4CC4)CC3)=O)C2)C)CC12CCCCCC2 52865,Cc1ccc(F)cc1C(N1CCN(C)CC1CNC(c1nccn1C(C)C)=O)=O 52866,n1(COC)ccc(C(=O)N(CCC(C)NC(=O)CCCNC(=O)C2CC2)C)n1 52867,C12(CNC(CCCN(C)C)=O)CCC(CC1)CN2C(=O)C(c1ccc(F)cc1)O 52868,c1(CC(=O)NCC23OCCC(NC(C(CC)C#N)=O)(C2)C3)nc2ccccc2s1 52869,N1(C(c2c(Cl)ccc(C)c2)C(=O)NC2CCC2)CCCC1C1CCCO1 52870,C(C(F)C(C)(C)O)NC(c1nc(C(C)NC(=O)CCc2ccsc2)oc1)=O 52871,C1(NC(Cc2ccc(SCC)cc2)=O)CC2CCC(C1)N2C(=O)C(C)(Cl)Cl 52872,Cc1ccc2[nH]c(C(=O)NCC(O)CCNC(=O)CCC(C)C)cc2c1 52873,C1(NC(C(C)SC)=O)CCN(CC2CCCCO2)C(C)C1 52874,N1(C(c2c(C)n(C)cn2)=O)CCCC(C)(C)C1C(=O)NC(c1nncn1C)C 52875,C1(N2CC(C)C(NC(c3ccc[n+]([O-])c3)=O)CC2)CCc2ccccc2NC1=O 52876,c1(C(N2CCCC(C)(NC(C3C(C)C3)=O)C2)=O)cncc2ccsc12 52877,c1(OC)ccc(-c2n[nH]cc2CN2CC(C(=O)OC)CC(CN(C)C)C2)cc1Cl 52878,N1(C(c2ccc(O)c(O)c2)=O)CC(C(N2CC3COCC3C2)=O)CC(F)(F)C1 52879,c1(NC(c2[nH]cc(COC)c2)=O)cccc(NC(C2(C)CCCO2)=O)c1 52880,N1(C(c2ccc(OCCO)c(F)c2)C(=O)NC)CCOC(C(F)(F)F)C1(C)C 52881,c1(Nc2cc3c(cc2)OC(C)C3)nccc(=NC2CCCn3nccc32)[nH]1 52882,N1(C(c2csnc2Cl)=O)CC2OCCN(C(C3CCCN4CCCCC34)=O)C2C1 52883,C1(CC(=O)NCC2CCN(C(=O)CSC(F)F)C2)CC(O)C12CCC2 52884,C1(C(=O)NCC2(NC(CCNS(CC)(=O)=O)=O)CC2)CC12CCC1(CC1)CC2 52885,c1(COCC)cccc(NC(=O)C(c2ccc(Cl)cc2)OC(CC(C)(C)C)=O)c1 52886,C1(C(=O)OC)CC2CN(C(=O)C(N3CCCC(O)C3C(=O)OC)=O)CC12 52887,c1(OCC)ccc(NC(=O)CN2CCC(c3ccccc3F)C2)cc1 52888,C1(C(N2CCC(NC(Cc3cc(C)no3)=O)C2)=O)CCCCC1c1nncn1C 52889,N1(C(c2[nH]cc(C#N)c2)=O)CCCCC(CNC(=O)C=CC(F)(F)F)C1 52890,c1(C(N2C(CNC(C(C(=O)NC)(C)C)=O)CC(O)C2)=O)cc2[nH]nc(C)c2cn1 52891,C1(C(=O)NC2(C#C)CC(F)(F)C2)C(C2CC2)CCN1C(=O)C=Cc1ccoc1 52892,N1(C(c2n(CC)cnn2)=O)CCC2(CCCC2NC(c2ccc(C)s2)=O)C1 52893,C(C(CC(C)C)NC(c1cccnc1CO)=O)NC(C(COC)C)=O 52894,c1(CCC(=O)NCC(C)NC(=O)C(F)(F)c2ncc[nH]2)nnc(C2CCCC2)o1 52895,C1(OC)CN(C(=O)CCC2CCC(C(N)=O)O2)CC1NC(c1cccc(Cl)c1)=O 52896,C1(C(=O)NCCNCCN(C)Cc2ccccc2Cl)COc2ccccc2O1 52897,N1(C(C(c2n(C)cnc2)O)=O)CC2(CCC(NC(c3ccccc3)=O)CC2)C1 52898,C(=O)(CC(C)CC(F)(F)F)NC1CCC(NC(c2nn(CC)c(C3CC3)c2)=O)C1 52899,c1(NC(C2C3(CN(C(Cc4nnc(C)o4)=O)C3)C2)=O)cc(Br)cnc1I 52900,c1(SCC2(C)C(C(C)O)C2)ccc(C2CC2)cc1 52901,C(=O)(CC1CCc2ccccc21)NC1CCN(C(c2snc(C)c2N)=O)C1C 52902,C(=O)(CS(=O)(=O)C1CC1)N1CCC(NC(CC2C=NN(C)C2=O)=O)C1 52903,CCCC(C(=O)NCCCCCNC(=O)C=Cc1cn[nH]c1)S(N)(=O)=O 52904,C(=O)(C(C)(C)CCCC(=O)N(C1CN(C(c2nc(Cl)c(Cl)s2)=O)C1)C)OC 52905,C1(CNCC(c2ccc(Br)cc2)C)CCC2(C1)CC2(F)F 52906,C1(CS(C)(=O)=O)(C(CN2CC(N(C)C)C2)=O)CCCC1 52907,C1(NC(CCc2cc(C)on2)=O)CN(C(=O)CN2CC(C)(C)C2)CC(C)(C)C1 52908,Cc1nc(C(N2CCN(C(c3c[nH]cc(F)c3=O)=O)CC2C(C)C)=O)cc(O)n1 52909,c1(C(N2C(CNC(=O)CC3CC4CCC3CC4)CC2)=O)c(F)cc(F)cc1Cl 52910,CC(N=c1ccc(Br)c(S(=O)(=O)N2CC=C(Br)CC2)[nH]1)c1cccc(F)c1F 52911,N1(C(C(Cc2c(C)n[nH]c2C)C)=O)CCCC2(NC(c3n[nH]cc3Cl)=O)CC2C1 52912,N1(C(CSC)C)CCC2(CC1)OCCc1sc(C(N3CC(F)(F)C3(C)C)=O)cc12 52913,C1(CNC(CCC)=O)CN(C(C2CCCCC23CC3)=O)CC12CCC2 52914,N(C(=NCCCF)NCCCS(=O)(=O)CC1CC1)C1C(C)(OC(C)C)C1 52915,C#Cc1cccc(C(=O)NCC2CCN(C(=O)CC3CCCC3)CC2O)c1C 52916,c1(N2C(C)CC(NC(c3c(C)cc(Cl)cc3)=O)C2)cc2nnc(C)n2cn1 52917,C(=O)(C1=CC(C)(C)C1)NC1C=CCN(C(C(c2ccc(N)cn2)C)=O)C1 52918,C(CS(=O)(=O)CC(=O)N(C)CC1CCCN(C(c2ccc(OC)s2)=O)C1)OC 52919,Cc1cc(C(=O)NC(Cn2ccnn2)C(=O)NCC2(C)CCCC2O)nn1C 52920,C(CC(C)(C)CBr)(c1nnnn1C(C)C)NCC(C)C(F)(F)F.C1CN1 52921,C1(CC)COCC1NC(=O)C(C)(C)NC(=O)C(C)=CC(C)(C)C 52922,c1(C(=O)NCC2N(C(C(CC)OC)=O)CC2)ccc([N+](=O)[O-])cc1C(F)F 52923,N1(C(C(C)Cc2cnc[nH]2)=O)CCC(C)(CNC(=O)CCc2nncs2)C1 52924,C1(NC(C2C(OCC)C2)=O)CC1C1CCCN(C(c2cccnc2Cl)=O)C1 52925,c1(OCC)nc(C(=O)NC(C)(C)C(C)NC(=O)C(C)NC(=O)C(C)(C)C)ns1 52926,C(=O)(CC(C)C(C)C(C)C)N1CC(C(C)(C)O)(CNC(C(CCCC)C)=O)C1 52927,C1(C(=O)NC(C(=O)OC(C)C)C)CC2(C1)CC(N=c1ncnc3[nH][nH]c(I)c1-3)C2 52928,C12(CNC(c3ccc(-c4ncc[nH]4)nc3)=O)CC1CN(C(c1coc(O)n1)=O)C2 52929,c1(C(N2CC(NC(C(C)NC(C)=O)=O)C(F)C2)=O)cc(Br)c(F)cc1Cl 52930,c1(C(N2CCC(C(C(=O)NCC(CC)(C)C)F)C2)=O)nn(C)cc1C 52931,C1(NC(N(C2CCCC2C#N)CC(C)C)=O)CC2C=CC1CC2 52932,c1(OC)ccc(Br)c(C)c1C(=O)NC1CCN(C(c2cc(C)c(C)cn2)=O)C1 52933,C(=O)(C1=CC(C)CC1)N1CCC(N(CCOC)C(c2cc(C)ccn2)=O)CC1 52934,C1(C(N2CCCC(N(C)C(c3scnc3Cl)=O)C2)=O)CCc2cncn2C1 52935,c1(COC)cc(CC(=O)N(CC(C)NC(c2c[nH]nc2C(C)C)=O)C)no1 52936,C(=O)(C(C)(C)C(F)F)N1CC(OCCNC(c2cc(C)c(C)s2)=O)C1 52937,c1(NCC(=C)C)cc(N2CCCC(OCC)C2)nc(C(F)(F)F)n1 52938,N1(C(c2n(C)nnc2)=O)CC2(CC2)CC1CC(=O)NCC1(C)CC1(F)F 52939,CC1CN(C(=O)C(C)(C)NC(=O)CCNS(C)(=O)=O)CC2(CCN(CC#N)C2)O1 52940,N1(C(C2(CF)CCN(C(C(C)C#N)=O)C2)=O)C2CCC1CC1(C2)N=N1 52941,C(=O)(CCCN(C)C)N(C(C)C(=O)NCC1(CO)CCCC1)C 52942,CC(C)C(O)CC(=O)NC12CC(NC(=O)CCC3(C)CC3(F)F)(C1)C2 52943,c1(CCC)nc(=NC(CNC(=O)C(C2CCCCCC2)OC)CO)s[nH]1 52944,CC1(CNC(=O)CCCCNC(N)=O)CCCN(C(=O)C(F)OC(F)(F)F)C1 52945,c1(C(N2CCCC(N(C(=O)C#CC3CCC3)CCO)C2)=O)cn2ccccc2n1 52946,c1(-c2cncc(NC(c3c(C(C)=O)c(C)ccc3)=O)c2)c(F)cc(CO)cc1F 52947,c1(C(C(=O)NC2(NC(C3C=CCC3)=O)CC2)O)cc(F)c(F)c(F)c1 52948,C1(N(C(c2c(COC)ncs2)=O)C)CC2CCC(C1)N2C(c1ccc(F)s1)=O 52949,C1(CC2(CNC(C3(O)CC3)=O)CC2)CN(c2ncns2)CCC12CCOC2 52950,C(=O)(N=c1cc[nH]cc1I)NC(C1(F)CC1)C 52951,N1(C(CSCC=C)=O)CCCC2C1CCN2C(=O)COCC1(F)CC1 52952,CC(C(=O)NC(CNC(=O)CCCn1c(O)nnc1O)C(C)(C)C)C(C)(F)F 52953,C1(NC(COC)=O)CN(C(C2(C(F)F)CC(Nc3cc(OC)no3)C2)=O)CC1F 52954,c1(C(=O)NC2C(CC)N(C(c3cc(C)nn3CC)=O)CC2)ccnc2[nH]nnc12 52955,c1(CC)nn(C)c(NC(=O)NC2CC2c2cccc(F)c2F)c1Cl 52956,Cc1cc(C(=O)NC2CC3CCC2(NC(C2CC(C)(C)C2)=O)C3)nc(O)c1 52957,C1(C(N2CC(C)=C(C)CC2)=O)N(C(c2cn(C3CC3)cn2)=O)CC12CCCC2 52958,O=C1CC(CC(=O)N2CCC3(CC2)CC3NC(c2ccsn2)=O)=NN1 52959,C1(CNC(Cc2cnn(C)n2)=O)CC2(CO1)CN(C(c1nc(Cl)ccc1N)=O)C2 52960,N1(Cc2c(Cl)ccc(Cl)c2)CCc2c(Cc3ccccc3)cccc21 52961,CC1=C(C(=O)N2CCCCC(CNC(c3cnc(-c4ccoc4)s3)=O)C2)CCC1 52962,C1(CC(=O)N(C2CCN(c3nnc(C4CC4)s3)C2)C(C)C)(COC)CCCC1 52963,C(=O)(CC(C)CN(C)C(=O)NCc1cc(C)nn1C)OC 52964,C1(C(=O)OC(c2ccc(Cl)cc2)C)CCC(=O)C(C)C1 52965,C(CCCCCNC(C1OC2CCC1C2)=O)n1cc(-c2cc(C(=O)OC)on2)nn1 52966,c1(CC(=O)N(CCNC(=O)CCc2cnc[nH]2)C2CC2)ccc(Cl)nc1 52967,N#Cc1ccnc(N2CCN(C(C3CCN(Cc4n[nH]cc4Cl)C3)=O)CC2)c1 52968,CC1CN(C(C23CC2COC3(C)C)=O)CCN1C(c1[nH]cnc1C#N)=O 52969,CCCCC(C)C(=O)N1CC2(CC2)CC1CNC(=O)CCCN1C(=O)CNC1=O 52970,C1(CC)CCCCC1C(=O)NCc1ccc(CNC(C2CCCC(=O)N2)=O)cc1 52971,C1(NC(C(Cc2ccccc2Br)NC(CCC=C)=O)=O)CC2CC1CC2CO 52972,c1(CN(C)C(=O)NCCCCC(=O)NCC(F)(F)F)ccc(F)c(Cl)c1 52973,C1(CNC(c2c(CC)nccc2)=O)CN(C(C2CCC(C)CO2)=O)CCN1C 52974,Cc1cc(C(=O)N(C2CCN(C(=O)CSc3n[nH]c(=N)s3)CC2C)C)nnc1C 52975,C(=O)(C1CCCc2nc(C)[nH]c21)NCCN(C(=O)C(C)n1ccnc1)CC 52976,C1(N(C(C2(CN(C)C)CCCC2)=O)C)CCCN(C(C2CNC(=O)C2)=O)CC1 52977,C1(NC(C2(C(C)C)CCC2)=O)CN(C(c2ccc(N)c(Cl)c2)=O)CCC1CO 52978,C(=O)(C(O)CC(C)C)NC(C(=O)NCc1c(C)cccc1)c1ccco1 52979,C1(CN2CCCC(C(N3CCN(C)CC3)=O)C2)CN2CCC1CC2 52980,C1(C(=O)NC2(CC=C)CCC2)CCC(CNC(=O)C=Cc2nc(C)cs2)CC1 52981,C(=O)(C1CNc2ccccc21)NCC(CNC(C(C)OCC)=O)O 52982,C1(N(C)C(C2CCCS2)=O)CCCN(C(=O)COC2CCCCC2)C1 52983,N1(c2n(C)nnn2)CC2CC(NC(C3CN(C4CCOC4)C3)=O)C2C1 52984,C(=O)(CCCC(F)F)N1C(CNC(=O)CCc2nc(C3CC3)no2)CC(OC)C1 52985,c1(CN2CCC(CNC(C3C(C)C3)=O)C2)ccc2ccc(Cl)cc2n1 52986,C(C)(C(O)C(=O)N1CC(CO)(NC(=O)Cc2cccc(C)c2)C1)SC 52987,C1(C(CNC(C2(CC)CCOC2)=O)C)CCN(C(c2cccn2COC)=O)CC1 52988,c1(CC(=O)NCCOCCNC(c2cc(O)cs2)=O)csc(-c2ccsc2)n1 52989,C1(C(C)C)CCCN(C(=NCC2CCN(C)C(=O)C2)NCC2CCCCO2)C1 52990,c1(C(=O)NC(CCNC(C(C)n2ccnc2)=O)(C)C)cc(F)cc(S(N)(=O)=O)c1 52991,c1(C(=O)NCCOC2CCN(C(CCNC(C)=O)=O)C2)c(Cl)ccc2c[nH]nc12 52992,Cc1c(C(=O)N(C)CCOCCNC(=O)CN2CCC(C)CC2)cccc1Cl 52993,N1(C(C(C)CN2CCOCC2)=O)CCC2CN(C(c3cc[nH]c3)=O)CC12 52994,c1(CC(=O)OC)ccc(C(=O)NC(C)(C)C(C)NC(C2CC23CCC3)=O)cc1 52995,CCS(=O)(=O)CC(=O)NCC(CC(F)(F)F)NC(c1cnc(CC(C)C)[nH]1)=O 52996,c1(NC(=O)NC(C(=O)OC(C)(C)C)CO)ccccc1-c1cnc(F)cc1 52997,CC1CC(C(=O)NC(C)(C)CN2CCN(c3ccccc3)CC2)C1(C)C 52998,c1(N(C(=O)COC)CCS)cc(C)ccc1C 52999,C1(C(CC)C(=O)N2CC(N(C)C(C3CCCO3)=O)C2)CCC(C)CC1 53000,C1(NC(=O)NCCCCCO)C2Cc3ccc(Br)cc3C12 53001,C1(C(=O)NC(C2(O)CCN(C(C3(C)CC(=O)C3)=O)C2)C)CCCOCC1 53002,N1(C(CC2CCCN(C(CC(CC)(C)C)=O)C2)=O)CCn2ccnc2C1C 53003,c1(C(c2n(CC)nnn2)NC2CCCC2CCOC)cccc(C)c1C 53004,c1(C(=O)NCC23CC(NC(=O)COc4ccsc4)(C2)C3)ccc(F)cc1F 53005,c1(OC)cnc(C(=O)NC2CCC2CNC(=O)COC2CCOC2)cn1 53006,N1(C(CCCNC(N)=O)=O)CC2CCC(C1)N2C(C1CC1c1ccc(Cl)cc1)=O 53007,C1(c2n(C(C(=O)OC)C)nnn2)(NCCS(=O)(=O)CCO)CC2(C1)OCCO2 53008,Cc1cc(F)c(N)cc1C(=O)NC1CC(F)CN(C(c2nnc(O)nc2O)=O)C1 53009,CC(C)CC(C)C(=O)NCCCN(C)C(c1nccc(Br)c1O)=O 53010,CC(C)C(C(=O)NCCC(C)NC(c1ccn(C(C)C)n1)=O)C1CCC1 53011,N1(C(c2c(CC)cc[nH]2)=O)CCC(CO)C(NC(C2(CCF)CCC2)=O)C1 53012,C(C(C(=O)N1CCCC1CNC(C)=O)C(C)(C)C)NC(CC(=O)OC)=O 53013,N(C(=NCCCCl)N1CCCC2(CCCOC2)C1)Cc1cccc(C#N)n1 53014,CCCCC(C(=O)NC)NC(=O)CCC1(NC(=O)CCn2cccn2)CCCC1 53015,CN1CCC(C(=O)NC2CCCN(C(=O)CC(C)(C)c3cccs3)C2)C1=O 53016,S(=O)(=O)(c1cccc(F)c1C)N1CCCC(CNC(c2ccc(C(C)N)cc2)=O)C1 53017,C(=O)(CC(C)CC(F)(F)F)NC1CN(C(c2c(OCC)nccc2)=O)CC12CC2 53018,c1(CC)ccc(C(N2CCNC(=O)C2)C(=O)NCCC2CC2)nc1 53019,C1(NC(CC(C)N2CCCC2=O)=O)C2CC1CN(C(c1ccc(Cl)c(Cl)c1)=O)C2 53020,c1(CCC(=O)N(CC(COC)C(=O)OC)CC(=O)O)cnc2ccccc2c1 53021,N1(C(CCNC(C2(O)CCSCC2)=O)=O)CCC(O)(CO)CC1 53022,c1(C(N2CC(CNC(c3cc(OC)nn3C)=O)OCC2)=O)cc(C#N)[nH]c1C 53023,c1(C(CCC(=O)NCCCCC(C)NC(CSC)=O)=O)cc(C)ccc1C 53024,CN1CCN(C(C2C3CCC(=O)C23)=O)C(CNC(c2ccno2)=O)C1 53025,C1(NS(CC(C)C)(=O)=O)CC2CCC(C1)N2C(=O)C(C)(C)C 53026,c1(CC)ccc(C(=O)NCCC2CC(NC(=O)C(n3cc(Br)cn3)C)C2)o1 53027,c1(OC(C)(C)C)cnc(NC(c2ccc(-c3cccc(C#N)n3)cn2)=O)c(F)c1 53028,c1(SC)cc(C(=O)N(CC(O)CN(C)C(c2ccc(C)cc2)=O)C)c(Cl)cc1Cl 53029,CCC(C)CC(C)N(C(=O)C(CCOCCO)NC(=O)C=CC(F)(F)F)C 53030,c1(CC(=O)NCC2C(CNC(CC(C=C)C)=O)C2)cccc(O)c1F 53031,c1(C(=O)NCCN(C(=O)C(C)(C)N(C)C)C)cccnc1N1CCCC1 53032,C(CC(C)C(=O)NC(CNC(c1coc(CS(C)(=O)=O)n1)=O)CO)=CC 53033,C1(C(N(C2(C(=O)NCC(C)C)CC2)C)=O)CCC(C)(C)OC1 53034,N1(C(CC(COC)C)=O)CCCC2(C1)CN(C(=O)CC(C)CN(C)C)C2 53035,C1(CNC(=O)CC2C=CCC2)CCC(CNC(=O)CN2CCCC2=O)CC1 53036,c1(C(=O)NC2(C)CCN(C(C3C(C)C3C)=O)C2)cc(O)nc2ccc(F)cc12 53037,CN1C(=O)C(=O)N(CC(=O)NC2CC2NC(C2CCC(N=[N+]=[N-])CC2)=O)C1=O 53038,c1(OCCCC(=O)NC2CC(CNC(c3c(CC)n[nH]c3)=O)C2)cccc(F)c1 53039,C(=O)(C(C)CC1CCC1)NCC(CC)NC(=O)CSCc1cccs1 53040,CCC(C)(C(=O)NCC1(C(C)NC(=O)CC2C(C)(C)C2(C)C)CC1)OC 53041,n1(CC)ccc(=NC(=O)C2C3CC2N(C(=O)C(c2ccnn2C)O)C3)[nH]1 53042,n1(CCC(=O)NCCCN(C(C(C)=C(C)C)=O)C2CC2)nc(C)cc1C 53043,O=C(CNC(=O)COCCCF)N=c1ccn(CCF)[nH]1 53044,C1(C(=O)NC(CN(C(=O)C=NOC)CC)C)CCN(c2cnccn2)CC1 53045,N1(C(C2C(C)C2C)=O)CCC(NC(C2(c3ccno3)CCC2)=O)C1C 53046,c1(NC(=O)NC2CCCN(C3CCCC3)C2)ccc(F)c(Br)c1F 53047,c1(C(=O)NC(C(C)NC(CCc2c(C)noc2C)=O)C(C)C)cc(Cl)ncc1O 53048,C=CCC(CC=C)C(=O)N1CCCC(C)C1CNC(c1cnc(S)nc1)=O 53049,C(CC1CC1)(C(=O)N(C)CCC1CCCN1C)NC(CC1CC(C)C1)=O 53050,c1(OCC(N2CC(CNC(C(n3c(C)cc(C)n3)C)=O)C2)=O)ccc(Cl)c(F)c1 53051,Cc1c(Cl)ccc(C(=O)NC2CCC(N(C(=O)COCC(C)(C)C)C)C2)c1N 53052,c1(C(=O)NC2(CC#C)CCCN(C(=O)OC(C)(C)C)C2)cc(Br)cc(O)c1C 53053,Cc1nc2ccc(C(=O)NC(CNC(C3CC(=O)N(C)C3)=O)C(C)C)cc2s1 53054,c1(C(=O)NCCNC(CC2CC(C)(C)OCC2)=O)cc(Br)cn2ncnc12 53055,C12(NC(CC3(CSC)CC3)=O)CCCC1N(c1nc(C(C)(C)C)ns1)CC2 53056,c1(C(=O)NCC2(CCNC(CC(CC)CC)=O)CC2)[nH]c2cc(C)ccc2c1C 53057,C(CCS(=O)(=O)NCC(=O)NCCOC1CCN(C(=O)C=NOC)C1)OC 53058,C#Cc1ccc(OCC(=O)NCCNC(=O)CC2CC(CC)=NO2)cc1 53059,N1(C(C2OCCN(C)C2)=O)CC2CC(C1)C2NC(=O)CCN(S(C)(=O)=O)C 53060,CC(CCCO)N=c1[nH]c(N2CC(C)OC(C)(C)C2)nc2c1SCC2 53061,c1(C(=O)NCC(C)(C2CC2)NC(c2ccnc(C3CC3)n2)=O)cc(F)cnc1O 53062,C1(NC(C(C2CCCC2)OC)=O)CCN(C(C2CCCC(OC)C2)=O)C1(C)C 53063,CC1(C)CC(NC(=O)CC2COCC(C)(C)O2)CN(C(c2coc(CO)c2)=O)C1 53064,Cc1cc(C(=O)Nc2nc(Cl)cc(Cl)n2)cc2nc[nH]c12 53065,c1(OC)ccccc1C1(C(=O)NC(C)CNC(=O)OC(C)(C)C)CCC1 53066,c1(CC)cc(CC(=O)NC2(CN(C(=O)C(C)(C)C3CCCCC3)C)CC2)n(C)n1 53067,c1(C(=O)NC2CC(C)(CC)N(C(=O)CNC(N)=O)C2)ccc(OC)c(F)c1N 53068,n1(CC(=O)NCCC(CC)(CC)NC(C(CC)C)=O)ccc(=O)c2ccccc12 53069,Cc1c(C(=O)NC2CCCC2NC(=O)CC2(N(C)C)CC2)cnc2ncnn12 53070,CC(C)(O)C#CC(=O)NC1CN(C(=O)COCC(C)(C)C)CC1(C)C 53071,N1(C(C=C(C)C(F)F)=O)CCCCC(CNC(=O)Cc2nc(C(C)(C)C)cs2)C1 53072,Nc1cc(F)c(C(N2CC=CC(NC(=O)C3=CCCC3)C2)=O)c(F)c1 53073,CC1(C)CN(C(c2ccn3nncc3c2)=O)C(CNC(C2(C)CC2(F)F)=O)CO1 53074,c1(C(N(C)CCOCCNC(=O)CCC(N)=O)=O)coc2c(F)cccc12 53075,CCCCC(CC(=O)NC(COC)CCO)NC(C1(C2(C)CC2)CC1)=O 53076,C12(C(=O)NCC3(CNC(c4c(CCC)nco4)=O)CCC3)CC3CC1C2C3O 53077,c1(C(=O)NCC2C3CN(C(CCC(N)=O)=O)C2CCC3)cc2cccc(F)c2o1 53078,c1(CC)n[nH]cc1C(=O)NCCCCCN(C)C(c1cn(C(F)F)cn1)=O 53079,c1(C(N2C(CNC(CC(=O)N(C)C)=O)CC2)=O)cc(CO)ccc1Cl 53080,N1(C(Cc2ccc(C(C)C)cc2)=O)CCN(C(c2ncccc2F)=O)CC1C#N 53081,c1(CC(=O)NCC(CC)NC(c2cc(O)cc(N)c2C)=O)ccc([N+](=O)[O-])cc1 53082,N1(C(C(C(C)C)NC(C)=O)=O)CCCN(C(c2sc(F)cc2Cl)=O)CC1 53083,c1(CCC)cccc(C(N2CC(NC(=O)C3=NOCC3)C(O)C2)=O)c1 53084,C1(O)(CCNC(c2cnc(O)c(Cl)c2)=O)CCCN(C(c2ccncn2)=O)C1 53085,Cc1cccc(Br)c1C(=O)Nc1cccc(CNC(c2c(C)nn(C)c2C)=O)c1 53086,c1(C(C(=O)OC(c2cccc([N+](=O)[O-])c2)CC)=O)cc2c(cc1Cl)OCCO2 53087,Nc1ccc(C(=O)NCC2(NC(C3CCOC3C3CC3)=O)CCC2)cc1Cl 53088,c1(OC)ccc(CCC(=O)NC2CN(C(=O)Cc3c(C)cccc3Cl)C2)c(F)c1 53089,CC(CCO)C(=O)N1CCC(CNC(c2ccc(Cl)cc2)=O)C1 53090,C=CCC(CNC(c1ccc(C#N)n1C)=O)C(=O)N1CC(C)(COC)C1 53091,N1(C(C(=O)NCC)=O)CCC(NC(c2cn(CC(N)=O)nn2)=O)C(F)C1 53092,C12(C(N3C(CCC)CCC3)=O)CC1CN(C(C1(O)CCCCC1)=O)C2 53093,CCCC(CCC)CC(=O)N1CCC(O)C1C(=O)NCC(O)C1(Cl)CC1 53094,C1(CC)CCCN(C(=O)C(COC)CNC(C2CCC=CCCC2)=O)CC1 53095,c1(NC(CC2N(C(C(CC)CC)=O)CC(O)C2)=O)cc(C#N)cnc1C 53096,c1(C(=O)NC(CNC(c2nnc(C)s2)=O)C(C)C)cccc(S(=O)(=O)CF)c1 53097,C1(c2ccccc2)(NC(CC2CC(C)C2)=O)CC(NC(=O)C(C)CO)C1 53098,C1(C(=O)NCc2cnc(C)s2)CC(O)CN1C(C1CC1[N+](=O)[O-])=O 53099,C1(NC(C(C=CC)O)=O)C(C)(C)C(NC(=O)CCc2scnc2C)C1(C)C 53100,C=C(C)CCCC(=O)Oc1cc(NC(CC)=O)c(-c2nnc(C)o2)cc1 53101,c1(C(N(CCC)CCNC(c2ccc(OCF)cc2)=O)=O)cc(N)ccc1O 53102,S(=O)(=O)(CC(=O)NC1CN(C(c2cnc(N3CCCCC3C)s2)=O)CC1C)NC 53103,c1(C(=O)NC(C)CNC(C2(C)CCCCC2)=O)cncc(F)c1Cl 53104,N1(C(C(C=CC)O)=O)CC2(C1)CN(C(c1ccc(Cl)cc1C)=O)CC2CO 53105,N1(C(=O)NC(c2cc(C3CC3)no2)C)CC(C)OC2(CCOC2)C1 53106,C1(C)(C(N(C)CC2CN(C(C3CCCC3)=O)CCO2)=O)CCCCNC1=O 53107,c1(-n2cc(C3(C)CN(C(Cc4scc(CC)n4)=O)C3)nn2)ccc(Cl)cc1 53108,c1(C(N(C)CCN(C)C(c2cc(C(N)=O)c[nH]2)=O)=O)cc(C(F)(F)F)n(C)n1 53109,CC1=C(C)CC(C)(NC(=O)C(C)CN(C)C(c2cc3ccncc3[nH]2)=O)CC1 53110,N1(C(CCCC=C)=O)CC2(CCN(C(=O)Cc3csc(CC)n3)CC2)C1CCOC 53111,Cc1cccc(C)c1C(C(=O)O)NC(c1nc(N(C)C)sc1Cl)=O 53112,C1(C(N(CC)CC2CCCN2C(=O)CP(C)(C)=O)=O)OCC2CCCC12 53113,c1(C(=O)OC)nc(C(=O)NCC2(NC(=O)C(CO)N(C)C)CCC2)co1 53114,C(=O)(C(O)CC(C)C)N1CC(N2CCN(C(c3c(C)nns3)=O)CC2)C1 53115,C=CC(C)(C)C(=O)NCCOC(C)(C)CNC(=O)C(C1CC(F)(F)C1)OC 53116,c1(C(=O)OC)cc(C(=O)NCC(O)CN(C)C(c2ccn(C)n2)=O)c(C)s1 53117,C=CCC(CC)C(=O)NCC1CN(C(c2nonc2CC)=O)CC1C 53118,c1(C(=O)NC2CN(C(COC(C)(C)C)=O)C3C2C3)cc(S(N)(=O)=O)ccc1Cl 53119,N1(C(c2nc(CNC(C3C(=C)C3)=O)oc2C)=O)CCCC2C1CCN2C 53120,C1(C(=O)NC(CCCC)CNC(c2cc3cscc3s2)=O)CCCC(F)(F)CC1 53121,C1(C)(CCNC(CN(C(C)=O)C)=O)CCN(C(c2sccc2Cl)=O)C1 53122,C1(C(=O)NCC(COC)C)CCN(C(=O)CC2C(C)(C)C2(C)C)CC1O 53123,C1(CNC(COCc2nc(C)sc2)=O)CC2CCC1N2C(=O)C(C)(C)C1CC1 53124,c1(SC)nn(C)cc1C(=O)NCC1(O)CN(C(=O)C=C(C2CC2)C2CC2)C1 53125,C=CC(C)(O)CC(=O)NCCOC1CCN(C(=O)CCC2CCC(=O)NC2)CC1 53126,N1(C(C(C(C)O)C)=O)CC(C)(C)OC2(C1)CN(C(c1nnn3c1COCC3)=O)C2 53127,C1(NC(C(CC)n2cccn2)=O)CCCCCN(C(=O)C=Cc2cnc[nH]2)C1 53128,Cc1ccc(F)c(C(N2CC(OCC(=O)NCC3CC(C#N)C3)C2)=O)n1 53129,c1(CC)nc(C(N2CCC2c2cn(CCCN3C(C)CCC3C)nn2)=O)c(C)o1 53130,c1(C(=O)NC2(CCOC)CCN(C(c3ccns3)=O)CC2)cnc2nccn2c1 53131,C(CN=c1nc(-c2ccccc2)nc[nH]1)(N(C(C(CCC)C)=O)C)C1CC1 53132,c1(N2CCCC(CC=C)(C(=O)OCC)C2)nc2c(cc1C#N)CCC2C 53133,N1(CC(N2CC(CNC(=O)Cc3ccsc3Br)C2)=O)CCCNC1=O 53134,N1(C(=O)Cc2csc(S)n2)CCCCC2(C1)CN(C(C1CC=CCC1)=O)C2 53135,CCC(CC)C(F)C(=O)N1CCC(CC(N2CCCNC(=O)C2)=O)C1(C)C 53136,c1(OC)ccc(C#N)cc1NC(C1CCCC1NCc1occc1Br)=O 53137,C1(CCCNC(C2N(CC)CC2)=O)CCN(C(=O)CCC2CCC(=O)C2)CC1 53138,C1(C(N2CCCC(SC(C)(C)C)C2)=O)CC(c2ccccc2[N+](=O)[O-])=NO1 53139,C(C(=O)NNC(=O)c1cc(-c2nn[nH]n2)on1)OC(c1ccc(C)cc1)C(C)=O 53140,N1(C(c2c(C)cno2)=O)CC(NC(c2c(Cl)cncc2Cl)=O)CC(O)C1 53141,C(COC)(N=c1cc(C)nc(NC(C)C2CC2)[nH]1)c1ccc(CC)o1 53142,N(C1CCc2c(Cl)cc(Cl)cc21)C1CCC(Oc2ccc(C)cn2)CC1 53143,C1(NC(C=CSC)=O)CCCC(N(C)C(c2cc(N(C)C)ccn2)=O)C1 53144,C1(CC)C(NC(C2(CO)CCCO2)=O)CCN1C(=O)CCC(=O)OC(C)(C)C 53145,N1(C(C=CC(=O)OCC)=O)CCC2(C1)CN(C(C1(C)CCOC1)=O)CCO2 53146,c1(CC)nc(C)cc(=NC(CCN(C)C(C2CC3(CCOCC3)C2)=O)C(C)C)[nH]1 53147,C1(C(=O)Nc2c(OC)cccc2Cl)CCC(N=c2ccn3ncc(Br)c3[nH]2)CC1 53148,C1(CCC(=O)NCC(CC)N(C)C(C2CC(=O)N(C)C2)=O)CCCCN1C 53149,NS(=O)(=O)c1ccc(CN2CCSC(C(N3CCCC4(CCO4)C3)=O)C2)cc1 53150,C1(C)(C(N2CCOCC(NC(CSCCC)=O)C2)=O)CCCNS1(=O)=O 53151,C(=O)(C1CCCc2scnc21)N1CC(O)CCC(NC(c2n[nH]c(C)c2C)=O)C1 53152,N1(C(C(CSC)OC)=O)CCCC(N(C(=O)Cc2cc(C)cs2)CC2CC2)C1 53153,Cc1oc(Cl)nc1C(=O)NCCCCC1CN(C(=O)C(=O)NCC(F)(F)F)C1 53154,C1(C#N)(C(=O)NCCC2CN(C(c3c(C)n(C)nn3)=O)C2)CCOCC1 53155,c1(-c2scc(C(=O)Nc3cc(Cl)ccc3Br)n2)c(F)cc(F)cc1F 53156,C1(CC)CN(C(C2(C(N)=O)CC2)=O)CCC1NC(=O)CCc1ncc[nH]1 53157,CC(C)C(F)(F)CC(=O)NC1CCCC1NC(c1cc(Cl)cn1C)=O 53158,c1(COC)cnc(OC)c(C(N2CC(CNC(C3(C4CC4)CC3)=O)CC2C)=O)c1 53159,c1(OC)c(C(N2CCC(C(N3CC(O)C3)=O)C2)=O)cnn1-c1ccccc1 53160,Cc1nc(CCC(=O)NCCC2CCN(C(c3c[nH]nc3C(C)(F)F)=O)C2)cs1 53161,c1(OC)ccc(CN(C)C(=O)NC2CCCOC2c2cn[nH]c2)c(OC)c1 53162,C1(NC(C(NOC)=O)=O)C2CCC1CN(C(=O)COc1cccc(C)c1)C2 53163,C1(CONC(C2C3CC4C(C3)C24)=O)CCCCN1C(C1CCCCC1O)=O 53164,CC1CN(C(=O)C(C)(C)C(F)(F)F)CC(C)C1NC(=O)C(c1ccc(F)cc1)=O 53165,N1(C(C(C)NC=O)=O)CCC(CCNC(c2cc(CCO)on2)=O)C1 53166,c1(C(N2C(C)CC(CNC(CC3CC(=C)C3)=O)C2)=O)ccc2nccn2n1 53167,n1(CC)ncc2c(NC3(CNC(=O)CC(C)(O)C4CC4)COC3)ncnc12 53168,C1(CC(=O)NC2CCN(C(COCCOCC#C)=O)C2)CCCN(S(C)(=O)=O)C1 53169,N1(C(=O)OC(C)(C)C)CCC2CCN(C(C3CC3c3ncccc3Br)=O)C2C1 53170,C1(O)(C(N(CCCCNC(=O)C(C)(C)c2ccccc2)C)=O)CC2CCC1C2 53171,C1(C(=O)NCC(CN(C(C2(CC=C)CC=CC2)=O)C)O)CC(F)(F)C1(C)C 53172,c1(C(=O)OC(C#C)C)ccc(-n2nc(C)cc2C)c(F)c1 53173,c1(C(=O)NCC(CNC(C2C(C)C2)=O)O)cc([N+](=O)[O-])cnc1O 53174,c1(OC)cnc(C(N2CC=CC(C(N3CCC3C(=O)N(C)C)=O)C2)=O)cn1 53175,CC1(C)C(C(N2CC(O)(CNC(=O)C(F)=C3CCCC3)C2)=O)C1(F)F 53176,C1(NC(c2scc(OC)c2)=O)COCCN(C(=O)C(F)(F)c2cnccn2)C1 53177,C(=O)(C(O)C(F)F)OC(CC(C)C)C.C1CCC(C)NC(=O)O1 53178,N1(C(c2ccc(C(C)C)nc2)=O)CCCC(NC(c2ccn(C)c2)=O)C1C 53179,c1(C(N2CC(C)C(C)(CO)C2)C(=O)NCCC)cc(Cl)c(Br)cc1F 53180,N1(C(C2=CCCC2C)=O)CCC(C(=O)NCC2CC3CCCC3C2)C12CCC2 53181,c1(C(=O)NC(C)C(C)NC(C2(CCO)CC2)=O)cnc(-c2ccccn2)nc1 53182,N1(C(c2n(C)ccn2)=O)CCCC1(C)CNC(=O)CC1(c2ccon2)CCC1 53183,C#Cc1ccc(C(=O)NCCC(C)CCNC(=O)CSc2ccccn2)c(C)c1 53184,N1(C(C23C(C(=O)OC)(CCC2)C3)=O)CCCCC(NC(C2(C)CC(C)(C)C2)=O)C1 53185,c1(OC)c(C(=O)NCCC(C)NC(C2(C)COC(=O)N2)=O)cnn1C 53186,C1(NC(CC2N(C(c3n(CC)ccc3)=O)CC(O)C2)=O)CCCCC1(C)O 53187,N1(C(CC=CC=C)=O)CCCC2(CNC(C34CCC(C)(C3)OC4)=O)CCCC12 53188,C(CCC(=O)NCC1CCCCC1)(C(C)C)NC(c1nccc(C)c1N)=O 53189,Cc1ccc2c(N3CCCC3CCCNC(c3ccc(Cl)cc3)=O)ncnc2c1 53190,c1(C(N(CCC(C(C)C)NC(c2ccoc2)=O)C)=O)cccc2nc(CO)[nH]c12 53191,n1(CC)cc(C(=O)NCC(C)NC(=O)CCC2NC(=O)NC2=O)c2ccccc12 53192,c1(-c2cc(Br)cc(SC)c2F)cn2c(n1)CN(C(=O)OC(C)(C)C)CC2 53193,N1(C(CSCC)=O)CCc2ccccc2C(NC(=O)CC2(COC)CC2)C1 53194,c1(CNC(=O)CC2(O)CNC2)ccc(CNC(=O)C(c2ccccc2)F)cc1F 53195,CCC(C)(C)C(C(=O)N(C)CCOCCN(C)C(C1(SC)CCC1)=O)OC 53196,c1(C(C)NC(c2c(C#C)c[nH]n2)=O)cc2ccccc2n1C 53197,C1(CC(=O)NCC2CN(C(C(OC)OC)=O)C(C)(C)C2)NC(=O)CN(C)C1=O 53198,C1(F)(CNC(C2Cc3cccnc3C2)=O)CCCN(C(C2(CO)COC2)=O)CC1 53199,c1(N2CCC(CCC)C2)nc2ccccc2c(=NCC(F)(F)Br)[nH]1 53200,C1(C(=O)NCCOC2CCN(C(c3cc(CO)on3)=O)C2)CCc2nc[nH]c2C1 53201,N1(C(CCC=C)=O)CCC2CCCN(C(=O)CSCc3ccccc3)C2C1 53202,Cn1cc(C2CC(C(N3CCC(N4CCOC4=O)CC3)=O)C2)c(C(F)F)n1 53203,N1(C(CNS(NC)(=O)=O)=O)CCCOC(CNC(=O)C(C2CCCCCC2)O)C1 53204,N1(C(c2c(CC)con2)=O)CC2CC1CC2NC(c1cc(C(=O)OC)co1)=O 53205,c1(C(C)N2C3(CCC3)CC2=O)cc2ccccc2o1.C1(O)(COC)CCCCC1 53206,Cn1cc(C(=O)NCC23CC2CN(C(=O)COCc2nc[nH]n2)C3)cc1Br 53207,N1(C(C(=O)Nc2cnc(OC)nc2)=O)CCn2c(C(C)(C)C)nnc2C1 53208,C(=O)(C(CCC)=CCC)NC1C(NC(C2(C=C)CC2)=O)CC1 53209,c1(SCCC)ccc(C(=O)N(C)CC2(C)CC2)o1.C1(=O)C(CC)N(CC)N1 53210,c1(CC2CCN(C(c3c(CN)occ3)=O)C2)ccc(Cl)cc1 53211,c1(C(=O)NCC2(CNC(CCN(C(CCC)C)C)=O)CC2)csc(Cl)c1Cl 53212,Cc1nn2c(C(=O)NCCCCNC(=O)C(C)C(C)C)c(C)nc2s1 53213,Cc1cc(=NC(=O)Cc2csc(=NCc3ccc(I)c(O)c3)[nH]2)[nH][nH]1 53214,N12CCCC(C)(CC1)CN1CC(COC)(C1)C2=O.C1(C)(C(=O)OC)CCCCC1 53215,c1(C(N2CCC(CC=C)(NC(C3COC(C)C3)=O)C2)=O)cc2ccccc2cn1 53216,c1(C(=O)NCCC(C)NC(c2c(CC)ncnc2)=O)c[nH]nc1[N+](=O)[O-] 53217,C1(CNC(CCCCN(C)C(c2ccn(C)c2)=O)=O)CCCC(C)(C)C1 53218,C1(OC)(OC)CC2(CC(NC(=O)NCCc3ccccc3)C2)C1.C1CCCN1 53219,CC(CCNC(C1CCC(C(N)=O)CC1)=O)CCNC(=O)C(c1ccnn1C)C 53220,C(C)(C)(CCCCNC(=O)CC1CC2CCC1O2)NC(C1CCN(CC)C1)=O 53221,c1(C(=O)NCc2nc(CNC(C3C(C)(C)C3)=O)sc2)cc(S(N)(=O)=O)ccn1 53222,C1(NC(C2(C#C)CN(C(=O)C(C)C#N)C2)=O)CCOCC12CCC2 53223,C1(C(=O)NCC(N(C(c2cnc(C(C)C)s2)=O)C)C2CC2)CCC(=O)N(C)C1 53224,N1(C(c2cn(CC)nc2)=O)CCC(C(=O)NCC2CC(CC(N)=O)C2)C12CCC2 53225,N1(C(c2c(CC)c[nH]n2)=O)CC(C)(C)CC1CC(=O)NCCC1(C)CC1 53226,c1(C(C)=O)ccc(C(N2CC(NC(c3c[nH]nc3OC)=O)CC2CO)=O)cc1C 53227,N1(c2nc(SC)nc(C)c2)CCC2CC(CNC)CCC2C1.C(=O)(C(C)C1CC1)NO 53228,O=C1CC2CC(C(N3CCC(C(=O)NC4(CO)CC5(CCC5)C4)C(O)C3)=O)C1O2 53229,CC1CN(C(c2cc(Cl)cn2C)=O)CCCN1C(C1CCc2n[nH]cc2C1)=O 53230,CCCC(C)CC(=O)N1CCCC(CNC(c2ccc(-c3cc[nH]n3)s2)=O)CC1 53231,Cn1cc(Cl)c(C(=O)NCC2CCN(c3ncncc3Cl)C2)n1 53232,c1(C(N2CC(COC)(CNC(=O)C(F)(F)C3CCCC3)C2)=O)ccnc(C)c1O 53233,C1(NC(C(C)n2ccnn2)=O)CCC(C)(NC(C2COCCOC2)=O)CC1 53234,C1(CC)CCN(C(=O)C(F)F)C(C(=O)NCC2(C)CCCOC2)C1 53235,N1(C(c2c(C)ocn2)=O)CCN(C(=O)CNC(c2ncn(C)n2)=O)CC1 53236,c1(CC)cc(NC2CC(NC(=O)CCC(C)C)C2(C)C)ncn1 53237,C(=O)(C(O)C(F)(F)F)N1CC(N(C)C)C(NC(=O)CC(=O)NCC2CC2)C1 53238,c1(C(N2C(CNC(=O)C(O)C3CC3)CC(O)C2)=O)cnn2c1OCCC2 53239,C1(N(CCC(C)C)C(=O)CN2CCCC2CO)CCN(C(=O)C2CC2)CC1 53240,N1(C(c2cnc(CCC)s2)=O)CCCC(N(C)C(c2ccn(C(C)C)n2)=O)CC1 53241,C12(C(=O)NC3CC(NC(c4c(Cl)ccc(C)n4)=O)C3)C3C4C1C1C2C3C41C(N)=O 53242,N1(C(C(C)C2CCCC2)=O)CC2CCC1C2NC(c1ccc(Cl)c(O)c1)=O 53243,Cc1ccc(C=CC(=O)NC2CCN(C(C3CS(=O)(=O)CCO3)=O)CC2F)nc1 53244,N1(C(CC2C(C(=O)OC)CC2)=O)CCC(OCC2CC2)C1 53245,C=CCCCC(C(=O)N1CCn2ncnc2C1)NC(c1cc[nH]c1C)=O 53246,Cc1c(CC(=O)NCCCNC(=O)CC2C=CCC2)cccc1[N+](=O)[O-] 53247,c1(CC)cc(C(=O)NCC(C(C)C)NC(=O)C(C2CCC2)OC)ncn1 53248,CC12CCN(C1)C2=O.C1(OCC(=O)NCC(F)(F)F)CC(=O)N1 53249,C1(OC)CC2(C1)CC(C(=O)NC1CC3CC1N(C(=O)C(O)CSC)C3)C2 53250,C1(NC(C2CCN(C(c3cn(CC=C)nc3)=O)C2)=O)CCN(C)CC1C#N 53251,C1(C(=O)NC(C)CC2CCOCC2)CCC(C)N1C(=O)CC1CC1C1CC1 53252,C(CCN=c1[nH]c(N2CCOC(CF)C2)nc2c1SCC2)OCC(C)C 53253,c1(CNC(C2CC(O)CN2C(c2nccnc2Br)=O)=O)ccc2cc[nH]c2c1 53254,Cc1cccc(C(=O)N(C)CC2CCCC2NC(C2(O)CCC(C)CC2)=O)c1N 53255,N1(c2ncc(OCC)cn2)CC(C(=O)O)C2(CCN2S(=O)(=O)CCBr)C1 53256,C1(NC(C2C(C)CCC2)=O)(CNC(C2CC(F)(F)C2)=O)CCOCC1 53257,C1(CNC(C2CN(C(=O)CO)CCO2)=O)COc2ccccc2O1 53258,C(c1cncnc1O)=CC(=O)NC1CCC(N(C(C=CSC)=O)C)C1 53259,C1(CC(C)NC(c2cn(C3CCOC3)nn2)=O)CCN(C(=O)CSC(F)F)CC1 53260,C1(C(=O)NCC(C)CC2CC2)CCC2CCC1N2C(=O)Cn1cnnc1O 53261,c1ccc2c(c1)CCC(n1nc(C3CCOC3)nc1-c1n[nH]c3c1CCC3)CC2 53262,CC(CC(=O)NOC(c1ccccc1)CNC(=O)C(F)(F)CO)C1CCCC1 53263,C(=O)(CC(C(F)(F)F)OC)N1CC(F)(CNC(CC2(CC=C)CCCC2)=O)C1 53264,N1(C(C2(CC#C)CCCCO2)=O)CCC(Nc2ncnc(=N)[nH]2)C(F)(F)CC1 53265,C(=O)(C1=CC2CCCC12)N(C1CCN(C(c2c(O)cccc2O)=O)C1)CC 53266,N1(C(C(CCF)NC(C(CC=CC)C)=O)=O)CCCNC(=O)C1 53267,C1(F)(C(=O)NC2C3CN(C(CC(CC)C)=O)C2C3)CS(=O)(=O)CC12CCC2 53268,N1(C(C(CC2CCC2)NC(Cc2cccc(C#C)c2)=O)=O)CC(F)(F)CCC1C 53269,c1(OCCC)ccc(NC(=O)NCCOC2CC2(F)F)cc1OC 53270,Cc1sc2ncnc(N3CCC4CCC(NC(C5CCC(C)C5)=O)C3C4)c2c1C 53271,c1(C(N2CCC(CNC(CC(C)OC)=O)CC2)=O)ccc2c(c1)CC(C)(C)C2 53272,c1(CNC(=O)CCN2CCOC2=O)ccc(-c2ccccn2)cn1 53273,C=CC(F)(F)C(=O)N1CC2C(n3cc(-c4cc(C)nn4C)nn3)C2C1 53274,N1(C(c2cnn(CC)n2)=O)CCCC(NC(c2ccnc(Cl)c2O)=O)C1C 53275,C#CC1(COC)COCCN1C(C(=O)NC1CC(F)(F)C1)c1csnn1 53276,C1(C(N2CCSCC2C2CCC2)C(=O)NC2(C)CC2)CCOC2(CCOCC2)C1 53277,N1(C(CC(CC)O)=O)CC(C)CN(C(c2[nH]cnc2C)=O)CC1C 53278,Cc1c[nH]c(=NCCC2CCCN(C(c3ccnc4ccnn34)=O)C2)nc1O 53279,C1(C(=O)NCC(CN(C(=O)C(C)(C)N2CCCC2)C)(C)C)CCCCC1C(N)=O 53280,c1(CN(C(C(=O)N(C)C)=O)C)ccc(CNC(C2C3CCC2CC3)=O)cc1 53281,CC1CN(C(c2cc(C3CCCC3)no2)=O)CCCN1C(C1CCCCC1O)=O 53282,Cc1sc(O)nc1C(N1CCCC(NC(c2cnc(Br)s2)=O)C1)=O 53283,C(=O)(CCCCC(N)=O)NC(C1CCN(C(c2cc(Cl)c[nH]2)=O)CC1)C(C)C 53284,N1(C(C2CC(C)(C)C2)=O)CC2CCCC(NC(c3nc(Cl)c(Cl)s3)=O)C2C1 53285,C1(C(N(C)CCNC(c2cccc(=O)o2)=O)=O)CC(C)(C)OC1(C)C 53286,C(=O)(C(C)(C)S(C)(=O)=O)NC1CN(C(c2c(OC)c(F)ccc2)=O)CC(C)C1 53287,CC(C)CCC(=O)NC1CC1C(=O)NC1(NC(C2(C(=O)NC3CC3)CC2)=O)CC1 53288,C1(C#N)(C(CN2CCCC(N(CCN3CCOCC3)CC)C2)=O)CC12CCC2 53289,N1(C(Cc2n(C)cnn2)=O)CCN(C(=O)CCc2cccc(F)c2Br)C2CC12 53290,C1(C(N2C(C(N(CCC(C)C)C3CC3)=O)CC2)=O)CC(C)(F)C1 53291,N#Cc1ccc(=NCC(=O)N2CCC3(CC2)CC(NC(=O)C2=CCCS2)C3)[nH]c1 53292,C(CN=C(NCc1cc(Cl)ccc1Br)N1CCC(C2CCOC2)C1)N(CC)CC 53293,N1(C(CC(CC)OC)=O)CCC2(C=C(C(=O)N3CCN4CCCCC4C3)C2)C1 53294,c1(CC(N2CCCC(N(C(=O)CC(C)(C)F)C)C2)=O)noc2ccc(O)cc12 53295,Nc1c(C(N2CC(O)CCC2C(=O)NCc2ccc(F)cc2)=O)cccc1F 53296,C12(CS(=O)(=O)C1)C(=O)N2.C(C(C1CC1)N)SC.C1(CC=O)(NC(C)(C)C)CC1 53297,c1(CC)cc(N)c(C(N2CCCC(C)CC2)=O)cc1F 53298,c1(C(=O)NCC2(O)CN(C(C(CC)C(C)O)=O)C2)cnc2c(F)cccn12 53299,CC1(C)CCCCC1CCc1nc(C2CCCCCCC2)no1 53300,c1(NC(C)=O)ccc(C(=O)NC2(C)CCN(C(C34CCC3C4)=O)CC2)cc1Cl 53301,C1(C(N(C2CCN(C(C3CC3C#N)=O)CC2)CCC)=O)CN(C)CCO1 53302,c1(C(N2C(C(C)NC(C3ON=C(C)C3)=O)CCC2)=O)cc2cccnc2s1 53303,c1(CC)ncc(C(=O)NCCC2COCCN2C(=O)C(O)CCN(C)C)c(O)n1 53304,Cc1nc(N2CC(NC(=O)Cc3ccccc3Br)C3(CC3)C2)c2c[nH]nc2n1 53305,C1(NC(C=CC=CC)=O)CS(=O)(=O)CC1NC(C1(S(C)(=O)=O)CC1)=O 53306,C1(C(N(c2cccc(O)c2)CC)=O)CCC2CCC1N2C(=O)C(O)CC(C)C 53307,C1(C(N2CCC(CCC(=O)NC(C)C(=O)NCCF)C2)=O)CCNC(=O)C1 53308,C(=O)(C(CC(C)C)OC)NC1CC(C(=O)NCC(=O)OCCCC)C1 53309,CCCCC(=O)C(=O)N1CC(C)CC1C(N1CCCC(CN(C)C)C1)=O 53310,C1(C(N(C)CC2CCCN2C(c2ccc(Cl)o2)=O)=O)CC2CC1C1CC21 53311,C1(CNC(C(C)C)=O)COCC2(CCN(C(C3(F)CCC3)=O)C2)O1 53312,CCCCCC(=O)N1CCC(F)(CNC(=O)C(C(C)C)c2cnn(C)c2)C1 53313,C(=O)(C1CCCc2cn(C)nc21)NC(C)CCC(C)(C)O 53314,C1(C2CCN(C(c3cncc(Cl)c3)=O)C2)(NC(C(Cc2c(C)nc[nH]2)O)=O)CC1 53315,C(=O)(CCC(C)S(C)(=O)=O)NC1CN(C(c2c(C)nc(CO)s2)=O)CC12CC2 53316,C1(CNC(c2n(C)cnc2)=O)CCC(F)(CNC(C2(C)CCCNC2=O)=O)CC1 53317,N1(C(C(CCC)C(C)C)=O)CCC2(CC1)COC(CNC(c1cscn1)=O)C2 53318,c1(OCC)cc(CCCNC(N2CCCC23CC3)=O)cc(F)c1F 53319,CC(C)CCC(O)C(=O)NC1CCN(C(=O)C2=COCC2)CC(O)C1 53320,N1(C(c2c(C)scc2)=O)CCCC2(NC(=O)Cc3ccccc3[N+](=O)[O-])CC2C1 53321,Cc1oc(Br)c(C)c1C(=O)NC1CCC(C)N(C(C2CC(O)C2)=O)C1 53322,N1(C(C=COCC)=O)CCOCC1CN(C(C1(C)CC1c1ccccc1)=O)CC 53323,Cc1c(F)ccc(C(N2CCOCC2)C(=O)N(C2CC2)Cc2ccccc2)c1Cl 53324,c1(Nc2cccc(OCC(C(F)(F)F)OC)c2)cc(C)nc2c(F)cccc12 53325,C1(CC(N2CCCC(C)C2CNC(=O)C=C2CCCC2)=O)Cc2ccccc2N1 53326,N1(C(c2cn(C)nc2C(F)(F)F)=O)CC2CCC(C1)N2C(=O)CC1CCC1 53327,C1(C(N2CC(C(N)=O)(CNC(C3CC34CC4)=O)C2)=O)CC2CCC1C2 53328,N1(C(C2CC(CCC(=O)NCc3ccc(SC)o3)C2)=O)CCOCC1C(C)C 53329,Cc1coc(C)c1C(=O)NCC(C)CN(C(=O)CSCc1csc(=N)[nH]1)C 53330,n1(CC)nc(C)cc1C(=O)NCC1CCC1NC(=O)CCN1CCCCC1C 53331,CCC(O)C(C)C(=O)NCC(C)(C(C)C)NC(c1oc(C(F)(F)F)nc1C)=O 53332,c1(CC)nccnc1CNC(=O)C(C)(CSC)NC(=O)C=CC1(C)COC1 53333,Cc1cn2c(n1)C(C)CC(C(=O)NC1CCC1NC(=O)CCC(C)(C)C)C2 53334,N1(C(C(CC=C)CNC(=O)C=Cc2cncn2C)=O)CC2CCC(CC2)C1 53335,c1(C(N2CCC(C)(NC(c3n(C)c(S)nc3)=O)C2)=O)nc2c(s1)COCC2 53336,C(=O)(CCC(F)(F)CN=[N+]=[N-])NC1CC(C)(CNC(C=CCOCCOC)=O)C1 53337,CC1(C)CCN(C(C2CCCC(=O)N2)=O)C1CNC(C1(C(N)=O)CC1)=O 53338,C(=O)(CC1CCCc2ccccc21)NC1CC(CNC(C2(C)CC=CCC2)=O)C1 53339,C(=O)(C1=COCCC1)NCC1CCN(C(C(C(C)C)OCC(C)C)=O)C1 53340,N1(C(C(CC)=CC)=O)CC(NC(=O)CC(C)n2ccc(C)n2)C(C)C1 53341,n1(CC)nc2c(c1C(N1CC3CC1CN3C(=O)C(F)CCC(C)(C)C)=O)CCCC2 53342,CN1CCCC1(C)CNC(=O)Nc1nc(-c2ccncc2)cs1 53343,C1(OC)CC(C(=O)NCC(C)(C)CN(C)C(C2CCN(C)CC2)=O)C12CCC2 53344,C(=O)(C1=CCCN(C(c2ncccc2F)=O)C1)NC(c1ccc(O)nc1)C 53345,C1(C(=O)NC(c2ncc[nH]2)C)CN(C(=O)C(c2ccn(C)n2)C)CC12CCC2 53346,c1(OC)cc(NC(=O)C(C)N(C(=O)CC(C)n2ccnc2)C)ccc1F 53347,c1(C(N(C)CCOCCNC(C2COCC2c2ccccc2)=O)=O)cn(C)c(O)n1 53348,N1(C(C2C(CC(C)C)C2)=O)CC2CN(C(=O)C=CC3COC(C)(C)O3)CC2C1 53349,c1(N(CCC)CCNC(=O)CC2=NNC(=O)C2)cnc2cc(F)c(F)cc2n1 53350,n1(C(C(=O)N(CC(C)C)C(C)C)C)cc(CNC=O)nn1 53351,C1(OCC=C)CCN(c2nnc(C3CC3)n2CC2(O)CCSC2)CC1 53352,C#CCC(C)(C)C(=O)NCC(CC=C)C(=O)NCCN1CCCC1 53353,CC1=NN(C)C(=O)C1CC(=O)NCC1CC1CNC(=O)COCC1CCC1 53354,C1(C(N(C(C)CNC(=O)CC2COCCO2)C)=O)CCCCN1C 53355,N1(C(C(C2CC2)OCC)=O)CCC(CN(C)C(C2C(C(F)F)C2(C)C)=O)CC1 53356,C1(NCc2ccc(C(=O)OC)cc2)CC2(C1)CC(NC(c1cccnc1)=O)C2 53357,c1(OC)ccc(C(N2CCN(C(=O)CNC(C)=O)CC2)C(=O)NCCC#N)nc1 53358,C1(C(N(C(C)CNC(=O)Cn2ccnn2)C)=O)CCCC(=O)C1 53359,c1(C(=O)OC)cc(C(=O)NC2CCC2NC(=O)COC2CC=CC2)ccc1F 53360,N1(C(C(CC)COC)=O)CCCC2(CCCN2C(=O)C2=C(Cl)CCCC2)C1 53361,c1(NC(C2CCN(C(C=CCN(C)CC)=O)C2C)=O)cc(C)cnc1O 53362,C1(CCC)CC(C(=O)NC2CN(C(=O)Cc3cnco3)CC2C)CCO1 53363,CC#CCCC(=O)NC(CC1CCC1)C(=O)NCC(N1CCCCC1)C 53364,c1(C(=O)NC2CC(CNC(c3cnc(Cl)s3)=O)C2)nnc2ccccc2n1 53365,N1(C(C(N2CC(C)C2)C)=O)CCCCC1C(=O)NCCn1cccn1 53366,Cc1cc2c(CC(=O)NC3COCCC3NC(C3(C)CC=CCO3)=O)csc2s1 53367,N1(C(CCC2N(C(c3c(C)nc(C)[nH]3)=O)CCC2)=O)CC=C(c2ccccc2)CC1 53368,C(=O)(C1=C(C)OCCC1)NC1C(NC(c2nc(OC)c(F)cn2)=O)CCC1 53369,c1(SC)cncc(NC(=O)C(C)(C)C2CCN(C(=O)CC3CCC(=O)N3C)C2)c1 53370,Cc1ccnc2sc(-c3nc(CCCC#N)nn3CC3CC3C)c(C)c12 53371,c1(C(=O)NCCN(C(COCCOCCOC)=O)C)ccc(O)c(=O)o1 53372,CC1=CCC(C(=O)NCCCC2CCCCN2C(=O)C(F)=CC2CC2)CC1 53373,N1(C(Cc2scc(C)c2)=O)C2CCC1CC(NC(c1ccc([N+](=O)[O-])s1)=O)C2 53374,c1(CC)ccc(Cn2nccc2NC(C2ON=C(C)C2C)=O)cc1 53375,C1(C(N(CCCOC)CCO)=O)CCC(C)(C)N(C(=O)C(CO)C(F)(F)F)C1 53376,N1(C(C(COC)N(C)C)=O)CCCCC1C(=O)Nc1cccc(C)n1 53377,Cc1cc(NC(C2CC(CCNC(c3[nH]ccc(=O)c3C)=O)C2)=O)ccc1F 53378,C1(NC(C(CC)N(C)C)=O)CCC12CCN(C(c1oc(SC)cc1C)=O)CC2 53379,N1(C(C2C3CN(C(c4ccc(OC)cc4O)=O)C2C3)=O)CCCC2(COC2)C1 53380,N1(C(C(=O)NCCC)CC2CC2(Cl)Cl)CCOCC1(C)Cc1ccccc1 53381,C1(CC)CN(C(=O)CN2CCC(F)CC2)CC1C(=O)N(C)CCSC 53382,c1(C(=O)NCCCC(C)NC(C2(F)CC=CC2)=O)nn(C)c2c1CS(=O)(=O)CC2 53383,C1(C(=O)Nc2nc(C)ncc2Br)(OC)CCN(C(C2CC2F)=O)CC1 53384,N1(C(C2C(=C)C2)=O)CCN(C(C2C(C(C)=O)C2(C)C)=O)C(C2CCCC2)C1 53385,C1(N(C(C(C)N(C)C)=O)C)CCN(C(=O)CCc2ccco2)C1.C1(C)CCCO1 53386,C1(CNC(c2cccnc2)=O)(CF)CCN(C(=O)CSc2ccc(C3CC3)o2)C1 53387,c1(C(N(CCNC(c2c(C)nc(CCC)o2)=O)CCC)=O)cncc(Cl)c1C 53388,C(C(CC(=O)NCCC1CCC(C)(C)O1)NC(=O)C(O)CCSC)OC 53389,N1(C(CC2CC(OC)C2)=O)CC2CC1CN(C(c1cc(F)ccc1C1CC1)=O)C2 53390,C(=O)(CCC(C)N(C)C)NCC(=CC(=O)NCC1(COC)CCCO1)C 53391,c1(CC(N2CCCC(C)(OC)CC2)=O)ccc2c(c1)CC(C)O2 53392,C(=O)(CCP(C)(C)=O)N1CCC(N(CC#C)C(c2nc(C)oc2C)=O)C1 53393,CC1CCC2(CC1)NC(=O)N(NC(=O)CN(C)C(C1CCCCC1)=O)C2=O 53394,C(C(=O)N1CCN(C(C2CCCCN2CC(F)F)=O)CC1C)(C(C)(C)C)SC 53395,Cn1ccc(C(=O)NCC2CCCN(C(C3(C(F)F)CC3(F)F)=O)C2)cc1=O 53396,c1(C(C)(C(=O)NCC(CNC(=O)CCCC2CC2)CO)N(C)C)ccc(F)cc1 53397,N1(C(c2cc(N)c(Cl)cn2)=O)CCOC2CN(C(=O)CC3C=CCC3)CC12 53398,C(C(CCO)N(C)C)N(C)C.C1(C2=NOCC2)c2nnnn2CCCN1 53399,n1(CC)cc(NC(c2cc(C(OC(F)(F)F)=O)[nH]c2)C(=O)NCC2(CC)CC2)cn1 53400,N1(c2c(C)c(NCCC(C)(C)F)ncn2)CCC(S(=O)(=O)C(F)F)C1 53401,C1(C(=O)NC2C(C(N3C(C(=O)OC)CCC3)=O)CCC2)CC2C=CC1C2 53402,N1(C(C2(CC(C)C)CC2)=O)CC2ON=C(CNC(c3cn(C(C)C)nn3)=O)C2C1 53403,c1(C(=O)NCC2C(NC(c3cnc4[nH]cncc3-4)=O)C2)ccc(Cl)c(F)c1F 53404,N1(C(C=CCCC)=O)CC2CC(C(N3CCC(CO)C(C)C3)=O)C(C2)C1 53405,Cc1ccccc1C=CC(=O)NC1CC2(C1)CC2NC(C1CCC(=O)N1C)=O 53406,N1(C(CC(CC)(C)C)=O)CC2CC(CNC(=O)C(C)(C)SC)CC1C2 53407,CCC(CC(=O)NC(C)CCCNC(c1nc(C(C)C)oc1C)=O)C1CC1 53408,c1(C(CC)C)ccccc1OCC(=O)NCc1ccn(C(C)CC)n1 53409,C(=O)(C(O)CC(F)(F)F)N(CCN1CCC1)CCO.O=C(CCOCCOCCO)N 53410,Cc1cc(C2CC2)c(CC(=O)NNC(=O)c2cc(C)c(C(=O)O)c(C)c2)cc1Cl 53411,C1CCC2C(N3CCC(OCC4CCCO4)C3)C2CC1 53412,CCC(CC)N(CCOC)C(=O)NC1CC1C1CCCO1 53413,C1(C(N2CC(OCCOC)C2)=O)CCC(CNC(=O)CCCF)O1 53414,C1(CN(C(CC(CC)C2CCC2)=O)C)CCCN(C)C1c1ccnn1C 53415,N1(C(C2CNC(=O)N2)=O)CC(NC(c2ccoc2Br)=O)C2(CCC2)C1 53416,c1(C(=O)NCC2C(NC(=O)C=C3CCOCC3)C2)c(Br)ccc2c1OCO2 53417,C1(NC(C(CC2CC2)OC)=O)(COC)CCN(C(C2CCN(C(C)=O)CC2)=O)C1 53418,N1(C(C2C3CN(C(C4C(OC)CCCC4)=O)CC32)=O)CC2CC2C2CC12 53419,c1(C(=O)NCCCN(C)C(c2cnc3ccoc3c2)=O)cncc(P(C)(C)=O)c1 53420,C(C1=NOC2CCCC12)NC(CCOCCCNC(CNS(N)(=O)=O)=O)=O 53421,C1(O)(CC(N2C(CNC(=O)C(O)c3cnc[nH]3)CC2)=O)CCCOC1 53422,c1(N2CCN(C)CC2)cncc(C#N)n1.N12CCCC1C2=O.C1CCN1C(N)=O 53423,c1(CNC(N2CC(C)(C#N)C2)=O)ccc(N=[N+]=[N-])cc1 53424,C1(N(C(c2cscc2Br)C(=O)NC(C(=O)OC)C)C)CCC2COC1O2 53425,c1(C(N(CC(CC)NC(C2(CO)CCC2)=O)CC)=O)ncn2ccc(C)cc12 53426,CCC(C)CCC(O)CC(=O)N1CCCC1C1CCN(C(=O)CCCNC(C)=O)C1 53427,C1(CNC(C2C(C(N)=O)C2)=O)C2CC1N(C(C1CCCC1F)=O)C2 53428,c1(C(=O)NC2C(CNC(Cc3n(C)nc(CC)c3Cl)=O)C2)nc2c(s1)COCC2 53429,C1(C(C(=O)CC2(C(=O)NNC3CC3)CC2)=O)C2CN(C(=O)Cn3cncn3)CC12 53430,c1(COC(C2(C(=O)OCC)CC23CC3)=O)cc2sc(C(=O)OCC)cc2o1 53431,CCC(C)(C)C(C)CC(=O)N1CCN(C(c2nocc2C(C)C)=O)CC1CO 53432,c1(C(N2CC(NC(c3c(C)onc3CO)=O)C2)=O)ccc(S(=O)(=O)C(F)F)cc1 53433,c1(CC)cc(Br)ccc1NC(c1ccc(NC(c2ccno2)=O)cn1)=O 53434,C(=O)(CC(N)C(C)(C)O)NCC(C(=O)OC)(C)O 53435,N#Cc1ccc(C(=O)Nc2cccc(NC(=O)CC3CC4CC4C3)c2)cn1 53436,c1(C2CN(NC(C3C(C)(C)C3)=O)C2)ocnc1-c1cn(CCC=CCO)nn1 53437,CC1(C#CC(=O)N2CCCc3[nH]ccc3C2)CN(C(=O)OC(C)(C)C)C1 53438,c1(C(C(=O)NC2CCCCC2)N(CC(=O)OC)CC(C)C)cc(F)c(F)c(Cl)c1F 53439,N1(C(C(C)N(C(C)=O)C)=O)CCCN(C(c2cnc(C(C)C)nc2)=O)CC1C 53440,n1(CC)ccnc1C=CC(N1CCOC(CCNC(C2CCS2(=O)=O)=O)C1)=O 53441,C(=O)(C(F)C1=CCCCC1)NCC(C1CCCC1)NC(c1c(CC)n[nH]c1)=O 53442,c1(CNC(CSC)=O)cc(C(=O)NC(C)CC(N)=O)no1 53443,N1(C(C(C)SCC)=O)CCCC(C)(CNC(=O)CCc2cc(C)nc(C)c2)C1 53444,C1(NC(CCN(C(CC2(NC(C)=O)CC2)=O)CCO)=O)CCCC2(C1)N=N2 53445,C1(NC(C(C=C)C)=O)CCCCC1NC(=O)CCc1cc(C)no1 53446,c1(CNC(=O)Cc2ccon2)nc2c(s1)CN(C(=O)C(O)(C1CC1)C1CC1)CC2 53447,CC(C)CCC(F)C(=O)NC(Cc1cnc[nH]1)C(=O)NCCC1CCC(=O)N1 53448,c1(C(=O)NC(CNC(C2(C)CC2Br)=O)CO)cncc2sccc12 53449,O=C(N=c1cc[nH]cc1F)C12CCN(C(c3ccc(Cl)c([N+](=O)[O-])c3)=O)CC1C2 53450,N1(C(C(n2cc(-c3ccc(OC)cn3)nn2)C)=O)CCC(C)C(C)C1 53451,c1(NC(C2C(NCc3nc(C)sc3)C2)=O)c[nH]c2ccc(Cl)cc12 53452,c1(CC(=O)NC2CCC(NC(c3cn[nH]c3)=O)C2)csc(Br)c1 53453,C1(CNC(C(c2cncnc2)C)=O)CC2CCC1N2C(c1ncccc1Cl)=O 53454,C1C(C)(C)CC(=O)S1.Cc1oc(C(C)(C)C)cc1CN1CCCCC1 53455,CCCC(C)(C)CC(=O)NC1CCC(NC(=O)C(C)(C#N)CC)C1 53456,c1(C(N2CCN(C)CC2CNC(c2ccnnc2O)=O)=O)cc2c(o1)CCCC2 53457,C1(NC(c2cc(N)sc2)=O)CC2(NC(c3cc(-c4ccco4)no3)=O)COC1C2 53458,CON=C(C(=O)N(C(CNC(=O)C(C)(C)C1CCCO1)C1CC1)C)c1ccco1 53459,N1(C(C2CCCCN(C(CC3CC(OCC)C3)=O)C2)=O)CCC2(CC1)CC(O)C2 53460,c1(C(=O)NC2C(C)N(Cc3cnon3)CCC2)ccc2c(c1)ncn2C 53461,N1(C(C(C2CCN(C(CS(CC)=O)=O)CC2)C)=O)CCc2nn[nH]c2C1 53462,c1(C(N)=O)cccc(C(N2CC(F)CC2CNC(c2cnn(CCO)c2)=O)=O)n1 53463,N1(C(c2c(CC)nc(C)o2)=O)CC(NC(=O)C(C(C)C)C2CCC2)CC(F)C1 53464,c1(C(=O)NC(C#C)C(C)OC)n[nH]c2c1CN(C(=O)CC(CC)CC)C2 53465,c1(C(=O)NC(CN(C(CCCOCCC)=O)CC)CC)cc(Cl)ccn1 53466,c1(C(C(=O)NCCCN(C(C23CCC(CC2)O3)=O)CC)=O)cc(F)cc(Cl)c1 53467,N1(C(c2c(C)n(CCO)cc2)=O)CCC(NC(c2cc(C3CC3)no2)=O)C12CC2 53468,C1(NC(C(CSC)O)=O)CCCC(C(=O)N(C2C3CCCC23)C)CC1 53469,N1(C(C(C)CO)=O)CCC(CCC(=O)NC2CCOC2)CC1 53470,c1(OC)ccc(CC(=O)NC(C)(C)CNC(c2cc(CN(C)C)on2)=O)c(C)c1 53471,c1(C(=O)NCC(CC)(C)NC(C2CC2F)=O)ccc(F)cc1OC 53472,C1(C(=O)NCCC(CCC)O)CCCCN(C(c2cnn(C)c2OC)=O)C1 53473,C=CC(C)C(=O)N(CCC(=O)N(C1CCC1)CCO)C 53474,C1(C(=O)NCc2cn(C3CCN(C(CC)=O)CC3)nn2)CCS(=O)(=O)C1(C)C 53475,N1(C(=O)Cc2ccoc2)CCC2(CCN(C(c3cnc(S)n3C3CC3)=O)C2)C1 53476,Cn1ncc(NC(C23CC(CN2C(C2CCCC(F)C2)=O)C3)=O)c1C(N)=O 53477,Fc1cncc(OC2(CN3CCCC(c4nn[nH]n4)C3)CC2)c1 53478,C(N=c1[nH]c(=NC2CC=CCC2)[nH]c2cc[nH]c12)c1cc(C(F)F)no1 53479,C1(N)CN(C(=O)C=CC(c2cnn(C)c2)=O)CC12CCC2.CC1CCN1CC(=O)N 53480,C1(CNC(C2(OC)CCC2)=O)CC2(CCC2)CN1C(=O)CCC1CC(F)(F)C1 53481,C1(NC(c2n(C(CC)C)ncc2)=O)(CO)CCCN(Cc2ccc(Br)s2)C1 53482,C(=O)(C(C)P(C)(C)=O)NCC(C)NC(c1occc1C(n1cc(Br)cn1)C)=O 53483,C1(C)(CC(=O)NCc2snc(C)n2)CCN(C(c2sccc2F)=O)C1 53484,N1(C(CCC2C(C)C2)=O)CCOCC1CCNC(c1cc(C2CCCC2)no1)=O 53485,C=CCC(C)(C)CC(=O)NC1CN(C(=O)Cc2cccc(F)c2Cl)CCC1CO 53486,c1(-c2ccc(CNC(CC#N)=O)s2)cc(OC(F)(F)F)cc(F)c1 53487,n1(CCC(=O)NC(CNC(CCNC(C)=O)=O)C(C)(C)C)ccc2ccccc12 53488,CC(C)CC(O)C(=O)NC1CCCC(C(=O)NCC(F)(F)CO)C1 53489,c1(OC)ncnc(N2CCOC(C)(CNC(C3(F)C(C)(C)C3(C)C)=O)C2)c1OC 53490,N1(C(c2nccc(OC)c2)=O)CC2CCN(C(=O)CS(N)(=O)=O)C(C2)C1 53491,C(=O)(C(C)(C)S(C)(=O)=O)NCC1C(C)CCN1C(=O)Cn1ccc(C(F)F)n1 53492,N1(C(=O)NC(C(C)C)C)c2ccc(Cl)cc2OCC1C 53493,N1(C(C2(CCC=C)CN(C(c3cccc(C)c3O)=O)C2)=O)CC2CCCC2C1 53494,C12(C(=O)NCC3(NC(c4ncccn4)=O)CCCC3)COCC1CS(=O)(=O)C2 53495,C=CC(CCC)CC(=O)N(C)CC1CN(C(c2ccccc2)=O)CCO1 53496,CC1(Cc2cc(COC3CC3)cs2)CCN(C(=O)CCC2CCOCC2)C1 53497,C=CCC(C)(CC)C(=O)N1CCC(NC(c2ccnc(C(F)(F)F)n2)=O)CC1 53498,C1(C#N)(C(N2CC(NC(c3ccc(OC)s3)=O)C(C)C2)=O)CCSCC1 53499,c1(C(N2CCC(CNC(=O)COCC3CCCO3)C2)=O)cccc2[nH]cc(Cl)c12 53500,C=CCC(C)(C)CC(=O)NC(CCF)C(=O)NC(CN(C)C)CC(C)C 53501,C1(C(=O)NCC2(C)CC(C)C2)CC1C1CN(C(C2CCCC(C#N)C2)=O)C1 53502,c1(C(=O)NC2(C)CN(C(C(CCC)CC)=O)C2)cc2c(C)cccc2[nH]1 53503,N1(C(C(C)(C)C)=O)CC(NC(=O)CCc2nc3ccccc3s2)C(C2CC2)C1 53504,N1(C(C(C)N=[N+]=[N-])=O)CC2COCC2(C(N2CCSC(C)C2)=O)C1 53505,C(=O)(C1OCCc2ccccc21)NC(CCCNC(c1c(COC)nn[nH]1)=O)C 53506,CC1(C)CC(COC(c2ccc(F)c(CO)c2)=O)OC1=O 53507,C#CC1(C(=O)Nc2ccc(COC)cc2)CCN(C(=O)CCc2nncn2C)CC1 53508,N1(C(CN(C2CC2)CC)=O)CC=CC(NC(c2cccc(C(C)(C)C)n2)=O)C1 53509,CCCCCCC(CNC(c1nc(C)c(C)nc1C)c1nnnn1C)CC 53510,CN1CCN(C(=O)CCc2nccs2)C(C(=O)NC2C3CCC(F)(F)C23)C1 53511,c1(N2CCC(NC(c3c(C)nco3)=O)C2)cc(-c2ccc(Cl)cc2)ncn1 53512,c1(C(=O)NC2CN(C(=O)Cc3ccc(O)c(Cl)c3)C2)n[nH]c2c1CC1CC21 53513,C1(N)CN(C(=O)OCC(=O)NCC2CC(=C)C2)CC2CCCC12.C(C)(C)(C)O 53514,c1(-c2ccc(C(=O)NCCSCC)c(C)c2F)cc2cc[nH]c2cc1F.CCCCN 53515,N1(C(C(C=C)O)=O)CC2(CC(NC(c3c(C)cc(C)nc3S)=O)CO2)C1 53516,c1(CNC(c2nnc(C)n2C)c2n(CCOC)nnn2)cccc(Br)c1 53517,C(=O)(C(CCC(C)C)NC(C1CC(C)(O)C1)=O)NC1C(COC)COC1 53518,C1(NC(C2OCCN(C)C2)=O)CCCC12CN(C(=O)C=Cc1ccccc1F)C2 53519,Cc1cncc(CC(=O)NC2C=CCN(C(c3sccc3CC#N)=O)C2)c1 53520,C(C(C(F)(F)F)N1CCOCC1)NC(=O)CCCn1cc(Cn2cncn2)nn1 53521,N1(C(C(C2CC2)SC)=O)CCC(C(N2CCC(F)(C#N)C2)=O)C(C)(C)C1 53522,c1(C(=O)NCCCCn2cc(CNC(N)=O)nn2)cc(Br)sc1Cl 53523,Cc1cccc(C)c1NCC(N1CCCN(C(=O)CCC2CCC(C)O2)CC1)=O 53524,NC1CN(C(C2(Cc3ccc(F)cc3)CCCN2)=O)CCc2ccccc21 53525,C1(C(=O)NC2(CO)CCN(C(C=CC=CC)=O)C2)CCn2nccc2C1 53526,C1(NC(C(=O)NC)=O)(CNC(C2CCC(C)S2)=O)CCC(F)(F)CC1 53527,c1(C(N2C(C(=O)NCc3cnc(C)nc3)CC3CC32)=O)ccc(Cl)c(Br)c1 53528,c1(C(=O)NCCN(C)C(C2CCOC2C2CC2)=O)ccccc1OC(F)F 53529,CC(C)C#CC(=O)N1CCC(O)(C(C)NC(=O)C(C)(C)c2ccn(C)n2)C1 53530,C1(CCC(=O)NC(C(C)NC(CCCCCC)=O)CO)CCc2cnn(C)c2C1 53531,Cc1[nH]c2ccccc2c1C(N1CC(C)CN(C(=O)CCOC2CC2)C(C)C1)=O 53532,c1(C(=O)NCCCN(C(C2(n3nccn3)CC2)=O)CC)ccc[nH]1 53533,CCN=C(NCC1(O)CCCCC1(C)C)N1CCN(S(C)(=O)=O)CC1 53534,C(C(F)(F)C(=O)NC1CCC(NC(=O)C(c2cccc(Cl)c2)C)C1)OC 53535,CN=c1[nH]nc(CC(=O)NCC2(O)CCN(C(=O)Cn3ccccc3=O)C2)s1 53536,C1(C(=O)NCC(N(C(C)=O)C)C2CC2)CC(C)CCN1C(=O)C(C)SCC1CC1 53537,N1(C(c2c(C)n(C3CC3)cc2)=O)CCN(C(=O)C(C)OCCN(C)C)CCC1C 53538,c1(CN2C(CNC(=O)C=CCN3CCCC3)CSCC2)c(Cl)ccc(F)c1F 53539,C(=O)(C(C)(C)S(=O)(=O)C1CC1)N(CCN(C(c1cccc(COC)c1)=O)C)C 53540,N1(C(C2C(C#N)C2)=O)CC2CC2(CNC(c2cn(CCO)nn2)=O)C1 53541,N1(C(Cc2c(C)ocn2)=O)CCC2CCC(NC(c3c(Br)nnn3C)=O)C12 53542,C1=CC(=O)Nc2c(N)ccc1c2.C1(CC=C)C(OC(C)(C)C)CC1OC 53543,n1(CC)nc(C(=O)NC(CO)C(C)NC(C2CCNC(=O)C2)=O)cc1C 53544,c1(CC)nn(C)c(C(=O)NC(C)C(CO)NC(C2CC(C(C)C)C2)=O)c1Cl 53545,N1(C(=O)C(O)C(F)F)CCC2(CCCN2C(c2ccc(N3CCC3)nc2)=O)C1 53546,c1(C(=O)NC(CC)(C)CNC(=O)C=C(C)Cl)cc2c(cn1)NC(=O)CO2 53547,N1(C(COCC=C)=O)CC(C(=O)NCCc2cnn[nH]2)(SC)C1 53548,c1(C(N(C2CC2)Cc2ccc(OC)c(F)c2)=O)n[nH]c2c1CC1CC21 53549,C1(O)(C(=O)NC2CN(C(C(COCC)N=[N+]=[N-])=O)CC2C)CCCC(C)CC1 53550,C1(O)(CNC(CC(C)c2ccncc2)=O)CCCN(C(C2(F)CCCCC2)=O)C1 53551,N1(C(CS(CC)(=O)=O)=O)C(C)CC2CN(C(=O)Cn3nccc3C)CC12 53552,CC#CCC(C(=O)NCC1CC1c1ccco1)NC(c1c[nH]c(C)c1)=O 53553,C1(NC(C(N2CCC(N(C(c3cscc3Cl)=O)CC)C2)=O)=O)CCC(F)CC1 53554,c1(C(=O)NC2CCN(C(=O)C3=CCCC3)C(C3CC3)C2)ccn2cccc2c1 53555,N1(C(C(CN(C)C)N(C)C)=O)CC2CCC(C(=O)Nc3cncnc3O)(C2)C1 53556,c1(SC)c(C(=O)NC23CC(NC(=O)COCCN(C)C)(C2)C3)cnn1C 53557,N1(C(C(CC(C)C)F)=O)CCc2sccc2C1CNC(=O)CC(C)(C)CC(F)F 53558,N1(C(c2c(=N)[nH]cnc2)=O)CC2CCOCC2(NC(=O)C=Cc2cccnc2)C1 53559,CC(C(=O)NOCC(N1CC(CO)(CO)C1)=O)C1CCCC1 53560,C(=O)(C(CCCCC(=O)OC)N1CCCC(CCO)C1)NCCC 53561,Cc1ncc2c(n1)CCC(C(=O)NC1CN(C(=O)C#CC3(C)COC3)CC1C)C2 53562,N1(C(C2CCOC2)=O)CC2OCCN(C(c3cc(C4CCOCC4)[nH]n3)=O)C2C1 53563,C(=O)(CCOCCN(C)C)OC(C(N1CCC1)=O)C.C=CCOC(C)=O 53564,c1(CC)nocc1C(=O)NCCN(C(=O)C(C)COC)C 53565,C(=O)(CC(C)(O)CCC)NC1C(C)CCN(C(C(C=C)c2ccccc2)=O)C1 53566,c1(C(=O)Nc2ccc(OC3CCCC3)cc2)cccnc1N1CCOCC1 53567,N1(C(=O)NCc2cnc3n2CCCCC3)CCCCC(C2CCOCC2)C1 53568,N1(C(C(C=C)O)=O)CCC(CO)C(NC(c2ccc(Br)c(C)c2)=O)C1 53569,c1(C(=O)NC2CC(F)(CNC(C(CC=C)CC)=O)C2)cc2nn[nH]c2cc1F 53570,Cc1ccc2c(c1)CCN(CCc1cc3cc(Cl)ccc3[nH]1)C2 53571,c1(C(=O)NC(C(CO)NC(c2cnc(C)[nH]2)=O)C)nc(O)c(C)s1 53572,N1(CCNc2scc(-c3ccc(Br)cc3)n2)CCC2CCCC(C1)N2 53573,N1(C(c2ccc(SC)s2)=O)CC(NC(=O)CCSC(F)(F)F)C(C)C1 53574,c1(CC)[nH]nc(Cl)c1C(=O)NC1CC2C(NC(c3ncsc3C)=O)C2C1 53575,N1(C(C)=O)CCCCC1CC(=O)NC1(C)CC(NC(C2CCNC2=O)=O)C1 53576,Cc1cc(CC(=O)NCC2CN(C(=O)CCCF)CCC2C)cc(C)c1Br 53577,C(=O)(CCN=C(NCc1cncc(C(F)(F)F)c1)NC(C)C)NCCC 53578,c1(C(=O)NC(CNC(C=C(CCC)C)=O)CO)ccc(C(C)C)c(Cl)c1 53579,c1(NCc2csc(C3CCC(OC)C3)n2)c(OC)ccc(S(N)(=O)=O)c1OC 53580,c1(N(CC(C)C(=O)N2CCCC2)C)ncnc2ccc(Cl)cc12.C(C)(C)(C)N1CC1=O 53581,C#Cc1cnn(CC(=O)NC(CC2CCC2)C(=O)NC2CC(N3CCCC3)C2)c1 53582,c1(N(CC(=O)OC(C)(C)C)CCOC2CCCC2)ncc(C(C)(C)C)s1 53583,Cc1ccc(-c2ccc(C(=O)NCCCN(C(=O)C(Cl)=CCl)C3CC3)s2)s1 53584,CCCC(C#N)C(=O)NCC(CNC(c1cccc(Br)c1)=O)OC 53585,c1(OC)cc(NC(C2C3CC2N(Cc2cc(Cl)ccc2I)C3)=O)ccc1C 53586,c1(NC(c2c(CNC(C3CCN(C)C(=O)C3)=O)occ2)=O)cncc2ccccc12 53587,c1(C(=O)NCC2CCCN2C(=O)CSc2nc[nH]n2)cccc(-c2nccs2)c1 53588,c1(C(N(CC)CC2CCCN2C(=O)CC(C)(C)O)=O)cc(Cl)cc(Cl)c1 53589,N1(C(CCCN(C(C)=O)C)=O)CCC(C)(C)C1C(=O)N(C1CC(O)C1)C 53590,C1(N(C(=O)CC2CC2)CC#C)CCN(C(=O)C(C2CCOCC2)F)CC1 53591,C(CC(CC)C(=O)NC1CC(C)(NC(=O)C(CC)C(=O)OCC)C1)=CC 53592,c1(NC(CN(C(=O)CN2C(C)CCC2C)CCC)=O)ccc(F)c(O)c1 53593,C(=O)(CCCCCCC(=O)N1CCN(Cc2c(O)cccc2Br)C2CC12)OC 53594,Cc1cc(C(=O)NCCN(C(=O)C(O)CC(N)=O)C2CC2)cc(S(N)(=O)=O)c1C 53595,C(=O)(C(C(C)C)NC(=O)C(C1CCCCC1)C)NCC#CCC 53596,N1(CC(=O)N(CCNC(C(OC)OC)=O)C2CC2)CC(=O)N1 53597,Cc1nc(=O)c2c(C)c(C(=O)OCCC(C)NC(=O)OC(C)(C)C)sc2[nH]1 53598,C1(CCOC)(C(=O)Nc2cncnc2C)CCN(C(=O)C(C(C)C)SC)C1 53599,C(=O)(CS(=O)c1ccc(Cl)cc1)NCC(C1CC1)NC(=O)Cc1cnsc1 53600,Cc1oc(C#N)cc1C(N1CCCC(C(=O)NC2(CC(N)=O)CCC2)C1)=O 53601,c1(-n2c(C)cnn2)ccc(C(=O)NCC2CCCC2NC(=O)CC(C)C)cc1 53602,C(=O)(N=c1[nH]onc1C1(CO)CCC(=O)N1)NC(CCC(=O)OCCCC)=O 53603,C(N=c1[nH]c(=NCCCNS(=O)(=O)NC)[nH]c2cc[nH]c12)c1cn(C)nc1C(F)F 53604,c1(C(N(C2CCN(C(=O)C(C)OCC(C)C)C2)CC)=O)cncc(C(C)C)c1 53605,CC1(CNC(C2(F)CCCC2)=O)CCCN1C(C1CCCCO1)=O 53606,CS(=O)(=O)c1ccc(CSCC(=O)NCc2nc3ccccc3s2)s1 53607,N1(C(CC=CCC)=O)CCN(c2ncncc2C)CC1C 53608,C1(C(=O)N(C)Cc2nnc(O)o2)(NC(C2C(C(C)C)C2)=O)CC1(C)C 53609,C(=O)(C1CCCc2scnc21)NC1CCC(CNC(c2coc(Br)c2)=O)C1 53610,C(=O)(CC(C)C(C)C)N(CC(=O)NCc1c(C)noc1C)CC(C)C 53611,C(=O)(CC(F)(F)C(F)F)N(CC(CC)NC(c1cc(Br)n[nH]1)=O)CC 53612,C1(N(C(CC2(C)CCOC2)C(=O)NCCC2CC2)C(C)C)CCC(C2CCCO2)C1 53613,N1(C(Cn2c(C)c(Br)cn2)=O)CCCC2(NC(c3nccnc3N)=O)CC2C1 53614,c1(C(=O)NC2CN(C(C(C)(C)c3ccc(Cl)s3)=O)CC2F)ncc(F)cc1F 53615,C1(NC(Cc2c(C)con2)=O)CCCCC1NC(=O)C(C)(C)c1ccn(C)n1 53616,N1(C(CC2(CSC)CC2)=O)CCCCC1CN(C(=O)C(C)=C1CC1)C 53617,N1(C(CCCC)=O)CCC2(CC1)CN(C(c1n[nH]c3c1CC1CC31)=O)CC(C)O2 53618,c1(C(=O)NC2CCC(C)N(C(=O)CCc3cncs3)C2)ccc2c(ccn2C)c1 53619,c1(C(N(C2CCCC(NC(c3ccc(C)s3)=O)C2)C)=O)cc(C)c(C#N)cn1 53620,c1(C(C(=O)NCC(C)CC2CC2)NC(=O)CN(C)C(N)=O)cccnc1 53621,C(=O)C#CC1CCCCC1.N1(N2CC(CC=C)(C=O)C2)CCC(C)C1CC 53622,N1(C(C(C)Cc2ccco2)=O)CC(C(N2CCS(=O)CC2)=O)CC(F)(F)C1 53623,N1(C(c2n[nH]c(CC)c2Cl)=O)CC2(CCCC(CNC(c3oncc3C)=O)O2)C1 53624,C1(CNC(C=Cc2cc(OC)ns2)=O)CC2CC(C1)N(C(=O)CC(C)C)C2 53625,C1(CCC)CN(C(=O)C(C)(C)COC(C)C)CCN1C(C1CCCS1)=O 53626,N1(C(CC(C=C)C)=O)CC2(C1)CN(C(c1nnn(CC)c1CC)=O)CC2CO 53627,CC(C)CC(C)(CNC(=O)CN(C)C(=O)C1CC1)NC(c1cnc(O)c(Cl)c1)=O 53628,c1(C(=O)NC(C(=O)OC)Cc2cn(C)cn2)cnn2c(Br)cccc12 53629,C(=O)(C(C)C(O)CCCC)NCCCCCC(=O)N1CC(CC(C#C)C)C1 53630,N1(C(CCC(CC)NC(c2cnn3c2OCC3)=O)=O)CCCC2(CCCO2)C1 53631,Cc1cc(C(=O)N(C)CC=CC(N2CCCCC2CCO)=O)cc(O)c1 53632,C1(NC(C2C(=O)NCCCC2)=O)CCN(C(C2(Cl)CCCCC2)=O)CCC1CO 53633,c1(Cc2nc(C(C)SCC)nn2-c2ccnc(Cl)c2)cc(Cl)ccc1Cl 53634,Cn1cncc(C(=O)NC2(O)CC2NC(=O)NC2COC3(CCC3)C2)c1=O 53635,N1(C(CCOCC)=O)CC2CN(C(=O)CC(CC)C3CCC3)CCC12 53636,Cc1cc(NC(C2CC3CC3N2C(=O)C(C)Oc2cccnc2)=O)c(C)cc1Br 53637,CCCS(=O)(=O)C(C)C(=O)NC1C2CC1N(C(c1cc3cccn3cn1)=O)C2 53638,c1(OC)ccc2c(c1C(=O)NCCN(C(=O)C1=CCCSC1)C1CC1)CCC2 53639,c1(C(=O)NCC2C(C)CN(C(c3cnc(N(C)C)o3)=O)C2)cc(F)cc(Cl)c1N 53640,N1(c2nccc(N3CC=C(C)C3)n2)CCCC2(CC=CCO2)C1 53641,c1(C(=O)NCCN(C(=O)CCn2cccn2)C)ccc2cc(F)c(F)cc2n1 53642,C1(CNC(c2cnc(CCC)s2)=O)CCCC2(CN(C(=O)CC(C)C3CC3)C2)O1 53643,C1(CCO)CC(C)(C)CC(C)(C)C1.Cc1cccc(-n2nc(-c3cc[nH]n3)nc2)c1 53644,c1(C(N(CCC(C(C)(C)C)NC(CCC=C(C)C)=O)C)=O)ccc2nccn2c1 53645,c1(C(=O)NC2C(CC)N(C(=O)Cc3nc[nH]n3)CC2)cnn2c(C)cccc12 53646,c1(C(N)=O)oc(CSCc2nncs2)nc1-c1ccccc1 53647,c1(C(=O)NC2CCC(CNC(c3cnc(Cl)nc3)=O)CC2)ccc(I)cc1Cl 53648,C(=O)(CCCC(F)F)NC(c1ccc(CC)cc1)CNC(=O)Cc1nnc(O)s1 53649,C(CCCCC(=O)N1CCCc2n[nH]cc21)NC(=O)C1=C(Cl)CCC1 53650,c1(C(C)C)cccc(NC(C2CC2CNC(=O)Nc2cccc(CO)c2)=O)c1 53651,c1(C(=O)NC2(CC=C)CN(C(C3SCCC3C)=O)C2)ccn2ncc(C)c2n1 53652,C1(CC(=O)N(CCNC(C)=O)C2CC2)CN(C(=O)CCC2CC2C)CCO1 53653,C1(C(=O)NCC(C)(C2CC2)NC(=O)CSC(F)(F)F)CC1[N+](=O)[O-] 53654,C1(C(=O)NCC(c2ccccn2)C)C2Cc3ccc(Cl)cc3C12 53655,C(=O)(C(F)CC(C)(C)C)NC(CNC(c1ccc(C(=O)OC)cn1)=O)C 53656,N1(C(C2C(CC)C2)=O)CCCN(C(c2c(OC)cccc2C)=O)C(C)C1 53657,O(C1(OCC)c2cccnc2CCC1NC(c1csc(Cl)c1)=O)CC 53658,N1(C(C2(C)CC2(Cl)Cl)=O)CC2C3CCC(C2C1)N(C(=O)CCN1CCOCC1)C3 53659,N1(C(C=CC=CCC)=O)CC(N=[N+]=[N-])CC1C(=O)NC1CCC(CCO)CC1 53660,Cn1[nH]nnc1=NC1CC2CCC1N(C(C1Cc3nccnc3C1)=O)C2 53661,C1(CNC(CC=CC(C)(C)C)=O)CC2CCC1N(C(=O)CSc1ccccc1)C2 53662,C1(OC)CC(NC(=O)Cn2ccc([N+](=O)[O-])n2)C12CCN(C(=O)C(F)=C(C)C)CC2 53663,c1(CN(CC(=O)NCCCN(C)C)C)ccc([N+](=O)[O-])o1 53664,C1(NC(C=C(C)C)=O)CCOC(CNC(c2ccc(F)cc2)=O)C1 53665,C(CCCC(C)(C)C(=O)NNC(=O)C(C)(C)O)NC(CCC(=O)NS(C)(=O)=O)=O 53666,Cc1cc(C#N)ccc1C(N1CCC(C(=O)NCCS(C)(=N)=O)C(O)C1)=O 53667,N1(C(C2C(C)N(C)CC2)=O)CCCC(C)(NC(=O)CCc2ccc(Cl)nc2)C1 53668,Nc1c(C(N2CCC(NC(C3CC3(F)Cl)=O)CC2)=O)ccc(F)c1F 53669,C(C(O)C(=O)NC(C1CCCN1C(c1cc(C(C)C)on1)=O)(C)C)SC 53670,N1(C(C2(OC)CC2)=O)CCC(C2CC2NC(=O)CN(CC(C)(C)C)C)CC1 53671,N1(C(Cc2c(SC)cccc2)=O)CC(C)CN(C(=O)C=C(C)Cl)C(C)C1 53672,C1(CCNC(c2ncn(C(C)C)c2)=O)CN(C(=O)C(c2cncnc2)C)CC1C 53673,c1(C(c2nnnn2C)NCC(CCC)C)cc(S(N)(=O)=O)ccc1F 53674,c1(C(N2CC(=C(F)CC(C)(C)C)C2)=O)cc(C(=O)NC2(C3CC3)CCC2)ccn1 53675,C1(CC(=O)NC2(c3cccs3)C(C)C2)CCCS1(=O)=O 53676,N1(C(c2n(CCC)ccc2)=O)CC(C(=O)NC2(CCOC)CC2)CC(C)C1 53677,C1(N(C)NC(C(=O)NCCC(OC)OC)=O)CCCN(CC(C)C)C1 53678,C(=O)(C1=CCCOCC1)N1CC(O)(CN(C(C2(CCCC)CC2)=O)CC)C1 53679,C1(C)(COC)CC(NC(=O)Cc2sc(O)nc2O)CN1C(=O)Cc1cnn(C)c1 53680,C(C(CCCC)NC(=O)CNS(=O)(=O)N(C)C)NC(CC(=C)Br)=O 53681,S(=O)(=O)(CC(=O)NC1(C(=O)NCC2CCCO2)CCSC1)NC 53682,c1(NC(C(C)NC(C2CCC2)=O)=O)cnn2c1CN(C(=O)CNC(N)=O)CC2 53683,N1(C(C2C(OCC)C2C)=O)CC2(CCN(C(C3CC4(C)CC3CO4)=O)C2)C1 53684,CCCCC(C(=O)NCCC1(C(C)(C)O)CC1)N(C)C.C12(CC1)C(=O)NC2 53685,Cc1cc(C(=O)NC2CC(NC(=O)C(C)Sc3ccc(Cl)cc3)C2)c(C)s1 53686,C(=O)(C(F)C(=O)NC(C)(C)CC(=O)N1CCC(CCOC)C1)OCC 53687,c1(C(=O)NC(CC)CNC(c2c[nH]c(=N)o2)=O)sc2cccc(F)c2c1Cl 53688,c1(NC(N2CCN(c3cncs3)CC2)=O)nc2ccccc2[nH]1 53689,N1(C(CC2(C)CC2)=O)CCC2(CNC(c3ccccc3CO)=O)CCCCC12 53690,Cc1ccc2ccnc(NCc3nc(C(=O)O)c(C)s3)c2c1 53691,N1(C(C=CCN)=O)CCCC(F)(CO)C1.CC(C)(O)CC=O 53692,c1(CC(N2CCCC(NC(=O)Cn3cccn3)CC2)=O)ccc2c[nH]nc2c1 53693,N1(C(C(CC)NC(C2C(C)C2C)=O)=O)CCC(CC)C1CC 53694,C(=O)(C(O)C1=CCCCC1)N(C1(C(=O)NCCC(CCCCC)O)CC1)C 53695,C1(C(N2CC(C)(NC(CCC(=O)NC)=O)C2)=O)CCC(=O)C(C)C1(C)C 53696,c1(C(=O)NCC(C)N(C(C(C)n2ccnc2)=O)C)cc(S(N)(=O)=O)sc1Cl 53697,C12(C(N(C3CCC3)C)=O)CCCC(CN1C(=O)C(O)CN1CCCC1)C2 53698,C1(CN(C(CC=CCC)=O)C)COCCN1C(=O)CC1CCCC(C)O1 53699,N1(C(C(CC)OC2CCCCC2)=O)CCCC2(CCCN2C(C)=O)C1 53700,C1(NC(c2ccc(F)cc2O)=O)C2COCC1CC(NC(C1CCCCO1)=O)C2 53701,c1(C(=O)NCC(CNC(C(C)OCCCCCC)=O)OC)cccc(C)n1 53702,C1(NC(CC2(C=C)CCC2)=O)(CO)CCN(C(C2CN(CC)CCO2)=O)CC1 53703,N1(C(C(CC2CCCC2)OC)=O)C2CCC1CC(CNC(C1(CO)CCC1)=O)C2 53704,C1(CNC(C2(C)CC(=C)C2)=O)CCCN(C(c2ccnn2CCC)=O)C1 53705,N(C(=NCCN(C)C)NCc1ncccc1N(C)C)CC(C)(C)OCC 53706,N1(C(c2cc(C)n(C)n2)=O)CCCN(CCNC(C2CC2CF)=O)CC1 53707,CC1(CCC2(O)CCN(C(=O)Cn3cc(C(O)C4CC4)nn3)CC2)NC(=O)NC1=O 53708,c1(C(C(=O)NC(CNC(c2c[nH]c(=NC)s2)=O)C)C)cccc([N+](=O)[O-])c1 53709,C12(C(N3CC(NC(CCc4ccc(C(C)C)cc4)=O)C3)=O)CC(C)(C1)OC2(C)C 53710,c1(N2CCCC(NC(=O)CCc3cscn3)C2)ncnc2sc([N+](=O)[O-])cc12 53711,C1(NC(c2c(N)ccc(Cl)c2)=O)CCC12CCN(C(C1CC3C=CC1O3)=O)CC2 53712,C(=O)(C(F)CC(CC)CC)NC1(C(=O)NCCC=CCCC)CC(F)C1 53713,N1(C(C(c2ccc(OC)cc2)C)=O)CC2CC(C)N(C(=O)CSC(C)(C)C)C2C1 53714,N1(CC(C)NC(=O)NC(C(=O)OC)C)CCN(S(=O)(=O)Cc2ccccc2)CC1 53715,c1(CCC)cc(C(=O)NCCNC(=O)C(C)NC(=O)OC)no1 53716,C1(C(=O)NC)CCCCN1C(=O)CC=CCNC(=O)CC1(CSC)CC1 53717,c1(C(=O)NC23CC2CN(C(=O)COCC2CCCO2)C3)ccc(OCF)c(F)c1 53718,CC1c2ccccc2CC1N(C(=O)C(=O)NC1CC(c2cccc(Cl)c2)C1)C 53719,Cc1cc(C)c(CC(N2CCC(NC(=O)C(F)(F)C(C)O)CC2)=O)c(C)c1 53720,Cc1nncc(C(=O)NC2(c3cn(C4CCCC(C)C4)nn3)CCC2)c1C 53721,N1(C(CC(C)n2ccnc2)=O)CC(C(=O)N(C2CC3CCC2CC3)C)C2(CC2)C1 53722,c1(C(=O)NC2CN(C(c3c(OC)nsc3)=O)CC(F)C2)cc2nccnc2[nH]1 53723,CCC(CC(=O)NCc1nocc1C(=O)NCCC1CCCC12CC2)C1CCC1 53724,C(=O)(C(C)CC(C)(C)C)NCc1ccccc1CN(C)CC1CCC(C)C(C)C1 53725,N1(C(c2cc3n(c2)CCSC3)=O)CCC2CN(C(=O)C(O)C3CC3)CC2C1 53726,c1(C(N2CC3CSCC3(C)C2)C(=O)NC(C(=O)OC)C)cn2cc(F)ccc2n1 53727,C(C)(C(=O)N1CC(O)(CCNC(=O)C2CC2)C1)(C1CC1)OC 53728,C(CC(C(C)(C)C)NC(=O)Cc1nc([N+](=O)[O-])n[nH]1)N(C)C(C1CCSC1)=O 53729,CC1(C)CC=CCN(C(C2(NC(C3CC3(C)C(F)F)=O)CCCC2)=O)C1 53730,C12(C(=O)OC)CCC(C(=O)N(C3CN(C(=O)Cc4sccc4C)C3)C)(C1)C2 53731,C(N=c1ccnc(N2CCCCC(N3CCOCC3)C2)[nH]1)c1ccc(C#N)cc1 53732,C1(CNC(=O)NOC(C2CCCC2)CO)CCCCO1 53733,c1(-c2cc(C(N(CCCCCNC(C3C(C)CC3)=O)C)=O)n[nH]2)ccccc1Cl 53734,Cc1cc(C(N2CCC(C(C)NC(=O)CC3COCC3(C)C)C2)=O)nc(O)c1 53735,c1(OC)cccc2cc(CNC(c3cnc(C)cc3C)c3nnnn3C)oc12 53736,C1(C2CC2)(CNC(CC2CCC(C)(C)CO2)=O)CCN(C(=O)C(Cl)=CCl)C1 53737,C(C1=NOC2CCCC12)NC(CCC1CCN(C(C2CCC(=C)CC2)=O)C1)=O 53738,C(=O)(CC(C)C(C)C)NC(C(=O)NCCCC(=O)NC)C1CC1 53739,CCC(C(=O)N1CCC(C(=O)N(C)CC2CCOC2)(C(C)C)C1)C(F)(F)F 53740,C1(C(=O)NCCC(C)NC(c2ccn(C)c2)=O)CCC2(CC1)NC(=O)NC2=O 53741,CC1(CNC(C2CC2CNC(=O)CNC(=O)C2CC2)=O)CC2(CC2)C1 53742,C1(NC(c2c(C)nc[nH]2)=O)CC(C2CCN(C(c3csc(S(C)(=O)=O)c3)=O)C2)C1 53743,c1(N(CC(C)CO)C)nccc(N2CCOC(c3n[nH]c(CO)n3)C2)n1 53744,N1(C(c2ncn(C)n2)=O)CCCC2C1CCCN2C(c1csc(CO)n1)=O 53745,n1(CCC)cccc1C(=O)NCC(O)CNC(C1CC1C)=O 53746,C1(C(=O)NCC(CC(C)C)NC(=O)CN2CCCCCC2)CC(=O)CC12CCC2 53747,c1(NC(=O)NCC(c2ccoc2)C)ccc(OCC2CCC2CO)cc1 53748,C12COC3(C1)CN(C3)C2=O.c1(NC(C(N2CCC(C)C2)=O)=O)ccc(C#N)[nH]1 53749,N1(Cc2c(O)ccc(C)c2)CCC2(CC1)CC(C(N1CCOCC1CO)=O)CO2 53750,C1(NC(C(C)n2ccnc2)=O)CCCC12CN(C(=O)C1CC1)C2 53751,N1(C(COC(C)(C)C)=O)CCOCC(NC(=O)NC2CCCC(CC(N)=O)C2)C1 53752,C(CCF)(C(=O)NCCC1CC(C)C1)NC(C1CC(OCC)C1)=O 53753,C1(CC(=O)OC)CN(Cc2ncc(C(C)(C)C)s2)C2(CC2)CO1 53754,c1(C(=O)NCC2(C(=O)OC)CC2)cc2c(-c3cccc(OC)c3C)cccc2s1 53755,N1(C(C2(C#N)CC(=O)C2)=O)CCC(C2(NC(C3CC3C3CCCC3)=O)CC2)CC1 53756,C1(CCNC(COCCC)=O)CCCN(Cc2coc(-c3cccc(F)c3)n2)C1 53757,c1(C(N2C(CC)CC(C)C2)C(=O)NC)cc(Br)c(C(F)(F)F)cc1F 53758,c1(CC)ccc(C(=O)N(CC(C)NC(C2(c3ccno3)CCC2)=O)C)cc1N 53759,CCCC(C)CC(=O)N(CCNC(=O)CC1CCCCC1(F)F)CCOCCO 53760,N1(C(C2C3CC2N(Cc2ccc(C(=O)O)[nH]2)C3)=O)CCC2(CCCO2)C1 53761,N1(c2c(C)cncn2)CC2CC1CN2C(C1(C)CC=CCC1)=O 53762,C(CC(N)CC(C)C)NC(c1ccc(OCC=C)cc1)=O 53763,C1(NC(C2CCCC23CC3)=O)CCCN(C(=O)Cc2cscc2Br)CC1 53764,C(CCC(=O)NC1CCC(CNC(=O)C(F)=CC2CC2)C1)OCC 53765,c1(CC)ccc(C(=O)N(CCNC(c2ccc(C)o2)=O)CC2CC2)c(F)c1 53766,C1(CN(C(=O)Cc2csc(C3CC3)n2)CC)CCCN(C(=O)CN2CC=CC2)C1 53767,CCC1=NOC(C(=O)NCCCCC(C)NC(c2cncnc2C(C)(C)C)=O)C1 53768,CCCN=C(NCCC(C)(C)O)NCC1(OC)CCC1 53769,CC1CCN(C(=O)CC2CSCCO2)CCN1C(=O)CC1C=NN(C)C1=O 53770,C(C(=O)NNC(=O)CCSC1CCCCC1)c1c(C)n[nH]c1C 53771,C1(C(=O)NC(CNC(c2cnc(CC)[nH]2)=O)C(C)C)CCC(F)(F)CO1 53772,N1(C(c2nccc(SC)n2)=O)CCN(C(C2CCC(C)=C(C)C2)=O)CC(C)(F)C1 53773,c1(C(=O)NCCC(CNC(C2C(=C)C2)=O)O)ccc(OC)c(S(=O)(=O)N)c1.C1N=N1 53774,CCC(CC)C(F)C(=O)N1CC(C(=O)NC(C2CCC2)C2CC2)C2(CCC2)C1 53775,c1(C(=O)NCCC2CCN(C(c3ccc(CC)o3)=O)C2)cncc2ncn(C)c12 53776,C1(NC(COCCC=C)=O)CC(NC(C2CC(F)(F)C2)=O)C12CCOCC2 53777,C1(CC=C)(NC(=O)CCC2CC2)CCCN(C(=O)CC(N2C(=O)CCC2=O)C)C1 53778,C12C3C=CC4(CN(C(=O)C14)C2)O3.N1(CC(=O)OC)CC(OC)CS1(=O)=O 53779,c1(C(N2C(CN(C(C3(OC)CS(=O)(=O)C3)=O)C)COCC2)=O)ccc(O)nc1Cl 53780,C(c1cnn(C)c1C)=CC(=O)NCC(CNC(CN(C)CC)=O)C 53781,c1(CC(C)C(=O)O)ccc(-c2cc(NC(=O)CC3CCOCC3)ccn2)cc1 53782,C1(NC(c2cn(CC=C)nc2)=O)CN(C(C2CCCCC2(F)F)=O)CCC1CO 53783,O=C1COC(CNC(C2CN(Cc3ccccc3I)CCO2)=O)CN1 53784,c1(C(N(CCN(C(C(CC#C)C)=O)C)C)=O)cc(-c2ccc(C)o2)ccc1F 53785,c1(C(=O)NC)ccc(CC(=O)NCC(C)NC(c2cnn(C)c2C(C)C)=O)cc1 53786,N1(C(c2ccn(C(CC)CC)n2)=O)CC(CNC(=O)Cc2cc(OC)no2)C2CC12 53787,c1(CNCc2ccc(-c3ccc(OC)cc3)s2)n[nH]c2ccc(C)cc12 53788,C(=O)(CCCCNC(C)=O)NCCN(C(C(C)(C1CCOCC1)OC)=O)C1CC1 53789,C(c1ncco1)=CC(=O)NCC1CCN(C(c2ccoc2C2CC2)=O)C1 53790,CC(C)(C)C1=NOC(C(=O)NCCC2(NC(c3n[nH]c(C4CC4)n3)=O)CCC2)C1 53791,C1(C(N)=O)CN(C(=O)Cc2nc[nH]n2)CCN1C(C1CC1c1ccccc1)=O 53792,Cn1cc(C(N2CCC(CO)C(NC(=O)CC3CC4CC4C3)C2)=O)c2sccc12 53793,C1(NC(c2c(C)cc(C)o2)=O)(CO)CCN(C(C2CC(=O)C2(C)C)=O)CC1 53794,C1(C(=O)NCC2=CCCCC2)C2CCN(C(c3ccsc3Cl)=O)CC12 53795,C1(CC)(NC(c2coc(C(C)(C)C)n2)=O)CCCN(C(C2CSCCS2)=O)C1 53796,c1(C(C)=O)ccc(C(=O)NC(CNC(=O)CCC(F)F)CC(F)(F)F)cc1F 53797,C1(C(=O)NCC(C2CC2)NC(C(CN(CC)CC)F)=O)CCC(C)CC1 53798,N1(C(c2cnn(C(CC)CC)c2C)=O)CCC(C)C(NC(c2csc(=N)[nH]2)=O)C1 53799,NS(=O)(=O)CCC(=O)NCCNC(C1CCCN(C(c2cnns2)=O)C1)=O 53800,c1(C(N2CC(O)(C(C)NC(C3CC(C(F)F)C3)=O)C2)=O)cc2c([nH]1)CCCC2=O 53801,C=C=C(C)CC(=O)NC1C2CCN(C(=O)CCC(=O)NC)C12.C1(C=O)CCC(C)CC1 53802,C#Cc1ccccc1CNC(C1CCN(C(=O)C(C)C=CC)CC1O)=O 53803,c1(C(=O)NC(CN(C)C)C(=O)N2CCC(N3CCCC3)C2)cncn(C)c1=O 53804,N1(C(Cc2c(C)ccnc2)=O)CCCC(C(=O)NC(c2ncn(C)n2)C)CC1 53805,c1(CC)ccncc1CNC(c1cccn1C)c1nnnn1-c1ccccc1 53806,N1(C(C(C)NS(C)(=O)=O)=O)CCN(C(c2nnn(C)c2C(F)F)=O)CC(O)C1 53807,Cc1nccc(C(=O)NCC2(F)CC(CNC(=O)C=Cc3nccs3)C2)n1 53808,N1(C(c2c(OCCCC)nccc2)=O)CCCC(C)(NC(=O)CCC(C)(C)F)C1 53809,C1(CS(N2CCN(c3nccc(OCCC)n3)CC2)(=O)=O)CC2(CCNCC2)C1 53810,N1(C(c2c(C)n(C(C)C)nn2)=O)CC2(CCCCN2C(C2(C)CCOC2C)=O)C1 53811,C(CC(C(N)=O)NC(C1(NC(C2CC2(Cl)Cl)=O)CCOCC1)=O)OC 53812,N1(C(CC2CCC(C)CO2)=O)C2CCC1CN(C(C1CCn3nncc3C1)=O)C2 53813,c1(N2CC(C(C)NC(c3ccc(C(F)(F)F)[nH]3)=O)OCC2)ncccc1C#N 53814,c1(C(=O)NCCCCCN(C)C(C2C=CCC2)=O)cnn2c1OCC(O)C2 53815,CCCCCC(F)C(=O)N(C(C)C(=O)NOCCCO)C 53816,Cc1nsc2ncc(C(N3CC4(C3)CN(C(c3cccn(C)c3=O)=O)C4)=O)cc12 53817,c1(C(=O)NCCCOCCN(C)C(C2C3COCC23)=O)nn(C)cc1S(C)(=O)=O 53818,C12(C(N3C(CNC(c4ccccn4)=O)C4CC4C3)=O)CCC(F)(CC1)CC2 53819,Cc1ccc(F)c(C(=O)NCC2CC(F)(CNC(c3ccn(C)c3C)=O)C2)c1 53820,c1(C(=O)NCC2CCC(NC(C(C)OC3CCCC3)=O)C2)cc(Cl)c(Cl)cc1N 53821,C(=O)(C(C)(C)C(F)(F)F)NC1CCCN(C(C(C2CCCC2)NC(C)=O)=O)CC1 53822,C1(C2CC2)(NC(CC(C)N(C)C)=O)CCN(C(c2coc3c2CCCC3)=O)C1 53823,CN1CCN(C(=O)Cc2cnns2)C(CNC(=O)CC2CCCCC2(C)C)C1 53824,c1(SC)nc2sc3c(C(C)(C)OC(C4C(OCC)C4)=O)c2c(=O)n1CCCC3 53825,C12(CNC(CCCOCC=C)=O)CC1CN(C(=O)C(C)Cc1cnc[nH]1)C2 53826,C(N=c1nc2ncn(C)c2c(NCCC#CCO)[nH]1)c1c(C)cncc1 53827,CC1(C)CCC(CNC(C2CCC(=O)NC2)=O)N(c2nnco2)C1 53828,c1(C(=O)NCCC2CCC(NC(=O)CCCC3CC3)C2)occ2c1CCOC2 53829,CS(=O)(=O)CCCCCCCC(=O)NC1(C)CN(C(=O)C2=CCCCCC2)C1 53830,N1(C(=O)Nc2n(C)ncc2C2CCC2)CC2C3CCC(C(O)C3)C2C1 53831,C(CCC(C)C(=O)N(CCCN(C(=O)Cn1cnc([N+](=O)[O-])n1)C)C)OC 53832,c1(C(=O)NC)ccccc1OCc1cscc1Br 53833,C1(NC(C(COC)C)=O)CN(C(=O)Cc2ncc(C)o2)C(C)(C)C1 53834,C1(C(=O)OC)CC(C(=O)NCCCCNC(=O)C(C)(C)C2CC2)C1(C)C 53835,c1(OC)cc(F)cc(C(N2CCOCC(CNC(=O)C3=NOCC3)C2)=O)c1N 53836,c1(CC(=O)NC23CCN(C(=O)CC4CCOCC4)CC2C3)c[nH]c2nccc-2c1 53837,c1(OC(N(CCCC(=O)N(CC(=C)C)CC(=C)C)C)=O)ccc(C)c(F)c1 53838,C(=O)(C(C)(C)C(C)O)N1CC(CNC(C2(CC=C)CCC2)=O)C(C)C1 53839,c1(C(C)OC)nc(C)c(C(N2CC(CNC(=O)C=CSC)C(O)C2)=O)s1 53840,CC(C(=O)NC1CN(C(=O)CC(F)F)CCC1c1ccccc1)S(N)(=O)=O 53841,C1(C(C)NC(c2n(C(C)C)ncc2)=O)CN(C(=O)CC2CN(C)C2)CCO1 53842,C(=O)(C#CC1CCCO1)N(C)CC1(O)CCN(C(c2nn(CC)c(O)c2)=O)C1 53843,Cc1ccc(-c2csc(CC(=O)NCC(CC3CC3)NC3CCCO3)n2)cc1 53844,C(=O)(C(C)CC(C)(C)C)N1CC(NC(CN(C(C)C)C)=O)C(C(F)(F)F)C1 53845,C=CCCCCCC(=O)N(C1CCCCN(C(=O)C(C)(C)OCCC)C1)C 53846,N1(C(C2(C)CCCC2O)=O)CC2(CC(CNC(c3cccn3C3CC3)=O)C2)C1 53847,C1(NC(C=CCCC)=O)CC1C1CCCN(C(=O)Cc2ccccc2OC)C1 53848,N1(C(c2c(C)cco2)=O)CCC(C)C(N(C)C(c2cncc(C(F)(F)F)n2)=O)C1 53849,c1(C(=O)OCC)c[nH]c(=NC2CCC3CCC23)cn1 53850,C1(NC(CONC(CN(CCOC)C)=O)=O)CCCCC1F 53851,c1(C(=O)NC(CNC(CCC(C)(F)F)=O)C2CC2)cc(N)c(Cl)c(O)c1 53852,N1(C(c2c(C)nc(C)o2)=O)CCCC(C(N2CCC(CC(F)F)C2)=O)C1C 53853,C(=O)(CC1=CCN(C)CC1)NCCCC(CCC)NC(C1CCC(C)=C(C)C1)=O 53854,C=CCCCC(C)NC(C1C=CCCN1C(c1cc(C)oc1C)=O)=O 53855,c1(NC(C2N(Cc3ccc(C)nc3)CC2)=O)cccc([N+](=O)[O-])c1F 53856,NC(=O)CCC(=O)N1CCCC1CCNC(c1csc(Br)c1Cl)=O 53857,c1(N2CCC(NC(c3c(C)nsc3)=O)C(C)C2)ncc2cc(F)cc(Br)c2n1 53858,C1(C(C(=O)OC)N(C(=O)COC(=O)CCC2CC2(F)F)C)CCCOC1 53859,C1(NC(COc2ccc(C(=O)NC(C)C)cc2)=O)CCN(C(=O)N(C)C)C1C 53860,c1(C(=O)NC2CCC(CNC(C3ON=C(C)C3)=O)C2)ccc2c(c1)CC(C)O2 53861,N1(C(C(=O)NCCSC)c2cccs2)CCc2c(Cl)cc(Cl)cc2C1 53862,Cn1cc(CNC(=O)C(=O)NC2CC3CCC2O3)c(-c2ccnn2C)n1 53863,C1(CNC(=O)CC2C=CCCC2)(NC(C2CCCCC2O)=O)CCCCC1 53864,c1(OCC=C)ccc(Cl)c(C(=O)NC2CCC2NC(C2(C)CC3CCC2O3)=O)n1 53865,Cc1cc(C(=O)NC2CCOCC2C(=O)N(CCCO)C2CCC2)c(C)n1C 53866,Cc1nc(CO)sc1C(=O)NCC1CCCC(NC(c2cc(C(C)C)on2)=O)C1 53867,C1(NC(c2ccccc2F)=O)CN(C(c2ccc(C3CCOC3)s2)=O)CC1F 53868,C1(C(=O)NC(CN(C)C(C2(CCF)CC2)=O)(C)C)CC12CCOCC2 53869,C(=O)(C1=CSCCO1)NCC1N(C(C(CC2CCC2)OC)=O)CC1 53870,c1(C(N(C2CC(NC(C3CC3c3ccn(C)n3)=O)C2)C)=O)nccnc1N 53871,CC1CC(N(C(=O)C(F)C2CC(NC(c3c[nH][nH]c3=N)=O)C2)C)CCO1 53872,c1(C(=O)NC2CC(CNC(C(C)N(C)C)=O)C(O)C2)ncc(Cl)cc1F 53873,C12(C(=O)NC(C3CCN(CCOC)CC3)C)CCCC1C2(F)F 53874,C(=O)(C1=NOC2(CCC2)C1)NC(CCC)CCCNC(=O)C(C)(F)F 53875,CC1CCC1CC(=O)NCCC1CC(NC(C2(C(N)=O)CC2)=O)C1 53876,C(=O)(CC(C(F)F)NC(c1cnco1)=O)NC(C)(C)C(F)F 53877,c1(C(N2C3CC(NC(=O)COCCF)CC2CC3)=O)ccc(F)c2[nH]ccc12 53878,C1(C(=O)NCCN(C(=O)CCNCCCNC(N)=O)C(C)C)(OC)CCC(C)C1 53879,N1(C(c2c(CC)con2)=O)CC2(CCN2C(=O)CCN2CCC(F)C2)C1 53880,c1(SCC2C(C(N(CCCNC(=O)Cc3ccccc3)C)=O)C2)ccccc1F 53881,c1(CCC)onc(C)c1C(=O)NCC1(C)CCC(NC(c2ccc(C)cn2)=O)C1 53882,N1(C(c2n(C)nc(O)c2)=O)CCC2(CC1)CC2C(N1CC2CCC(CC2)C1)=O 53883,N1(C(CN(CC)CC)=O)CCCC12CCN(C(=O)C(C)CC1CC1)C2 53884,C1(C(N(C2CC(F)(F)C2)C)=O)CN(C(c2ccn(CCF)n2)=O)CC1(F)F 53885,C1(O)(CN(C(C2(COC)CC2(F)F)=O)C)CCN(C(C2CC2(C)C)=O)C1 53886,C1(n2cc(CNC)nn2)CCN(C(C23CCCC2CC3)=O)CC1 53887,C(=O)(C1CCCn2cncc21)NCC(C(C)C)NC(COC(C)C)=O 53888,CC(CC(C)(C)C)C(=O)N1CCC1CNC(c1ccncc1Br)=O 53889,Cc1ccnc(Cl)c1C(=O)NCC1CCCCC1Nc1cncc(Cl)n1 53890,N1(C(CC2C(C)C2)=O)CCC2(CC1)CCN(C(C1CC13CC(C)(C)C3)=O)CC2 53891,c1(CC(N2CC3C(CNC(C4(CCCC)CC4)=O)C3C2)=O)cc(F)ccc1Cl 53892,c1(C(N2CC3CC(NC(c4c(CC)cccc4)=O)C3C2)=O)ccn2nccc2n1 53893,C(CCOC)(C(=O)NCCC(C)C1CCCC1)NC(C(C)OCC)=O 53894,C(=O)(C(CCC(C)C)NC(=O)C1=CCC(C)CC1)N(C)Cc1nc(C)[nH]n1 53895,CC(C)C(CCN(C)C(c1ccc(-c2ccccn2)nc1)=O)NC(=O)C(C)O 53896,Cc1cc(CC2CC3COC2C3)c(C)n1C.C1CCC(=O)NC12CCC2 53897,c1(CC(C(=O)N(CCCNC(C2(CC#C)CCCO2)=O)CC)C)ccc(F)cc1 53898,Cc1ccc(S(=O)(=O)NC2CCC(C(=O)Nc3ccccc3CO)CC2)cc1Cl 53899,C1(CNC(C(C)Cc2ccncc2)=O)CC2(CC2)CN1C(c1nccnc1N)=O 53900,CCC(CC)CC(F)C(=O)N1CCCC(CCNC(c2cc(C#N)n(C)n2)=O)C1 53901,c1(C(N2CCC(N(C(COCC=C)=O)CC)C2)=O)cccc2nc(O)[nH]c12 53902,C(=O)(CC(O)C1CC1)NC1CC(CCNC(=O)OC(C)(C)C)C1 53903,C1(NC(C=CC(C)(C)SC)=O)CN(C(=O)CCc2ncc[nH]2)CC1C(F)F 53904,C1(CN(C(=O)C=CC2CCCO2)C)CCN(C(c2cnoc2-c2cccs2)=O)C1 53905,Cc1ccc(CNC(=O)CC2CC(C)N(C(=O)C(C)CC3CC3)C2)c(C)c1 53906,Cc1ccc(CCNC(=O)C(C)CNC(=O)C(n2ccnc2C)C)cc1 53907,c1(C(N(CC(CC)NC(=O)COC2CCCOC2)C)=O)ncc(C)cn1 53908,c1(CN(C(=O)CN2CCSCC2)CCNC(C2CC(C#N)C2)=O)cccc(Cl)c1 53909,N1(C(CC(C)C2CCCO2)=O)CCC(NC(=O)CSC2CCOC2=O)C(C)(C)C1 53910,c1(C(N(CC(C)N(C(=O)Cc2cccc(F)c2F)C)C)=O)cc(F)ccc1F 53911,c1(C(N2CCCCC(NC(C3N(N=O)CCCC3)=O)C2)=O)cc2cn[nH]c2cn1 53912,c1(NC2CCC(CCC(=O)N(CCCN(C)C)C)O2)ccc(S(N)(=O)=O)cc1Cl 53913,CC1(C)OC2(CC(c3ccc(F)c(O)c3)=O)CCC1(C(=O)O)CC2 53914,CC(O)C(C(=O)N1CCC(C)(NC(c2cnn(-c3cccnc3)c2)=O)C1)N(C)C 53915,c1(NC(C(CC2CC2)NC(C(CC2CCC2)OC)=O)=O)cnc(C)c(Cl)c1 53916,c1(CCC(=O)NC2CN(C(=O)CC34CCCC3C4)CC2O)cccnc1F 53917,C(CN=c1[nH]c2cccc(F)c2s1)(C1CC1)NC(=O)C#CC1CCCCC1 53918,CS(=O)(=O)c1ccccc1C(N1CCCCC(NC(=O)C2=COCCC2)C1)=O 53919,C1(NC(CC(C(C)OC)NC(=O)Cn2ccccc2=O)=O)CC2(CNC(=O)O2)C1 53920,C1(CC)CCCCC1OCC(=O)Nc1nc(CNC(=O)CC2CCC2OC)cs1 53921,C1(OC)CN(C(=O)CC2CCC=CCC2)C(C)(CNC(=O)Cc2csnc2C)C1 53922,CN1C(=O)OCC12CN(C(=O)NCc1ccnc(OC3CCCC3)c1)C2 53923,CC(C)C(C)(O)C(=O)NCc1cn(CC(=O)NC2CCC3CCC23)nn1 53924,N1(C(CCC(C)SC)=O)CC2CCCC2(NC(=O)Cc2ccn(C)n2)C1 53925,N1(CCCCNC(C(C)Cc2cnc[nH]2)=O)CCCC(NC(=O)CCCSC)C1 53926,c1(NC2CN(C(c3c(C)[nH]nc3Cl)=O)CC2C)cc(=O)n(C)cn1 53927,N1(C(CSCC)=O)CCC2CCN(C(c3cnc(-c4ccccn4)s3)=O)CC12 53928,c1(C(N(C2CCN(c3ncc(Cl)c(O)n3)CC2)CCC)=O)coc2c1COC2 53929,C(=O)(CCCC(=O)N(CCCN(C(=O)CN1CC(C)C1)C)C)NCCC 53930,N1(C(c2cccc(NCC)c2)=O)CCC(C2CC2)(CNC(C2CNC(=O)C2)=O)C1 53931,CC(C)CCC(=O)NCC(=O)NC1CC(CNC(c2ncn(C)n2)=O)C1 53932,C(=O)(CC(COC)NC(=O)CC1(OC)CCC1)NCC1(CO)C(C=C)C1 53933,N1(C(=O)CNC(C2(n3nccn3)CC2)=O)CCC(C2CCCC2)C1 53934,C(=O)(C(C)CCN(C)C)N1CC(CCNC(CC(=O)OCC)=O)(OC)C1 53935,c1(CNC(C(C2CCOC2)OC)=O)ccc(C(=O)NCC2CC2[N+](=O)[O-])o1 53936,N1(C(c2cncc(C(C)C)c2)=O)CC(C)CCC1CNC(=O)Cc1cnnn1C 53937,C#CC1(C(N2CC(CC(F)F)C2)=O)CCN(C(=O)C(C)C2CC2)CC1 53938,c1(COC)nc(C(=O)NC(C)C(CO)NC(=O)C(F)=C(C)C2CC2)n[nH]1 53939,C1(C(=O)NCC(F)(F)C(C)(C)O)(CC)CCCN(C(=O)C=Cc2cc(C)no2)C1 53940,N1(C(CC=C=C)=O)CCC(C(=O)NC2C=CCCC2)C1(C)C 53941,CC(CSC(F)(F)F)C(=O)N(CCCCCNC(=O)CCC1CNC(=O)N1)C 53942,Cc1c(C(=O)N(CCC(C(C)C)NC(C2COCCO2)=O)C)cccc1F 53943,c1(C(=O)NCC2(CCNC(CC3C(C)CCC3)=O)CC2)c(F)cc(F)cc1Cl 53944,C1(CC)(CC)CC(O)CN1C(=O)C(C1CCN(C(c2cc(F)n(C)n2)=O)C1)F 53945,n1(CCOC)nnnc1C(c1cncn1C(C)C)NC1CCC(NC(N)=O)C1 53946,C1(CNC(C2(CC)CC2(F)F)=O)CN(C(=O)CCc2cccn2C)CCC1(C)C 53947,C1(N(C(C(CC#C)C2CC2)=O)C)CN(C(c2ccc(C(N)=O)cc2)=O)CC12CC2 53948,C1(NC(C2CCC3CCC23)=O)CCN(Cc2ccc(-c3ccc(Cl)cc3)[nH]2)CC1 53949,C1(CNC(C2CN(C)C2)=O)CC(NC(c2ccc(Cn3cccn3)o2)=O)C(O)C1 53950,C1(C)(NC(C(N2CCCC(C)C2)=O)=O)CCCN(C(c2ccnc(O)c2)=O)C1 53951,Cc1nc2cccc(C(=O)NCC3CC3NC(C3(CC(C)C)CCCC3)=O)c2[nH]1 53952,CC1CCOC1CO.c12cn(nn1)C1CC(C1)C(=O)N(CCCO)CC2 53953,N1(C(C(C)CC2CCCC2)=O)CCCCCC1CNC(=O)CCCCCN(C)C 53954,N1(C(c2ccc(NC)cc2)=O)CCCCC(CNC(=O)C(C)CN2CCCC2)C1 53955,c1(CC)nccnc1C(=O)NCC(C)CC(=O)NC1CC2CCC1O2 53956,C(=O)(C1=CC2CCCCCC12)N1CCC(C(C)NC(c2ccc(C(C)=O)s2)=O)C1 53957,C(c1ccc(S(=O)(=O)NC)cc1)=CC(=O)NCC(CC=C)NC(=O)CC1CC1 53958,C=CCCC(C(=O)OC)NC(C1(NC(=O)C(C)SC)CCSC1)=O 53959,C1(CN(C(=O)Cc2cccs2)CC)CCN(C(=O)C(F)COCCSC)CC1 53960,Cc1nsc(C(N2CC(F)(CNC(=O)CSC(F)(F)F)C2)=O)c1N 53961,O(C1CCc2c(Br)cccc21)C(=O)C(c1ccc(F)c(F)c1)=O 53962,N1(C(C2(F)CCN(C(C(C=CC)O)=O)C2)=O)CC(C)OC(C)(C)C1C 53963,C1(C)(C(=O)NCCN2CCN(C(C3OCCC(C)C3)=O)CC2)CCS(=O)(=O)CC1 53964,c1(C(N2CC(c3ccc(C)cc3C)OCC2)=O)cc(N)cc(O)c1Br 53965,c1(C(=O)NCCC2(CNC(C3CC3C(=O)O)=O)CC2)cc2c(cn1)CCCC2 53966,Cc1nsc(N)c1C(=O)NC(CNC(=O)CC(C)n1ccnc1)C(C)(C)C 53967,N1(CC)CCN(C2CN(C(C)C(OC)OC)C2)CC1.C(C)(C(=O)O)OCCO 53968,Cc1c(NC(c2ccnc(O)c2)c2nnnn2CC(F)F)ccc(Br)c1Cl 53969,C1(CNC(CCCCC#C)=O)CCCC2CN(C(=O)Cc3ccc(F)nc3)CC12 53970,n1(CC(=O)N(C2CN(C(=O)COCCN(C)C)CC2F)C)cnc2ccccc12 53971,Cc1cnn(CC(=O)NC2CC(CCNC(=O)C(C)Oc3cccnc3)C2)c1 53972,CCC(CC(=O)NCCCOCCCNC(C1OCCC1C)=O)C(F)F 53973,N1(C(C2C(C=C)OCC2)=O)C2CCC1CC(NC(=O)C(C)(C)c1cncnc1)C2 53974,N1(C(C2C(C)=C2)=O)CC2CCCC(C1)N2C(=O)CC(C)c1ccco1 53975,C1(C(=O)NC(CCNC(Cc2ccn(C)c2)=O)(C)C)CCNC(=O)C1 53976,C(=O)(C1=Cc2ccccc2C1)N(CCC(=O)NC1COCCC1O)CC=C 53977,C(=O)(C1=C(Cl)CC1)NCC(O)COC(N(CC(=O)NCCOC(C)(C)C)C)=O 53978,N1(C(CN(CCC)C)=O)CCC2(NC(C3CCN(C(C)=O)CC3)=O)CCCCC12 53979,C=C(C)C1CC=C(C(c2nnnn2CC)NCc2cc(F)cc(Br)c2)CC1 53980,N1(CC(=O)CCNC(=O)C(c2ccc(Br)cc2)(F)F)CCC(C(O)C(F)F)CC1 53981,c1(C(N(C2CCCCCC2)CCN)=O)cc[nH]c(=N)n1.C(=O)(CCC1CCCO1)OC 53982,Cc1ccc(CC(=O)NCC2CCN(CCN(C3CCCO3)C3CC3)C2)c(C)c1 53983,N1(C(c2c(CC)nc[nH]2)=O)CC2CCC(C1)C2CNC(=O)C(C)NC(=O)COC 53984,C12(C(=O)NCC(C(C)C)O)CCC(NC(=O)CC(C)O)(CC1)C2 53985,CC(C)CC(CNC(=O)C1=CCCOCC1)C(=O)N1CCc2nn[nH]c2C1 53986,C(=O)(CC(O)CNC(C1CCCC1O)=O)NCC(=O)N(CC)CC 53987,Cn1nc(CNC(c2cc[nH]n2)=O)c2c1CCN(C(=O)CC1CCOC1=O)C2 53988,c1(CC)ccc(C(C)C(=O)N(CCNC(=O)CC(C)C2CCCO2)C(C)C)cc1 53989,C(=O)(C(CC(C)C)NC(C)=O)N1CCC(OC)(CNC(c2sccc2C#N)=O)C1 53990,C(=O)(C1=CCCC1(C)C)N1CC2C(NC(c3cn(C)nn3)=O)(CC2)C1 53991,c1(C(N(CCCNC(=O)Cc2ccnn2C)CC)=O)cnc(Cl)c(F)c1N 53992,c1(COCC)nnc(N2CCCC2CCNC(=O)C2CC2)s1 53993,CC1CC(NC(c2cc(C#N)n(C)n2)=O)CCN1C(c1cnc(C(C)(C)C)[nH]1)=O 53994,C=CCN(OC)C(=O)CCC1CCCN(C(=O)CC2CC(F)(F)C2)C1 53995,C(C1=NOC2(CCC2)C1)NC(C1CCN(C(C(CC)N(C)C)=O)C1)=O 53996,Cn1ccc(-c2cc(C(=O)NCC3CCN3C(=O)CC3CCSCC3)n[nH]2)c1 53997,c1(OC)cc(CC(=O)NCCc2ccc(-c3ccccc3)[nH]2)cc(OC)c1O 53998,C1(C(=O)NC(c2nccn2C)CC)CCCN(C(c2nn(C)cc2C)=O)C1 53999,C1(N(C)C)(C(=O)NC2CCCC(N(C(=O)C=Cc3cc[nH]n3)C)C2)CCCCC1 54000,c1(CC)nc(C)n(C)c1C(N1CC(F)(CNC(C2(C)CC(C)=NO2)=O)C1)=O 54001,Cc1nc(CC(=O)NC(Cc2cn[nH]c2)C(=O)NC2(C)CC2)n[nH]1 54002,C1(NC(CCc2nc(C)c(C)[nH]2)=O)CN(C(=O)CC2CCCCC2)CCC1C 54003,c1(-c2cc(NC(C3CCCCCC3)C)sc2)ccc(F)cc1 54004,c1(C(=O)NC(C)CNC(C2CCN2S(C)(=O)=O)=O)cnc2n1CCS2 54005,C1(CNC(C2CCC(C)(C)C2)=O)C(C2CC2)CCN1c1nccnc1F 54006,CCCCC(CC)CC(=O)NCCCCCCN(C(=O)C(CC)C(C)(C)CC)C 54007,c1(CC(C(=O)N(CCOCCNC(C2(CC)CCOC2)=O)C)C)ccccc1Cl 54008,C1(C(=O)NCC2N(C(c3cc(C)sc3C)=O)CC(F)C2)CCCC2(CC2)C1 54009,C1(CNC(C(c2c(F)cccc2F)(C)C)=O)C2CCC(C2)C1N 54010,C1(NC(c2c(COC)cc[nH]2)=O)CC(C)CN(C(=O)COCCF)C1 54011,Cc1cc(Br)ncc1NC(=O)CCC1CCCN1Cc1cnn(CC(C)C)c1 54012,N1(C(C2CN(C(Cc3cccc(C)n3)=O)CC(F)C2)=O)CCC(O)C(C)(CO)C1 54013,c1(NC(C)C)ncccc1C(=O)NC1CCCC1NC(C1CCOC1C1CC1)=O 54014,c1(NC(CNC(C(C(C)C)NC(COC)=O)=O)(C)C)cc(C)ncc1C(=O)OC 54015,Cc1cc(F)ccc1C(C)Nc1ccc(=O)n(CC2CCNCC2)c1 54016,C(C)(C)(CC(F)C(=O)N(C1CCOC(C)(C)C1)C)NC(C1C(C)OC(=O)N1)=O 54017,CC1(C)CC=C(C(=O)NCC(C)(C2CC2)NC(c2ccc(O)nn2)=O)CC1 54018,C1(CNC(CN(C2CN(C)CCO2)C)=O)CCN(C(c2ccccc2)=O)C12CC2 54019,C1(NC(CCN(C(=O)C(C)CC2CC2)C(C)C)=O)CC1C1CC1 54020,N1(C(c2ccno2)=O)CCCC2(CCN(C(c3nccc4ncccc34)=O)C2)C1 54021,C1(OC(C)(C)C)CCCCN1CC.c12ncc(s1)C(=O)OCCO2.C1(=O)NC1 54022,C1(CNC(C2C(=C)CC2)=O)CC2(CO1)CN(C(=O)CC=Cc1cccc(F)c1)C2 54023,C1(CC(=O)NC)CN(C(=O)CC2(CSC)CC2)CCN1C(=O)C(C)C(C)(F)F 54024,S(=O)(=O)(CC(=O)N(C)CCOCCCNC(=O)CC1(C)CCCC1)NC 54025,C1(NC(CCNC(C2CCC2)=O)=O)CC2CC1N(C(C1C3COCC13)=O)C2 54026,CN1CC(C(=O)NCC(C)(C)NC(=O)COC(F)F)c2ccccc2C1=O 54027,C1(NC(C2N(C)CC(F)C2)=O)CC12CCN(C(C1CCc3nn[nH]c3C1)=O)CC2 54028,N1(C(C(CC=C)C)=O)CCC2(CC1)CC2(CO)CNC(c1ccccc1CC)=O 54029,C1(NC(c2c(F)ccnc2F)=O)CC1C1CCCN(C(=O)C2=C(Cl)CC2)C1 54030,N1(c2nc(OC)c(Br)cn2)CC2CCCC(C1)C2C(=O)NC(C)C1CC1 54031,C(=O)(C1=C(C)CCCC1(C)C)N(CC)CC1CCCN1C(=O)Cc1cccc(N)c1 54032,c1(NC(C(CC2CC2)NC(c2cnn(CCF)c2)=O)=O)cccc2c1CCC2 54033,Cc1nc(CNC(=O)CCC(=O)N(C)C)oc1C(=O)NC(C)Cc1nc[nH]n1 54034,C1(CNC(C2(O)COC2)=O)CCC2(CCN(C(C3CC(C4CC4)=NO3)=O)CC2)O1 54035,Cc1cc(C(N2CC(F)(F)CC2CNC(=O)CCc2cnc[nH]2)=O)cc(N)c1O 54036,C1(NC(C(C)OCC=C)=O)C2CCC1N(C(c1nc(C)n(C)n1)=O)C2 54037,c1(SCC(=O)N(CCCN(C(=O)C(C)(C)C)C)C)ncnc2[nH]cnc12 54038,N1(C(c2cc(C)ns2)C(=O)NCCC)CCOCCc2ccccc2C1 54039,C(C(=O)NNC(=O)c1ccccc1CC(F)(F)F)C1(C)CC1(F)F 54040,c1(C(=O)NCC2CCN(C(C3C(C)(Br)C3)=O)C2)coc2ccc(F)cc12 54041,Cc1cccc(F)c1CC(=O)NC1CC1CNC(=O)C(C)(C)CF 54042,C(C(C)CN=c1cc(C)nc(C2CC2)[nH]1)NC(C=Cc1cccc(OCC)c1)=O 54043,c1(OC)cccc(OC)c1S(=O)(=O)NC1COC2(COC2)C1 54044,C1(NC(CCN(C(c2cc(C)[nH]c2)=O)C(C)C)=O)CCC12CCCC2 54045,CC12COC(C(N3CCC(O)(CNC(c4ccns4)=O)C3)=O)(C1)C2 54046,c1(N2C(CNC(C(CCC)OC)=O)C(C)CC2)ccc([N+](=O)[O-])cc1 54047,c1(CCC(N2CC3C(C2)N3C(c2ccc(O)c(Cl)c2)=O)=O)cc(Br)ccc1I 54048,c1(C(=O)NC2C(CC)CN(C(=O)CC(F)F)CC2)nn(C)c2c1CSCC2 54049,Cc1nn(C)c(Cl)c1C(=O)NC12CC(CNC(c3ncccc3O)=O)(C1)OC2C 54050,N1(C(C(C)SCC)=O)CC2(CNC(c3[nH]c(O)nc3C)=O)CCC1CC2 54051,c1(OCCN(C(=O)CCCn2cc(CN)nn2)CC)ccc(C)c(C)c1.C(CO)O 54052,c1(OC)cc(O)c(C(=O)NCCNC(C2CC2c2cccs2)=O)cc1S(N)(=O)=O 54053,C1(CNC(c2cccc(C(C)(F)F)n2)=O)CC2COCC2N1C(c1cnn[nH]1)=O 54054,Cc1c(C(N2CCN(CCNC(=O)C=CC(F)(F)F)CC2)=O)cnn1CC(F)F 54055,C(=O)(Nn1ccccc1=O)C1CC(NC(C(C2CC2)OC)=O)C1 54056,N1(C(CC2C(C)CC2)=O)CC(NC(C2CC(N3CCC3)C2)=O)CC1(C)C 54057,C(C(=C)CCNC(C)=O)NC(=O)C(C)(C)OC1(CC=C)CCC1 54058,c1(C(=O)NCC(C2CCCCC2)NC(C(C)SC(C)C)=O)cccc(N(C)C)n1 54059,C1(C(N2CCC(NC(=O)Cc3ccc(Cl)s3)C(F)C2)=O)CN=C2N=CNN2C1 54060,N1(C(C(C2CN(C(=O)CC3CCC4CC34)C2)OC)=O)CCOC(C(=O)N(C)C)C1 54061,C(CCCCCF)N(C(=O)C=CC(F)(F)F)CCOC 54062,Cc1cn2c(=O)c(C(N3CCC(O)(C(C)CNC(=O)C(C)(F)F)C3)=O)cnc2s1 54063,Cc1nn(C)cc1C(C)C(N1CCC(CNC(=O)C(c2ccn(C)n2)C)CC1)=O 54064,c1(CC)cc(C(=O)NC(CC2CC2)Cc2ccccc2Br)cc(Cl)c1 54065,N1(C(c2cc(C)cc(C)c2C)=O)CCOC2(CCN(C(C3CCN3C)=O)C2)C1 54066,c1(C(=O)NC2CC(C)N(C(c3cc(Cl)n(C)n3)=O)C2)ccc2ncsc2c1 54067,c1(C(N2CCN(C(C3CCC(C)CC3)=O)CC2)=O)cc2cc(Cl)ccc2n1C 54068,c1(C(N2CC(C(C(N3C(C(=O)OC)C=CC3)=O)OC)C2)=O)ccnnc1C 54069,S(=O)(=O)(c1c[nH]c(C(=O)NCC(C)(CO)NC(=O)CC2CC(F)(F)C2)c1)NCC 54070,C(=O)(CCCCNC(=O)C(C)C1CCCO1)NCCSCCOC 54071,N1(C(C(CCC)C)=O)CCN(C(c2ccc[nH]2)=O)CC1c1cn[nH]c1 54072,N1(C(C(COC(C)=O)C)=O)CCC(C)(C(=O)OCc2ccccc2C)C1 54073,N1(C(c2cc(CC(C)C)on2)=O)CCN(C(=O)C=CC2CCC2)C(C)C1C 54074,C12(NC(Cc3ccc(C#C)cc3)=O)CCN(C(=O)CC(C)CCC)CCC1C2 54075,N1(C(C2C(C(C)C)C2)=O)CC(C)(CNC(c2onc3ccccc23)=O)CC1(C)C 54076,CC(C)CC(C)CC(=O)N1CCC(C)C1CNC(C12CCCCC1C2(F)F)=O 54077,c1(OC)cncc(C(=O)NC2CCCC(C(N3CCC(F)CC3)=O)C2)c1 54078,C1(NC(C2C(OC)C2)=O)C2CC(O)C1N(C(=O)CNC(c1cscn1)=O)C2 54079,c1(NC(C2CN(c3ccncn3)CCO2)=O)ccc2c(=O)[nH]ccc2c1 54080,c1(C(N2C(CC(N3CCC(C#C)CC3)=O)COCC2)=O)cc(Br)c(O)c(Br)c1 54081,C1(C(=O)OCC)CN(N(C)CCCOC)CC1c1noc(C2COCCO2)n1 54082,C1(S(N)(=O)=O)(C(=O)NC(C)CN(C(=O)CCC#N)C)CCCC1 54083,CCCC(CNC(=O)CC1(O)CCCC1)NC(=O)CC1CCOC1C 54084,C(=O)(C(C(C)O)N(C)C)NCC1(NC(C=C(C)C)=O)CC1 54085,N1(C(C(C)NC(N)=O)=O)CC2(C1)C(NC(c1ccoc1)=O)CCS2(=O)=O 54086,c1(CCN(C(c2n[nH]c(C)n2)C(=O)NC2CC2)C(C#C)C)ccccc1 54087,C(=O)(C1=CCCCO1)NC(C)CNC(C1(Oc2ccccc2)CC1)=O 54088,CCCCC(CNC(=O)CCOC(C)=O)NC(=O)C(N1CCCCC1=O)C 54089,c1(OC(C(N2CCC(OCC=C)C2)=O)C)c(F)cccc1F 54090,N1(C(=O)C(F)=C2CCC2)CCCc2cc(C(F)(F)F)ccc21 54091,c1(C(=O)NC2CC(CNC(CC(CCC)O)=O)C2)cc(F)cc2nccnc12 54092,c1(CCC(=O)N(C)CC2N(C(CCSC)=O)CCC2)ncc(F)cn1 54093,N1(C(c2c(CC)noc2)=O)CCN(C)C(C(=O)NCC2CCCCS2)C1 54094,O=C1CC2CC(Nc3ccc(N4CCN(CCO)CC4)cc3)C1C2 54095,C1(C(=O)OCC)(C(C)C)CCN(Cc2ccc(-c3scnc3C)cc2)CC1 54096,c1(C(N(CC(=O)NCC2(O)CCC(C)C2)CC#C)=O)cccc(CC)c1 54097,c1(C(=O)NC2CCC(N(C)C(c3ccccc3Cl)=O)CC2)cc(F)ccc1F 54098,c1(CN(CCNC(=O)NCC2CC(CC(C)C)OCC2)C)ccc(Cl)cc1Cl 54099,CC(C)CC(C(=O)NC1CCN(C(=O)C(C)SC(C)C)CC1)N1CCCCC1=O 54100,N1(C(CC(COC)(C)C)=O)CCC2(C=C(C(=O)NCCc3ccc(O)cn3)C2)C1 54101,C1(C(C)C)CCC(CC(C(=O)NC2(C)CC2)N(CC(C)(C)CO)C)CC1 54102,N1(C(C(CCCC)O)=O)CCCC(C2CCCN(C(=O)CC3CC(OC)C3)C2)C1 54103,c1(C(=O)NCC2C(CNC(CCC(=C)Br)=O)C2)cc2ccccc2n1C 54104,N1(C(C2CC3C=CC2CC3)=O)CC2CCN(C(c3cnc4cccnn34)=O)C2C1 54105,C(=O)(CCCC(=O)OC(C)(C)C)NC1(CCNC(Cc2n(C)cnc2)=O)CC1 54106,c1(CCC)onc(C)c1C(=O)NC(CNC(c1cc(C(F)F)ccn1)=O)C1CC1 54107,N1(C(C2(F)CCOC2)=O)CCC2(CC1)CC(NC(C13CCC(CO)(CC1)C3)=O)C2 54108,c1(C(=O)NCC2C(C(=O)O)C(C)C2C)ccc(F)c2[nH]ccc12 54109,C12(NC(CC(=C)C)=O)CCC(CNC(=O)CCCOc3ccccc3F)(C1)OC2 54110,c1(CC(=O)N(CCCC(C)C)Cc2ccc(C)s2)cn2ccccc2n1 54111,C1(NC(COCCCCC)=O)CCN(C(=O)CC(O)C(C)C)CC1O 54112,C(c1cn(C)cn1)=CC(=O)N(CCC(C)NC(=O)C(=Cc1c[nH]cn1)F)C 54113,C1(CNC(C2CN(C)C(=O)C2)=O)CC(C(=O)NCc2cn[nH]c2)=NO1 54114,CCCC1CC(=O)C2CC3C(C(Nc4cc(C)cnc4OC)C2C3)C(=O)N1 54115,CCCCCCC(C(=O)NCC=CCNC(C1(C)CC=CCC1)=O)NC(C)=O 54116,C1(CC(=O)N(CCNC(CC2N(CC)C(=O)CC2)=O)C(C)C)CC2C=CC1CC2 54117,c1(-c2scc(C(C(=O)NCc3ccco3)N(C(C)C)CC)n2)cccc(C)c1 54118,c1(C(N2CC(CNC(C=C)=O)C(C(F)(F)F)C2)=O)c(OC)cccc1F 54119,C1(CNC(CN(C(COC)=O)C)=O)CCC2(CN(C(c3c(C)n[nH]c3C)C)C2)O1 54120,N1(C(Cc2c(C)occ2)=O)CC(NC(c2cocc2C(N)=O)=O)CC(F)C1 54121,c1(C(=O)NCC2C(NC(C(=O)NCC)=O)C2)ccc(F)cc1Br 54122,c1(C(=O)NCCNC(C(C)O)=O)ccn(CC(F)(F)F)c(=O)c1 54123,N1(C(c2cc(C)ns2)=O)CCCN(C(C2CCn3nccc3C2)=O)C(C)C1 54124,c1(C(N2C3CN(C(c4ccc(C(N)=O)cn4)=O)CC2C3)=O)ccc([N+](=O)[O-])cn1 54125,N1(CC(=O)NCC(C)N(C(c2c[nH]c(=N)s2)=O)CC)CCCCCC1 54126,N1(C(C2C(CNC(C(C)O)=O)CC2)=O)CC(C)c2ncccc21 54127,N1(C(CC2CCC(C)(O)CC2)=O)CC2(CCCC(CNC(C3(Cl)CC3)=O)O2)C1 54128,N1(C(CC2ON=C(C)C2)=O)CCC(O)(CCNC(c2cc(C(F)F)cs2)=O)CC1 54129,CC(C)CCCCC(=O)NCCCC(O)C(=O)NCc1cc(Cl)ccn1 54130,C1(NC(CCN(C(C)C)C(C2C=CCS2)=O)=O)C(O)CC1O 54131,c1(C(N2CCC(NS(C)(=O)=O)C2)C(=O)NCCCSC)ccc(C(C)(C)C)nc1 54132,c1(NC(=O)NCC2CCCC2NC(=O)C(Cl)(Cl)Cl)cnncc1Cl 54133,C(=O)(CCCCCCCCN)N1CCN(CC(=O)Nc2c(OC)cccc2)CC1 54134,c1(CNC(=O)OC(C)(C)C)ccc(O)cc1O.C12CCC(C1)C(=O)O2 54135,CC1(NC(C2CCCC2O)=O)CCN(C(=O)Cn2nnc(=N)[nH]2)C1 54136,C1(CNC(COCC)=O)CN(C(=O)C(C2CC2)SC)CCC1(C)C 54137,C1(C(N(CCC(=O)N2CC(n3cc(CO)nn3)C2)CC)=O)Cc2nccnc2C1 54138,Cc1c(C(=O)NCC(C)CNC(=O)C(C(C)C)NS(C)(=O)=O)ccc2c1CCC2 54139,N1(C(CN2CC(CC)C2)=O)CCN(C(=O)CC2(OC)CC2)C2CC12 54140,c1(NC(C2(C)CN(Cc3cc(Cl)cnc3Cl)C2)=O)ccc(C(F)(F)F)cc1[N+](=O)[O-] 54141,C1(C(C)C(=O)N(c2ccn(C)n2)C2CC2)CCCN(C(c2cnc(=N)[nH]c2)=O)C1 54142,c1(CNC(c2cnn(C)c2C)c2n(CC)nnn2)cn(C)c2ccccc12 54143,C1(NC(c2c(CC)nn[nH]2)=O)CC(CNC(=O)CNC(=O)CN(C)C)C1(C)C 54144,N1(C(CCN(C(C)=O)C)=O)CCN(C(=O)C(Cl)=CCl)CCC1C 54145,C#CCC(C(=O)NCC(C)C(=O)OCC)NC(c1cc(CC)nn1C)=O 54146,c1(SC)cccc(F)c1C(=O)NCC1COCCN(C(c2cnccn2)=O)C1 54147,C1(CC(=O)NC2C(NC(c3cc(=N)[nH]cc3)=O)C2)CCC2(CC1)OCCO2 54148,c1(C(C(=O)NCCCCCN(C(C2CC(C)C2)=O)C)O)ccc(F)c(Cl)c1F 54149,c1(CNC(CC(C)NC(=O)CC2CCOC2(C)C)=O)ccccc1C#N 54150,C(=O)(N1OC2CCC1CC2)C1(C#C)CCNCC1 54151,Cc1cc(C(=O)N(CC(C)N(C)C(C2CCCN2C)=O)C)ccc1C(F)(F)F 54152,CCCCC(CC)C(=O)NC1CCCC1NC(=O)C(C)(C)c1cnc[nH]1 54153,C1(NC(c2cc(-c3nc(C)sc3)oc2)=O)CCN(C(c2nnn(C)n2)=O)CC1C 54154,C=CCC(C)(O)C(=O)NC1CCCC1C(=O)NOCC(=C)Cl 54155,c1(CCCC(=O)NCC2CC2NC(=O)Cc2ccc(Cl)s2)nc2ccccc2s1 54156,c1(N2CCOCC(CNC(C3OCCN(C(C)C)C3)=O)C2)cc2nncn2cn1 54157,C1(NC(C2C(C)C2)=O)CN(C(=O)C(C)S(C)(=O)=O)CCC12CCC2 54158,CC1(C)CCC(C)(NC(=O)CC2(NC(=O)C=CCN3CCC3)CCC2)C1 54159,Cn1nc(CNC(=O)C(C2CCOC2)NC(=O)OC(C)(C)C)cc1C(F)(F)F 54160,N1(CC(=O)NCC(C2CCC2)NC(c2cccnc2O)=O)CCS(=O)(=O)CC1 54161,C(=O)(C1=CC(O)C(NC(C2CC23CC3)=O)C1)N1CC(C2(C)CC2)C1 54162,C(C(C)C)(C(O)C(=O)NC(CNC(c1cc(C)ns1)=O)CO)OC 54163,c1(C(c2nnnn2C2CC2)NC2(C=C)COC2)cn(C(C)C)nc1Br 54164,CCCCC(C(=O)NC1(C2CN(C(=O)C3=CCOC3)C2)CC1)N(C)C 54165,C1(CC(=O)N(C)CC2N(C(C(F)OC)=O)CCC2)CCCN(C(C)C)C1 54166,Cc1cccc(C(N2CC=CC(NC(C3CC(N=[N+]=[N-])C3)=O)C2)=O)c1F 54167,C(=O)(CCCC(C)(F)F)N(C1CCCN(C(C(C=CCCC)O)=O)C1)CC 54168,N1(C(=O)CCC2CCC2)C2CCC1CC(CNC(C1(N3CCOC3=O)CC1)=O)C2 54169,C(=O)(CC(C)(C)CC(F)(F)F)N1CCC(COC)(NC(=O)C(F)=C(C)C)C1 54170,C1(NC(c2cc(CC)n(CCO)n2)=O)CN(C(C2CC(=O)N(C)C2)=O)C(C)(C)C1 54171,N#CCCCC(=O)N1CC(F)CC1CNC(c1cccnc1-n1nccn1)=O 54172,c1(OC)c(Cl)ccc2[nH]c(C(N3CCCC(CNC(=O)C4=CCCS4)C3)=O)cc12 54173,C=CC1(CC(=O)NC2(C)CCN(C(c3c[nH]c(=N)nc3C)=O)C2)CCCCC1 54174,CCC(CO)CN=c1cc(C)[nH]c(=NCCN2CCC(F)(F)CC2)[nH]1 54175,c1(C(N2CC(NC(C(C=C)(C)C)=O)C(C)C2)=O)c(C)ccn1C 54176,C1(CNC(CCOCC#C)=O)CCN(C(=O)CCCCc2cnc[nH]2)CC1(F)F 54177,N1(C(C2CC(C(C)C)C2)=O)CCC2(NC(=O)C=Cc3cnc[nH]3)CCCCCC12 54178,N1(C(C2OCCN(CC)C2)=O)CC2(CCN(C(=O)CCC(C)C)CC2)CC1C 54179,CC1CCCCN1C(=O)CN(C(=O)C(=O)N(C)C1CC1)CC1CC1 54180,N1(C(C(F)=CC)=O)CCN(C(=O)C(CC(F)F)c2ccc(F)cc2)C(CCC)C1 54181,c1(CC)cc(NC(=O)CC2(OC)CCOCC2)nc(CC)n1 54182,C(C(C)C(C)C(=O)N1CC(O)CC1CNC(=O)C(C)=CC1CC1)OC 54183,C(=O)(CC(C)CC(C)C)NCCC(C(=O)NCCCOC=C)(C)C 54184,c1(CC)cc(C(=O)NC(c2cccc(C)c2)CNC(=O)C(C)OCC)ccc1Cl 54185,N1(C(C2CCCN(C)C2)=O)CCC(NC(C2CC3C(C2)C3(F)F)=O)C(CO)CC1 54186,N1(C(C2(C)CCCO2)=O)CC2(NC(=O)CCC3(C#N)CCC3)CC1C2 54187,C=CCC(C(=O)NC1(CC(=O)NC(C)Cc2ccncc2)CC1)C(C)C 54188,C1(COC(C2CCC(C)CC2)OC)CCN(C(c2cccc(OC)n2)=O)CC1 54189,c1(C(=O)NC(CC(C)NC(c2c(C)ccnc2C)=O)C)n[nH]c2cccnc12 54190,c1(C(=O)OCC)nc(=NC(C)CNC(=O)Cc2cc(O)nc(O)n2)cc[nH]1 54191,C12(CNC(C(CC#C)(C)C)=O)CCCC(CN1C(=O)CNC(=O)OCC)C2 54192,C1(CCC)CN(C(=O)Cn2ccc(C)n2)CC1C(=O)N(C12CC(C1)C2)C 54193,C1(C(=O)NC(C(C)C)(C)CNC(=O)Cc2cnn(C(F)F)c2)CC2(CCC2)CO1 54194,C1(C(=O)NCC2N(C(c3c(OC)c(C)ncn3)=O)CCC2)CCCC1S(C)(=O)=O 54195,CC1COCCN1C(C1CC1c1cccc(Br)c1)=O 54196,C1(NC(C2CC=CCO2)=O)CCOC12CCN(C(=O)Cc1ccccc1F)CC2 54197,C12(C(=O)NC(CC(=O)N3CCC(C(=O)NC)C3)COC)C(=O)C3CC1C2C3 54198,C#CC1(C(N2CC(OC)CC(NC(c3cccc(F)c3C)=O)C2)=O)CCOCC1 54199,c1(OC)nc2ccc(C(N3CCCC3c3cccc(C)c3)=O)cc2[nH]1 54200,c1(OC)ccc(OC)c([N+](=O)[O-])c1C(N1CCC(NC(=O)C(O)CC2CC2)C1)=O 54201,c1(CC(=O)NC(c2cnn(C)c2)C(=O)NCC(CSC)(C)C)ccc(C)c(C)c1 54202,N1(C(C2CCN(CC)C2)=O)CCN(C(=O)COc2ccc(F)cc2F)CC1CF 54203,N1(C(c2c(CC)c[nH]n2)=O)CC(O)CC1(C)C(=O)NCC(C)C(C)(F)F 54204,N1(C(C(CCC)(C)C)=O)CC2CCN(C(c3c(F)cc(Cl)cc3Br)=O)CC2C1 54205,C(=O)(C(O)CCS(C)=O)NCC(C)CN(C(=O)CN1Cc2ccccc2C1)C 54206,c1(NC(C(C2CN(C(=O)CC(C)=C(C)C)C2)OCC)=O)ccc(CO)c(F)c1 54207,CC1(C)CCCOC1C(=O)NCCOCCCNC(=O)CSc1cccs1 54208,C1(C(=O)NOCCCN(Cl)Cl)CN(C(C2CCOC2)=O)CC1F 54209,c1(N2CCC(c3scc(CC)n3)CC2)ccc(S(=O)(=O)N2CCC2C(C)C)cn1 54210,c1(C(N2CC(CNC(C3N(C)CCC3)=O)C2)=O)cnc2c(c1)CNC(=O)N2 54211,c1(C(=O)NCCCN(C(C2CC23CCC3)=O)CC)scnc1C(F)F 54212,c1(COC)ccc(C(=O)NC(CNC(=O)CC2CC2(Cl)Cl)C2CC2)o1 54213,C1(CC(C)NC(c2cncc(F)c2)=O)CC2CCC(C1)N2C(C1CCCC1)=O 54214,N1(C(c2[nH]cc(OC)c(=O)c2)=O)CC2CCCC(C1)N(C(c1[nH]nnc1C)=O)C2 54215,c1(C2C(NS(C3(c4cn(CCN(CC)CC)nn4)CC3)(=O)=O)C2)cccc(F)c1 54216,O=C(C1=COCCO1)NCCC1COCCN1C(C1CC1C(F)(F)F)=O 54217,Cc1nonc1C(=O)NC1(C(=O)NC2CSC2)CCSC1 54218,N1(C(c2ccc(CNC(C(CCC)CC)=O)s2)=O)CCC(C)C(F)(F)C1 54219,C1(CC(=O)N(C(C)C(=O)OC(C)(C)C)C2CCCC2)COCC1O.N(C=O)C(C)C 54220,C(=O)(C1=C(Cl)CCCC1)N(C(C)CN(C)C(c1ccsc1-n1cnnn1)=O)C 54221,c1(CN2C(C(=O)NCc3c(C(N)=O)nccn3)C(O)CC2)nc2ccccc2[nH]1 54222,C1(CN(C(C2CC(N(CC)CC)C2)=O)C)CCCN(C(=O)CC2COCCO2)C1 54223,c1(N(C)C)ccc(F)c(C(=O)NC2CCN(C(=O)CCS(N)(=O)=O)CC2O)c1 54224,C1(C(=O)NCCC(C)NC(c2cnc(C(F)(F)F)s2)=O)CCCOC1C1CC1 54225,C1(C(N(C(CNC(Cc2ccc(CC)cc2)=O)C)C)=O)CC12CCS(=O)(=O)CC2 54226,c1(CCC)cc(C(=O)NCCC(C)(C)NC(C2CCC2(OC)OC)=O)n[nH]1 54227,C1(CC)CCCCC1C(=O)NC(COC)C(=O)NCc1cccc(CO)n1 54228,C#CC1(O)CC(C(=O)NCCCOCCC(=O)NC(C(N)=O)C2CCCC2)C1 54229,C1(C(N(CCCNC(=O)CCc2nccs2)CC)=O)CNC(=O)CC12CCOC2 54230,c1(C(C)NC(c2cccc(Br)c2)c2nccn2C)ccc(F)c(F)c1F 54231,Cc1cn2cc(C(N3CCC(F)C(NC(c4ccc(O)cc4F)=O)C3)=O)sc2n1 54232,CCC(C)(C(=O)NCC(CC)(CC)NC(C1CCN(C)C1)=O)C(N)=O 54233,N1(CC(=O)NCC(C2CCC2)NC(=O)CCc2ccccc2)CSCCSC1 54234,CCC(C)C(C(=O)N1CC(NC(C2C(C(C)N(C)C)C2)=O)C1)N(C)C 54235,C1(NC(C=CC=CCC)=O)C2CN(C(c3ccc(-c4ccc(F)cc4)[nH]3)=O)CC12 54236,CC1CN(C(=O)Cc2ccncc2OC(=O)C(C)(F)F)CC1Cc1ccccc1 54237,C#CC(CC)(CC)NC(C1CC(O)CN1C(=O)CC1CSCCO1)=O 54238,n1(CCOC)cc(C(=O)N(C2CCN(C(=O)C=Cc3cncs3)C2)C)nn1 54239,C#Cc1ccnc(C(N2CC3(C2)CN(C(=O)CC(F)(F)CC)C3)=O)c1 54240,S(=O)(=O)(c1ccc(C#N)cc1)NC(C1CNC(=O)C1)=O.CC12CN(C1)C2 54241,N1(C(c2c(N)cccc2F)=O)CCN(C(=O)CC2CC3(CCC3)CO2)CC(O)C1 54242,c1(C(=O)NCCC2CN(C(C(C3CCCOC3)OC)=O)C2)nonc1N 54243,C1(NC(=O)CC2CCC(F)(F)C2)CN(c2ccncc2[N+](=O)[O-])CCC12CCC2 54244,C1(CC)(CC)C(OC)CC1N(C)C(=O)NC1CC1c1ccc(C(C)(C)C)cc1 54245,C1(F)(C(=O)NC(C2CN(Cc3c(OC(C)C)cccc3)C2)C)CCC(F)(F)CC1 54246,C(=O)(N=c1ccn(CCCO)[nH]1)C1N(C(c2ccc(COC)cc2)=O)CC(C)C1 54247,C1(C(=O)NC2CCC(Cn3cc(Cn4cccn4)nn3)CC2)(CC)CCCCO1 54248,N1(C(c2cc(C)c(O)cc2)=O)C(C(N2CCC([N+](=O)[O-])CC2)=O)C2CC(O)C1C2 54249,C(=O)(CC(CNC(c1c[nH]cc1C(C)C)=O)C1CCC1)NC(COC)CO 54250,c1(OC)ccc(NC(=O)N(C)CCN(C)C(=O)C2CC2)cc1Br 54251,C(=O)(C1=CCC(C)(C)CC1)NCC(CNC(c1c(C)c(C(N)=O)ccc1)=O)O 54252,C1(CNC(=O)CC2CC2)CC12CCN(C(c1ncc[nH]c1=O)=O)CC2 54253,C(=O)(C1CCCc2ncnn21)N1CCC(C(C)NC(=O)CC2=CCCCC2)CC1 54254,c1(NC(N2CC(OC3CCCCC3CC(F)(F)F)C2)=O)ccc(F)nc1 54255,c1(NC(C(n2cc(-c3cc(C)ncc3)nn2)C)=O)coc(S(C)(=O)=O)c1 54256,C1(NC(CNC(C(CC)C)=O)=O)CCCCN(C(C2(C)CC2C)=O)C1 54257,Cc1cc(C(N2CC3C(CNC(C4CCC(=O)N4)=O)C3C2)=O)c2sc(=N)[nH]c2n1 54258,CCC(C)CN(C)N(CCCNC(C1CCCC1)=O)CC(=O)OC(C)(C)C 54259,N1(C(CCC=C)=O)CCC(NC(C2CC(=C(F)F)C2)=O)C(F)C1 54260,c1(CCOCC(=O)NCCCN(C(=O)CC2C=CCCC2)C(C)C)ccccc1 54261,Cc1cc(Cl)c(C(N2C3CCC2CC(NC(=O)C(C)O)C3)=O)cc1N 54262,C1(COC)CC(O)C(O)CC1C(=O)NC1(C)CCCO1 54263,CCC(CC(C)C)C(=O)N1CCCC(F)(CNC(c2cc(C)c(C)cn2)=O)C1 54264,C(C)(CN=c1[nH]c2c(c(=NCCCN=c3cc[nH]c4ccccc34)[nH]1)COC2)SC 54265,C(=O)(CCCCCO)NCCOC1(CNC(C2CC(C)OC2)=O)CCOCC1 54266,CCC(C)(C(=O)N1CCCC(COC)(NC(c2ccc(Cl)c(C)c2)=O)C1)C(N)=O 54267,C1(C(N2CCC(NC(c3ccnn3C3CCC3)=O)(CF)C2)=O)CN2CCC1CC2 54268,c1(OCC(CNc2cccc(C(CC)O)c2)O)cc(N)cc(Br)c1 54269,N1(C(C(C=CC)O)=O)CCCC2(CCCCC2NC(c2cc(C)c(C)cn2)=O)C1 54270,c1(COC(c2c(C)[nH]nc2CO)=O)cc(Br)ccc1Cl 54271,c1(C(N2CC(N(C(C(Cc3c(C)nc[nH]3)O)=O)C)C2)=O)cc([N+](=O)[O-])cn1C 54272,N1(C(CCCC(C)=O)=O)CC2(CC(C(=O)NCCc3nc(C)cs3)CO2)C1 54273,C1(NC(CN(C(CCOCCC)=O)C(C)C)=O)CCOC(CC)C1 54274,C1(C(N(C(CNC(C(CC(=O)OC)C)=O)C)C)=O)Cc2cccnc2C1 54275,c1(C(=O)OCC)nc(C)oc1OC.C12CC(C1)NC2=O.N12CCC1C2=O 54276,N1(C(=O)Cn2cccc2)CCC(C(N2CC3CC3C2)=O)C(O)C1 54277,c1(C(=O)NC(C(C)NC(C2(O)CCCCC2)=O)CO)ccc(Cl)c(C#N)c1 54278,CC(C(=O)N1CCCC(CNC(=O)CNC(N)=O)CC1)C(C)(F)F 54279,Cc1cc(C(=O)NCCCCNC(c2cncc(C(N)=O)c2)=O)sc1Br 54280,C1(C2CCC2)(C(=O)NC2C(NC(C3(C(F)F)CCCO3)=O)CCC2)CC1 54281,N1(C(C(C)OC)=O)CCCN(C(c2cc(C)n(C(C)(C)C)n2)=O)C(C)C1 54282,CC(C)C(CC(=O)NC12CC(NC(c3ccnc(S)c3)=O)(C1)C2)C(C)C 54283,C1(N(C)C(c2cnc[nH]2)=O)CCCN(C(C2NC(=O)OC2(C)C)=O)CC1 54284,O=C(CCN1C(=O)CSc2ccccc21)Nc1ccc(OCC(F)(F)N)cn1 54285,c1(C(=O)NC(CC)CNC(=O)C(C2CC(F)(F)C2)OC)nn(C(F)F)cc1Cl 54286,c1(C(=O)NC(C2CCCCC2)CNC(C(C=C)(C)O)=O)nccc(C)c1F 54287,C1(C(=O)NCC2(O)CC(CNC(c3cc(COC)sc3)=O)C2)CC(=O)N(OC)C1 54288,N1(C(C#CC)=O)CCc2cccc(C(=O)Nc3nccc(Cl)c3OC)c2C1 54289,c1(C(N2C(C(C)(C)C)C(NC(C3(C)CC3)=O)CC2)=O)csc2ccncc12 54290,c1(CC)ccc(C(N2CCN(C(=O)C3CC3)C3CC23)=O)cc1[N+](=O)[O-] 54291,c1(C(=O)NCC(CCNC(Cc2cn(C)nc2)=O)(C)C)c[nH]c2ncccc12 54292,C1(NC(CCC2C(C)C2)=O)CCN(C(c2ccc(NC=O)cc2)=O)C1(C)C 54293,N1(C(c2ccn(CC(F)F)n2)=O)CCN(C(c2cnc(O)o2)=O)C(C2CC2)C1 54294,c1(NC(COC)=O)cccc(NC(=O)NC(c2ccn(C)c2)C)c1 54295,c1(CC)cc(C(=O)NCC2CCC2NC(C2(Br)CC2(F)F)=O)n[nH]1 54296,CCCC(CC)CC(=O)NC1CCN(C(=O)C=CC(c2ccc(C)cc2)=O)C1 54297,C=C1CC(C(=O)N(C2CC(C)C2)C)(CNC(c2cc(Cl)cs2)=O)C1 54298,N1(C(=O)NC(c2n(C)ccc2)C2CC2)CC(O)CCCCCC1 54299,c1(NCCC(C)(C)SC)cc(C)c(S(=O)(=O)NC(c2ccncc2)CCO)cn1 54300,C#Cc1cccc(C(N2CCC(=C)CC2C(=O)OC)C(=O)NC2CCOC2)c1 54301,C1(CC(=O)NC2CONC2=O)OCC2CCN(C(=O)Cn3ccccc3=O)CC12 54302,CC(F)(F)C(F)C(=O)NCC1CN(C(=O)CSCC(F)F)CC12CC2 54303,c1(C(N2CCN(C(c3cc(C)nn3C)=O)CC(O)C2)=O)cc2cc(Cl)ccn2n1 54304,C#CCCC(O)C(=O)NC1CN(C(c2ncc(C(F)F)s2)=O)CC1O 54305,C(CCCCNC(c1c[nH]nc1-c1ccoc1)=O)N(C(C(F)OC)=O)C 54306,N1(C(c2occ(C)c2)=O)CC(NC(=O)CC2CCC(=O)NC2=O)C2CCCC12 54307,C1(C(N(C)CC2CCCN2)=O)CC(O)CN1C(c1ccsn1)=O 54308,C(C1CCCN1C(=O)CC1CC(OC)C1)=CC(=O)N(C)CC1CCN(CC)C1 54309,C(N=c1ccc(S(=O)(=O)NC2COc3cc(CO)ccc32)c[nH]1)C1C(C)C1 54310,C(c1ccc(F)cc1Cl)=CC(N1C(C(C)C)CN(C(c2ccn(C)n2)=O)CC1)=O 54311,C1(N(CCC(=O)N2CC(N3CCCCC3)C2)C)CC1C1CC1 54312,c1(CNC(C(=O)OCC)Cc2ccccc2)cccc(CS(C)=O)c1 54313,N1(C(CC(C)C)C(=O)NCCN2CCOCC2)CC(C)(C)OC2(CCCOC2)C1 54314,c1(C(N2CC3(CN(C(CC(=O)NCC#C)=O)C3)C2)=O)cc(S(N)(=O)=O)cs1 54315,N1(C(CCC(CC)C)=O)CCCN(C(c2cnc(CC3CC3)s2)=O)CCC1 54316,N1(C(c2cc(CCC)n(C)n2)=O)CCC(C)C(NC(c2ocnc2CCC)=O)C1 54317,c1(-c2cc(C)c(OC(C)C)nc2)ccc2[nH]c(C(N3CCCC3C(N)=O)=O)nc2c1 54318,C1(C(=O)NCc2cnsc2)(CNC(CC(C)n2ccnc2)=O)CCCCC1 54319,C(=O)(C(F)CC(C)(C)NC(c1ccns1)=O)NC1CCN(C)C1=O 54320,c1(CC(=O)N(C2CCN(C(=O)Cc3cccn3C)C2)CCC)ccc(Cl)c(F)c1 54321,c1(OCC)ccc(F)c(C(=O)NC2CCCC2CNC(=O)COCCN(C)C)c1 54322,CCC(CN(C)C)C(=O)N1CC(CC(=O)NC2CCC(=O)NC2)(OC)C1 54323,Cc1ccnc(C2(NC(=O)N(C(C)CS(C)=O)C)CCC2)n1 54324,CC1CCC(NC(c2cc(Cl)no2)=O)CN1C(=O)C(N1CCN(C)CC1)C 54325,[N-]=[N+]=NCCCOCC(=O)NC(C(=O)NCCC(O)C1CCC1)C1CCC1 54326,C(=O)(CCCCC(=O)N1CCN(C(c2cccc(OC)c2)=O)CC1C1CC1)NC 54327,CCCC(C)(O)CC(=O)N1CCCCC(NC(=O)Cc2nc(C(C)(C)C)cs2)C1 54328,N1(C(c2nnn(C)c2N)=O)CC2CCN(C(C3CCCOC3)=O)C2C1 54329,n1(CC(N2CC(N(C)C)C2)=O)cc(CNC(=O)C(O)C2CCCC2)nn1 54330,N1(C(N2CC(c3nc(C)on3)C2)=O)CCC2C(CCCN2C2CC2)C1 54331,n1(CC(=O)N(CCC2CN(C(C)=O)C2)C(C)C)cc(C)cn1 54332,c1(CC(N2C(CNC(C3CC(=C4CC4)C3)=O)CC2)=O)ccc(O)c(F)c1 54333,C1(C(=O)NC(CCOC)CO)CCN(C(=O)Cc2ncccc2F)CC1 54334,C1(N(C(=O)COCC2CCC2)CC#C)CCN(C(=O)Cc2csnn2)CC1 54335,C1(NC(CCCC=C)=O)CCN(C(C2CC3(CSC3)C2)=O)C(c2ccccc2)C1 54336,c1(C(Cc2nc(-c3cccc(CC)c3)nn2CC(F)(F)F)O)c(F)cccc1Cl 54337,C(CCCC(=O)NCC1C(C)CCN1C(=O)C1=CCOC1)N(C(C)C)C 54338,CC1CC2CC2CC1C(=O)NC1CCC(C)N(C(=O)CCC2CCCOC2)C1 54339,C1(N(C(CC(=O)NCC)=O)C)CS(=O)(=O)C12CCN(C(C1CCCCC1)=O)CC2 54340,N1(C(c2ccc(OC)o2)=O)CCN(C(=O)C(C)SC(C)C)C(c2cccnc2)C1 54341,C(=O)(C1=NOC2(CCC2)C1)NCC(CC)NC(=O)Cc1ccc(Cl)nc1F 54342,C(CCCCCCNC(C1(CC)CCC1)=O)n1cc(COC(C)C)nn1 54343,C1(C(N2CCC(CC(C)NC(C(C=C)O)=O)CC2)=O)Cc2ccccc2C1 54344,c1(CC)cc(N)ccc1C(=O)NCC1CCC(NC(c2cnoc2C2CC2)=O)C1 54345,C(=O)(C(F)CC(C)(C)NC(=O)CC(C)(C)CN(C)C)Nc1c(CC)noc1 54346,C1(c2ccc(C)cc2)CC1N=c1[nH]c(=NCCC(C)O)[nH]c2c1COC2 54347,c1(C(=O)NCC2N(C(CCC(C)OCC)=O)CCC2)ccc(S(N)(=O)=O)cn1 54348,C1(C(=O)NCC2CC(F)CN2C(C23CCC2C3)=O)CCN(C2CC2)CC1 54349,N1(C(COC(CC)C)=O)CCCCC(C2CN(C(c3cnc(OC)nc3)=O)C2)C1 54350,Cc1n[nH]c2cc(C(=O)NC3CCCC3NC(c3ncccc3F)=O)ncc12 54351,c1(NC2CC(NC(c3ccc(F)c4occc34)=O)C2)c(Cl)cncc1[N+](=O)[O-] 54352,CC1CCN(CCOC(C2(c3ccccc3)CC3(CC3)C2)=O)CC1 54353,c1(N(C)NCc2cc(C)on2)nc2c(c(=NCc3ncn(C4CC4)n3)[nH]1)CCC2 54354,Cc1cc(C(N2CCN(C(C3CCCCC3O)=O)CC2C)=O)ncc1C#N 54355,C1(C(=O)NC(CC(C)C)c2ccccc2)(CF)CCN(C(=O)OC(C)(C)C)CC1 54356,C1(OC)CN(C(=O)C(O)CNC(C2CC2C(N)=O)=O)CC12CC2 54357,C(=O)(C1CNc2ccccc21)NCCCCC(C)NC(C(C)OCC1CC1)=O 54358,N1(C(=O)Nc2cc(C(N)=O)cc(Br)c2F)CCc2c(F)cccc2C1 54359,N1(C(COC)=O)CCC2(CCC(C(=O)NCC3(N4CCOCC4)CCCC3)C2)C1 54360,N1(C(C2C(C)CCC2)=O)CCCC(CCNC(=O)COCC2CCOCC2)C1 54361,c1(CC(N2C3CC(NC(c4cncc(C)n4)=O)C(C3)C2)=O)cc(F)c(C)cc1F 54362,c1(NC)ncccc1C(N1CC(NC(=O)Cc2ccsc2Cl)C(C)C1)=O 54363,C#CC1(C(=O)Nc2ccc(OC)nc2C)CCN(C(=O)C2=C(C)CC2)C1 54364,C1(Nc2cccn2CC)CC(NC(C2CCCC(C(=O)OCC)C2)=O)C12CCC2 54365,N1(C(C2C(C)C2C2CC2)=O)CC2CC3CC2C1C3NC(C1COCCO1)=O 54366,n1(C(C)C)ncc(C(=O)NCC(C2CC2)NC(C2(O)CC2)=O)n1 54367,c1(C(N2CC3C(NC(CN(C)CC)=O)CC(C3)C2)=O)cn2cc(C)ccc2n1 54368,c1(C(=O)OC)cc2c(s1)CCC2NC(c1cncc(N)n1)=O 54369,CC1CN(C(=O)CCOCCNC(=O)CC#N)CC1CO 54370,C(C(C(=O)NCC12CCC(CC1)CC2)C(C)C)NC(C(C(C)C)OC)=O 54371,N1(C(CCC2CNC(=O)N2)=O)CC2CCC(C1)N2C(=O)C(F)OC(F)(F)F 54372,c1(C(=O)NCC(CNC(c2cccs2)=O)OC)cc2ccc(F)cc2o1 54373,c1(OC)ccc2[nH]c(C(=O)NCC3CCN(C(=O)CC(C)C)CC3C)c(C)c2c1 54374,N1(C(Cc2n(C)ncc2Br)=O)CC(NC(c2cc3sccc3[nH]2)=O)CC(F)C1 54375,C1(NC(CCN(C(CCCOCCOC)=O)CC2CC2)=O)CCCN(C)C1C 54376,CC(C)CC(C(=O)NC(CC(C)(C)C)C(=O)N(C)Cc1ccnn1C)C(C)C 54377,C1(C(N(CCCNC(=O)Cn2cnnn2)CCC)=O)CC(=O)N(CCOCC)C1 54378,c1nc(CC(C(=O)OC)NC(C23CC(C(=O)OC(C)=O)(C2)C3)=O)n[nH]1.CC(C)C 54379,C1(NC(=O)C(c2ccccc2)Sc2ccc(F)cc2)CCc2ncnn2C1 54380,CN1C(=O)CCC1C(N1CC(O)CC1C(=O)NCCN1CCCC(O)C1)=O 54381,C1(NC(=O)C2CC2)CC2(CCN(C(C34CC(CO3)C4)=O)CC2)C1 54382,C1(C(=O)NC(C)CC(C)NC(=O)C(C)Oc2cccnc2)CCN(C(N)=O)CC1 54383,c1(C(N2CCCC(C(=O)NCC=Cc3ccccc3)C2)=O)ccc2cncn2c1 54384,C1(O)(CNC(C(CC)(C)C)=O)CCCN(C(=O)CC2CCCC(C)(C)O2)CC1 54385,O=C(CCCC(F)(F)F)NC1CN(C(C2(CO)CC2(F)F)=O)CC12CC2 54386,C(C1=CCCN(C)C1)NC(C(C(C)NC(c1cnc(N)cn1)=O)C)=O 54387,C1(N(C(Cc2nc(C(C)C)sc2)=O)C)CCN(C(c2csc(=N)[nH]2)=O)CC12CC2 54388,N1(C(COCCCCC)=O)CCN(C(C2CCCN2CC(C)C)=O)C(C2CC2)C1 54389,CC1CC(C)N(C(c2nn3c(c2Br)CCC3)=O)CCN1C(c1cccnn1)=O 54390,c1(N(C2C(OC)COCC2)C)ncnc2c([N+](=O)[O-])cccc12 54391,C1(c2nnnn2CC(F)F)(NCCOC(CC)(C)C)CCC(CCOC)C1 54392,c1(C(CO)NC(C2(NC(COCC(=O)OC)=O)CC2)=O)cccnc1 54393,C(c1cn(C)nn1)=CC(=O)NC1(CNC(C2C(C)C2)=O)CC1 54394,C=C(C)C1CCC(C)CC1NC(Cc1ccc(F)cc1)C(C)(C)C 54395,C(=O)(C1=CC(c2ccc(F)cc2)=NS(=O)(=O)N1)N(CC(=O)OC)C 54396,C1(O)(CNC(C2CCC2)=O)CCN(Cc2cccc(-c3ccccc3)n2)CC1 54397,C=C=CCCC(=O)NC(C1CCN(C(c2cc(C)cs2)=O)C1)C 54398,N1(C(COCC(=O)OC)=O)CCCC(C2CCCCN2C(=O)C(O)CSC)C1 54399,n1(CC)cc(C(=O)NCC2(CCNC(=O)CC3CC34CC4)CC2)nn1 54400,Cc1ccc2c(C(=O)NCC(C)CNC(=O)CCc3ccc(F)nc3)coc2c1 54401,c1(C(N2C(CNC(=O)C3=CC(C)(C)C3)CCC(C)C2)=O)ccc2c(c1)CCC2 54402,Cc1cc(C(=O)NC2CC3(C2)CC3NC(=O)Cc2ccc(Cl)cn2)cn(C)c1=O 54403,C(=O)(C(C)(F)C(C)(C)F)N1CC(CN(C)C(c2cn3cnnc3cn2)=O)OCC1 54404,n1(CC)cc(Cl)c(C(=O)NCC2CCCN2C(c2sc(C)cc2C)=O)n1 54405,c1(C(N(C2(C3CCCN3C(=O)C3=CCC3)CC2)C)=O)cc2ccccc2o1 54406,C(=O)(C(CC1CCCC1)NC(=O)C=CCN1CCC1)NCCCCSC 54407,C(=O)(CCCCC(=O)NC)NC12CCN(C(C(=O)NCCOC)=O)CC1C2 54408,CC(C)CC(C(=O)N1CCOCC1C1CCC1)Nc1c[nH]c(Br)c1 54409,C1(NC(c2nnnn2C2CC2)C2CC(CC)C2)Cc2ccc(Br)cc2C1 54410,N1(C(C2CC(CC)C2)=O)CCC2OCCN(C(c3ccn4cncc4c3)=O)C2C1 54411,CC1CC(C(N2CCCC2CNC(c2cccc(C3CC3)n2)=O)=O)CC(C)C1 54412,c1(C(=O)OC)c(C)cc(C)nc1NC(C)CC(C)NC(=O)CC(C)CC(C)C 54413,C1(C(=O)NCCOCC#C)CN(C(c2ncc(C(F)(F)F)s2)=O)CCC1O 54414,C(c1cncc(F)c1)=CC(=O)NC1C(CNC(=O)CCCF)CCCC1 54415,CC(C)C(C)(CNC(c1cnc(S)n1C)=O)NC(=O)C(c1ccc(Cl)s1)C 54416,c1(CCC(=O)NCC(C)(C2CCC2)NC(C(C)OCCCC)=O)c(C)n[nH]c1C 54417,c1(C(=O)NCC(CC(=O)NCCN(CC(C)C)CC)O)cnn(C)c1C#N 54418,C(CC(C)C)(C(=O)NC1CC2(C1)CC2NC(=O)CC1(CS(C)(=O)=O)CC1)OC 54419,C1(C(N2CC(CNC(c3ncccc3F)=O)C3(C2)CC3)=O)CC2(C1)CC(F)(F)C2 54420,N1(C(C(C)SCCCC)=O)CCC(CNC(=O)C(CO)OC)C1C 54421,N1(c2nc(C)c(=O)n(C)n2)CCCC2(CCCO2)CC1 54422,C(CN=C(NCc1ncc(C)s1)N1CCC2(CCCOC2)C1)N(C(=O)OC)C 54423,C(C1=CCN(C2CCC2)CC1)Oc1cncc(NC(C=CC(C)(C)SC)=O)c1 54424,C(=O)(C1CCCc2nn[nH]c21)NCC=CCNC(CC(n1c(C)cc(C)n1)C)=O 54425,C1(C(N(CC(=O)OCC)C)=O)CC2CC2N1C(=O)CCc1nc(=N)[nH][nH]1 54426,Cc1nn(C)cc1C1CC1C(=O)NCCCNC(C1CC2CCC1O2)=O 54427,c1(C(c2nnnn2CC(F)F)NC(c2c(C)n(C)nc2)C)nn(C)c2c1CCC2 54428,C(C(C)C)(C(O)C(=O)NCC1CCOC1C(=O)N(C)Cc1ncco1)OC 54429,C1(C)(C(N(CCCC(=O)NCC(CC)(C)Cl)C)=O)CC(F)(F)C1 54430,C(=O)(C1=CC2CCC(C1)C2)N1CCCC(NC(c2c(COC)nn[nH]2)=O)(CO)C1 54431,C1(C)(CNC(C(C)NC(c2cc[nH]c2)=O)=O)CCCC1 54432,Cc1ncccc1C(=O)N(CCCNC(C12CC(O)C1C2)=O)C 54433,N1(C(C(COC)O)=O)CC(NC(c2ccc(F)s2)=O)C2CCCCC12 54434,CC1=C(CNC(=O)C(c2ccns2)NC(=O)OC(C)(C)C)S(=O)(=O)CCO1 54435,S(=O)(=O)(c1c(Cl)cc(Br)cc1Cl)N1CC(C)(C(=O)Nc2cc(Cl)cc(Cl)c2F)C1 54436,C1(C(NOC(C(=O)OC)C)=O)CC(C)(NC(=O)C(=O)N(C)C)C1 54437,N1(C(C2C(CCOC)C2)=O)CC23CCCC2(C1)CN(C(C1CCC(OC)C1)=O)C3 54438,C1(C(=O)OC)CCN(S(=O)(=O)N2CCSC(C)C2)CC1 54439,c1(C(=O)NCC2N(C(C(C(=O)OC)C)=O)CC(C)(C)C2)cccc2c1cnn2C 54440,C1(C)(C(N(CC(=O)NCC(c2ccccc2)O)C)=O)CC(C#N)C1 54441,c1(NC(C(=O)NC(CC=C)CO)=O)ccc(OC(F)(F)F)c(Cl)c1 54442,C(=O)(CC(F)(F)CNC(=O)OC(C)(C)C)NCc1c(OC)nccc1 54443,C(=O)(C(C)(C)C(N)=O)N1CCC(CCNC(c2c(N(C)C)cncc2)=O)C1 54444,CCC(C)C(C)C(=O)NCCN(C)C(c1cnn(-c2cccc(Cl)c2)c1N)=O 54445,N1(C(C(C)SCC)=O)CCC2CN(C(=O)C=Cc3cnccn3)CCC12 54446,c1(C(=O)OC)cccc(C(=O)NCC(C)(C)CNC(=O)CCF)c1C 54447,c1(C(=O)NCCCN(C(C2CN(C(=O)NC)C2)=O)C2CC2)ccc(C)c(F)n1 54448,CCC(C)(C)CCCC(=O)N(C1(C(=O)NCCOCCC2CC2)CC(O)C1)C 54449,C1(CN2CCC(NC(c3c(CC)nn(C)c3)=O)C2)CCC(F)(F)CC1 54450,c1(C(c2nnnn2C(C)(C)CC)NCC(COCC)C)c(C)cc(Br)cc1C 54451,CCC(CNC(=O)CN1CCCS1(=O)=O)(CC)NC(C1C=CCCC1)=O 54452,CC(CNC(c1ccccc1O)=O)C(F)C(=O)NCc1c(F)cncc1F 54453,N1(C(C(C)=C2CC2)=O)CC2CCC(CNC(c3n[nH]c4c3NCCC4)=O)(C2)C1 54454,CS(=O)(=O)CCC(=O)NC1CCN(C(c2csc(-c3cccnc3)n2)=O)C12CC2 54455,[nH]1cccc([N+](=O)[O-])c1=O.C(=O)(C(C)(C)CCCF)N1CCC(C)C1c1c[nH]nn1 54456,CCCCCC(F)C(=O)NCCCN(C)C(C12CC(C)(C1)OC2(C)C)=O 54457,CC1(C)CC(CC(=O)NC2COCCC2NC(=O)CC2CC3(CC3)C2)CO1 54458,C1(CC)CCC(C)CN1C(C1CC2(CCC2O)C1)=O.C1=CC(=O)NC(C)(C)C1 54459,Cc1coc2ccc(C(=O)N(CC(C)NC(c3cc(Cl)cc(F)c3F)=O)C)cc12 54460,c1(CC)nnc(N(C2CCCC(C)C2)C)n1CCn1cc(Br)cn1 54461,N1(C(C2(F)CCN(C(c3cc(C)ncc3C)=O)CC2)=O)CCCC2C(O)CC12 54462,Cc1[nH]c2ncccc2c1C(=O)NCC1CN(C(=O)CCC2CCOC2)CCO1 54463,C1(CCOC)(NC(=O)C(C)Cc2cnco2)CCN(C(=O)CSS(C)(=O)=O)CC1 54464,C1(C(=O)N(CC(C)C)C)(CC)CCN(C(=O)CCC2CCOCC2)C1 54465,c1(C(N2CC(F)CC(NC(C(C)c3ccco3)=O)C2)=O)c(N)c(F)cc(F)c1F 54466,C(C(C)C)(C(O)C(=O)NC1CC(N(C(=O)CCc2cc(C)no2)C)C1)OC 54467,N1(C(c2ccn(CC)c2C)=O)CC(N(C(=O)CP(C)(C)=O)C)C2(CC2)C1 54468,C1(C)(C(N(CC=C)CCOC)=O)CN(C(C2CCC(C(N)=O)C2)=O)CC1C 54469,n1(CCC)nnnc1C(c1cc(C)[nH]n1)NCCc1cnoc1 54470,CC(CNC(=O)COCC1CC1)C(=O)NC(CO)CCC1CC1 54471,C1(C(=O)NCC(C)SC)C2CCC(C2)C1NC(C1(O)CC1)=O 54472,CCC(CC(=O)N1CC(=C(F)CNC(=O)CSC(F)(F)F)C1)C(F)F 54473,CCCC(CC)C(=O)N1CC2CC2(NC(c2cc(C(C)(C)C)c[nH]2)=O)C1 54474,C1(NC(CCSC)=O)CCN(C(c2ccc(CF)cc2)=O)CC1C 54475,C(=O)(C(CCCC(C)(F)F)N1CCC2C(CCCN2C(C)=O)C1)NCCOC 54476,C(=O)(CN=c1cc[nH]cc1)N1C(C(=O)NCC2N(C(C)=O)CCC2)CCCC1 54477,C(=O)(C(C)C(=O)NC(C)C(=O)Nc1cncnc1O)OC 54478,C(=O)(C1CNC(=O)c2ccccc21)N1C(CNC(C2(CC)COC2)=O)CCC1 54479,C(=O)(CCCCCS(N)(=O)=O)NC1C(NC(c2ccnc(OC)n2)=O)CCC1 54480,C1(CNC(c2n(COC)ncc2)=O)CN(C(c2csc(CO)n2)=O)C2CCN1C2 54481,c1(C(=O)NC(C(C)NC(c2ncc(OCC)nc2)=O)C(C)C)cc(C)cc(O)c1 54482,CC(CCCCCO)N=c1[nH]c(=NCCN2CCC2)c2ccccc2[nH]1 54483,c1(C(N2CC(c3c(CNC(C(CC)F)=O)nco3)C2)=O)cc2cscc2s1 54484,Cc1c(N)c(C(=O)N(CC(C)CNC(c2ccc(C(F)F)c(F)c2)=O)C)nn1C 54485,C(CCCCCF)NC(C1CC(NC(=O)CC2CCC2)C1)=O 54486,c1(C(C)C)ncc(Cl)c(C(=O)NCC2CCN(C(C3CCC3C(F)F)=O)CC2)n1 54487,N1(c2ncc(C(=O)OCC)nc2)CCC(CNC(c2csc(NC)n2)=O)C(C)C1 54488,C1(NC(=O)CCC2CCCCN2C(C2CCC3CC2CO3)=O)CCCCCC1F 54489,CC1=C(C(=O)NCC(C2CCCN2C(=O)CSCCC(C)C)F)CCC1 54490,C1(C(=O)NC2CC(C(=O)NC(CCCCC)C)CC2O)CC(=O)CC(=O)N1 54491,C1(F)(CS(C(=O)NCCSCc2ccc(C(F)(F)F)cc2)(=O)=O)CCCCCC1 54492,CC1CCN(c2ncc(C(=O)NC3CCCN(C(=O)C(CO)N(C)C)C3)s2)CC1 54493,C(=O)(C(C)(C)C(=O)N1CCC(F)(C(=O)NC(C)CN(C)C2CC2)CC1)OC 54494,Cc1cc(C(=O)N(C2C3CN(C(C4CN(C)CCO4)=O)CC23)C)c(Cl)cc1F 54495,CC1Cc2ccccc2C1NC(=O)C(C(C)(C)C)NC(C1CN(C(=O)NC)C1)=O 54496,c1(C(=O)NC2N(C(C(C)Oc3ccc(C)cc3)=O)CC3CC32)cc(C#N)cn1C 54497,C1(C(N2CCN(C)C(=O)C2)=O)CC(C)(C)CCN1C(C1CN2CCC1CC2)=O 54498,N1(C(CNC(CC)=O)=O)CCC=CC1C(=O)NCC1CC(F)(F)CO1 54499,N1(C(C2CCC(N(C)C)CC2)=O)CC2(CCN(C(c3cn(C)c(=O)cn3)=O)C2)C1 54500,C1(NC(COCCOCC#C)=O)(CF)CCN(C(c2c(C)ncn2C)=O)C1 54501,c1(C(=O)NCC(CNC(=O)CCc2ncco2)OC)cnc[nH]c1=N 54502,N1(C(c2c(CC)cc(Cl)cc2)=O)CCC12CCCN(C(=O)C(C)OC)C2 54503,C1(NC(CN(S(CC)(=O)=O)C)=O)C2CCN(C(c3cc(F)c[nH]3)=O)C12 54504,c1(-n2c(C(=O)NC(COC)(C)C(=O)NCCn3cncn3)cnn2)cc(Cl)ccc1Cl 54505,CCC(C)C(O)CNC(=O)COC1CC(NC(C2(CC)CCCCO2)=O)C1 54506,N1(C(C2(SC)CC2)=O)CCOC(CCNC(N2CC(OCC)C2)=O)C1 54507,CC(C)CC(CC(C)C)C(=O)NCC1CC(CNC(=O)Cc2cn(C)nn2)C1 54508,c1(C(=O)NC2CN(C(c3c(CC)cno3)=O)C(C)C2)sc2[nH]cnc(=S)c2c1C 54509,CC1(C(=O)NCCCC2CCCN2C(c2cnc[nH]2)=O)CCCC1(F)F 54510,C1(C(C)C)(C(=O)NCCCCN(C)C(c2coc(CC3CC3)n2)=O)CCCO1 54511,c1(CC)onc(C)c1C(N1CCCC(NC(C2CCCN2C(=O)C(C)C)=O)C1)=O 54512,C1(CC(=O)NC(C)C(C)NC(c2ccccn2)=O)CCCCC12CC2 54513,C1(C(NNc2cc(C)nc(C)n2)=O)CCN(S(=O)(=O)N2CCNCC2C)CC1 54514,Cc1[nH]nc2c1CC(C(N1CCCC(F)(CNC(=O)C(C)(C)C(F)F)C1)=O)CC2 54515,N1(C(CC(=O)NCC#C)=O)CC=C(C(=O)NC2CCOC2C(=C)C)CC1 54516,c1(C(=O)NCC(O)CCNC(C2CN(C3CCOC3)C2)=O)cccc2[nH]ccc12 54517,c1(C(N2CC3C(NC(CCCCSC)=O)(CCC3)C2)=O)cccc(S(N)(=O)=O)c1 54518,N1(C(C2CCCN(C3CC3)C2)=O)CC(C2CCN(C(C3CC(N(C)C)C3)=O)CC2)C1 54519,c1(OC)csc(C(=O)NC2CCC(CNC(=O)CCCc3cccnc3)C2)c1 54520,CC#CCCCC(=O)NC(CNC(c1nnsc1C(F)F)=O)CC(C)C 54521,c1(C(=O)NCCCC2CCCN2C(C2CCC(F)(F)C2)=O)cccn2nncc12 54522,N1(C(C2CCC(C)(C)C2)=O)CCc2[nH]nc(CNC(C3CCOC3)=O)c2C1 54523,CC1CCc2onc(C(=O)NC3CC4C3CCN4C(c3cn[nH]c3)=O)c2C1 54524,c1(OC)cc(OC)nc(NC(CC2N(C(C3CCN(C)C(=O)C3)=O)CC2)=O)n1 54525,c1(CC(=O)NCCC2CCN(C(CCCc3onc(C)n3)=O)C2)cccc(F)c1 54526,N1(C(C)=O)CCOC(C(=O)NC2CCC(N(C(=O)C=CBr)C)CC2)C1 54527,Cc1nn(C)c2c(N(CCCn3ccnc3C)C)nc(=NC3CCCOC3)[nH]c12 54528,c1(OC)cncc(C(N2CC(CCNC(=O)C(=O)N(C)C)C(C)C2)=O)n1 54529,C(=O)(CC(C=C)CCC)N1CCC(N(C(=O)C(C)(C(C)C)OC)CC#C)CC1 54530,C1(C(N2CCN(c3ccccc3O)CC2)=O)CN(Cc2ncc[nH]2)CC(F)(F)C1 54531,C1(CC(N)=O)CCCN(C(=NCCC2CCOC2)NCC(CO)C(F)(F)F)C1 54532,c1(C(N2CCCCC2CC=C)C(=O)NCC=C)ccccc1Br 54533,N1(C(=O)CCc2ccccn2)CCCC(CO)(NC(C2CC3C=CC2O3)=O)C1 54534,c1(C(=O)NCC(CC(C)C)NC(=O)CC2CN(C)C2)ccnc(C(F)(F)F)c1N 54535,Cc1[nH]c(C)c(C(=O)NCC(C2CCC2)NC(=O)CCCOC(C)C)c1C 54536,N1(C(C(CCCC)F)=O)CCC2(CC(C(=O)N(C3CC(C(N)=O)C3)C)C2)C1 54537,N1(C(C(C=C)O)=O)CCCN(CCNC(=O)C(C)c2cncs2)CC1 54538,C1(NC(c2nc(C)sc2)=O)CCCN(C(=O)COC2CCCC(C)C2)C1C 54539,CCCC(CCC)CC(=O)NC1CC2CC1N(C(c1ccc(F)c(C)c1)=O)C2 54540,C1(C(=O)NCCN(C(C(CCCC)O)=O)C(C)C)Cc2nccnc2C1 54541,c1(C(=O)NC2C(C)CN(C(c3cc4scnc4[nH]3)=O)C2)cnc2ccncc2c1 54542,c1(N2CCC(=CC)C2)cc(C)c(S(=O)(=O)N2CCOC(c3ccccc3)C2)cn1 54543,C1(CNC(COCCOC)=O)(NC(=O)C(C)CO)Cc2ccccc2C1 54544,CC(C)CC(CNC(=O)CC1CC2(CCC2)C1)NC(=O)CCc1cccc(Cl)c1 54545,N1(C(C2CC(C)(C)C2)=O)CCN(C(C2CCC(C(F)(F)F)CC2)=O)CC(O)C1 54546,N1(CC)C(=O)NC(c2ccc3nc(C4CC4)oc3c2)C(C(=O)OCC)=C1COC 54547,Cc1cccc(CCC(=O)NCC=CCNC(C2CCCN(C)C2)=O)c1 54548,N1(C(c2cn(CC=C)nc2)=O)CCC(N(C(=O)C(N2CCCCC2)C)C)C(C)C1 54549,N1(Cc2ccc(COC(C)=O)o2)CC(C(=O)O)C2(CN(C(=O)CS(C)(=O)=O)C2)C1 54550,CC(C)C(CNC(C1CNC(=O)C1)=O)C(=O)NC1CCCCCC1CO 54551,c1(C(=O)NC2C(NC(C3C(OC)C3)=O)CCC2)csc2ccc(Br)cc12 54552,c1(C(c2nnnn2CCCSCC)NCCC(CC)C)nc(C)[nH]c1Br 54553,Cc1cc(C(=O)NCCOC2CCN(C(=O)CC(C)C)C2)c(C)n1C1CCOC1 54554,n1(C(C)C)ncc2c1CC(NC(=O)NC1CCCC1C(N)=O)CC2 54555,c1(OC)cc(OC)nc(C(=O)NC2CC3CC(NC(=O)C=C4CCC4)CC23)n1 54556,C1COC(CNC(=O)CCNC(C2CC2)=O)C1.O=C(COC)NC1CCC1 54557,N1(C(c2n[nH]c(CC)c2C)=O)CC(C)C(NC(=O)CNS(=O)(=O)CC)C(C)C1 54558,c1(CNC(C2(CC=C)CCCN2C(=O)CN2CCCC2)=O)cc(C)ccc1C 54559,c1(C(=O)NC2CN(C(c3n(C=C)ncc3)=O)CC(F)C2)cccc(F)c1NC 54560,CCC(C)C(O)C(C)C(=O)N1CC(OC)CC1C(=O)NCc1ccc(F)c(Cl)c1 54561,C1(C(N(CC)CC2CCC2)=O)CCCN(C(=O)C(CN(C)C)C(C)C)CC1 54562,C(CCC)(C(=O)N1CCCC1C(N1CCCC1CCCC)=O)=CCC 54563,c1(CNC(C2C(=C)C2)=O)nc(CNC(C2COCCN2C)=O)cc(O)n1 54564,C1(CCC(=O)NC2CN(C(C(N)=O)=O)C2)CCC(=O)NC1 54565,c1(Nc2cncc(-c3ccc(C)cn3)c2)cc(N2CCCC2)nc(C)n1 54566,c1(C(N2CC(N(C(c3c(CCC)nco3)=O)C)C(F)C2)=O)ccc(O)c(C)c1C 54567,c1(N2CC(SCCCCCC)C2)ncnc2c1ncn2CC(CC)(CC)C(C)O 54568,C#CCC(C(=O)NCc1nn(C)cc1Cl)NC(=O)CCCCN(C)C 54569,Cc1nc2ccccn2c1C(=O)NC(C)CNC(c1nc[nH]c1C(F)(F)F)=O 54570,c1(C(=O)Nc2ccc(NC(C(COCC)C)=O)c(C)c2)c(C)[nH]c2ccccc12 54571,c1(C(N(C)CC2(O)CCN(C(C3CC(O)C3)=O)C2)=O)ccc(Cl)c2cccnc12 54572,N1(C(c2cnc(SC)s2)=O)CC(NC(=O)CC2CC(C)(C)CO2)C2(CCCC2)C1 54573,c1(C(=O)NCC(C2CCOC2)NC(c2cnccn2)=O)ccn2ccccc12 54574,C1(C(=O)NC(CC)CNC(C2(CC)CCC(O)CC2)=O)CCC2C(C1)C2(F)F 54575,C1(n2cc(C(c3ccncc3)C)nn2)CCCN(C(=O)Nc2cncc(Cl)c2)C1 54576,CCC(CC)CC(F)C(=O)NC1C2CC3C1C3C2C(N1CC2(CCC(O)CC2)C1)=O 54577,C(C(C)CC(=O)NC1COCCC1NC(c1snc(Cl)c1Cl)=O)OC 54578,C1(C(N2C(COC)(CNC(=O)C(C)=C3CCCC3)CCC2)=O)CNC(=O)CC1C 54579,N1(C(Cc2ccc(C)c(C)c2)=O)CCC2CN(C(=O)CC(C)(C)O)CC2C1 54580,N1(C(CC(C=C)C)=O)C2CCC1CC(O)(CNC(=O)CC1=CCCC1)C2 54581,c1(C(N(CCCNC(C2(C)CC2Br)=O)CC)=O)c[nH]cc1COC 54582,C1(C(F)(F)F)(C(N2CC(N(C(CSCCC)=O)C)C2)=O)CCOCC1 54583,c1(CC(=O)NCC(C)(C)NC(C2CCC(C(=O)OC)C2)=O)cc(F)ccc1OC 54584,CC1(C)CN(C(=O)C(c2ccns2)NC(=O)OC(C)(C)C)Cc2ccccc21 54585,c1(OCCC#C)ccc(CNC(C2CCNCC2C)=O)cc1 54586,C1(C(=O)NCCN(C(C)C)CC)CC(C)CCN1C(c1cnc(C)c(C)c1)=O 54587,Cc1ccc(S(=O)(=O)NCC(N2CC3(C2)CN(C(C2CNC(=O)N2)=O)C3)=O)cc1 54588,C1(COC)CN(C(C2CCN(C)S2(=O)=O)=O)CCN1C(c1ccc(O)nc1C)=O 54589,C1(c2nnnn2Cc2nnc(COCC)s2)(OC)CCC1C1CCC1 54590,C12(C(N3CC(C)C(NC(c4cnn[nH]4)=O)C3)=O)CCC(C1)C2(C)C 54591,c1(OC)cc(CC(N2CCC(CN(C)C(C3C(C)CC3C)=O)CC2)=O)ccn1 54592,C1(NC(c2cc(C)ncn2)=O)CC(C2CCN(C(c3cccc(C#N)c3)=O)C2)C1 54593,C1(NC(=O)COCCOCCO)COCCN(C(=O)Cn2cccn2)C1 54594,C12(C(N3CC(CNC(Cc4cncc(OCC)c4)=O)C3)=O)CCCN(CC1)C2 54595,C1(NC(CCOCC)=O)CC2C1CCN2C(c1ccc(C(C)(C)C)c(Cl)c1)=O 54596,N1(C(c2c(CC)cc[nH]2)=O)C(C(=O)NC(c2snnc2C)C)CCC1C1CC1 54597,CON=CC(=O)NCCCCCNC(c1nnsc1N)=O 54598,C1(C(N2CC(OC)C(NC(=O)CCc3cscn3)CC2)=O)CC1C1CC(F)(F)C1 54599,c1(C(=O)NCC2(C)CCCN2Cc2cccs2)c(Cl)cc(Cl)cc1Cl 54600,C1(C(=O)NC(CCCOC)C)(NC(c2ccc(CC3CC3)cc2)=O)CCCCC1 54601,N1(C(c2cc(C3CC3)on2)C)CCC(C(C)C(=O)NC2CCOC2)CC1 54602,CC1(C)CC(=O)NC1CNC(C1OCCC1NC(=O)CN1CCCCC1=O)=O 54603,c1(C(=O)NC2CC2NC(C2(c3ccccc3)CC2(F)F)=O)cc2cccn2cn1 54604,C(C(CO)CC(C)C)NC(C1(C)N(C(c2cc(C)sc2N)=O)CCC1)=O 54605,Cc1nc(NC(C)(CNC(C2(C(F)F)CCCO2)=O)C2CC2)cc2nncn12 54606,C1(CNC(=O)CCc2cccs2)CCCN(C(=O)CC2CCC(F)(F)CO2)CC1 54607,c1(OCC(N2C(CNC(COC(C)(C)C)=O)CC2)=O)ccc(Br)cn1 54608,c1(C(=O)NCC(CN(C(=O)CC2COC(=O)N2)C)(C)C)cn2ccccc2n1 54609,N1(C(c2nn(CC)c(O)c2)=O)CC(NC(=O)CNC(c2ccsc2)=O)CCC1C 54610,Cc1cc[nH]c1C(=O)NCCCCc1cn(C2CCCC2N)nn1 54611,c1(CC)ccc(C(N2CCC(CNC(c3coc(Br)c3)=O)C(C)C2)=O)cc1N 54612,Cc1nc(C(=O)NC(C2CN(C(=O)C(C(C)C)NC(N)=O)C2)C)[nH]c1C 54613,S(=O)(=O)(c1cccc(=NCC2SCCS2)[nH]1)NC1C(OC)C2(C1)CCC2 54614,C1(C)(CC)CC(NC(c2c(OC)cccc2O)=O)CN1C(c1cnc(S)nc1)=O 54615,N1(C(C(C)(C)C2CCC2)=O)CCCC(C2CCN(C(C3(F)CC=CC3)=O)C2)C1 54616,C12(NC(c3cc4occc4s3)=O)CCCN(C(=O)Cc3ccoc3)CC1C2 54617,c1(NC(C2CC(NCc3cnc(OC)s3)C2)=O)cnc2sccc2c1 54618,CC1COC2(CCC2)CN1C(=O)CSCCNC(=O)C(O)Cn1cncn1 54619,c1(SCC)cc(NC(=O)NCCOc2ccc(Cl)cc2Cl)ccc1OC 54620,C(=O)(C1=COCCO1)N1CCC(C)(NC(c2nncc(C)c2)=O)C1 54621,C1(C2CC2)(C(=O)NCc2cc(C(=O)NC(C)CC3CCC3)n[nH]2)CC(=O)C1 54622,c1(NC(C2CCCN2C(=O)CN2C(=O)CCCC2=O)=O)ncc(I)nc1Cl 54623,CS(=O)(=O)CCC(=O)NCC1(O)CCCN(C(=O)CC2CCCS2(=O)=O)C1 54624,N#CC1(NC(c2cccc(F)n2)=O)CCN(C(c2ccc(Cl)nc2Cl)=O)C1 54625,c1(C(=O)NC(C(=O)NCCCCN(CC)CC)C)occ2c1CCC2 54626,Cn1ncc2nc[nH]c(=NC3CC(C(N4CCC(c5ccccc5)C4)=O)C3)c12 54627,CC(C)(CCC(=O)N1CC(C)(C(=O)NC2CCCCC2(F)F)CC1(C)C)[N+](=O)[O-] 54628,CC1CCN(C(c2sccc2C2CC2)=O)CC1NC(c1nscc1N)=O 54629,c1(C(N2CCC(N(C)C(c3cnc[nH]3)=O)C2)=O)cc([N+](=O)[O-])cc(S(C)(=O)=O)c1 54630,c1(OCC(=O)N(C(C(=O)NC2(CCOC)CC2)C)C)ccncc1 54631,C(C(C(=O)NCCC(C)O)C(C)(C)C)NC(c1ncc(CC)cn1)=O 54632,C(CC1CC1)(C(=O)NCCN1CC=CC1)NC(C1C(C)C1C)=O 54633,C(=O)(C(F)C(C)CC(C)(C)C)NCC1N(C(c2c(CC)occ2)=O)CC(C)(C)C1 54634,C(=O)(C1CCc2cccnc21)N1C(CN(C(CCSCC)=O)C)COCC1 54635,N12CC3C(C3C1)C2=O.c1(NCc2cnc(CC)s2)ccc(Cl)cn1 54636,N1(C(C23OCC(C(C)C)(C2)C3)=O)CCN(c2ccc(C(=O)O)cn2)C(C)C1 54637,c1(C(N2CCC=C(Br)C2)C(=O)NCC)cccc(C(=O)OC(C)(C)C)n1 54638,C1(C(N2CC(C)=C(C)C2)=O)CC2CCCC2N1C(C1Cc2nccn2C1)=O 54639,c1(C(=O)NC(CNC(Cc2nnc(C)s2)=O)C(C)C)c(Cl)cnn1C 54640,c1(CC)cc(C(=O)NCC(C)CNC(=O)CCCC2CCOCC2)ccn1 54641,c1(OC)cc(C(N2CCC(F)(C(=O)Nc3cn(C)nc3C)C2)=O)cc(OC)c1Br 54642,C(CC(=O)NC1CC(NC(C2(c3cccc(C)c3F)CC2)=O)C1)(C(F)(F)F)OC 54643,c1(CNC(=O)NCc2n(COC)ncc2)cccc([N+](=O)[O-])c1C 54644,C1(C(=O)NCC=CCNC(C2(c3cccs3)C(C)C2)=O)CCC(F)(F)CC1 54645,C=Cc1cncc(C(N2CCC(NC(c3ncncc3F)=O)C(F)C2)=O)c1 54646,C=Cc1ccc(C(=O)NC2CC2CNC(=O)Cn2nnc(-c3ccco3)n2)cc1 54647,c1(N2CC(OC)(CNC(=O)Cn3nnc(C)n3)C2)cc(=O)n(C(C)C)c(O)n1 54648,N1(C(c2cnc(OC)c(C)c2)=O)CC2(CCC(NCc3c(F)cccc3F)C2)C1 54649,c1(N(C(C2CS(=O)(=O)C2)=O)Cc2cccc(OC)c2)ccc(S(N)(=O)=O)cc1 54650,c1(OCC)nc(Cl)ccc1C(=O)NC1CCN(C(C2CC3(CCC3O)C2)=O)C1C 54651,c1(C(=O)NC(C(C)NC(=O)COC(F)(F)F)C)cccc(OCCN(C)C)c1F 54652,C12(C(N(CC(C)NC(C3CN(CCC)C(=O)C3)=O)C)=O)CCOC(C)(C1)C2 54653,C(=O)(CCCCC(=O)N1CCC(NC(=O)CCn2nc(C)c(C)c2C)C1)NC 54654,c1(C(N(CC(CNC(c2n(C=C)nnc2)=O)C)C)=O)cc(Br)ccc1O 54655,N1(C(CN(CC)CC)=O)Cc2ccccc2C(NC(c2ncc[nH]c2=O)=O)C1 54656,n1(CC)cnc(C(N2CC(NC(C3CCC(COC)C3)=O)C2)=O)c1 54657,C=CCC(C(=O)N(CCCNC(c1cc(F)ccc1C(F)(F)F)=O)CC)C(C)C 54658,Cc1ccc(C(F)F)cc1C(N1CCOC(C)(CNC(=O)C=CCF)C1)=O 54659,Cc1cccc(C(=O)NCC2CC(NC(C3(C#N)CC3)=O)CC2O)c1Br 54660,N1(C(C2C(C)CCC2)=O)CCC2(CC1)CCN(C(=O)Cc1c(Cl)cccc1Cl)C2 54661,c1(CNC(CCCCC)C2CC2)ccc(Cl)c(Cl)c1 54662,O=Cc1c[nH]c2cc(C(N3CC(c4cc(O)n[nH]4)C3)=O)ccc12 54663,C1(C)(C(=O)NCCN(C(=O)C(C(C)C)NC(N)=O)CC)CCC(C)=C(C)C1 54664,N1(C(CC2CCN(C)C2)=O)CCN(C(c2cnoc2-c2cccs2)=O)CC(O)C1 54665,N1(C(C)C)CCC(C(=O)NCC2CCCC2NC(=O)C2=CCOC2)CC1 54666,C1(NC(c2c(CC)cncc2)=O)CN(C(c2c(Cl)cncc2Cl)=O)CCC1C 54667,N1(C(c2ccc(OCC)cc2)=O)CCC(F)C(NCc2ccc(I)cc2)C1 54668,C(CC1=CCN(C(C2CCOC2C)=O)CC1)NC(c1cc(C)sc1)=O 54669,C=C1COCCN(C(=O)C=CC(C)NC(=O)CC(C)n2cccn2)C1 54670,O=C(CCCn1cncn1)NCCC1CCN(C(c2ccco2)=O)C1 54671,c1(C(=O)NCC2(NC(=O)COc3ccncc3)CC2)cnn(C2CC2)c1Cl 54672,C1(NC(C(C)Cn2ccnc2)=O)CC2(C1)CC2NC(=O)CCC(=O)c1ccc[nH]1 54673,C(C(=O)NC(CC(=O)NCc1cc(OC)ns1)c1ccccc1)(C(C)C)NCC 54674,c1(C(N(C)CCN(C(=O)C(CO)N(C)C)C)=O)cc2c(C(F)F)nn(C)c2s1 54675,c1(C(C)NC(C2(O)CCN(C(c3cnc(Br)o3)=O)C2)=O)ccc([N+](=O)[O-])cc1 54676,C1(C)(C(=O)NOCc2n(CCC)nnn2)CCC2(CC1)CC2 54677,N1(C(C(CC(F)F)NC(C(CSC)OC)=O)=O)CCC(F)(F)C(F)C1 54678,C1(C(=O)NCC(C2(CC#C)CC2)=O)CC(=C)CCN1C(=O)CN(C)C(=O)C1CC1 54679,N1(C(CN(CCC)C)=O)CCOCC1CN(C(=O)C(F)C(C)C)C 54680,S(=O)(=O)(c1cccnc1C(F)(F)F)NC(CCN1C(C)C(C)N(C)CC1)(C)C 54681,c1(COC)cnc(OC)c(C(=O)NN(C)C(N)=S)c1 54682,CCC(C#N)C(=O)N1CCC=CC1C(=O)NCc1cc(C)ns1 54683,c1(CC)ccc(C(=O)NC2CC(N(C(=O)C=C(C)C)C)C2)c(F)c1 54684,C1(C(=O)N)CCn2nnnc2C1.Cc1noc(C(C)C)n1 54685,C1(C(=O)NCCC2(NC(c3c(Cl)cn(C)n3)=O)CCCC2)CC12CC(F)(F)C2 54686,c1(C(N2CC(NC(CCCC=C)=O)CC23CCC3)=O)cc2nccnc2cc1F 54687,CC1(C)CCC(C(CO)NC(=O)CNC(=O)Cc2ccccc2)CC1 54688,c1(NC(CC)(C)COC)ccc(S(=O)(=O)N2CCC(CCCO)C2)cc1C#N 54689,C1(C(N2C(CCCNC(CN3C(C)CC3)=O)CCC2)=O)CN2CCC1CC2 54690,C1(NC(C23CC(C)C2C3)=O)CN(C(c2ccc3n[nH]cc3n2)=O)CC2(CC2)C1 54691,N1(C(c2n(CC)cc(Cl)c2)=O)CCC2(COC)CCCC12 54692,C1(CNC(=O)CC2CCNC2=O)CCCCC1Nc1ncc(O)cn1 54693,O=S(=O)(c1ccc(=NCCCOCC2CCCO2)[nH]c1)NCC12CCCN(CC1)C2 54694,C12(NC(C=CC(C)(C)SC)=O)CC(CNC(=O)Cn3cncn3)(C1)OC21CCC1 54695,C1(C(=O)NCCN(C)CCO)CC2(CCC2)CN1C(c1[nH]nnc1C1CC1)=O 54696,C(=O)(CS(=O)(=O)NC(N)=O)NC1(CN(C(C2(CCC=C)CC2)=O)C)CC1 54697,C(=O)(C(C#N)C(C)(C)C)NC(C(NOCC(=O)OC)=O)C 54698,c1(C(=O)NCCCN(C(c2cc(Cl)cnn2)=O)CC)ccc2c(c1)N(C)CC2 54699,C1(C)(C(=O)NCC2(OC)CN(C(c3c(C)oc(C(C)C)c3)=O)C2)CCCS1(=O)=O 54700,N1(C(C2CC(=C)C2)=O)CC2CCC(NC(c3n[nH]c(C)n3)=O)CC2C1 54701,N1(C(CC(CC)NC(C2(c3cccnc3O)CC2)=O)=O)CCOCCC1C1CC1 54702,C1(COC)CC(CNC(c2csc(=N)[nH]2)=O)N(C(c2[nH]c(O)nc2C)=O)C1 54703,C1(F)(C(=O)NCC2C(NC(C=NOC)=O)C2)CCCOC1 54704,CC1C(O)CC2CCC1N2C(=O)OC(C)(C)C.c1(C23CC(C2)N3)cccc(Br)c1 54705,c1(C(=O)OC)cc(C)nn1CC(=O)NC(C)CC(C)NC(=O)C(C)CC1CCC1 54706,c1(OCC(=O)NCC2N(C(CCC=CC)=O)CCOC2)ccc(Cl)cc1Br 54707,c1(C(=O)NCC2N(C(C3N(C(C)=O)CC(O)C3)=O)CCC2)ccc(N)cc1Cl 54708,CON(C(=O)CCC1(C)CN(C(C2C(C)(C)C2(F)F)=O)C1)C1CCC1 54709,CCC(CC)(CO)C(=O)NC1CCN(C(=O)C(c2ccc(F)cc2)C)CC1 54710,C(C(C)C)(C(O)C(=O)N1CC(C(C(=O)NCC2CCOC2=O)OC)C1)OC 54711,C1(C(CNC(CC(C)N2CCOCC2)=O)C)CCN(C(=O)C(C)(C)CF)CC1 54712,C(C(C)(C)C(=O)NC1CCCC1CC(=O)NOCC=CCl)N(C)C 54713,c1(C(N2CC(F)(CNC(C(CCC#C)O)=O)C2)=O)cc(F)c(F)c(Cl)c1F 54714,Cn1ncc(NCc2cccnc2P(C)(C)=O)c(Cl)c1=O 54715,c1(SC(C(=O)NCC(=C)CCNC(=O)CN2CCC(C)C2)C)ccc(Cl)c(Cl)c1 54716,c1(C(=O)NC(CNC(CCC(C)OCC)=O)CO)cc(=O)n(C)cc1Br 54717,C1(C(=O)NCc2c(C)nn[nH]2)CC2(CC(NC(C3CCCC(=O)N3)=O)C2)C1 54718,C1(COCC)CCN(C(c2nonc2C)C(=O)NCc2ccccc2)C1 54719,N1(C(=O)NCc2ccn(C(C)C)n2)CCN(C2CCCOC2)CC1 54720,N1(C(Cc2ccc(C)s2)=O)CC=CCC1C(N1CCCC1CCO)=O 54721,N1(C(c2ccc(CC)s2)=O)CCCC2CN(C(=O)Cc3ccc(C)c(C)c3)CC12 54722,c1(CC(N2CCC(N3CCN(c4nncs4)CC3)C2)=O)ccccc1Cl 54723,c1(C(C(=O)NC2C(NC(Cc3c(C)scc3)=O)C2)C)ccc(F)cc1 54724,c1(CCN=C(NCC2OCC(C)C2)NCc2ccccc2)c[nH]c2ccccc12 54725,C1(c2ccccc2)(C(N(CCCOCC)NC(C2(CC)CC2)=O)=O)CC(OC)C1 54726,C1(CC)CCCCC1N(C(=O)C(C)(C)C1CCN(C(c2ccco2)=O)C1)C 54727,c1(C(=O)O)cc(CN2CC3(CC(C(=O)Nc4cc(O)nc(O)n4)C3)C2)cc(F)c1 54728,C(C(C)C(F)C(=O)NCC(n1ccnn1)C)NC(c1c(C)cc[nH]1)=O 54729,C(=O)(C(CC)(CC)CC)NC1CCC(C(=O)NC(CCC=C)C(=O)OC)CC1 54730,N1(C(CCSCCC)=O)CCCC(C)(NC(c2cccnc2S)=O)C1 54731,c1(CC(N2CC(CNC(c3cc(CCC)[nH]n3)=O)(COC)C2)=O)cnccc1C 54732,c1(C(=O)NCC2C(C)CN(C(=O)Cc3csc(Cl)c3)C2)cc(Cl)cc(F)c1N 54733,CC1CCCCC1CC(=O)NCC1(C)CC(C)(C)C1.C12CC(C1)NC2=O 54734,N1(C(C(CCSC)O)=O)CCOCC(C(=O)N(CCC(C)C)CC(C)C)C1 54735,C(c1cccc(Cl)c1)=CC(=O)NCC1CC(NC(c2cn(C)[nH]c2=N)=O)C1 54736,C1(NC(C2(CC#C)CC2)=O)COCCC1C(=O)NCc1ncc(CO)o1 54737,n1(CC(=O)NC2CC(CCNC(C=CC(CC)C)=O)C2)cc(C#N)c(O)nc1=O 54738,c1(C(=O)NC2C(NC(c3nccc(C)n3)=O)COC2)ccc2cccnc2c1N 54739,N1(C(C2(C(=O)O)CCC(F)(F)CC2)=O)CCN(C2=NCCCN2)CC1 54740,C(C)(CCC(=O)N1CCC(C)(CCNC(c2cc(F)n(C)n2)=O)C1)SC 54741,C#CCCCC(C)C(=O)NCC(C(C)C)NC(=O)Cc1cccc(SC)c1 54742,C1(NC(CC2CN(C(C)=O)C2)=O)CC12CC(NC(c1cccc[n+]1[O-])=O)C2 54743,N1(Cc2c(C)cccc2S(C)=O)C(=O)NC2(CCCCC2)C1=O 54744,C(=O)(NNC(=O)NC1CC1c1cccnc1)C1(NC(=O)OC(C)(C)C)CC1 54745,C1(CC)CN(C(=O)CC2CC(C)=NO2)CC1NC(C1CCC(N(C)C)CC1)=O 54746,C1(NC(CCc2ccc(OC)c(OC)c2)=O)CCNC12CCOCC2 54747,N1(C(CSC)=O)CCC(C)(CNC(c2c(C)coc2C)=O)C1 54748,C(=O)(CN=c1cc[nH]cc1)N1C(CCNC(C2(O)C(C)(C)OCC2)=O)CCCC1 54749,CC(C)C(O)C(C)C(=O)NCC12CC(NC(c3ccc(F)cc3O)=O)(C1)C2 54750,CC1(O)COCCN(C(c2cc(CNC(=O)C(c3ccccc3)F)no2)=O)C1 54751,N1(C(CCC#CC)=O)CC(NC(C2(OC)CCOCC2)=O)C(C2CC2)C1 54752,Nc1c(C(=O)NCCOCCCNC(C2CC23CC3(F)F)=O)cccc1Cl 54753,Cc1[nH]nc(Cl)c1NC(=O)N(C)Cc1cnn(C2CC2)c1C 54754,Cc1c([N+](=O)[O-])c(C(N2CC(NC(=O)C(=O)N(C)C)CC3(CC3)C2)=O)nn1C 54755,C1(CNC(=O)CCc2ccccn2)C(C2CC2)CCN1C(=O)Cn1cccn1 54756,c1(C(=O)OC(C)(C)C)ccc(OCC2CC2)c(C)c1.C1(OC)COC(=O)NC1 54757,C(=O)(C(=O)NNc1cc(C)c(Cl)cn1)NCc1c2ccc(C)cc2oc(=O)c1 54758,C1(CC#C)CCN(C(=O)C(C)N(C(C2(C#N)CCC2)=O)C2CC2)C1 54759,C1(C2CC2)(CNC(c2ncc(Cl)cc2F)=O)CCN(C(C2(O)CCOCC2)=O)C1 54760,N1(C(c2ccc(N)c(C)c2C)=O)CCN(C(C23CCCCC2C3)=O)CC(C)(C)C1 54761,C(C(CC(=O)N1CCCC1CN(C)C)NC(=O)C(C)CCN(C)C)OC 54762,N1(C(c2cc(CCC)c(C)s2)=O)CC(NC(=O)CCNC(C)=O)C(C)(C)C1 54763,C1(c2cn(CC3CCN3C(C3CN(C4COC4)C3)=O)nn2)(N(C)C)CCCC1 54764,N1(C(C(CCC)CC)=O)CCCC2(C1)CN(C(C1(CCO)CC1)=O)C2 54765,C1(NC(C(CSC)O)=O)CC2CCC1CN(C(C1(F)CCCCC1)=O)C2 54766,c1(C(=O)NC(CC)CNC(=O)CCOC(C)=O)cnoc1CC(C)C 54767,N1(C(C(CCCNC(C2ON=C(C(C)C)C2)=O)O)=O)CCCN(C=O)CC1 54768,O=C1NC2(CCO1)CN(C(=O)CC1CCCC1NC(C1CCC=CCCC1)=O)C2 54769,C1(C)(C(=O)NC2(CC)CC2)CC(O)CN1C(=O)C(CC1CCC1)OC 54770,CN1CCCC(CNC(C2CC(NC(c3cc(F)n(C)n3)=O)C23CCC3)=O)C1=O 54771,C(=O)(C(C)(F)C(=O)OC)N1CC(C)(NC(C(CC=CCC)C)=O)C1 54772,C1(NC(c2cc(COC)sc2)=O)CN(C(c2n[nH]c(C)c2Br)=O)CC1C 54773,C(=O)(C(CO)C(C)(C)C)NCCC(C)(C)NC(CN(C)C(c1ccoc1)=O)=O 54774,c1(N2CC(O)(CNC(C(CCC)OC)=O)C2)ncc(C)c(SC)n1 54775,Cc1sc(CN2CCC(CC3(O)CC3)CC2)c(Br)c1C 54776,c1(OC)cc(C(C(=O)NC(C)(C)C)N(C2CCC(=O)NC2=O)C(C)C)cc(F)c1 54777,c1(C(C)C)nccc(C(=O)NC(c2cccc(Cl)c2)CNC(C2CC2C)=O)n1 54778,NS(=O)(=O)c1ccc(C2CCN(c3ccc(Br)c(C(=O)O)n3)CC2)cc1 54779,c1(N(c2cccc(CNC(C3CCCN3)(C)C)c2)C)c(O)ccc2ccccc12 54780,c1(SC)nc(C(=O)N(CCCN(C)C(C2CC(F)CN2C)=O)C)c2ccccn12 54781,c1(C(N2C(C(C)NC(C3(C)CCC(=O)N3)=O)CCC2)=O)cc2nc[nH]c2cn1 54782,N1(C(C(F)OC)=O)CCC(NC(c2ccccc2N2CCCCC2)=O)C(C)C1 54783,C(C(CNC(=O)CCc1cnn(C)n1)CO)NC(C1CN(C(C)=O)C1)=O 54784,N(C1CCCc2c(I)n[nH]c21)C(c1coc(C(F)(F)Br)n1)=O 54785,CC1(C)CCCC(NC(C2(C)CCN(C(c3nccnc3N)=O)C2)=O)C1 54786,c1(OC)cc(-c2csc(CO)c2)ccc1OC(F)F 54787,N1(C(c2cc(C)sc2)=O)CCN(C(c2cc(C3CC3)ns2)=O)CC1CCO 54788,C12(NC(C3C4CN(C)CC43)=O)CCC(NC(C3(C#N)CC4CC4C3)=O)(CC1)C2 54789,C(=O)(CCC(=O)C1CC1)NC(C(C)NC(c1n[nH]cc1CN(C)C)=O)CO 54790,c1(C(N(CC(N2CCN(C(C(C)C(C)O)=O)CC2)=O)C)=O)cc(F)c(Cl)cc1Cl 54791,C1(N(C)C(C2(N(C(C34CC(C)(C3)C4)=O)CCO)CCC2)=O)CCCC(C(F)(F)F)C1 54792,c1(CC)cncc(C(=O)NCCCCNC(=O)Cc2ccnc(Br)c2)c1 54793,c1(NCC(N2CC(c3c(CNC(C(CSC)O)=O)nco3)C2)=O)ccc(O)cc1 54794,c1(CCCSCCNC(N2CSCCSC2)=O)ccc2ccccc2c1 54795,N1(C(C2(CC)CC2)=O)CCC2(CCN(C(c3cc(F)c4cn[nH]c4c3)=O)C2)C1 54796,c1(C(N(CC(CNC(C(C)OC(C)=O)=O)O)C)=O)ncc(C)cc1C 54797,c1(N(CCNC(=O)CC(C)C2CCCCC2)CC)ncnc(Cl)c1Br 54798,N1(C(Cn2c(C)ccc2C)=O)CCCC(N(C(=O)C(c2ccccc2)O)C)CC1 54799,N1(CCc2nnn(C(C)(C)C)n2)CCC(NC(CCC(=O)OC)=O)CC(C)(C)C1 54800,C12(C(N3C(CCNC(Cc4nc(C)oc4)=O)CCC3)=O)CCC(F)(CC1)C2 54801,C1(NC(c2ccc(CC)o2)=O)C2CC3C1C3C2C(=O)NCCc1cc(C)no1 54802,c1(NC(C)=O)sc(Cl)cc1C(=O)NCCC(C)(C)NC(=O)C(F)C1CC1 54803,C1(NCc2cnn(C)c2Cl)COC2(CCN(C(c3cccc(O)c3)=O)CC2)C1 54804,C1(CN(C)CCC2C(CC)CCCC2)CC12CCOCC2 54805,n1(CC=C)nnnc1C(c1csc(Br)n1)NC(c1nnc(CO)s1)C 54806,c1(C(=O)NCC2N(C(c3cc(C)c(N)cn3)=O)CC2)ccc(S(N)(=O)=O)cc1 54807,O=C(CS(=O)(=O)C1CC1)NC1COC2(C1)CN(C(c1cnc3cccnn13)=O)C2 54808,Cc1nc(NCCc2ncccc2C)cc(=NCC(C)N2CCCCC2)[nH]1 54809,C#CCCCCCNC(=O)C(CCC1CCC1)NC(C1CC1C(N)=O)=O 54810,S(=O)(=O)(c1ccc(NCCCCn2cnnc2)cc1Br)N(CCCC(=O)NC)C 54811,C(=O)(CCCCC(C)C)N(C1CCN(C(c2c(SC)nn(C)c2)=O)CC1C)C 54812,N1(C(C=CC2CCN(C(C(CC)C(F)(F)F)=O)CC2)=O)Cc2ccnn2CC1C 54813,CC1(C)C(CO)CN1c1nc(-c2ccccc2Cl)no1 54814,C1(C(=O)NC(C)(C)CS(C)(=O)=O)CN(C(=O)CC2CCC(=O)NC2)CC12CC2 54815,CC1(C(=O)NCC2CCN(C(=O)CCCc3ccccc3Br)C2)CC(F)(F)C1 54816,Cc1c(N2CCOCC2)ncnc1N1CCC(NC2COCC2C)CC1 54817,C1(C(=O)Nc2cccc(OC)c2)CCCN(C(=O)C=CCF)C1C 54818,C1(CNC(C2NC(=O)OC2)=O)(CNC(c2cccnn2)=O)CCCCC1 54819,c1(NC(C(CCOC)NC(=O)C(=O)N(C)C)=O)cn(CC)nc1C#N 54820,c1(C(N2CC(C(C)NC(c3cc(C)ns3)=O)C2)=O)c(C)ccnc1O 54821,c1(C(N2CCC(CC#N)C2)C(=O)NC)cccc(Cl)c1F 54822,S(=O)(=O)(CCC(=O)NCC1C=CC(NC(=O)C(c2ccccc2)O)C1)NC 54823,c1(CNC(c2c(CC)cc[nH]2)=O)ccc2c(c1)CCN(C(c1c[nH]nc1C)=O)C2 54824,c1(NC(C2CC2C(N2C3COCC2C3)=O)=O)cnc(I)cn1 54825,N1(CCC)CCCC(C(=O)NC(C)CCNC(c2cc(CC)no2)=O)C1 54826,C(N=c1[nH]c(=NC2CCCC(F)(F)C2)c2ccccc2[nH]1)c1nc(C)c(C)[nH]1 54827,c1(C(=O)NCCC2N(C(CCC#CC)=O)CCC2)ccc2c(c1)OCCO2 54828,Cc1nc([N+](=O)[O-])cn1CCC(N1CC(NC(C2(C)CC(C)(C)C2)=O)CC1C)=O 54829,c1(C(=O)NC2C(OC)CN(C(c3ccc(F)c(N)c3)=O)C2)cc2c(s1)CCCC2 54830,Cc1cn2c(CC(N3CCC(CNC(C4(C)C(C)(C)C4(C)C)=O)C3)=O)csc2n1 54831,c1(C(N2CCCC(C(C)NC(C(COC)NC(C)=O)=O)C2)=O)cnc(Cl)c(N)c1 54832,c1(C(=O)NC2C(SC)CN(C(c3nc(O)sc3C)=O)C2)cnc2sccc2c1 54833,C1(CNC(CCC(=O)OC)=O)CC2CCCC2N1C(=O)COCc1cc(C)on1 54834,Cc1cc(C)c([N+](=O)[O-])c(C)c1C(N1CC(CC(C)NC(c2ccon2)=O)C1)=O 54835,c1(C(=O)NCCN(C(C2(O)CCC(CC)C2)=O)C2CC2)cccc2c1CC(=O)N2 54836,c1(C(=O)NCc2c(C(N3CCC(CC=C)C3)=O)con2)ccc(O)nn1 54837,C1(=CC(=O)NC(C2(O)CN(C(=O)C=Cc3ccsc3)C2)C)CCSCC1 54838,c1(C(=O)Nc2nc(Cl)ccc2Br)c[nH]c2cc(-c3cnn(C4CCC4)c3)cnc12 54839,C1(NC(c2cc(CNC(C(CC)=CCCC)=O)no2)=O)CC(C)(C)OC1=O 54840,Cc1ncc(Cl)c(C(N2CCC(F)(CNC(=O)Cc3scnc3C)C2)=O)n1 54841,c1(C(=O)NC(C)CNC(c2cncn2-c2ccccc2)=O)c([N+](=O)[O-])cnn1C 54842,C1(C(=O)NC(CC)(C)CN(C)C(C2(C(C)=O)CC2C)=O)CC(C#N)(OC)C1 54843,Cn1cc(C2=CCCC2)cc(C(N2CCN(C=O)CC2)=O)c1=O 54844,C1(C(N2CCC(C)C2CNC(c2cn(C)cc2C(F)(F)F)=O)=O)CC2(C1)CC2(F)F 54845,C1(C(N2CC(CCCNC(c3c(OC)n[nH]c3)=O)OCC2)=O)OCCN(C)C1=O 54846,n1(CC(=O)NCCC2(O)CN(C(COCCCC)=O)C2)ncc2ncccc12 54847,c1(OC)c(F)cc(C(=O)NC(C)(C)C(C)NC(=O)CC2CC=CCC2)c(N)c1F 54848,c1(C(N2CCC3CN(C(COCC#C)=O)C3C2)=O)coc2c1C(=O)CCC2 54849,c1(C(N2CCC(C(C)NC(c3cc(CCO)on3)=O)CC2)=O)ccc(O)cc1Cl 54850,C1(C(N(C2CCCC(C)(C)C2)C)=O)CN(C(=O)C(F)n2ccnc2)CC(C)(C)C1 54851,c1(CC)ccc(C)c(NC(C2CCC(C)N2C(=O)CCC2CC2(F)F)=O)c1 54852,N1(C(CCN(C(CCC(C)CN(C)C)=O)CC2CC2)=O)CCOCC(C)(O)C1 54853,CCC(C(=O)N1CCC(CNC(=O)CC2CCC(F)(F)CC2)C1(C)C)C(C)(F)F 54854,C(N=c1[nH]c(N2CCCC3(CC2)CC3)nc2cc[nH]c12)C1(F)CC1 54855,C(C1CCCN1C(=O)CC1CC1)=CC(=O)NCC(C)C1CCC1 54856,c1(OCCC)ccc(CNC2(CC)CCNC2)cc1C 54857,C1(C(N2C(C)CCC(CNC(CCC(=O)NC)=O)C2)=O)CC2CCC1C21CC1 54858,N1(C(C2C(C)CCO2)=O)CCC(F)(C(=O)NC2(C)CCCC2O)C1 54859,Cn1cc(C(F)=CC(=O)NCCCCNC(=O)Cc2cccnc2O)cn1 54860,C1(CNC(c2ccc(F)cn2)=O)C(C2CC2)CCN1C(=O)COCC1CCC1 54861,c1(C(=O)NC(CNC(C2(COC)CCC2)=O)CO)cc(OC)ccc1C 54862,C(C1c2ccsc2CCN1C(=O)COCC(C)C)NC(CCCCCCC=C)=O 54863,C1(CC)(CC)CCC(NC2(c3nn[nH]n3)CCOC2)CC1 54864,C1(N(C(=O)C(F)CC2CN(C(C)=O)C2)CC)CCCN(C(=O)Cc2cn[nH]c2)C1 54865,Cc1c(C(=O)NCC2(CNC(C3CCCC(=O)N3C)=O)CC2)[nH]c2ccccc12 54866,C(=O)(C1=NOC(C)C1C)NC1CC(CNC(Cc2c(C)nc(S)s2)=O)C1 54867,C1(CC(=O)NC(C)CC2CC2)CCN(C(C23C(=O)C4CC2C3C4)=O)C1(C)C 54868,C1(C(N2CC(O)(C(C)CNC(C3CCCC(F)(F)C3)=O)C2)=O)CCC(C)(C)CC1 54869,c1(C(N2CCC(N(CC#C)C(C3CCC3OC)=O)CC2)=O)cc2sc(C)cc2[nH]1 54870,c1(C(=O)NCC(C(=O)N(CC(C)(C)N(C)C)C)OC)ccc(CO)cn1 54871,C(CC(=O)NC1CCCOC1)(C(F)F)NC(=O)CC1CC2(CCC2)C1 54872,Cc1csc(CNC(=O)C(c2ccnn2C)NC(=O)COCCF)c1 54873,N1(C(C(CO)OC)=O)CCC(C(=O)NC2CC3CCC2C3)(C(C)C)C1 54874,C(=O)(CCCCC(C)CC)Nc1c(CC)cc(C(F)(F)F)cc1.N12CC(C1)C2=O 54875,c1(C(N(CC(CN(C(=O)CN2CCCC2)C)O)C)=O)cc2sc(Cl)cc2s1 54876,c1(C(N2CCCC(CNC(C(CC)CN(C)C)=O)C2)=O)ccc(C)nc1C 54877,c1(CN(C2CN(C(=O)C(O)Cc3ccc(O)cc3)C2)C)cc(Cl)cc(Cl)c1O 54878,c1(C(N(C(CNC(C=C(CCC)C)=O)C2CC2)C)=O)ccnn1CC 54879,c1(-c2cn(-c3ccc(NC(C(C)CN)=O)cc3)nn2)cc(F)ccc1Cl 54880,CC1(CNC(C2(N(C(=O)CC34CCCC3C4)C3CC3)CC2)=O)CCCCC1O 54881,c1(C(N2CCN(C(C3CCC(OC(F)F)CC3)=O)C3CC23)=O)nnc(O)cc1O 54882,Cc1c(C(N)=O)cccc1C(N1CC2(CCC2NC(C2C3CC4C(C3)C24)=O)C1)=O 54883,Cc1c(C(F)(F)C(N2CCCCC2C(C)NC(=O)C2=CCOC2)=O)cnn1C 54884,CCC(CC)C(C(=O)NC(CN(C)C(C1(Cl)CC1)=O)Cc1ccccc1)OC 54885,CC(C)(C)CC(O)CC(=O)NC1CC2(C1)CC2C(=O)NC1(C(O)CO)CC1 54886,CCC(CC)(C(=O)NC1CCC(CNC(c2ccc(=O)n(CCF)n2)=O)C1)OC 54887,C1(CNC(CC=CCC)=O)(CO)CCCN(C(=O)C(F)C2CCC2)C1 54888,C1(OC(C)C(=O)NCc2ncoc2C2CN(C(=O)C=CCO)C2)CCCCCC1 54889,C1(CCC(N2C(CNC(c3c(C)coc3)=O)C=CC2)=O)CCCCN1C 54890,CCC(C#N)C(=O)N1CC(F)CC1CNC(=O)COCC(C)C 54891,N1(C(C(c2cccc(O)c2)C)=O)CCC2(C1)CN(C(=O)C(C)C(C)O)CCO2 54892,n1(C(C)(C)C)cc(C(=O)NCC2CC2NC(C2CCC(C(F)(F)F)O2)=O)nn1 54893,N1(C(Cc2n(C)ccn2)=O)CCC2CN(C(C3OCC4CCCCC34)=O)C2C1 54894,Cc1nc2ccc(C(N3CC4(CC(NS(=O)(=O)CCCl)C4)C3)=O)cc2o1 54895,N1(C(CNc2nccc(OC)n2)=O)CCOCC(NC(=O)CCC2CC2(F)F)C1 54896,CCC(C)(CC)C(=O)NC(C1CCN(C(=O)C(=O)Nc2cccc(C)c2)CC1)C 54897,C1(C(N)=O)Cc2cc(NC(NC3CCCc4sccc43)=O)ccc2O1 54898,CCC(CCC(=O)N(CCC(=O)NC1CCN(C(C)C)CC1)C1CC1)OC 54899,c1(CC)cc(C(=O)NC2CCC2NC(=O)CCc2cccnc2)sc1C 54900,C1(NC(C23OCC(COC)(C2)C3)=O)CCCCN(C(=O)C(C(C)O)N(C)C)C1 54901,N1(C(CCc2ccc(C)nc2)=O)CCC2(CC(NC(C3(C)CCOCC3)=O)C2)C1 54902,c1(CC)nn(C)cc1CN(C(C)C(=O)NC)C 54903,N1(CCCNC(C=C(CC)C)=O)CCN(C(c2ncoc2C2CCCO2)=O)CC1 54904,C1(NC(c2cc(CCCCC)[nH]n2)=O)CC(F)(F)CC1NC(=O)C1=CCSC1 54905,Cc1cc(C(=O)NCC2(F)CC(NC(=O)C(C)NC(C)(C)C)C2)n(C)n1 54906,O=C(C1=CCN(C(=O)C2=CCSC2)CC1)Nc1cncc(C2CC2)c1 54907,c1(-n2cc(C(CC(N)=O)NC(C(CC)OC3CCC3)=O)nn2)c(C)cccc1Cl 54908,N1(C(c2cccc(C#C)c2F)=O)CCC(NC(=O)CSCC)C(F)(F)CC1 54909,N1(C(C(C(=O)NC)(C)C)=O)CCN(C(=O)CCNC(C2CCCO2)=O)CC(O)C1 54910,CCCC(CC)CC(=O)N1CCN(C(c2c[nH]nc2C(C)(C)C)=O)CC1C 54911,C1(O)(CN(C)C(c2cnccn2)=O)CCCN(C(c2ccnc(C3CC3)n2)=O)C1 54912,C(N=c1nc2c(cnn2C)c(Nc2cnc[nH]c2=N)[nH]1)C1CCCC(CC)CC1 54913,N1(C(C2C(CC)CCO2)=O)CC(S(=O)(=O)N2CCN(C(C3CC3(F)F)=O)CC2)C1 54914,c1(C(=O)NC(CC)CNC(=O)CNC(C)=O)ccc2c(c1)CCCN2C(C)=O 54915,N1(C2CCN(CCN(C)C)CC2)CCCC(C(N2CCCCC2C(N)=O)=O)CC1 54916,N1(C(COCC)=O)CCC(C2CCCCN2C(c2ccn(C3CCC3)n2)=O)CC1 54917,c1(C(=O)NC2CC(F)(CNC(C3CC(C)N(C)C3)=O)C2)cccc(S(N)(=O)=O)c1 54918,Cc1c(C(=O)NCC(C)NC(=O)CC(C)C)cc(O)cc1N.c12ccc(cc1)o2 54919,C1(C(N(CC(N2CCC2C2CCCC2)=O)C(C)C)=O)CCCC(=O)N1 54920,C1(C(=O)N(c2ccsc2)C)(CNC(CC2CC(=C)C2)=O)CC=CC1 54921,C1(N(C(Cn2cc(-c3cccc(C)n3)nn2)=O)C)CCCCC1(C)C 54922,C1(C(N(C2CCCN(C(CCC=CC)=O)C2)CC)=O)OCCOC1(C)C 54923,n1(CC(=O)NC2CCN(C(C(C)CF)=O)CC2O)nc2n(c(=O)c1=O)CCOC2 54924,c1(C(=O)NCC23OCC(CNC(C(CC)(F)F)=O)(C2)C3)cc2ccccn2c1 54925,C(CNC(=O)Cc1csc(Cl)c1)(C(C)C(C)C)NC(Cc1cnc(C)[nH]1)=O 54926,C(=O)(CCCC(C)NC(N1CCOC(C(F)F)C1)=O)OC(C)C 54927,c1(OCC)cccc2c(NC(=O)NC3CCC(SC)CC3)c([N+](=O)[O-])cnc12 54928,N1(CC(N2C(C(=O)NC(C3CC3)C3CC3)C=CC2)=O)C(=O)CNC1=O 54929,C1(C(=O)NCCC(C)(C)NC(CC(C)c2cccnc2)=O)C(C)(C)C1(C)C 54930,C(C)(CC(C)NC(=O)Cc1cncs1)NC(CN(CCOC)C)=O 54931,C1(NC(C(COC)(C)C)=O)CCN(C(c2cccc(CCN(C)C)c2)=O)C(C)C1 54932,C=Cc1cncc(C(N2CCCC(N(C(=O)CC(C)C(F)F)C)C2)=O)c1 54933,Cc1nsc(N)c1C(=O)OCC(C1CC=CCC1C(F)(F)F)=O 54934,C1(NC(C(=Cc2cn[nH]c2)C)=O)CC(C)N(C(c2nnsc2N)=O)C1 54935,Fc1ccsc1C(c1cn[nH]c1)NCc1cccs1 54936,N1(C(c2n(C(C)C)ccc2)=O)CCN(C(=O)CCc2nccn2C)CC12CC2 54937,c1(N(C)Cc2ccn(C)n2)nc(N2CCN(CC(F)(F)F)C(C)C2)nc2sccc12 54938,c1(C(N2CCN(C(C(C)SCC)=O)C(CCOC)C2)=O)cc2ccsc2c(O)n1 54939,CC(C(=O)NC1CC(CCn2cc(-c3ccncc3F)nn2)C1)C(F)F 54940,N1(C(C2N(C)CCC2)=O)CCCC2C1CCN2C(c1cc(Cl)ccc1[N+](=O)[O-])=O 54941,c1(C(=O)NCC(CO)NC(C(C(C)C)O)=O)cc(Cl)ccc1C(F)F 54942,C1(CC(N2C(CC)CN(C(c3nc(C)sc3C)=O)CC2)=O)NC(=O)CN(C)C1=O 54943,N1(C(c2c(CC)nccn2)=O)CCCN(C(=O)C(O)Cn2cncn2)C(C)C1 54944,CCCC(C)(CCC)C(=O)NC1COCC1CNC(=O)C=Cc1ccoc1 54945,C(C1=CCCN(C)C1)NC(N(Cc1ccc(OC)cc1)Cc1ccccc1)=O.OC 54946,CCC(CC(=O)N1CCC(C(C)NC(=O)CCn2ccnc2C)C1)C1CCC1 54947,C(=O)(CCCC(F)(F)F)N1CC(CC(C)NC(c2cn(C(C)C)nc2)=O)C1 54948,C(CC1=CCN(C)CC1)N1CC(=O)N(C(C(N(OC)C)=O)C)C1=O 54949,C1(C)(c2nc(SCc3c(C(=O)OC)[nH]cc3C)on2)COCCN1CCCOC 54950,CC1(C)CC(CNC(c2cnc(=N)[nH]c2)=O)N(C(=O)C(N)=O)C1 54951,C1(C(=O)NCc2n(C)cnn2)CC2(CCC2)CN1C(C1CCC1)=O 54952,C(=O)(C#CC1CCC1)NCC(CC=C)NC(=O)Cc1cccc(C(N)=O)c1 54953,C1(N(C)C(c2coc(C(N)=O)c2)=O)CN(C(c2cn(CCF)nn2)=O)CC12CC2 54954,N1(C(CCSCCCC)=O)CCCC1(C)C(=O)NC(CO)CCF 54955,N1(C(C23CC(NC(CC4CC(=C)C4)=O)(C2)C3)=O)CC(C)CC(C)(C)C1 54956,CCC(C)(C(=O)NC1CC(C)N(C(=O)C(=O)NOC)C1)c1ccccc1 54957,Cc1onc(-c2ccsc2)c1C(=O)NCC(n1cc(C2(C)CC2)nn1)C 54958,C1(NC(CC(C(F)F)NC(C=CC(C)C)=O)=O)CCn2ncnc2C1 54959,c1(OCC(N2CC(O)(CNC(c3c(CC)cco3)=O)C2)=O)ccc(O)cc1 54960,c1(C(=O)NC(CCC)CNC(=O)C(F)CC2CCOC2)oc(C)nc1CC 54961,c1(C(=O)NC2CC(C)(NC(C3CN4CCN3CC4)=O)C2)cccc([N+](=O)[O-])c1N 54962,C1(C(N2CCC(N(C(Cc3ncc(CC)[nH]3)=O)C)CC2)=O)CCCCNC1=O 54963,O=S(=O)(c1nc(N2CCOC3(CCCCC3)C2)ccc1Br)NC1(CO)CC1 54964,C1(NC(C(CC)C#N)=O)(CO)CCCN(C(C2CC3CC(=O)C2O3)=O)C1 54965,c1(CN(CC2C(=O)N2CC)C(=O)COC)cn(C)nn1.C(C(C)C)OC 54966,C1(OC)(OC)CCN(C(C(=O)NCCCSCC)C(C)C2CC2)C1 54967,N1(C(C(C)SCCCC)=O)CC2CC(NC(=O)CCc3ccncc3)CC1C2 54968,c1(CCC(=O)NCC(CNC(c2c(CC)occ2)=O)(C)F)cccc(F)c1 54969,C12(NC(CC3(C=C)CN(C(c4cnn(C(C)C)c4)=O)C3)=O)CCC(CC1)C2(C)C 54970,C1(C(N(CCNC(=O)CSC2CC2)CC)=O)CC(=O)C1C 54971,Cn1cc(CCC(=O)N2CC(CNC(C3C(c4ccccc4)C3F)=O)C2)cn1 54972,C1(NC(C2C(C(C)C)C2)=O)CC2CCC1CN2C(C1CCC(C)CC1)=O 54973,c1(CC(=O)N(CC(C)NC(COCCC)=O)CC)ccc(C)nc1 54974,c1(C(N2C3CN(c4nccc(C)n4)C(CC3)C2)=O)cc(Br)c2ccccc2n1 54975,C(=O)(C1CN(C)C(=O)c2ccccc21)NC(C)CNC(=O)C=CCF 54976,c1(NC)cnccc1C(=O)NCCCN(CCO)C(C1CCC1OC)=O 54977,C1(C2CCN(C(c3ccc(S(C)(=O)=O)o3)=O)C2)(NC(CS(CC)=O)=O)CC1 54978,C1(NC(C(C=C)(C)CC)=O)CC2CN(C(=O)C(CCC)C(C)C)CC2C1 54979,C(C1=NOC2COCC12)NC(C1(CC)CCCN(C(=O)Cc2cscn2)C1)=O 54980,CCCCC(CC)C(=O)NC(C)(C)CNC(=O)CC1CCN1C(=O)OC(C)(C)C 54981,C(CNC(c1c(C)n[nH]c1C)=O)(C(C)(C)C)NC(C(C)OCCC#C)=O 54982,C12(CNC(c3c(Cl)cn(C)n3)=O)CCC(C1)N(C(C13CC(F)C1C3)=O)C2 54983,C(C(O)(C(F)(F)F)C1CCC1)NC(NC(CC)C)=NCCC1CC1 54984,N1(C(CCCC=C)=O)CCN(C(c2ccc(-c3ccccc3)[nH]2)=O)C(CCC)C1 54985,Cc1cccc(C(=O)NCC2(C)CCCN2C(=O)COc2ccccc2)c1F 54986,Cc1cc(C(N2CCN(C(C3C4CC5C(C4)C35)=O)CC2CC(F)F)=O)nnc1C 54987,c1(C(N2CCCCC(CNC(C3CC(C#C)(O)C3)=O)C2)=O)c(F)ccc(C)c1Cl 54988,C1(CC(C)C)CN(C(=O)CC(C)(C)C)CC1NC(=O)CC1C=NN(C)C1=O 54989,c1(OC)cc(C(=O)N(C2CCC(NC(c3[nH]ccc3C)=O)CC2)C)cc(F)n1 54990,CS(=O)(=O)c1cc(C(N2CCN(C(=O)C3=C(Cl)CC3)C(CO)C2)=O)ccc1F 54991,c1(OC)c(Cl)cc(C(=O)N(CC(C)(C)NC(C2CC(C)C2)=O)C)cc1Cl 54992,CCCC(CNC(c1cnn(C2CC2)c1)=O)C(=O)NCc1ncccc1O 54993,c1(CNC(CN(C(=O)C(COC)NC(C)=O)CC)=O)ccc(C)c(C)n1 54994,C(=O)(CCC(N)C(=O)O)N1CCN(Cc2c(OC)cccc2)CC1C 54995,Cc1ccc2c(c1)N(C(=O)N(CC1=CCCOC1)CCO)CCC2 54996,c1(C(=O)NCC(N(C(CCOC(C)C)=O)C)C2CC2)cc(Br)c2cccnn12 54997,N1(C(c2ccn(CCCC)n2)=O)CCN(C(c2cnn3ccsc23)=O)C2CC12 54998,CC1CC(CNC(c2cc(CN(C)C)no2)=O)CN1C(=O)CCn1cncn1 54999,N1(C(c2cc[nH]c(=N)c2N)=O)C(CNC(=O)Cc2ccc(Cl)s2)CC2COCC12 55000,C1(C2CN(C(=O)CCc3nc(O)n[nH]3)C2)(NC(C2N(C)CC(O)C2)=O)CC1 55001,C(N=C(NCC1CCCO1)N1CCC2(C1)CC2(F)F)c1cc(C)cc(C)n1 55002,c1(NCC(=O)Nc2cccc3[nH]ccc23)cc(F)c(N2CCCCC2)c(F)c1 55003,C1(NC(COCCCC)=O)CC2CCC1N2C(=O)C(C(C)C)OC 55004,C1(CC)(NC(c2nccn2C)=O)CCN(C(c2c[nH]nc2C)=O)CC1 55005,N(C1CCc2cccnc21)C(c1ccc(CNC(c2cn(CCC)nn2)=O)o1)=O 55006,CC(O)C(C(=O)NCC(C)(C)CNS(C)(=O)=O)N(C)C 55007,C1(CCC(=O)NC2C(C(=O)OCC)CC2)CCCN1C(=O)CCCN(C)C 55008,CCS(=O)c1ccc(-c2ccc3nnc(C(=O)NC(C)C)n3c2)cc1 55009,C1(Nc2cccc(OCC#N)c2)CCCC2CNCCC12 55010,Cn1nccc1C1OCCC1C(=O)NCC(C1CCC1)NC(C1CC(F)(F)C1)=O 55011,C1(C(=O)NCC(C(=O)NC(C(=O)OCC)CC)C)CCC(C)(C)CC1 55012,N(C(=NCCC1CCCN(C(C)=O)C1)NCC1CC1)C(C=C)C.c1cnccc1Cl 55013,CCC1=NOC(C(=O)N(CC(C)(C)CNC(C2(C)CNC(=O)C2)=O)C)C1 55014,c1(NCC23C(CN(C(=O)OC(C)(C)C)C2)C3)nc(O)c2ncnc-2[nH]1 55015,C1(NC(c2cn(CC(C)C)nc2)=O)CCCCCN(C(=O)CC(C)F)C1 55016,CC1(C(=O)NCC2(F)CN(C(C3CC3CF)=O)C2)CC(c2ccccc2Cl)=NO1 55017,CC1(F)CCN(C(=O)CC2(C)CCN(C(=O)CC3(O)CCCOC3)C2)CC1 55018,CCC(F)(F)CC(=O)NCC1CN(C(=O)C(c2ccccc2Cl)N(C)C)CC1C 55019,c1(C(=O)NC2CN(C(=O)COCCCF)CC2CO)c(O)cccc1F 55020,C1(OCC(=O)NC(C)CC2CCCCN2C(=O)C2=CCCC2)CCCCC1C 55021,c1(C(=O)NCC(C)(C(C)C)NC(C(CCOC)C)=O)nc[nH]c2nccc1-2 55022,C1(C(=O)NC(C2N(C(C(C(C)C)F)=O)CCC2)C)C2(CCC2)C12CCC2 55023,CCCCCCCCC(=O)NCCC1(OC)CN(C(C2(n3cncn3)CC2)=O)C1 55024,C1(CN(C(C2C(C(N(CC#C)C)=O)C2)=O)C)CCN(C(c2cnc(S)[nH]2)=O)CC1 55025,C1(CC(=O)NCC(C)CNC(=O)CC#N)CCCCC1(F)F 55026,c1(NC(C(C(C)CNC(=O)C=C2CCOCC2)F)=O)cccc(N=[N+]=[N-])c1 55027,c1(Cn2cc(-c3cnc(OC)s3)nn2)cc2c(cn1)CCCC2 55028,C(=O)(CCC1CCc2ccccc21)NCCCn1cc(C(C(C)C)O)nn1 55029,C#Cc1ccc(C(=O)NC(C)CN(C(=O)CS(=O)(=O)NCC2CCCO2)C)nc1 55030,C(=O)(CCC(C)(C)NC(c1ccn(CCF)n1)=O)NCC(c1cn(C)nc1)O 55031,C(=O)(C(CO)C(F)(F)F)N1CCCC(CC(N2C(C)CC2)=O)CC1 55032,c1(C(N(C)CC2C(NC(CCCN(C)C)=O)CCC2)=O)cc(O)cc(F)c1 55033,C1(NC(CCCCC=CC)=O)CCOC2(CCN(C(=O)CCCCC)CC2)C1 55034,Cc1ncc(CNC(C2(CCNC(=O)CCCn3ccnn3)CC2)=O)o1 55035,N1(C(C2CCC3(CC3)C2)=O)CCCC2(CCCN2C(=O)CC2CCCOC2)C1 55036,C1(NC(=O)CC)CCCN(C(C2(COC)CN(C(c3nc(Cl)sc3Cl)=O)C2)=O)C1 55037,Cc1cc(NC(C2CCCN2C(=O)CC2CCC(C)(C)C2)=O)cc(O)c1 55038,C1(C(N(C)C)=O)Cc2ccccc2CN1C(c1cccc(S(C)(=O)=O)c1)=O 55039,n1(CC(N2CC(C(C)NC(Cc3c(C)occ3)=O)C2)=O)ccc2c(C)cccc12 55040,C(=O)(C1(C)OC(=O)c2ccccc21)NCC1CCc2c(cnc(C)n2)C1 55041,C#CCCCCC(=O)N1CCC1C(N1CCCC(CCCO)C1)=O 55042,C(=O)(C(C(C)(C)C)NC(=O)CCOCCC)NCC(CCC=C)O 55043,c1(CC(=O)NCCCCC(C)NC(C23CCCC2C3(F)F)=O)cccc(Cl)c1F 55044,c1(C(N2CC(CNC(c3ccc(SC)o3)=O)C2)=O)ccc(N)c2c1CCCC2 55045,Cc1c2cccc(NC(C3CC3C(=O)NCC3CCCOC3)=O)c2nn1C 55046,c1(NCc2c(N3CC(C)OCC3)cccc2)cc(OCC(=O)O)ccc1F 55047,n1(CC)cccc(NC(c2sccc2CNC(=O)Cc2ccoc2)=O)c1=O 55048,c1(NC(C)C)ncc(Br)c(C(=O)NC(C)(CNC(=O)C(C)C2CC2)CO)n1 55049,C1(CNC(CN(C2CCC2)C)=O)CC(NC(=O)C(C)(C)CF)CC1O 55050,O=C(N=c1cc(C(F)F)[nH][nH]1)N(C1CCCCC1)CCF 55051,N1(C(c2cc(C3CC3)nn2CC)C(=O)NCC)CCC2CCN(C)C(=O)C2C1 55052,N(C(=NCC1CCCC12CC2)Nc1ccccc1Cl)CCNS(CC)(=O)=O 55053,N1(C(C2(COC)CN(C(C3CC(O)(CC#C)C3)=O)C2)=O)CC(O)(C#C)C1 55054,c1(C(=O)NCC(CCCC)NC(C2CCC(OC)C2)=O)c(COC)nn(C)c1Cl 55055,c1(C(C)C(=O)NC(C)(CNC(=O)Cn2cncn2)CO)cccc(Cl)c1 55056,N1(C(C2C(C)=CCS2)=O)CCC2(CC2NC(C2CC2c2ccccc2)=O)C1 55057,N1(C(c2c(Cl)nc(N(C)C)s2)=O)CC2(CC(NC(C3CCC(F)(F)C3)=O)CO2)C1 55058,C1(NC(C(CN(C(C2(CC)CCOC2)=O)C)C)=O)CCCCCC1C 55059,N1(C(C)=O)CCC(Nc2ncnn2C2CN(C(=O)OC(C)(C)C)C2)C2CCC12 55060,Cc1nc2ncc(C(=O)NCC=CCNC(=O)C(C)N3CCC3)c(=O)n2[nH]1 55061,c1(C(=O)NCC(C(C)C)NC(c2cnc(O)s2)=O)ccn2ncnc2c1 55062,C1(C)(CC)CCN(C(=O)CCN2CCC(NC(=O)CN3CCOCC3)CC2)C1 55063,c1(C(N2CCC(O)(CC(C)NC(COCCCC)=O)C2)=O)nc(Cl)c(=O)[nH]c1N 55064,CC(C)(F)C(=O)NCC1CCN1C(c1cc(-c2ccccc2)on1)=O 55065,c1(OC)cccc2c1CN(C(=NCC(C)c1ccncc1)NCCSC)CC2 55066,c1(C(=O)NCC(C)NC(c2c(C#C)c[nH]n2)=O)cccc2c1ccn2CCOC 55067,c1(C(C)C)cc(C(=O)NC2CC(NC(C3CCN(C)C3)=O)C2)on1 55068,n1(CCC)cc(C(N2CC(CCc3cn(-c4ccc(Cl)cc4)nn3)C2)=O)c(C)n1 55069,c1(NC(C2(CC#C)CCCO2)=O)cccc(CNC(=O)C(C)C(F)F)c1 55070,Cc1nn(C)c(C)c1CC(=O)NCC1C(C)CCCN1C(c1cnco1)=O 55071,c1(C(=O)NCCN(C(=O)C(C)c2cc[nH]n2)CCOC)nc(O)sc1C 55072,C1(NC(COC)=O)CC2CCC1N2C(=O)CCNC(c1ncccc1O)=O 55073,c1(-n2cc(CCN(C(COCCOC)=O)CC)nn2)ccc(N2CCC(O)C2)cc1 55074,CC1C(OC(C)(C)C)CCCN1N(CCO)CCO 55075,Cc1snnc1C(=O)N(C)CCN(C(=O)C(F)C1(NC(=O)OC(C)(C)C)CC1)C 55076,Cc1ccc(Br)nc1CNC1C2CC3C(C2)C13CO 55077,n1(-c2c(OC)cccn2)c(-c2csc(C(=O)NC3CC3)n2)nc2c(C)ccnc12 55078,c1(N(C)C(=O)Nc2cc(C3(O)CC3)[nH]n2)ccc(OCc2ccccc2)cc1 55079,N1(C(c2c(C)cccn2)=O)CCCC(C2CN(C(=O)C3=CC4C=CC(C3)C4)C2)C1 55080,N1(C(C)=O)C(C)CN(CC(=O)NC2CC3(C2)CC3(F)F)CC1C 55081,N1(CC(=O)N(C2C3CN(C(CC(C)OC)=O)CC32)C)CCCCS1(=O)=O 55082,N1(C(c2ccc(SCC)nc2)=O)CCC(NC(C2(CCF)CC2)=O)C(C)C1 55083,N1(C(CN2CCC(=O)CC2)=O)CC(NC(=O)CCc2cnn[nH]2)C(C2CC2)C1 55084,C(=O)(C(C1CN(C(=O)Cc2cscn2)C1)OC)N(CC(C)C)CC 55085,N1(CC(=O)NC2(C)CN(C(C3CCC(=O)O3)=O)C2)CCC(F)(F)C1 55086,c1(C(C(=O)NCC2(CC(=O)N(CCC#C)CCOC)CC2)F)ccccc1 55087,c1(OC(CC(=O)NCC(C2CC2)NC(CC)=O)C)cc(Cl)cc(Cl)c1 55088,N1(C(C2(CNC(c3cccnn3)=O)CCCC2)=O)CC2CCCC(O)C2C1 55089,c1(C(N2CCN(CC)C(C)C2)C(=O)NCC2CCOC2)ccc2c(n1)OCCO2 55090,c1(SCC(=O)N(CCCN(C(C2CN(S(CC)(=O)=O)C2)=O)C)C)ccccc1O 55091,CC(C)C(C(C)NC(=O)Cc1csc(-c2nc[nH]n2)n1)NC(=O)Cc1ccsc1 55092,N1(C(c2c(C(C)C)ccs2)=O)CC(NC(C2CN(C(N)=O)C2)=O)CC(F)C1 55093,C(=O)(C#CC1CCOC1)ONC(C1(NCC2(NC(=O)C)CCCC2)CCC1)=O.CO 55094,C1(C)(CNC(C2C(C)CC2)=O)CCN(C(=O)C(O)C2CCC2)CC1 55095,N1(C(CC2CC(NC(C)=O)C2(C)C)=O)CC(N2CCCC2)CC1C(N)=O 55096,N1(C(c2c(C(=O)OCCCNC(=O)C(F)C(C)C)nns2)=O)CCC(OC)CC1 55097,Cc1nc2[nH]n(C)c(=O)c2c(C)c1CC(N1CCOc2cccc(C(C)C)c21)=O 55098,N1(C(C(C2CC2)NC(N(C)Cc2ccccc2)=O)=O)CC(C)(C)NC(C)(C)C1 55099,c1(C(=O)NCC2N(C(C(C(C)C)CN(C)C)=O)CC2)nc2cc(F)ccc2s1 55100,c1(C(N2CC3C(NC(c4ccc(C(=O)OC)cn4)=O)(C3)C2)=O)cc(C)c(C)cn1 55101,C1(CNC(c2c(C(C)C)noc2)=O)CC2COCC2N1C(=O)CC1CCC2CC12 55102,C(C(=O)NCCN(C)C)(C(C)OC)NC(c1c(CC)ncs1)=O 55103,C(=O)(C(CO)C(F)(F)F)N1CCC2(C(C(=O)NCCc3n(C)nnc3)C2)C1 55104,c1(C(C)=O)c[nH]c(C(=O)NC(c2cn(C)nn2)C(=O)N(CCCF)C)c1 55105,N1(C(c2c(C)nco2)=O)CCC2(CCC2NC(C2CC23CCCCCC3)=O)CC1 55106,C(=O)(C(CC(F)F)C1CCC1)NCC1CC(NC(=O)CCc2nc(O)n[nH]2)OC1 55107,C1(NC(=O)C2=CCC2)CCN(c2ncncc2I)CCC1CO 55108,c1(COC)nc(C(=O)NC2(CO)CN(C(=O)C(C)C3CCOC3)C2)co1 55109,C(=O)(C(O)CC(F)(F)F)N(CC)CC1CCCN(C(=O)CCn2cnnn2)C1 55110,C1(C(=O)NC2C(C(=O)NC(C3CCCC3)C)CC2)CCCC1F 55111,N1(C(COC2CC(NC(C(CCCC#C)C)=O)C2)=O)CCN2C(=O)OCC2C1 55112,C1(NC(c2cc(C)c(C)o2)=O)CC2(C1)CC(C(=O)NCC1CC(O)CCO1)C2 55113,Cc1c(C(N2CCN(C(=O)CCc3ccoc3)C3CC23)=O)ccc2c1CCC2 55114,c1(C(CC)(C)O)cn(Cc2ncoc2CNC(c2ccc(F)s2)=O)nn1 55115,C1(CNC(c2c(C)onc2)=O)CN2CCCCC2CN1C(=O)C1=CCOCC1 55116,C1(NC(c2cc(C)oc2C)=O)CC(C)CN(C(C2(O)COC2)=O)C1 55117,c1(CNC(=O)CCCC2CCCCC2)cnn2c1CN(CCF)CC2 55118,Cc1c(CC(N2CC3CC3(CNC(C3CCCC3(C)C)=O)C2)=O)ncn1C 55119,c1(C(N2CCCC(N(C(C3C(C=C)OCC3)=O)C)C2)=O)cnc(CC)nc1O 55120,c1(CC)ccc(C(F)(F)C(N2CC(NC(c3cnc(O)n3C)=O)C(O)C2)=O)cc1 55121,C(=O)(C(C)(C)n1cc(NCc2ncnn2C2CCOCC2)cn1)OC 55122,C1(CC(=O)NCC(C)OCC)(CC2CCCC2)OCCO1 55123,N1(c2n(CC)c(COc3ccc(Br)cc3)nn2)CCc2cc(C)ccc2C1 55124,Cc1cccc(O)c1C(=O)NCC1(F)CC(CNC(=O)C=CCOC(C)(C)C)C1 55125,Cc1cc(C)c(S(N)(=O)=O)cc1N1CC(NC(=O)OC(C)(C)C)CC2(CC2)C1 55126,C=CCC(C)(C)CNC(=O)C(=O)NCC1CCOC1C 55127,Cc1cccc(CC(=O)N(CCCNC(=O)C(C)Cn2cccn2)C(C)C)c1Cl 55128,C12(CC(N3C(C)CC(CNC(C4(F)CCC4)=O)C3)=O)CC3CC(CC(C3)C1)C2 55129,Cc1cc(N2CCC3CCC(NC(c4sccc4F)=O)C2C3)ncc1[N+](=O)[O-] 55130,Cc1cc(Cl)cc(Cl)c1OCC(=O)N(C)CCNC(c1ncn(C)n1)=O 55131,C1(C(N2CC(CNC(C3CC34CCOC4)=O)OCC2)=O)CCc2nn[nH]c2C1 55132,c1(NC(CC2N(C(COCC)=O)CCOC2)=O)ncc([N+](=O)[O-])cc1O 55133,N1(c2cc(C)ncn2)CCC(NC(C2CCC3(C2)CC3(F)F)=O)C12CCC2 55134,c1(CNC(=O)NCCC(=O)Nc2c(CC)cccc2)cc(Br)cnc1C 55135,Cc1cnc2n1C(C(=O)N1CC(CO)(NC(c3cc(=O)cc(Cl)[nH]3)=O)C1)CCC2 55136,Cc1cc(C(=O)N(C2CN(C(c3nnc(S)n3C)=O)C2)C)c2c(c1)CCO2 55137,C1(C(=O)NCCCCC=C)CCC2(CC2)N1C(=O)Cc1n[nH]c(C)n1 55138,CCC(CC)C(F)C(=O)N1CCCC1C(=O)NC1CN(CC(F)F)C1 55139,CCCC(C(=O)N1CC(C)(OCC(=O)NCc2n[nH]cc2CC)C1)OC 55140,C(=O)(CCC(=O)N1CCC(C(=O)NC2CCN(C3CC3)C2=O)(CO)C1)NC 55141,c1(NC2CCC3CN(C(c4c(C)ncs4)=O)CC3C2)nc(Cl)nc2[nH]c(O)nc12 55142,N1(C(C(CC=C)C)=O)Cc2ccc(CNC(=O)Cc3cc(COC)no3)cc2C1 55143,c1(C(N2CC(O)CCC(NC(CC(COC)C)=O)C2)=O)ccc2c(c1)OCCN2 55144,C1(O)(CCNC(c2ccn(C(C)C)n2)=O)CCN(C(C2CCCCC2F)=O)CC1 55145,CN1CC2CCN(C(C3CC(C)(NC(C4C5COCC45)=O)C3)=O)CC2C1 55146,CC1(NC(=O)CNc2nccs2)CC(NC(c2csc(-c3ncccn3)n2)=O)C1 55147,N1(C(CNC(C2CCC2)=O)=O)CCC2(CCN(C(C3CCSC3)=O)C2)C1 55148,N1(C(C(CCNC(=O)CSC(F)F)OC)=O)CC2(CNC(=O)C2)C1 55149,c1(C(N(CC(CNC(Cc2nc(CC)sc2)=O)C)C)=O)cccc(NC(N)=O)c1 55150,C1(OCCC)CCCCC1C(=O)N(C)CCN1CCN(C(=O)CC(C)(F)F)CC1 55151,CC1CCCC(CC(=O)NCCCCNC(=O)C=C2CCN(C)CC2)C1 55152,CCCC(C(O)C(=O)NC(CC)(CC)C(C)C)NC(c1ccc2c[nH]nc2c1)=O 55153,c1(OC)cc(C#N)ccc1C(c1nnnn1C1CC1)NCCC(C)(C)C(=O)OC 55154,Cc1ccc([N+](=O)[O-])cc1C(N1CC2CC(NC(=O)Cc3scnc3C)C2C1)=O 55155,Cc1cccc2ncc(C(N3CC(C4CCCO4)CCC3C3CCNCC3)=O)n12 55156,N(C(=NCC1(F)CC1)N1CCCC(O)(c2ccc(Cl)cc2)C1)CC(C)C 55157,c1(C(=O)NC2CCC(N3CCOCC3)C2)ccnc(Cl)c1O 55158,Nc1ccc(C(=O)NC(Cc2ccccc2)CCNC(=O)CSCCO)cc1F 55159,C(=O)(CCC(C)(C)C#N)N1C(CNC(c2cnc(SC)s2)=O)CCCC1 55160,C12(C(=O)NC3CCCN(C(C4C5CC(F)(F)CC45)=O)C3)CCCCCC1OCC2 55161,c1(C(=O)NCCN(C(CCSCC)=O)C2CC2)cccc(F)c1 55162,C12(CNC(C3(C)CC=CC3)=O)CCC(CNC(C3(O)COC3)=O)(CC1)CO2 55163,N1(C(CSCCC)=O)CC2CCC(C1)N2C(=O)C=Cc1ccc(OC)c(C)c1 55164,C1(C(=O)NCC(C)CNC(=O)C(C)(C(F)F)c2ccccc2)CN2CCN1CC2 55165,CN1CCCC1CCCNC(C1(CC(F)F)CCNC1)=O 55166,N1(C(C(C)=CC)=O)CCC2(CCN(C(=O)CC3COC(=O)C3)C2)C1 55167,N1(C(C(C)C2CC2)=O)CCC(F)(CNC(=O)CNC(=O)C=Cc2cccnc2)C1 55168,N1(C(C(C)C)=O)CC(NC(=O)C(C)Oc2cccnc2)C(C#N)C1 55169,CCCCC(C)(CO)NC(C1CC=CC(NC(=O)CCc2cscn2)C1)=O 55170,c1(CNC(C(=Cc2cnc[nH]2)C)=O)cccc(Br)c1.C12CCC(C1)NCC2 55171,C1(C(=O)NCCC#C)CN(C(C2(CN(C)C)CC2)=O)CCO1 55172,C1(NC(C(CC=C)(C)C)=O)CC1C1CCCN(C(C2CCCC(O)C2)=O)C1 55173,c1(OC)c(CN2CCCC(C(=O)Nc3c(C)ncnc3C)CC2)cc(Cl)cc1Cl 55174,Cc1nncn1NC(=O)C1C=CCCN1C(C1CCCCCN1C)=O 55175,c1(OC)ccc(CN(C(=O)C(=O)Nc2csnc2C2CC2)C)c(C(F)(F)F)c1 55176,C(=O)(CC(CC)C(F)F)N1C(C(=O)NC(CC)C(=O)N(C)C)CC(OC)C1 55177,C1(C(=O)NC(CCCC=C)C)N(C(c2ccnnc2C)=O)CCCC1(C)C 55178,CCC(C)(CO)C(=O)N(C1CCN(C(=O)CNS(=O)(=O)CCCOC)CC1)C 55179,C1(F)(C(=O)NC2(C(=O)NCC3(CC)CCCC3)CSC2)CCOC1C 55180,N1(C(c2nncc(OC)c2)=O)CC(NC(c2cc(C(F)F)[nH]n2)=O)CC12CCC2 55181,C12(CNC(C(CC)OC)=O)CCC(CC1)N2C(=O)C(c1cccs1)SC 55182,C1(NC(=O)C2=COCC2)CC(F)CN(C(c2ccc(=O)n(C3CC3)c2)=O)C1 55183,c1(CC(C(=O)OC)NC(C2OCC3CCCC2C3)=O)c(F)c(F)c(F)c(F)c1F 55184,Nc1c(F)cc(C(N2CC3(CCCC3NC(c3cncnc3)=O)C2)=O)c(F)c1F 55185,C#CCCCC(=O)NCCC1CSCCN1C(=O)COC(C)(C)CC 55186,CC1C(O)CCCN1C(c1n[nH]cc1CNC(c1ccc(=O)n(C)c1)=O)=O 55187,c1(C(N2CCC(NC(C3C(=O)NCC3)=O)C2)=O)cc2cccc(Br)c2s1 55188,c1(C(N2Cc3[nH]nc(-c4ccnnc4)c3C2)=O)ccn2ncc(Br)c2n1 55189,C12(NC(Cc3c(C)scc3)=O)CCC(CNC(=O)C(n3cc(Cl)cn3)C)(C1)OC2 55190,S(=O)(=O)(CC(C)C#N)N1CC(OC)OCC1 55191,c1(CC(=O)NC2C(NC(C(CC)OC3CCCC3)=O)C2)cccc(NCC)c1 55192,N1(C(C(c2cccs2)SC)=O)CCCN(C(=O)COC(C)=O)CCC1 55193,c1(NC(C)C)cccc(C(N2CCC(CN(C(=O)CCc3cnc[nH]3)C)C2)=O)c1 55194,C1(C(N2CC(NC(C3CCN4CCCC4C3)=O)(CF)C2)=O)CCc2cnnn2C1 55195,CCC(C)(F)C(=O)N1CCCC(NC(=O)NC2CCCC2)C1 55196,N1(C(C2(C=C)CC2)=O)C2CCC1CN(C(C1(C3CC3)CCC1)=O)C2 55197,C(=O)(CC(CC)C1CC1)N(CCCC(=O)NCCc1noc(CC)n1)CCC 55198,O=S(=O)(NCCc1ccc(Br)cc1)N1CCC(S(=O)(=O)c2ccccc2)C1 55199,CCCCC(C(=O)N1CC2CC1CN2C(c1n[nH]cc1Cl)=O)N1CCCS1(=O)=O 55200,CCCCCCCCC(=O)NC1CCC(CCC(=O)NCCN(CCC)C(C)C)C1 55201,C(=O)(C1=NOC2COCC12)NC(CNC(c1nn(CCCC)c(=O)cc1)=O)CC 55202,O=C1Cc2c(N3CCC3C(=O)Nc3ccc4nncn4c3)ncnc2N1 55203,c1(CNC(C2(C)CCN(C(C(CCC)OC)=O)C2)=O)cccc(F)c1F 55204,n1(C2CCN(C(N3CCCc4[nH]ccc4C3)=O)C2)nc(C(=O)O)c2c1CCCC2 55205,C1(CC(=O)NCCCCC2C(C)C2)(NC(C2CC3CCC3C2)=O)CCCCC1 55206,N1(C(c2ccn(C(C)C)n2)=O)CC2CN(C(c3ccnc(S)c3)=O)CC(C1)O2 55207,C1(C(=O)NCC(CNC(c2ccncc2C)=O)OC)CC2(CCCCC2)S1(=O)=O 55208,c1(C(=O)NCCN(C(CCC(C)OC)=O)CCOCCO)ccc(N)c(Cl)c1O 55209,C1(C(=O)Nc2c(C(=O)OC)csc2)CCN(C(c2cscc2OC)=O)CC1O 55210,C#CC1(C(=O)NCC2CCC(F)C2)CN(C(=O)CC2CC(N(C)C)C2)C1 55211,c1(CNC(C)=O)ccc(C(=O)NCC2CC2(C)C)nn1.C12CCC(C1)NC2=O 55212,c1(C(=O)NC(CNC(c2onc(C)c2C)=O)C2CCC2)cc2c(nc1N)CCC2 55213,N1(C(C(COC)C)=O)CC2CCCC(C1)N2C(c1ccnnc1O)=O 55214,c1(CN2CCN(CCC(=O)NC3CN(C)C3)CC2)c[nH]c2cccc(F)c12 55215,N1(C(C(C2CCN(C(CN(C)CC)=O)C2)F)=O)CCC12CC(CC(N)=O)C2 55216,c1(C(C(=O)N(C)CCn2cc(Cc3ccccc3)nn2)O)ccc([N+](=O)[O-])cc1 55217,CCC(CNC(C1CCCOC1CN)=O)(CC)NC(C1CC(F)(CO)C1)=O 55218,C(=O)(CCS(C)(=O)=O)NC1C(CNC(c2ccc(CC)[nH]2)=O)CCCC1 55219,c1(C(=O)NCC(CO)NC(C2CCS2(=O)=O)=O)ccn2c(C(F)(F)F)nnc2c1 55220,CC1CCN(C(C23CCCCC2OCC3)=O)C(C)C1NC(C1CC=CCN1C)=O 55221,N1(C(c2c(CC)non2)=O)CCC(NC(=O)C=C2CCCC2)C(F)C1 55222,CC(C)CCN=C(NCC1(C2CCC2)CCC1)NCC1(CO)COC1 55223,C(=O)(C1=CC2CCC(C1)C2)N(C1CCC(NC(C(C(C)C)C)=O)CC1)C 55224,N1(C(Cc2cc(OC)no2)=O)CC(C)N(C(=O)Cc2cc(Cl)ccc2Cl)CC1C 55225,O=C(C1=CCCCC1)NC1C=CCC(C(=O)NCC(Cl)Cl)C1 55226,C1(C(=O)NC(CC#C)CC)CNC(=O)CN1C(=O)C(C)N(C)C(C)=O 55227,CC(C(=O)NCCCC(=O)N1CC(O)(CO)C1)C(F)F 55228,C1(NC(C2C(C)C2)=O)CN(C(C2CCCSC2)=O)CC2(CCC2)C1 55229,N1(C(C(CC)CO)=O)CCC2(CC1)CC2n1cc(-c2ccc(N)cc2OC)nn1 55230,c1(C(N2CC(CNC(C3(C)CCOCC3)=O)C3C2C3)=O)ccc(Cl)nc1N 55231,C1(NC(C(CCC)NC(N)=O)=O)CCCN(c2nnc(CCC)s2)CC1 55232,N1(CC2N(Cc3cn(C)nn3)CCC2)CC=C(CNC2CCCC(F)(F)C2)CC1 55233,CC1(C(=O)NC2CC(CCNC(c3conc3C(C)(C)C)=O)C2)CCCCC1 55234,c1(C(=O)OC)c(S(=O)(=O)NC2CCOC23CCCC3)n[nH]c1C 55235,c1(CN2CCN(Cc3c(C)cccc3Br)CC2)nc2ccccc2c(=O)n1C 55236,C(=O)(C(O)CNC(=O)C(C)CNC(C)=O)NCC1CC(C(=O)OC)C1 55237,c1(COC(=O)C(C)C(=O)OCCC(C(=O)OC)OC)ccc(C#N)cc1F 55238,c1(CC)nc(C(N2CCC(C(C)C(=O)NCC(O)CF)CC2)=O)c(N)s1 55239,C(=O)(C(CO)C(C)(C)C)NCC1(C)C(C)CN(C(=O)C(C)(C)CC2CC2)C1 55240,Nc1cc(F)cnc1CO.C1C(CC(=O)O)NC(=O)C2CC(n3cc1nn3)C2 55241,c1(NCCOC)cccc(-c2cn(CC(C)NC(=O)CCCCC3CC3)nn2)c1 55242,c1(CC)cc(-c2cn(C3CCN(C(C)=O)C3)nn2)n[nH]1 55243,c1(CC)onc(C)c1C(=O)NCC1CC1NC(=O)CCCN1C(=O)CCC1=O 55244,c1(C(=O)NCC(C)(C2CCC2)NC(C(C)NC(CC)=O)=O)cc([N+](=O)[O-])c(C)s1 55245,Cc1cc(C)c(C(=O)NC2CCNC2C2CC2)cn1 55246,CCCC(C(=O)N1CCC(NC(c2cnoc2-c2ccco2)=O)C1)OC 55247,Cc1nc(C)n(CC(=O)NC2(CCNC(=O)Cc3sc(S)nc3C)CC2)n1 55248,c1(C(N(CCNC(C2CC3(CCO2)CC3)=O)CC)=O)cnc2ccncc2c1 55249,N1(NC(c2nncn2C)CC)CCC(C#N)(c2ccc(C)cc2)CC1 55250,c1(C(=O)NC2CCN(C(c3ccco3)=O)CC2O)cc2cnccc2o1 55251,CC1(C)CN(C(c2c(F)cncc2F)=O)c2cc(-c3cccc(O)c3)cnc21 55252,CC(C)CC(C(=O)NCC1CCN(C(c2cncc(Cl)n2)=O)CC1C)C(C)C 55253,N1(C(C2C(C(C)C)OCC2)=O)CC=CC(C(=O)NCCCC2(C)CC2)C1 55254,Cc1nscc1CNC(=O)CN(C)C(C1CC2CC2C1)=O 55255,c1(C(=O)NC(CC)(CNC(=O)Cc2ccc(Cl)s2)CC)cccc2nccnc12 55256,c1(C(N2C(C)CC(CNC(C(CC)NC(C)=O)=O)C2)=O)ccnc2ccsc12 55257,C1(CC)C(NC(c2ccn(C)c2C)=O)CCCN1C(c1ccc(=O)n(C)n1)=O 55258,C1(C(=O)NCC2(NC(=O)C=CCO)CCC2)CNC(=O)N1 55259,c1(CN2CCC(F)(C(=O)NC(C)C3CC3)CC2)cnc2ncccn12 55260,C1(NC(c2c(Cl)cc(C)s2)=O)C2CC(CN(C(c3cc(CF)on3)=O)C2)C1CO 55261,C1(F)(CNC(C2(C)CCSCC2)=O)CC2CCC(C1)N2C(=O)C=C1CCC1 55262,CCC(C)CC(=O)C(=O)N1CCCC(C(=O)NCC2(SC)CCC2)C1 55263,C(c1ccc(OC)cc1)=CC(N1CC(N(CC)CC)C1)=O.O(C(F)F)CCN 55264,c1(C(=O)NCC2(C)CCN(C(C(CCCOC)C)=O)CC2)ccc2occc2c1 55265,C(c1csc(S(=O)(=O)N2CCC2)c1)=CC(N1CC(C(=O)OC)C12CCOCC2)=O 55266,C(=O)(C1=C(C)OCCS1)N1CCC(CCOC)(NC(C2CCC2(F)F)=O)C1 55267,c1(OC)ccc2ccnc(C(C)NC(c3cc(F)ccc3C(=O)O)=O)c2c1 55268,C1(CC(=O)Nc2cc(C(C)(C)C)no2)CCN(c2ncncc2I)CC1 55269,N1(C(c2cc(OCC)no2)=O)CCCCC1C(C)(C)CNC(c1cnsc1)=O 55270,CC1(C=CC(=O)NCCC2CC(NC(c3cnc(C4CC4)s3)=O)C2)CCOCC1 55271,Cc1ccc(CC(=O)NCC2(C)CCCN2C(=O)C=Cc2ccncn2)cc1C 55272,c1(C(=O)NC2CN(C(C(CC)(C)C)=O)CC2C#N)c(Cl)ccc(OC)c1F 55273,C1(C)(CNC(CC2CC(OC)C2(C)C)=O)CCN(C(=O)CN2CC(C)(C)C2)CC1 55274,N1(C(c2c(C)nc(O)s2)=O)CC2CCCC2(NC(c2cccc3ccnn23)=O)C1 55275,CC(O)(C(=O)NCCCOCCNC(=O)CC1(C(F)F)CC1)C1CCC1 55276,C1(NC(c2ccn(CC3CC3)n2)=O)CCOCC1NC(C1(CF)CCOCC1)=O 55277,c1(C(N2CCN(C(CCOCC)=O)CC2C(C)(C)C)=O)cn2c(n1)CCCC2 55278,N1(C(C(CC)C)=O)CC(O)(C2(CNC(C3CCC(N(C)C)C3)=O)CC2)C1 55279,C(=O)(CCCCCF)N1CCC(NC(c2c(C)cc(CC)o2)=O)(COC)C1 55280,N1(C(C(CCCC)N(C)C)=O)CCCCCC(NC(=O)CC2CCC2)C1 55281,C1(CC=C)(NC(=O)C(C)CN(C)C(c2csnc2OC)=O)CCOC1 55282,N1(C(CCC=C=C)=O)CCCCC(CNC(C2CCCOC2)=O)C1 55283,C1(NC(c2n(COC)ncc2)=O)CCN(C(=O)CNS(=O)(=O)N(C)C)C12CCC2 55284,C1(NC(c2cn(CC)nn2)=O)CN(C(c2coc(C(N)=O)c2)=O)CC1O 55285,C12(C(=O)NCc3ncc(CC)[nH]3)CCC(NC(c3cnsc3)=O)(CC1)C2 55286,c1(C(C(=O)NCCC2CC(NC(C(C)(O)C3CCC3)=O)C2)O)ccc(Cl)c(F)c1 55287,c1(C(=O)NCCCOCCCNC(C2(SC)CC(O)C2)=O)cc(Cl)c(C)cn1 55288,O(N(C)C(=O)CN=c1[nH]c2c(c(=NC(C)c3ccncc3Br)[nH]1)COCC2)CC 55289,C(=O)(CC(CN(C)C)CC)NC1CCC(N(C(C2CCC(CC)O2)=O)C)CC1 55290,C(=O)(C#CC1CCCCC1)N1C2(CN(C(CC3CC(=C)C3)=O)C2)CC1 55291,c1(-c2ccc(C)cc2)nc(=NC(=O)N2CC=C(Br)CC2)s[nH]1 55292,C(C1(O)CCc2ccccc21)N(C(C1CC2=C(C)NNC2=NC1)=O)C 55293,Cc1nn(CC(=O)N(C(CNC(C2(Cl)CC2(F)F)=O)C2CC2)C)cc1[N+](=O)[O-] 55294,c1(N2CCCC(CS(=O)(=O)NC)C2)cc(Br)cc(F)c1C#N 55295,Cc1nc(Cl)ccc1C(=O)NC(C)CNC(=O)CSC(F)F 55296,C(=O)(C1=CNS(=O)(=O)N=C1C)N1CC(CNC(CC(C(F)(F)F)OC)=O)OCC1 55297,c1(CNCC2OCCN(C(C3N(C)CCC3)=O)C2)ccc(Br)cc1C#N 55298,N1(C(C(C(C)C)C#N)=O)CC2CC(NC(=O)CSC(F)F)C(C2)C1 55299,N#Cc1cnn(CC(=O)NCCCCCNC(c2cc(C3CC3)on2)=O)c1 55300,C(=O)(CCC(C(C)C)NC(=O)C(F)C(C)(F)F)NC(CC)CCCO 55301,N1(C(CC2N(Cc3ccc(OC)cc3F)CCOC2)=O)C2COCC1CC(F)C2 55302,c1(NC2CCCN(C(CNC(C(C)NC(N)=O)=O)=O)CC2)cn(C)c(=O)nc1O 55303,C1(NC(c2cncc(OC)n2)=O)CN(C(=O)C2=COCCC2)CC(F)(F)C1 55304,c1(C(=O)NC2(CC(=O)NC3(CCF)CCOCC3)CC2)cccc(F)n1 55305,CCCCC(=O)C(=O)NC(C)(CNC(=O)C=CS(C)=O)C1CCC1 55306,CCC(F)(C(=O)OC)C(=O)NC1CCCCC1NC(C12CC(C)(C1)OC2(C)C)=O 55307,c1(CC2N(C(c3csc(C)c3C)=O)CCC2)ccc(S(C)(=O)=O)cc1 55308,N1(C(C=CC=CC)=O)CCC(C2(O)CN(C(=O)C3=CSCS3)C2)CC1 55309,c1(C(CNC(=O)CCC2CC2(F)F)(F)F)ccc(Cl)cc1Cl 55310,c1(-c2n(CC=C)c(N(C)CC3COCCC3(F)F)nn2)ccc2ccccc2c1 55311,CC(C)CC(C)CC(=O)N1CCC(C(=O)NCCc2c[nH]nc2O)CC1C 55312,C1(CC)CN(C(=O)COC)CCN1C(c1cn(CCN2CCOCC2)nn1)=O 55313,c1(C(C)(C)C)cncc(C(=O)NCCC2CCN(C(=O)C(C)(C)C3CC3)CC2)c1 55314,N1(C(CC)C(=O)OC(C)(C)C)CC2(CC2C(=O)NCC(N2CC(C#N)C2)=O)C1 55315,C1(C(=O)OC)C2CN(C(C3CCC4(CC4)C3)C(=O)NCCSC)CC12 55316,N1(C(CCC#CC)=O)CCCC(COC)(NC(=O)C=NOC)C1 55317,C1(NC(C2C(OC)CC2)=O)CCN(C(C2CC(SC)C2)=O)CC1(C)C 55318,C(=O)(C1=CC2CCCCC12)N1CC(NC(c2sc(CC)c(C)c2)=O)C(C)C1 55319,N1(C(c2c(C(C)C)[nH]cc2)=O)CCC(C)N(C(C2CCC2(F)F)=O)CC1 55320,c1(C(=O)NC2CC(C)(NC(C3C=CCC3)=O)C2)cccc([N+](=O)[O-])c1O 55321,N1(C(c2c(C)nc(C)o2)=O)CCC2(C)CN(C(C3CCC(C)C3)=O)CC12 55322,c1(C(=O)NCC(CNC(C2CCN(C)C2)=O)(C)O)oc2ccccc2c1Br 55323,CC1CN(C(C2COCCN2C=O)=O)CCCN1C(=O)CCC(F)(F)F 55324,N1(N2C(C=O)CCC2)CCc2nncn2CC1.C12CC3CCC1N3C2=O.CC=O 55325,C1(C2CN(C(=O)COC(F)F)C2)(NC(=O)COc2ccc(Br)cn2)CC1 55326,c1(C(=O)NCCC(CNC(C2CC2(C)C)=O)OC)ccc(C(C)C)cn1 55327,CC1C=C(C(=O)NC(c2cn(C)nn2)CNC(C2(C)CNC(=O)N2)=O)C1 55328,C(=O)(NNc1ccc(Cc2ccccc2)cc1)NC(c1csnn1)C 55329,c1(CC)ccoc1C(=O)N(C1CCOC1C)NC(COC1C(N)COC1)=O 55330,C1(F)(NC(N2CCC(COC)C2)=O)CCC(C(=O)OC)CC1 55331,Nc1nc2ncccc2cc1C(N1CC2(NC(C3CCC(=O)NC3)=O)CC1C2)=O 55332,C1(NC(C2(SCC)CC2)=O)CC2CCC(C1C)N2C(c1cccc(N)n1)=O 55333,Cc1ccc(C)c(CC(=O)NC2CCC2CNC(=O)CN2CC(=O)N(C)C2=O)c1 55334,c1(CN2CCC(NC(c3c(C)cccc3)=O)(CO)CC2)cccc2cccnc12 55335,c1(CNC2CCC(C(=O)Nc3c(C#N)cc(F)cc3)C2)ccc(Cl)c([N+](=O)[O-])c1 55336,S(=O)(=O)(c1ccc(N2CCCC(S(N)(=O)=O)C2)c(Cl)c1)NC(=O)OC(C)(C)C 55337,Cc1cc(C(N2CCC(NC(c3cc(CO)[nH]n3)=O)C2C2CC2)=O)ncn1 55338,c1(OC)ccc(C2(CSC3CCC(NC(C4(OC)CC4)=O)C3)COC2)cc1Cl 55339,C1(NC(c2ccc(C(C)C)o2)=O)C=CCN(C(=O)CNC(=O)CCCCO)C1 55340,N1(CCNC(=O)Nc2n(CC)ccn2)C(=O)NC(C)(C2CCCC2)C1=O 55341,Cc1cnc(O)n1-c1cccc(NC(=O)C(=O)NC(C)CN2CCCC2=O)c1 55342,c1(CSC)ccc(-c2nc(C3CC3Cl)n(Cc3ccc(C(F)(F)F)nc3)n2)cc1 55343,CC(Cc1ccncc1)N=c1cc[nH]c(=NCCCc2ccccc2)[nH]1 55344,c1(CCC)nc(C(=O)NCCOCCCN(C(=O)C=CC(C)(C)SC)C)co1 55345,C(=O)(C1CCc2nccn21)NC1CN(C(C2(SC)CC2)=O)CC1C 55346,C1(C(=O)NC(C(C)NC(=O)Cc2cccnc2Br)C)CC2CCC1CC2 55347,c1(C(N(C)CCOCCNC(C2CCCC(C#N)C2)=O)=O)cnc2ccccn12 55348,C=C1CCCN(C(=O)CSCCNC(c2ncn(CC)n2)=O)C1 55349,C(=O)(CCCCC(C)C)N1C(CNC(CCCc2onc(C)n2)=O)CC(C)(C)C1 55350,C(=O)(CC1CCc2ccccc21)NCC1CCC(NC(C(C)NC(=O)NC)=O)C1 55351,C12(NC(C3CC(NC(C4CCC(C)CC4)=O)C(O)C3)=O)CC=CC(C1)OC2 55352,N1(C2CCC(NC(c3c[nH]nc3F)=O)C2)CCN(C(=O)C2=CCSC2)CC1 55353,Cc1ccc(CC(=O)NCCC(C)NC(=O)CC2CC(C3CC3)C2)cc1Cl 55354,c1(CCC(=O)NCC2(CNC(=O)C(C3CCC3)C3CCC3)CC2)ncc(F)cn1 55355,c1(-c2c(C)noc2)cnc2cc(C(=O)NCCc3ccsc3)ccn12 55356,Cc1ccn2cnc(C(=O)NC3C=CCN(C(C4CC4CC(C)(C)C)=O)C3)c2c1 55357,C1(CC(=O)NCCCOCCNC(C(C)c2cccs2)=O)CCOCC1(C)C 55358,C(=O)(C1CCc2nccn21)NC1CCC(CNC(c2c[nH]c(=N)s2)=O)CC1 55359,C1(N(C(C2CCCN(C(C3C(C(C)C)C3)=O)C2)=O)C)CCCC(C)C1C 55360,C12(C(C)C)CCC(NC(c3ncoc3CNC(C34CC3CNC4=O)=O)=O)C1C2 55361,C=C=C(C)CC(=O)N(CCCOCCNC(=O)C(CC)NC(C1CCC1)=O)C 55362,C1(C(C)(C)C)(C(=O)NCCOC2CN(C(CC3C(C)CCC3)=O)C2)CCCCC1 55363,c1(C(N(C(C)C(=O)NCCS(C)(=N)=O)CCC)=O)cc(C(C)C)no1 55364,c1(CNc2c(CC(=O)Nc3ncc(C)c(F)c3)cccc2)ccc(F)c(C)c1Cl 55365,c1(CC(=O)NCC(C)(CC)NC(C(CCC)O)=O)ccc(S(N)(=O)=O)cc1 55366,c1(CC(=O)NC(CCNC(C(CC)NC(C)=O)=O)C)c[nH]c2cc(OC)ccc12 55367,c1(C(N2CC3C(CNC(c4cnn5c4CCC5)=O)(C3)C2)=O)snc2ccccc12 55368,c1(NC(CN(C(=O)NC2C(OC)CC2)C2CC2)=O)ccc(C(N)=O)cn1 55369,C1(C(NOCC2CC(=C)C2)=O)C2CC1N(C(=O)C=Cc1ccncc1)C2 55370,CCC1=C(C(=O)NCC2(C(C)NC(=O)C=CC3CCOC3)CC2)CCCO1 55371,c1(OC)cccc2ccc(C(=O)NC(C)CN(C(=O)CS(C)(=O)=O)C)nc12 55372,S(=O)(=O)(c1ccc(Nc2ncccn2)cc1)N1CC2C(N(C)C)(CC2)C1 55373,C(=O)(C(F)C(C)CC(C)(C)C)N(C)CC1CCCCN1C(=O)C(=O)N=S(C)(C)=O 55374,S(=O)(=O)(c1ccc(N2CCS(=O)(=O)CC2)c(Br)c1)NCc1ccc(OC)cc1C 55375,c1(CNC(C2CC(C)OCC2)=O)cnn2c1CN(C(C1CCN(C)CC1)=O)CC2 55376,C=CC1CN(C(=O)CCCn2ccnn2)CC1NC(=O)CC1CNC(=O)C1 55377,c1(N2CCN(C(=O)Cc3cc(F)ccc3F)C3C2C3)ncnc2cc(Br)ccc12 55378,Cc1nc(C)c(C(N2CCC(O)(C(C)NC(=O)Cc3nn(C)cc3Cl)C2)=O)s1 55379,Cc1cc(C)c(CN2CCN(C(=O)C=Cc3ccoc3)C3CC23)cc1C 55380,C=CC1(CO)CCN(C(C2CCOC2CNC(=O)CC(C)N(C)C)=O)CC1 55381,c1(C(=O)Nc2c[nH]nc2C(=O)Nc2cc(F)ccc2I)cc2sccc2[nH]1 55382,c1(C(N(CC(C)(C)CNC(c2cc(C(F)F)[nH]n2)=O)C)=O)cccc(F)c1Cl 55383,C(=O)(C(CC)C(F)(F)F)NC1(C)CCC(NC(CNS(CCCC)(=O)=O)=O)CC1 55384,C(=O)(C(C)(C)CSC)NC(CN(C(c1cnc(-c2ccccc2)o1)=O)CC)C 55385,N1(C(C=CCC=C)=O)CCC2CCC12CNC(c1cn(Cc2ccccn2)nn1)=O 55386,N1(C(CC)C(=O)O)CCC2(CC1)CC2(C)C(=O)NC1CCOC(c2cccs2)C1 55387,c1(C(C)C)c(C(=O)N(CC(O)CN(C)C(c2ncccn2)C)C)cnn1C 55388,c1(C(C)NCc2cc(C3CCC3)no2)coc2ccccc12 55389,c1(C(=O)NCCn2cc(CNC(C(C)C(F)(F)F)=O)nn2)cc2cccn2cn1 55390,c1(NC(COC)C)nc(N2CC(OC)C(OC)C2)nc2sccc12 55391,CN1CCC(C)(C(=O)NCC2(C)CCN(C(C3(c4cc[nH]n4)CC3)=O)CC2)CC1 55392,C1(C(=O)NCC2CCC(NC(C(c3cnn(C)c3)C)=O)CC2)CC2CCC(C1)O2 55393,c1(C(=O)Nc2cccc(C(=O)NC3CC(C)(C)OC3)c2)cc(O)ncc1F 55394,C(=O)(CS(=O)(=O)C(C)C)N1CCC(NC(C2(C=C)CCCCC2)=O)C1C 55395,CN1CCN(C(=O)Cc2csnn2)CC1CNC(=O)COc1ccon1 55396,N1(C(C(=O)NCCCC)CC2CCC(C(C)(C)C)CC2)CCC2C(O)C(C)(C)C12 55397,C(=O)(C#CC1CCCC1)NCCCCC(C)NC(C1(c2cccc(O)c2)CC1)=O 55398,C(=O)(C(C(C)CC1CC(F)(F)C1)NC=O)NC1CCN(CCCOC)CC1 55399,Cc1ccc(NC(C2C3CC3CN2C(=O)Cn2c(C)ccc2C)=O)cc1F 55400,c1(CC(=O)N(C2CCN(C(=O)C#CC3CCCO3)C2)CC)cccc2sccc12 55401,C1(NC(c2n(CCC)ccc2)=O)CCN(C(c2cn[nH]c2)=O)C1(C)C 55402,N1(C(c2c(C)cno2)=O)CCC2(C1)CN(C(c1nc(C(=O)N(C)C)no1)=O)C2 55403,CC(=O)CCCC(C)C(=O)NC(CC(=O)N1CCCC(F)C1)CC(C)C 55404,CC1(C)COc2cc(C(=O)Nc3ncc(-c4cncc(F)c4)s3)nn2C1 55405,CCC(CC)C(C(=O)N1CC(C(C(N2CC([N+](=O)[O-])C2)=O)OC)C1)OC 55406,N1(C(c2ccc(C(C)C)o2)=O)CCCC(C)(CNC(c2cnc(O)cc2O)=O)C1 55407,Cc1cc(CN(c2nnnn2CC2CCSC2)C)cc(C)c1Br 55408,C#CC(C)(C)C(=O)NC1(CNC(c2nnc(C(C)C)s2)=O)CC1 55409,C1(C(=O)NCC(CC(=O)N(CCCO)CC)O)CC2C(C1)C2(C)C 55410,N1(C(CCC2CC(C)C2)=O)CCCC(CO)(CNC(=O)CS(C)(=O)=O)C1 55411,C(=O)(C(C)(C)CCCNC(C1CCC(=O)C1)=O)NCC(n1ccnn1)C 55412,C1(CC(=O)NC)CN(C(C2CCC2(C)C)=O)CCN1C(C1CCC=CCC1)=O 55413,C#CC(CNC(=O)C(Cn1cncn1)NC(=O)CN1CC(C)(C)C1)CC(C)(C)C 55414,n1(CC)nc(C2CC2)cc1C(N1CC(NC(=O)CCCc2cccs2)C1)=O 55415,C(=O)(C(O)P(C)(C)=O)N(CCCNC(=O)CCCc1cncs1)C 55416,c1(C(C)(C)C)ccc(CNc2ncccc2Br)cc1 55417,N1(C(=O)NCC(N2CCCCCC2)C)C2CCCC1CN(C)C2 55418,CC(C)CC(N)C(=O)N(c1ccnc(C(C)C)n1)C1CNCCOC1 55419,C1(C(N2CC(C(C)(C)O)(CNC(C3(SC)CCC3)=O)C2)=O)CC2(C1)CC(F)C2 55420,Cc1ccc2nc(C(=O)NC3CN(C(=O)CS(C)(=O)=O)CCC3CO)cn2c1 55421,c1(C(N(C(C)C)Cc2cccc(C)c2C)=O)ccc2c(c1)OC(C)C2 55422,Cc1nccc(C(=O)NCC2(C)CCCN2C(=O)Cc2ccc(F)cc2Cl)c1N 55423,C12(C(=O)NCC(c3ccc(O)cc3)N(C(=O)C(Cl)=CCl)C)CC3CC1C2C3 55424,CC1(CNC(c2cnc(C3CC3)s2)=O)CCCN1C(C1CC1C(N)=O)=O 55425,C#CCC(CC#C)C(=O)NCCCC(CCC)NC(c1csc2c1CCCC2)=O 55426,C1(NC(CC(=O)OC(C)(C)C)=O)CC=C(C(=O)NCc2occ3c2CCC3)C1 55427,CC#CCCC(=O)N(CC(C)(C)CNC(c1cncnc1C1CC1)=O)CC 55428,c1(SC)cncc(C(=O)NC2CC(NC(=O)C=CC3CCOC3)C2)c1 55429,N1(C(C2(C)CS(=O)(=O)C2)=O)CCC(C2CCN(C(=O)CC#N)C2)C1 55430,C1(NC(=O)CCN(C(c2scnc2Cl)=O)CC2CC2)CN2CCC1CC2 55431,N1(C(CCC=CCC=C)=O)CCC(C)(NC(=O)C(C)CC2CCC2)C1 55432,n1(CC(N2CC3C(NC(c4ccnc(C)c4N)=O)(C3)C2)=O)cnc2c1CCCC2 55433,C(C)(CCCC(=O)N(C)CC1(O)CCCCC1)NC(COC(C)=O)=O 55434,C1(C(=O)NC(CCC2N(C(COC)=O)CCCC2)(C)C)(CF)CC2(CCC2)C1 55435,c1(NC(C(C(C)C)NC(C(CCC)NC(N)=O)=O)=O)cc(C#N)ccc1O 55436,N1(C(c2c(C)ocn2)=O)CCN(C(c2csc(CC(F)(F)F)n2)=O)CC1 55437,S(=O)(=O)(c1cccc(=NC2CCC=CCCC2)[nH]1)NC1CN(C)C2(C1)CCOCC2 55438,c1(C(N2CCC(CC=C)(CNC(=O)C(F)(F)C(C)O)C2)=O)cc(C)c(C#N)cn1 55439,CC1CC(C(N2CC(CN(C)C(C3(C4CC4)CCC3)=O)C2)=O)CCC1C 55440,c1(C(N2CCC(C3N(C(C(F)OC)=O)CCC3)C2)=O)ccc(F)nc1F 55441,C1(C(C)NC(C(C)=C(C)C)=O)CCN(C(c2cc[nH]c2C2CC2)=O)C1 55442,CC(CC(=O)c1cccc(Br)c1)C(=O)NCC(O)(Cc1ccccc1)C1CC1 55443,C1(NC(c2scc(OC)c2)=O)CS(=O)(=O)CC1NC(=O)C=CSC 55444,C(C)(C)(CC(=O)NC1COCC1CO)NC(Cc1ncn(C)c1)=O 55445,N1(C(C(C)OCCCC)=O)CC2(CCC(NC(C3C=C(C)CS3)=O)CC2)C1 55446,S(=O)(=O)(C=Cc1ccccc1)N1CCN(C(=O)C=Cc2ccccc2)C2C1C2 55447,n1(CC=C)ncc2c(O)nc(=NNC(=O)CC3CN(C(=O)C(O)CC[S+](C)C)C3)[nH]c12 55448,C(=O)(NN1CCCC1C(=O)NC1CCC2CC12)c1cc(C(N)=O)[nH]c1 55449,N1(C(C(C)NC(=O)NC)=O)CCCC(CO)(NC(=O)CC2C=CS(=O)(=O)C2)C1 55450,C1(NC(C2C(CC)C2)=O)C=CC(CC(=O)NC2CCCCC2)C1 55451,C1(NC(C2C(NC(CCCC3C(C)C3)=O)CCC2)=O)CCOC1(C)C 55452,C1(C(=O)NCCC2(CNC(=O)COC3CC(F)(F)C3)CC2)CCCCCS1(=O)=O 55453,c1(C(=O)NCCN(C(=O)CC2OCCCO2)CCC)coc(OC)n1 55454,C1(C(=O)NC(C)C(=O)O)CC=CC(n2cc(-c3ccc(F)cc3)nn2)C1 55455,c1(C(=O)NC(C(C)(C)C)CNC(C23CCC2CC3)=O)cc2n(n1)CCCC2=O 55456,C1(CN(C(=O)C(=O)N(C)C)C)CCN(C(C2CC(=C3CC3)C2)=O)C1.C1CN1 55457,C12(NC(C(CC#C)CC#C)=O)CCOCC1CN(C(=O)CS(=O)(=O)CC)C2 55458,CCC(c1ccnc(Cl)c1)=CC(=O)NC(C)CCC(=O)OC 55459,N1(C(C(C)(C)OCC)=O)CCOCC(CNC(c2nc(C)n(C)n2)=O)C1 55460,C=CC1(C(N2CSCC2C(=O)NC(C)CC(C)C(F)F)=O)CCCCC1 55461,N#CC1CN(C(C2(C3CC3)CC2)=O)CCN1C(c1ccc(OCF)cc1)=O 55462,N1(C(CCC=CC)=O)CCCC2(CCC(NC(c3cnnn3C(C)C)=O)C2)C1 55463,c1(CC(C(=O)NC(C(=O)OC(C)C)Cc2ccccc2)N)cccnc1F 55464,c1(NC2CCCCN(C(CC(CC)O)=O)C2)c(Cl)cc([N+](=O)[O-])cc1Cl 55465,C(=O)(CCCCCN=[N+]=[N-])N1C(C(=O)NCCCc2c(C)n[nH]c2)CCC(C)C1 55466,c1(C(N2CCC(CN(C)C)C2)=O)cncc(C(=O)O)n1 55467,C1(CC)C(NC(C2CCC(CC)CC2)=O)CCCN1C(=O)CCn1ccnn1 55468,n1(CC(=O)N(C)CC2CCN(C(C3(COC)CCCC3)=O)C2)ncn(C)c1=O 55469,N1(C(c2c(NC(CC)=O)cccc2)=O)CC(C2CCCCC2)CC1C(=O)O 55470,N1(C(CCC=C)=O)CCC(C(=O)NCC2(c3ccnc(Cl)c3)CC2)CC1 55471,Cc1ccc2c(c1)CCC(C(=O)NCC1CCCCC1NC(c1csnn1)=O)O2 55472,C(=O)(C#CC1CCOCC1)N(CCCNC(=O)CCc1cnn(C)n1)C(C)C 55473,N1(C(C2C(C)CC=CC2)=O)CCC(F)CC1C(=O)NCC1(C#N)CC(C)(C)C1 55474,C(=O)(C(C)CC(C)C)NCCCSCC(=O)N(C)CCOC 55475,CCC(CN(C)C)CC(=O)N1CC(O)(CNC(=O)CCCC(=O)OC)C1 55476,c1(COC)cccc(CC(=O)NC2CCC2CNC(c2cccc(CO)n2)=O)c1 55477,C1(CC)CN(C(c2cc(=O)n(C)o2)=O)CCN1C(C1CCCOCC1)=O 55478,c1(OC)ccc(CNC(=O)NNC(C)Cc2ccccn2)c(F)c1Br 55479,C1(N(C(=O)C(=O)NCCOC(C)(C)C(F)(F)F)C)CCS(=O)(=O)C1 55480,Cc1cc(C(N2CCC3(NC(=O)C(F)C4CCCC4)CC3C2)=O)cc(C)c1O 55481,C1(C(N(CC(C)NC(=O)CNC(N2CCCC2)=O)C)=O)COC(C)CO1 55482,OC1COCCN(N2CCC2C2CCC2)C1.c1ccco1 55483,c1(C(=O)Nc2cc(C)c(NC(c3ccnnc3C)=O)cc2)ccn2cncc2c1 55484,C(CCC(=O)NC1CC(C)(NC(c2ncsc2Br)=O)C1)OCC=C 55485,O=C(C1=CCOC1)NCC(C1CC1)NC(C1CCSC1)=O 55486,CCCCCCC(CC)C(=O)N1CCCCC1Cn1cc(CNC(N)=O)nn1 55487,c1(C(N2CC3CC3(C(=O)NCCO)C2)=O)cn2c(Cl)cccc2n1 55488,C1(CN(C)C(=O)N(C(C)(C)C)C)CC1C1CC1 55489,c1(OC)nccc2c(C(N3CCCC3CNC(C3CC4(C3)CC4(F)F)=O)=O)c[nH]c12 55490,Nc1ccc(C(=O)NC2CC(CCNC(=O)CC3(N(C)C)CCCC3)C2)c(O)c1 55491,c1(C(=O)NCC(CNC(C(COC)(F)F)=O)F)cccc2c1ncn2C 55492,C(=O)(NN1CCCC1C(=O)NC1CC2(CCCCC2)C1)c1cc(CCC)[nH]n1 55493,c1(OC)cc(C)c(C(=O)NC2COCC2NC(c2ccc(Cl)cc2C)=O)cn1 55494,c1(C(=O)NCC2OCC(CNC(C(CC)COC)=O)C2)ccc(N(C)C)c(F)c1 55495,C1(C)(CCC)CCCN1C(c1ccc(N(C(c2ccc(C)cc2)=O)CC)nc1)=O 55496,C1(n2cnnn2)(C(=O)NC2(C)CN(C(c3cc(C4CC4)no3)=O)C2)CCOCC1 55497,N1(C(c2c(OC(C)C)n[nH]c2)=O)CC(NC(C23CCCC2C3)=O)C2(CCC2)C1 55498,c1(C(=O)NC(C(CO)NC(C2C(CC)CCC2)=O)C)ccc(C)nc1C 55499,Cc1nccc(C(=O)NC2CC(CNC(C3SCCCS3)=O)C23CCC3)c1C 55500,c1(C(=O)NC(C(C)O)C(=O)N(C)C)cnc(F)c(F)c1 55501,CC1(C(=O)NCC2CCN(C(c3[nH]cnc3C#N)=O)CC2)CC(C2CC2)=NO1 55502,C1(CC)(NC(=O)CN2CCCC2C)CCCN(C(c2ccc(Cl)c(OC)c2)=O)C1 55503,c1(C(=O)NC(CN(C(=O)C=CCF)CC)C)cc2c(OC)cc(OC)cc2[nH]1 55504,CC1(C(=O)NC2(C3CCC3)CC2)CCN(C(=O)C=CCN2CCC2)CC1 55505,N1(Cc2sc(C)c(Br)c2)CCC2(CC1)CN(CC(=O)O)N2CCO 55506,Cc1cc(C)c(C(=O)NC2(C)CN(C(C34COCC3C4)=O)C2)cc1C 55507,N1(C(c2[nH]c(CC)c(Cl)n2)=O)CCC12CN(C(=O)CC(C)(C)C)C2 55508,CC(C)C(C(=O)NC1CCN(C(=O)C=CC2CC2)C1C)Sc1ccccc1Cl 55509,c1(C(=O)NCC2N(C(C(C=C)O)=O)CCN(C)C2)ccc2[nH]ccc2c1F 55510,c1(NC(C)=O)ccc(C(=O)NCC2(O)CC(NC(C3CCC3(F)F)=O)C2)s1 55511,c1(C(=O)NCCC2OCC(C(=O)OC)C2)ccnnc1S 55512,Cc1cc(C(N2CCCC(N(C(=O)C(C)C3=CCCC3)C)C2)=O)cc2nc[nH]c12 55513,c1(C(=O)NC2C(CC)N(C(C)=O)CCC2)c(Cl)ccc(Br)c1F 55514,Cc1[nH]c2ncccc2c1C(=O)NC(CO)C(C)NC(=O)CC1(C)CCCC1 55515,C(=O)(C1=CCCCC1)NC(C1CCN(C(c2ccc(CCCC#N)cc2)=O)C1)C 55516,C(=O)(C1=CC=CN2CCS(=O)(=O)N=C12)NCC(C)(CO)NC(=O)CCC(N)=O 55517,N1(CCN(C(=O)CC2CC=CCN2C)C)CCN(C(c2ccns2)=O)CC1 55518,C1(NC(Cc2ccc(CCC)cc2)=O)CCC(C)N(C(C2C(C#N)C2(C)C)=O)C1 55519,C(=O)(CC(C)n1ccc(C)n1)NCCCN(C(=O)C=Cc1cocn1)CC 55520,CCCCCC(CCCCC)C(=O)NC1CC(NC(c2cc(C#N)oc2C)=O)C1 55521,Cc1cc(Br)c(N)cc1C(=O)NCCN(C(=O)CCCC(F)(F)F)C 55522,c1(C(=O)NC(CCNC(c2cn(C)[nH]c2=N)=O)(C)C)cccc2nsnc12 55523,N1(C(c2ccc(C(N)=O)s2)=O)CCC2(CC1)CC(NC(C1C3CC4C(C3)C14)=O)C2 55524,c1(C(=O)NC2(C)CC(NC(=O)CC3(C(F)F)CC3)C2)ccc2c(c1)C(=O)C(=O)N2 55525,C1(=CC(=O)NCC2CC2NC(=O)CCc2cc(Cl)cs2)CN2CCC1CC2 55526,c1(C(N2C(CNC(=O)C(O)C3CC3)CCC2)=O)cnn2cccc(Cl)c12 55527,N1(C(c2cc(C)[nH]c2)=O)CCN(C(=O)CC(C)C(F)(F)F)CCC1C 55528,c1(C(=O)NCC(CNC(c2ncc(C)cn2)=O)O)c(N)sc2ccccc12 55529,c1(C(N2C3CC(CC(NC(CSCCC)=O)C3)C2)=O)ccc2n[nH]cc2c1Cl 55530,c1(NC(CC)C(=O)N(C)CC2(NC(=O)C(N)=O)CC2)cccnc1Cl 55531,C(=O)(C1=CCN(C(c2cnnc(O)c2)=O)C1)NC(C(C)C)CO 55532,N#Cc1ccc(C(=O)NCC#CC(N2CCCCCC2C(N)=O)=O)nc1 55533,Cn1cc(C(=O)NC2CCCCC2CNC(=O)C(C)(C)c2cscn2)n(C)c1=O 55534,c1(CC(=O)NC2(COC)CCN(C(C3(C)CC(C)(C)C3)=O)C2)ccc(C#N)cc1 55535,C1(C(N(CC(C(=O)OC)C)C)=O)CC(C)(C)CN1C(c1cc(C)c(F)cn1)=O 55536,N1(C(CCOCC#C)=O)CCC(C)C(N(C(=O)Cc2csc(C)n2)CC)C1C 55537,CC(C)CC(C(=O)NCC1(C)CN(C(=O)CC2CCOCC2)CC1C)C1CCC1 55538,C(=O)(C1=CC2CCCCCC12)NC1(CO)CN(C(CN(C(=O)OC)C)=O)C1 55539,N(C(=NCCCSC)NCC1CC(=O)N(CC)C1)Cc1ccc(OCCC)cc1 55540,C(=O)(C(CC(C)C)n1ccnc1)NC(CC=C)CNC(C1(CN(C)C)CC1)=O 55541,c1(C(=O)NC2CCC(CNC(C3(C)CC4CCC3O4)=O)C2)ccc(Cl)c(N)c1Cl 55542,c1(C(N2C(CNC(CC(C)P(C)(C)=O)=O)CC2)=O)cc2c(cn1)COCC2 55543,CCCCC(C(=O)N=c1cc(C)n(CC(F)(F)F)[nH]1)C1CCC1 55544,C1(OC)CC1C1CCN(C(C2(C#N)CCN(C(=O)OC(C)(C)C)CC2)=O)CC1 55545,Cc1nc(C(N2CCOC(CNC(=O)CC3CCC(F)(F)C3)C2)=O)[nH]c1C 55546,C1(CCC)(CO)CCN(C(=O)C=CC(C)NC(=O)C(C)C2CCC2)C1 55547,c1(C(=O)NCC2N(C(c3c(C)coc3)=O)CCC2)ccc([N+](=O)[O-])cc1Br 55548,c1(CNC(C(C)n2ccnn2)=O)ccc(C(=O)N(C)Cc2cnco2)s1 55549,Cc1ccc(C)c(OCCCNC(c2ccc(N)cc2Br)=O)c1 55550,Cc1onc(Br)c1C(N1CC(CNC(c2ccc(O)nn2)=O)C(C)C1)=O 55551,c1(C(=O)NCCC)cccc(NC(=O)NCC(n2cccn2)O)c1 55552,c1(C(N2CC(CC(=O)N(CCF)CC)OCC2)=O)ccn2ccnc2c1 55553,Cc1cc(C(=O)NCC2CC(NC(c3cc(Cl)sc3Cl)=O)C(O)C2)cn(C)c1=O 55554,C(=O)(CCC(C)(C)[N+](=O)[O-])NC1C(CNC(CN(CC(C)(C)C)C)=O)C1 55555,C1(NC(CN(C)CC)=O)CC2(CCCN(C(C3CCCC(=O)N3)=O)C2)C1 55556,N1(C(C(c2ccccc2)C)=O)CCOCC1(C)c1cn(CCCCCO)nn1 55557,C(=O)(C(CO)C(C)(C)C)NCCCN(CCC)C(c1ccc(CC(C)C)s1)=O 55558,S(=O)(=O)(C(F)(F)F)CCC(N1CC(C2CCCO2)(OC)C1)=O 55559,c1(Nc2n(C)c(Br)cn2)nc2c(c(=NCCS(C)=O)[nH]1)CSC2 55560,c1(CCC=C)ccc(C(=O)NCCN(C(C2(c3ccc(F)cn3)CC2)=O)CC)cc1 55561,N1(CC(=O)Nc2ccc(C=CC(=O)OCC)cc2)C2CCC1CC(SC(C)C)C2 55562,C12(C(=O)OC)CCC(CC1)N(C(c1cc(-c3ccccc3)co1)=O)C2 55563,C1(C(=O)NC2CCC(N(C)C(c3cnsn3)=O)CC2)OCC2CCCC1C2 55564,C1(NC(C(=O)NCC2(OC)CCC(C)C2)=O)CC(C)NC(C)C1.C1CCO1 55565,c1(OC)cc(C)cc(-c2cccnc2C(N2CCC(N(C)C)C2)=O)c1F 55566,c1(CCC(=O)NCC(CC)NC(C2CCC(C(F)(F)F)O2)=O)c(F)cccc1F 55567,CC1(C)CC(NC(C2CC2)C2CC2)CC(C)(C)C1.C(=O)(CCCC1CC1)O 55568,Cc1cc(C(=O)NC(C(=O)N2CC(C(F)(F)F)C2)C2CCOC2)nn1C 55569,Cc1ncc2c(n1)CN(C(=O)OC(C)(C)C)C2C(=O)Nc1cnccn1 55570,N1(C(c2c(COC)cccn2)=O)CCC(C(=O)NCCNCCO)C(O)C1 55571,C12(C(=O)NC(C3CCN(C(c4cc(F)ccc4O)=O)C3)C)CCCCN1CCC2 55572,CC1CC(NC(C2(C)CC2(F)F)=O)CCN1C(c1coc(O)n1)=O 55573,C1(C(=O)NCc2ccc(C#N)cn2)CN(C(=O)CCCC2CC2)CC12CCC2 55574,N12CC3(CCC1C3)C(=O)NCCCNC2=O.c1(C=O)cscn1.CC(C)(C)O 55575,C(=O)(C1CC=Cc2ccccc21)NC1CC(NC(COC(C)(C)C(F)(F)F)=O)C1 55576,C(=O)(CCCC(C)(C)C#N)OC.C1(=O)C(C(C)C)NC(=O)OCC(OC)CN1 55577,c1(C(=O)NC2CCN(C(c3c[nH]cc3C3CC3)=O)CC2O)cc2ncccn2n1 55578,CCCC(C(F)(F)F)NC(=O)CNC(C(CC1CCCC1)Cc1ccncc1)=O 55579,CN1CCN(C(=O)NC2CCC(N3CCOCC3)C2)CC1CC1CC1 55580,n1(CCNC(C(C2CC2)SC)=O)ccc(C(=O)NC(c2nncn2C)CO)c1 55581,N1(C(c2cccc(OC)c2N)=O)CCC(NC(=O)C(C)CC(N)=O)C12CCCC2 55582,C(CCC(=O)N1CCCC1CC(N1CC(N(C)C)C1)=O)NC(C)=O 55583,C1(C(N(CCCCC)CC#C)=O)CC(NC(=O)CNC(=O)OCC=C)C(O)C1 55584,N1(C(C=C(C)C)=O)CC(NC(C2CCOC2c2cccnc2)=O)CCC(O)C1 55585,C(c1ccc(O)c(OC)c1)=CC(=O)NC(CC)CNC(c1csnc1Cl)=O 55586,C(=O)(CCCNC(=O)OC)NCCCNC(C(C1CCC1)OCC)=O 55587,CC(CNC(c1cc(C(O)C2CC2)ccn1)=O)CC(=O)NC(C)C(C)C 55588,CCCC(CNC(C1CCN(OC)CC1)=O)C(=O)NCCN1CC(C)(O)C1 55589,C1(C)(C(=O)OC)CCN1C(=O)CC1CCCN1C(=O)C=CCF 55590,c1(NC(CCCC#CC)=O)nc(N(CCCSC(=O)OCC)C)nc(C)c1OC 55591,C1(C)(NC(c2cc(C)ns2)=O)CCN(C(c2cc(CC3CCC3)c[nH]2)=O)C1 55592,C12(C(=O)NCCN(C(Cc3cc(OC)no3)=O)C3CC3)CC=CC(C1)OC2 55593,c1(CCC(=O)NCC(C)NC(=O)C(C)OC2CCCCCC2)nnc(O)nc1O 55594,C(C)(C(=O)NCCC(=O)N1CCCC1)(C(F)(F)F)NC1(CC)CC1 55595,N1(C(CCC2(C)CN(C(c3cc[n+]([O-])cc3)=O)C2)=O)CCC(C)(O)C(O)C1 55596,C1(C(=O)NC2CCC2O)CC12CCN(C(=O)Cc1cn[nH]c1)CC2 55597,CCC(C)(CC)C(=O)N(CCCCNC(=O)CNC(c1ccccn1)=O)C 55598,c1(C(N(CC(CN(C(c2c(C)cncc2)=O)C)O)C)=O)c(Cl)cccc1[N+](=O)[O-] 55599,c1(C(=O)NC(CCNC(c2c(C)nc(C)[nH]2)=O)(C)C)cccc2oc(C)cc12 55600,c1(C(=O)NC2CC(C)(CNC(c3n(CC)ccn3)=O)C2)ccc(F)cc1C 55601,c1(C(=O)NCC2C3CC2N(C(=O)C(O)C(F)(F)F)C3)cc2c(F)c(F)ccc2[nH]1 55602,c1(CNC(=O)CCc2cnc[nH]2)cc2ccccc2[nH]1 55603,C1(NC(CC(C)(C)O)=O)CC2CCC1CC2NC(c1cc(-c2cccs2)[nH]n1)=O 55604,C1(NC(CCC(C)OC)=O)CCCCCC1CNC(=O)CC1(O)CCC1 55605,CCC(CCCC(=O)NCCC(C)(CC)OC)NC(=O)C(C)CC(C)(C)C 55606,C(=O)(C1=NNC(=O)CC1)NCC1CCC(F)(CNC(C=CC(CC)C)=O)CC1 55607,c1(C(=O)NC2C(NC(=O)C=CI)CC2)ccc(Cl)s1 55608,N1(C(C(C)OC)=O)CCCN(C(=O)C(C)CC(=O)c2ccccc2F)CC1 55609,CCC(O)C(C)C(=O)NC(C)(C)CCC(=O)NC1(c2cccnc2)CC1 55610,c1(C(=O)NC2CC(C)(NC(C(C)OC)=O)C2)cccc(C(F)F)c1Cl 55611,C(=O)(C1=CC2(CN(C(C3(C)CC(=O)N(C)C3)=O)C2)OC1)NCCCOC(C)C 55612,N1(C(C(COC)NC(C)=O)=O)CCC2C(CCCN2C(=O)C#CC2CC2)C1 55613,CC1(C)CN(C(=O)C(O)Cc2ccccn2)CCC1NC(c1coc(C#N)c1)=O 55614,CC1(C)CCOC1C(=O)NC1C=CCN(C(c2cnc(-c3ccccc3)s2)=O)C1 55615,CC(C)C(=O)C(=O)Nc1ccc(C2CCOCC2)cc1.C12CCCN(C1)C2=O 55616,N1(C(c2cc(COC)oc2C)=O)CC2CC(NC(=O)C3=CCCC3C)C1C2 55617,C12CCCC(C1)NC2=O.C(CCOCC(=O)N(C)C)NC.C1CO1.CCO.O 55618,N1(C(C2CN(C(CC(CC)O)=O)C(C)(C)C2)=O)CC(O)C(N=[N+]=[N-])C1 55619,C(CS(=O)(=O)CC(=O)NCC(C1CCC1)NC(C1(c2ccno2)CCC1)=O)OC 55620,C(=O)(C(C)(C)C(C)NC(C1CCOC1)=O)Nc1cncc(C)c1 55621,C1(C(N2C(C(N3CC4(CCOC4)C3)=O)CC(C)C2)=O)CC2(CCC2=O)C1 55622,O=C(CCCCCNC(c1ncncc1N)=O)Nc1ccc(F)nc1 55623,C1(C)(CNC(c2ccc(OC)cn2)=O)CN(C(=O)CC2CC2)C(C)(C)C1 55624,C(CCF)(C(=O)NCC1CC1(Cl)Cl)NC(Cc1cn(CC)nn1)=O 55625,C(=O)(C#CC(C)(C)CNC(=O)CC1CCC(C)O1)N1C2CC(OC)C2CC1 55626,CC(C)C(F)C(=O)NC1CCCCC1NC(=O)CCSc1ccccn1 55627,Nc1ccnc(C(=O)NC2CCCC2NC(C2CC2C2CCCO2)=O)c1Cl 55628,c1(C(=O)NC2C(NC(C(C)OCC3CC3)=O)CCC2)cc(F)cc(S(N)(=O)=O)c1 55629,c1(C(=O)NC(CNC(C2(NC(N)=O)CC2)=O)CO)cc2n(n1)CC(F)C2 55630,c1(SC)ncc(C(=O)NCC(C)CNC(c2ccnnc2)=O)s1 55631,CC(C)CC(C)(CNC(=O)CC1CC1)NC(c1ccc(N2CC=CC2)cc1)=O 55632,C#CCCCC(=O)NCCOCC(N1CCCC1C1CCCC1)=O 55633,C1(CNC(C2N(C(C)=O)CCC2)=O)CC2(CO1)CN(C(c1sccc1C)=O)C2 55634,C12(C(=O)NCC(CC=C)NC(C3CC4C=CC3O4)=O)CCC(O)(CC1)CC2 55635,CC(C)CC(C(=O)N1CC(NC(C2(C)CCN(C)C2=O)=O)CC(F)C1)C(N)=O 55636,Cn1c(C(=O)NCCC23CCC2CN(C(=O)Cc2ccns2)C3)cc2ccsc12 55637,N1(C(c2c(C)ocn2)=O)CCC(NC(=O)Cn2cc(CO)nn2)C12CC2 55638,c1(N(C)C)cccc(C(N2CCC2CNC(C2CCN(C)C2=O)=O)=O)n1 55639,N1(C(CC(=C)C)=O)C2CCC1C(F)C(NC(c1nc(Cl)ccc1Cl)=O)C2 55640,C=CCC(C(=O)NCC1CC1CNC(C1CC2(CC2)CO1)=O)C(C)C 55641,c1(OCC(=O)NCCC(C)(C)NC(C(COCC)C)=O)cccc(F)c1F 55642,O=S(=O)(c1cnccc1N1CCCC(c2nncs2)C1)NCc1ccccc1 55643,C(N=c1cc(C)[nH]c(=NCCN2CC(C)CC(C)C2)[nH]1)c1ncc(C)nc1 55644,CC1(CC(=O)NCCCN(CCCNC(=O)CCc2cscn2)C)CCCC1 55645,C1(O)(CC(N2C(CC(C)C)CCC2)=O)CCN(C(C2CCCC2)=O)CC1 55646,CC(C)(C)C(CNC(c1ccc(=N)[nH]c1)=O)C(=O)NC1CCC2(CC2)C1 55647,CCCC(O)C(=O)NC1CC(F)(CNC(=O)CC2CC2)C1 55648,C(=O)(C(F)(F)CCn1cccn1)NCC(=O)NC(C)(C)C 55649,c1(C(N2CCC(OCCNC(C=COCC)=O)C2)=O)cnn2cccc(Br)c12 55650,Cc1cc(CC(=O)NC2CN(C(c3cccnc3C)=O)CC2C)cc(O)n1 55651,C1(NC(C2CCC(C)O2)=O)CC1C1CCCN(C(C2(CO)CC2)=O)C1 55652,c1(CCCC(N2CC(O)(CCNC(CC(C)O)=O)C2)=O)ccc(CN(C)C)cc1 55653,N1(C(C2(CC)CC2(F)F)=O)CCCN(C(=O)CC2CCC2(C)C)CC1 55654,N1(C(C2(C)CCCOC2)=O)CCN(C(c2cc(CF)on2)=O)C(CO)C1 55655,CC(c1cccnc1)=CC(=O)NC1(C)CCN(C(=O)CC(O)CN(C)C)CC1 55656,Cc1ccc(OCC(=O)NCCCC(C)NC(C2(S(C)(=O)=O)CC2)=O)cc1 55657,C1(C(=O)NC(CC)CNC(C2CCSC(C)C2)=O)Cc2ccccc2N1 55658,c1(C(=O)NCC(CC=C)NC(=O)C(C)S(C)(=O)=O)coc2cc(F)ccc12 55659,C(=O)(CC1CCOc2ccccc21)NC(C(=O)OC)Cc1ncccc1C 55660,C(N=c1nc(N2CCCC(F)C2)c2ccc(C)cc2[nH]1)C1CCCN(CC)C1 55661,c1(CC(N2CC(OCCNC(C3C(C)CC=CC3)=O)C2)=O)cnn2ccccc12 55662,C1(C(=O)NC2C(NC(C34CC(C(C)(C)C)(C3)C4)=O)COC2)COC(=O)N1C 55663,N1(C(=O)Nc2c(OC)cc(C(N)=O)cc2)CC2(CCCC2)C1c1ccco1 55664,c1(C(=O)NC(C)(C)C=CC(=O)NCCC23CCCCC2C3)ccc(CO)cn1 55665,Cc1cc(Cl)c(Cl)cc1C(N1CC2CC2(C(=O)Nc2ccnc(O)c2)C1)=O 55666,C1(NC(CC2C(C)C2)=O)CC2(CCN(C(C3(Sc4cccs4)CC3)=O)CC2)C1 55667,CC(C)(C)C(=O)CCC(=O)N1CC(C(=O)NC2CC(=O)N(O)C2)C(C)(C)C1 55668,CC1ON=C(C(=O)NCCOC2CCN(C(c3cc(O)nc(O)c3)=O)C2)C1C 55669,c1(C(N2CCC(F)(n3cc(C4(C)N(C)CCC4)nn3)C2)=O)cnc(N)c(N)c1 55670,C=CC1(CC(=O)N(CC(C)O)CCNC(=O)C(C)CC2CCC2)CCOCC1 55671,C(c1ccccc1)=C(C(=O)NC(COC)CNC(C1(CO)CCCC1)=O)C 55672,C(=O)(CS(=O)(=O)C1CCCC1)NCCCC(C)NC(c1c(OC)csc1)=O 55673,Cc1nc(=N)[nH]c(=NCC(C)N(C)C(c2ccc(F)o2)=O)[nH]1 55674,C(=O)(CC(C)(C)CC(F)F)N(C1CCCC1)C(C1(O)CNC1)C 55675,c1(OC)ncc(CNC2CCC(C(=O)Nc3cnc(C)nc3)C2)cn1 55676,c1(CC)cccc(C(=O)NC2CC23CC(NC(=O)CCNC(=O)CC(C)C)C3)c1 55677,C1(OCC#C)CCCN(C(C2CCC=CC2NC(=O)CC2CCOC2)=O)C1 55678,c1(CC(=O)N(C2CCN(C(=O)C(F)CC3CC3)C2)C)ccn(C(C)(C)C)n1 55679,CC(C)CC(C(=O)NC1CN(C(c2cnn(C)c2C#N)=O)CC1O)NC(N)=O 55680,CC1(C)CN(C(c2ncoc2CNC(=O)CCC2(C)CC2)=O)CC(CO)O1 55681,Cc1nc2cc(C(=O)NCC#CCNC(=O)CC3CC(O)C34CCC4)ccc2o1 55682,c1(C(=O)OCC)ccc(C2CCCCN2C(C2COC(C)C2)=O)n1C 55683,C(=O)(C1(C)CCc2ccccc21)N1CC(F)CC(NC(COCC(=O)OC)=O)C1 55684,CC(O)C(C)(C)C(=O)N1CSCC1C(N1CC2CSCC2C1)=O 55685,C(=O)(C1CCc2nccn21)N1CC2N(C(c3cc(OC)cc(C)n3)=O)C(CC2)C1 55686,C(C(=O)NN1CCCC1C(=O)N(CC1CC1)CC1CC1)c1c(N)cncc1 55687,S(=O)(=O)(c1ccc(Cl)cc1F)NC1C(C#N)CN(C(=O)Cc2cccs2)C1 55688,c1(CCNC(C2OCCN(C(c3ccccc3)=O)CC2)=O)c[nH]c2cc(F)ccc12 55689,C(CCc1ccccc1)(C(F)(F)F)NC(C(n1ccc(C2CC2)n1)C)=O 55690,Nc1cc(F)cnc1C(=O)NC1CC(CCNC(c2sccc2C2CC2)=O)C1 55691,N#Cc1ccsc1C(=O)NCc1ncccc1C(=O)NOCC1CCCCC1 55692,C=CC1CN(C(=O)CCOCCNC(C2CC(C)=NO2)=O)CCO1 55693,C12(NC(Cc3c(C)noc3Cl)=O)CCCC1N(C(=O)C(O)CC(C)(C)C)CCC2 55694,C1(SC)CN(C(=O)Cc2nccn2C)CC1NC(c1ns[nH]c1=O)=O 55695,C(=O)(C1(C)CCn2ccnc21)NCC1(CNC(C=Cc2cn(C)nc2)=O)CC1 55696,c1(C(N(CCNC(CC=CCC)=O)CCC)=O)cc(Cl)cn1CC 55697,N1(C(C2(CC=C)CN(C(=O)CCSC)C2)=O)CCC2(CCC(OC)C2)C1 55698,C1(NC(CCCCCC)=O)CN(C(c2cnn(C)n2)=O)C2(CCOC2)C1 55699,C1(C(N2C(C(=O)NC3C(C(C)(C)C)C3)C(O)CC2)=O)CC2CC(=O)C1O2 55700,CC1(C)CC(NC(=O)CCC2CCCCO2)CN1C(=O)CC1CCCCC1O 55701,C(=O)(C1c2c[nH]nc2CN1C(C1CC12CCCCC2)=O)NC1CC(CC(=O)OC)C1 55702,c1(C(=O)NC2CC(C)(NC(=O)CC3CC=CCC3)C2)cc(F)ccc1F 55703,C=CCCCCC(=O)N(CC(C)N(C)C(C1CCN(CC)CC1)=O)C 55704,C1(C(=O)NCC(C(C)C)NC(C2CCN(C3CCCCC3)C2)=O)CCCC2CC12 55705,c1(C(=O)NCC2C(NC(C(CCSC)O)=O)C2)occ2c1CCOC2 55706,c1(C(=O)NC2C(NC(C=NOC)=O)CC2)cnc2c(c1)NC(=O)CS2 55707,N1(C(C2(C#N)CCCC2)=O)CCC2CCC(C1)N2C(C1CCCS(=O)(=O)N1)=O 55708,C(=O)(CC(C)C(F)(F)F)NCC(C(=O)N(C)Cc1nnc(C)o1)N(C)C 55709,c1(SCC(=O)NC2C(NC(=O)C=Cc3ccccc3)C2)cc(F)ccc1F 55710,N1(C(C(N2CCSCC2)C)=O)CCCOC(CCNC(=O)CC(C)CN(C)C)C1 55711,C=CCCC(C)(C)C(=O)N1CC(CNC(=O)CC(C)N(C)C)C(O)C1 55712,C1(C)(NC(C=CCCC)=O)CCN(C(=O)Cc2c[nH]c(=N)nc2O)CC1 55713,C(=O)(C(O)C(C)(C)C)NC1C(NC(C2C(C(=O)Nc3cc(C)sc3C)C2)=O)C1 55714,c1(C(N2CC3(CCCN(C(C(C)C(F)F)=O)C3)C2)=O)cn(C)c(=O)c2cncn12 55715,c1(C(N2CCC(NC(C3C(CC(C)C)C3)=O)CC(O)C2)=O)ccc(F)c2occc12 55716,N1(C(c2c(OC)nsc2OC)=O)CCC(NC(c2cc(C)no2)=O)CC1C1CC1 55717,CC1c2ccsc2CCN1CCOc1cc(F)ccc1Br 55718,N1(C(C(C(=O)OCC)F)=O)CCN(C(c2cc(COC)on2)=O)C(C(C)(C)C)C1 55719,C(=O)(C1=C(C#N)CCC1)N(C(C)CC(=O)N1CCC(CCCO)C1)C 55720,C12(CNC(CCOC3CN(C(CCC(N)=O)=O)C3)=O)CCCC1OCC2 55721,C12(NC(c3ccc(OC)nn3)=O)CCC(CNC(=O)C(O)C3CCC3)(CC1)OC2 55722,C(=O)(C(=O)C(C)CC)N(CC(=O)NC(COCC)C)CC1CC1 55723,C(C)(C)(CCC(=O)NC1CC2(C1)CC(C)C2)NC(C(c1ccccc1)C)=O 55724,N1(C(CCC2OCC(C)(C)C2)=O)CCOCC(NC(c2cccc(Cl)c2Cl)=O)C1 55725,c1(CC(N2CCC(CCNC(CC(CC)OC)=O)CC2)=O)ccc(OC)cc1F 55726,C(C1=CCCSC1)(c1n(CC(=C)C)nnn1)Nc1ccc(CC)c(Cl)c1.C1CO1 55727,c1(C(N(C)CC2N(C(C3ON=C(CC)C3)=O)CCOC2)=O)ccc2ncnn2c1 55728,S(=O)(=O)(c1ccc(N2CCC(C)C2)cc1Cl)NCc1cccc(OC)n1 55729,C(=O)(CC(C)C(F)F)NCc1c(C(N2CCCC(C(=O)NC)C2)=O)nco1 55730,CC1c2c[nH]nc2CCC1C(=O)NC1CCN(C(=O)C(=O)C(C)(C)C)CC1C 55731,c1(C(N(CC(C)NC(C(C(C)C)OCC)=O)C)=O)ccc(Cl)cc1[N+](=O)[O-] 55732,C(CCC(C)C(=O)N1CCC(OCCNC(C23CC(C(C)=O)(CO2)C3)=O)C1)OC 55733,C(=O)(C1SCc2cccnc21)N1CC(CNC(CN(C)CC)=O)C(F)(F)CC1 55734,c1(OCC(=O)NC2CN(C(=O)Cc3ccon3)C2)ccc2c(c1)CCCC2 55735,C(CC(C(=O)N(C)Cc1ccoc1)NC(c1c[nH]nc1C)=O)OCC 55736,N1(C(COc2cccc(C)c2)=O)CC(NC(=O)CC(C)F)CC(C)C1 55737,c1(OC)ccc(C(=O)NC2CCN(C(c3nc(C)nn3C)=O)CC2C)c(F)n1 55738,C(=O)(C#CC1CCCOC1)N(CC)CC1CCCN(C(=O)CCC(F)(F)F)C1 55739,C1(NC(COC(CC)C)=O)CN(C(=O)CCSC)CC1CC 55740,c1(OC)cc(CC(C)NCC(C)OC(C)(C)C)ccc1O 55741,CCCCC(C(=O)N1CCOC(C(C)NC(c2ccsc2COC)=O)C1)C(C)C 55742,C(=O)(CCC(N)=O)NC1(C(N(C)OCc2ccccc2)=O)CC1 55743,CC1OCCC1C(=O)NC(C1(CNC(c2ccc(CCN(C)C)s2)=O)CC1)C 55744,Cn1ncc2cc(CNc3ccccc3CC(N3C4CCC3COC4)=O)ccc12 55745,N1(C(C2(C(F)(F)F)CCOCC2)=O)CC2CC(C1)C2N=c1[nH]ncs1 55746,N1(C(c2cc(CC)ncn2)=O)C2CCCC1CN(C(C13CCCN1CCC3)=O)C2 55747,N1(C(C(Cc2ccc(OC)cc2)C)=O)CCN(C(=O)C=CCBr)C(C(F)F)C1 55748,c1(CC)c(C(=O)N(C)CC2CCN(C(=O)CNC=O)C2)nnn1C 55749,N1(C(c2cc(COC)no2)=O)C(C(=O)NC(c2cncs2)C)CC2CCCC12 55750,C(C(N=[N+]=[N-])C(=O)N1CC(NC(C2CC2(C)Br)=O)CCC1C)OCC 55751,CN1CCN(C(c2cc(Cl)cs2)=O)C(C(N2CCCC2(C)C(C)(C)C)=O)C1 55752,C(CC(=O)NOCC(F)(F)F)(C(C)OC)NC(C(CC=C)CC=C)=O 55753,c1(NCc2ccccn2)ccc(-c2cncnc2)cc1 55754,Cc1ccc(C(=O)NCC2CCCCN2C(c2cnsc2)=O)c(N)n1 55755,c1(C(=O)NCC2N(c3nccc(OCC)n3)CCOC2)cc(F)cc(Br)c1C 55756,CCCC(CCC)=CC(=O)NCC1(CNC(C2CN(C3CCC3)C2)=O)CC1 55757,CC(C)C1=NOC(C(=O)N(C)CC2(O)CCCN(C(=O)C=CC(C)(C)SC)C2)C1 55758,Cc1ccnc(C(=O)NCC2CCCC(NC(=O)CSCc3ncc[nH]3)C2)n1 55759,C(=O)(C1=CC2C=CC(C1)C2)N1C(C)(C(N2CCC=C(C)C2)=O)CC(O)C1 55760,N1C(=NCCC(C)C)NCC(C)(O)c2cccc(c2)C1.C1(=CCC)CCNC1.SC 55761,C1(NC(c2nc(-c3ccc(C)o3)sc2)=O)CN(C(C2(O)COC2)=O)CC1C(F)F 55762,c1(C(=O)NCCC(CNC(CCc2cc(C)on2)=O)O)cccc(CC#N)c1 55763,C(CCN=c1[nH]c2ccc(Br)cc2s1)OCCNC(C1CC2C=CC1C2)=O 55764,c1(C(=O)NC(CNC(c2c(C(C)C)ncs2)=O)C(C)C)ccc2nnn(O)c2c1 55765,CC1(CNC(c2ncoc2-c2cccs2)=O)CCCN1C(=O)CSS(C)(=O)=O 55766,C#Cc1cnc(C(=O)N(CCC(C)NC(c2cccc(CC)c2F)=O)C)c(C)c1 55767,n1(CC=C)c(SCC2CCCC(C)O2)nnc1-c1cc(C)n(C)n1 55768,c1(NCC(=O)NCc2ccc(N(C3CCCC3)CC)cc2)cccc(F)c1[N+](=O)[O-] 55769,C1(c2nnnn2C)(C(=O)NCCCN(C(C)(C)C)CC)CCCCC1C 55770,c1(CNC(CN(C(c2cc(CC)oc2C)=O)C(C)C)=O)nn(C)c(=O)n1C 55771,c1(C(=O)NC(C(=O)NCC(N2CCCC2)C)c2ccco2)cccc(O)c1F 55772,C12CCN(C1C)C2=O.C1(OC)CCN(C(=O)C(N)=O)CC1 55773,C1(C(=O)NC2CC(NC(c3ccc(C)s3)=O)C23CCC3)Cc2nccnc2C1 55774,C(=O)(C(C)CCCOC)N1C(CC(NOCC(CC)C)=O)CCC1 55775,C1(CNC(CCOCC#C)=O)CC2(CO1)CN(C(=O)C(C)(C)CC=C)C2 55776,C1(CNC(CNC(=O)OC)=O)CCC2(CO1)CC(NC(C1(C)COCCO1)=O)C2 55777,C1(C(N(C)CC2CN(C(CC=CC)=O)C2)=O)CCC(C)C1 55778,C12(CNC(C3CC(C#C)(O)C3)=O)CCCC1N(C(=O)Cc1occc1C)CCC2 55779,c1(OCOC)ccc(C(=O)NC2CC2c2ccc(-n3cnnn3)cc2)cc1 55780,n12nc(nc1-c1ccc(CCC(F)(F)F)nc1)CCC2.c1(COCC)ccccn1.OC 55781,C(CCCC(C)NC(C1CC12CC2)=O)NC(C1(CCOC)CC1)=O 55782,C=C1CON(C(=O)CC2CCN(C(=O)COc3ccc(C)cc3)C2)C1 55783,N1(C(C(COC)(C)O)=O)CC(NC(c2ccc(OCCF)cc2F)=O)CC(O)C1 55784,N1(C(C(=O)NCC(CC(C)C)N)=O)CCc2cc(Cl)ccc2C1 55785,CC1(C)CC(NC(=O)CC2Cc3ccccc3N2)CN1C(C1CNC(=O)C1)=O 55786,C1(NC(C2(COC)COC2)=O)CCCCC1CC(=O)NC1CCC(=O)NC1 55787,N1(C(=O)Cc2ccsc2)CCN(C(N2CCC(c3cc(O)ns3)C2)=O)CC1 55788,C1(C(N(CC(C)O)CCNC(c2ccn(CC(F)F)n2)=O)=O)CC12CC(F)(F)C2 55789,C1(O)(C(C)NC(Cc2n(C(C)C)cnn2)=O)CCN(C(=O)C=CC2CCOC2)C1 55790,CC(CC(=O)N(C)CC1CCCCN1C(C1CCCO1)=O)P(C)(C)=O 55791,CC(C)C(CNC(C12CCC(CC1)C2)=O)C(=O)NC1CCCC(O)C1O 55792,CCCC(CCC)=CC(N1CCC(CNC(=O)Cc2nc[nH]n2)(OC)C1)=O 55793,CC(C)CC(O)CC(=O)NC(C1CCCN1C(=O)CCC1CC1(F)F)C 55794,C1(OC(C)(C)C)CCN(CCNC(C2(F)C(CNC(=O)OC(C)(C)C)C2)=O)CC1 55795,C(=O)(CCCCCO)N1C(C)CC(NC(c2ccc(C(=O)CF)cc2)=O)C1 55796,N#Cc1c[nH]cnc1=NCC1(F)CC(NC(c2ccnc(Cl)c2Cl)=O)C1 55797,C1(CNC(C2(C(F)F)CC(=C)C2)=O)CC2CCC(C1)N2C(=O)CC(C)SC 55798,C1(C(=O)NC)CS(=O)(=O)CCO1.[N+](C)(C)(C)CCN 55799,c1(C(N2C3CC(=C)C(C3)C2)C(=O)NCCOC)cc(OC)c(F)cc1F 55800,N1(C(C(=CC2CCCC2)C)=O)CCCC(CCNC(c2cc(C)ccn2)=O)CC1 55801,c1(C(=O)NCC2N(C(c3c(C)cn(C)c3)=O)CCC2C)cc2c(C)n[nH]c2cn1 55802,C12(C(=O)NCC(CC)NC(c3cc(C(N)=O)n[nH]3)=O)CC(c3ccccc3)(C1)C2 55803,c1(CN2C(C(=O)Nc3ccc(CCO)cc3)CC(F)(F)C2)cc(Br)c(O)cc1O 55804,C#CCC(C)(C)C(=O)N1CCC(COC)(NC(C2CC2CC(C)C)=O)C1 55805,c1(CC(N2C(C)(CNC(C(C)OCCC#C)=O)CCC2)=O)cc(F)cc(Cl)c1 55806,c1(C(N2CCC(NC(CC3CC(=O)NCCC3)=O)C2)=O)ccc(F)c2ccsc12 55807,c1(NCC(C(C)C)O)ccc(S(=O)(=O)NC2CC3OCCCC23)c(Br)c1 55808,N1(C(C(CO)OC)=O)CCN(C(c2cc[nH]c(=N)c2)=O)CC1C1CCC1 55809,C(=O)(CC1CCCc2c1[nH]c1ccccc21)NC1C(C(=O)OC)C2C1CC2 55810,C1(COCC2CCOCC2)CN(C(=O)C(F)=C(C)C)CCN1OC 55811,C1(CC(N2CCCC(Cn3cc(CSCCO)nn3)C2)=O)C=CS(=O)(=O)C1 55812,N1(C(CC(=O)N(C)C)=O)CCCC(O)(CNC(c2ccc(=O)n(C)c2)=O)CC1 55813,C1(OC)CC2CC(C(=O)NCCC(C)(C)CNC(=O)CS(C)(=O)=O)CC12 55814,N1(C(CCN(CC)CC)=O)CCC2CN(C(c3nccc4[nH]ccc34)=O)CC12 55815,C1(C(N2CC(SC)C(NC(=O)CC3CCOC3(C)C)C2)=O)COCC(C)(C)O1 55816,N1(C(COC(CC)C)=O)CCCCC1CN(C)C(c1sc(F)cc1Br)=O 55817,c1(CC)ncoc1C(=O)NCCCOCCNC(C1CC(C(F)(F)F)CO1)=O.OC 55818,c1(C(N2CC(Cn3cc(CC(C)C)nn3)OCC2)=O)cc(C(F)F)cc(Cl)c1 55819,C12CN(CC1CC(C)(C)C)C(=O)C(=O)N2.c1(C(CC2CC2)OC)ccccc1 55820,C1(NC(c2cn(CC)nn2)=O)CC2CC(C1)N(c1ncc(Br)c(O)n1)C2 55821,Cn1cncc1C(=O)NCc1ocnc1C(=O)NCCC1CC1C1CC1 55822,Cc1ccc(C(=O)NC(=O)C(=O)NCC2CCCN(c3ncccn3)C2)c(C)c1 55823,C1(O)(CCNC(=O)C(O)C2CCC2)CN(C(=O)CC2CCOC2=O)C1 55824,C(C(CC(C)C)C(=O)NC(c1cn(C)cn1)C)NC(C(C1CC1)OC)=O 55825,c1(C(=O)NCC(C)N(C(c2cccc(CC)c2)=O)CC)cnc2n1CCC(C)C2 55826,Cc1cnc(CN2CCCC(C(N3CCCC(CCN(C)C)C3)=O)C2)cn1 55827,C(=O)(C1=CCCSC1)NC1C(C(N2CC(CO)CC2CO)=O)CCC1 55828,c1(C(N2CCC(O)(CNC(C3(C#N)CCC3)=O)C2)=O)cc([N+](=O)[O-])ccc1Cl 55829,c1(NC(C2CCC(C)(C)CC2)C(=O)OC)cc(=O)n2cc(Cl)ccc2n1 55830,c1(CN(C2CN(C(C34CC(C(=O)OC)(C3)C4)=O)C2)C)ccc(OC)c(OC)c1 55831,c1(OCC)cncc(NC(=O)C(C)C(C)NC(=O)CSc2nc[nH]n2)c1 55832,CCCCC(O)C(=O)NC(C1CCN(C(c2cccc(CN(C)C)c2)=O)C1)C 55833,C1(CNC(C2CC2C(F)(F)F)=O)COCCN(C(c2cnco2)=O)C1 55834,C(c1cccnc1)=C(C(N1C(CCNC(C(C=CC)O)=O)CCC1)=O)C 55835,c1(C(C(=O)NCCCSC)N(CCC=C)CC)nccc(Cl)c1F 55836,c1(C(C(=O)NC(C)C)N(CC=C)Cc2cccnc2)c(Cl)c(C)nn1C 55837,c1(CC(=O)N(c2cccnc2)CC=C)ccoc1C 55838,c1(C(=O)NCC2CN(C(=O)C(F)(F)CC3CC3)CC2(F)F)cccc2c1CCO2 55839,N1(C(C(c2ccccc2)C)=O)CCC(CCCNC(C2CC2Cl)=O)CC1 55840,C(=O)(C(C)C1=CCCC1)N1CCCCC(N(C(c2cccc(C#C)c2)=O)C)C1 55841,CC(C)CCN=C(NCCF)NCC1C(O)CCN1C(=O)OC(C)(C)C 55842,CCC(C)C(C)NC(C1(C(C)NC(=O)C(C)c2cccs2)CC1)=O 55843,CCC1=NOC(C(=O)NCC2CC(C)N(C(=O)CCc3cnccn3)C2)C1 55844,c12ccc(nc1)c(=O)[nH]2.CCC(C(=O)NCC(C)(O)C1(C)CC1)NC(C)=O 55845,c1(C(=O)NC)cc[nH]n1.C1(=O)CCN1.C1(=O)COCC(=O)NCC(C2CC2)N1C.CN 55846,C(CC(C)C(=O)NC1CC(N(C)C(c2cnc(N3CCOCC3)s2)=O)C1)OC 55847,c1(N2C(=O)CC(C(N3CCC(OC)C3)=O)C2)ccc(Cl)c(F)c1 55848,c1(CC(N2CCC(C(C)NC(C3(CC=C)CCC3)=O)CC2)=O)ccc(F)c(C)c1 55849,CCCCCCC(C)C(=O)NC(CC1CCC1)C(N1CC2CCC(C1)O2)=O 55850,CC(Cc1ccnn1C)C(=O)N1CCC1CNC(=O)CCc1ccccc1 55851,c1(N2CC(C)C(CO)CC2)nc2c(c(=NCCN(C)C)[nH]1)CCCCC2 55852,c1(CNC(C=C2CCC(C)CC2)=O)cc(O)nc(CNC(=O)CC2OCCO2)n1 55853,Cc1ccc2c(c1)C=C(C(=O)NC1CCOC(CNC(C3CC3F)=O)C1)CO2 55854,N1(C(C(CCC)O)=O)CC2CC(C1)CN(C(=O)C(F)C(F)(F)F)C2 55855,C(=O)(C(CC1CCCC1)C(C)C)N1CCC(NC(Cc2c(C)onc2)=O)CC1 55856,C(CC(F)CN=[N+]=[N-])NC(C(CC=CC)NC(C1OC2CCC1C2)=O)=O 55857,c1(OC)[nH]c(=N)ccc1C(N1CCN(C(C)CNC(C2(CO)CCC2)=O)CC1)=O 55858,N1(C(c2cnn(C)n2)=O)CCC(CNC(C2CCN2C2CCCC2)=O)C1(C)C 55859,CC1CN(C(=O)CC(F)F)CC(CCNC(=O)C(c2ccccc2F)(C)C)O1 55860,CCC(C)C(O)C(=O)N1CCCCC1CNC(C1(O)CC1)=O 55861,CC(C)C(CCC(=O)NC(C)(C)CF)NC(=O)Cc1cn(C)cn1 55862,C#CCCC(C(=O)OC)NC(=O)NCc1ccc(CC2CCOC2=O)cc1 55863,c1(C(C)=O)ccc(C)nc1NCC(C)CNC(C1CCOC(C)(C)C1)=O 55864,C1(C(=O)NCCCNC(=O)C(Cc2cccc(Cl)c2)=NO)CCC2CCC(=O)N12 55865,C1(F)(CNC(=O)C=Cc2ncco2)CC2CCC(C1)N2C(=O)CC1CCCCC1 55866,C(=O)(C(F)C(F)(F)F)N(C(CNC(c1cccc(CC)n1)=O)C)CC 55867,C(=O)(C1=NNC(=O)CC1)N(CC(CC)NC(c1ccc(Br)c(N)c1)=O)CC 55868,C=CCC(C(=O)NCCC1(CNC(=O)CN=S(C)(C)=O)CC1)C(C)(C)C 55869,CC1=C(C(=O)N2CC(NC(C3(C)CCCS3(=O)=O)=O)C2)SCCO1 55870,N1(C(C(CC)CO)=O)CCC(NC(C2(O)CCSC2)=O)C(C)C1 55871,[N-]=[N+]=NCC(C(=O)NCCOC1CCCC1)NC(C1CC2(CC2)CO1)=O 55872,c1(C(N2CCC(N(C(c3cnc(C)[nH]3)=O)CC)C2)=O)cnc(OCC(F)F)cn1 55873,N1(C(C(CCC)C)=O)CCC2(CC1)CN(C(C1C=C1C)=O)C2C(C)C 55874,c1(OC)ccccc1CC(=O)N1CCC1CNC(c1oncc1C)=O 55875,c1(CC)cc(C(N2CCC(=CCNC(=O)C(C)SC(C)C)CC2)=O)c(C)nn1 55876,CCC(CC)C(=O)NCC1CC(NC(c2cncc(C(=O)OC(C)(C)C)c2)=O)C1 55877,C1(C(=O)NC2CC(C#C)C2)COCCN1C(c1cnn(C(C)C)c1)=O 55878,C1(CC=C)(NC(c2cnn(C3CC3(F)F)c2)=O)CCN(C(C2CCSC2)=O)C1 55879,N1(C(C2C(=C)CC2)=O)CCC2CN(C(C3(n4cc(Br)cn4)CC3)=O)CC12 55880,c1(C(=O)NC2CN(C(C3(C(C)(C)C)CCC3)=O)CC2F)ccc(=O)n(CCF)n1 55881,CC1(C)CC(c2nnnn2C2CC2)(NC2CC3CCC2O3)CCO1 55882,C(CCCCC(=O)N1CC2CC(C1)C2NC(c1ncc(N)cc1Cl)=O)OC 55883,N1(C(c2cc(CCC)on2)=O)CC2CCC2(CNC(=O)CC23COCC(C2)C3)C1 55884,CC1(C)CCN(C(C2CCN(C(=O)CC3CCC(=O)N3)CC2)=O)CC1 55885,c1(CC(=O)N(C)CCNC(C2(Cc3cc[nH]c3)CC2)=O)ccc([N+](=O)[O-])cc1Cl 55886,C(C(=O)N1OC2CCC1CC2)N1CCN(C(=O)Cc2ccon2)CC1 55887,Cn1nc(C(N2CC=C(CNC(=O)Cc3cccs3)CC2)=O)c2c1CCSC2 55888,C(=O)(CC(CC)C(C)(C)C)NC(COCC)C(=O)NC1(CF)CC1 55889,CC1(C)C2CCC1(CC(N1CCN(C(=O)C#CC3CC3)CC1C(F)F)=O)CC2 55890,N1(C(C(CC)n2ccnc2)=O)CCCCC(CNC(=O)Cc2ccoc2C)C1 55891,c1(NC(C2CC23CCN(C(=O)C=Cc2ccoc2)C3)=O)cc(I)ccc1CO 55892,N1(S(c2cnc(N(C)CC3N(C(C)=O)CCCC3)s2)(=O)=O)CCC(C)C(F)(F)CC1 55893,c1(C(=O)NC2C(C)CN(C(=O)C(c3ccnn3C)O)C2)nnn2c1CSCC2 55894,N1(C(c2ccnc(C)c2C)=O)CCOC2(CCN(C(c3[nH]cnc3C#N)=O)C2)C1 55895,N1(C(C2CCC(N(N3CCOCC3)CC(F)(F)F)CC2)=O)CCCC(CO)CC1 55896,C=CCC(CNC(=O)CCn1cncn1)C(=O)Nc1ccc(O)nc1 55897,c1(CNC2(CC(=O)Nc3ccnc(Cl)c3I)CCC2)c(Cl)[nH]c2ccccc12 55898,C1(C(N2CCC(CC(C)C)CC2)=O)CC2(CC2)CN1C(C1CC(OC2CC2)C1)=O 55899,c1(C(=O)NCC2CC(OC)CN2C(c2cnccc2Cl)=O)ccc(=O)n(C)n1 55900,CC(C)CCCC(=O)N1CC(O)CCC1C(=O)NCc1cccnn1 55901,Cc1cc(C(=O)NC2CC2C(=O)NCCOc2ccc(Br)cc2)c(C)n1C 55902,c1(C(=O)NC(C(C)C)(C)CNC(C2(O)CC2)=O)ccn2cnnc2c1 55903,c1(NC(=O)NCc2noc3c2CC(C)CC3)cc2c(cc1O)OCO2 55904,c1(NC(c2nc(C)sc2)C)nc(N2CCc3sccc3C2)nc2sccc12 55905,C(=O)(CCCCC(N)=O)NC1CCCC(NC(COc2c(C)cccc2Cl)=O)C1 55906,C(C(CC(F)(F)F)NC(C1(CC)CC1(F)F)=O)NC(c1cnc(OCC)nc1)=O 55907,C(C)(CNC(c1cnc(C(C)C)s1)=O)(CO)NC(C(C)OCCC(C)C)=O 55908,Cc1coc(C)c1C(=O)NC(C)(CNC(C1CCC(C)O1)=O)C1CC1 55909,c1(C(=O)NCC(CNC(CCC=CC)=O)CO)cnn(C(C)CC)c1C 55910,c1(OCC)nc(C(=O)NC(CNC(c2ccn(C3CCOCC3)n2)=O)CC)ns1 55911,c1(CCC(=O)NC(C2CN(C(CCNC(=O)NC)=O)C2)C)cccc(F)c1 55912,c1(CC)cc(Cl)ccc1NC(=O)N(C(C)(C)CC)C(c1cccc(Cl)c1)C 55913,N1(C(C(CC)(C)OC)=O)CCC(C2CCN(C(=O)Cc3c(C)noc3C)C2)CC1 55914,C1(F)(NC(C2C(CNC(CCCCOCC)=O)CCO2)=O)CCCCCC1 55915,C12(C(N3CCC(COC)CC3)=O)CC(CO1)N(C(=O)C=CC(F)(F)F)C2 55916,C(=O)(CCC(C)CN(C)C)NC(C(N1C(C)(C(=O)OC)CCC1)=O)C 55917,CC1(C)CCCN(C(c2cncs2)=O)C1C(=O)NC(CCO)C1CC1 55918,C#CCCN=C(NCCc1cnccn1)NCC1CCCOC1 55919,c1(C(N2C(CNC(C3(C)CCOC3)=O)CC2)=O)ccc(Cl)cc1C(N)=O 55920,C1(C2CC2)(C(N2CCC(NC(c3sccc3F)=O)CC2)=O)CC=CC1 55921,c1(C(=O)NCC2(CCNC(CC)=O)CC2)cccc(C2(S(C)(=O)=O)CC2)c1 55922,C(=O)(C(CNC(=O)CCC1CC1(F)F)CC(C)C)NCCc1ccc(C)s1 55923,C(=O)(C(CO)C(C)(C)C)NC(CCC)C(=O)NCC1(C)CCCC1O 55924,N1(C(C(=O)Nc2cccc(C)c2)=O)CCN(C(c2cnc(C)n2C)=O)C(C)C1C 55925,Cc1cc(F)ccc1CCNC(c1ccncc1)(c1nnnn1C1CCC1)C 55926,c1(C(=O)NCC2CN(C(c3cocn3)=O)CCCO2)cccc(C#CCO)c1 55927,C12(CC(=O)NCC(C)N(C(=O)Cc3cnns3)CC)CCCC1CCC2 55928,c1(CNC(=O)Cc2cnoc2)ccnc(C(=O)NC2CCS(=O)CC2)c1 55929,C(CN=C(NCCN1CCCC(C)C1)NCCSC)=CCC 55930,N1(C(C(C)n2cncn2)=O)CCOCC1CN(C)C(c1nccnc1C(N)=O)=O 55931,c1(NCC(C)S(N)(=O)=O)ccc(S(=O)(=O)N2CCC(c3ccc(Cl)s3)C2)cc1Cl 55932,O=C1CN(CC2CC2(Cl)Cl)C(=O)N1CCC1(C(F)(F)F)CC1 55933,CC(C)C(C(=O)NCC(C(C)C)NC(=O)COc1cnn(C)c1)NS(C)(=O)=O 55934,C1(CCNC(C(C=C)(C)O)=O)CN(C(=O)C(C)OC2CCOC2)CCCO1 55935,N1(C(CC(=C=C)C)=O)CC2(CCN2C(c2ccc(OC(C)=O)cc2)=O)C1 55936,C1(CCN(C(C(Cn2ccc(C)n2)C)=O)C)CCN(C(=O)CSCC(N)=O)CC1 55937,CCC(C)CC(C)C(=O)N(C(C)CN1CCCCC1)CC 55938,c1(NC2C=CC(C(=O)NCc3ccc(C)c(Cl)c3)C2)ccnc2ccnn12 55939,N1(C(C(Cc2ccc(C)cc2)NC=O)=O)CCCN(C(C2C=CCC2)=O)CC1 55940,N1(C(c2c(C)cn(C)c2)=O)CCCC(O)(CCNC(=O)C=C2CCC(C)C2)C1 55941,C12(CNC(c3ccc(C#C)o3)=O)CCCC1CN(C(=O)C(F)(F)CCC=C)C2 55942,C(N=c1ccnc(NC2CCC2C2CC(C)(C)CCO2)[nH]1)c1ccc(C)c(Br)c1 55943,C1(C#N)(C(=O)NC2CC(CCNC(C(CC)N(C)C)=O)C2)CCSCC1 55944,c1(C(=O)OC)ccc2c(c1)CC(O)CN2Cc1nnc(-c2cccnc2)s1 55945,C(N=c1[nH]cnc2[nH]cc(C(F)F)c12)C1CCCN(C(c2ccc(F)s2)=O)C1 55946,C=C=CC(C)C(=O)N1CCC(OCCNC(C2CCC(=O)N2CC)=O)C1 55947,Cc1nn(CC(=O)NC2CC(NC(=O)C(C)CN(C)C)C(O)C2)c(C)c1[N+](=O)[O-] 55948,c1(NC2C(C)COCC2)[nH]c(=NCc2sncc2Br)nc2c1ncn2C 55949,c1(C(N2CCCC(CCNC(CC(C)F)=O)C2)=O)ccn2ncccc12 55950,CC(C)(CNC(=O)CC1CCC1)CC1CN(C(c2cnc(C(F)(F)F)s2)=O)C1 55951,CCCCCC(=O)NC1COCCC1NC(c1cnc(C2CC2)[nH]1)=O 55952,C1(CNC(C(C)OCCC=C)=O)CCN(C(c2ccc(CC)[nH]2)=O)C(C)C1 55953,c1(CCNC(=O)Nc2cn(CC(=O)OC)nn2)cccnc1O 55954,C1(CC=C)(NC(c2cnn(C)c2OC)=O)CCN(C(=O)CC2CC2C)C1 55955,C(=O)(C1=NOC(C)C1C)NC(C1N(C(c2ccc(OC)cc2OC)=O)CCC1)C 55956,C(CC(C)(C)C)(C(=O)NCCC1CC(C(=O)N(C)Cc2cn(C)cn2)C1)OC 55957,c1(C(N(C)Cc2ccc(C)cc2Br)=O)n[nH]c2cccc(F)c12 55958,C1(NC(CCc2cn(C)nc2)=O)CN(C(C2CCCS(=O)(=O)C2)=O)CCC1F 55959,Cc1ccc(C=CC(N2CCC(NC(=O)CC3(C)CCCO3)CC2)=O)s1 55960,C(CN=c1[nH]c(=NC2CCC(C3CC3)CC2)[nH]c2c1SCC2)OCCOC 55961,C1(C(N(CCC(C)NC(c2ccnc(OC)n2)=O)C)=O)COc2ccccc2O1 55962,CN1C(=O)CCC1CC(=O)NC1CC(CC(=O)NCC(F)F)C1 55963,CC(C(=O)N1CCCC(NC(c2cnc(N)c(CO)c2)=O)C1)C(C)(F)F 55964,C(C(=O)NCCCN(C(=O)CO)C(C)C)(C1CC1)SC 55965,C1(C)(C(N2CC(C(C)NC(c3ccc(CO)nc3)=O)C2)=O)CC(C2CC2)=NO1 55966,N1(C(C(CC=C)C(=C)C)=O)CCC2(CCC2C(=O)NCc2cc(Cl)ccn2)CC1 55967,C(=O)(CC(O)CC(C)(C)C)NC1CCC(NC(C(C(C)C)n2cncn2)=O)CC1 55968,Cc1c(C(=O)NC(C)C(C)CN(C)C)ccn1CCO 55969,c1(C(N2C(CNC(CC(C)N(C)C)=O)CC3(CC3)C2)=O)cccc2nccn12 55970,C1(NC(c2c(C)cc[nH]2)=O)CN(C(=O)Cc2ccccc2CS(N)(=O)=O)CC1O 55971,N1(CC)CCOC(C)(CNC(=O)CC(c2cccs2)NC(C2(Br)CC2)=O)C1 55972,N1(CC(=O)NCCCCC2CN(C(Cc3c(C)ncs3)=O)C2)CCN(C)C(=O)C1 55973,N1(C(C(COC)C)=O)CC2(CCN(C(=O)C(C)Cc3ccncc3)CC2)C1 55974,N1(C(c2cccc(C(=O)OC)c2)=O)CCC(C)(CNc2ccc(I)cc2Br)CC1 55975,c1(CCC(C)=O)nc(-c2ccnc(N3CCCCC3)c2)nn1CC(C)O 55976,C(C)(C(CC(=O)NCCC(C(C)C)OC)NC(C1CN2CCC1CC2)=O)OC 55977,Cc1cnc(CC(=O)N(C2CCN(C(C3CCSC3)=O)C2)CCO)s1 55978,N1(C(C2CC=C(C)CC2)=O)CCCC(CCNC(=O)C=CC(C)C)CC1 55979,C1(CNC(CSCCOC)=O)CC2(CC(NC(=O)C(c3c(C)n[nH]c3C)C)C2)C1 55980,C1(C(C)NC(=O)C(F)Cc2ccccc2)CN(C(c2cnoc2)=O)CCO1 55981,C(CC(C(=O)NCCC(C1CC1)C1CC1)NC(=O)CSC(C)(C)C)OC 55982,Cc1c(C(N2CCOC(CC(=O)N(C3CN4CCC3CC4)C)C2)=O)c[nH]c1C#N 55983,Cc1c(C(N2CCC(CN(C(=O)C(C)NC(C)(C)C)C)C2)=O)sc(Cl)c1Cl 55984,C1(C(=O)NC(CC)CSC)CN(C(c2ccc(CO)cc2)=O)CC(C)(C)C1 55985,C1(O)(C(CNC(COCCC#C)=O)C)CCN(C(c2nocc2C(C)(C)C)=O)C1 55986,c1(C(=O)NCCN(C(C2CC3OC(=O)OC3C2)=O)CC)nn(C)c2c1CCC2 55987,C1(NC(c2occ(C)c2)=O)CCCCC12CCN(C(c1cnc(F)c(C)c1)=O)C2 55988,C(=O)(C1=NOC(C)C1C)NCC(C)NC(C1(C(C)C)CCC1)=O 55989,N1(C(c2c(C)nc(O)cc2)=O)CC(CNC(=O)C(C)n2cnnn2)CC(C)(C)C1 55990,C1(NC(C(C)NC(N)=O)=O)CCC(N(C(=O)Cn2cnc(Br)n2)C)CC1 55991,N#Cc1ccc(CN2CCOC(NC(=O)NCCCCl)C2)c(Br)c1 55992,c1(N2CCC(CCNC(c3cc(O)ncn3)=O)CC2)nc2ccccc2o1 55993,N1(C(c2ccc(C)c(C)c2)=O)CCC(NC(c2cnc[nH]2)=O)C(CO)CC1 55994,C1(NC(c2n(CC)nc(C)c2)=O)C2CCC1N(C(=O)CN1CC3CC3C1)C2 55995,CN1CC(C(=O)NC2(C(=O)NCC3(CO)CCCCC3)CCSC2)CCC1=O 55996,N1(C(C(C)(C)OC)=O)CCCC(CCNC(c2ccc(C)nn2)=O)CC1 55997,c1(C(=O)NCCC(=C)CNC(C2CCC(C)=C(C)C2)=O)cccc(O)c1F 55998,C1(CNC(C(CC)NC(C)=O)=O)C2CN(Cc3ncsc3Br)CC12 55999,N1(C(c2ccnc(OC)n2)=O)CCC(C)N(C(c2ccncc2O)=O)CC1 56000,c1(C(N(C(CNC(c2cc(C(=O)OC)no2)=O)C)C)=O)noc2c1COCC2 56001,C1(CC(=O)NC(CCC)CO)CN(C(=O)Cc2ccsc2)CCC1C 56002,C(=O)(CC(CCC)NC(C1(C2(C)CC2)CC1)=O)N1CCC(C=C)C1 56003,C1(C(=O)NCCC(C)N2CCCC2)(CC)CCN(C(C2CC2C(F)(F)F)=O)C1 56004,C1(C(F)(F)F)(C(N2CC(CC(C)NC(=O)CCc3cncs3)C2)=O)CCCC1 56005,C1(CO)CN(N2CC3CCCC(C3)C2)CC12CCOCC2 56006,N1(C(C2(C)CC(C)(C)C2)=O)CCN(C(C2C=CCCC2)=O)C(CC(F)(F)F)C1 56007,c1(C(=O)NCc2cn(CCNC(CC=CC=C)=O)nn2)ccccc1C 56008,N1(C(C(=O)N(C)C)=O)CC2(NC(c3cnco3)=O)CC1C2 56009,n1(CC)ccc(C(=O)NC(CNC(C2(CC(C)C)CCC2)=O)CC(C)C)cc1=O 56010,C1(NC(CC2CC(C)NC2)=O)CCC2(CCC2)C1 56011,n1(CC)cnc(C(=O)NC2CCCC2CNC(C23CCC2C3)=O)c1 56012,N(C=CC(=O)C(F)(F)F)C(=O)CC1CN(C(c2cccc(Cl)c2O)=O)CCO1 56013,C12(CNC3(n4cc(-c5c(C)ccc(N)c5)nn4)CC3)CCC(C(=O)O)(CC1)CO2 56014,c1(C(=O)OC)cnc2ccccc2c1N1CCC(C(=O)NCc2nccs2)CC1 56015,C1(NC(C2CCC3(CC2)CC3)=O)CS(=O)(=O)C12CCN(C(=O)CCC(F)F)CC2 56016,CC1(C)C(C(F)F)CCN1C(c1cc(C(F)F)ncn1)=O 56017,N1(C(C(COCC)C)=O)CCN(CC(=O)NCCCC(O)CO)CC1 56018,N1(CC(=O)NC(C(C)C)CNC(=O)CCC2CCC(=O)N2)CCS(=O)(=O)CC1 56019,CCCCC(C)(F)C(=O)N1CC2CCCC2(NC(c2cccc(C)n2)=O)C1 56020,c1(-c2cc(N(CC)CC)ncc2)c[nH]c2cc(C(=O)NCCSC)ccc12 56021,C(=O)(C(C)S(N)(=O)=O)NC(C1N(C(c2cc(SCC)ncc2)=O)CCC1)C 56022,c1(CC)ccnc(C(N2CCC(C(=O)N(C)CC3(O)CCC3)C2C(C)C)=O)c1 56023,C1(CN(C(C2C(C=C(C)C)C2(C)C)=O)CC)CCCCN1C(c1n[nH]cc1C)=O 56024,CCC(CC(=O)NCC(CO)NC(c1cnc(C2CC2)s1)=O)C1CC1 56025,N1(C2CCN(C(C(C3CCCCC3)=O)=O)C2)CCN(C(=O)CCC2CCC2)CC1 56026,c1(NC(=O)NCCC2COCC2O)ccc(I)c(Br)c1 56027,C=C1CC2CCC(C1)N2C(=O)C(F)C(C)CNC(C1(C(N)=O)CCC1)=O 56028,c1(-c2cc(C)nn2C)ccc2[nH]c(C(=O)NCc3ccncc3)cc2n1 56029,C1(CNC(C2(OC)CCC2)=O)CCN(C(c2cccc(=O)n2C)=O)C12CC2 56030,C1(O)(CNC(CC2(C)CCN2C(=O)CCc2ccc(O)nc2)=O)CCCCCC1 56031,c1(C(N2CCCC(n3cccn3)C2)=O)ccc(-c2ncc(C(F)F)s2)cc1 56032,CC1(C)CC(CNC(=O)C2=COCC2)N(C(=O)CC2(O)CC2)C1 56033,C1(C(=O)NC2(CC=C)CCN(C(c3nsnc3O)=O)C2)C2CCCCCC12 56034,C1(NC(Cc2n(C)ncc2)=O)CC2CCC(C1)N2C(c1c[nH]c2nccc-2c1)=O 56035,c1(O)ccc(C(=O)C(C)C)cc1.C1(=O)CN(CC)CCN1CC.CCCCCC 56036,c1(CN2C(C(=O)Nc3nnc(C)o3)CC(C)C2)c(C)nn(C)c1Cl 56037,C=C(C)CN=C(NCC1COCC(C)(C)O1)N1CCC(F)(F)C(C)C1 56038,C1(CC(=O)NC(CNC(C=CC)=O)C2CC2)CC(=O)c2ccccc2C1 56039,c1(C(=O)NCC23N(C(C=C4CCC(C)C4)=O)CC(C2)C3)cc2c(s1)CCC2 56040,c1(C(=O)NCC(C2CCC2)NC(c2ccc(CC)o2)=O)nccc2n[nH]cc12 56041,C(c1ccc(O)cc1)=CC(=O)NC1(CO)CCN(C(C=CCN(C)CC)=O)C1 56042,C1(NC(C(COC(C)C)NC(c2ccc(CC)o2)=O)=O)COCC1C1CC1 56043,c1(C(=O)NC2CCC(NC(C(CC=CCC)C)=O)CC2)c(C)nn(CC)c1C 56044,C1(CN(C(=O)Cc2cccs2)C)CN(C(=O)CCNC(C2CCC2)=O)CCO1 56045,C(=O)(CC(O)C(C)C)NCC1(OC)CN(C(c2ccnc(-n3cccn3)c2)=O)C1 56046,Cc1nsc(C(N2CCC3C(NC(c4ccnc(S)c4)=O)C23)=O)c1N 56047,c1(COC)ccnc(C(=O)NCCC2CCC(NC(=O)CP(C)(C)=O)C2)c1 56048,C(=O)(C(O)(C(F)(F)F)C1CC1)NCC1(C)CC=CC1 56049,C1(C(=O)NCC(C(C)C)(C)NC(=O)C(N)=O)CCC(F)(F)CC1(C)C 56050,C1(CNC(c2c(C)nc(C)[nH]2)=O)CC(C(C)(C)C)CN(C(=O)CC(C)C2CC2)C1 56051,C1(CC=C)(C(=O)NC2CCN(C(=O)Cn3cc(C#N)cn3)C2CC)CCCCC1 56052,CCC(C(=O)NCC1CCCC1NC(=O)C(C)(C)F)NC(C)=O 56053,C1(C(=O)NCC2(NC(C(C(C)C)OC)=O)CCCC2)CCC(F)(F)CO1 56054,C(=O)(C1=Cc2ccccc2C1O)NCC1CCCN(C(C=NOC)=O)C1 56055,CCS(=O)(=O)CCCN=C(NCC1CCOCC12CCC2)NC1CCC1 56056,C(C(=O)NCC(C)N(C(=O)CCc1cnn(C)c1C)CC)(C(C)C)OCC 56057,CCCCCC(O)C(=O)N(c1ccc(F)cc1C)C(C1C(N)C2CCCCC12)=O 56058,N1(C(CCC(C)OCC)=O)CCC(C)(C)C(NC(c2cc(C(F)(F)F)no2)=O)C1 56059,Cc1nc2cccc(C(N3CCN(C(C4COC(=O)O4)=O)C(C4CC4)C3)=O)c2[nH]1 56060,N1(CC)CCC(C(=O)NC(C)(CSC)C(=O)N(CCCC(C)C)C)CC1 56061,C1(C(C)OC)CCCN(C(=O)CCN(c2cc(C)co2)C(c2cccs2)=O)C1 56062,c1(CNC(CSCC(=O)OC)=O)nc2c(s1)CN(C(=O)CCOC(C)C)CC2 56063,N1(C(C(CC)N2CCCC2=O)=O)CC2CN(C(=O)Cn3c(C)ccc3C)CCC12 56064,C1(O)(C(=O)NCCC(C)NC(c2ccc(CO)o2)=O)CCCC(C)(C)CC1 56065,N1(C(C2(COC)COC2)=O)CC(C)CN(C(=O)Cc2c[nH]nc2C)C(C)C1 56066,C1(CC(=O)N(C)CCN(C)C(c2cc(C)c(C)s2)=O)(OC)CCCCC1 56067,C(=O)(N=c1nn[nH]n1-c1ccc(F)cc1)NCCCCC1C(C)C1 56068,c1(C(C)C(=O)NCCCCC2CN(C(=O)CC3COCCO3)C2)cccc(Cl)c1 56069,c1(CC(=O)OC)occc1C(N1CCCC1C1CCN(C(c2csc(Cl)n2)=O)C1)=O 56070,C(=O)(CC1=CCOCC1)N1CCC(CNC(c2c(Cl)c(C)n(C)n2)=O)C(C)C1 56071,C(=O)(CCCC(CC)NC(=O)CCCCCC)NC(C1CCOC1)C#C 56072,N1(C(C(CC)F)=O)CC2C(CNC(=O)CCc3nnc(C(F)F)o3)C2C1 56073,N1(C(C(F)=C(C)C)=O)CCC2CCN(C(c3csc(Br)n3)=O)C2C1 56074,N1(C(C2(c3ccc(OC)cc3)CCC2)=O)CCN(C(=O)C=CCN(C)C)CC1C 56075,Cc1cc(N)c(C)nc1C(=O)NCCCNC(=O)C=CC1CC1 56076,c1(-c2ccc(OCC)cc2F)nc2ccc(C(N3CCC(C(N)=O)C3)=O)cc2s1 56077,NS(=O)(=O)c1cncc(C(=O)NC23CC2CN(C(C2CCCCC2)=O)C3)c1 56078,N1(CCC)CC(C(=O)NC(C)CNC(C2CCCN2N=O)=O)CC1=O 56079,N1(C(CCC#C)=O)CCC(C)C1CNC(=O)CCSc1nnnn1C 56080,CON(C)C(=O)CNC(=O)CCC1CC(NC(=O)C(C2CC2)C2CC2)C1 56081,C(CS(=O)(=O)CCCN1CCCC(C)(C(N2CCCCC2)=O)C1)OC 56082,C1(NC(c2cncnc2)=O)CN(C(=O)CCN2C(=O)CCC2=O)C2(CCOC2)C1 56083,c1(CSC)cccc(C(N2CC(C)(NC(=O)Cn3cnc(C(F)(F)F)c3)C2)=O)c1 56084,C1(C(N(C)CC2(O)CN(C(=O)CN3CCSCC3)C2)=O)SC2C=CC1CC2 56085,C1(C(=O)NCC(CN(C(CCCOC)=O)C)C)OCCOC12CCC2 56086,Cc1coc(C(C)C)c1C(=O)NC1(CO)CN(C(C23CCC(C2)OC3)=O)C1 56087,Cc1cc(C(c2nnnn2C(C)C)NC(C)Cn2cnnc2)c(Br)cc1F 56088,c1(C(N2CC(SC)C(NC(=O)CCC3CC(F)(F)C3)C2)=O)n[nH]c2c1CSCC2 56089,N1(C(=O)OC(C)(C)C)CCC(NS(=O)(=O)NCC2CC2c2ccncc2)CC1 56090,C1(NC(C23OCC(C(C)C)(C2)C3)=O)CC2(CCN(C(C3CSCC(=O)N3)=O)C2)C1 56091,C#CC1CCN1C(=O)C(Cn1ccnn1)NC(=O)C(C)=CC(C)(C)C 56092,CCC(CCC(=O)Nc1ccccc1CCO)NC(C1CCCCC1O)=O 56093,C1(NC(C2CC2[N+](=O)[O-])=O)CC2C1CCN2NC(c1ccnc(S)c1)=O 56094,N1(C(=O)COCC(F)F)CCC(O)(CCNC(C2(c3ccc(F)cn3)CC2)=O)C1 56095,N1(C(C=CCOCCOC)=O)CCN(C(c2coc(C)n2)=O)C2CS(=O)(=O)CC12 56096,N1(C(CC(=O)NC)=O)CCC2(CC1)CC(NC(=O)CNC(c1cccc(O)c1)=O)C2 56097,C1(C)(NC(CCOCCC)=O)CCCN(C(c2[nH][nH]c(=N)c2Br)=O)C1 56098,C(CCN(C)C)(C(=O)NC1CCCCC1)NCc1nc(NC(C)=O)sc1 56099,CC(C)C(C)(O)CNC(c1cc(NC(C2(n3nccn3)CC2)=O)nn1C)=O 56100,CC1CN(C(=O)CCc2ccnc(Cl)c2)CCC1NC(c1c(Cl)csc1Cl)=O 56101,C1(N(C)C)CCC(C(N2CCC(CCNC(=O)CCc3nccs3)C2)=O)CC1 56102,N1(C(=O)C(F)C2CCCC2)CC2CC1CN2C(C1(F)CCC1)=O 56103,N1(C(c2c(CC)nco2)=O)CC(C)OC2(CCN(C(=O)CSCC(C)C)C2)C1 56104,c1(CN(C)C)ccccc1C(=O)NCC1C=CC(NC(C2COCCOC2)=O)C1 56105,C1(F)(CNC(Cc2ccn(C)n2)=O)CCN(C(C2CC(N3CC(O)C3)C2)=O)CC1 56106,C1(NC(=O)CSCc2cccnc2)COC2(CCN(C(c3ccc(F)o3)=O)C2)C1 56107,CN1CCC(F)(F)CC1C.CCC(CC)(CC(=O)OC)OC 56108,c1(Cc2cnc(N3C(C)(C(=O)O)CCCC3)s2)ccc2nc[nH]c2c1 56109,CCC(O)C(C)C(=O)NC12CC(C(=O)OC3(c4ncc(C)[nH]4)CCC3)(C1)C2 56110,C1(O)(CC)CCN(C(=O)C(C)(C)CN(C(=O)CCCSC)C)C1 56111,N1(C(CCNS(CC)(=O)=O)=O)CCC2(COCC(CNC(c3cnco3)=O)O2)C1 56112,Cc1ncc2n1CC(C(=O)NC1CN(C(C3CCOC(C)(C)C3)=O)CC1C)CC2 56113,N1(C(C(c2ccnn2C)C)=O)CC(NC(=O)Cc2nc[nH]n2)CC12CCCOC2 56114,C1(CCC(=O)NCC(CC)(C)NC(=O)COC(C)C)CCC(O)CC1 56115,N(C(=NCC=C1CCOCC1)N1CCC(c2nncs2)C1)CCOC(C)C 56116,c1(CNC(C(N2CCC(N(CC(CN(C(C)C)C)O)C)C2)=O)=O)cccc(F)c1 56117,S(=O)(=O)(c1ccc(F)cc1Cl)NC(c1ccc(S(C)(=O)=O)cc1)C 56118,N1(C(C2C(OC)C2)=O)CCC(C)C(CNC(=O)C=CC=C(Cl)Cl)C1 56119,C1(C(=O)OC(C(C)N(CC(=O)NCCOC)CCSC)=O)CCCC12CC2 56120,C12=C(Cl)N=CNC1=NCC1(CC13CCC3)CN2.c1(C(=O)OC)cncc(N(C)C)c1 56121,C1(CC)C(C(=O)NC(CCN(C(=O)CSc2ccncc2)C)C(C)C)CCN1C 56122,Cc1ccn(C(C)CC(=O)NCC2(C)CC(NC(c3cc(F)cs3)=O)C2)n1 56123,N1(C(C(CC=CC)NC(=O)CCC(C)N(C)C)=O)CC(C)N(CC)C(C)C1 56124,C#CCCC(O)C(=O)NCC12CC1CN(C(=O)Cc1cccc(Cl)c1F)C2 56125,C1(C(=O)NCc2oc(C)c(C(=O)NCc3cc[nH]n3)n2)CC2(CCC2O)C1 56126,c1(C(N2CCN(C(c3cc(OC)no3)=O)CC23CC3)=O)ccc([N+](=O)[O-])cc1I 56127,CCCC(C(=O)NCC(C)(C)CNC(c1cc(Br)cc(N)c1C)=O)C(C)C 56128,CC1=C(C(=O)N2CCC(C3(NC(c4sccc4F)=O)CC3)C2)CCCC1 56129,c1(C(=O)NCC=CCNC(C=C(C)C(C)C)=O)cc(F)cc(Cl)c1O 56130,c12cccc(c1)C(=O)N2.N1(CC)CCOC(c2cn[nH]c2)C1 56131,N1(CCC(=O)NCc2ncoc2C2CCCN2)CCCCC1 56132,CCCCC(CN(C(=O)CC1(N(C)C(C2CC23CCCC3)=O)CC1)C)CC 56133,c1(CC(N2CC(O)CC23CCC3)=O)ccc2ccccc2c1Br 56134,C1(NC(C2CC3CCC2O3)=O)C=CCN(C(=O)CCc2ccsc2)C1 56135,CC1(C)CC(NC(C2CC3CC2C3)=O)CN(C(c2coc(OCC(F)(F)F)n2)=O)C1 56136,c1(CCC(=O)NC(CNC(CCOCC(C)C)=O)(C)C)cc(Cl)no1 56137,N1(C(c2ccn(CC)c2C)=O)CCCC(C)(C(N2CCC(F)(CF)CC2)=O)C1 56138,c1(NC(C)=O)ccc(-c2csc(NC(c3cc(Cl)c(Cl)s3)=O)n2)cn1 56139,CC(CC(C)(C)C)C(=O)NCCOCCCNC(=O)CSc1nncn1C 56140,c1(C(c2nnnn2C2CC2)NCC(CCC)OC)cnc2ncccn12 56141,c1(CN2CC3C(C(N=c4nc(C)[nH]s4)=O)C3C2)ccc2c(c1)CC(C)O2 56142,N1(C(C(C)N(C)C)=O)CC2CC1CCC2NC(c1ccc(OCC2CC2)nc1)=O 56143,Cc1c(Cl)c(C(N2CC(CNC(=O)Cc3cccnc3Cl)CC2C)=O)nn1C 56144,C(=O)(CCCCC(F)F)NC(C)C(CO)NC(c1cnccn1)=O 56145,N1(CCC(=O)NCCNC(C(CC)F)=O)CCCCCC1 56146,c1(OC)ccc2c(c1)C(NC(=O)C(N1c3ccccc3CCC1C)=O)CC2 56147,c1(C(N2CC(C(=O)Nc3cn(CC)nc3C)C(F)C2)=O)cnc(C)cc1C 56148,C(=O)(CCc1ccsc1)NCCN(C(=O)COC)CCC.C1(=O)CCN1 56149,Cc1nc(C)c(C(N2CC(NC(c3ccnn3C(F)F)=O)C(C)(C)C2)=O)nc1C 56150,CC(C)C(CNC(=O)CCCSC(C)(C)C)NC(=O)Cc1cnn(C(F)F)c1 56151,Cn1cc(S(N)(=O)=O)cc1C(O)C(=O)NCCC1CCCCN1C(=O)CC(F)F 56152,c1(OCC(=O)NC2CC(C)N(C(C3CC4CC3C3CC43)=O)C2)ccccc1C#N 56153,CCCCC(O)C(C)C(=O)NC(c1cnn(C)c1)C(=O)NC(C1CCOC1)CO 56154,c1(C(N(C2CN(C(Cc3cnc(C)o3)=O)CC23CC3)C)=O)ccn2cccc2c1 56155,C12(CNC(c3cc4n(n3)CCC4)=O)CCC(CC1)N(C(C1CCCC(CF)C1)=O)C2 56156,Cc1cccc(CC(=O)NC2CC2NC(=O)C(C)C2CCCC2)c1 56157,N1(C(Cc2n(C)nnc2)=O)CCC2(CCOC2)C(CNC(C2(CCO)CC2)=O)C1 56158,C(N=C(NCC(C)(C)C)NC1CCN(C2CCCC2)CC1)C1C(OC)CCC1 56159,C1(C(=O)NCc2ccc(N(C)CC)cc2)CC2CCCC2C1 56160,N1(C(C2C(C)(COC)C2)=O)CC(NC(=O)Cn2cc(Cl)cn2)C(CO)C1 56161,C1(NC(CC(CC)CC)=O)CC2CC1CN(C(c1ccc3nncn3c1)=O)C2 56162,C1(NC(=O)Cc2ccccc2)CN(C(C2CCC3(CCC3)OC2)=O)CC2(CC2)C1 56163,Cc1c(C(=O)NC2CCCC(NC(=O)C(F)=C3CCCC3)C2)sc2ccccc12 56164,c1(C(N2CCN(CCNC(CCCSC)=O)CC2)=O)ccnc2ccc(O)cc12 56165,N1(C(CC#C)=O)CC2CCCC2(NC(=O)Cc2cc(OC)cc(Cl)c2)C1 56166,O=C(C#CC1CC1)N1CCCCC1C1CCCN(C(c2ccccc2O)=O)C1 56167,C1(C(=O)NC(Cc2cn(CCOC)nn2)C(=O)OC)CCC2(CC1)CC(O)C2 56168,C1(NC(CNC(=O)OCC)=O)CN(C(=O)C(C2CCCCC2)F)C2(CCCC2)C1 56169,C(=O)(CCCCC#N)NCCC1CC(NC(C2(C)COCCO2)=O)C1 56170,N1(C(c2c(CC)cncc2)=O)CC(C(=O)NC(c2n[nH]c(CO)n2)C)CC(C)C1 56171,C1(C#N)(NCCNC(CCCC(=O)N(C)C)=O)CC2C=CC1C2 56172,C(CN=c1[nH]c(=NCc2cc(C(C)C)n[nH]2)[nH]c2cccc(F)c12)OC(CC)C 56173,c1(C(N(C2C3CN(C(C4ON=C(C)C4)=O)CC32)C)=O)ncc2c(F)cccn12 56174,C=CCCC(C(=O)NC(c1csc(O)n1)CCSC)NC(C1CC(COC)C1)=O 56175,C1(NC(C2C(C)(C)C2)=O)CCCCCC1C(=O)NCC1(C(C)(C)O)CC1 56176,C1(CN(C(c2c(C)nsc2)=O)C)CCCC(NC(c2cc[nH]n2)=O)C1 56177,C1(NC(c2ccc(COC)o2)=O)CC2CCC1N(C(=O)C(C)n1cnnn1)C2 56178,C(=O)(CC(C(F)(F)F)n1ccnc1)N1CCC(Sc2cc(C(C)=O)nn2C)CC1 56179,C1(C(N(CC(=O)N(C)C)C)=O)CCC2(CC2)N1C(C1CCCCC(=O)C1)=O 56180,c1(OC)ccc(C(N2CC=CC2(C)C(=O)NCCCn2cnnc2C)=O)cn1 56181,N1(C(c2cc(OC)ns2)=O)CC(C(N2CCNC(=O)C2C(C)C)=O)CC(C)(C)C1 56182,Cc1cccc(Br)c1C(C(=O)NC1(C)CC(C)OC1=O)NC(=O)Cc1ccsn1 56183,C=CC(C)(O)C(=O)N(CC(=O)NC(c1ccco1)CC)Cc1csc(-c2cocn2)n1 56184,CN1CCOc2c(C(N3CC(NC(=O)C(O)C(F)(F)F)C3)=O)cccc21 56185,c1(C(=O)NCC(C2CCC2)NC(C2C(CC(C)C)C2)=O)nsnc1O 56186,C12CN(C1)C2=O.C1(CCOC)(C(=O)NCC2CC(C(=O)OC)C2)CCC1 56187,C(C)(C)(CCCCC(=O)NC1CCN(C(c2ccc(Cl)c(Cl)c2)=O)CC1)OC 56188,Cc1cnnc(O)c1C(=O)NCc1cc(C(N2CCC(C)C2CO)=O)no1 56189,CC(CN=c1nc(N2Cc3cncnc3C(C)C2)c2c(ncn2C)[nH]1)N(C)C 56190,C1(C(=O)NCC2(C)N(C(C3OCCN(C)C3)=O)CCC2)CC(C)(C)CN1C 56191,c1(C(N2CC3C(CN(C(C(C=C)O)=O)C)C3C2)=O)cc(C)cc(C)c1 56192,CCCCC(C)(C)NC(=O)C(C)Sc1ccc(C)cc1 56193,CC1CC=C(C(=O)NCC2CCC2NC(=O)CSc2nnnn2C2CC2)CC1 56194,Cc1ccc2c(CC(N3CCN(C(C45CC(C)(C4)C5)=O)CC3)=O)c[nH]c2c1 56195,c1(CNC(C(C)c2cccs2)=O)ccoc1C(=O)NCc1ccnn1C 56196,C(C1=C(C(=O)O)C(c2ccccc2)NC(=O)N1)C(CC1NN=C(C(=O)OC)C1)=O 56197,N1(C(C(C(=O)OCC)(C)C)=O)Cc2occ(C(=O)NCCCSCC)c2C1 56198,N1(C(CC2C(C)CCC2)=O)CCC2(CC(NC(=O)C=Cc3cncs3)C2)C1 56199,CC1CN(C(c2cn(CCNC(=O)CC3CCCC(=O)N3)nn2)=O)CC(=O)N1 56200,C(=O)(C(C)(C)CCCCC)NC1CN(C(CC2(C(=C)F)CCC2)=O)CC(C)C1 56201,C1(N(C(c2cc(CC)no2)=O)C)CC2CC1N(C(=O)C(C)(C)CN(CC)CC)C2 56202,N1(C(C2(F)CCN(C(c3cc(C)ncc3C)=O)C2)=O)CCCC12CCCOC2 56203,N1(C(CS(C)(=O)=O)=O)CCC(NC(=O)C=CC=CCO)CC1C1CC1 56204,c1(C(N2CCC(CC3CN(C(c4cnco4)=O)C3)CC2)=O)ccn2ccnc2c1 56205,CC1(C)CN(C(=O)CC2(C(F)(F)F)CC2)CCC1NC(c1cc2ccsc2s1)=O 56206,C(=O)(CCCCCC#N)NC(C(=O)NC(C#C)CC(C)(C)C)(C)C1CCC1 56207,Cc1cc2nc(-c3nc(CC(C)C)nn3CC3CCCCC3)ccc2c(=O)n1C 56208,C=CCCCCC(=O)N1CCN(C)C(C(=O)NCCNC(=O)CC)C1 56209,Cc1cc2c(cc1C)OC(C(N1CCN(C(=O)CC3(CO)CCC3)C(C)C1)=O)C2 56210,C(=O)(C(C)C(=O)NCc1cc(C(=O)NC(C)C(=O)C2CCCC2)no1)OC 56211,c1(CC(=O)NCCN(C(=O)CSc2cccs2)CCOC)ccc2c(c1)COC2 56212,CC1CCC(C(N2CCC(CN(C(=O)C(C)(F)F)C3CC3)CC2)=O)CC1C 56213,N1(C(C2(NC(C3C(C)C3)=O)CCCCC2)=O)C2CCC1CN(C)C2 56214,N1(C(C2(CC)CCN(C(C3CC34CCCC4)=O)C2)=O)CCC(C)(C2CC2)C1 56215,Cc1nc2n(c(=O)c1CCN1CCCC3(CCCCCO3)C1)CCCC2 56216,c1(OC)cc(C(=O)Nc2ccc(C(=O)Nc3csc(C#N)c3)cn2)ccc1Br 56217,c1(C(C)C)[nH]nc(C(N2CC(O)CC2Cn2cc(CCC3CC3)nn2)=O)c1Br 56218,CN1N=CC(CC(=O)NC2CC(NCCNC[Si](C)(C)C)CC2O)C1=O 56219,S(=O)(=O)(CC(=O)N(CCCNC(=O)Cc1cnn(CC)c1)CC)NCC 56220,Cc1ccc(C(F)F)cc1C(N1CCC1CNC(c1cccc(C#N)c1)=O)=O 56221,C12(C(=O)NCC(CN(C(CCC(=C)C)=O)CC)(C)C)CCC(C(F)F)(CC1)C2 56222,c1(OC)cccc2c(N3CCCC(CC(C)C)C3)ncnc12 56223,c1(C(N(C)Cc2ncc(-c3ccccn3)[nH]2)=O)ccc(-c2cccs2)cc1 56224,C=C1CCC(C(=O)N(C2CCCCC2NC(=O)Cc2cnnn2C)C)CC1 56225,C(C(O)CC(=O)NC1CN(C(=O)C(C)(C)N2CCCCC2)CC1F)N(C)C 56226,C(=O)(CCS(N)(=O)=O)N1CCC(C(=O)NC2CCOC2=O)(OC)C1 56227,C(=O)(CCCC(C)(C)NC(=O)C(C#N)C(C)(C)C)NC1CCN(CC)C(C)C1 56228,Cc1ccc(C)c(C(N2CC(CCNC(C3CC(C(C)C)=NO3)=O)C2)=O)c1 56229,c1(N2CCC(C)C2)ncnc2c1ncn2CC1CCCCC1O 56230,CC1(C)COC1C(N1CCCC1CCNC(=O)Cc1cc[nH]n1)=O 56231,Cc1scc(C(=O)NCCN(CCCN(C)C)C(=O)CC2CC3CC3C2)c1C 56232,N1(C(CNC(CCC)=O)=O)CCC2CCN(C(=O)Cc3cccc(OC)c3)C2C1 56233,C1(CNC(CC(CC)(C)C)=O)CC2CCC(C1)N2C(C1(COC)CCCCC1)=O 56234,c1(C(=O)NC)ccc(NC(C2(C)CCCN2Cc2cnc(C)[nH]2)=O)cc1 56235,N(C1CCCc2c(Br)cncc21)N1CCC(c2ccc(N(C)C)cc2)C1 56236,CC1CCN(C(=O)C(=O)NC2(CNC(=O)CC3(C)CC3F)CC2)CC1 56237,C(=O)(C1=NOC(C)(C)C1)N1CCCC(C(=O)NCCC(C(C)C)OC)(CO)C1 56238,c1(NC(C)=O)nnc(S(=O)(=O)NC2CCC(F)(F)C(C)C2)s1 56239,C1(C(=O)OC)CN(N(Cc2cccs2)CCCO)CC1S(=O)(=O)c1ccccc1 56240,c1(C(=O)OC)cc(NC(=O)NCC2CC(c3ccccc3)C2)cc(C)c1C 56241,C1(CC(=O)NC(CCNC(CC=CCC)=O)(C)C)CCCC(C)(C)C1 56242,c1(OC)cc(C(ONC(=O)C(CSC)OC)=O)cc(SC)c1 56243,C1(CCC)(NC(=O)Cc2cccc(C)c2)CCN(C(C2COCC2(C)C)=O)CC1 56244,c1(NCc2ccn(CC)n2)[nH]c(=NCc2cnn(C3CC3)c2)nc2scnc12 56245,N1(C(C(CC(C)C)(C)O)=O)CC2(C=C(C(=O)NCC3CCSC3)CO2)C1 56246,CCCCC(N)C(=O)N1CCC(O)C(C(N2CCN(C)CC2CCO)=O)C1 56247,N1(C(COC)=O)CC2CCN(C(c3cc(O)cc(O)n3)=O)CCC2C1 56248,C1(NC(C(C)CC2CCCC2)=O)CC12CCN(C(=O)CC1CCCN1C)C2 56249,C1(NC(C(c2cc(C)oc2C)C)=O)CCCCN(C(=O)C(F)(F)c2nccs2)C1 56250,C1(NC(c2c(CC)occ2)=O)(CC)CCN(C(C2(C)COC2)=O)CC1 56251,C1(NC(C2CC(C)(CC)C2)=O)(CO)CCCN(C(=O)C(F)(F)c2cscn2)C1 56252,c1(C(CNC(c2ccon2)=O)NC(C2CN(C)C(=O)C2)=O)ccc(F)cc1F 56253,C(=O)(C(F)(F)CC(C)C)OCC(c1c(C)onc1-c1c(F)cccc1Cl)=O 56254,c1(C(=O)NC(CC)CN(C)C(c2cc(C)cs2)=O)cc(N)c(Cl)c(O)c1 56255,C12CCCCC1NC2=O.C(=O)(C(C(C)C)N(C)C)NCC1N(CCC)CCC1 56256,C1(C(N(C(CF)CF)C)=O)CC1C1CN(C(C2CN3CCC2CC3)=O)C1 56257,C1(CC(=O)NCC(CC)NC(c2nnsc2C(F)F)=O)CC(C)(C)OC(C)(C)C1 56258,N1(C(C2C(C)C2)=O)CCCCC1CNC(=O)CCc1cnn(C)n1 56259,N1(C(c2c(C)cnnc2)=O)CC(CNC(C2CCCC23CCC3)=O)C(C)(C)C1 56260,C(=O)(C1=CCC2CCC1N2C(C1(C2CC2)CC1)=O)N(CCCOC)CCO 56261,C(=O)(CS(=O)(=O)c1ccccc1Cl)NC1CCC(NC(C23OCC(C)(C2)C3)=O)C1 56262,c1(N(CCC)C)ccc(C(=O)NCCCN(C(C2CC(CO)CO2)=O)CC)cc1 56263,C1(C(C)C)(C(N2CCC(C(C)(C)O)C2)=O)CCN(C(=O)CSCC(F)F)C1 56264,O=C(C(O)CC(F)(F)F)NC1CCN(C(=O)C=Cc2cccc(O)c2)C1 56265,Cc1nnc2n1CC(C(=O)OC1CCC1)CC2 56266,O=C(N=S1(=O)CCNC(c2ccccc2)C1)c1cc2c(Br)cccc2s1 56267,c1(C(N2CC3C(CNC(COCCCC)=O)(C3)C2)=O)nccc(Cl)c1C 56268,C(=O)(CCCC1CCCC1)NCC1(CCNC(C(C)N(C(C)=O)C)=O)CC1 56269,N1(C(Cn2ccc(OCCOC)c2)=O)CCC(CO)C12CC2.N1CC(OC)C1=O 56270,N1(C(c2c(C)coc2C)=O)CCN(C(=O)Cn2nnc(=O)[nH]2)C(C)C1C 56271,C(CC)(C(=O)N1CCC(c2ncco2)C1)N(C(CSCC)=O)C 56272,c1(OC)cc(C(=O)NCCc2ccccc2C)c(NC(c2ccccc2)=O)cn1 56273,c1(C(=O)NCC2(F)CN(C(c3ncc[nH]c3=O)=O)C2)cc([N+](=O)[O-])n[nH]1 56274,C1(C(=O)NCCC(=O)NC)CCN(C(=O)c2cnn(C)c2OC)O1 56275,C(CC(=O)NC1CC2OCCCC12)(C(C)OC)NC(c1cnc(CC)o1)=O 56276,C1(CNC(c2cc(C(=O)OCC)on2)=O)CC(C(=O)OC)CC(C(F)(F)F)C1 56277,c1(CNC(N2C(C)CSCCC2)=O)c(Br)ccc(Cl)c1F 56278,CC(CC(C)(C)C)C(=O)N1CC2CC(C1)N(C(=O)CNc1ncccn1)C2 56279,Cc1ccn2nc(C(=O)NCCNC(C3CC4CC4C3)=O)nc2n1 56280,Cc1c(C(N)=O)cccc1C(=O)NCCCC1CCCN1C(=O)C(F)C(C)(C)O 56281,C1(C(=O)NCC2CC3(CCC3)C2)CCN(C(c2cc[n+]([O-])cc2)=O)C12CC2 56282,c1(OC)ncc(C=CC(=O)NC2CCCN(C(C3CCCN3C)=O)C2C)cn1 56283,c1(C(C)=O)ccc2c(c1)NC(=O)C1(CC(C(=O)NC(=O)NC(C)C(=O)O)C1)CC=N2 56284,c1(C(N2CCOCC2)C)cc(CN2CCN(C(=O)OC)C(=O)C2)cc(Br)c1 56285,C(=O)(CCS(=O)(=O)C1CCCC1)N1CCCC(C)(NC(=O)C(CO)NC(N)=O)C1 56286,N1(CCN(C(CCC)C)C)CC(C)OC(C)C1 56287,n1(CC)cc(CN(C(=O)CNC(=O)CNC(=O)C(C)CO)C)nn1 56288,CC1CC(CCNC(c2cc(Cl)no2)=O)CCN1C(=O)Cc1ccc(F)nc1 56289,N1(C(c2ccc(CC)[nH]2)=O)CC(NC(C2CC(OC(F)(F)F)C2)=O)CC1C 56290,N1(C(CC(C)CF)=O)C2CCC1CC(NC(=O)CN1CSCCSC1)C2 56291,CC(CCCCNC(=O)CNC(=O)C(F)(F)F)NC(=O)CCn1cccnc1=O 56292,C1(NC(c2c(Cl)cn(CC)n2)=O)CN(C(=O)CC2CCC3CC3C2)CC1(C)C 56293,C1(C(=O)NC2CCN(C(C(CC)c3ccccc3CC)=O)CC2)CCCC(C)(C)O1 56294,c1(C(C(=O)NC(C)C)N(CCC)C)cnc(C(F)F)s1 56295,CC1CCCc2cc(NC(N3CCSc4ccccc43)=O)nn21 56296,CC1CC(N(C(C(=O)NCCC2CC2)c2cnc[nH]2)C)CCN1C 56297,C=C(C)CC(C)C(=O)NCC(CC)NC(=O)C(C)(C)C(F)F 56298,N(C(=NCCc1ccccc1F)NC(C)(C)CF)CCC(=O)N(C)C 56299,CCCC(CC(C)C)C(=O)NCCc1ocnc1CNC(=O)C(C)SC(F)(F)F 56300,CC1CN(C(C2CCC3(CC2)N=N3)=O)CCC1NC(C1SCCCS1)=O 56301,Cc1cc(N)c(C(N2CCC(O)(C(C)CNC(c3ccc(Br)o3)=O)C2)=O)c(F)c1 56302,C1(C(N2CCC(C)(NC(=O)CC3COC(=O)C3)C2)=O)C2Cc3ccccc3C12 56303,C(=O)(CC(C)CC(=O)NC1CN(C(c2cc(C3CC3)no2)=O)C2(CCC2)C1)OC 56304,c1(C(=O)NC(C(C)NC(c2c(C)nc(CCC)s2)=O)C)ccc(OC)nc1Cl 56305,Cc1cn2cc(C(=O)NC3CCN(C(=O)COc4ccn(C)n4)C3)nc2s1 56306,c1(OC)c(C(=O)NC2CCN(C(c3occc3C)=O)CC2C)cccc1Br 56307,c1(C(=O)NCCCOCCCNC(=O)CC2C=CCC2)cscc1C1CC1 56308,C=CCCCCCCCC(C(=O)OC)N1CC2CCCN2CC1CC 56309,CC(CCC1CNc2ccccc21)n1cc(Cc2ccccc2)nn1 56310,c1(CC)cnn(C)c1C(C(=O)NCC1CC1)N(CCCNC(=O)OC(C)(C)C)C 56311,NS(=O)(=O)c1cccc(C(=O)NC2C3CC2CN(C(c2ccc(CO)o2)=O)C3)c1 56312,N1(C(C)=O)C(C(N2CCC(C(=O)Nc3cnc(Cl)nn3)C2)=O)CCC1C 56313,CCC(CO)(C(=O)N(C)CCN(C)C(c1cnc[nH]c1=N)=O)OC 56314,C1(CNC(C2CC23CCCC3)=O)CNCCC12CCOCC2 56315,C1(O)(C(C)NC(CC2C(C)CC2)=O)CCN(C(C2(CF)CC2)=O)C1 56316,N1(C(c2n(C)nnc2)=O)CC(NC(C2CCOC2)=O)C2CCCC2C1 56317,c1(C(=O)NCC2(CNC(C3CC4(CCC4)CO3)=O)CC2)nccc2occc12 56318,N1(C(CC#C)=O)CC2COCC2(C(N2CCCC2C(C)(C)O)=O)C1 56319,c1(OC)cc(Br)c(C)nc1NC(C1CC(F)CN1c1cc(C)ncn1)=O 56320,N1(CC(=O)NC)CC(O)CC2(CCNCC2)C1.C12(CC1)C(=O)N2 56321,CCC(CC(C)C)C(=O)NCC1(C(N2CCC(OCCF)C2)=O)CCCCC1 56322,C1(N(C(C(CNC(c2nc(C)sc2)=O)N(C)C)=O)C)COC(C)(C)C1 56323,CCCCN=C(NCCc1ccc2c[nH]nc2c1)NCC(C)C#N 56324,N1(C(C2N(C(c3c(C)ncc(Cl)c3)=O)CCSC2)=O)Cc2cccc(O)c2C1 56325,N1(C(CCn2cnc(=N)[nH]2)=O)CCC2CCN(C(=O)CCF)CC12 56326,CC(C)CC(C(=O)N1CCC(O)(CO)CC1)NC(=O)Cc1ccccc1 56327,C1(CNC(C(CC)SC)=O)CC2(CCN(C(c3ccc(C(C)C)cc3)=O)CC2)C1 56328,C1(NC(COCC=C)=O)CCCN(C(=O)Cc2csc(C3CCS(=O)(=O)C3)n2)C1 56329,C(C(=O)NC1CCCCC1NC(=O)C#CC1CC1)(C(C)C)(C(C)C)NC(C)=O 56330,Cc1ccccc1COCC(N1CC(NC(C2CC3(CC3)CO2)=O)C(O)C1)=O 56331,CCC(C)(CO)CN=c1cc(NCCc2csc(C3CC3)n2)nc[nH]1 56332,C1(NC(N2C(NS(C)(=O)=O)CCC2)=O)CCC2C3CCC(C3)C12 56333,CC(C)CCC(F)C(=O)N1CCC(O)(CCNC(C2CCCCCC2)=O)CC1 56334,c1(OC)cc(NCC2(OC(C)=O)CC(c3nnnn3CC(F)F)C2)cc(O)c1 56335,c1(C(=O)NC2CCCC(NC(CN(C)C)=O)C2)ccc(Cl)c(N2CCCC2)n1 56336,c1(OC)ccc(F)cc1CC(N1CC2CN(C(c3cc(O)ncn3)=O)C2C1)=O 56337,C1(C(=O)NCC)C(C2CC2)CCN1Cc1nnc(N2CCCC(N(CC=C)CC)C2)s1 56338,C1(C(=O)Nc2ccc(COC)cc2)CCOCCN1C(c1cnn[nH]1)=O 56339,N12CCC(CC1)CN(C(=O)CC1(C)CCOC1)CC2=O.C1(OCC)CCCOC1 56340,c1(C(C(N2CC(CNC(CN(CC)CC)=O)OCC2)=O)(C)C)cccc(C#N)c1 56341,N1(C(C(C=C)(C)C)=O)CCC(C(F)(F)F)C(NC(c2nnc(C)cc2O)=O)C1 56342,CCCCC(O)C(C)C(=O)NCC1(C)CCN(C(=O)COCc2nc[nH]n2)CC1 56343,c1(C(N2CC(OCCNC(C3C(C=C)C3)=O)C2)=O)cc(Cl)c(Cl)cc1O 56344,c1(OC)ccc(C2(NC(=O)N(C3CC3)Cc3ccnc(SC)n3)CC2)cc1OC 56345,c1(-n2c(C)ncc2)ccc(CN2CCC(N(CCCn3ccnc3)C)CC2)cc1 56346,N1(C(CCOCCCC)=O)CCN(C(=O)C(C)N(CC)CC)C2(CC2)C1 56347,c1(C(=O)Nc2ccc(C)nc2Br)cc(-c2ccc(C)cc2)n2cnc(CN)c2n1 56348,C1(C(=O)NCCN(C(=O)COC2CCCOC2)C(C)C)OCC2COCCC12 56349,C1(C(=O)OC)CN(C(=O)C(=O)NCC2(C)CCN(C)CC2)C(C)(C)C1 56350,c1(OC)cc(C2(C(=O)NC3CCC(CNC(=O)CC4CC=CC4)C3)CC2)ccc1C 56351,c1(CC)nc(C)c(C(=O)NC(C(=O)NOCC2CC3C=CC2C3)C2CC2)o1 56352,N1(C(CCCC#C)=O)CCC(NC(C2CCCN(C(C)=O)C2)=O)C1(C)C 56353,CCC(C)(C)C(C(=O)NC1(CNC(=O)Cc2csc(C)n2)CCOCC1)OC 56354,C1(CNC(CC(C)N2CCCC2=O)=O)CCN(C(C2CCC(=O)N2)=O)C(C)C1 56355,c1(C(N2C(C(=O)NC(C(=O)OC)C3CC3)CC3CC32)=O)ccc(F)c(Br)c1F 56356,C1(NC(=O)Nc2ccnc(N3CCOC3=O)c2)CCc2cc(Br)ccc2C1 56357,N1(C(C2=C(C)OCC2)=O)CC2(CCC(NC(c3ccncc3F)=O)C2)C1 56358,C12(NC(c3cc(-c4ccoc4)[nH]n3)=O)CC1CN(C(c1ccnn1C1CC1)=O)C2 56359,N1(C(C2N(C(C(C)CC(N)=O)=O)CC3CC32)=O)CC2(C1)NC(=O)NC2=O 56360,Cc1cc(C)cc(C=CC(N2CCCC2CN(C(=O)CCSCC(N)=O)C)=O)c1 56361,N(C1CCNC(=O)c2[nH]ccc21)C(C1CCC(C(=O)OC)CC1)=O 56362,c1(CC)ccc(N2CC(C(=O)NC3CCN(C)C3)CC2=O)cc1 56363,C1(C(N2CCN(Cc3nc(C4CCCCC4)no3)CC2)=O)CC2(CSC2)C1 56364,N1(CC)CCCC(NC(=O)C(CO)NC(=O)CCC(C)N(C)C)C1 56365,C1(C(=O)NC)C2CC1N(C(c1cnc(Cl)s1)=O)C2.C1(n2cccn2)COC1 56366,C12(NC(c3cc(C)sc3)=O)CCCC1CN(C(c1cc[nH]n1)=O)C2 56367,C1(CNC(=O)C2=NOCC2)CN(C(=O)C(F)Cc2ccccc2)CC2(CCC2)O1 56368,C1(CC#C)(C(=O)NCc2snnc2C)CCN(C(c2cccc(C)n2)=O)C1 56369,CCC(CC(=O)N1CC2C(CNC(C3CC4(CCOCC4)C3)=O)C2C1)C(C)C 56370,c1(C(=O)NCC23CC(CO2)N(C(=O)CC=C(Cl)Cl)C3)c(F)ccc(Cl)c1F 56371,C1(NC(CCCC)=O)CC(C2CCN(C(c3ncnc(C)c3C)=O)C2)C1 56372,C1(OCC(=O)NCCCN(CCCF)C)CCC(F)(F)CC1.C12CC1NC2=O 56373,C(C)(C)(CN=c1[nH]nc(C#N)s1)C1CN(C(=O)NCc2c(C)cc(Cl)cc2C)C1 56374,C12(NC(C3(N=[N+]=[N-])CC3)=O)CCCC1CN(C(=O)CCC1CCC1)C2 56375,Cn1cc(CCC(=O)NC(C(N2CCC(c3cnn[nH]3)C2)=O)C2(O)CCC2)cn1 56376,c1(OC(C)C(=O)Nc2c(O)n[nH]c2Cc2ccccc2)ccccc1F 56377,CC1CC(N(C(=O)C(C)(C)CN(C(=O)Cc2cncnc2)C)C)CC(C)O1 56378,N1(C(C2(c3cccc(OC(F)F)c3)CCC2)=O)CC(NC(=O)C2CC2)CC(O)C1 56379,N1(C(CC(N)Cc2ccc(OC(F)(F)F)cc2)=O)CC2NCCOC2C1 56380,C(=O)(C(C)CC(C)C(C)=O)NC1C(C(=O)NCC2(CC(=O)OC)CC2)CC=CC1 56381,CCCC(CC)C(=O)NCCCNC(=O)C(O)Cc1c(F)cccc1Cl 56382,C(CN=c1[nH]c(=NCC2CN(C)CCN2C)[nH]c2c1COC2)N(CCC)CCC 56383,c1(OC)cc(NC(C2CC2NC(c2cc(Br)ccc2C)=O)=O)cc(C#N)c1 56384,c1(C(=O)NCC(c2cccc(Cl)c2Cl)F)cc(Cl)c([N+](=O)[O-])[nH]1 56385,n1(CC)c(NC(=O)CSc2nccc(C(C)C)n2)nc2ccc(Br)cc12 56386,N1(C(c2cc(C)n(C)c2)=O)CC(NC(C2CC3(CCCO3)C2)=O)CCC(O)C1 56387,c1(OC)ccc(C(=O)NCCN(CCC)CC)c(OC(c2cnn(C)c2C)=O)c1 56388,c1(C(N2CCC(F)(C(=O)Nc3ncc(Cl)nc3Br)CC2)=O)cc(Cl)cc(Cl)c1O 56389,C=CCC(C(=O)N(C)CCN(C(=O)C(O)c1ccsc1)C)C(C)(C)C 56390,C(=O)(C(C)(C)S(=O)(=O)C1CC1)NCC1N(c2snc(C)n2)CCC1 56391,C1(C#CC(=O)N2CCCC2CNC(=O)Cc2ccc(O)c(OC)c2)(CC)CC1 56392,N1(C(c2c(C)nc(O)s2)=O)CCN(C(=O)CCc2cn(C)nn2)CC(C)C1 56393,N1(C(C=COCC)=O)CC(NC(c2cnc(OC(C)C)cn2)=O)CC2(CC2)C1 56394,c1(C(=O)Nc2cc(OC(F)F)n[nH]2)n[nH]c2c1CN(Cc1cnnc(Cl)c1)CC2 56395,C1(C(NOC(C)C)=O)CCC(NC(=O)COCCF)CC1 56396,Cc1cncc(C(=O)NCCC(C)CCNC(=O)C(F)CC2CCCCC2)c1 56397,CC1=C(Br)CN(C(c2ccc(C)c(Br)n2)C(=O)NC2COC2)CC1 56398,c1(C(=O)NCCN(C(=O)C(C)N2CCC2)CC)cc(C(=O)OC)c[nH]1 56399,c1(OC)cc(Cl)c(-c2cn(CC3CCCN3C(=O)Cc3cnns3)nn2)cc1Cl 56400,c1(C(=O)NC2C(NC(CCc3nc(C)c(C)o3)=O)CC2)ccc(F)c(C2CC2)c1 56401,c1(SC)cc(C(=O)NCC2CC(F)(CNC(=O)Cc3csnn3)C2)c(C)o1 56402,c1(C(N2C(C(N3CCC(C)(C#N)C3)=O)CCC2C)=O)ccc2cc(O)ccc2n1 56403,C1(NC(CC2N(C(C(C)SC(C)C)=O)CC(O)C2)=O)CCC(C)(C)CC1 56404,Cc1cc(NC(=O)CSCCNC(C2CC3(C2)CC32CC2)=O)c(F)cc1F 56405,C(CC(C(=O)NCCC(C)(C)N(C)C)NC(=O)CCCSC)SC 56406,C(=O)(CS(=O)(=O)CC(=O)OC)NC1C(NC(C(COC)C)=O)CCC1 56407,CC1CC(C(=O)NCC2(F)CN(C(c3cc(O)cc(O)n3)=O)C2)Cc2nn[nH]c21 56408,C1(C(=O)NC2CC(CO)C23CCC3)(CC)CCCN(C(=O)CC(C)F)C1 56409,N1(C(c2cc(C)nc(O)n2)=O)CC2(CCCN(C(c3ccc(CF)cc3)=O)C2)C1 56410,C1(C)(NC(c2ccc(C(C)C)nc2)=O)CCN(C(C2CCC(F)C2)=O)CC1 56411,CC1CC(=O)NC(C(=O)NC(C2CC2C(=O)NCC=C2CCSCC2)C)C1 56412,C(C(C)(C)C#CC(=O)NC1CN(C)CC1O)NC(Cn1c(C)ccc1C)=O 56413,Cc1cnc(C(=O)NC(C2(O)CN(C(=O)C3=CCCOC3)C2)C)cc1C 56414,C1(CNC(C(C)N2CCC2)=O)CCN(C(=O)C(C(C)(C)C)N(C)C)CCC1(F)F 56415,c1(C(=O)NC2C(NC(C(=Cc3cccs3)C)=O)CCC2)cc(Cl)ccn1 56416,N1(C(C2(NC(c3ccncc3O)=O)CC(OC)C2)=O)CCC2(C1)CC2(F)F 56417,N1(C(c2c(CC)[nH]cc2)=O)CCN(C(=O)C(C)NC(C)=O)CC1C(F)F 56418,Cc1cncc(C)c1C(N1CCOC(CCNC(C2CCC(C)(C)OC2)=O)C1)=O 56419,CC1CCC(CNC(=O)C=CBr)N(C(=O)Cc2ccc(C(F)(F)F)cc2)C1 56420,C1(NC(CCC#CC)=O)CCN(C(=O)Cc2c(C)noc2Cl)CC1C 56421,C1(O)(CNC(C2CC(N(C)C)C2)=O)CN(C(=O)COc2ccon2)C1 56422,C1(OC)CCC(C(N2CC(N(C)C(c3cnn(C(C)C)c3F)=O)C(O)C2)=O)CC1 56423,c1(OC)cc(CN(C(c2csc(Br)n2)C(=O)NCCC2CC2)C)c(OC)cc1C 56424,CCC(C)(CO)C(=O)N1CC2(CCN2C(c2cc(OC)n[nH]2)=O)C1 56425,CCCCCC(F)C(=O)NC1CCSC12CN(C(c1cnc(O)o1)=O)C2 56426,C1(OC)CN(C(C2CC=CCO2)=O)CC1c1cn(-c2ccncc2)nn1 56427,C1(CCC(=O)NCCC(C)(C)F)CCCCN(C(=O)C=CC2CCOCC2)C1 56428,CC1CN(C(=O)C(C2(O)CCCCC2)(F)F)CC1(C)CNC(=O)CS(C)(=O)=O 56429,C(CC(C)C(=O)N(C(C)C(=O)N(C1CC(C)(C)C1)C)C1CC1)=CCC 56430,CC(O)CC(C)(C)CNC(C1(F)CCN(C(C2(C(F)(F)F)CC2)=O)C1)=O 56431,c1(C(=O)NCC(CC)N(C)C(c2csc(F)c2)=O)ncc2[nH]ncc2n1 56432,Cc1ncccc1NC(=O)C(C)CN(C(=O)C(O)C1CC1)C 56433,C(C(=O)NC1CCCC1(F)F)(C(C)OC)NC(C(CC)=CCCC)=O 56434,N1(C(C2(CCOC)CCC2)=O)CCC(NCCCC2CCOC2)C(C)C1 56435,C=CCCC(C1CC1)NC(=O)C(c1ccnn1C)NC(=O)C(c1ccn(C)c1)C 56436,c1(C(=O)NCC2N(C(C(CC#C)C)=O)CCC(C)C2)ccc2nc[nH]c2c1F 56437,C(=O)(C(CC)CC(F)(F)F)N1CCC(CNC(c2cc(CC)on2)=O)C12CC2 56438,c1(C(=O)NCCNC(C2CCCN(C(C(CC)F)=O)C2)=O)cc(C)ccc1N 56439,c1(N2CCC(NC(C3C(C)=C3)=O)C(C)C2)ncc(C#N)cc1Br 56440,C(=O)(C1=C(C#N)CCC1)N1CC(NC(c2ccc(-c3nc(C)on3)cc2)=O)C1 56441,c1(OC)cccc(CNCC(C(=O)C2C(CSC)C(O)C2)(F)F)c1 56442,N1(C(c2cc(C)oc2)=O)CCN(C(c2ncc3[nH]ncc3n2)=O)CC2(CC2)C1 56443,CC1CC(C(N2CCC(O)(CN(C(=O)C3=COCCO3)C)CC2)=O)CC(C)O1 56444,c1(CCC(=O)N(CCCNC(C2CC3(F)CC2C3)=O)C)ccc2c(c1)CCO2 56445,C1(C)(C(N(CC(=O)N(CCC#C)CCOC)CC)=O)CC2CCC1C2 56446,Cc1ccnc(C(C)NC(=O)CC2CN(C(=O)OC(C)(C)C)CC2C)n1 56447,C=CC(C)(C)C(=O)N1CCC(CCCCCNC(c2cc(C)n(C)n2)=O)CC1 56448,c12ccc(cc1)[nH]c2=O.c1(CNC(C)=O)cccc(Br)n1 56449,C1(CNC(CCCN(C(C)=O)C)=O)CCCCN(C(c2cocc2C(N)=O)=O)C1 56450,C1(F)(C(=O)OCC)CN(C(c2cn[nH]c2Br)=O)CC12CNC2 56451,N1(C(CN(C(=O)COCC(C)(C)C)CCOC)=O)CCC(CO)(CO)C1 56452,c1(C(=O)NC2C(CNC(C(CCCOC)C)=O)C2)cccc2c1OC(C)(C)CC2 56453,Cc1csc2c(C(N3CCCCC3CNC(=O)CC34CCCC3C4)=O)cccc12 56454,C(=O)(C(C)CC(C)(C)C)NCC(CC)N(C(=O)CSC(F)F)C 56455,c1(C(N2CCCC(N(C(c3nc(C)c(C)s3)=O)CC)C2)=O)nc(C)ccc1F 56456,C(=O)(C(F)CC(C)C)NCC1(CO)CCN(C(CC=C=C)=O)C1 56457,C1(C)(C(=O)NCC(C)CN(C)C)CCN(C(C2CC(C)(C)C2)=O)C1 56458,c1(C(=O)NCc2cc(C(=O)NC(C(=O)OC(C)C)C)ncc2)ccc(=O)n(C)n1 56459,N1(C(C(C)OCC)=O)CC2(CCCC(CNC(c3nn(C)cc3[N+](=O)[O-])=O)O2)C1 56460,C(N=c1[nH]c(=NCC(=O)N2CCCO2)c2c(F)cccc2[nH]1)c1scc(CC)n1 56461,Cc1cc(C=CC(=O)N(C)CC2(O)CCCN(C(c3cnns3)=O)C2)ccc1F 56462,N(C(=NCc1nccs1)NCC(C1CCOCC1)(F)F)CC(=O)NCC(F)(F)F 56463,C=C(CNC(=O)Cc1ccsc1)CCNC(C1CCN1C(C)=O)=O 56464,C=C(C)C(C)(C)C(=O)NC1CCC(C)(CNC(=O)CNC(C)=O)CC1 56465,C(c1ccccc1F)=CC(=O)NCC1(NC(=O)Cc2cc[nH]c2)CCOCC1 56466,c1(OC)cc(CNC(C2CCCC2NC(=O)CCC2CC2)=O)cc2c1OCO2 56467,c1(C(=O)NC2C(CNC(CC(=O)N(C)C)=O)CCC2)cc2cc(Cl)c(Cl)cc2[nH]1 56468,C1(NC(CC(C)(C)C)=O)CCN(C(=O)COc2ccccc2Cl)CC(O)C1 56469,c1(C(=O)NCCC(C)CCNC(=O)CC2CC(F)(F)C2)cc(F)c(F)cc1O 56470,c1(OC)cc(CN2CCCC2CNC(c2cc([N+](=O)[O-])cs2)=O)c(OC)cc1C 56471,c1(C(=O)NC23C(NC(c4cnns4)=O)CC(CC2)C3)cc2sccc2cn1 56472,c1(N(C(c2ccco2)=O)CC)ccccc1C 56473,C(=O)(CCCCCC(C)(C)C)N1C(CNC(=O)C=C(C)C2CC2)CC(COC)C1 56474,Cc1cnsc1C(=O)NCC1(NC(C2CCC2CN(C)C)=O)CCCC1 56475,N1(C(CCCC2(NC(C3C(C)C3)=O)CCC2)=O)CC(S(C)(=O)=O)C1 56476,c1(C(N2CC=CC(NC(C(C=C=C)C)=O)C2)=O)cc([N+](=O)[O-])n[nH]1 56477,N1(C2CCN(C(CC3(OC)CCC3)=O)C2)CCN(C(C2CC3CC3C2)=O)CC1 56478,N1(C(c2cncc(SC)c2)C(=O)NC(C(=O)OC)C)CCC(O)C2CCCCC12 56479,C1(CC)CN(C(=O)COCC2CC2)CCC1NC(C1CC(O)(C#N)C1)=O 56480,CCCC(C(=O)N(CCNC(=O)C(c1ccccc1)F)CCOCC)NC(N)=O 56481,c1(NC(c2ccc(CCC(N3CC(F)C(F)C3)=O)[nH]2)=O)cnnc(Cl)c1 56482,C1(NC(CN(C)Cc2nnc(C)n2C)=O)CC2CC1N(C(C1CC=CCC1)=O)C2 56483,N1(C(CC2C(C)(C)CCCO2)=O)CC2CC(C1)CN(C(C1C3CCCCC13)=O)C2 56484,Cc1ccccc1N=c1[nH]c(CN2CCCS(=N)(=O)CC2)nc(=N)[nH]1 56485,c1(Oc2cncc(N3CCC(COC)CC3)n2)nc(C)c(C)c(C)c1C#N 56486,Cc1nc2sccn2c1C(=O)NC1(C2CCCN2C(C2COCCO2)=O)CC1 56487,CC1(C(=O)NCC(c2ccc(O)c(O)c2)O)CCCN(CCN2CCCCC2)C1 56488,c1(C(=O)NC2C(CNC(C(COCC)(C)C)=O)C2)ccc(P(C)(C)=O)nc1 56489,c1(C(=O)NC(c2cccc(F)c2)C)nc(C2=CCC(O)CC2)c2ccccn12 56490,c1(C(N(C2CCCN(C(=O)C(F)=CCCF)C2)CC)=O)cnc(C2CC2)nc1O 56491,CCN=c1ccc(C(=O)NC2CCCC2NC(c2ccc3cnoc3c2)=O)c[nH]1 56492,c1(CCC(=O)NCCCN(C(C=CC(CC)=CC)=O)C2CC2)nccn1CC 56493,C1(CC=C)(C(=O)N(C(C)C(C)SC)C)CCN(C(=O)C(CC2CCC2)OC)C1 56494,N1(C(c2c(SCC)nccn2)=O)CCN(C(=O)C2=CCCC2)C(C(C)C)C1 56495,C1(NC(C=C(CC)C)=O)CC2(C1)CC1(CC(NC(c3ccc(CO)cc3)=O)C1)C2 56496,C1(NC(Cc2cc(CC)nn2C)=O)CC(O)CN(C(=O)CCC2(C)CC2)C1 56497,c1(C(=O)NC(CNC(CN(CCC)C)=O)C(C)C)cc(C)c(C)c(S(N)(=O)=O)c1 56498,c1(OCC(=O)NC(CN(C(c2cnc(C(=O)OC)s2)=O)C)C)ccc(F)cn1 56499,CCC(C)C(O)C(C)C(=O)NCCC1(NC(=O)C(C)=CC(C)(C)C)CCCC1 56500,CC1C(NC(=O)C=Cc2ncco2)CCCN1C(c1csc(Br)c1)=O 56501,Cn1ncc(C(N2CCCC2CNC(c2cnn(C3CCC3)c2)=O)=O)n1 56502,c1(OC)c(Cl)ccc(C(=O)NC2(C)CN(C(c3cc(N(C)C)ccn3)=O)C2)c1N 56503,C1(C(N2C(c3c(C)ccs3)CCC2)=O)CC(F)(F)CCO1 56504,N1(C(C(C(=O)OCC)F)=O)CCC(NC(c2ccc(CC)cc2F)=O)C12CC2 56505,C(CCN=c1[nH]c(=NC(C)c2nccs2)[nH]c2c1CSC2)OCC 56506,C(C)(CC(C)NC(=O)CNC(c1cscn1)=O)NC(C1(CCOC)CCC1)=O 56507,N1(C(CNC(C)=O)=O)CC(O)CC1CNC(=O)C(CO)c1ccccc1 56508,c1(OC(F)F)ccc(-c2ncn(C3CCC3)n2)cc1.C1(C2CC2)CCCO1 56509,C1(NC(c2cc(C)cc(F)c2)=O)CCC(O)CN(C(=O)COCC(F)(F)F)C1 56510,N1(C(c2cc(CC)oc2C)=O)CCC(CC(=O)NC23CC(C2)C3)C(O)C1 56511,N1(C(c2csc(C)c2C)=O)C(C)CC2CN(C(=O)CCC3(C)CC3(F)F)CC12 56512,Cc1ccc2oc(C(=O)NC3(C)CC(NC(=O)COC4CCCCC4)C3)cc2n1 56513,CCC(CC)(CC)C(=O)N1CCN(C(=O)Cc2nc(C(C)C)c(C)s2)C(C)C1 56514,N1(C(CCNC(COC)=O)=O)CCN(C)C(CNC(c2cc3ccsc3[nH]2)=O)C1 56515,C(=O)(CCCN=c1nccc[nH]1)N1CCC(NC(c2c(C)nsc2C)=O)CC1C 56516,C(N=c1[nH]c2cc(Cl)c(S(=O)(=O)NCC(Cl)(Cl)Cl)cc2s1)C1C(C)OCC1 56517,C1(NC(c2c(CC)non2)=O)COC2(C1)CN(C(C1(C)CCC(C)CC1)=O)C2 56518,C1(F)(CNC(C2CCC(=C)CC2)=O)CCCN(C(C2(F)CC=CCC2)=O)CC1 56519,N1(C(c2cccc(C)c2Br)=O)CC(NC(C2(O)CCC2)=O)CC12CCCC2 56520,c1(Cc2ccc(C(N3CCCC3CF)C(=O)NCC(F)F)cn2)ccc(F)cc1 56521,C1(C(=O)NCC(CC)N2CCCC2)CCCCN1C(C1CC(F)CN1C)=O 56522,C1(CNC(C2CC3CCC2O3)=O)CN(C(=O)CSc2ccccc2O)CC1(F)F 56523,c1(C(N2CC(C)C(NC(C3(C)C=CCCC3)=O)C2)=O)cnc2c(Cl)cccn12 56524,N1(C(C2C(C)=C2)=O)CCCCC(CNC(C2CNC(=O)CC2C)=O)C1 56525,c1(CN(C(CCN(S(C)(=O)=O)C)=O)C2CN(Cc3cccnc3)C2)ccc(F)cc1 56526,N1(C(=O)OC(C)(C)C)CCC2CCN(Cc3ccccc3)C2C1 56527,CCS(=O)(=O)c1ccc(CN2CC(NC(=O)CCC(=O)NC)C(F)(F)C2)cc1 56528,c1(C(N(CCCNC(C2CC23CCOC3)=O)C)=O)ccc(Br)c(F)c1F 56529,C1(CCC(=O)Nc2c(SC(c3cccs3)CC)c[nH]c2)(NC(C)=O)CCCCC1 56530,c1(C(=O)NC2C(NC(C=CCC)=O)CC2)cc2ccc(Cl)cc2c(=O)o1 56531,Cc1c(C(N2CCC(O)(CNC(=O)C(C)(C)CO)C2)=O)cc(Br)cc1N 56532,C(=O)(CC(C)(C)Cc1ccc(Cl)cc1)NC(CC)(C)CNC(c1cccnn1)=O 56533,n1(CCCC)nnnc1C(c1cccn1C1CC1)NCC(C)(C1CC1)OC 56534,c1(C(N2CCCC(CCC(=O)NCCCNC(=O)OC)C2)=O)ccc(C)c(O)n1 56535,C12(C(=O)OC)CC1CN(C(=O)C(CSC)NC(=O)C(C(C)C)N(C)C)C2 56536,CCCC(C(=O)NC(C(=O)NC)C1CCCC1)NC(c1cnn(C)n1)=O 56537,c1(N2CCOCC(NC(CC(C(F)(F)F)OC)=O)C2)nc(Cl)nc2c1ncn2C 56538,C#CC1CN(C(=O)Cc2ncc(F)cc2F)CCN1C(C1CCC=CCCC1)=O 56539,c1(-c2cn(CCN(C(C=C(CC)CC)=O)C)nn2)c(F)cccc1F 56540,C1(NC(c2nc(C)oc2C)=O)CC2(NC(=O)C(C)c3cccs3)COC1C2 56541,Cc1cc(=NCCCC(C)(C)NC(=O)CCc2ncc(F)cn2)[nH]c(C(C)C)n1 56542,C1(C(C)C)CCN(C(=O)C(C#N)C2CC2)CC1.C(=O)(CC(C1CC1)C1CC1)N 56543,C1(C(N(C)CC2CCC2)=O)CC2C=CC1N(C(C(CO)C1CC1)=O)C2 56544,C(=O)(C(F)C1=CCCCC1)N1C(CN(C(COCCSC)=O)C)CCC1 56545,c1(C(=O)NC2C(NC(C(Br)=C(C)C)=O)CC2)cc2ncccc2o1 56546,N1(C(c2ccnc(C)n2)=O)CC2CCCCN2CC1CNC(c1oncc1C)=O 56547,N1(C(C(C=C)O)=O)CC2CCC1C1CN(C(c3c(F)cc(F)c(F)c3F)=O)CC21 56548,C1(OC)COCCC1(c1nnnn1C1CCC1)NCCC(=O)Nc1ccccc1 56549,c1(C(=O)NC(C)CCCNC(=O)CC2CCCS2(=O)=O)ncccc1C#N 56550,O=C(C(F)CC1CC1)NC1CCCC1NC(c1cnn(C2CC2)c1)=O 56551,C(=O)(C(C)C(C)CC)N1CCC(NC(CCc2ccc(OC)cc2)=O)C1C 56552,c1(C(=O)OC)ccc(CN(C)C(C2CCCN(C(=O)OC(C)(C)C)C2)=O)cc1Cl 56553,N1(C(c2ccc(OCC)cc2)=O)CCN(C(C2(C)CC2C)=O)CC1c1cn[nH]c1 56554,CCC(c1ccc(C)cc1)=CC(=O)NC(CNC(c1n[nH]cc1OC)=O)CO 56555,c1(C(N(C)CCOCCN(C)C(C2(C)CC2F)=O)=O)ccc2c(c1)OCC2 56556,N1(C(C2CCCC(OC)C2)=O)CC2(CCN(C(c3ccc4c(c3)NCC4)=O)C2)C1 56557,C(=O)(CCC(=O)NC(C)(C)CC(=O)NCCC1(COC)CCC1)NCC 56558,CC1(CNC(=O)NC2(c3cccc(O)c3)CCCC2)CCCCCC1 56559,C1(SC)CN(C(c2c(C)nsc2C)=O)CC1NC(=O)CCc1cscn1 56560,c1(SC)ccccc1-n1nc(CNC(C)=O)nc1-c1cccc(C2CCOC2)c1 56561,c1(C(c2nnnn2CC(F)F)NCCCc2n(C)ncc2)snc(OCO)c1Br 56562,N1(C(CC(CC)(C)C)=O)CCC2(CCCN2C(c2sccc2C)=O)C1 56563,C1(C(=O)NC2CCCC2NC(C2(CO)COC2)=O)CC12CC(F)(F)C2 56564,CCCCC(C(=O)NCC1(F)CCN(C(=O)C(O)(C2CC2)C2CC2)C1)C(C)C 56565,N1(C(C(F)=CC)=O)CCC(C2CCCN(C(c3n[nH]c(CC)c3Cl)=O)C2)C1 56566,C12(NC(C3CCCOC3c3ncc[nH]3)=O)CC1CN(C(C1(O)CC1)=O)C2 56567,C1(CNC(COCCC(C)C)=O)COCCN(C(C2OCCOC2C)=O)C1 56568,c1(C(=O)OC)cc(Cl)c(OC)cc1CN1CCCC(CS(C)(=O)=O)C1 56569,C1(C(=O)NC(CC)(C)CC)N(C(c2c[nH]c(=NC)o2)=O)CCCC1(C)C 56570,N1(C(C2CC2C2CC2)=O)CC2(CNC(C34CCCC(O)(CC3)C4)=O)CC1CCO2 56571,Cc1nc(Cc2ccccc2)oc1C(=O)NCC1CCN1C(C1CC1F)=O 56572,C1(NC(CC(CC)O)=O)CC2CCC(C1)N2C(=O)C(c1ccc(F)cc1F)C 56573,C(c1cccc(Br)c1)=CC(=O)N(CCC#C)CC 56574,C(=O)(C(=O)N=c1ccn(C2CC2(F)F)[nH]1)N1C(c2n(C)cnc2)CCC1 56575,C(CNC(=O)CC1(C)CCOCC1)(CC(=O)NCCC1(C)N=N1)OC 56576,C1(NC(CCNC(=O)NC)=O)CCN(C(c2c(C)ccoc2=O)=O)CCC1(F)F 56577,c1(C(=O)NCC2(O)CN(C(C3CC(OC)C3)=O)C2)nn(-c2cnn(C)c2)nc1C 56578,c1(OC)cc(C(=O)NCC(COC)NC(C2(C)CCCCC2C)=O)cnc1C 56579,N1(C(C2C(C)(CC)C2)=O)CC2(C(=O)Nc3cn(C)nc3C#N)CCC1CC2 56580,c1(CNC2C(c3ccc(OC)cc3)C2)ccc(C)nc1O 56581,N1(C(CCSCCCC)=O)CC2CC(N=c3[nH]nc(C(F)(F)F)s3)CC1C2 56582,N1(C(c2cn(C)c(=O)cn2)=O)CC2CCN(C(=O)CC=C(Cl)Cl)CCC2C1 56583,CC1NC(=O)CCC1CNC(C1(CNC(c2ccncc2)=O)CCCO1)=O 56584,c1(CC(=O)NC(=O)CO)cccc2cc[nH]c12.C1C2=CCN(CC2)CC(=O)NCC1 56585,C1(CC)CCN(C(=NCC2SCCS2)NCC(=O)NC(C)C)C1 56586,N1(C(c2cc(OC)cc(Cl)c2)=O)CC(NC(C2COC(=O)C2)=O)CC2(CC2)C1 56587,c1(C(=O)NCC2(C)CCCN2C(C2CC3C(C2)C3(F)F)=O)ncc2[nH]ncc2n1 56588,N1(C(C(C)=C(C)C)=O)CCC(NC(C2(C)CC2(F)F)=O)C(C)C1 56589,C1(OC)CN(C(C2CC3(CCC3)C2)=O)C(C)(CNC(c2ccc(F)cc2Cl)=O)C1 56590,N1(C(c2c(C)cns2)=O)CC(NC(=O)Cn2cc(C#N)cn2)C(C(F)F)C1 56591,CC1CCC(Cl)=C(C(=O)Nc2nc(-c3ccc(Br)s3)cs2)C1 56592,C(=O)(C1CCCc2nncn21)NC1C(C)CCN(C(C2C(C(=C)C)OCC2)=O)C1 56593,N1(C(C(C(C)C)OC)=O)CCC(CNC(=O)C(C)(C)O)C(F)(F)CC1 56594,c1(-n2cc(CN3CCN(C(CC4C(=C)CC4)=O)CC3)nn2)ccc(F)c(C)c1 56595,N1(C(CC2(C)CCOC2)=O)CCC2(CC2)CC1C(=O)NCC1(C#N)CCCCC1 56596,CC(C)C(O)CC(=O)N1CC(F)CC1CC(=O)Nc1ccc(Cl)nc1 56597,Cc1ccc(C(=O)NCC(=C2CN(C(c3ncccc3Cl)=O)C2)F)cn1 56598,C1(CC(N2C(COC)CCC2)=O)(NC(=O)Cn2nccn2)CCCCC1 56599,c1(NCCC(N2C(C)CC(CNC(=O)C(F)(F)F)C2)=O)ccccc1[N+](=O)[O-] 56600,C(c1cnc[nH]1)=CC(=O)NCC1(CNC(c2ncoc2C(F)(F)F)=O)CCCC1 56601,c1(C(N(C)CC2CCN(C(CCCCCC)=O)C2)=O)ccc2cccnc2c1 56602,c1(OC)ccc(C2CC2C(=O)NC2(C)CC(NC(c3ccc(C)s3)=O)C2)cc1 56603,CN1N=C(CC(=O)N2CCC3(NC(c4nsnc4O)=O)CCCCC23)CC1=O 56604,CC(C)(F)CCC(=O)N1CC(NC(=O)CC2COC(C(F)(F)F)C2)C1 56605,O=C1NCc2cc(CNC3CCCCC3Nc3ncncc3Br)ccc21 56606,C1(NC(C2OCCN(CC)C2)=O)(CC)CCN(C(C2(CC)CCCSC2)=O)CC1 56607,C1(NC(c2ccccc2CO)=O)CN(C(=O)CC2CCNC2=O)CC(F)(F)C1 56608,C1(C(N2CC(N3CCC3)C2)=O)CCC(O)CN1C(C1CC2(CSC2)C1)=O 56609,N1(C(C(C)OC)=O)CC2CCC(C1)C(NC(c1cccc(OC(C)C)c1)=O)C2 56610,N1(C(CCCc2nc(C)sc2)=O)CCCC2CN(C(=O)OC(C)(C)C)CCCC12 56611,C1(C2CCN(C(=O)CCc3nc(-c4ccco4)no3)C2)(NC(CC=C=C)=O)CC1 56612,CC1(C)CN(C(c2ccc(=N)[nH]c2)=O)CCC1NC(c1ccc(C(N)=O)cn1)=O 56613,C(=O)(C(F)CC(C)C)N(CCCc1ccc(OC)cc1OC)CCOC 56614,N1(c2nccc(OCC)n2)CCC(C)C(NC(C2CCCC2C)=O)C1C 56615,Cc1ccc(C2=CCC3(CN(C(C(=O)NCCCF)C4CC4(Br)Br)C3)CC2)cc1 56616,c1(NC(c2n(C)nnc2)c2nnnn2CCCF)ccc(O)c(F)c1 56617,C=CC1(C(N2CCOC(C#N)C2)=O)CCN(C(c2cc(CC)no2)=O)CC1 56618,C(=O)(C1=C(C)S(=O)(=O)CC1)NCCCNC(c1c(CC)ncc(Br)c1)=O 56619,C(=O)(C(C)(CC1CCC1)N1CCN(C)CC1)OC 56620,N1(C(C2CCCOC2)=O)CCCC2C1CCN2C(=O)COCCN1CCS(=O)CC1 56621,C(CCCCC(=O)N1CC(NC(=O)CNC(c2cscn2)=O)CC1(C)C)SC 56622,c1(CC)ccc(C)cc1C(=O)NC1CN(C(c2cc(Cl)n(C)n2)=O)CC1C 56623,N1(C(Cc2c(C)noc2)=O)CCC2CN(C(c3cccc(=O)n3C)=O)CCC2C1 56624,C#Cc1cc(C(=O)NC(C2CCN2C(=O)C(=CC2CCCC2)C)C)ccc1C 56625,C(CCCOC)(C(=O)NCCCN(CC(C)C)C)NC(c1c(CC)cno1)=O 56626,c1(NC(=O)CNC(=O)NCCC2CCCN2Cc2cccnc2)ccc(F)cc1 56627,c1(C(N2CCC(C(C)(C)NC(C(C)O)=O)CC2)=O)cc2occc2s1 56628,c1(C2C(C(=O)NCC3C(CNC(C(N)=O)=O)C3)C2)ccc(F)c(F)c1 56629,c1(CC)nnsc1C(=O)NCC(C)(O)CNC(=O)CCC1CCCOC1 56630,C(=O)(C(C)(O)CC(F)F)NCC(CN(C(CCn1c(C)nc(C)n1)=O)C)(C)C 56631,c1(C(C(N2CCC(NC(Cn3c(=N)nc[nH]3)=O)(CF)C2)=O)=O)ccc(F)cc1F 56632,O(NC(=O)C(CCOC)NC(=O)C(C)COC)C(C=C)C 56633,CC(C)(CC(=O)NCC1CC1NC(=O)CCn1cc(Br)cn1)CC(F)F 56634,c1(CC(C)C)ccc(C=CC(=O)NCC2CC(CNC(=O)CO)CO2)cc1 56635,Cc1ccc(-n2cc(C(C)N(C)C(C3CCN(C)C3)=O)nn2)c(Br)c1 56636,C(=O)(C(O)CC(F)(F)F)N1CC(CC(C)NC(=O)C(C)(C)C(F)(F)F)C1 56637,C1(NC(c2noc(C3CC3)n2)=O)C2CCC1CN(C(c1ccnc(Cl)n1)=O)C2 56638,c1(C(N(C)CC2(O)CCN(C(CCC#CC)=O)C2)=O)cnc(C)c(C)c1 56639,C=CCCCCC(=O)OCc1csc(C(C)(F)F)n1 56640,C1(C(N2CC3CC(NC(=O)C(C)c4cccs4)C2C3)=O)(CC)CCC(F)(F)CC1 56641,C(=O)(N=c1[nH]c(S(C)=O)ncc1Br)N1CCCC(COC(C)(C)C)C1 56642,N1(C(Cc2c(C)cco2)=O)CCc2sccc2C1CNC(=O)C(Cl)=CCl 56643,N1(c2nccc(OCC)n2)CC2(C)CN(C(c3ccncc3)=O)CC2(C)C1 56644,CC1CC(C(=O)NCC2CC(C(=O)NC3(C)CC=CC3)C2)CCS1 56645,C1(N=c2cnc3cc(F)c(F)cc3[nH]2)(CC)CCN(C(C2CCC(C)O2)=O)CC1 56646,C1(C(=O)NCC(C)OCCO)(CC)CCCN1C(=O)CN1CCOC1=O 56647,C1(NC(CCc2ncc(C)[nH]2)=O)(CO)CCN(C(c2occc2Br)=O)CC1 56648,S(=O)(=O)(c1cccc(C(=O)O)c1)N1CCN(C)C(CC2CC3N(OC)C(CC3)C2)C1 56649,c1(C(=O)O)ccc2c(c1)CCC2NC(c1nc(F)ccc1Cl)=O 56650,C1(CC)(NC(=O)C(C)CC(N)=O)CCCN(C(=O)C(c2cccc(C)c2)OC)C1 56651,c1(CC)ccc(C(c2nnnn2C2COC2)Nc2ccc(C)nc2)c(C)c1 56652,N1(C(CN(C)CC)=O)CCC(Nc2nccc(C(F)(F)F)n2)C(C)C1 56653,Cc1nc(C(N2CC(NC(c3cn(C)c(=O)n3C)=O)C3CC23)=O)c(C)n1C1CC1 56654,C(=O)(NN1CCc2ccc(F)cc21)NC1CCCN(C(=O)OC(C)(C)C)CC1 56655,CC(C)CC(C(=O)NCc1conc1C1CC1)ONC(=O)CC1CCOCC1 56656,C(=O)(C(O)CC(C)C)N1C(CCNC(c2c(OC)noc2C)=O)CSCC1 56657,c1(C(=O)OCC)cnc(NC(C2CCCN2C(=O)NC2CC2C)=O)cn1 56658,N1(C(CCOCC)=O)CC2(CCC(NC(=O)C(=O)NCC(F)F)CC2)C1 56659,c1(C(=O)NCC2C(NC(CCOC)=O)CC2)ccc(CN2CCCCC2=O)cc1 56660,c1(OC)c(C(N2CCCC(CCF)C2)=O)sc2nccnc12 56661,C1(NC(C(=O)NCc2nc(C3CC3)cs2)=O)CCOc2ccccc2C1 56662,C1(C2(O)CCOCC2)(C(=O)NC2CC3CC(NC(C(CC=C)C)=O)C2C3)CC1 56663,C=CCC(C(=O)NC1(CNC(=O)C(C)CC(F)F)CCCCCC1)C(C)C 56664,N1(C(CCCCC(=O)OC)=O)CCC2C(CCN2Cc2ccc(Br)cc2I)C1 56665,C1(C(=O)NCC(O)C(=O)NC2CC(CO)C2)CCC(O)CC1 56666,CN1CCN(C(C2(CO)COC2)=O)CC1CNC(=O)CSCc1ccncc1 56667,C(=O)(CCCCCC#N)NC(CCCC)CNC(=O)Cc1ccc(F)cc1 56668,C(=O)(C(CC(N)=O)NC(c1cn(C(C)C)nn1)=O)NCC(CC(C)C)O 56669,C1(c2nnnn2C)(NCC2(CC(C)C)CCC2)CCCN(C)C1 56670,C(=O)(C1=CCCN(C(C2CCN(C(c3ccc(Br)cc3)=O)CC2)=O)C1)OC 56671,c1(CONC(c2ccc(CNC(CC(C)(C)O)=O)o2)=O)ccc2c(c1)CC2 56672,c1(C(=O)NC2CC(O)(CNC(C3C(C)C3)=O)C2)cnc2[nH]nnc2c1 56673,CC1(CC(N2CCC(OCC3CC3)C2)=O)CN(C(=O)CCN2CCC2)C1 56674,c1(C(N2CCN(C(C(CC)C)=O)C(c3ccccn3)C2)=O)ccn2cncc2c1 56675,c1(CCC(=O)N(CCNC(=O)CC(C)C)CC)cccc(C(F)(F)F)c1 56676,N1(C(C)C)CCN(C(C23CC(CN2C(=O)C(F)(F)CO)C3)=O)CC1 56677,c1(NC(c2[nH]nc(SC)c2C#N)=O)ccc2ncc(-c3cccc(F)c3F)n2c1 56678,C1(NC(C(C)Cc2cccnc2)=O)COCCN(C(c2cc(F)ccc2N)=O)C1 56679,c1(C(=O)NC(CN(C)C(C2(Cl)CC2(C)C)=O)(CO)CO)ccc2ccoc2c1 56680,C(=O)(C1=NOC(CNC(c2cncc(NC)c2)=O)C1)Nc1cc(COC)no1 56681,c12ncccc1OCN2.n1(C(C)(C)C)nccc1-c1cn(CC2CS(=O)(=O)C2)nn1 56682,C(=O)(C(O)C(C)C)NC(C(N1CC(O)(CC=C)C1)=O)CO 56683,c1(CN(C(=O)CC2(c3ccccc3)COC2)CC=C)cccc(F)c1F 56684,c1(C(N(C2CC(C(=O)OCC)C2)CC)=O)ccc(N2CCOCC2)c(F)c1 56685,N1(C(c2c(C(C)C)cnn2C)=O)CCC(C)C(NC(=O)C=CCO)C1 56686,CN1CCC(Nc2cc(NCc3nc(C(F)(F)F)n[nH]3)ncn2)CC1=O 56687,c1(C(=O)O)ccc(C(N2CC(Cc3ccc(Cl)c(F)c3)C2)=O)c(F)c1 56688,c1(C(N2C3C(NC(c4c(CC)onc4)=O)CC(C3)C2)=O)c(C)ccc2n[nH]cc12 56689,C(CC(=O)NC(CO)C(N)=O)(C(C)(C)C)NC(C(C)n1cccn1)=O 56690,N1(C(CC=CCNC(CCCNC(=O)OC)=O)=O)CC2CC1C1CC21 56691,C1(C(=O)NCC23CC(CNC(=O)CCn4cccc4)(OC2)C3)CC2OC1C1CC21 56692,S(=O)(=O)(c1cc(F)c(F)cc1[N+](=O)[O-])NC(c1ccc(C(F)C(F)(F)F)cc1)=O 56693,N1(C(c2cc(C)c(F)cc2Cl)=O)CC(C)CN(C(c2ccc(N)cc2)=O)C(C)C1 56694,N1(CC(=O)OCCC2CCOCC2)CCN(C(=O)Nc2ccccc2)CC1 56695,c1(CC)nc(N2CC(CNC(c3cc(OC)n[nH]3)=O)(OC)C2)cc(C(C)(C)C)n1 56696,c1(C(=O)NC2C3CCN(C(CCN(CC)CC)=O)C32)cc2ccc(OC)cc2[nH]1 56697,C1(NC(COc2cccc(C)c2C)=O)CN(C(=O)Cc2cc[nH]n2)CCC1(F)F 56698,c1(CC(=O)N(C(C)CN(C(=O)C(O)c2ccco2)C)C)ccccc1C1CC1 56699,CC1CN(C(=O)CC(=O)NC2CC2)CC1CC(=O)N(C)CC1(C)CCCO1 56700,C1(C(=O)NCCC(C)CO)(OC)CCN(C(=O)C(O)C(C)C)C1 56701,N1(C(CCOCCOC)=O)CCC(CC(=O)NC2COCC2F)C1(C)C 56702,C(=O)(C1=CCCCCC1)N1C(CNC(C2CC(OCC)C2)=O)C(C)CC1 56703,N1(C(C(C=C=C)C)=O)CCC(C2CCN(C(c3ccc(=O)n(C)c3)=O)CC2)CC1 56704,C1(C(CC)CC)CC(C(N2CCN(C(=O)CCO)CC2)=O)CCO1 56705,c1(NC(C(CCC2CC2)NC(CCC(CC)=O)=O)=O)cn(C)c(=O)cc1C 56706,C1(NC(c2ccc(CC)s2)=O)CC2CC(NC(C3(c4ccoc4)CC3)=O)C2C1 56707,C1(C(=O)NCC(CC)(C)C(N)=O)CC(C)(C)CCN1C(c1ccc(C(F)F)o1)=O 56708,C1(CN=[N+]=[N-])CCCN(C(=O)CCN(C(=O)CCCC2CC2)C2CC2)C1 56709,N1(C(c2c(COC)cc[nH]2)=O)CCN(C(=O)Cc2ccc3c(c2)CC3)C2(CC2)C1 56710,CCC(CC(F)(F)F)C(=O)NC12CCCC1N(C(=O)C1=NNC(=O)C1)CC2 56711,Cc1cc(C)c(CC(=O)NC2CCC2NC(C2CCC3(CCC3)O2)=O)c(C)c1 56712,C=CC(C)CC(=O)NCC(O)CNC(c1sc(Br)cc1C)=O 56713,CCCC(O)CC(=O)NC1(CF)CCN(C(=O)CN(CC)Cc2ccccc2)C1 56714,c1(NCCOC)ccc(S(=O)(=O)NC2CCC3CC23)cc1Cl 56715,c1cc(=NC2CCCSCC2)[nH]c(C2CC2)n1 56716,C(C)(C)(C(=O)N1CC(C(C(=O)NCC2(COC)CCC2)OC)C1)OC 56717,c1(OC)ccc(OCC(N2CC(NC(=O)CSC(C)(C)C)CC2C)=O)cc1 56718,N1(C(CN2CC(=O)NCC2)=O)CCN(C(C2CCC3CC23)=O)C2(CC2)C1 56719,C(=O)(CC(C(F)(F)F)ON)N1C(C(C)NC(=O)C(F)(F)C(F)F)CCC1 56720,c1(N(CCCOC)C)nc(NC)nc(-n2cccn2)n1.c12ncc(s1)[nH]2.C(C)C 56721,CC1(NC(c2cccc(C3(C)CC3)c2)=O)CCN(C(c2ncccc2Cl)=O)CC1 56722,C(C(C)C(F)C(=O)NCCC(F)(F)C(C)C)NC(c1cc(C)ns1)=O 56723,C1(N(C(CCC(=C)Cl)=O)C)CCCN(C(c2nocc2Br)=O)CC1 56724,CC(=O)C(C)(C)CC(=O)NCCOCCCNC(c1cc(C(N)=O)c[nH]1)=O 56725,C(=O)(C1=CCS(=O)(=O)C1)N1CCCC(CN(C(CC(CCC)C)=O)CC)C1 56726,c1(C(=O)NCCNC(c2cn3c(n2)SCC3)=O)cc2ccc(Cl)nc2s1 56727,C(=O)(C(CC(F)F)N(C)C(C1CCOC1C(C)C)=O)NCC(=C)CC 56728,C1(N2C(=O)C2C2CCCC2)CCSCC1.c1(CC2CCOC2)ccccc1 56729,C(=O)(C(C)(C)CC(C)C)N(CC(C)(C)NC(C(F)=CCC)=O)C.C1(=O)CN1 56730,Cc1ncc(C(=O)NC(C)C(C)(C)C(=O)NC2CN(C(N)=O)C2)c(=N)[nH]1 56731,C(=O)(CCC(F)(F)C(F)(F)F)N(CCC)CCNC(C1(C)CCOC1)=O 56732,C1(NC(C2N(C(CCC)=O)CSC2)=O)CC2CC1N(C(c1cc[n+]([O-])cc1)=O)C2 56733,c1(C(=O)NCC2C(C)CN(C(C3C=CCC3)=O)CC2)cc2cc(F)ccc2s1 56734,c1(C(=O)NCCCNC(CC)=O)ccc(CNC(=O)C(C)CN(C)C)cn1 56735,N1(C(c2c(C#C)cnn2C)=O)CCC2(NC(=O)CCC(=O)NC)CCCC12 56736,Cc1sc(Cl)c(C(=O)NC2CC2CNC(=O)C=CC(=O)N(C)C)c1C 56737,N1(C(C(=O)NCC(C)C)CC(C)C)Cc2c(Cl)cccc2C(C)C1 56738,c1(OC)ccc2c(c1)CCC2NC(c1cccc(Cn2nc(C)cc2C)c1)=O 56739,Cc1cc(C(C)(C)NCc2ncoc2C(F)F)ccc1F 56740,C1(C(N(CCCO)CC#C)=O)(OC)CCN(C(C2(C#N)CCCC2)=O)C1 56741,c1(C(=O)NCC(C(C)(C)C)NC(c2c(NC)snc2C)=O)cc(OC)cnc1F 56742,CC1CCCC(CCNC(C2CCN(C(=O)CCCc3cnn[nH]3)C2)=O)C1 56743,CCC(CC)CC(=O)N(C1CCN(C(=O)C(C)(C)C(C)C)C1)C 56744,Cc1cccc(C(=O)NCCOC2CN(C(C3(C(C)(C)O)CC3)=O)C2)c1F 56745,c1(C(=O)NC2CCN(C(Cc3cncc(C)c3)=O)C2)ccc2c(c1)CCC2=O 56746,C1(C(=O)NCCC(C)N(CCC)C)C=CCCN1C(=O)Cc1ccsc1 56747,C(c1ccc(Cl)cc1Cl)=CC(N1CCN(CCc2c(OC)ccc(Cl)c2)CC1)=O 56748,N1(C(COCC(=C)C)=O)CCCC(N(C)C(c2ccc(Cl)s2)=O)CC1 56749,c1(NC(=O)CCc2ccc(-c3nn[nH]n3)cc2)ccc(F)cc1O 56750,c1(COC)cccc(C(=O)NC2CCCC(NC(=O)CSC(C)(C)C)C2)c1C 56751,C1(C)(NC(C(C)CC2CCC2)=O)CCN(C(=O)CCF)C1 56752,CC1(C)CC(C(N2CCCC(NC(=O)Cc3ccsc3)CC2)=O)CC(C)(C)S1 56753,C1(C(=O)OC)CC12CCC(NC(c1sc(C(F)(F)F)cc1Br)=O)CC2 56754,c1(CC(=O)NC2(CCNC(Cc3cc(C)n(C)n3)=O)CC2)ccc(Cl)c(Cl)c1 56755,C12(CNC(C(CC)NC(N)=O)=O)CCC(CC1)N(C(c1ccc(Cl)c(C)c1)=O)C2 56756,c1(OC)cc(F)cc(F)c1S(=O)(=O)NC(C)(C)Cc1cc(F)cc(F)c1 56757,c1(-c2ccc(C(C)(C)O)cc2)cccc2c(C(=O)Nc3ncc(Br)s3)[nH]nc12 56758,N1(C=O)CCC12CCN(C(c1cc(C)nc(O)c1)=O)CC2.C=C(C)C(=O)OCC 56759,C1(C(N(CC(=O)OC)CC#C)=O)CC12CCN(C(=O)CC(C)(F)F)CC2 56760,c1(C(c2n(CCC)nnn2)NCCCOC(=O)NC)c(Cl)cc(Br)cc1Cl 56761,c1(C(C)NC(CC(CC)(F)F)c2nnnn2CC2CC2)nnc2n1CCOC2 56762,c1(CC(=O)NCC2(F)CC(NC(C=CC(=O)NC3CC3)=O)C2)csc2nccn12 56763,c1(C(=O)NCC2(COC)CN(C(C3CC4CC4C3)=O)C2)cnc2n1CCCC2 56764,C(CC(C(=O)NC(c1cn[nH]c1)C)NC(c1[nH]ccc1C)=O)OCC 56765,C(=O)(C(C)(F)C(=O)NCC(C)(F)CNC(=O)C(C)(C)c1cccnc1)OC 56766,S(=O)(=O)(c1ccc(I)cc1)N1CCN(C(c2ccc(NC)cc2)=O)CC1C 56767,N1(CN2C(C(CC)(C)C)CCC2)CCCC(C(=O)NCC(O)CO)C1=O 56768,C1(NC(C2CC23CCC3)=O)(CNC(C2CCCS2)=O)CC2CCC1CC2 56769,N1(C(C(CC=CCC)C)=O)CC(NC(=O)CC2(C#N)CC2)CC(C)C1 56770,C(C(C)(O)CC(=O)NCC1CC(C)(C)CN1C(c1cc(Cl)ns1)=O)OC 56771,Cc1ccc(C(C)C(N2CCCC2(C)C(=O)Nc2cncnc2Cl)=O)cc1 56772,c1(C(=O)NC2(C(F)F)CC(=C)C2)cccc(C2CC2)n1 56773,C(=O)(C1c2c[nH]nc2CN1C(c1cc(CO)on1)=O)N(CCCC)CCO 56774,S(=O)(=O)(c1ccccc1N)N(c1ccc(NCCCc2ccccc2)cc1)C 56775,CC(O)(CNC(c1coc(CNC(C2CC23CCCC3)=O)n1)=O)CCO 56776,c1(C(=O)Nc2ccc(NC(C3(CC)COC3)=O)c(C)c2)ccc2c(n1)CCC2 56777,C1(NC(c2cccc3ncsc23)=O)CN(C(c2cnco2)=O)CC12COC2 56778,c1(C(N(CC(C)NC(=O)CC2CCCCC23CC3)CC)=O)ccc(S(N)(=O)=O)s1 56779,N1(C(C2CCN(C)C2=O)=O)CCC(C)(NC(c2cc(O)nc(Cl)c2)=O)CC1 56780,O=C(CCC(=O)c1cccnc1)NC1CCCCC1NC(C1(CC2CC2)CC1)=O 56781,c1(C(=O)NCCCCNC(C2C(C)CCOC2)=O)c(F)ccc(Cl)c1[N+](=O)[O-] 56782,C1(O)(C(C(=O)NC2CCC(C(=O)NC(C3CCCCC3)C)C2)N(C)C)CCCCC1 56783,C(C(=O)N1CC2CC1(CNC(=O)C(F)(F)CC1CC1)C2)(C(C)C)OC 56784,C1(NC(c2c(C)coc2C)=O)C2CCC1N(C(=O)Cc1cscc1Br)C2 56785,n1(CC)nnnc1C(c1nc(C(=O)OC)cs1)NC1CC1c1ccccc1 56786,C(C(=O)OCC)(C(C)C)O.CCC(C(=O)C(=O)NCc1nc(CN)sc1)C1CCC(=O)N1 56787,Cn1nccc1C=CC(=O)NC1CC(NC(c2ccsc2C#N)=O)C1 56788,N1(C(c2c(CC)nccc2)=O)CC(O)CC1(C)C(=O)NC1CC(N2CCCC2)C1 56789,N1(C(C2(CC)CCCCC2)=O)CC2(CC(NC(C3(O)CCC3)=O)c3nccn32)C1 56790,CC1(C)CC(C(=O)NCC(O)(CO)CO)CN(C(=O)Cn2cnnc2O)C1 56791,c1(-c2cccc(OCC)c2F)c(C(=O)NCc2cccn2C)[nH]c2ccccc12 56792,C(=O)(C(F)C(C)CNC(=O)CC1CCSC1)N1CC(CSC)C1 56793,CC1CC(NC(C2COCCOC2)=O)CN(C(c2ccsc2)=O)C1 56794,N1(C(C(C2CCCCC2)=O)=O)CC2(C=C(C(=O)N3CCOC4C(O)CC34)CO2)C1 56795,Cn1ccc(C(N2CCC2CNC(c2n[nH]c(C3CC3)c2Cl)=O)=O)c1C1CCC1 56796,CCCC(C)CC(=O)NC(C)CN(C(c1cc(C)no1)=O)CC 56797,N1(C(c2n(C)cnc2)=O)C2CCC(C2)C1CC(N1CC2(CSC2)C1)=O 56798,N1(C(=O)C(F)F)CCCC2C(CCCN2C(c2cc(F)c[nH]2)=O)C1 56799,C1(N(C(=O)CCNS(C)(=O)=O)C)CC(C)(NC(C2CC(C(F)(F)F)C2)=O)C1 56800,C(=O)(C#CC1(C)CCCO1)NC(C1CCCN1C(c1cnccc1Cl)=O)(C)C 56801,c1(C(N2CC3C(CNC(c4cnc(C(C)C)s4)=O)C3C2)=O)ccc(Cl)c(F)c1N 56802,c1(N)cccc(Cl)c1O.CC(O)C=O.C1(C)C=CC(=O)N1CCO 56803,C(=O)(CCCCCCCC)N1CCC(O)(CN(C(CC2CC(=C)C2)=O)C)C1 56804,Cc1snnc1C(=O)NCC1CCC(NC(C2CC(O)C2)=O)C1 56805,N1(C(c2n(CC)ncc2)=O)CC2(C(=O)NC(COC)C(C)C)CCC1CC2 56806,C1(NC(C(C)(CO)NC(C(CN(C)C)N(C)C)=O)=O)CN(C)CC1(F)F 56807,C(C(C)(F)C(C)C)NC(c1c(CNC(CSC(C)C)=O)cco1)=O 56808,n1(CC(C)(C)CO)nc(-c2ccco2)nc1-c1cc(C2CC2)on1 56809,C1(C(N(C2CCC(O)(c3ccccc3)C2)C(C)C)=O)CC(C)CC(C)(C)C1 56810,N1(C(c2sc(C)cc2C)C(=O)NCCC(=O)OCC)CCC(C#N)CC12CC2 56811,C1(CC(=O)N(C)CC2CCCN2C(=O)Cn2cc(Br)cn2)COCC(C)(C)O1 56812,c1(CNC(C2CC(=C)CN2C(=O)CCc2ccc[nH]2)=O)cc(CC)cc(Cl)c1 56813,C1(CNC(CCCOCCOCC)=O)CN(C(C2CCNC2=O)=O)CC1C 56814,c1(C(N(CCN(C(=O)Cc2sccc2C)CC)CC)=O)nn[nH]c1Cl 56815,C=C(C)CCC(=O)N1CCC(NC(C2CC(C)=NO2)=O)C1CC 56816,C1(CNC(C2CCCC2)=O)COCCN(C(C2CCCOCC2)=O)C1 56817,Nc1cc(C(=O)NC2CC3(C2)CC(NC(c2ncncc2F)=O)C3)cc(F)c1O 56818,N1(C(c2c(C)n(C3CC3)nc2)=O)CCC(NC(=O)C2=COCCO2)CC1C1CC1 56819,C(=O)(C(CC(C)C)C(N)=O)NC(C(=O)N(CC#C)C)C(C)C.C1CO1 56820,C(CNC(C1CC1C1CC1)=O)(C(C)(C)C)NC(c1n(CC)ncc1)=O 56821,C(c1cccc(F)c1F)=CC(N1CCC(NC(c2cc(=N)[nH]cc2)=O)(CO)C1)=O 56822,N1(C(c2c(O)ncc(CC)c2)=O)CCCN(C(=O)CCOC)C(C)C1 56823,c1(CCC(N2CC(NC(C(CC)OC)=O)C(C(F)F)C2)=O)cnc2ccccn12 56824,Cc1cc(Br)c(C(=O)NC2CCC(F)(F)C2)cc1Br 56825,C1(NC(CN2CCN(C)CC2)=O)CCSC12CN(C(c1n[nH]cc1Cl)=O)C2 56826,CC1Oc2ccc(C(=O)OCC(=O)N(C)Cc3ccccc3F)cc2NC1=O 56827,c1(C(N2CCC(O)(CNC(C3(C)CC=CCO3)=O)C2)=O)nnn2c1CCC2 56828,c1(C(=O)NCC2C(NC(COC)=O)COC2)cc2ccccc2cc1OCC1CC1 56829,C1(C(=O)NC(C2CN(C(c3c(CC)c(C)sc3)=O)C2)C)CCC(N=[N+]=[N-])C1 56830,N1(C(C2C(C)C2)=O)CC(CNC(=O)Cc2nc[nH]n2)C2(CCC2)C1 56831,c1(CN2CC(CC(=O)Nc3cc(Cl)cnc3Br)OCC2)cc(Br)c(O)cc1O 56832,C(=O)(C1CCc2nccn21)NCCC1(C)CCN(C(COCC(=O)OC)=O)CC1 56833,C(=O)(C1=NOC(CNC(=O)CCc2ccco2)C1)N1C(C#C)CCC1 56834,c1(C(=O)NC(C2CN(C(c3c(NC)cncc3)=O)C2)C)ccc2nc(O)cn2c1 56835,Nc1nonc1C(=O)NCC1(CC(N2CCC(F)C2)=O)CC1 56836,C1(CC#N)CCCN(c2ccnc(NCC3CC3c3cccnc3)n2)C1 56837,CCN(Cc1ccc(F)cc1)N1CCc2cc(CO)ccc2C1 56838,N1(C(C(c2ccccc2)NC(C(C)NC(C)=O)=O)=O)CC2C=CCC(C2)C1 56839,c1(CC(N2C(CN(C(C(F)=C(C)C)=O)C)COCC2)=O)c[nH]c2ccc(Cl)cc12 56840,Cc1cn(C)cc1C(=O)N(CCNC(c1ccccc1C1CC1(F)F)=O)C1CC1 56841,C(CCCCN(C)C(C12CCCC1C2)=O)NC(C1(C(=O)OCC)CC1)=O 56842,c1(C(N2C(C=CC(=O)N(CC(C)(O)C3CC3)C)CCC2)=O)cccc2ccnn12 56843,c1(Cc2nc(C(CC)OCC)n(-c3ccccc3)n2)ccc(Cl)cc1Cl 56844,N1(C(c2c(C)nc(COC)s2)=O)CCCN(C(C2(COCC)COC2)=O)CC1C 56845,c1(C(C)(CO)N(C(c2cn(C3CC3)nn2)=O)CC2CC2)c(F)cccc1F 56846,c1(C(=O)NC2CC(NC(C#CC)=O)C2)ccc(I)c(C)c1 56847,C1(CC(=O)NC(C2CCN(C(c3ncoc3C3CC3)=O)C2)C)CC(=O)NC(=O)C1 56848,Cc1cc(C(=O)NCC2CC2CNC(=O)C(C)N(C)C)nc2ccccc12 56849,N1(C(C(=O)NCCOC)=O)CCC(CO)(CNC(C2CC(=O)N(O)C2)=O)CC1.C(C)=O 56850,CS(=O)(=O)c1ccc(F)c(C(=O)NCC2(F)CC(NC(=O)C(F)F)C2)c1F 56851,c1(C(N(C2CCN(C(=O)C(O)CN3CCCC3)C2)CC)=O)ccc(=O)oc1 56852,C#CC1CC2(CC(C(N3CCN(C(=O)CNC(N)=O)CC3CO)=O)C2)C1 56853,CC(C)CC(C)(CNC(C1(Cl)CC1(C)C)=O)NC(c1cccc(C2(C)CC2)c1)=O 56854,Cc1cc(C(=O)NCCOC2CCN(C(=O)Cn3cccc3)C2)cc2ccsc12 56855,CCC(C(=O)N1CCC(C(=O)N(CC(C)(C)O)C2CCC2)C1)C(C)(C)CC 56856,c1(OCC)cccc(C(N2CC(NC(C3CCC3(F)F)=O)CC2CO)=O)c1N 56857,C1(C(=O)NCCN(CCC#C)C)CC2(CCC2)CN1C(=O)C(F)C1CCC1 56858,c1(C(N2CCCC(N(C(C(CC)N(C)C)=O)C)CC2)=O)cc2n(n1)CCNC2=O 56859,N1(C(=O)NCc2ccc(OC)s2)CCCCC1C1OCCO1 56860,N(C=CC(=O)C(F)(F)F)C(=O)CC1CN(Cc2cc3ncccc3[nH]2)CCO1 56861,CC(C)CC(C)CC(=O)N1CCN(C(=O)C2=CCCC2C)C2(CC2)C1 56862,C1(NC(CN(CC(C)C)C(c2n(CC#C)cnn2)=O)=O)CCC2(CCC2)C1 56863,C#Cc1cccc(C(=O)NC2CC(CNC(c3cc(OC)n[nH]3)=O)C2(C)C)c1F 56864,c1(C2(C(=O)Nc3c(CC(=O)OCC)onc3)CC(N)C2)cccc(F)c1 56865,N1(C(C2CCC(C)C2)=O)CCOC2(CCN(C(c3cc(Cl)ccc3N)=O)C2)C1 56866,C1(CC(=O)NC2(C(N(CCOC)C)=O)CC2)CCC(C#N)C1 56867,c1(C(=O)NCC2(F)CC(CNC(COCCC(C)C)=O)C2)ccc(F)c(N)c1F 56868,CCCC(C(=O)N1CCC(NC(c2cncs2)=O)C(O)C1)C(C)C 56869,N1(C(c2c(C)ncs2)=O)CCC2(CCCC2NC(c2cc(O)nc(O)c2)=O)CC1 56870,N1(C(CC)=O)C2CCC1CN(C(c1c(C3CC3)cccc1C1CC1)=O)C2 56871,c1(CCC(=O)NC2CCC(NC(=O)CCC3CNC(=O)N3)C2)c(F)cccc1F 56872,c1(OCCC(=O)NC2(C)CCN(C(=O)CC3CC3)C2)ccc(F)cc1Cl 56873,c1(CCC(N2CCC(NC(COCC=C)=O)C(F)C2)=O)csc2ccccc12 56874,C1(CN(C)C)CCN(C(=O)C(O)CNC(c2ccccc2CC#N)=O)CC1 56875,CCC(CC)CC(C(=O)NCSc1ccccc1)N1CCCC(C)C1C 56876,C1(F)(C(N2CCC(NC(=O)C(Cl)=CCl)C2)=O)CCN(Cc2ccccc2)CC1 56877,C1(C(NOCC(=O)NCc2cc(Cl)cs2)=O)CC2(C1)CC(O)C2 56878,N1(CC(N2C(CN(C(c3cncnc3C)=O)CC)CCC2)=O)CCn2nccc21 56879,c1(CC(N2C(C(C(=O)NCCCC3CC(C)C3)(C)C)CCC2)=O)cccc(O)c1 56880,Cc1nc(=NCC2CCN(C(c3ccc(C)n3C)=O)CC2C)[nH]cc1Br 56881,C1(CNC(C(C)OC)=O)CCC(NC(C2CCOC2)=O)CC1 56882,C1(NC(C2CC(F)CN2C(=O)Cn2ncnn2)=O)CCn2ncnc2C1 56883,C#CCC(CC(F)F)C(=O)NC(CNC(c1nccnc1C(N)=O)=O)CC(C)C 56884,Cc1cccc(C2CCCN2C(=O)C(C(C)O)NC(C2COCCC2C)=O)n1 56885,N1(C(c2ccno2)=O)CCC2(CC1)CCN(c1ncc3ccccc3n1)CC2 56886,C(=O)(CC(C)(C)NC(C1COCCC1C)=O)NCC1(OCC)CC1 56887,c1(CC(=O)NC2CC(CC)(CC)N(C(=O)CNC=O)C2)cnn2ccccc12 56888,Cc1nn(CCO)cc1C(=O)N(CC(C)N(C(=O)C(C(C)C)N(C)C)C)C 56889,Cc1ccnc(C(=O)NCCC(C)N(C)C(C2CCC2(F)F)=O)c1N 56890,c1(C(N2CC(NCc3ncccc3Br)CC(F)C2)=O)cc(Br)c(O)c(Br)c1 56891,Cc1cncc(C(=O)NCCN(C(=O)Cc2cnc(C3CC3)[nH]2)C2CC2)c1 56892,S(=O)(=O)(c1cccc2nsnc12)NC(C)C(N1CCC2C(C(=O)O)C2C1)=O 56893,N1(C(C(N2CCNC2=O)C)=O)CCN(C(=O)COCC2(F)CC2)C(C)C1 56894,CCCC(C(=O)NC1CC2C(NC(c3[nH]nnc3C(F)F)=O)C2C1)OC 56895,C=C1COCCN(C(C2(N)CC=CC2)=O)C1 56896,S(=O)(=O)(c1cc(C(F)(F)F)ccc1Cl)NC1CCN(C(c2cscn2)=O)CC1F 56897,N1(C(CC(C=C)C)=O)CCN(C)CC1CNC(c1ccn(CCF)n1)=O 56898,c1(OC)ccc(F)c(N)c1C(N1CCC(C(C)NC(C2C(C)(C)C2(C)C)=O)C1)=O 56899,N1(C(CCN(C(C2(C)CCCO2)=O)CC)=O)CCC(O)C(C)C1 56900,C(=O)(C(CC(C)C)N(C(=O)C(C#N)C(C)C)C)NC(c1c(C)nc(C)[nH]1)C 56901,C(CCN(C)C)(C(=O)NC1CCOC1CN(C)C)NC(C(c1ccncc1)C)=O 56902,CCCCCCC(F)C(=O)N1CCC(CC)C1CNC(c1cc(C)no1)=O 56903,S(=O)(=O)(c1ccc(NCCNS(=O)(=O)NC)c(F)c1)N1CC(COC)OCC1 56904,CCCCCC(O)CNC(=O)CC(CNC(c1c[nH]nc1C(C)C)=O)C1CCC1 56905,C1(NC(N(C2CN3CCC2CC3)C)=O)CN(C)C(C)(C)C1 56906,N1(C(CCNC(C(C)(C)C)=O)=O)CCC(O)C(NC(=O)Cc2csc(Cl)c2)C1 56907,N1(C(c2ccccc2F)=O)CCC2CCCC12C(=O)NCC1C=CCCC1 56908,C1(CC)CN(C(C2CCOC2CNC(c2cccnn2)=O)=O)CCCO1 56909,c1(C(N2C(CCOC)CN(C(=O)C(C)(O)C3CC3)CC2)=O)cc2ccccn2c1 56910,C1(C(=O)NCCN(CCCCCC)C(C)=O)(Cc2ccccc2)CCNC1=O 56911,C1(C(=O)NCC(C(=O)NC2(C(C)O)CC2)N(C)C)(CC)CCOC1 56912,C1(C(C)(C)C)C(NC(C2CC2F)=O)CCN1C(=O)C(=O)N(C)C 56913,C(C)(C(CC(=O)NCC1CCCC1(C)C)NC(C1CCOC1)=O)OC 56914,c1(C2CN(CC(=O)N(C)C(=O)Oc3c(C(=O)OC)scc3)C2)cccc(Br)c1 56915,c1(CC)ccc(C=CC(=O)N(C2CCC(NC(C3(OC)CCC3)=O)C2)C)cc1 56916,c1(CCC(N2CC(O)(CNC(CCCOCC)=O)C2)=O)cccc(C(F)F)c1 56917,C(=O)(C(CC)C(C)C)NC(C(=O)N(CCOCC#C)C)CCC1CC1 56918,C(=O)(C1=NOC(C)C1C)NCC(CCOC)NC(c1ccc(C(F)F)c(Cl)c1)=O 56919,C1(CNC(CCCC(C)(C)C)=O)CN(C(=O)CCC2(C)N=N2)CCC12CCC2 56920,N1(C(c2ccc(OC)s2)=O)C2CCC1C1CC1(NC(c1cc(C)sn1)=O)C2 56921,N1(C(C(CCC)OCC)=O)CCC(CNC(c2cc(C(C)C)on2)=O)CC1C 56922,C(C(C)(CO)NC(c1sccc1NCS(C)(=O)=O)=O)NC(C)=O 56923,C1(CNC(C2(OC)CCOC2)=O)CN(C(c2coc(C)n2)=O)C2(CCC2)C1 56924,c1(C(N2CCCC(NC(Cc3c(C)nccc3)=O)CC2)=O)ccc(Cl)c(C)c1F 56925,N1(C(C(C)=CC2CC2)=O)CCC(NC(c2ccnn2C(C)(C)C)=O)C(CO)C1 56926,C12(CNC(c3cc(COC)no3)=O)CCCC1N(C(C1CCC(=O)C1)=O)CCC2 56927,C(CC1=CCN(CC2CCS(=O)(=O)C2)CC1)NC(CCC(C)OC)=O 56928,c1(OC)cc(C(=O)NC(Cc2ccc(O)cc2)C(N)=O)ncc1-c1cscn1 56929,C(=O)(CCCCCF)NC1C(NC(C(N2CCCCC2=O)C)=O)CCCC1 56930,c1(NC(C2CC3(CCCCC3)C2)Cc2ccc(Cl)cc2)cncc([N+](=O)[O-])c1 56931,C(=O)(C1CCCc2c1ncn2C)NC1CC(C)(NC(CC=C(C)C)=O)C1 56932,c1(C(=O)NCC(CNC(C2CC2C(F)F)=O)OC)cnc[nH]c1=N 56933,N1(C(c2n(C)nc([N+](=O)[O-])c2)=O)CCC2(CC1)CC(CNC(c1cocn1)=O)C2 56934,CCCCC(C(=O)NCCOCCOCC)N(C)C.c1(=O)c(=O)[nH]1 56935,N1(C(C=CC)=O)CCC2(CC1)CC(CNC(C1CC(=O)N(CCC)C1)=O)C2 56936,c1(C(=O)NCC(CC)NC(c2n[nH]c(C)n2)=O)cc(C2CCOCC2)on1 56937,N1(C(c2cc(CC)[nH]n2)=O)CCC(C)(C)C(C(=O)NCc2cc(C)[nH]n2)C1 56938,C(=O)(C1=CC(O)CCC1)NC(C)C(C)(C)NC(C1SCCCS1)=O 56939,C1(C(=O)NCC2(C#N)CC2)CC2C=CC1N(C(C1CCCC(=O)C1)=O)C2 56940,C1(N(C(CCC(=O)NC)=O)C)CCCN(C(c2ccc(O)nn2)=O)CC1 56941,c1(C(=O)NCC2C(NC(C(C)n3cnnn3)=O)C2)coc2cccc(O)c12 56942,Cc1c(CN2CC(C)CC2c2ccccc2F)cccc1F 56943,N(C1CCc2cc(Cl)ccc21)c1ccnc(NC2CCN(C(=O)OCC)C2)n1 56944,N1(C(Cc2nc(=N)[nH][nH]2)=O)CCC(C(N2CC(C3CCCO3)C2)=O)(CO)C1 56945,CCCC(C)(CCC)C(=O)NCCN(C(C1CSCCS1)=O)CC 56946,N1(C(C2N(C(=O)OC(C)(C)C)CSC2)=O)CC(NC(=O)CSC2CC2)CC(F)(F)C1 56947,c1(NCC(C(C)C)O)ccc(S(=O)(=O)N2CCCC(O)C2)cc1F 56948,c1(OC)ccc(Cn2cc(C(C)N(C)CC3CC3(Cl)Cl)nn2)cc1.C1C(=O)O1 56949,CC1CC(F)(F)CCN1C(C1CCN(C(=O)CCn2cccc2)CC1)=O 56950,Cc1c(CC(=O)NCC2(CCNC(C3CC3C(N)=O)=O)CC2)cnn1C 56951,c1(C(=O)NCC2CC(NC(C(CCC)C#N)=O)C2)[nH]c2cc(Cl)ccc2c1C 56952,CCCC(C(O)C(=O)N1CCOC(CF)C1)NC(c1cc(C)c(CC)o1)=O 56953,C(=O)(C(C(C)CC1CC(F)(F)C1)N1CCC(Oc2cccnc2)C1)NC 56954,c1(C(=O)NC(C)C(=O)NCC2CC3(CCCO3)C2)cc(F)cnc1O 56955,S(=O)(=O)(C(F)(F)F)N1CC(NC(=O)CCc2cnc[nH]2)C1 56956,N1(C(CC(C)(C)O)=O)CC(NC(c2csc(Cl)c2)=O)CC(O)C1 56957,C(C1=CCN(C(c2ccc(N(C)C)nc2)=O)CC1)NC(C(C)SCC)=O 56958,N(C(=NCCC1COC(C)(C)C1)NCCF)CC.c12ccc(cc1)c(=O)o2 56959,CC1CCCN(C(c2cncc(NS(C)(=O)=O)c2)=O)C1CCNC(=O)CO 56960,N1(C(C2(S(N)(=O)=O)CC2)=O)CC(NC(=O)Cn2cc([N+](=O)[O-])cn2)C(C2CC2)C1 56961,N#Cc1ccc([N+](=O)[O-])c(CN2CCCC2C(=O)Nc2ncc(Cl)nc2Br)c1 56962,C(=O)(CC(C)(F)F)NC(CN(C(=O)Cc1ccnc(C(F)(F)F)c1)CC)C 56963,C(=O)(C(F)(F)C=Cc1ccccc1)NCCn1cc(C2(C(=O)OC)CCC2)nn1 56964,C(=O)(CCC(C)(C)C#N)NCc1ccc(OC)cc1.C12CC(C13CCC3)C(=O)N2 56965,C(CN=c1[nH]c(C(=O)OC)ns1)(CC(C)C)NC(C1CC(C#C)(O)C1)=O 56966,Fc1ccc(Cl)c(F)c1CNCc1cc(I)ccc1Cl 56967,c1(OC)ccsc1C(=O)NCC(F)CNC(c1ccn(CC(F)(F)F)n1)=O 56968,C(=O)(CC(C)(C)C)NC1CC(C(C(=O)N(C)Cc2cnccn2)F)C1 56969,c1(OC)cccc2c1CN(C(C1C3CC(CC3F)N1Cc1ccc(C)s1)=O)C2 56970,C1(NC(c2c(C)cc(Br)o2)=O)COCCN(C(=O)C(C)O)C1 56971,c1(OC)ccc(C(=O)NCC(CNC(C2(C)SCCCS2)=O)CO)cc1N 56972,Cc1c(C(N2CCOCC2CCNC(=O)CC(C)N(C)C)=O)cccc1Cl 56973,c1(CCNC(=O)NCCP(C)(C)=O)nnc2c(=O)[nH]ccn12 56974,C1(C(=O)NCC)CCCN(S(=O)(=O)CC)C1.C1(=O)C(=O)NCCCN1CC 56975,N1(C(C(CC)N(CC)CC)=O)CC2=C(C1)CN(C(c1cc3n(c1)CCCC3)=O)C2 56976,C(=O)(C1CCc2nccn21)NCc1occ(C(N(C2CCC2)CCN(C)C)=O)n1 56977,C1(CNC(=O)C2CC2)(Cc2occ(C(=O)NCC(C3(C)CC3)SC)c2)CC=CC1 56978,C1(N(C(C2(NC(CC(C)O)=O)CC(O)C2)=O)C)CCN(C)C1=O 56979,Cc1c(C(=O)NCC(C)CNC(=O)COCC2CCOC2)ccc(F)c1F 56980,CC(C)C(F)(CNC(c1ccn(C)c1)=O)C(=O)NC1C(O)C2CCOC12 56981,C=CC1(C(=O)NC(C)CN(C(C2C=C(C)CS2)=O)CC)CCOCC1 56982,c1(NC(=O)NC2CC(CCSC)C2)ccc2c(c1)OCCO2 56983,N1(C(C2C(C(=O)OC)C2)=O)CC(CNC(=O)CC(C)(C)SC)OC(C)(C)C1 56984,C1(CC)C(C(=O)NC2(CF)CN(C(c3cnc(C)nc3)=O)C2)CCN1C 56985,N1(C(C2N(C(CCC)=O)CCCC2)=O)CC2(NC(C3CCC3C)=O)CCC1CC2 56986,c1(C(=O)NCCCC(C)NC(C2C3CCCC23)=O)cc2c[nH]cnc-2n1 56987,CCC(C)(C)C(=O)N1CCC(C(C)CNC(=O)Cc2csnc2C)CC1 56988,N#Cc1cc(Cl)cnc1N1CCCC(C(N2CCCC2c2ccncc2)=O)C1 56989,C1(NC(C(n2c(C)ncc2)C)=O)CN(C(c2scnc2C(C)C)=O)CCC1F 56990,Cc1cc(CNC(c2cnn(CCNC(=O)C(O)C(C)(C)C)c2)=O)cnc1F 56991,N1(C(c2c(Cl)cc(C)s2)=O)CC(C)CCC1CNC(c1ccc(F)s1)=O 56992,CCC(C)CC(=O)NCC(O)CNC(=O)NC12CC(CC(=O)OC(C)(C)C)(C1)C2 56993,C(CSC(C)(C)C)(C(=O)N1CC(CNC(c2csc(C)c2)=O)C1)NC(C)=O 56994,c1(SCC)nc(C(=O)NCC(C2CCOC2)NC(=O)COCC2CC2)cs1 56995,C=CCC(C)C(=O)NC1CCN(C(c2ccc(-c3ccc(F)cc3)o2)=O)CC1 56996,C(=O)(C(C)CCCC(C)C)N1C(C(N2CCC(SC)C2)=O)CC(F)CC1 56997,c1(NC(C2CC(NCc3ccc(C)cc3Br)C2)=O)ccc(C#N)c(Cl)c1 56998,N1(C(c2nc(C(C)C)sc2)=O)CC(NC(=O)C2=CCSC2)C2(CCC2)C1 56999,C1(NC(c2cc(CNC(CC(C)C)=O)[nH]n2)=O)CCCC1(C)C 57000,N1(C(CC(C)n2cccc2)=O)CCC(F)(CN)C1 57001,C(CC)(CC)(CCNC(c1cccc(Cl)c1F)=O)NC(C(CC)n1ccnc1)=O 57002,N1(C(CC(=O)NCC#C)=O)CCC(C)(C)C1C(N1CCC1(C)CCO)=O 57003,c1(NC(C(C(C)C)NC(CCC=C)=O)=O)cnc(Cl)nc1C 57004,C1(OC)CN(C(c2cc(C(C)=O)[nH]n2)=O)C(C)(C(=O)NOCC2CCOCC2)C1 57005,C(C(C1CCCCC1)NC(=O)CCF)(C(C)C)NC(c1ccc(SC)s1)=O 57006,C=CCC(C)(CC)C(=O)NC1CN(C(C2(O)CCOCC2)=O)CC2(CC2)C1 57007,N#Cc1ccc(CCNCc2nnco2)cc1 57008,c1(NC(c2nc[nH]n2)C)[nH]c(=NCC2CC(C(F)(F)F)C2)nc2c1ncn2C 57009,n1(CC)cc(C(=O)NCC23CC(CN2C(=O)CSC)C3)c(C(C)C)n1 57010,c1(COCC(=O)NCC)cn(CCCNC(c2cnn(C(F)F)c2)=O)nn1 57011,c1(CC)[nH]ccc1C(=O)NC(CC1CC1)C(=O)NCC1CC1(F)F 57012,c1(N2CC(C(C)NC(C(n3ncc(C)c3)C)=O)C2)ncnc2[nH]c3ccccc3c12 57013,c1(C(=O)NC2C(OC)CN(C(=O)C(CO)N(C)C)C2)cc2cc(Cl)ccc2n1C 57014,n1(CCOC)ccnc1NC(=O)NC1CCCC1Cc1ccccc1 57015,c1(COC)ccc(NC(C2CN(C(=O)CCc3ccc(F)nc3)CCS2)=O)cc1 57016,c1(C(C)C)cnc(N2CC(C(=O)Nc3ncncc3Cl)C2)c(Cl)c1 57017,N1(C(CCCOCC)=O)CCCC(CN(C(=O)C(n2cc(Cl)cn2)C)C)C1 57018,N1(C(CC(C)C)=O)CCCC(C2CN(C(C3CCc4n[nH]cc4C3)=O)C2)C1 57019,c1(N2C(C3CCN(C(c4ccns4)=O)C3)CCC2)nc(Cl)nc2[nH]ccc12 57020,C1(CCC)C(=O)NCCN1C(=O)NC(c1ccncn1)C 57021,C1(CCOC)(NC(=O)CC(C)(C)C2CC2)CCN(C(c2coc(C(F)F)c2)=O)C1 57022,N(C(=NCc1coc(C)n1)N1CCC(Cc2ccccc2)C1)C(C=C)C 57023,Cc1cc(N2CCN(C(=O)C(C)(C)C)C(C)C2)nc(C2(C)CCCO2)n1.CCO 57024,C12(NC(CNC(=O)OC)=O)CC(C(=O)N(C3CC3)Cc3ccco3)(C1)C2 57025,C1(CNC(c2nnnn2C2CCC2)C2C(c3ccsc3)C2)CC2(CCC2O)C1 57026,N1(C(N)=O)CCC(CNC(=O)Nc2cccc(SC3CC3)c2)CC1 57027,c1(C(=O)NC(CN(C(COCCC=C)=O)C)(C)C)cc2ccccc2nc1O 57028,Cc1cc(C(=O)NCC2CC(F)(CNC(C3(C)CC3(F)Cl)=O)C2)ccn1 57029,c1(OC)ccc(C(=O)C(N2CC3CC3C2C(=O)NOCC(O)CO)=O)cc1Cl 57030,N1(C(=O)NCC2C(C)(C)C2(F)F)CCn2nnc(CO)c2C1 57031,CC1COCCN1CCNC(C1CC12CC(NC(=O)Cc1ccc(O)cc1)C2)=O 57032,CP(C)(=O)C(O)C(=O)N1CCC(CCCCNC(C2CCC(=O)O2)=O)CC1 57033,NS(=O)(=O)CCCC(=O)N1CCN(C(=O)CCCN2CCCCC2)C2CC12 57034,c1(OC)cc(CN2CC=CC2C(=O)Nc2ccc(C)cc2Cl)ccc1OC(C)C 57035,c1(CC(N2CCN(Cc3ccncc3Br)C3CC23)=O)c(F)cccc1Cl 57036,N1(C(C2(C3CC3)CN(C(C(C3CC3)SC)=O)C2)=O)CC(C2=NOCC2)C1 57037,CC12CCCC1N(C(=O)C1=NOCC1)CCN(C(=O)CCC1CCCCCC1)C2 57038,c1(OC)c(C(=O)NC23COC(C2)C(OC(C)C)C3)nc(O)nc1O 57039,C1(=CC(=O)NC2CCC(CNC(Cc3ccn(CC)n3)=O)C2)CN2CCC1CC2 57040,C1(C(N2C(C3CCN(C(c4ccc[n+]([O-])c4)=O)C3)CCC2)=O)OC2CCC1CC2 57041,C(=O)(C(F)(F)C(F)F)N1CCC(CNC(c2ccsc2)=O)CC1 57042,c1(C(=O)NC(CC)CNC(=O)C(C)N(CC)CC)cc(F)ccc1C(F)(F)F 57043,C#CCC(CCCO)NC(C1CCCC1NC(C1CC2(C1)CC21CC1)=O)=O 57044,c1(CC(=O)NCCCN(C(C2C(SC)CCC2)=O)C)ncn2c1COCC2 57045,c1(SCC(=O)NC2CCN(C(C3CCCC3O)=O)C2)n[nH]c(O)n1 57046,C(=O)(CCC(=O)NC1C2CC1N(C(=O)C(C1CCCCCC1)C)C2)NCCC 57047,C1(C(=O)NCC(CNC(C2(N3CCCC3)CCC2)=O)OC)CC(C)CC(C)(C)C1 57048,c1(NC(N2CCC(CC3CCC3)C2)=O)ccc(C(F)(F)F)cc1O 57049,CCCC(CC(C)C)C(=O)NC1CCC(CNC(=O)C(F)(F)c2cncs2)C1 57050,c1(NC(C2(NC(C=CCOC)=O)CC(F)C2)=O)ccc(F)cc1C 57051,C(CC(C)(C)CC(=O)N1CC(NC(c2cn(CCO)nn2)=O)CC1C)OC 57052,C=CCC(CN(C(C)CC)C)C(=O)N(C(=O)CCC(=O)N(C)C)C 57053,c1(C(=O)NCC(CC)NC(=O)C(c2cccnc2)C)nn(C)c(Cl)c1Br 57054,N1(C(C2CCN(C)S2(=O)=O)=O)C2CCC1CN(C(C1CC(CCO)C1)=O)C2 57055,Cn1cc(Cl)cc1C(=O)NCC1CC1CNC(c1cnccc1C(F)(F)F)=O 57056,N1(C(Cc2c(C)n[nH]c2)=O)CC2CCN(C(c3cccc4nsnc34)=O)CC2C1 57057,CC(C)C1=NOC(C(=O)N(C)CCOCCNC(=O)Cn2cc(Br)cn2)C1 57058,Cc1cc(NC(=O)NC(Cn2cc(C(C)(C)O)nn2)CC(C)C)c(C)s1 57059,CC1CCC=C1C(=O)N1CC2CC2(NC(=O)Cn2ccc([N+](=O)[O-])n2)C1 57060,c1(CNC(C2C(C(C)C)CCO2)=O)cnn(C)c1C(=O)NC(C(C)C)C1CC1 57061,C1(C(N2CC(F)(C(=O)NC3(C(N(OC)C)=O)CC3)C2)=O)CC12CCOC2 57062,N1(C(c2ncnc(C)c2C)=O)CC2CCCC1C2CNC(c1ccc(F)cn1)=O 57063,c1(-c2nc(COC)nn2-c2c(CO)cc(Br)cc2C)noc2c1CC(C)CC2 57064,CC1(C)CCC(C(N2CCCC(CC(=O)Nc3cccc(CO)c3)C2)=O)C1 57065,C(=O)(CCCCCCCC1CC1)N1CC(NC(C(CC=C)CC)=O)C(C(F)F)C1 57066,C(C)(C)(C(C)CC(=O)N1CC(C)CC(O)C1)NC(C(C)OCCN(C)C)=O 57067,C1(CNC(=NCCC)NCCC2CCOCC2)CCC2(CCCC2)O1 57068,CC(O)CCCNC(=O)CC1CCCC1NC(c1ccsn1)=O 57069,c1(C(N2C(C(C)NC(Cc3c(C)con3)=O)CCC2)=O)cn(C)c(=O)cc1Cl 57070,N1(C(C(CC)SC)=O)CCCC2(CCN(C(C)C(=O)N(C)C)C2)C1 57071,c1(-c2cn(C(C(N)=O)Cc3ccccc3)nn2)cccc(C(=O)O)n1 57072,c1(C(=O)NC(CNC(CSCC(=O)OC)=O)CO)ccc2c(c1)CCCS2 57073,C(=O)(C(O)CC(C)C)N1CCCC(CN(C(C2CN(c3nncs3)C2)=O)CC)C1 57074,c1(N2CCN(CC3(C(=O)OC)CCNC3)CC2)ccc(F)c(OC)c1 57075,C1(c2cn(Cc3c(CC)ccs3)nn2)C(C)CCN1C(=O)C(C)N1CCC1 57076,c1(C(=O)NC(C2CCOC2)CNC(C2(CC)CC2)=O)ccnc2ccc(F)nc12 57077,N(C1CN(C(C2CCS(=O)(=O)C2)=O)Cc2ccccc21)C(CCS(=O)(=O)NC)=O 57078,c1(CCNC(c2c(C)nn(C)c2)C(=O)OC)ccc2occc2c1 57079,C1(CC(=O)NC(C2(C(=O)NCC(C)Cn3ccnc3)CC2)C)CCCCO1 57080,Cc1cc(-c2cc(C)ccc2F)ccc1CN(CC(C)(C)CO)C 57081,C1(NC(c2c(OC(C)C)n[nH]c2)=O)CCN(C(c2n[nH]cc2Cl)=O)C12CC2 57082,C(=O)(C(C)C(C)COC)N1CC(C(F)(F)C(=O)O)(OC)C1 57083,C(=O)(C(O)C(C)(C)CC)NC1CN(Cc2nc(CCC)on2)CC1(C)C 57084,C1(CC=C)N(c2ncnc(NCCC(O)C(C)C)c2C)CCCC1(C)C 57085,Cn1ncc2nc(Cl)nc(N3CCC(NC(=O)CCC(N)=O)C34CCC4)c12 57086,C1(NC(C2C(CNC(C3(CCC)CCC3)=O)CCC2)=O)CCC(O)C(O)C1 57087,C(=O)(C(C)C(C)(C)C)N1CCC(C2N(C(C(C)OC)=O)CCCC2)C1 57088,c1(C(=O)NCC2CC(NC(C3C(C)C3)=O)C(O)C2)cc([N+](=O)[O-])c(F)cc1N 57089,CC1CCN(C(=O)C(F)C2CCC2)CCN1C(c1cnc(N)c(O)c1)=O 57090,c1(C(N2CC3C(NC(C4C(CCC)C4)=O)(C3)C2)=O)cc(Cl)ccc1N 57091,C(=O)(C#CC1CCCCC1)N1C2CN(C(c3c(NC)cnnc3)=O)C(C2)C1 57092,C1(C(=O)NC2C(C)CCN(C(c3cccs3)=O)C2)CCC2CCCCC2C1 57093,N1(C(C2CCC(NC(C3CCC(C)(CC)O3)=O)C2)=O)CC2CCCCC12C 57094,c1(C(CNC(CCCC)=O)NC(c2[nH]cnc2C)=O)ccc(Cl)cc1 57095,N1(C(C2(CC)CCC2)=O)CCC2(CCOC2)C(CNC(=O)CCC2(O)CCC2)C1 57096,C(=O)(CCCCCN(C)C)NC1(CC=CCNC(C(CC)C)=O)CCC1 57097,CCC(CC(=O)N1CCCC1CCNC(=O)C=C1CCC1)SC 57098,C#CCC(CO)NC(c1n[nH]cc1CNC(c1c[nH]cc1CC)=O)=O 57099,C1(C(C)(C)NC(C=CCOC)=O)CCCN1C(=O)C(n1nccc1C)C 57100,N1(C(CCN(C)CCO)=O)CCC(NC(C2(C)CC(O)CN2C)=O)C(F)C1 57101,C1(C(=O)NCC2(SCC)CC2)CNC(=O)CN1C(=O)C=CC1CCCN1C 57102,C(=O)(CS(=O)(=O)CC(=O)N1CCN(C(=O)C(C)N(C)C)CC1CF)OC 57103,C(=O)(C#CC(C)(C)C)NCCOC1CCN(C(c2nn(C)c(Br)c2)=O)C1 57104,C1(CNC(=O)COC2CCC2)CC2(CO1)CN(C(C1CCC(=O)O1)=O)C2 57105,c1(SCC(=O)N(C)CC2CCN(C(CCSCC)=O)C2)ccc(Cl)cc1 57106,CN=c1[nH]cc(C(N2CC(O)CC2C(=O)NCC2COC(=O)N2)=O)o1 57107,C1(NC(C2CC2C2CC2)=O)CN(C(C2CCCCC2)=O)CCC1(F)F 57108,C1(C(=O)NC2CN(C(c3ccn(C)c3)=O)CC23CC3)CCC2(CC1)CNC(=O)C2 57109,C(=O)(CC(C)C(=O)N1CCC(CNC(c2cnc(S)n2C2CC2)=O)CC1C)OC 57110,C1(C(N(C2(C(=O)NC(C(=O)NC(N)=O)C3CC3)CC2)C)=O)OCCCC1(C)C 57111,N1(C(CSCC)=O)CCCCC1C(=O)NC(c1ccc(C)cc1)C(F)(F)F 57112,Cc1ccc(S(=O)(=O)N2CCCC(NCc3c(C4CC4)cccc3F)C2)cc1C 57113,CCC(O)C(C)(C)C(=O)NCCCN(C)C(c1csc(-c2ccc(Cl)cc2)c1)=O 57114,C(=O)(C(C)(CO)NC(C1CC(C#N)(OC)C1)=O)NCc1n(CC)ncn1 57115,Cc1nc(C2CCCO2)sc1C(=O)NC1COCC1NC(c1ccccc1O)=O 57116,N1(C(=O)OC)CCCC(C(=O)NCC=CCNC(=O)CC2CCCC23CC3)C1 57117,c1(C(N)=O)cc(Cl)ccc1NC(=O)CCC1CNC(=O)N1 57118,C1(NC(C2CCN(C(CC)=O)C2)C(=O)N(C)C)CCC(C(=O)NC)CC1 57119,C1(O)(CNC(C(C)C2CC2)=O)CC2CCC(C1)N2C(c1cnc(S)nc1)=O 57120,N1(c2ccnc(NCc3ccc(F)c(C)c3F)n2)CCCC2(CC1)CNC(=O)C2 57121,N#Cc1cc(S(=O)(=O)N2Cc3c[nH]c(=N)nc3C2)ccc1NCC1(F)CCOC1 57122,C1(C)(NC(C2C(=C)C2)=O)CCN(C(c2ncccc2C(F)(F)F)=O)CC1 57123,C1(N(C(c2cn(-c3ccc(OC)cc3)nn2)=O)C)CN(C(=O)CCF)CC12CC2 57124,CC1OCC2(CCN(C(C3CN(Cc4cccc(Cl)n4)CCS3)=O)CC2)C1N 57125,N1(C(C(C)OC2CCOC2)=O)CC2CC1CN2C(C1CC(C)(C)CN1C)=O 57126,C1(CC(=O)NC(CC=C)CNC(=O)Cc2sccc2C)CCCC(C)(C)CC1 57127,C1(NC(C(C)C2CC2)=O)CCC2(CC1)CN(C(=O)Cc1csc(S)n1)CCO2 57128,Cc1cccc(C)c1CC(N1CCC(CO)C(NC(c2[nH]c(O)nc2C)=O)C1)=O 57129,N1(C(C(C)C(F)(F)F)=O)CCN(C(=O)COc2c(F)cccc2F)C2(CC2)C1 57130,N1(C(C(C)OCC)=O)CCC(N(CC(C)C)C(c2cccnc2CC)=O)CC1 57131,N1(C(C(C)C#N)=O)CCOCC1CC(=O)N(C)CC1(O)CN(C)C1 57132,C1(NC(CCCC)=O)CCCN(C(=O)C=CCOCC(F)(F)F)C1 57133,C1(C)(CCCC(C2CCN(C(c3c(C)cncn3)=O)CC2)=O)NC(=O)NC1=O 57134,C12(CNC(C(C)(C)F)=O)CN(C(c3ccc(OC(F)F)cc3F)=O)CC1CCO2 57135,c1cc2c(NCCOC3CCOCC3)[nH]c(=NCCC(O)C3CCCC3)nc2s1 57136,n1(CC(=O)NC2CCCN(C(C3N(CC)CCC3)=O)C2C)ncc2cccnc12 57137,C(c1ccc(C2CC2)cc1)=CC(N1CCNCC1C1CCCC1)=O 57138,N1(CC(=O)NC(C(=O)OC)C2CCC2)CCN(c2cc(Cl)ncn2)CC1 57139,N1(C(CC(C)(C)O)=O)CCC2(CCCC2NC(c2[nH]nc3ncccc23)=O)C1 57140,CCCC(CN=c1ccc(Br)c(S(=O)(=O)NC(c2nccnc2C)C)[nH]1)OC 57141,c1(C(=O)NC2(CC)CC(F)(F)C2)ncc(NC(=O)COC(C)C)cn1 57142,CC(C)C(CNC(=O)CCC1CCCCO1)NC(=O)CCCN(C)C 57143,C1(C(CC)O)CCCN1C(=O)C=CCNC(=O)CC1(COC)CC1 57144,c1(OC)cccnc1-c1cn(C2(C(=O)NC(C)CC3CCOC3)CCC2)nn1 57145,N1(C(C2(CSS(C)(=O)=O)CC2)=O)CCCN(C(C2CC(C(=O)OC)C2)=O)CCC1 57146,O=C1CCOC(C(N2CCCC2c2cn(CC3COCCO3)nn2)=O)C1 57147,C1(NC(=O)OC)CCCN(CCC(=O)CCOc2ccc(C(C)(C)C)cc2)C1 57148,C1(CCC)CN(C(=O)C(C#N)CC)CCN1C(c1ccnc(O)c1)=O 57149,N1(C(C2(CCC=C)CN(C(=O)C(O)C(C)C)C2)=O)CC(C)(C)C1COC 57150,N1(C(C=C(C)C)=O)CCN2CCN(C(=O)CCc3ccccn3)CC2C1 57151,CC1(C(=O)NCC2(O)CCN(C(=O)C3=CCOCC3)C2)CCC(F)(F)CC1 57152,c1(C(=O)NCC2N(C(C(COC)C)=O)CC2)nc(-c2ccco2)oc1C(C)C 57153,CC(C)C#CC(=O)NCCC(C)NC(=O)CC(C)NC(C1CCCC1)=O 57154,C1(NC(C2C(C)CCOC2)=O)C2CC3C1C3C2C(=O)NCC1(O)CCCCC1 57155,C1(C(N2CC(NC(c3nn(CC)c(O)c3)=O)C3C(C2)C3)=O)CN2CCCN1CC2 57156,c1(N2CCCC(CCNC(CSC(C)C)=O)C2)ccc(C#N)cc1[N+](=O)[O-] 57157,Cc1ncc(Br)c(N2CCC(C(N3CC(O)C(O)C3)=O)C2)n1 57158,C(=O)(CCS(=O)(=O)C1CCCC1)N1CC2CCN(C(CC(C=C)C)=O)CC2C1 57159,Cc1nscc1C(N1CC=CC1CNC(c1cc(C(C)(C)C)n[nH]1)=O)=O 57160,C1(NC(Cc2c(C)non2)=O)CN(C(c2csc(O)n2)=O)CC1C(F)(F)F 57161,c1(C(COC(CNC(C2C(C)CCC2)=O)=O)N(C)C)cccc(C(F)(F)F)c1 57162,C1(C(=O)NC2C(C(=O)OC)CCC2)CCCCN1C(=O)Cc1ccoc1 57163,C(=O)(CC(C)CC(=O)N1CC(=O)CC1C(N1CCOC(C2(C)CC2)C1)=O)OC 57164,C1(C(N(CCC(C)C)CC(C)C)=O)CCC(C)(C)N(C(C2CC=CCC2)=O)C1 57165,c1(C(N2C(C)(C(=O)Nc3cc(C)cc(F)c3)CC2)=O)cnc2ccccc2c1 57166,C1(CC)(NC(C2C(C)C2C)=O)CCCN(C(c2ncc(OC)cn2)=O)C1 57167,CC1=C(C(=O)NC2CCN(C(=O)CC(C)P(C)(C)=O)CC2(C)C)S(=O)(=O)CCO1 57168,Cc1nnc(O)c(C(=O)NCC(O)CN(C(=O)Cc2cn3ccsc3n2)C)c1C 57169,CC1(C)CC(CNC(=O)CNC(=O)C(C)(C)C)N(C(C2SCCCS2)=O)C1 57170,c1(C(N2CCN(C(C(CC(C)C)N(C)C)=O)C(C)C2)=O)c[nH]c2ccccc12 57171,CC1CCN(C(c2cccc(SC(F)F)c2)=O)CCN1C(C1CCCC(=O)N1)=O 57172,c1(CCC(=O)N(CCNC(=O)Cc2cc[nH]c2)CC)c(F)cccc1F 57173,C(=O)(CC(C)(C)C#N)NCC1C(C(=O)NC2CCN(CC)CC2)C1 57174,N1(C(C2CC(C#C)(O)C2)=O)CCC(C)C(NC(C2CC(O)C2)=O)C1 57175,CC(c1ccccc1F)=CC(=O)NC1CC(NC(C2(F)CCCC2)=O)C12CCC2 57176,N1(C(=O)Cn2cccnc2=O)CCC2C(CCCN2C(=O)C=CC2CC2)C1 57177,c1(CC(=O)N(C(CCNC(C(C)SC)=O)C)C)ccccc1[N+](=O)[O-] 57178,CC(C)C(C(C)NC(=O)Cn1cnccc1=O)NC(=O)CCn1cnccc1=O 57179,CN1CCN(C(C2(C#N)CCSCC2)=O)CC1CNC(=O)Cc1cncs1 57180,CC1(C)CCC(O)(CNC(c2ccc(CNC(=O)CC3CCCSC3)nc2)=O)C1 57181,C(=O)(C(C)(C)C(=O)NCC(C)(O)CNC(C1CC2CC2C1)=O)NC 57182,c1(N2CC(C(N3C(C)CCCC3C)=O)C(O)CC2)ncc2[nH]ccc2n1 57183,N1(C(C(C)NC(=O)OC)=O)CC2C(CN(C(=O)CN3CC4CC4C3)C)C2C1 57184,c1(C(N2CCC(O)(C(C)NC(CC=C=C)=O)C2)=O)[nH]c2cc(OC)ccc2c1C 57185,c1(C(=O)NC(C2CCCN2C(=O)CN(C2CCSC2)C)C)nnnn1C(C)(C)C 57186,Cc1[nH]c2ccccc2c1C(=O)NC(C)CN(C(=O)CC1CC(F)C1)C 57187,C1(C)(C(=O)NC(CN(C(c2ccc(C(C)C)nc2)=O)C)C)CC(C(F)(F)F)=NO1 57188,C(=O)(C1CCCn2cncc21)Nc1c(OC)cccc1 57189,Cc1ccc(C(=O)NC2CCN(C(=O)Cc3nc(=N)[nH][nH]3)C(C)C2)cc1C1CC1 57190,CC(C(C)(C)C(=O)NC1CCN(C2CC2)C1=O)NC(=O)C1=COCC1 57191,Cc1cc2[nH]c(C(N3CCCC(NC(c4cc(F)n(C)n4)=O)C3C)=O)cc2o1 57192,c1(C(=O)Nc2ccc(CS(CCOC)=O)nc2)c(SC)nc2ccccc2c1C 57193,C(CCCCNC(c1cnn(CC(F)(F)F)c1)=O)NC(=O)Cc1cncnc1 57194,C1(NC(C(C2(O)CCCCC2)CC)=O)CCN(c2cc(C(C)=O)ncn2)CC1O 57195,c1(C(=O)NC2CCC(NC(Cc3cc(C)ns3)=O)C2)ccc(-n2cncn2)cc1 57196,CCCC(CC)CC(=O)NCC1(NC(C23CCC(N=[N+]=[N-])C2C3)=O)CCCCC1 57197,c1(CNC(C(CCC)O)=O)cccc2c1CN(C(c1sc(CO)nc1C)=O)C2 57198,c1(CCCC(=O)NCCN(C(C2C(C=C)C2)=O)C)ccccc1Br 57199,Cc1nn(C)c(Br)c1C(N1CCCC(N(C(=O)CCOC2CC2)C)C1)=O 57200,C(=O)(CCCC(C)(C)CC)N1CC2C(CNC(c3ccc(C=C)cc3)=O)C2C1 57201,C1(NC(C2C(C)(C)C2)=O)C2CC1CN(C(C1CCN(c3nccs3)CC1)=O)C2 57202,c1(C(=O)NC(C2OCCN(C(c3[nH]cc(CC)c3)=O)C2)C)nccc(Cl)c1Cl 57203,c1(CC)cc(C(=O)N(CC(O)CNC(=O)CN2CC(=O)NC2=O)C)ccc1C 57204,C1(NC(=O)COC2CC(F)(F)C2)CCN(C(c2csc(O)n2)=O)CCC1CO 57205,N1(C(CN(CCC)C)=O)CCC(O)(C(C)NC(c2cc(Br)cn2C)=O)C1 57206,O=C(C1=NOC2(CCC2)C1)NC1CC1CNC(=O)COc1c(Cl)cccc1Cl 57207,C1(NC(C2(OCC)CCSCC2)=O)CN(C(=O)CSc2cnn(C)c2)CCC1F 57208,C1(C)(C(N(CC(C)SC)C)=O)CCCN1C(c1sccc1CO)=O 57209,n1(CC)ncc(C(N2CCOCC2CC(N2CC(O)C2)=O)=O)c1C 57210,CC(C)CCCC(C)NC(C1CC2(C1)CN(C(=O)Cc1noc(C(C)C)n1)C2)=O 57211,C1(CNC(C(C)OCCC(C)C)=O)(CNC(=O)C(N)=O)CC1(F)F 57212,CCCCCCCC(=O)N1C2CCC(C2)C1CNC(C1CCCS(=O)(=O)C1)=O 57213,CCCCCCCCC(C(=O)NCCCSC)N1CC2CSCC2C1 57214,C=C(C)CC(C(=O)N1CCC2(CC2C(=O)NCCCc2ccccn2)C1)OC 57215,C(CS(=O)(=O)CC(=O)NC1C2CC1N(C(C1CCc3nc[nH]c3C1)=O)C2C)OC 57216,c1(N(C(CCN(C(C)=O)C)=O)CCNC(=O)CN(C2CCC2)C)ccccc1F 57217,c1(C(=O)NCC2CC(NC(c3c(CC)cno3)=O)C2)ccc(Br)c(N)c1 57218,C1(CC(=O)NCC(C)CNC(c2ccnn2CCN(C)C)=O)CC=CCN1C 57219,CCC(C(=O)N1CCC(CF)(NC(=O)CCc2ccccc2Cl)C1)C(C)C 57220,c1(OC)ccnc(F)c1C(N1CC(CNC(=O)C(C)SC(F)(F)F)(OC)C1)=O 57221,N1(C(c2c(COC)ccs2)=O)CCN(C(=O)C(F)C(C)(C)O)CC12CCC2 57222,CCC(CCCO)NC(=O)CCSc1cccc(OC)c1 57223,CCC(CC)(CO)C(=O)NCC1CCC2(CN(C(c3sc(F)cc3C)=O)C2)O1 57224,N1(C(C2C(=C)C2C(=O)OC)=O)CCCN(C(C2CC2(Cl)Cl)=O)CCC1 57225,Cc1cc(C(C)C(=O)NC2(CCCCNC(=O)C3=NOCC3)CC2)c(C)o1 57226,c1(CC(=O)NC2CC(C(N3CC(C)OCCC3)=O)C2)cnc2ccccn12 57227,c1(C(=O)NC(C(C)(C)NC(C(C)NC(C)=O)=O)C)c[nH]c2ccc(F)cc2c1=O 57228,C1(NC(C2C(OCC)C2C)=O)CCCN(C(=O)C(C)=C(C)C)C1 57229,C(=O)(CC1=NNC(=O)C1)N1CCN(CCCNC(c2ccnc(C)n2)=O)CC1 57230,C1(NC(CN(S(CC)(=O)=O)C)=O)CCN(C(C2CC2C2(C)COC2)=O)C(C)C1 57231,C(C(C)S(C)(=O)=O)(c1ccc(C)cc1)NC1CN(C(=O)NCc2ccco2)C1 57232,C(=O)(C(C)S(C)(=O)=O)NC1(CCCC(=O)Nc2cccc(C(C)C)c2)CCC1 57233,C1(OCCNC(C(C)OCOC)=O)CCN(C(=O)CC(C)(C)C)CC1 57234,N1(C(C(CCC)O)=O)CCC(C)CC1CNC(c1ccc(CSC)cc1)=O 57235,N1(C(CCCSC(C)(C)C)=O)CCCC2(CNC(c3ccc([N+](=O)[O-])o3)=O)CC12 57236,N1(C(C(CSC)O)=O)CCC12CN(C(=O)CC1(C)CCOCC1)C2 57237,c1(OC)c(Cl)cc(C(N2CCCC2C(=O)NCCC23CC(CCO2)C3)=O)cc1Cl 57238,CS(=O)(=O)CCC(=O)NCC(C1CCOC1)NC(c1cocn1)=O 57239,C(N=c1cc(NCC2CC3CCC3C2)nc[nH]1)C1(COC)CCC1 57240,n1(CCC(=O)NCC2N(C(C(C)C(C)(C)C)=O)CCCC2)cnc2ccccc12 57241,CCC(C)CCC(=O)NC(Cn1cccn1)C(=O)N(C1CCCC1C)C 57242,N(C(=NCCC(=O)N1CCCCC1)NCc1cccs1)CC(CC)(CC)N(C)C 57243,c1(CC)cccc(C(N2CCC(C(C)(C)NC(C3SCC=C3C)=O)CC2)=O)n1 57244,C12(C(=O)NCC3CCN(C(C(CC)c4cccnc4)=O)C3)CC(CN1C1CC1)C2 57245,C(=O)(CC(C)(C)CNC(C)=O)N1CC(OC)C(NC(=O)C(C2CCCCC2)F)C1 57246,C1(C(=O)NC(CC)C(=O)c2ccccc2)CCc2nc(C(C)C)ncc2C1 57247,n1(CC(=O)NCCC(C)NC(=O)CC2CCC23CCC3)nc2ccccn2c1=O 57248,Cc1cc(C(=O)NCC(CC(C)C)NC(c2cc3sccc3[nH]2)=O)nc(C)n1 57249,Cc1n[nH]c(C)c1C(=O)N.C1CCCN(C(c2cnn(Cc3cccs3)c2)=O)C1 57250,CCCCC(O)C(C)C(=O)NC(C)CN(C)C(c1ncc[nH]c1=O)=O 57251,C1(CC)CN(C(c2cc(OC)cs2)=O)CCC1NC(=O)CCc1ncc(C)[nH]1 57252,n1(C(C(=O)N(C(CNC(c2c(CC)n[nH]c2)=O)C)C)C)cnc(C#N)n1 57253,C(=O)(C(C#N)CC)N(CC(=O)NC(C=C)(C)CC)CCC 57254,CC1CC=C(C(=O)N2CC(NC(=O)CCOC3CC3)CC3(CC3)C2)CC1 57255,C1(CNC(CC#N)=O)CCC2(CO1)CC(NC(=O)CCC1CCCCCC1)C2 57256,Cc1[nH]nc2c1CC(C(N1CC(C(N)=O)(CNC(C3COC(=O)N3)=O)C1)=O)CC2 57257,N1(C(C(C)NC(c2ccoc2)=O)=O)CC2(CC(NC(c3cnccn3)=O)CO2)C1 57258,Cn1nc(C(=O)NCCCCCC(=O)NCCc2csnn2)cc1C#N 57259,c1(CC(=O)NCCCN(C(C2ON=C(CC)C2)=O)CC)c[nH]c2cccc(C)c12 57260,C1(NC(C2CN(C)C(=O)C2)=O)CC12CCN(C(c1nccc(C(F)F)n1)=O)CC2 57261,c1(C(=O)NCCCN(C(CC2(COC)CC2)=O)C)cc(C#N)ccc1C 57262,Cc1ccc(Sc2ccccc2C(=O)COC(=O)CC2CSCCO2)c(C)c1 57263,N1(C(C2(OC)CCCOC2)=O)CCC(NC(=O)CCn2nc(C)nc2C)C(O)C1 57264,Cc1cc(C(=O)NC2CC(CCNC(=O)COc3ccsn3)C2)c(N)c(F)c1 57265,c1(C(C2CC2)NC(=O)C(=O)NCC2(F)CCCC2)cnn(-c2ccccc2)n1 57266,N1(C(CC2CCCC(OC)C2)=O)C2CCC1CC(CNC(c1ccc(Cl)s1)=O)C2 57267,O=C(N=c1[nH]nco1)C12CC(C=O)(C1)C2.N1(CCn2ccnc2)CCC(O)CC1 57268,CN1CCC(CO)(CNC(C23CC2CCN3C(=O)C(O)C2CCCC2)=O)C1 57269,C12(C)CCCN(C1)C2=O.C12CCN(CC1)C(=O)N2.c1(COC)ccc(C#N)s1 57270,N1(C(C2C(CC)OCCC2)=O)CC2(C1)CN(C(c1cccc(OC(F)F)c1)=O)C2 57271,Cc1cccc2c1OCC2C(=O)NCCOC(C)(C)CNC(=O)CC1CCOC1 57272,C1(C(C)OC(=O)N(C)C)(CO)CCOCC1.c12cn(nn1)CC(=O)NC2C(C)C 57273,C12(CNC(C3(CNC(C4N(C)CCCC4)=O)CCCC3)=O)CCC(CC1)CC2 57274,Cc1cc(NC(=O)CC2C3CN(C(=O)C=Cc4ccccc4)CC23)cc(C)c1F 57275,CCC(CC)CC(F)C(=O)NC12CC(NC(C3(N4CCOCC4=O)CC3)=O)(C1)C2 57276,C(CNC(=O)C(F)OC(F)(F)F)(C(=O)NC(C(F)(F)F)C1CC1)OC 57277,N1(CC)CC(C)N(c2nnc(-c3nc(N)sc3I)n2CCC#N)CC1C 57278,C1(CNC(c2cccc(C3CCC3)c2)=O)C2CCC(C2)N1C(=O)CC1(O)CCC1 57279,Cc1cc2ccc(C(=O)NC(C)(CNC(=O)CC3(C#N)CCC3)C3CC3)cc2o1 57280,CCC(C)C(=O)C(=O)NCCc1cc(C(N2CCCCC2C(N)=O)=O)no1 57281,C(=O)(CCCC(=O)NC1CCCCC1CNC(C1CC2CCC1C2)=O)NC 57282,c1(C(N(C(C)CC(=O)NC(C)C(F)(F)F)C)=O)cc(F)ccc1F 57283,C(CCC(C(=O)N(C1CCOCC1C)C)NC(c1ccn(C2CC2)n1)=O)OC 57284,c1(C(=O)NCCCN(C(c2nc(OC)oc2)=O)C2CC2)c(Cl)oc2ccccc12 57285,C(=O)(C#CC(C)(C)C)NCC(c1ccc(C)cc1)NC(C(CC)OC)=O 57286,c1(C(N(CCCN(C(C(C)C(C)C(C)(C)C)=O)C)C)=O)cc([N+](=O)[O-])ccc1Cl 57287,C1(OC)CN(C(=O)C=CC2CCCN2C(=O)Cc2ncn(C)c2C)CC12CC2 57288,CC(C)C(F)C(=O)NC1CCN(C(C)C(N2CCCC(C)C2)=O)CC1 57289,c1(C(=O)NC2C(NC(CCC)=O)C2)cccc(N)n1 57290,c1(CC(=O)NCCN(C(=O)CN(C(=O)C(C)C)C)CC)csc(-c2ncccn2)n1 57291,c1(CNC2CN(C(COC)=O)CC2C)cccc(CNC(=O)OC(C)(C)C)c1 57292,C1(C(N2CCC(COC)(NC(=O)CCC(F)F)C2)=O)OC(C)(C)OC1(C)C 57293,CCC(C)CC(C)C(=O)N1CC2CC(C1)N2C(C1(Cl)CC1)=O 57294,CC(C)C(C(=O)N1CCC(CO)C1)C(C)NC(c1nnsc1N)=O 57295,N1(C(C(C(C)C)NC(N)=O)=O)CCCN(C(C2SC3C=CC2CC3)=O)CC1 57296,c1(C(=O)NCC(CNC(C(N2CC(C)C2)C)=O)(C)C)ccccc1C(=O)N(C)C 57297,Cc1n[nH]c(C)c1CCC(=O)NC1(CNC(c2c(C(F)(F)F)cnn2C)=O)CC1 57298,CC1(C)COC(CC(=O)NCCOCCNC(C2(c3ccns3)CC2)=O)C1 57299,C1(NC(CCOCC#C)=O)CCCN(C(c2cc(N)nc(Cl)c2)=O)C1C 57300,c1(N(C)C)ccc(C(=O)NC(C)CCNC(C2CC(OC3CC3)C2)=O)cc1F 57301,c1(C(N2CCCC(C(C)NC(CC=C=C)=O)C2)=O)c(OC)cccc1Cl 57302,CC1=C(C(=O)NCC2CC(NC(c3ccc(Cl)c(Cl)c3)=O)C2)CCCC1 57303,c1(C(N2CCC(CCNC(c3cc(C(N)=O)no3)=O)C2)C)ccccc1Br 57304,C1(NC(C2C(=C)C2)=O)CC2(CCCCN2C(=O)CCc2ccccc2C(N)=O)C1 57305,N1(C(C2CN(S(C)(=O)=O)C2)=O)CCCC(O)(CNC(c2cnc(C(F)F)s2)=O)C1 57306,c1(CC)cn2c(n1)CC(C(N1CC(OCCNC(=O)C(O)C(C)(C)C)C1)=O)CC2 57307,CCCCC(C(=O)OC)NCC1CN(C(=O)OC(C)(C)C)C(C)(C)C1 57308,c1(CC)oc2ccccc2c1CC(=O)NCC(C)N(C)C(c1ccnc(O)c1)=O 57309,C12(C(N3CC(C)C(NC(c4ccnc(O)c4)=O)C3)=O)CCCC1CCC2 57310,N1(C(Cc2c(C)scc2)=O)CC2(C1)CN(C(C1CC(S(C)(=O)=O)C1)=O)CC2CO 57311,N(C1CSCc2ccc(Br)cc21)C(=O)C(c1ccc(O)cc1)O 57312,N1(C(=O)NC(C)Cc2ccccc2)CCC(N)CC1.c1(-c2ccccc2)ccncc1 57313,C1(n2cc(COC)nn2)(C(=O)NC(C)COCCc2ccccc2)CCOCC1 57314,C(=O)(C(C)C(=O)NC1CCCC(NC(=O)C(Cl)=CCl)C1)OC 57315,c1(C(c2n(C(CC)(C)C)nnn2)NC(C)(C)CF)ccc(F)cc1Br 57316,c1(-c2n(C(c3cccc(Br)c3)CC)ccn2)c(C(=O)O)nn2ncccc12 57317,c1(CC)cn2cc(C(N3CCC(N(C(=O)COC(F)(F)F)C)C3)=O)cc(F)c2n1 57318,C1(C(N(C)CC2CCCN2C(c2cc(Br)cn2C)=O)=O)CCCCCC(=O)C1 57319,C1(C(=O)NCC(C)N(C)C(c2csnc2Cl)=O)CCCCC12CCC2 57320,C1(CC(=O)NCC(C2CCN(C(c3scnc3Cl)=O)CC2)C)COCCOC1 57321,C1(Nc2n(C)c(Br)nc2)CCCC(C(=O)NC2CC2)CC1 57322,CC1(C(=O)NCc2ccc(CNC(C3CCC(=O)NC3)=O)cc2)CCCCCC1 57323,N1(Cc2sc(C=O)c(Br)c2Br)CCC2(CC1)CC(CCN1CCCC1=O)CO2 57324,C12(C(=O)OC)COC(COC(=O)C(F)Cc3ccccc3)(C1)C2 57325,C(C(C)(C(N)=O)NC(=O)CCCN(C)C(C1CCCCCC1)=O)OC 57326,C1(NC(c2cc(O)ncn2)=O)C2CCN(C(=O)CCCC3CCCCC3)C12 57327,c1(NC(CCN(C(=O)CCOC2COC2)C)=O)cncc(C(N)=O)c1 57328,C(=O)(C(F)CC(C)(C)NC(c1ccc(CO)s1)=O)N(C1(C#C)CC1)C 57329,C1(F)(CNC(C(=O)NCC)=O)CCC(NC(=O)C=C(C)Cl)C1 57330,N1(C(c2cc(CC)c(F)cc2)=O)CC(C)N(C(=O)CC(F)(F)CC)CC1C 57331,N1(C(=O)CC2CCC(C3CC3)O2)CCN(C(=O)C(O)C2CCCC2)C(C2CC2)C1 57332,C(=O)(C(CCNC(C1(O)CCCC1)=O)OC)N(C(C#C)C1CCC1)C 57333,C=C(C)C(C)(O)C(=O)NC1CCC(NC(c2ccc(CNC(C)=O)cc2)=O)CC1 57334,C1(C(=O)NCc2c(C)ccc(C)c2)CC2CCCCC2N1C(c1cocn1)=O 57335,C1(C(N2CCCC(CNC(C(C)C3CCCO3)=O)C2)=O)CCCCC12OCCO2 57336,C1(CNC(C2CC(CC)C2)=O)(OC)CCN(C(=O)C(O)Cc2cnn(C)c2)CC1 57337,C1(OC)CC(C(N2CC(C(C)C)C2)=O)N(C(=O)Cc2ccns2)C1 57338,c1(C(=O)NCC(CC)NC(C2(C)C=CCCC2)=O)cc2n(n1)CC1(CC1)C2 57339,C(=O)(C(C)(C)S(C)(=O)=O)N1CC(O)(CN(C)C(C2CCC3(CCOC3)O2)=O)C1 57340,N1(C(C(CCCCC)O)=O)CC2(CCCCN2C(C23CC(C)(C2)OC3(C)C)=O)C1 57341,c1(CC(=C)Br)nnc(N2CCC(CCF)CC2)n1CCCc1ccc(OC)cc1 57342,C1(F)(CNC(c2n(C=C)ncc2)=O)CCCN(C(c2ccc(C(F)F)o2)=O)CC1 57343,N1(C(c2cnc(C(C)C)nc2)C(=O)NCC=C)CCC(C2CCOC2)CC1 57344,c1(C(=O)NCC2N(C(COCC)=O)CC(C(F)(F)F)OC2)ccc2occ(C)c2c1 57345,C=CCCC(C)NC(=O)C(C)=CCNC(=O)CCc1cnn[nH]1 57346,Cc1cc(Br)c(C(=O)Nc2ccc(C)c(C(C)(C)C)c2)cc1Cl 57347,C1(C)C2CC3C(C2NC(=O)C2=CCCCO2)C13.CC(C)(CO)C1(OCC(=O)N)CC1 57348,c1(NC(C23CC2CN(Cc2cnn(C4CC4)c2)C3)=O)cc(F)ccn1 57349,Cc1ccc(O)cc1C(=O)NC(CC1CC1)CC(=O)N1CCC(C(F)(F)F)C1 57350,c1(CCC(=O)NC2CCN(C(C(C)=CC)=O)CC2)cccc(C#N)c1 57351,C(=O)(C1CCc2ccccc21)NC1CCC(NC(=O)Cc2cc(C3CC3)on2)C1 57352,CCC(C)CC(C)C(=O)NCC1(C)CCN(C(c2ccnc(F)c2OC)=O)C1 57353,c1(NC(C2CN(C(CC(C)(C)OC)=O)C(C)CC2)=O)cccc2c1OCC2 57354,CC1(C)CN(C(=O)CSC2CC2)C(CNC(C2SCCS2)=O)CO1 57355,C1(O)(C(C)CNC(=O)Cc2cnns2)CCN(Cc2cc(-c3ccoc3)[nH]n2)C1 57356,C1(S(C)(=O)=O)(C(=O)NCC(CC)(C)NC(C2CCN(C)C2C)=O)CCC1 57357,C1(C(=O)NCCCCC=C)CCC2CCC1N2C(c1cnn2c1CCC2)=O 57358,Cc1ccc(NCCC(N2CC(NC(=O)C(Cl)=CCl)CC2C)=O)cc1 57359,C(=O)(CCC=C(C)C)NCC(CNC(C1(CCCC)CCC1)=O)OC 57360,c1(OC(C)C)ccccc1C(=O)NC(C)CNC(C1CCCN1C(C)C)=O 57361,N1(C(=O)COc2ccc(Cl)c(Cl)c2)CCC2(CC1)CN(C(C1C=CCC1)=O)C2 57362,c1(C(=O)NCC(C)CNC(=O)CC2CC23CC3)c[nH]c(C(N)=O)c1 57363,C1(C(=O)NC(C2CCC2)C)CCCN(C(c2cccnc2S)=O)C1 57364,C1(NC(C2CC(C)(C(=O)OC)C2)=O)CCC(NC(c2ccc(=O)oc2)=O)CC1 57365,c1(C(=O)NCc2c(CCNC(C(CC)C(C)C)=O)ocn2)cc(S(C)(=O)=O)co1 57366,C12CCCN(C1)C2=O.C1(NN(C(=O)COC2CCN(C)CC2)C)CCC(CO)CC1 57367,c1(C(C)SCc2nnnn2-c2ccccc2)cccc(Br)c1 57368,C(=O)(CCCC(CC)NC(=O)CCOC(C)C)NC(CCC)C(C)(C)C 57369,CCC(F)(C(=O)OC)C(=O)N1CCC(O)(CNC(=O)C(F)=CC2CC2)CC1 57370,N1(C(Cc2c(C)n[nH]c2)=O)CCC2(CCN(C(=O)CNC(C3CC3C)=O)CC2)C1 57371,N1(C(C2CCC(CC)O2)=O)Cc2[nH]nc(C(N3Cc4c[nH]nc4C3)=O)c2C1 57372,C1(C(N(CCC)Cc2cn[nH]c2)=O)CCCN(CCOc2ccccc2C)C1 57373,C1(NC(C2CCC(CNC(C3C(C)=CCS3)=O)O2)=O)CC(=O)N(O)C1 57374,N1(C(c2nc(C)oc2)=O)CCCN(C(=O)CCn2ccc3cccnc23)CC1C 57375,C(c1c(Cl)nc2ccccn12)=CC(=O)NCC1(F)CC(NC(C2CCCO2)=O)C1 57376,C(CCC(=O)N1CC(OCC(=O)NCC2CC2[N+](=O)[O-])C1)SC 57377,c1(C(N2CCCC2C2(NC(C3CCCO3)=O)CC2)=O)ccc(OC2CC2)cc1Cl 57378,C1(CN(C)C(C2C3CCCCC23)=O)CCCCN1C(=O)CCC1CCOCC1 57379,N1(C(C(CSCC)NC(c2ccco2)=O)=O)CCCN(C)CC1CC 57380,Cc1c(F)ccc(NC(C2CCCC2CNC(=O)Cc2cccnc2F)=O)c1F 57381,CC1CN(C(c2cnc(O)c(F)c2)=O)CC2(CCN(C(C34CCC(C3)C4)=O)C2)O1 57382,C1(CC(=O)NC2C(CC)N(C(C3CNC(=O)C3)=O)CC2)CCC2(CC1)OCCO2 57383,CC(C)CCC(O)C(=O)N1CCC2(CC2NC(=O)C2=COCCC2)C1 57384,c1(CC)cc(C(N2CC(CNC(=O)C3CC3)(OC)C2)=O)n[nH]1.C1(C)C(=O)N1 57385,c1(CNC(C(C2C(C)(C)C2)N(c2cc(F)ccn2)C2CC2)=O)ccc(F)cc1 57386,N1(C(c2nccc(CC)c2)=O)CC(C(N2CC3CCCC23)=O)CC(C)(C)C1 57387,CC1CC2(CC(C(=O)NC34CCN(C(c5cnn[nH]5)=O)CC3C4)C2)C1 57388,C=C(F)C1(CC(N2CCCCC2CCN(C)C(c2nc(C)c(C)s2)=O)=O)CCC1 57389,CCCCCCCC(F)C(=O)NC1CCN(C(C2CN(C)C(=O)N2)=O)C(C)C1 57390,Cc1cnc(Cl)c(C(=O)N(C)CC2CCCN2C(=O)C(=O)C2CCCC2)c1 57391,c1(NC(C2C(NCc3ncc(C)c(Br)c3)CCC2)=O)ccc2oncc2c1 57392,C(=O)(CCCC(=O)NCC=C1CCN(C(C2(C(F)F)CCCO2)=O)CC1)NCC 57393,C1(CNC(COCC(=C)C)=O)CN(C(=O)CCOC2CCCC2)C2CC12 57394,C(=O)(CCN(OC)C(=O)c1cccnc1O)N1C(C(CCC)C)CCC1 57395,c1(C(=O)OCc2ccc(C)o2)cccc(Cn2ccnc2)c1 57396,C(C(C)C(F)C(=O)N(C)CCn1cnnc1)NC(c1cnc(C)n1C)=O 57397,CCCCC(CN(C)C(C1CCN(C(C2(CCOC)CCC2)=O)CC1)=O)CC 57398,Cc1cccc(C(N2CC(O)(C(C)(C)CNC(=O)C(O)C3CCC3)C2)=O)c1F 57399,N1(C(C2C(C(C)(C)C)C2)=O)CCC2(CC1)CC2NCC=C1CCSCC1 57400,N1(C(c2c(C)snc2)=O)CCC2C(CCCN2c2ncnc3c(C)csc23)C1 57401,C1(C(=O)NCC2CCSCC2)(CC)CCCN(C(c2cnccc2C)=O)C1 57402,CCCCC(C(=O)NC)NC(=O)C(C)(C)C(C)NC(=O)CC1CC1CC 57403,c1(CC(=O)NCC2N(C(CSCC#C)=O)CCN(C)C2)cccc2c1OCCO2 57404,c1(OC)cncnc1NCCCOCC1CC1.C1(=O)CC(C)N1 57405,C=CCC(CC)C(=O)NCCC1(NC(=O)Cc2csc(-c3ccoc3)n2)CC1 57406,C1(NC(c2cc(C)c(C)o2)=O)CC(C)CN(C(C2(CC3CC3)CC2)=O)C1 57407,C(CC(O)CNC(c1cn(C2CCC2)nn1)=O)NC(=O)Cc1cscn1 57408,Cc1scc(C(=O)NC2CC3C(NC(=O)CC4CCCCC4O)C3C2)c1C 57409,N#CC1CCC(CC(=O)NCC2(F)CC(CNC(c3cc(Cl)sc3Cl)=O)C2)C1 57410,n1(CC(=O)NCCCN(C(C23CCC(C2)C3)=O)CC)nc2n(c1=O)CCOC2 57411,C(c1cn(C)c(=O)n(C)c1=O)=CC(N1CC(NC(c2c(C)ccs2)=O)C(C)C1)=O 57412,c1(C(N2CC(NC(=O)CSc3ccc(Cl)cc3)(CO)C2)=O)cccc(F)c1O 57413,C(N=c1[nH]c(=NC(C)CF)[nH]c2c1CCC2)c1scc(COC)c1 57414,c1(C(=O)NC(c2nc(C3CC3)no2)C)cc2n(c1)CCS(=O)(=O)C2 57415,CC(C)(CNC(C1CCC2(CCC2)C1)=O)CC(=O)NC(C)(C)C(C)(C)CO 57416,N1(C(C(c2cccc(Cl)c2)C)=O)CC2CCN(C(=O)Cn3cnnc3)CC12 57417,CC(C(=O)N1CC(N(C)C(c2coc(C3CCCC3)n2)=O)C(C)(C)C1)S(C)(=O)=O 57418,Cc1nc2sccn2c1C(=O)NCC(F)CNC(=O)COCC(C)(C)C 57419,c1(C(=O)NCC(CC)NC(=O)CC2NC(=O)CNC2=O)cc2c(C)ccc(F)c2o1 57420,C(=O)(C(C)S(N)(=O)=O)NCCn1ncc(C(=O)NC(COC(C)C)(C)C)c1 57421,O=C(CN=c1cc[nH]cc1)NC1(C(=O)NCCC2(O)CCOC2)CC(CO)C1 57422,C1(NC(=O)C(CO)c2ccccc2)CCCCCN(C(c2nccc(Cl)c2F)=O)C1 57423,C1(C(N(C)CC2(CNC(c3ccnnc3)=O)CC2)=O)CCC=CCCC1 57424,CC(C)(C)C(O)CC(=O)N1CC(NC(=O)COC2CCCC2)C(O)C1 57425,c1(C(=O)NC(C2CCN(C(c3n[nH]cc3Br)=O)C2)C)cccc(CO)c1 57426,C(=O)(C1CNC(=O)c2ccccc21)N1CCCCC(CNC(C2(C#C)CC2)=O)C1 57427,c1(C(N2CC3C(CNC(=O)Cc4cnccc4Cl)(C3)C2)=O)cc2n(n1)CCC2 57428,c1(CC)occc1C(=O)NCC.c1(C(C(N2CC(OC(F)F)C2)=O)ON)ccccc1 57429,N1(C(CCC(C)C)=O)CC2(CC(NC(=O)CC3CCOCC3(C)C)CO2)C1 57430,N1(C(C(F)=CC)=O)CCC2(CC1)CC(C)N(C(C1CC13CC3)=O)C2 57431,N1(C2C(C)SCC2)CCN(c2ccccn2)CC1.C12CCN(C1)C(=O)C2 57432,C1(C)(CNC(c2cc(COC)[nH]n2)=O)CCN(C(c2snnc2C)=O)C1 57433,Cc1cc(C(=O)NC(c2cnn(C)c2)C(=O)NCC2C=CCCC2)ns1 57434,C1(OC)CCC12CC(C(=O)NCCCC(C)(C)NC(=O)CCc1ccnn1C)C2 57435,N1(C(CCS(N)(=O)=O)=O)CCCCC12CC(NC(=O)C(=Cc1cccnc1)F)C2 57436,c1(CC(=O)N(CC(=O)N(C(CC2CC2)CO)C)C2CCC2)cncnc1O 57437,N1(C(CCCNC(=O)OCC)=O)CC(NC(=O)CSC2CCCCO2)C(C)C1 57438,c1(C(=O)NCCCOCCCNC(c2cc(OCC)n[nH]2)=O)cn(C)nc1C 57439,Cc1cc(NC(C2CSCCN2Cc2ccc(Br)cc2O)=O)c(C)cc1Br 57440,N1(C(C2COCCN(C(Cc3ccn(CC)n3)=O)C2)=O)CCCN(C)C(=O)C1 57441,C1(NC(COCc2ncc(C)o2)=O)CN(C(C2CCOCC2)=O)CCC1F 57442,C=CC1(C(=O)NCCOCCCNC(=O)CCS(C)=O)CCOCC1 57443,Cc1c(C(=O)NC(C2CCCN(C(C3(C(N)=O)CC3)=O)C2)C)cnc2ccnn12 57444,CC#CCC(C(=O)N(CCC(=O)OCC)C)NC(=O)CCc1cn[nH]c1 57445,c1(C(N2CCC(C)C(N(C)C(c3cnco3)=O)C2)=O)ccc2cccnc2c1 57446,N1(C(C(=O)NCC)=O)CCCC2(NC(=O)CSc3c(C)n[nH]c3C)CC2C1 57447,C1(C(=O)NCCCCCNC(C(C)OCCOC)=O)(OC(C)(C)C)CCCC1 57448,c1(-n2cc(-c3ccc(SC)cc3)nn2)c(F)cc(C(=O)OC)cc1F 57449,c1(C(N(C2C(C)CC2)C)=O)coc2c1CN(C(=O)CCc1nccn1C)C2 57450,N1(C(C2CCC(C(N)=O)O2)=O)CCCC2(CCN(C(c3cccnc3F)=O)C2)C1 57451,C(=O)(CCCC(C)(C)C)NC1CC2(CC(NC(C(C)c3ccsc3)=O)C2)C1 57452,C1(C)(C(=O)NC(C(C)O)CO)CCCN(C(=O)CCC2CC2C)C1 57453,c1(C(=O)NCCCCCOC)ccnc(CNC(=O)C(C)C2CCCO2)c1 57454,C1(C(N2CCC(CN(C)C)CC2)=O)C2CCC(C2)N1C(C1CC2COCC2C1)=O 57455,c1(N(C)C)cncc(C(N2CC3CC2(CN(C(=O)C=CC(N)=O)C2CC2)C3)=S)c1 57456,c1(CC)sc(=N)[nH]c1C(=O)NCC1CC1CNC(c1cn(C)c(C)n1)=O 57457,CC12CN(C(=O)Cn3cnc([N+](=O)[O-])c3)CC1CN(C(C1CCS(=O)(=O)C1)=O)C2 57458,c1(C(=O)NCC2CN(C(C3(CO)CCOCC3)=O)C2)cccc2c1CCCCC2 57459,C1(CNC(COCCCC(C)C)=O)CCN(C(c2cncn2C)=O)C12CCC2 57460,CC(C(=O)NCCC1CN(C(=O)CCN2CCN(C)CC2)CCCO1)C(C)(F)F 57461,C=C1CC2(C1)CC(C(=O)NC1CCN(C(C3CCC=CCC3)=O)CC1C)C2 57462,C1(CC)CNC(=O)CN1C(=O)C(C)(C1CC1)N(C)C(c1cc[nH]c(=NC)c1)=O 57463,c1(N2C(C)(C(=O)NC(c3ncccn3)CC)CC2)ncnc2c1ncn2C 57464,CCC(C)CC(=O)N(C1CC(NC(=O)CCOc2ccccc2F)C1)C 57465,c1(C(=O)NC(CCN(C(C(CCC)CC)=O)C)C)ccc([N+](=O)[O-])cc1CC 57466,N1(C(c2ncc[nH]2)=O)CCCC(C2CCN(C(C3(C(F)F)CCC3)=O)C2)C1 57467,CCCCCCC(=O)N(C)CC1CCN(C(C2(C(=O)OC)CC2)=O)CC1 57468,C1(NC(c2cc(C)on2)=O)CN(C(=O)CC2(O)CCCCC2)CC12CCCC2 57469,C(C1CCC(C)CC1)=C(C(N1CCC(N(C(C2CCN(C)C2=O)=O)CC)C1)=O)C 57470,C1(C(N2CC(N3C(=O)CC(OC)C3)C2)=O)COc2cc(OC)ccc2C1 57471,C(=O)(CS(=O)(=O)C(C)C)N1CCN(C(c2snc(C)c2N)=O)C(c2ncc[nH]2)C1 57472,C(=O)(C(C)(CC)C(N)=O)NC1(COC)CN(C(c2ccc(Cl)cc2OC)=O)C1 57473,c1(C(=O)NCCCCCN(C(c2n(CC)ncn2)=O)C(C)C)occ2c1CCC2 57474,N1(C(C2N(C)C(=O)OC2)=O)C2CCC1CN(C(=O)CC1CCOC(C)(C)C1)C2 57475,C1(C(=O)OC)N(C(=O)CCC(C)NC(=O)Cc2cnn(C)c2)CC1(C)C 57476,N1(C(CC(C(C)C)NC(=O)Cn2cncn2)=O)CCN(C)CC(C)C1 57477,CN(C)NC(=O)CCC(=O)N1CCC1CNC(c1ccccc1C1CC1)=O 57478,C(=O)(C(C(=O)N1CCCC1Cn1cc(-c2nccc(C)n2)nn1)OC)OC 57479,C1(C(N(CC(C)O)CCNC(c2cnn[nH]2)=O)=O)CCOC(C)C1 57480,C1(NC(c2cc(Cl)cs2)=O)CCN(C(=O)C=CCn2cncn2)C12CC2 57481,c1(C(=O)NC2CC(NC(CCc3c(C)nccc3)=O)C2)cccc(F)c1Br 57482,N1(C(COc2cn(C)nc2)=O)CC(NC(=O)CCN2CCCC2=O)CC1CO 57483,N1(C(CCc2cnc(C)o2)=O)CCCC(CNC(C2CC2(F)F)=O)CC1 57484,c1(C(C(=O)NCCC2CC(NC(c3ccns3)=O)C2)O)ccc(Cl)cc1 57485,C(=O)(C1Cc2c(Cl)cccc21)NCC1CC2N(C(CC3CN(C)C3)=O)C(CC2)C1 57486,C1(c2nnnn2C2CC2)(NCCCC(=O)OCC=C)CCCC(C=C)C1 57487,CC1CCC(NC(C2CNC(=O)C2)=O)C1 57488,N1(C(C2(C(C)C)CCN(C(CCC(CC)=O)=O)C2)=O)CCCC(C2CCC2)C1 57489,c1(OC)ccc(C(=O)NC2CCC(NC(=O)CSc3nccn3C)C2)o1 57490,C1(n2cc(CCNC(=O)CCOC3CCOC3)nn2)(CN)CCOCC1 57491,C(CCCC(=O)NCC1CC(CC)C1)NC(CSCC#C)=O 57492,Cn1[nH]c(C(=O)NCCC2CCN(C(=O)COC3COC3)CC2)nc1=O 57493,Nc1ncccc1C(N1CCC(N(C(=O)CC2CS(=O)(=O)C2)CC2CC2)CC1)=O 57494,c1(C(=O)NC2C(NC(CC3CC(=O)NCC3)=O)C2)cc(F)cc(Cl)c1 57495,C(=O)(CC(C)(C)c1ccccc1)NCC(Cn1cc(C(C)OCC)nn1)(F)F 57496,C1(F)(C(=O)NCC(CC)(CC)OC)CCCN(C(c2ccc(C)o2)=O)C1 57497,C1(NC(C(C(CC)C)O)=O)CC2CCC(C1C)N2C(=O)CNC(=O)OCC 57498,c1(-c2cccc(CC)c2)cccc2nc(CSCC)cn12.C1(C(N)=O)CNC(=O)N1 57499,Cc1cnn(C)c1CC(=O)Nc1ccc(OC)cc1.c1(CCCC)cn(CC)nn1 57500,C1(C(=O)NCC2OCC(C(=O)NCc3c(C(C)C)n[nH]c3)C2)CC(=O)NC(=O)C1 57501,C(c1cc(Br)ccc1OCC)=CC1=CCN(Cc2ccc(CCCC)cc2)CC1 57502,n1(CCC(=O)NC2C(NC(C3ON=C(CC)C3)=O)CCC2)cc(S(N)(=O)=O)cn1 57503,C1(S(N)(=O)=O)(N(CCCn2cc(COCC(=O)CNC(N)=O)nn2)C)CC1 57504,n1(CC(=O)N(CC(C)NC(c2sccc2-n2cccc2)=O)C)cc(CO)nn1 57505,c1(C(=O)NC(C)Cc2cccs2)ccc2nn[nH]c2c1O 57506,C1(c2n(CCCC)nnn2)(NCC2(N(C)C)CCS(=O)CC2)CCCN(C)CC1 57507,c1(CNC(CN2CC(CC)C2)=O)cn(C2CCN(C(=O)CCF)C2)nn1 57508,N1(C(C2C(C)(C)C2(C)C)C(=O)NCCCOC)CCc2ccc(Cl)cc2C1C 57509,C(=O)(CC1=NNC(=O)C1)N(C(C)CNC(c1ccc(CO)c(F)c1)=O)CC 57510,C1(C(=O)NCC(C2CCC2)NC(=O)CCOc2ccccc2)SC2C=CC1CC2 57511,C(=O)(C(Cc1cnc[nH]1)N(C)C)N1CC(NC(=O)NCC)C1.C12CN(C1)C2=O 57512,O(NC(=O)C(CNC(=O)CCCCCSC)C(C)(C)C)CC(CC)C 57513,N1(C(=O)NC2C(=O)NCC2)CCN(C(=O)CC2COCCOC2)CC1 57514,c1(C(N(CC(C)CNC(C2CC2C)=O)C)=O)cncc(-c2ccc(F)cc2)c1 57515,C=CCC(CNC(c1ccc(CC(C)C)s1)=O)NC(c1csc(C(C)(C)C)n1)=O 57516,c1(C(=O)NCC2(F)CCC(NC(CS(CC)(=O)=O)=O)C2)cn2cc(C)ccc2n1 57517,N1(C(C2N(C(C)=O)CCC2)=O)CCN(C)C(C(N2CC=CCC2)=O)C1 57518,c1(C(N(CC(CNC(CC(=C)C)=O)O)C)=O)cn2cc(Br)cc(C)c2n1 57519,C(N=c1nc[nH]cc1C#N)C1CC(NC(c2ccc(C)nc2)=O)C1 57520,C1(C(=O)NCC(C)C)CCCN(C(C)Cc2ccc(C(C)(C)C)cc2)C1 57521,CS(=O)(=NCC(=O)NCCn1cc(CNC=O)nn1)c1ccc(Cl)cc1 57522,N1(C(CCN(C(C2CCC(=O)CC2)=O)C2CC2)=O)CC2(CCC2)CC1CO 57523,c1(OCCNC(c2cnsn2)C)ccccc1F 57524,c1(C(=O)NC(CC)CNC(c2ccc(-c3ncc[nH]3)cc2)=O)cc(=N)[nH]c(Cl)n1 57525,CC1CC2(CO1)CN(C(=O)CC(C1CC1)NC(C1CC1C(N)=O)=O)C2 57526,C=CCC(CNC(C1CC1(C)C(F)(F)F)=O)NC(=O)C=CC(C)(C)C 57527,N1(Cc2cn(-c3ccc(C)cc3)nc2)CCCN(C(C2CCCO2)=O)CC1 57528,N1(C(C2(C)CCN(C(C)=O)C2)=O)CC2CCC(C1)N2C(C)C(=O)NC1CCOCC1 57529,c1(C(=O)NC(CNC(C(CCCC)O)=O)C2CC2)n[nH]c(C(C)C)c1[N+](=O)[O-] 57530,c1(C(=O)NC(CC)C)ccc(CC2(c3ccccc3)CC2)cc1 57531,c1(C(N(CCC(=O)NCC2C(OC)CCC2)C(C)C)=O)csc(C)c1C 57532,c1(CC)cc(C(N2CC(CNC(c3ccc(CSC)o3)=O)C(C)C2)=O)cc(N)c1 57533,C(=O)(CC1=CCOCC1)N1C(C(=O)NCc2c(CC)nn(C)c2)CC(F)CC1 57534,CC1(C)CCCN(C(=O)Cc2nnc(O)s2)C1CNC(c1cnc(Cl)s1)=O 57535,c1(OC)ccc(C(C)C(=O)N(C(C)CCNC(=O)C(C)(F)F)C)c(C)c1 57536,C1(CC(N2CCC(N(CCCOC)CCO)CC2)=O)CCn2cncc2C1 57537,N1(C(C2C(NC(C(C)C(F)(F)F)=O)CCC2)=O)Cc2n[nH]cc2C1CO 57538,CN1CCC(CC(C(=O)O)NC(C2CCCC2CN)=O)CC1 57539,C1(NC(c2nc(COCC)sc2)=O)CC2CCC1N2C(c1cn(C)ccc1=O)=O 57540,C#CCCCCC(=O)N1CC(NC(=O)C(CCC)OCC)C(C)(C)C1 57541,N1(C(C2(F)CCN(C(C(C)N(CC)CC)=O)C2)=O)CC2CCC2(OC)C1 57542,C(=O)(CS(=O)(=O)C1CC1)N(CCCCCNC(c1ncn2c1CCC2)=O)C 57543,c1(CC(=O)NCCC(C)CCO)cc(F)c(Cl)cc1[N+](=O)[O-] 57544,CC1=C(C(=O)NC2CCCC2NC(=O)CC2CC=CCN2C)CCC1 57545,Nc1ccc(C(=O)NCC(C2CC2)NC(C2(O)CC2)=O)cc1OCCO 57546,C1(NC(C(C)=C2CCC2)=O)CN(C(=O)CC2CCN(C)C2=O)C2(CCCCC2)C1 57547,S(=O)(=O)(c1ccc2c(c1)N(C(=O)Nc1ccc(S(C)=O)cc1)CCC2)N(C)C 57548,c1(C(N2CC3(C(NC(CS(CC)=O)=O)CC3)C2)=O)cccc(S(=O)(=O)CCO)c1 57549,N1(c2snc(C(=O)OC)n2)C2CCC1C(CNC(=O)C(c1cscn1)N(C)C)C2 57550,c1(CC(=O)NCC(F)CNC(c2cc(F)n[nH]2)=O)nccc2ccccc12 57551,CC(C)C(C(=O)NCC1(CNC(c2ccccc2)=O)CC12CCC2)N(C)C 57552,C(=O)(C1OCCc2cc(OC)ccc21)NC1C2CC3(C(=O)OC)C(C2)C31 57553,C1(C#CC(=O)NCc2ccc(C(=O)NC(C)CCOC)nc2)(CC)COC1 57554,c1(NCCNC(CC)=O)ccc(S(=O)(=O)NCCCC(F)(F)F)c(Cl)c1 57555,c1(C(=O)NC2(C)CCN(C(CC(CC)(C)C)=O)C2)cc2cccnc2nc1O 57556,C1(C(=O)NCCN(C(CCc2cc(OC)no2)=O)C(C)C)CCCCC12CCC2 57557,Cc1cc(CC(=O)NC2CC(CCNC(=O)C=CCO)C2)cc(C)c1 57558,c1(C(CNC(C(C)CC2CC2)=O)NC(=O)CN(C)C)cccc(Cl)c1Cl 57559,CC1OC(C)C(C(N2CCN(C(=O)CC3(C)CC3(Cl)Cl)C(CCO)C2)=O)C1C 57560,COn1cnc(C)c1C(=O)NC1COCCN(C(=O)CCCC(C)C)C1 57561,c1(C(=O)NCC2CN(C(c3c(C)nco3)=O)CC2C)cc2cccnc2s1 57562,N1(CCC)CCCCC1C(N1CCC(CF)(NC(c2nc(O)sc2C)=O)C1)=O 57563,C(=O)(CC(C)CC(=O)OC)NCC(CC)(C)NC(=O)CN(C)C(C)C 57564,N1(C(c2cc(CCCCC)[nH]n2)=O)CCCC(NC(C2(C)CCOCC2)=O)C1 57565,N1(C(C=CC(C)NC(C(C)=C(CC)C)=O)=O)CCC(CCN(CC)CC)C1 57566,CC(F)(F)C(C)(C)CC(=O)C1=CNN=CC(C(=O)N(CC2CC2)CO)CC1 57567,C1(COc2cccc(C#N)c2)CC2COCC2N1C(=O)OC 57568,NS(=O)(=O)c1ccc(C(N2CCC(F)C(NC(=O)CCC3CCCO3)C2)=O)nc1 57569,C(=O)(C(F)(F)C(F)(F)F)NC1CCCC1.N12CCCC1C1(CC1)CCC(C)C2=O 57570,C(CS(=O)(=O)CC(=O)NC1COCCC1C(=O)NCc1cc(Cl)ccn1)OC 57571,c1(C(=O)NC2CCN(Cc3nccc(C)c3)CC2O)cc2cnccc2nc1C 57572,C1(CNC(c2ccc(COC)[nH]2)=O)CCN(C(=O)CSCC2CCCO2)C12CC2 57573,C1(C(=O)NCC(C(N2CCC(NC(CC)=O)C2)=O)N(C)C)CCC2(CCC2)O1 57574,c1(CC(=O)NC2C3CN(C(C(C)(C)CO)=O)CC2C3)csc2c(F)cccc12 57575,N1(C(C2(CC)CN(C(=O)CC3CC=CCC3)C2)=O)CCC(C)(O)CC1 57576,O=C1CCC(CCC(N2CCCC2C2(NC(c3ccncn3)=O)CC2)=O)CN1 57577,N1(C(c2c(C)nsc2)=O)CC2CC2(NC(=O)C(C)OCC2CCCO2)C1 57578,c1(C(=O)NCC2CC(NC(C3C(=C)C3)=O)C(O)C2)ccn2c(C)cc(C)nc12 57579,C1(CCNC(c2c(C)con2)=O)CN(C(C2CC2(Cl)Cl)=O)CCO1 57580,N1(C(C(C=C)(C)C)=O)CCC(NC(c2oc(C)cc2C)=O)C(F)(F)CC1 57581,N1(C(C(C)C#N)=O)CCC2CCN(C(=O)CN3CC4CC4C3)CC2C1 57582,N1(C(C(C2CCC2)OC)=O)CCOCC(NC(C2CSCCS2)=O)C1 57583,CC1(C)CCCN(CCN(C(c2ccccc2N)C2CC2)C2CC2)C1 57584,N1(C(CCN(C(Cc2cccc(C#C)c2)=O)C2CC2)=O)CCOCC2(CC2)C1 57585,C1(C(=O)NC2C(NC(c3n[nH]c(C(C)C)c3Br)=O)C2)CCCCCN1C 57586,Cc1cc2[nH]nc(CNC(=O)N(C)Cc3ccc(C#N)cc3)c2o1 57587,C(C(C)(O)CC(=O)NCc1c[nH]nc1C(=O)NC1CCCCC1)OC 57588,Cc1cc(=O)c(C(N2CCC(C(=O)NCC34CC(F)(C3)C4)(CO)C2)=O)c[nH]1 57589,c1(-c2c(OCC)c(F)ccc2)cccc2sc(C(N3CC(=O)NC(=O)C3)=O)cc12 57590,C(=O)(C(CNC(=O)C(C)CC#N)C(C)(C)C)Nc1ccc(OC)cc1C 57591,C1(C(=O)NC2C3CC2N(C(=O)CN(C)C2CC2)C3)(OC)CCOCC1 57592,n1(CCNC(CN2CCN(CC(COC)O)CC2)=O)c(C)cc2ccccc12 57593,CC1CCN(CC(=O)NCC2CCN(C(=O)CNC(c3ccncc3)=O)C2)C1 57594,Cc1c(Br)noc1C(=O)NCC#CCNC(=O)C(C)OC1CCCCCC1 57595,Cn1nc(C(N2CC(NC(c3cscc3F)=O)CC(O)C2)=O)c(Cl)c1Cl 57596,C12(C(N3CCOCC3)=O)CC(c3ccccc3)(CO1)C2.O=C1NCCN1 57597,CCC(C)CCCC(=O)NCC(CC)(CC)NC(C12CC1CN(C(C)=O)C2)=O 57598,Cc1csc(C(=O)NCCCN(C2CC2)Cc2nc(CN(C)C)n[nH]2)c1Cl 57599,CCC(CNC(=O)C(CC1CCOCC1)NC(=O)CN1CCNC(=O)C1)C(C)C 57600,c1(NC(=O)NC2CCCC(NS(C)(=O)=O)C2)ccc(Br)c(F)c1F 57601,C(CC(=O)N(CC(=O)NC(CO)C1(O)CC1)C)SCC 57602,N1(C(CN(C(=O)OCC)C)=O)CCC2CC12C(=O)NCCCn1cccn1 57603,C1(NC(C)=O)CN(C(=O)Cc2csc(Cl)n2)CC1c1ccccc1 57604,c1(COC)nn(C)c(Cl)c1C(=O)NC(CCNC(C1CCC1(F)F)=O)CC(C)C 57605,N1(C(c2cccc(OCC)n2)C(=O)NCC(=C)C)CC2CCN(C)CC2C1 57606,C1(C(=O)NCCN(C(C=C(C)CN2CCOCC2)=O)C)CCCN1CC(C)C 57607,C1(NC(C)=O)C2CN(C(C3(NC(c4ccnn4C(F)F)=O)CCSC3)=O)CC12 57608,C(C)(CO)(C(=O)NCCN1CCCC1)NC(c1ccc(C(C)=O)o1)=O 57609,CC1=CCC=CC1C(N1CC(C)(CC(=O)NCC2(N(C)C)COC2)C1)=O 57610,C12CCCCN(C1)C(=O)N(C)C2=O.c1(C(C)=O)ccc(Br)cc1.C1(C=O)OCC1(C)C 57611,C1(CC(=O)NCC(COCC)C)CN(C(c2ccc(C#N)o2)=O)CCC1C 57612,N1(C(C(C)OCCCC)=O)CC2CCCN(C(c3cc4ccccn4n3)=O)C2C1 57613,C(=O)(C(C(C)C)C(C)C)N(C1CCN(C(=O)C(c2cncn2C)O)C1)CCC 57614,c1(CCC(=O)NCC(c2ccccc2)C)ccc(OC(F)(F)F)cc1 57615,c1(C(=O)NC2CC(NC(C(CC)OCC)=O)C2)ccnc(F)c1N 57616,C1(NC(c2cc(CCNC(c3ccn(C)c3)=O)on2)=O)C2CCCOC12 57617,C1(C(=O)NCCNC(CC2C(C)CCC2)=O)CCC(C)(F)CC1 57618,C(=O)(C(F)(F)CCn1cccn1)NCC(C)CNC(c1cc(Cl)cn1C)=O 57619,Cc1cc(C(N2CCCC(C(N3CCCC(O)C3C)=O)C2)=O)ccc1Br 57620,Cc1nc(C)c(C(C)NC(=O)C(C2CC2)N(C(=O)CCC(C)N(C)C)C)[nH]1 57621,c1(C(N2CC3C(N(C(c4cc(COC)on4)=O)C)C3C2)=O)cc(O)cc(C#N)c1 57622,CC1(C)CN(C(=O)NCC2CCC3(C2)OCCO3)CC2(CCOCC2)O1 57623,c1(C(N2CCC(C)(NC(C3C(C)CCCC3)=O)C2)=O)cnc2n1CCS2 57624,c1(C(=O)NCC2CC(C)(C)C2)ccc(CNC(=O)CNC(N)=O)nc1 57625,c1(CC(=O)NC2(c3cn(CCCC)nn3)CCC2)ccc(F)cc1C 57626,C#CCC(C)(CC)C(=O)N1CC(NC(=O)C(c2cnn(C)c2)C)C1 57627,C(=O)(C(C(CC)=Cc1cccnc1)N1CCCCC1C1CC1)NCCCC 57628,C(C1=C(C)OCCS1(=O)=O)NC(NCCN1C(CC)CCC1)=NC.C1(C)CC=CCC1 57629,N1(C(C(C(=C)Cl)(C)C)=O)CCCC(NC(=O)C2=C(C)OCC2)C(F)C1 57630,N1(C(CN(CCOC)C)=O)CCCC(O)(CNC(=O)CC(C)c2cccnc2)C1 57631,C(=O)(CCCCCN(C)C)NC(C(C)C)C(C)NC(C1CCCCS1(=O)=O)=O 57632,N1(C(C2C(C)(C)CCCO2)=O)CC2(CC(C(=O)N(CCO)CCO)CO2)C1 57633,c1(N2CCC(C(=O)OC)(COC)C2)ncc(S(C)(=O)=O)cc1Cl 57634,c1(C(=O)NCCC2CCN(C(C(CC)SC)=O)C2)cc(O)cc(F)c1 57635,CC1=C(C(=O)NC2CC(Nc3ncc4ccnc-4[nH]3)C23CCC3)CCS1(=O)=O 57636,C1(NC(c2c(C)cccc2)=O)CCN(C(c2ncc(Br)cc2C)=O)CC1CO 57637,c1(CC(N2CCCC2C2(O)CNC2)=O)ccc(Cl)cc1SC1CC1 57638,c1(C(=O)NC2(C)CCN(C(C(COC)(F)F)=O)C2)ccc2nnn(C)c2c1 57639,C(=O)(C(C)CC(=O)NCC(C(C)(C)C)NC(C1CSCN1C(C)=O)=O)OC 57640,C1(C(=O)NCCC(CCC)O)CN(C)CCN1C(C1CC(N(C)C)C1)=O 57641,O=C1CCCC(C(=O)NCCCCC(=O)NC(CO)CCF)CC1 57642,N1(C(c2cc(OC)n[nH]2)=O)CC(C)CN(C(C2CC3(COC(=O)N3)C2)=O)C(C)C1 57643,CC1(CNC(C2C3COCC23)=O)COCCN(C(=O)C2=NOC(C(C)(C)C)C2)C1 57644,Cc1cnsc1CNC(Cc1cn(CC(c2ccccn2)C)nn1)C(=O)O 57645,C1(N(C(=O)COCC(C)(C)C)C)CCN(C(C2COC(=O)O2)=O)C1 57646,N1(C(COCCC)=O)CCN(C(=O)C(c2cccc([N+](=O)[O-])c2)C)CC(O)C1 57647,C1(C(=O)NC(CN(CC)CC)C)CCC2CCC1N2C(c1cncn(C)c1=O)=O 57648,C1(N(c2c(Br)cnc(C)n2)Cc2cc(C(C)C)ccc2O)CC2CCCC(C1)N2 57649,C1(NCC(c2ccc(CC(C)C)cc2)N(C)C)CC2(C1)CC(C#N)C2 57650,c12ccccc1CC(=O)N2.c1(NC(C2C(C(N)=O)C2)=O)ccsc1 57651,C1(C(NOC(C(=O)OCC)(C)C)=O)CCCCN(C(c2ccc(C)c(F)c2)=O)C1 57652,N1(C(CNS(N(C)C)(=O)=O)=O)CCC(C)(C)C(NC(=O)CC2CCC(F)(F)C2)C1 57653,N1(C(C(C)NC=O)=O)CCC(C(=O)NCCC2CC(=O)C2)CC1 57654,c1(C(=O)NCC(=C)CCNC(=O)C=Cc2cnccn2)nncc2c1CCCC2 57655,C1(CCC(=O)NCC(O)CNC(C2(N(C)C)CC2)=O)(C(=O)OC)CCCC1 57656,C1(NC(=O)Oc2c(C)cccc2)CCCN(C(C)C(N)=O)CC1 57657,C1(C(N2CC(CN(C(=O)CCN3CCCS3(=O)=O)C)C2)=O)CNc2ccnn2C1 57658,Cc1cc(C(C)(C)C(N2CC3CC3C2CNC(=O)CC2CC2)=O)ccc1Br 57659,C(=O)(C1c2c[nH]nc2CN1C(=O)CCc1ccco1)NC(CCN(C)C)(C)C 57660,C(C)(CNC(=O)COCCC(C)C)(CNC(=O)CCc1nncs1)OC 57661,N1(C(c2c(CC)cno2)=O)CCC(C(CO)NC(=O)C(C)(C)COC)CC1 57662,c1(C(C(=O)NCCC2CC2)N(C2CCCS(=O)(=O)C2)C)ccn2ncnc2c1 57663,n1(CC(=O)NCC(CCCC)NC(CSCC=C)=O)ncc(=O)c2ccccc12 57664,N1(C(C(CNC(C2(OC)CC(C)C2)=O)N(C)C)=O)CCc2ccc(C#N)cc21 57665,C1(CC)CCN(C(C2CN3CCC2C3)=O)C1CNC(=O)C(C1CC1)OC 57666,C1(NC(=O)Cc2cscn2)CCC2(CCN(C(=O)C3=CC4(CCOC4)C3)C2)C1 57667,CCC(C)(C)CC(=O)N1CCC(CNC(c2cc(C)c(C(N)=O)cn2)=O)C(C)C1 57668,C1(NC(C(Cc2cn(C)nc2)O)=O)COCCN(C(=O)CN2CSCC2=O)C1 57669,c1(C(=O)NCC(CC)(C)C(=O)NCCn2ccccc2=O)cccc2ccnn12 57670,C(=O)(C(C)(C)c1ncco1)N1CC(CNC(C(C2CCC2)OC)=O)C1 57671,Cc1cc(C(C)C(=O)NC2CN(C(C3(C)COC3)=O)CC2C(F)(F)F)cc(F)c1 57672,C(CCN(C)C(C1CCC(C)(CC)O1)=O)(C(C)C)NC(c1nc(CCC)sc1)=O 57673,C1(COC)(NC(=O)C(n2nccc2C)C)CCCN(C(=O)CSS(C)(=O)=O)C1 57674,C1(CCN)(O)CN(C(=O)CN(C2CCCCC2)C(C)=O)C1.c1(C(=O)NCC)ccco1 57675,c1(C(N2CCC(n3cc(C(CC)O)nn3)C2)=O)cc(Br)c(Br)cn1 57676,N1(C(C2C(C)(C)CC2)=O)CC(CO)C2(C1)CN(C(=O)C(C)(O)c1ccccc1)C2 57677,N1(C(c2sc(C)c(O)n2)=O)C2CCC1CC(O)(CNC(c1ccco1)=O)C2 57678,N1(C(C2CCCN(C(CCCC)=O)CC2)=O)C2CCC1CC(OC)C2 57679,C12(C(=O)NC3(CCO)CN(C(c4ccc(OC)cc4)=O)C3)CCCCC1C2(F)F 57680,CCCCC(C)CCC(=O)NCCCC1(NC(c2ccn(C)c(=O)c2)=O)CC1 57681,c1(CC)sc(C(=O)NC(C)(C)CN(C)C(c2ccccn2)=O)cc1C 57682,C=CC(C)(C)CCNC(C1(OC)CCN(C(=O)COCC(C)(C)C)C1)=O 57683,c1(OCC(=O)N(C(CCNC(C=CCC)=O)C)C)cc(F)cc(F)c1 57684,c1(C(C)C)ccc(NC(=O)C(C)N(C(=O)C=Cc2ccsc2)C)cc1 57685,N1(C(c2cnc(NC(C)=O)o2)=O)CC2(CC(NC(C3CCCN3C=O)=O)CO2)C1 57686,C12(NC(c3ccoc3)=O)CN(C(c3cnsn3)=O)CC1CS(=O)(=O)C2 57687,N1(C(C2(CC)CCNC2=O)=O)CCN(C(=O)CC2(COC)CC2)C(CO)C1 57688,c1(C(=O)OC)sc(C(=O)N(C2CCN(C(C3(CCF)CC3)=O)C2)C)cc1N 57689,C1(CC(=O)NC2(N(C(CC3CC(OC)C3)=O)CC3CC3)CCC2)CCN(C)CC1 57690,C1(NC(C(c2cc(F)c(Cl)cc2Cl)C)=O)Cc2ccc(C#N)cc2C1 57691,N1(C(c2[nH]cc(-c3nc(C)sc3)c2)=O)CCCC(C(C)NC(=O)CSC2CC2)C1 57692,CC(C(=O)N1CCCCC1CCN(C)C(C1(F)CCC1)=O)C(F)F 57693,C=CCC(C)(CC)C(=O)N1CCC(CNC(=O)C(N2CCN(C)CC2)C)C(O)C1 57694,c1(C(=O)NCC(C(=O)N(C(CC)C)CCO)OCC)cnncc1OC 57695,N1(C(COCCCCC)=O)CC(CNC(c2c[nH]nc2OC)=O)CC1COC 57696,N1(C(C(C(C)O)N(C)C)=O)CCC2(CC1)CC(NC(=O)Cc1cn[nH]c1)CCO2 57697,c1(C(=O)NC2C(NC(CC3N(CC)CCOC3)=O)CCCC2)c(C)nn(C)c1C 57698,c1(OC(CC)C)cccc(CN2CCNCC2C(=O)NCC)c1 57699,C(=O)(C(F)(F)C(F)F)NCC(N1CCN(C(C(C)=CC2CC2)=O)CC1)C(F)(F)F 57700,c1(C(N2CCC(O)(CNC(C(CC)CC)=O)C2)=O)cc(C)c(C#N)cn1 57701,c1(COC)cncc(C(=O)N(C2CCCC(N(C(=O)CSCCOC)C)C2)C)c1 57702,C(C1c2ccsc2CCN1C(C1CCc2nc[nH]c2C1)=O)NC(CCP(C)(C)=O)=O 57703,Cc1cnc(F)c(-c2cn(C(C)C(=O)N(C)C(c3ccco3)C)nn2)c1 57704,C(=O)(CCCC(C)(F)F)N(C1C(C)CN(C(c2cc(O)cs2)=O)CC1)C 57705,C1(C)(C(=O)NCCC(CNC(c2ccc(CN(C)C)o2)=O)O)CC2CC2C1 57706,C1(NC(CCSC)=O)CN(C(C2(CC3CC3)CC2)=O)CCC1C(F)(F)F 57707,N1(C(c2ccc(CN(C)C)[nH]2)=O)CCCCC12CC(NC(C1CN(C)C1)=O)C2 57708,c1(C(N(C(C)CN(C)C(C2CCC(N(C)C)CC2)=O)C)=O)ccc(F)cc1F 57709,C#CCC(O)C(=O)N(C)CC1CCCN(C(=O)C(C)NC(=O)OC(C)(C)C)C1 57710,Cc1cc(C(=O)NC2CC(C(C)NC(C3CCC4CC34)=O)C2)ncc1Cl 57711,c1(N2CCC(N(C(=O)C(C)CN(C)C)C)C2)nc(C)nc2sc3c(c12)CCC3 57712,C1(CNC(C(N2CCN(C(c3ccco3)=O)CC2)C)=O)C=CS(=O)(=O)C1 57713,C1(C(N(CC(CC)NC(C2(CC#C)CCC2)=O)C)=O)CC(=O)N(C(C)CCC)C1 57714,n1(C(C)C(=O)NC(C)CC(C)NC(C2CC(=O)C2)=O)cnc2ccccc12 57715,C(N=c1[nH]c2c(c(=NCc3cccc(N)c3)[nH]1)CCCC2)C1CC(C)C1 57716,C1(NC(C(C)CC2CC2)=O)C2CC3CN(C(c4ccc(N)cc4O)=O)C1C3C2 57717,N1(C(CS(=O)(=O)NC)=O)CCCCC1C1CCCN1C(=O)CN1CCCNC1=O 57718,C1(CCNC(C2CC2CF)=O)CCN(C(C2CCCC2c2nc(S)n[nH]2)=O)CC1 57719,C(=O)(C(CCN(C)C)NC(=O)C(C)C#N)NC1C(C)CC1 57720,N1(C(C(CC)CC)=O)CC2OCCN(C(=O)C(C3CCOCC3)C)C2C1 57721,c1(CC)c(C(=O)NCC2CC(C)(C)CN2C(=O)C(C)OCC(C)C)cccc1C 57722,C(COC)(CC(=O)N1CC(c2cccc(C#N)c2)C1)NC(C(OCCOC)OC)=O 57723,CS(=O)CCC(O)C(=O)NCCCNC(=O)Cc1cccc(CC(F)(F)F)c1 57724,Cc1ccc(C2CCN(C(c3ccc(Cc4ccc(OC)cc4)cc3)=O)CC2)cc1 57725,N1(C(c2c(O)cc(C)c(Br)c2)=O)CC2CCCC(C1)C2C(N1CCC1CO)=O 57726,Cc1cc(N(C2CCC2)C)nc(=NCCOc2conc2C)[nH]1 57727,n1(CCC)cccc1C(N1C(C(=O)N(C)CCc2ncccn2)CC1C)=O 57728,CC(C)(CNC(N1CCOC(CCO)C1)=O)C(N)=O 57729,N1(C(C2CC(CNC(c3c(C(C)C)nco3)=O)C2)=O)CC2CC(C)C2C1 57730,Cn1nccc1CC(=O)NCC1CC1CNC(C1CCCCC1)=O 57731,N1(C(C=NOC)=O)CC2=C(C1)CN(C(=O)Cc1ccsc1C)C2 57732,C1(CNC(c2ncc(C)nc2)=O)CC2CCC1N(C(=O)CC1CC(C)(C)CO1)C2 57733,C1(c2n(-c3c(C)cccc3C)nnn2)(NC(C)CF)CCOC2(CCCCC2)C1 57734,S(=O)(=O)(c1ccc(N(C)Cc2ccc(Cl)o2)cc1Cl)NC1CC(C)N(C)CC1 57735,N1(C(c2ccc(CN(C)C)[nH]2)=O)CCCC(CNC(c2cc(Cl)n(C)n2)=O)CC1 57736,C1(C)CCCN(C(=O)C=Cc2cccnc2)C1.C(=O)(CCNC(N)=O)N(C)CN 57737,N1(C(c2c(C)[nH]cc2)=O)CCC(O)C(NC(=O)CSc2nnnn2C2CC2)C1 57738,CC1CN(C(c2cscc2C(F)F)=O)CCN1C(=O)CCSc1nnnn1C 57739,CC(C)(C)CC(O)CC(=O)N(CC(N1CCCC(CO)CC1)=O)C1CC1 57740,c1(N2CCCC(C)(C)CC2)nc(N2CCCOC(C(C)(C)C)C2)c2ncsc2n1 57741,C1(CNC(C(C(=C)Cl)(C)C)=O)C(C2CC2)CCN1C(=O)CCc1cnc(C)s1 57742,C1(C2(O)CN(C(c3ccc(C(F)F)o3)=O)C2)(CNC(c2ccnnc2)=O)CC1 57743,N1(C(=O)Cc2ccco2)CC2CCC(C(=O)NOCC3CCOC3)(C2)C1 57744,C12(C(=O)OC3CCC(c4n(C)cnn4)CC3)CCC(=O)N1CC1(CC1)C2 57745,c1(N(C)Cn2cc(Br)ccc2=O)ccc(Br)cc1NC(C1CCCC1C#N)=O 57746,C1(CN(C(c2ccon2)=O)CC)CCCN(C(=O)CN2CCC(C)(O)C2)C1 57747,C1(c2cn(C)nc2)CS(=O)(=O)CCN1C(=O)Nc1ccc(I)cc1O 57748,N1(c2nc(OC)nc(C)c2)CCC2(CC1)OCCCC2NC(=O)C(C)CN(C)C 57749,c1(CC)cc(C(N2CCC(C(F)C(=O)NCC(C)N(C)C)C2)=O)c(C)o1 57750,Cc1c(Cl)c(C(=O)NC2CCCN(C(=O)C(c3ccccn3)O)CC2)nn1C 57751,C12(C(N3C(C)(C)C(NC(=O)CCC[N+](=O)[O-])CC3)=O)CCOC1CCOC2 57752,C12(COC(c3c(C(=O)OC)cncc3)=O)CC(CNC(=O)C(F)(F)F)(CCO1)C2 57753,Cc1cc(O)nc(CNC(C2CCCC2C(C)C)=O)n1 57754,S(=O)(=O)(c1ccc(-c2cccc(C(F)F)c2)cc1)NC1CCC(=O)NC1 57755,O=C(CC1NC(=O)c2ccccc21)NCC1CCN(C(c2coc(O)n2)=O)C1 57756,N1(C(CSCC#C)=O)CCc2ccccc2C(NC(C2CCC(F)C2)=O)C1 57757,CCCC(C)CC(=O)NC12CN(C(c3cccc(OC)c3N)=O)C(COC)(C1)C2 57758,C1(C(=O)NC2C=CCN(C(C(n3cc(C)nc3)(C)C)=O)C2)CC2CCCC2C1 57759,N1(C(C=CS(CC)(=O)=O)=O)CCC2CN(C(C)C)C(C)C12 57760,c1(C(C)NC(c2ccc(-n3c(C)cc(C)n3)cc2)=O)nc2ccccc2[nH]1 57761,C1(NC(=O)NCc2cscc2Br)CCc2ccccc2C1 57762,c1(C(C)SCC)nc(COC)n(-c2ccnnc2)n1.C1CCCN1S(C)(=O)=O 57763,CCCC(CCC)=CC(=O)N(C1CC(C#N)C1)CC(=O)N(CCOC)CC1CC1 57764,C1(C(N(C)CCOC(=O)CCNC(N)=O)=O)CCS(=O)(=O)N1.C1CCNC1=O 57765,C1(C(=O)NC2CCC(NC(Cc3c(C)cccc3C)=O)C2)CCC12CCOCC2 57766,N1(C(=O)NC(C)Cc2cccnc2)CCc2ccn(C(=O)OC(C)(C)C)c2C1 57767,N1(C(c2csc3nccn23)=O)CCC2(CCCN2C(c2cc(O)cs2)=O)C1 57768,Cc1nnc2n1CCC2(C)C(=O)N1CC=C(CCNC(c2cccn2C)=O)CC1 57769,c1(CCC(c2n(CC(=C)C)nnn2)NC2CCC3CC23)ccccc1Br 57770,c1(C(N2C(C(N3CCC(NC(CC)=O)C3)=O)CC(F)C2)=O)ccnc(C)c1N 57771,Cc1ccc(Br)c(C(=O)NC2CCCCC2NC(C2CN(C)C2)=O)n1 57772,CN1CC2CC2(CNc2cccc(COc3ccc(F)cc3F)c2)S1(=O)=O 57773,C(=O)(C1=NOC(CC2(O)COC2)C1)N1CC(C)(NC(=O)CCOC2CC2)C1 57774,C(CCCCCCC(F)(F)F)NC(C1CC(c2ccc(C)cc2)(O)C1)=O 57775,Cc1ccnc(C(F)(F)C(=O)NCC2CCCN(C(C3CCCN(C)C3)=O)C2)c1 57776,N1(C(CC=CC)=O)CCC(OCCNC(=O)CCCc2ccccn2)C1 57777,N1(C(c2c(CC)n(CC)nc2)=O)CC2(CCC2)CC1CNC(C1OCC1(C)C)=O 57778,CCCC(C)(O)C(=O)N(CC(C)N(C(=O)Cc1ccco1)C)C 57779,CC#CCC(C(=O)NC1CC2CC(O)C1C2)NC(c1ccnc(C)c1)=O 57780,N1(C(CNC(=O)OC)=O)CCCC1C(C)NC(=O)CCc1cncn1C 57781,C(=O)(C(C(=O)OC)C(C)(C)C)N.N1(C(C2(C=C)CC2)=O)CCC(OC)(COC)CC1 57782,CC1CN(CCN(C)C(C2CN(CC(F)F)CC2C)=O)CC(C)O1 57783,c1(C(=O)NC2C(C)CN(C(=O)C3=CCCO3)CC2)cnn2c1CC(C)CC2 57784,C12(C(N3CC(NC(=O)COc4nc(O)nc(O)n4)C3)=O)CCCCC1OCC2 57785,c1(C(=O)NCCCC(C)NC(C(C(C)(C)C)SC)=O)cc([N+](=O)[O-])ccc1C 57786,c1(C(=O)NC2CN(C(=O)Cc3ccoc3)CC2O)cnc2ccccc2c1 57787,Cc1c(C(=O)NCC(F)CNC(=O)C(c2ccn(C)c2)C)cnn1C(C)C 57788,N#Cc1cc(C(N2CCC(C(=O)NCC3CCC(F)C3)C(O)C2)=O)ccc1O 57789,C1(C(=O)NCC2(NC(C3C(C)C3)=O)CC2)COC2CC1C2 57790,Cc1ccc2c(=NCC(=O)N=c3cc[nH]cc3)[nH]c(N3CCCC(C)C3)nc2c1 57791,n1(CC)cc(C(N2CCC(C(C)(C)NC(c3cc(C)cn3C)=O)C2)=O)c(C)n1 57792,N1(C(c2c(C)cc(Cl)cc2)=O)CC(C)(C)OC2(C1)CN(C(c1coc(O)n1)=O)C2 57793,C(=O)(CCCCCC#N)NCc1cc(C(=O)NC(CC(=O)OCC)C)ncc1 57794,N1(C(c2cccc(COC)c2)=O)CCC(C2CCN(C(=O)C=C3CCC3)C2)CC1 57795,C1(NC(c2n(C=C)ncc2)=O)CC2CN(C(c3ccc(F)c(N)c3)=O)CC12 57796,C1(NC(C(N2CCC(O)CC2)C)=O)CCN(C(C2CC(C)(C(C)(C)C)C2)=O)CC1 57797,C(=O)(C(F)CC(C)(C)NC(=O)CCn1ccc(C)n1)N1CC(C#C)C(OC)C1 57798,Cc1cccc2cc(C(=O)NCC3CN(C(=O)COCC(F)F)CCC3C)oc12 57799,C(CCCCCC(=O)N1CCC(NC(C2CC(OC(F)(F)F)C2)=O)C(O)C1)SC 57800,c1(COCC(=O)NC2CC(C)(NC(C3C(C)CC3)=O)C2)ccccc1 57801,n1(C(N2CCCC(NC(N(C(C)(C)CO)CC)=O)C2)=O)cnc2c(N)ncnc12 57802,CC1(C(=O)NCCC(O)C(=O)NCC(O)C2(Cl)CC2)C=CCCC1 57803,c1(C(N(CCN(C(=O)Cc2cc(C(C)C)no2)CC)CC)=O)cncc(C)n1 57804,CCC(C)C(C(=O)N1CCC=CC1C(=O)NCCOCC(C)(C)O)OC 57805,N1(C(c2n[nH]c(C)c2Cl)=O)CC2CCCC(NC(C3CN4CCN3CC4)=O)C2C1 57806,CC(CS(C)=O)C(=O)N1CC(CCNC(=O)CC2=CCCC2)C1 57807,C1(CC(=O)NCC(C)CN2CCCC2)CCCN(C(c2nc[nH]n2)=O)C1 57808,CC1(C)CCc2sc(C(c3nnnn3C3CCOCC3)NCCC3CC3)cc2C1 57809,CC(C)(COC(c1ccc(-c2cnc(F)nc2)cn1)=O)CC(F)F 57810,C(=O)(C1=CCOC1)N1CC(NC(CN(C)C(c2ccc(Cl)cc2)=O)=O)(CO)C1 57811,C1(N(C(C2(CSC)CC2)=O)C)CCC(NC(=O)CN2CCOCC2)C1 57812,C1(C(=O)NCC(C(C)O)C)CCOCCN1C(C1CCC(O)CC1)=O 57813,N1(C(C2CC(C)=C(C)CC2)=O)CC(NC(C2CCCCS2)=O)C2CCCC12 57814,CCCCCCC(C)CC(=O)NC1(COC)CN(C(c2c[nH]nc2[N+](=O)[O-])=O)C1 57815,c1(C(=O)NCC2(NC(C(F)OC)=O)CCC2)cc(-c2cccnc2)[nH]n1 57816,C(=O)(CCCC(=O)NCc1csc(C(N2CCC2)=O)c1)OCC 57817,CC(C)CC(C(=O)NC(CNC(=O)Cc1nccn1C)C1CCC1)n1ccnc1 57818,C(C(C)(C)CC1CN(C(c2csc(C(F)(F)F)n2)=O)C1)NC(CCOCC)=O.O 57819,C1(NC(C(N2C(=O)CCC2=O)C)=O)CCN(CCc2ccc(F)c(F)c2)CC1F 57820,c1(C2(C(N3CC(C)(NC(c4c(Cl)cn(C)n4)=O)C3)=O)CCC2)ccccc1C#N 57821,C1(OC)CCCC1C(=O)NC(C)CCNC(c1cn(C)cn1)=O 57822,C(C(CO)CC(C)C)NC(C1(CCNC(C(C)=C2CC2)=O)CCC1)=O 57823,N1(C(c2c(CNC(c3nc(CCC)oc3)=O)c[nH]n2)=O)CC(O)CC1CC 57824,c1(OC)cnc(C(=O)NC(C)(CNC(C2CCCC2O)=O)Cn2cccn2)cn1 57825,C1(NC(c2c(C)coc2)=O)CCCC(CN(C)C(c2nn(C)cc2Cl)=O)C1 57826,C(=O)(C1CCCc2cc(C#N)ccc21)N(CCNC(C(CN(CC)CC)F)=O)C 57827,C=CC(C)CN=C(NCC1CCCO1)NCC1(CO)CCOCC1 57828,Cc1c(C(=O)NCC#CCNC(c2[nH]c3ccccc3c2Cl)=O)nc2sccn12 57829,N1(C(=O)C=Cc2cnc[nH]2)CC2CN(C(=O)Cc3cccc(O)c3)C2C1 57830,C(CCC(O)CO)N(C(=O)CC1CC1CNC(C1(CO)CCCCO1)=O)C 57831,C1(CNC(C(c2ccc(C)s2)C)=O)CN(C(=O)CCc2cncc(F)c2)CC1C 57832,c1(C(=O)NC2CN(C(c3ccc(C(=O)OC)[nH]3)=O)C3C2C3)ccccc1[N+](=O)[O-] 57833,c1(NCC2CC(O)(CNC(c3c(CC)scn3)=O)C2)cc(C)nc2ncnn12 57834,c1(OC)cc(F)c(F)cc1C(=O)N(CCNC(=O)Cc1cnn(CC)c1)C(C)C 57835,C1(C(=O)OCC)CN(C)C(=O)CN1C(c1ccon1)=O 57836,C#CCC(CCOC)NC(C1COCCN1C(=O)CCS)=O.NCC 57837,CC1Oc2c(C(N3CC4(CCC4NC(=O)COCCF)C3)=O)cccc2NC1=O 57838,C1(C(N(CC(C)NC(c2cc(C(C)=O)oc2C)=O)C)=O)CCS(=O)(=O)N1C 57839,c1(SCCC(=O)N(C(C)CN(C(=O)Cc2ccoc2)C)C)ccccn1 57840,c1(CNC(C2CCN(C(=O)OC(C)(C)C)C2)C)ccc(Cl)cc1C(F)(F)F 57841,N(C1CCCOc2c(F)cccc21)C(c1ccc(SC(F)(F)F)c(F)c1)=O 57842,C(=O)(C(O)CCCNC(c1c[nH]c(=NC)s1)=O)N(CC=C)CCOC 57843,c1(OCC)ccc2ccccc2c1CN1CCC1C(=O)Nc1csc(Br)c1 57844,C1(C2CCCC2)(C(N2CC3(CC(NC(C4CCOC4C4CC4)=O)C3)C2)=O)CCC1 57845,CC1(C)CC1(c1cn(CCC(F)(F)Cl)nn1)NC(=O)CNCCNC=O 57846,c1(NC2C3N(C(c4cc(CCC)on4)=O)CC(CC3)C2)ncc(Cl)cc1[N+](=O)[O-] 57847,N1(CC(C)NC(=O)C(C2CCN(C(c3cc(O)cs3)=O)C2)F)CCCCC1 57848,N1(C(c2c(CC)noc2)=O)CCC(C)C(NC(c2cc3c([nH]2)CCCC3)=O)C1C 57849,c1(C(N2CC(NC(C=Cc3nc(C)c(C)[nH]3)=O)(CO)C2)=O)nccc2occc12 57850,N#Cc1cncc(OCC(=O)NCC2CCCCC2c2ccccc2)c1 57851,Cc1cc(C)c(NC(C2CC3CC3N2Cc2cnc(C3CC3)s2)=O)cn1 57852,C1(C(N2CCCC(Cn3cc(CCCC=C)nn3)C2)=O)CC2(CCOCC2)CO1 57853,C12(NC(CCCn3cc(C(C)(C)NC(C)C)nn3)=O)CC3CC(C1)CC(C)(C3)C2 57854,c1(CC)ccc(N)c(C(=O)NC23CCC(NC(C4CCCO4)=O)(CC2)C3)c1 57855,N1(CC)CCCC(NC(C2CC(F)CN2C(C2CC2CC(C)C)=O)=O)C1 57856,N1(C(c2c(C)nc[nH]2)=O)CC(C)CCC1CNC(=O)COc1ccsn1 57857,N1(C(c2c(C)nsc2)=O)CCC(CNC(=O)CC=Cc2ccccc2)C12CCC2 57858,C#CCC(O)C(=O)NCC1CC(NC(c2cnn(C(C)C)c2C(F)(F)F)=O)C1 57859,S(=O)(=O)(c1ccc2c(c1)NCC2)NCc1c(COC)cccc1 57860,N1(C(c2c(C)nns2)=O)CC2C(CNC(c3ccc(CN(C)C)o3)=O)C2C1 57861,C(=O)(C(C(C)(C)C)NC(c1ccn(COC)n1)=O)NC(CCOCC)C 57862,c1(C(N2CCC(S(N)(=O)=O)C2)C(=O)NCC(C)C)noc2c(Cl)cccc12 57863,N1(C(c2c(C(C)C)n[nH]c2)=O)CC2CC1(C(N1CC(CC(F)F)C1)=O)C2 57864,c1(C(N2CCC(N(C(C(F)=CC)=O)CC)C2)=O)ccc(S(N)(=O)=O)c(C)c1 57865,CC1ON=C(C(=O)N2CC(CCNC(=O)CN3CCCCCC3=O)C(C)C2)C1C 57866,c1(C(=O)NC(CCNC(C(C=C=C)C)=O)C)cccc2c1CC(C)(C)C2 57867,CCCCC(C)C(=O)NC(CNC(C1(CSC)CC(F)(F)C1)=O)CC 57868,CCC(C)C(O)C(=O)NCC1CC2CN(C(c3cc(C)cs3)=O)CC12 57869,C(=O)(C(C)C(C)C(C)(C)C)N(CC)CC1CCN(C(c2ccc(C)n2C)=O)CC1 57870,C(=O)(C1CC=Cc2ccccc21)N1CCC(C)C(NC(C2CC(C)(F)C2)=O)C1 57871,C(CCC(C)C)(C(=O)N(C)Cc1cc(C)cs1)NC(C(C=C)C)=O 57872,N1(C(c2c(CC)onc2)=O)CCC(NC(=O)C=NOC)C(F)C1 57873,C(=O)(C(CC(C)C)NC(C1CC2CCC1N2C(=O)C(=O)NC1CC1)=O)NC 57874,c1(C(N2C(CCNC(C=C(C)Cl)=O)CCC2)=O)cnc(C)cn1 57875,c1(-c2nn(CC(=C)C)c(-c3cn(CC4CCOC4)nn3)n2)ccc(OC)cc1Cl 57876,c1(C(=O)NC(CNC(CC(C)OC)=O)C(C)C)cc2cc(Cl)sc2[nH]1 57877,C(CCC(C)(C)C(=O)NC1CCn2nnnc2C1)NC(C(COC)C)=O 57878,c1(C(N2CC(OC)C(NC(=O)C3=CC(C)CC3)C2)=O)ccc(C(F)(F)F)c(N)c1 57879,C1(NC(COCC#C)=O)CCCC1(C)CNC(=O)Cn1ccnn1 57880,C(=O)(C(COC)CC(C)C)NC1CC(CNC(C(CC)SC)=O)C1 57881,CC1CC(NC(c2cc3n(n2)CCO3)=O)CCN1C(c1cc[n+]([O-])cc1)=O 57882,c1(OCC)ccccc1OCCNCC1COCC1(C)C 57883,N1(C(C(C)NC(C)(C)C)=O)CCCC1CCCNC(=O)Cn1cc(Br)cn1 57884,C1(NC(C2(SC)CC2)=O)CN(C(=O)CNC(c2ccsc2)=O)CC1C1CC1 57885,C12(NC(c3ccc(=O)n(CCF)n3)=O)CCCC1N(c1ncc(Br)cn1)CC2 57886,c1(C(N(C(CNC(c2cc(C)cc(F)c2)=O)C)C)=O)cc(Br)cc(C)c1C 57887,CC(C)CC(C)(CNC(C1CC1C)=O)NC(c1cc(CC2CCC2)c[nH]1)=O 57888,c1(N(CC=C)CC)[nH]c(=NC2CC(N3CCC3)C2)nc2scnc12 57889,c1(C(=O)NC(CC)CN(C)C(c2cnns2)=O)ccc(-c2cnn(C)c2)o1 57890,N1(C(C2(CC)CCCCC2)=O)CCCCC(CNC(c2nccc(Cl)c2C)=O)C1 57891,C1(CNC(=O)CCOCC2CCCO2)CCN(C(C2CC(=C(F)F)C2)=O)CC1 57892,C(CN=C(NCC1CCOC1)N1CCc2cc(C)ccc21)C1CC(OC)C1 57893,CC1(C)CC(C(=O)NC(C)(C)CCCNC(=O)CCc2nc[nH]n2)=NO1 57894,C1(CN(C(c2c(COC)noc2)=O)C)CCCC(NC(C2CCC2)=O)C1 57895,C12(NC(CC(=C=C)C)=O)CCCCCC1N(C(C1CC3(C1)CS(=O)(=O)C3)=O)CC2 57896,C1(CCC)CN(C(C2CC2[N+](=O)[O-])=O)CCN1C(=O)COCc1cccc(C)c1 57897,c1(C(N(C2(CC(N3CC(C(=O)OC)C3)=O)CC2)C)=O)csc(C)n1 57898,N#CC1(C(=O)NCC2CC(F)(CNC(=O)Cc3ccsc3Cl)C2)CCC1 57899,c1(C(=O)NCCCN(C)C(c2ccc3cnnn3c2)=O)ccc2c(c1)CCC2=O 57900,C1(NC(C(CO)OC)=O)CN(C(c2oncc2C)=O)C2CCCC12 57901,c1(C(=O)NCC(C)N(C(CC(C(=C)C)O)=O)C)ccc2c(c1)NCCC2 57902,CCCCC(CC)CC(=O)N(C1CCCC1)CCCNC(=O)CC(C)NC(N)=O 57903,N1(C(C2CCN2C(=O)CC2OCCCO2)=O)CC2CC3CC2C1C3 57904,C(=O)(CC(C)C(=O)NCC(C(=O)N1CC=CC1(C)CO)C(C)C)OC 57905,C1(NC(c2c(C)noc2)=O)CN(C(=O)C=C2CCCCC2)C2CCCC12 57906,c1(OC)c[nH]c(C(N2CCN(C)CC2CNC(=O)CC2CCC(=O)O2)=O)cc1=O 57907,Cc1[nH]c(=NC(C)C2COCCO2)sc1S(N)(=O)=O 57908,c1(CC)oc(C)cc1C(=O)NC(C1CC=CCC1)C(=O)NC1CC1O 57909,CC(CO)(C(F)F)NC(=O)CC1(NC(=O)C(N)=O)CC1 57910,C1(C(N(CC(C)CNC(=O)CC2(C)CCC2)C)=O)OCCN(C)C1=O 57911,c1(C(=O)NCC(CC)NC(C2(OC)CCCOC2)=O)cc(O)cc(F)c1F 57912,C1(NC(CCc2n(C)ccc2)=O)CC(NC(=O)Cn2nnc(C3CC3)n2)C(O)C1 57913,N1(C(CN(C)C(c2cnns2)=O)=O)CCN(C(=O)C(C)(C)CC2CC2)CC1 57914,Cc1ccc2[nH]c(=NCC3CC4(CC(NC(=O)CC5CCC6CC56)C4)C3)sc2n1 57915,C(CC(O)CO)NC(C1N(C(COCCOC)=O)CC1)=O 57916,CCC(N=c1cccc(S(=O)(=O)NC(C)(CO)C2CC2)[nH]1)c1cc(C)ccc1C 57917,c1(NC(C2C3(CN(C(c4c(C)ncnc4)=O)C3)C2)=O)c(I)cc([N+](=O)[O-])cc1I 57918,CC12CC1CCN2c1nnc(-c2ccc(Br)s2)o1 57919,N1(C(C(CC=C)C)=O)CCC2(CNC(c3c(F)cc(F)cc3F)=O)CCCCC12 57920,n1(CCC(=O)NC2CC(O)(CNC(C(C3CC3)OC)=O)C2)nc(C)cc1C 57921,CCC(C)(CNC(=O)C(C)OC(C)(C)C)C(=O)N(C)CCOCCO 57922,C(c1ccc(O)cc1)=CC(=O)NCC1CCC(NC(C(C2CCC2)OC)=O)C1 57923,c1(C(=O)NCCCCN(C(C=Cc2ncc(C)[nH]2)=O)C)cnc2ccccc2c1 57924,c1(OCC(=O)NC(CCCNC(CCNC(C)=O)=O)C)ccc(C)c(C)c1 57925,C#CC1(C(=O)NC2COCC2CN(C)C)CCN(C(=O)C(n2cc(C)cn2)C)C1 57926,N1(C(CC(C)n2cccn2)=O)CCCC(C)(NC(c2ccc(CO)cn2)=O)C1 57927,c1(C(=O)NCCN(C)C(C23C4C5C2C2C3C4C52CO)=O)csc2ccccc12 57928,C1(CNC(CNS(NC)(=O)=O)=O)CN(C(=O)CN2CCCC2CO)CCO1 57929,N1(C(C(C)=O)=O)CCCCC(Cn2cc(-c3ccc(N)c(F)c3)nn2)C1 57930,N1(C(c2c(C)c(N)ccc2)=O)CCC(C2CCCN(C(c3occc3Br)=O)C2)C1 57931,CC(C(C)(C)O)N(c1nc(C2CCCCC2)cs1)C(C1CC=CCC1)=O 57932,C12(CNC(CSc3c(OC)cccc3)=O)CCC1CN(C(=O)C1=CCOCC1)C2 57933,c1(C(=O)NC2C(CNC(C3N(C)C(=O)CCC3)=O)C2)cc(F)c2ccccc2c1 57934,c1(C(=O)NC2CC2)ccnc(-n2cc(C3CC34CCC4)nn2)c1 57935,N1(CC)CCCCC1C(=O)NCC1CC(C(=O)NCCC2CC(=O)N(C)C2)C1 57936,c1(C(N(C)CC2CCCN(C(COCCCC#C)=O)C2)=O)cc(F)c(F)cc1O 57937,N1(C(CC2ON=C(CC)C2)=O)CCN(C(c2cc(Cl)no2)=O)CC1C(C)C 57938,N1(C(c2ccc(=N)[nH]c2)=O)CCC(F)(CNC(=O)CC2CNC(=O)C2)CC1 57939,c1(C(=O)NCC(CNC(c2cc(C)c(C)nc2)=O)CO)ccc2cn(C)nc2c1 57940,CC1CN(CC(O)CNC(=O)NC2CC=CCC2)CCO1 57941,C(=O)(CN=c1cc[nH]cc1)N1C(CNC(c2ccc(F)c(C)c2C)=O)C(C)CC1 57942,C1(n2cc(CNC(CCC=C)=O)nn2)CCCN(C(c2cnn(CCO)c2)=O)C1 57943,c1(C(N2C(CNC(C(C)CC(N)=O)=O)CC(O)C2)=O)cc2ccccc2[nH]1 57944,c1(C(C)C(N2CCC(c3cn(CCCCC(=O)O)nn3)CC2)=O)cccc(C#N)c1 57945,c1(C(N2C(C(=O)Nc3cc(SC)n[nH]3)CSCC2)=O)cc(Cl)nc(Cl)c1F 57946,CC1(C(=O)NC2CCCC(NC(c3cccc(C(F)(F)F)c3)=O)C2)CCCCO1 57947,Cc1nc(N2CCC3CC(NC(C4CC4(F)F)=O)CCC3C2)ncc1[N+](=O)[O-] 57948,Cc1nc(=O)n(C2CCN(C(C3CCN(C4CCSCC4)CC3)=O)CC2)[nH]1 57949,C1(C(N2CCC(C(=O)NCC(c3cnn(C)c3)C)CC2)=O)C2CC3C(C2=O)C13 57950,C1(CC=C)(C(N2CCC(C)(N(C)C)C2)=O)CCN(C(=O)CN2CCN(C)CC2)C1 57951,C1(C(N2CC(NC(C(=CC3CCCC3)C)=O)C(n3cccn3)C2)=O)C(C#N)C1(C)C 57952,C=C=CCCC(=O)N(C)CCOCCC(N1CCCCC1C(C)(C)O)=O 57953,c1(COC(C)=O)ccc(C(=O)NC(C(=O)NC2(CCC)CC2)C2CC2)s1 57954,n1(CC)ccc(CC(=O)NCC2(C(=O)NC3CC(OC(C)C)C3)CC2)n1 57955,c1(CC)cc(C(=O)NC(C)(C)CNC(=O)C(COC)N(C)C)c(C)nn1 57956,C(=O)(CCCCC(F)F)NCCC(C)N(C(C(C)Cc1ccc(Cl)cc1Cl)=O)C 57957,c1(OC)ncc(C)cc1C(=O)NCC(C)(CNC(=O)C(F)CC(C)C)OC 57958,c1(C(=O)NC(C)CS(C)(=O)=O)coc2c1CN(C(c1cc3n(n1)CCO3)=O)C2 57959,c1(C(=O)NC2CCC(CNC(c3c(C)ncs3)=O)C2)cc(F)cnc1O 57960,N1(C(C2(NC(c3nccc(C)c3N)=O)CCCC2)=O)CCCC2CCCCC12 57961,Cc1cc(C(=O)NCC2CC2CNC(c2ccsc2)=O)c(C)s1 57962,C1(CNC(C2CCC(=O)O2)=O)CC(C(=O)N2CCCC2CO)=NO1 57963,c1(CN(C(C2C(NC(C(C)=C(CC)C)=O)COC2)=O)C)cccnc1O 57964,n1(C(C(=O)OC)C)nnnc1C1(C(c2cscn2)C)CN(C(=O)OCC)C1 57965,c1(CC)onc(C(=O)NC2CCOCC2NC(=O)CC(C)n2ccnc2)c1C 57966,CCC(C)(C(=O)NCc1ccccc1CN(C(=O)C(C)C(=O)OC)C)C(N)=O 57967,c1(CCC(=O)NCC2CC2NC(C23CCCC2C3)=O)cccc(Br)c1F 57968,Cc1nc(-c2ccc(Cl)s2)sc1CN(C(=O)OC)CCc1ccccc1Br 57969,C(=O)(CC1=CCCC1)NC1C(NC(C(N2CCC(O)CC2)C)=O)C1 57970,N1(C(Cc2ccn(C)n2)=O)C(C(=O)Nc2nc3c(s2)CCC3)C2CC(F)C1C2 57971,N1(C(C2CCC(C(=O)NC(C)C)CC2)=O)CCCC(NC(C2CC(F)C2)=O)CC1 57972,Cc1cnsc1C(N1CCC1CNC(=O)CCNC(c1cnccn1)=O)=O 57973,N1(C(C(=O)NC)C)CC2CCC1C1CN(C(=O)CCCN3CCCC3)CC21 57974,N1(C(C=CC(C)(C)C)=O)CCN(C(=O)COc2ccc(F)c(Cl)c2)C2CCC12 57975,CP(C)(=O)c1cccc(C(=O)NCC2CC(NC(c3ccc(Cl)nc3O)=O)C2)c1 57976,C1(CC(N2CCC(C)(CCC)C2)=O)CC(C)(C)CN1C(=O)CC(C)(C)C 57977,C(=O)(C1=CS(=O)(=O)CCC1)N1CCC2C(NC(c3n[nH]c(C)c3C)=O)C2CC1 57978,c1(C(=O)NCC(C)N(C)C(C2C(C)C2C)=O)cc(S(=O)(=O)NCC(N)=O)c[nH]1 57979,Cc1[nH]nc2ncc(C(N3CCN(C(=O)C(CO)NC(N)=O)C(C)C3)=O)cc12 57980,c1(NC(C2C(NCc3cc(C)sc3C)CCCC2)=O)c(C)ccc2n[nH]cc12 57981,N1(C(c2n(C=C)nnc2)=O)CC(C)CN(C(=O)C=Cc2cn(C)nn2)C(C)C1 57982,c1(C(=O)NC(C)CCCCNC(c2cccc(CO)n2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 57983,C1(NC(CCSCCCC)=O)CCC(CCC(=O)N(C)CCOC)C1 57984,c1(C(N2CCC(NC(CSC(C)C)=O)C(F)C2)=O)ccc(Cl)c2ccccc12 57985,CC1C(N(C)C(C2(C)CC(NC(c3cc(C#N)cs3)=O)C2)=O)CCCC1C 57986,c1(CS(=O)(=O)NCC2(S(C)=O)CC2)cc2ccccc2s1 57987,Cc1ccc(C(=O)NCC2CCN2C(=O)CCCc2ccccn2)c(C)n1 57988,c1(C(=O)NC2CCC(N(C(Cc3c(C)con3)=O)C)CC2)cnc(CO)nc1C 57989,N1(C(C(C)(C2CCC2)NC(C2CCOC2=O)=O)=O)CCC2(CC1)N=N2 57990,c1(C(=O)NCC2C(CNC(c3cc(C#N)sc3)=O)C2)ccc2c(c1)S(=O)(=O)NC2 57991,c1(C(N2C(CNC(CC3(C=C)CC3)=O)C(C)CC2)=O)cnc(OC)nc1C 57992,N(C1c2ccccc2CC1NC(=O)C(C)N(C)C)C(c1n(C(CC)C)ncc1)=O 57993,N1(C(CC(CC)CC)=O)CC2CCC1CN2C(=O)C(C)N1CCC1 57994,C=CC1(CC(N2CCC(C(C)C)(CO)C2)=O)CN(C(c2ccncc2NC)=O)C1 57995,C(CS(C)(=O)=O)(C(=O)O)NC(c1c(C(C)(C)C)nn(CC(F)(F)F)c1)=O 57996,C1(C2CCN(C(c3cc(NCC)cnc3F)=O)C2)(NC(CSCC)=O)CC1 57997,C1(CC(N2CC3C(NC(c4ccc(C(N)=O)[nH]4)=O)C3C2)=O)CCCC2(CC2)C1 57998,c1(C(=O)NCC2COCC2NC(C2CC2(Cl)Cl)=O)cc2c(nc1O)CCCC2 57999,C(=O)(C(CC)N(C)N1Cc2ccc(CC)cc2C1)OCC 58000,C1(CC(=O)NCC=CC(=O)NCC2(OC)CCOC2)CCCCC1O 58001,C1(NC(C2(NC(C)C)CC2)=O)CCC(CNC(C2(F)CCOC2)=O)CC1 58002,Clc1cccc2c1CCC2NCc1csc(C2CCCO2)n1 58003,N1(C(C2CC3(CC(NC(C4C5CCC(=O)C45)=O)C3)C2)=O)CCC2(CCCC2)CC1 58004,c1(C(=O)NC2CC(F)(CNC(C3CC34CC4)=O)C2)nn2cccnc2c1Cl 58005,c1(C(=O)NCC23C(CN(C(C(C)CC(N)=O)=O)C2)C3)ccc(Cl)c(O)c1N 58006,N1(C(c2ccc(C)nn2)=O)CCN(C(=O)C(C(C)(C)C)n2ccnn2)CC1C 58007,c1(OC)cc(F)c(F)cc1C(N1CCC(CN(C)C(c2cnc(C)n2C)=O)C1)=O 58008,c1(CC2CC(OC)CN2c2cc(SC)nc(C)n2)cnn2ncccc12 58009,C12(NC(=O)Cn3cccn3)CCCC1N(C(c1ncccc1O)=O)CC2 58010,c1(C(=O)NCC(C)NC(=O)CCc2cnn(C)n2)cccc2c1OC(C)C(=O)N2 58011,C(C(CC(C)C)C(=O)NCCOCCN(C)C(C1(Cl)CCC1)=O)OC 58012,c1(C(N(CC(C)NC(C2(c3ccno3)CC2)=O)C)=O)cccnc1-n1ccnn1 58013,N1(C(C(CNC(C2CCC(CC)CC2)=O)O)=O)CCC2(COC(C)C2)C1 58014,c1(C(N2CC=CC(NC(c3ccc(C)c(F)c3)=O)C2)=O)cccc2c1OCCC2 58015,N1(C(C(C)NC(N)=O)=O)CC23CCCC2(C1)CN(C(=O)CC(C)(F)F)C3 58016,C#CCC(O)C(=O)N1C(C(N2CCC2C)=O)CCC1C(C)C 58017,N1(C(C(C2CCN(C(C(C)(C)C3(O)CCC3)=O)C2)F)=O)C2CSCC1C2 58018,n1(CC)c(C(C)OC(C)C(=O)NCC(CC(C)C)OC)nc2ccccc12 58019,C1(NC(CC2C(C)CC2)=O)CC2CC(NC(c3cnn(C)c3C(F)F)=O)CC12 58020,N1(C(c2cnc(CC)nc2)=O)CC=C(CNC(C2CC23CCCCC3)=O)CC1 58021,c1(OC)ncc(F)cc1C(=O)N(C1CCCCN(C(C2CC(C)=NO2)=O)C1)C 58022,C(=O)(C(C)CC(N)=O)NC1C(NC(c2ccc(CSC)o2)=O)CC1 58023,c1(NC(N2C(CC(N3CCOC(O)C3)=O)CCC2)=O)cncc(C(F)(F)F)c1 58024,C1(C(=O)NCC(C)NC(C2CC(O)C2)=O)CCCC1O 58025,C1(C(C(=O)NC(C)(C)C)N(C)CC2(CC(C)C)CC2)CC(C)CC(C)C1 58026,N1(C(C2(C(=O)OC)CC2)=O)CC2(C1)CN(C(c1nc(C(C)=O)sc1N)=O)C2 58027,n1(CC)nc(C)c(COC(c2ccc(N3CCCC3)nc2Cl)=O)c1C 58028,c12ccc(cc1[N+](=O)[O-])c(=O)[nH]2.N1(CC)CCCC(C(=O)NCCOC)CC1 58029,CC1(CNC(C2CCCC(F)(F)C2)=O)CCN(C(c2sccc2C(F)F)=O)CC1 58030,c1(C(N(CCN(C(c2n(CC)ncc2)=O)C(C)C)C)=O)cnnc(Cl)c1 58031,N1(C(C(C)SCC(=O)Nc2ccc(Cl)cc2)=O)CCN(C)C(C)(C)C1 58032,CC1(C)C(NC(C2(c3cccs3)CC2)=O)CC1CNC(=O)Cc1nnc(O)s1 58033,Cc1cnccc1CCNC(=O)CC1CCCN(C(c2cnn(C)n2)=O)C1 58034,N1(C(C(CCC)N(C)C)=O)CC2CCC1CN2C(=O)C(O)CC(C)C 58035,N1(C(c2c(Cl)cc(C)s2)=O)CC2(CCC(CNC(C3(O)CCC3)=O)O2)C1 58036,c1(CC)nn[nH]c1C(=O)NCC(C)(C)CNC(c1ccn(CC)n1)=O 58037,c1(C(N2CCC(O)(C(C)(C)C)C2)=O)cc2cc(Cl)ccc2cn1 58038,CCCCCCCC(F)C(=O)Nc1ccc(C(C)C(=O)OC)cc1 58039,N1(C(C2C(OCC)C2)=O)CC(CNC(c2cccc(N3CCOCC3)n2)=O)CC1C 58040,C1(NC(c2c(C)n[nH]c2)=O)CN(C(=O)CC2(C)CC(F)(F)C2)CC12CCC2 58041,n1(CCCCNC(CN(C(=O)OC)C(C)C)=O)cnc2ccccc12 58042,N1(C(C(C)Cn2cccn2)=O)CC(CO)C2(C1)CN(C(=O)COCCCF)C2 58043,c1(CC)cncc(C(N2CC=CC(C(=O)NC(C3CCC3)C3CC3)C2)=O)c1 58044,c1(NC)cccc(C(=O)NC(C(C)NC(=O)CCCc2cccs2)C(C)C)n1 58045,C(=O)(C(O)C(F)(F)F)N(CC=CC(=O)NC(C#C)CCC)C 58046,CC1(C)COCCC1CC(=O)NCC12CC(NC(C3CC(O)C3)=O)(CO1)C2 58047,c1(C(=O)OC)csc2c1CCN(Cc1ccc(NC(C)=O)cc1C#N)C2 58048,c1(CCC)cccc(C(=O)O)c1.C12CCN(CC1)C(=O)N2C(C)C.C1CC1 58049,C1(CNC(C(C)OC)=O)(NC(C2(C)COC(C)(C)CO2)=O)CCC(F)(F)CC1 58050,N1(C(Cc2ccn(C)n2)=O)CCCCC(Cn2cc(Cc3ccccc3)nn2)C1 58051,C#CCCCCC(=O)N(C)CC1CCCN(C(=O)C(c2cc(Cl)cc(Cl)c2)C)C1 58052,N1(C(C(c2nc(F)ccc2Cl)C)=O)CCC(C2(NC(C3CC=CCC3)=O)CC2)C1 58053,c1(SCC(=O)N(CC(C)CNC(=O)C(C)c2ccsc2)C)ccc(F)c(F)c1 58054,Cc1cc(C(=O)NC(C)CC(C)NC(C2(O)CC2)=O)cc(Cl)c1 58055,c1(C(=O)NCC2(C)CCN(C(c3cnco3)=O)C2)ccc2sc(O)nc2c1 58056,CC1c2cc(Cl)cc(F)c2CCN1C(C1CC12CCOCC2)=O 58057,n1(CC(=O)N(CC(C)NC(C(CC)(C)C(N)=O)=O)C)ncc2ccccc2c1=O 58058,CC1CC(C(=O)N(C2(C(N3CCC(c4ncco4)C3)=O)CCC2)C2CC2)CCS1 58059,C1(F)(CNC(=O)C(=O)NCC2CC2)CN(C(c2csc(CO)n2)=O)C1 58060,C1(n2cc(C(N3CCCC3)(C)C)nn2)CCCN(C(C2CC23CCCC3)=O)C1 58061,c1(C(=O)NCCCNC(CCCC(CC)C)=O)ccc2c(c1)OCCN2 58062,c1(NCC)cccnc1C(=O)NC1CC(C)N(C(=O)CCSC)C1 58063,N#Cc1cc(NC(C23CC2CN(Cc2ccccc2Cl)C3)=O)cc(Br)c1 58064,c1(C(=O)NCC(CNC(C=C(C)C)=O)O)ccc(F)c(C(F)(F)F)n1 58065,C(CN=c1[nH]cncc1I)(N(C(c1ccc(C#C)cc1)=O)C)C1CC1 58066,N1(CC(C)(C)C)CCC(C(=O)NCC(C2CCCC2)N)CC1 58067,CCCS(=O)(=O)c1ccc(S(=O)(=O)NC(=O)OCC(C(=O)OC)C(C)(C)C)cc1 58068,O=C(C1COc2ccccc21)NCCOC1CN(C(=O)CC2(O)CC2)C1 58069,N1(C(=O)C=CC2CCOC2)CCC2CCC(C1)N2C(=O)C(F)C1CCOC1 58070,C=C1CC(C(N2CCCCC2c2ccccc2F)=O)N(C(c2ccncc2)=O)C1 58071,COn1cnc(C)c1C(N1CC(CNC(=O)Cc2ncc(Cl)s2)C(C)C1)=O 58072,C=CC1(CC(=O)NCc2[nH]nnc2CC)CN(C(C2(COC)CC2)=O)C1 58073,C1(C2CCN(C(=O)CCc3ccc(C)s3)C2)(NC(C(C)NC(C)=O)=O)CC1 58074,C(=O)(C(C)(C)C(C)NC(=O)CC1CNC(=O)O1)NCc1c(C)nccn1 58075,c1(C(N2CCC3CC3(C(=O)Nc3nc[nH]n3)C2)=O)cc2ccccc2[nH]1 58076,c1(NC(C2CCCN(c3cc(OC)nc(OC)n3)C2)=O)c(Cl)nc(C)nc1Cl 58077,c1(C(=O)NCC2(O)CCN(C(C3CCCCO3)=O)C2)cc(Br)cnc1S 58078,c1(SCC=C)ccccc1C(=O)NCCNC(c1cnn(C)c1CCC)=O 58079,C(=O)(C(C(C)(C)C)OC)NCCC1CCN(C(c2c(SC)nn(C)c2)=O)C1 58080,C1(C#CC(=O)NC(c2ccccc2)C(N2CCCC(SC)C2)=O)(CC)COC1 58081,C1(NC(C2CCC(C)(C)O2)=O)CC2(CCN(C(c3cc(Cl)c(N)cc3F)=O)C2)C1 58082,n1(CC(=O)NCCCCNC(=O)CSc2ccc(F)cc2)ccccc1=O 58083,C1(C(N2CC(C)(CO)C2)=O)(NC(=O)CSCCC#N)CCOCC1 58084,C1(NC(c2nnnn2Cc2cccc(F)c2)(C)C2CC2)CC(=O)N(C(C)(C)C)C1 58085,c1(C(N2CC(SC)C(NC(=O)CC3(CO)CCC3)C2)=O)c(F)ccc(C)c1F 58086,c1(OC)cccc(C(=O)NC2CN(C(C3(C(F)(F)F)CCC3)=O)CCC2C)c1F 58087,N1(C(c2c(C)cc(C(F)(F)F)s2)=O)CC(C2CN(C(=O)CC(C)(F)F)C2)C1 58088,c1(SC)nc(C(=O)NCC(O)CCNC(=O)C(O)CC2CC2)cs1 58089,N1(C(C2N(CC)CCC2)=O)CCC(C(F)F)(CNC(c2coc(N(C)C)n2)=O)C1 58090,Cc1c(NC(O)CC)cccc1F.C(CCC(C)(C)C)N1CCCC1c1ccccc1Cl 58091,C1(CNC(c2cc(C)n(C)n2)=O)CCCCN(C(=O)Cc2ccc(O)cn2)CC1 58092,C12(c3ccn(CC(=O)OC)n3)CCC(CC1)N2C(=O)C(N1CC2CC2C1)C 58093,N1(C(C(=O)NCc2c(C)nn(C(C)C)c2C)=O)CC2CCCOC2C1 58094,c1(C(=O)NC2C(C)CN(C(c3cnc[nH]3)=O)C2)cnc2c(c1)OCCN2 58095,Cc1ncc(C(=O)NCC2CC(NC(=O)CC34CC(C3)C4)C2(C)C)n1C 58096,N1(C(c2c(NC)cncc2)=O)CCN(C(C23CCC2CC3)=O)C(CO)C1 58097,c1(CNC(c2ccc([N+](=O)[O-])s2)c2n(CC=C)nnn2)cccc2ccccc12 58098,C12(NC(c3cc(C)n(CCO)n3)=O)CCCN(C(=O)C(C)(C)CO)CC1C2 58099,c1(C(=O)NC2(CO)CCN(C(C(CC)(C)OC)=O)C2)ccc2c(c1)CCO2 58100,N1(C(C(OC)OC)=O)CCC2(CCC(CNC(C3CC4CCCCC34)=O)O2)CC1 58101,c1(C(=O)NC)ccc(C=CC(=O)N(CC2=CCCOC2)C)cc1 58102,C1(OC(=O)CSC2C(C(=O)O)C2(F)F)Cc2ccccc2C1=O 58103,Cc1ccccc1COCC(=O)NC(CNC(C1CCC12CCC2)=O)C(C)C 58104,C1(C(C)NC(=O)C=CC(F)(F)F)CCN(C(=O)Cc2nccn2C)CC1 58105,Cc1cc(C#N)nc(NC23CCCC2CN(C(C2(C)C(C)(C)C2(C)C)=O)C3)n1 58106,Cn1ncc2ncc(C(N3CCC4(CCCN4C(C4CC4F)=O)C3)=O)cc12 58107,CCS(=O)(=O)CC(=O)NCCC1(O)CCCN(C(=O)CCCc2nc(C)cs2)C1 58108,C(C(C)C(F)C(=O)NCCCc1ccco1)NC(C(C)=CCC)=O 58109,Cc1onc(-c2cccs2)c1C(N1CC2C(CN(C)C(C3CCC3)=O)C2C1)=O 58110,C1(CNC(C(C(C)C)C)=O)CCN(C(c2ccc(-c3cccs3)o2)=O)CC1(F)F 58111,C1(CC(=O)NC)CN(C(=O)C2=CCSC2)CCN1C(=O)C=C(C)C(C)(C)C 58112,C1(N(C(=O)CSCc2ccncc2)C)CC2CC1N(C(=O)C(F)=C1CCC1)C2 58113,c1(NC(C2(C)N(C(c3n(C)cnc3)=O)CCC2)=O)ccc(F)cc1I 58114,Cc1cc(C(N2CCSCC2C(=O)N(CC(C)C)CC(C)C)=O)c(C)n1C 58115,CN1CCCCC1C(=O)NCC(C)(C)C(=O)NCCCC1(O)CC1 58116,N1(C(C(C=C)(F)F)=O)CC2CCCC(C1)N2C(=O)C=Cc1ccncc1 58117,C#CCCC(O)C(=O)NCC1(CCNC(=O)C(C)Cc2ccccc2Cl)CC1 58118,S(=O)(=O)(c1ccc(N(CC(O)CF)C)cc1Cl)N(C)Cc1c(C)ccs1 58119,C1(CNC(=O)COCCF)CCN(C(=O)COc2ccon2)CC1(F)F 58120,N1(C(CCCOCCOC)=O)CC2(C1)CN(C(c1cnc(C)n1C)=O)C2 58121,C1(NC(CC=C(C)C)=O)CC2(CCN(C(C3CC3Br)=O)CC2)C1 58122,C1(C(C(=O)NCC2CC(CC)C2)C)CCN(C(=O)CN2CC3CC3C2)C1 58123,c1(CN2CCCC(C(=O)NC(CC)C(=O)OC(C)(C)C)C2)nc2ccccc2n1C 58124,c1(C(=O)NCC(C)CN(C(=O)C(C)(C)C#N)C)nn(C)c(Cl)c1Cl 58125,c1(C(=O)NCCN2CCN(C(c3c(NC)cccc3)=O)CC2)ccc([N+](=O)[O-])o1 58126,C1(C)(CNC(Cc2ccn(CC)n2)=O)CC(F)(F)CN1c1nc(C2CC2)ns1 58127,Cc1c(NC(=O)C(C)OC(F)F)cc(F)cc1CO 58128,Cc1cc(C(=O)NC(CNC(=O)Cc2cnoc2)C(C)C)cnc1O 58129,CCCC(CNC(c1ccc(OC)o1)=O)C(=O)NC1CC12CCC2 58130,c1(OC)ccc([N+](=O)[O-])c(C(=O)NCC2CCN2C(=O)CC2CCC2)c1 58131,C1(CCC)CN(C(=O)CNC(c2cccnc2)=O)CCN1C(=O)C#CC(C)C 58132,c1(C(=O)NCC(CC)NC(C2CCCC(C#N)C2)=O)cc2c(C)cc(Cl)cc2[nH]1 58133,C1(C(=O)NCC(C)N(C(Cc2cc(C(C)C)no2)=O)C)CCC([N+](=O)[O-])CC1 58134,N1(CCCCCNC(C(CC)C)=O)CCC(n2cc(-c3ncc(F)cn3)nn2)CC1 58135,C(c1ccc(Cl)s1)=CC(=O)C(N(CCN(CC(F)(F)F)C)C)=O.N 58136,C1(NC(CC(C=C)(C)C)=O)CCC(O)CN(C(=O)CCOCC2CCCO2)C1 58137,c1(C(C)(C)NC(c2ccccc2)CO)ccc(F)cc1F 58138,CCC(C)CC(C(=O)NC)NC(=O)CCN1CCOC1=O.c12cnn(C)c1NC2=O 58139,C1(NC(C2C(C)(COC)C2)=O)CN(C(=O)CCc2cccc(OC)c2)CC1O 58140,C12(C(=O)NCCCCN(C(CC3CC(C(C)C)OCC3)=O)C)CCC(F)(CC1)C2 58141,c1(OC)ccc(C(=O)NCCn2cc(C(=O)NCC3CCOC3C)cn2)cc1 58142,C1(NC(c2c(OCCC)cccc2)=O)CCN(C(=O)CS(=O)(=O)CC)CC1CC 58143,C1(NC(CSc2nc(C)[nH]n2)=O)CCN(C(C2CC3C=CC2O3)=O)CC(C)(C)C1 58144,N1(C(CSc2cn(C)nc2)=O)CCC2CCN(C(=O)CC3CC3(C)C)CC12 58145,Cn1ccc2c(C(=O)NCC3CCCCN3C(C3CS(=O)(=O)C3)=O)[nH]cc2c1=O 58146,c1(S)cc(C)cc(C)c1OC.CCC(CN(CCC(=O)OC)S(C)(=O)=O)CC 58147,N1(C(CC(C)F)=O)CC2(C1)C(NC(c1cc3ccc(Cl)cc3[nH]1)=O)CCS2(=O)=O 58148,c1(SCCC(=O)NC2CN(C(=O)CN3CCCCC3)CC2O)ccc(F)c(F)c1 58149,C1(N(C(CNC(CCC)=O)=O)C)CCCC(NC(=O)CCOC)C1 58150,C(CNC(C)=O)(C(=O)O)N(C(CCSCC)=O)C 58151,C1(C(N(C2CN(C(Cc3c(C)nn(C)c3C)=O)C2)C)=O)CC2(C)CCC1(C)O2 58152,C(=O)(C(CC)(CC)CC)NCc1c(C(N2CCC(OCC=C)CC2)=O)scc1 58153,c1(NC(=O)NC(CCCC#C)c2ccccc2)ccc(S(=O)(=O)C2CC2)nc1 58154,C(CC(C)(C)C(=O)NC1CC(N(C(=O)CSc2cnn(C)c2)C)C1)OC 58155,Cc1cc(C(=O)NCC2(CNC(=O)C(F)CC3CCCC3)CCC2)nc(C)c1 58156,C1(NC(c2scc(C)c2Cl)=O)CCC2CCN(C(C3CC3(F)F)=O)C12 58157,c1(C(=O)NC(C2CCCN2C(c2cnc(O)o2)=O)C)cc(O)nc(Cl)c1 58158,C12(CNC(c3n(C)ncc3)=O)CC3CC(CC(C3)C1NC(=O)CSC(F)(F)F)C2 58159,CC(CNC(=O)CN1CCCC1=O)C(F)C(=O)NCC1(CF)CC1 58160,Cc1cc(NC(C2(CNCc3ccn(C)n3)CC2)=O)n(-c2ccccn2)n1 58161,c1(NC)cccc(C(=O)NC(CCN(C)C)C(=O)NC(CCOC)C(C)C)n1 58162,N1(C(=O)CC2CC3(CCC3)CO2)CC2OCCN(C(c3ns[nH]c3=O)=O)C2C1 58163,c1(C(N2CC(NC(c3sc(CC)c(C)c3)=O)C(F)CC2)=O)c(F)ccc(F)c1O 58164,C=C1CCN(C(c2cn(C)nc2OC)=O)C(C(=O)NCCC(O)CCO)C1 58165,C1(C(=O)NCc2c(C)cnn2C)CC(N=[N+]=[N-])CN1C(c1cc(F)n(C)n1)=O 58166,S(=O)(=O)(c1ccc(O)c([N+](=O)[O-])c1)NCCCC(=O)OC 58167,c1(N(C2CCN(C(c3ccsc3C(F)(F)F)=O)C2)C)cc(F)ncn1 58168,c1(OCC)ccc2c(C(=O)N(CC(=O)OC(C)(C)C)C)c[nH]c2c1 58169,CC#CCCCC(=O)NC1COCC1C(N1CC(OC)CC(C)C1)=O 58170,Cc1cc(C)c(C(=O)NC2CCN(C(=O)CCCOC(C)C)C2C)o1 58171,CN1CC(C(=O)NCCCOCCOCCNC(C2CC(F)C(=O)N2)=O)CC1=O 58172,c1(NCC)cccnc1C(=O)NC(C)CC(C)NC(=O)C(C1CCCC1)OC 58173,C1(O)(CN(C(C=CC(CC)=CC)=O)C)CCN(C(=O)CC2(O)CCC2)C1 58174,N1(C(C)=O)CC2CC2(C(=O)NC2(c3cccnc3)CC2)C1.N12CC(C1)C2=O 58175,c1(C(=O)NC(C)C(c2ccccc2)NC(=O)COCC(F)F)ccc(N)cc1O 58176,c1(NC(C)CN(C(=O)C2=CCSC2)C)ncnc2c1nnn2C1CC1 58177,c1(C(=O)NCC2(C)C(C)CN(C(=O)CC3CC(F)C3)C2)cc2c(s1)CCOC2 58178,N1(C(c2cc(C)sc2)=O)CCCOC(CNC(C2CCCN(C)C2)=O)C1 58179,O=S(=O)(c1ccc(=NCC2CCOC(C3CC3)C2)[nH]c1)NCC12CC(CCO1)C2 58180,c1(CC)noc(C)c1C(=O)NCc1csc(C(N2CCC2(C)CC)=O)c1 58181,N1(C(Cc2cc(C)sc2)=O)CC2(C1)CN(C(=O)C(C)OCC(F)(F)F)CC2CO 58182,C(CC(C)(C)C)(c1n(C(CC)C)nnn1)(C1CC1)NC(c1cccnc1)CCO 58183,c1(OCC)ncc(F)c(N2CC3CC2CN3S(=O)(=O)CCCCl)n1 58184,c1(N2CC(C)(C)C2C2CC2)ccc(C#N)c(CNS(C)(=O)=O)n1 58185,CC12CCC(C(=O)NC3CC3NC(c3cc[nH]c4nccc3-4)=O)(CC1)CO2 58186,c1(C(=O)Nc2c(CS(C)(=O)=O)cc(F)cc2)cc(F)c2c(c1)CCC2 58187,c1(C(N2CCC(NC(C(CC)n3cncn3)=O)C2CC)=O)ccn2nccc2c1 58188,C1(CNC(c2nccc(CC)n2)=O)CC2COCC2N1c1nnc(C(=O)OC)s1 58189,c1(CC)[nH]c(C(=O)NC2CC(CO)N(C(c3sc(F)cc3C)=O)C2)nc1Cl 58190,c1(C(N2CC(NC(C(CSC)O)=O)C(C)C2)=O)coc2c(C)cccc12 58191,C1(C(=O)NCC(C)NC(=O)Cc2cnccn2)CC(=O)N(C(C)(C)C)C1 58192,C(c1ccc(F)c2ccccc12)=CC(N1CC(NC(C(C)C)=O)CC(F)(F)C1)=O 58193,c1(C(=O)OC)c(C)ccc(NC(=O)NS(=O)(=O)CC2CCOCC2)c1C 58194,Cc1ccc(-c2noc(C(C)NC(=O)C(C)C(N)c3ccccc3)n2)cc1F 58195,C(=O)(C1CCCc2nccn21)N1CC(NC(c2ncc(OC)cn2)=O)(CO)C1 58196,c1(C(N(CCCOCCNC(C(C)C(F)F)=O)C)=O)n[nH]c2cccnc12 58197,c1(CC(=O)NCC(C)(C)NC(C23COC(CNC(N)=O)(C2)C3)=O)ccnc(O)c1 58198,CC1CC(C(N2CC(CC(C)(C)CNC(=O)CC3CCCCC3)C2)=O)C(=O)O1 58199,CCCC(C(=O)N1CC(NC(C2CC(C)CO2)=O)C(C)C1)N(C)C 58200,C1(C(=O)NCC2(C)CCCN2C(=O)Cc2ccoc2)CC2CCCCCCC12 58201,C(=O)(CS(C)(=O)=O)NCC(C)(F)CNC(=O)CCC(=O)C1CC1 58202,c1(NC(C2CCN(C(c3cnc(Br)o3)=O)CC2O)=O)cc(C(F)F)cc(Br)c1 58203,C1(CNC(c2ccncc2F)c2n(CCC)nnn2)OCCOC1(C)C 58204,N1(C(C(C)CCN(C)C)=O)CCCC12CCN(C(C1(O)COC1)=O)CC2 58205,N#Cc1cc(Cl)c(C(=O)NCC2CC2NC(c2c[nH]nc2-c2ccncc2)=O)s1 58206,c1(C(=O)NC(CNC(c2cn(CCC=C)nn2)=O)CC)noc2ncccc12 58207,c1(NC(C2N(Cc3c(C)nn(C)c3)C3C(C2)C3)=O)cccc2ccccc12 58208,C=CC1(NC(C2CC23CCN(C(=O)Cn2nccn2)C3)=O)CCOCC1 58209,N1(C(CC)=O)CCC(C2CCC2)(CNC(C2CCn3c(C)nnc3C2)=O)CC1 58210,N1(Cc2c(C)ncs2)CCCCC(NC(=O)C=Cc2ccnn2C)C1 58211,C(=O)(CCCCCCCC(=O)N1CCC(NC(=O)C#CC2CC2)CC1)OC 58212,c1(C(C)NC(CNC(C=C(C)C(C)(C)C)=O)=O)cccc(F)c1 58213,c1(C(=O)NC(CCOC)CNC(C2CC=CCC2C)=O)c(OC)ccc(Cl)c1F 58214,CC(C)(C)C(O)C(=O)NCC1CCCCN1C(=O)Cc1n[nH]c(=N)s1 58215,c1(C(=O)NCC2CCN(C(C=CCCC)=O)C2)ccc(F)c(C(C)(C)F)c1 58216,N1(c2cccc(C)c2)N=C(C(=O)NC2CC2NC(c2ccns2)=O)CCC1=O 58217,c1(N(CCC)CCNC(c2coc(C)c2)=O)ncccc1[N+](=O)[O-] 58218,C12CCCCN1C2.CCCC(CNCc1ccccc1)OC 58219,C(=O)(C(C)(C)CS(N)(=O)=O)N1CCC(N(C(c2coc(C3CC3)n2)=O)CC)CC1 58220,c1(C(=O)NCC(CNC(C(C)=C2CCC2)=O)(C)C)n[nH]c2ccc([N+](=O)[O-])cc12 58221,C12(CNC(=O)Cc3cccnc3Cl)CCC(CC1)N2C(c1cccc(CO)n1)=O 58222,CN1CCOCC1C(=O)NOCC(N1CC2CC2(C2CCO2)C1)=O 58223,C1(C(N2C(C3CCN(C(=O)Cn4cnnn4)C3)CCC2)=O)CC2(CCCO2)C1 58224,N(C(=NCCCN1CCOCC1)NCC(CC1CC1)CO)CCC1CCC(=O)N1 58225,c1(CC)ccc(C)c(C(=O)N(C2CCN(C(c3cncnc3)=O)CC2C)C)c1 58226,C1(CNC(CCc2ccc(OC)cc2)=O)C(C)CCCN1C(C1CCCCC1)=O 58227,C(N=c1[nH]c(=NC(C)c2ncc(C)cn2)c2c(ncn2C)[nH]1)C1(OC)CCSC1 58228,S(=O)(=O)(c1c(Br)cccc1[N+](=O)[O-])N1C(C)CC(C(F)(F)F)C1 58229,C1(OC)CCN(C(C2CCOCCN2C(C2CCSCC2)=O)=O)C12CCC2 58230,C12(NC(C(COC)OC)=O)CCCC1N(C(c1cc(C)cc(Br)c1O)=O)CC2 58231,c1(C(=O)NC2CCN(C(C3(C)ON=C(C)C3)=O)C2)ccc2c(ccn2C)c1 58232,c1(N2CCC(N(C(C(C)Cc3cnc[nH]3)=O)C)C2)ncc2c(n1)CCOC2 58233,C1(C(N2CCC3C(NC(c4cc(F)ccc4F)=O)C32)=O)CC2CCC(C1)C2(F)F 58234,c1(C(=O)NC(CC)CNC(=O)CC2CC2CC)cccc(COC)n1 58235,c1(C(=O)Nc2c(C(=O)OC)ccc(OC)c2)ccc2c(c1)N(C)C(=O)C2 58236,C1(C2(O)CN(C(C3CN(C)C(=O)N3)=O)C2)(CNC(c2ccc(C)cn2)=O)CC1 58237,C=CC(C)C(C)C(=O)N1CCC(CNC(c2cccc(Br)c2N)=O)CC1 58238,N1(C(CCNS(C)(=O)=O)=O)CCN(C(c2ccsc2)=O)C(C2CCC2)C1 58239,c1(OC)ccncc1C(=O)NCCC1(C)CCN(C(=O)Cc2n[nH]c(C)n2)C1 58240,C1(CN2CC3(C(C(N(CCCO)CCC)=O)C3)C2)C2CCC3(CNCC13)O2 58241,Cc1nc(C)c(CN2CCCCC2C(=O)NCCCS(=O)(=O)N(C)C)[nH]1 58242,c1(-c2n(CC3C(C)C3)nc(Cn3cncn3)n2)cc2ccsc2s1 58243,CC1(C(=O)NCC2CC(C(=O)NCCn3ncccc3=O)C2)C=CCCC1 58244,C1(CN(C(=O)COc2cccc(Br)c2)C)CCCN(C(=O)C=CC(F)(F)F)C1 58245,C1(CNC(C2C(C)(C)C2CO)=O)CCN(C(=O)Cn2nnc(C3CC3)n2)CC1 58246,N1(C(Cc2ncc(CC)[nH]2)=O)C2CCC1CC(CNC(C1(C)CCC(C)C1)=O)C2 58247,C12(C(N3CC4C(CNC(C(CCCC)C)=O)C4C3)=O)CC3CC(CC(C3)C1)C2 58248,CC1(C)C(NC(c2cccnc2C(F)F)=O)CCN1C(=O)C(F)C(F)(F)F 58249,C1(C(N(CC(O)C(F)(F)F)C)=O)CC2CCC(C1)N2C(C1CCC=CCC1)=O 58250,CCC(C(=O)NCc1ccc(CNC(C2CC3CC(=O)C2C3)=O)cc1F)C(C)C 58251,C(=O)(C(CO)C(C)(C)C)NC(CSNCC)C(=O)NOCCCC(F)(F)F 58252,c1(C(=O)NC2CCN(C(CCCSC)=O)C(C)C2)ccc2c(c1)CC(=O)N2 58253,C1(NC(CCOC(C)C)=O)CCN(C(c2cnc(-c3cccs3)o2)=O)CC(O)C1 58254,C1(N(C)C)CC(C(=O)NC(C(=O)NCCN2CCC2)C2CCCC2)C1 58255,c1(C(C(N2CCC(n3ccnc3)C2)C)=O)ccc(F)cc1 58256,n1(CC=C)cc(C(=O)NC2CCCC2NC(C2CCCN2C)=O)nn1 58257,C1(F)(C(=O)NC(CC(C)C)Cn2cc(C3CCCCC3O)nn2)CCCCCC1 58258,CC(C)CCC(C(=O)NCc1cnn(C2CC2)c1)NC(=O)C(C)NC(N)=O 58259,C(=O)(C(C)(C)S(C)(=O)=O)NCCC(C)N(C)C(c1coc(N(C)C)n1)=O 58260,CS(=O)C1(CNC(C2C=CCN2C(c2cc(C(N)=O)co2)=O)=O)CC1 58261,c1(SC)cccc(C(N2CCC(C(C)NC(=O)C(=O)N(C)C)CC2)=O)c1Cl 58262,N1(C(C2CC(C(=O)OC)C2)=O)CCCCC1C(C)(C)CNC(c1cnco1)=O 58263,CC12CCOC(C(=O)NC3CCN(C(c4scnc4C(C)(C)C)=O)CC3O)(C1)C2 58264,CCC(CC(=O)NC1(C)CC(NC(=O)C=Cc2cccc(C)c2)C1)CC(F)(F)F 58265,N1(CCC)CCC(C(N2CC(NC(c3ccc(C)o3)=O)C(C)C2)=O)CC1 58266,c1(C(=O)NC2CC3CN(C(C#CC(C)(C)O)=O)C2C3)cccn2cncc12 58267,C1(OC)CN(C)C(C)(C(=O)NCC2CN(C(=O)CCc3cccs3)CCC2C)C1 58268,C(=O)(CCCCC(C)(C)C)N1CC2CCC(N(C(Cc3cc(C)on3)=O)C)C2C1 58269,Cc1cccc(C(C)NC(c2cccc(Br)c2Cl)C)c1C 58270,N1(C(c2nc(C)n(C)c2)=O)CCC(C)(C)C1CC(N1CCC(N(C)C)C(C)C1)=O 58271,CC(CS(C)(=O)=O)C(=O)NCC1CN(C(=O)Cc2cocn2)CC(C)(C)C1 58272,c1(CC(=O)NCC2CN(C(C=CCC)=O)CC2O)cnc2n1CCCC2C 58273,N1(C(C2(C(=C)F)CCC2)=O)CCC(CC(=O)O)C(C2CC2)C1.CC#N 58274,Cc1cccc2c(C(=O)NCC3CCCN(C(C4COC(=O)C4)=O)CC3)cnn12 58275,C=C(C)CC(C(=O)N1CC2CC1C2NC(=O)C(C)OC)NC(C)=O 58276,C1(O)(CNC(CCCC#CC)=O)CCCN(C(=O)CCC(=O)N2CCCC2)CC1 58277,N1(C(C(C)C)=O)CCC(CCCNC(=O)CCc2ccnc(Cl)c2)CC1 58278,N1(C(=O)NCC2CCC(C)O2)CCN(C2CC2)c2ccccc21 58279,N1(c2nc(N3CCOCC3)nc(N3CC(C)OCC3)n2)CCC(O)C(C)(C)C1 58280,C1(C(N2CCC(C3(C)N=N3)C2)=O)(NC(C2N(C(C)C)CCC2)=O)CCN(C)C1 58281,c1(C(=O)NCC)ccncc1NC(C(Cc1ccco1)NC(=O)NCCF)=O 58282,CCC(C)(C(=O)NC1COC2(C1)CN(C(=O)CN(c1cnccn1)C)C2)C(N)=O 58283,c1(C(C(=O)NCCC(C)NC(c2cn(C)cn2)=O)C)c(F)cccc1F 58284,CC1(C(=O)NC2CC(C(=O)OC(C)(C)C)C2)CCC(NC(=O)CN(C)C2CC2)CC1 58285,C12(CNC(C(C)C3CC3)=O)CC(CO1)N(C(C1(c3cccs3)CC1)=O)C2 58286,c1(CCCNCC2(CC#C)CCOCC2)cc(C(=O)O)ccc1O 58287,c1(CNc2c(C(=O)Nc3cnc(C)s3)n[nH]c2)c(Br)ccc2c1OCO2 58288,N1(C(C2CCCCO2)=O)CCC2CN(C(=O)C(c3ccccc3F)O)CC2C1 58289,CS(=N)(=O)C1CC(NC(=O)NCc2ccnc(OCC3CC3)c2)C1 58290,c1(C(N2CC3C(CNC(C4C(C(C)C)CCC4)=O)(C3)C2)=O)n[nH]c2c1COCC2 58291,C(=O)(CCC(C)(C)[N+](=O)[O-])NCCCC(C)NC(CCCn1c(C)nc(C)n1)=O 58292,C1(C(=O)NC2(C(=O)NC(c3cccs3)C)CC(O)C2)CCC2(CCC2)O1 58293,c1(C(=O)NC(C)CC2CN(C(C3(n4cc(Br)cn4)CC3)=O)C2)cnn(C)c1 58294,Cn1ccn2ncc(C(=O)NC3CC(CNC(c4cccnc4O)=O)C3(C)C)c12 58295,CCC(CCC(=O)N1CCC(C)(C#N)C1)NC(=O)CN1CC2CC2C1 58296,N1(C(Cc2cc(C)[nH]n2)=O)CCC(CCNC(=O)CCNC(=O)C=CCl)CC1C 58297,c1(C(N(CCC(=O)NCc2scc(C)c2)CCCO)=O)cc(F)cc(F)c1 58298,CC1CN(C(c2cnc(F)c(Cl)c2)=O)CCC1CNC(C1(C(N)=O)CCC1)=O 58299,C1(CCC(=O)N(C2C3CN(C(C4(C)CCCOC4)=O)CC23)C)CCCCCC1 58300,C1(F)(C(=O)NCC2(F)CC(NC(CN(S(CC)(=O)=O)C)=O)C2)CC2(CCC2)C1 58301,N1(C(C(C)c2cc[nH]n2)=O)CCCCCCC1C(=O)NCC(F)F 58302,c1(C(N2C(C)C(NC(c3ncncc3Cl)=O)CC2)=O)cc2n(n1)CCCC2O 58303,N1(C(C2(C(=O)OC)CC2)=O)CC(C2(NC(=O)Cc3ccc(Cl)cc3OC)CC2)C1 58304,CC1CCC(CNC(=O)Cc2ccc(F)nc2)CN1C(c1cncn1C)=O 58305,C1(C(=O)NCCOCCC)CCOC1CNC(=O)C=C(C)C(C)(C)C 58306,CC1(C)CN(C(C23CCC(CC2)OC3)=O)CCC1NC(=O)CCc1cnn[nH]1 58307,CCC(C)CC(C(=O)N(CC(=O)NC)C)NC(c1cc(C)nn1CC)=O 58308,c1(C(=O)NC(CC)CNC(C2CC(O)(C(F)(F)F)C2)=O)cc[n+]([O-])cc1 58309,C1(C(C)NC(=O)C(=O)NCCC(N)=O)CCCN1C(=O)C(F)=CC1CC1 58310,c1(C(=O)NCC2(C(C)(C)O)CN(C(CC)=O)C2)cnc2c(Cl)cccn12 58311,N1(C(C2C(C(C)C)C2)=O)CCN(C(=O)Cc2c(Br)cnn2C)C(CCO)C1 58312,c1(N2CCC(Nc3c(-c4ccccc4)csc3)C2)nnc(C2CC2)n1CCC#N 58313,C12(NC(=O)CCn3cncn3)CCCC1(F)CN(C(C13CCC(F)(CC1)C3)=O)C2 58314,N1(Cc2cc(C)oc2C(F)(F)F)CCOC(CNC(c2nc(C(C)=O)sc2)=O)C1 58315,N1(C(COC2(C)CCOCC2)=O)CC=C(CCNC(C2CCC(=O)O2)=O)CC1 58316,Cc1nc(C(=O)NNC(=O)C(C)C2CCCC2)cn(C)c1=O 58317,c1(C(C(=O)NCCN(C2CCCCC2)C(c2cnc(C)[nH]2)=O)O)ccccc1Cl 58318,C12(C(=O)NC(C)CC3CCN(C(C4(C)CCCC4O)=O)CC3)CCC(CC1)CC2 58319,N1(C(C2CCC(=O)N2)=O)CCCOC(CNc2nccc(-c3ccnn3C)n2)C1 58320,C1(NC(CC2(C)OCCO2)=O)C2CN(C(C3CCCN(CC(F)F)C3)=O)CC12 58321,CC(C)C(O)C(C)C(=O)NCCCC(C)CO 58322,C1(CC(C)(C)C)CN(C(=O)CCC(=O)c2cccs2)CC1NC(=O)COC(F)(F)F 58323,C1(CN(C(C(C2CC2)NC(C(C)n2cncn2)=O)=O)C)COCCO1 58324,c1(C(N(CC(O)CNC(=O)C(O)CC2CC2)C)=O)c(Cl)cc(Cl)c2ncccc12 58325,C1(NC(c2cc(C)sn2)=O)CCC12CCN(C(c1cc(Cl)c(F)cc1Cl)=O)CC2 58326,CC1=NN(C)C(=O)C1CC(N1C2CCC1C(NC(c1cccc(F)c1Cl)=O)C2)=O 58327,C1(CCC(=O)NC2CC(=C)C2)CCCN(C(C2(C3(C)CC3)CC2)=O)C1 58328,c1(C(=O)NC(CNC(C(CC)O)=O)C2CCC2)cc(C)cc([N+](=O)[O-])c1 58329,c12cc[nH]c1C(=O)NC2.C1(C(=O)OC)CC(C(N2CC(N3CC(O)C3)C2)=O)C1 58330,N1(C(CN(C(=O)C(=O)NC(C)(C)C)CC#C)=O)CCC(N(C)C)C1 58331,CC(CCCCNC(=O)CC1C=CCCC1)NC(=O)C1=CCCC1 58332,c1(C(N2CCCC(Br)C2)=O)ccc(NCc2ccncc2Cl)cc1 58333,C1(C(N2CC(CNC(C(COC)C)=O)CC2(C)C)=O)CN2CCCN1CC2 58334,N1(C(c2c(SC)c(Br)ccc2)=O)CC(CC(=O)O)OC2(CCOC2)C1 58335,c1(CCC(=O)N(C2CCN(C(C3CC34CCC4)=O)CC2)C)cccnc1Cl 58336,C1(COC)CCCCN(C(=O)CC(C)CNC(=O)CC(C)O)C1 58337,c1(C(=O)NC(C(C)NC(=O)CNC(=O)NC2CCOCC2)CO)cccnc1O 58338,Cc1ccc(O)c(CNC(C2C=CCN(C(C3(C)CC4(CCC4)C3)=O)C2)=O)c1 58339,C12(C(=O)NCC(C3CC3)SC)CC(C)(CN1C(=O)CCn1ccnn1)C2 58340,N1(C(C=CCC)=O)CCC2(CCCC2NC(c2cnn3c2OCC3)=O)CC1 58341,C1(C(N2C(C)CC(NC(C3C(OC)CCC3)=O)C2)=O)Cc2cccnc2C1 58342,C(=O)(CC(O)C(C)C)NC1CCC(NC(C(CC)N(CC)CC)=O)C1 58343,N1(C(Cc2cc(C)sc2C)=O)CCC(C2CN(C(c3ccns3)=O)C2)CC1 58344,c1(C(CC(=O)OCc2ccc(CCCCCCC)cc2)O)ccc(O)c(O)c1 58345,CC1CCC(NC(c2ccc(CO)c(Cl)c2)=O)CN1C(=O)CCC1CCC1 58346,C(=O)(C(F)C(C)(C)O)NCC1N(C(c2nn(C)c(Br)c2)=O)CC(O)C1 58347,[N-]=[N+]=Nc1ccccc1NC(C1CC2CC1C1CNCC21)=O 58348,c1(CCC)ncoc1C(=O)NCC1CC(CNC(=O)CC(=O)N(C)C)CO1 58349,Cc1cccc(Cl)c1CC(=O)NCC1CCN1C(=O)C1=C(Cl)CC1 58350,Cn1nc(O)cc1C(=O)NCCCc1ncco1 58351,Cc1cnc(C(=O)NC2CCC(C(=O)NCc3ccnn3C)C2)cc1C 58352,c1(C(=O)NC(CNC(C23CCC(=O)N2CCS3)=O)CO)cc(=O)n2nccc2[nH]1 58353,N1(C(C(C)=CC)=O)CCN(C(CNC(c2ccsc2)=O)C(F)F)CC1 58354,c1(C(=O)NCC2C(NC(c3coc(Cl)c3)=O)CCC2)ccc(F)c(Br)c1 58355,C1(NC(c2ccc(OC)o2)=O)CCCC(NC(c2ccnc(C(F)F)c2)=O)CC1 58356,Cc1cc(C(=O)NC(c2cnn(C)c2)C)cc(C)c1O 58357,C(=O)(C1=Cc2ccccc2C1C)NCCN1CCCN(C(C(C)OC)=O)CC1 58358,c1(C(N2CCCN(C(C(CC(C)C)OC)=O)C(C)C2)=O)cccc2cnccc12 58359,CC1CCN(C(c2c[nH]nc2C(F)F)=O)CCN1C(=O)CCc1ccccc1F 58360,Cc1ncc(C=CC(=O)NCC=CCNC(c2cc(F)c(O)c(Cl)c2)=O)c(O)n1 58361,N1(C(c2c(CC)cco2)=O)C2CCC1C(C(=O)NCc1nc(C)co1)C2 58362,CC1(C)CC(CNC(=O)C2=CSCS2)CN1C(=O)COc1ccccc1 58363,Cc1cncc(C(=O)NC(C2CC2C(N2CCOC(CN=[N+]=[N-])C2)=O)C)n1 58364,S(=O)(=O)(c1cnc(Cl)nc1)N1C(C(=O)Nc2c(OC)cccc2)CC(O)C1 58365,C1(N(C(c2cnc(CC)s2)=O)C)CN(C(C2CC2C(C)(F)F)=O)CC1(C)C 58366,c1(C(N2CCC(N(C(C3CCCO3)=O)CC)C2)=O)cc(C)n(C)c(=O)c1 58367,O=C1NCc2cc(C(N3CCOC4(C3)CN(C(C35CCCC3C5)=O)C4)=O)ccc21 58368,c1(NC)cnc(C(=O)NC2CC(CNC(=O)C(S(C)(=O)=O)C3CC3)C2)c(Cl)c1 58369,CCCCC(CC)C(=O)NC1CC(F)(CNC(c2ccc(COC)c(F)c2)=O)C1 58370,c1(NC(CCC)CC)cc(NCCc2scnc2C)nc(C)n1 58371,C1(O)(C(C)NC(C(C)OC)=O)CCN(C(=O)C(F)CC2CC(F)(F)C2)CC1 58372,C1(NC(C(C)OCC#C)=O)CC2(CCCN(C(=O)C(CC(C)C)NC(C)=O)C2)C1 58373,C(=O)(CCCCC1CC1)NC(C1(C(=O)NCc2nnc(C)o2)CC1)C 58374,Cc1cc(=NC(C)C2CCCN(C(C3(N(C)C)CCC3)=O)C2)c([N+](=O)[O-])c(C)[nH]1 58375,CCCC(C(=O)N1CCC(CO)(NC(c2ccc(F)cc2CC)=O)C1)S(N)(=O)=O 58376,C1(C(N(C)Cc2ncn(C)n2)=O)CC12CCN(C(=O)C(CO)N(C)C)C2 58377,c1(OC)c(F)cc(S(=O)(=O)N(C)CC2CCCC2(C)C)cc1[N+](=O)[O-] 58378,CC1(C)CC(O)(CC(N2CCC(CNC(c3cc(O)ncn3)=O)C2)=O)CO1 58379,C(=O)(C(C(C)C)NC(c1cc(CO)oc1C)=O)NCCOCC 58380,C1(C(N2CCC(=CC)C2)=O)CCN(C(=O)Nc2ccccc2O)CC1 58381,CC#CCCC(=O)NC(CNC(c1onc(OC)c1Br)=O)C1CC1 58382,c1(OC)nc(C(=O)NCC2CN(C(c3ncc(C(F)F)s3)=O)C3CC23)sc1C 58383,C12(C(=O)Nc3c(OC)ccc(C)c3)CCCC1CCN2C(C1CCC1C)=O 58384,CCC(CC(C)C)C(=O)NCC1CCN(C(C2CCSCC2)=O)C(C)C1 58385,c1(OC)ccc(C2CC2)c(C(=O)NCC2(CCNC(=O)C3=CCCS3)CC2)c1 58386,C1(C(=O)OC)CC12CN(C(C13CC1CCN3C(c1cc(C)sc1C)=O)=O)C2 58387,C12(C(=O)NCC3CN(C(c4n[nH]c(C)c4Cl)=O)CC3(F)F)CCCCN1CCC2 58388,C(CC(C)C)(C(=O)NC(C)CC(C)O)NC(c1ccc(C)n1C)=O 58389,c1(C(=O)NCC(CN(C(CCOCC)=O)C)C)occc1F 58390,Cn1ccc(=NC(=O)CC(C2CC2)N(C2(F)CCC(=O)CC2)C(=O)OC(C)(C)C)[nH]1 58391,C1(C(N2CC(CC)(CC)C2)=O)CN(C(=O)C=C(C)C(F)F)CC(C)(C)C1 58392,C1(CNC(=O)NC2CC(NC(C3CC=CCC3)=O)C2)CCCCC1N1CCCC1 58393,n1(C(CC)C)nc(-c2cccc(C)c2)nc1-c1csc(N(C)C)n1 58394,C1(F)(CNC(CC2CCC(C)C2)=O)CCN(C(=O)Cc2csc(C(C)C)n2)CC1 58395,c1(C(N(C2CC3CCC(C2)N3C(C2CNC(=O)C2)=O)C)=O)cc(Cl)cc(Cl)c1Cl 58396,C12=CC=C(C=C1)C2C.C1(C(=O)NC(C)C)C2CN(C(C3CCC(=O)N3C)=O)CC12 58397,C1(C(=O)NC(CNC(C=C(C)CN2CCOCC2)=O)(C)CO)CCC(F)(F)C1 58398,c1(C(N2CC(F)CC(NC(C=C(CC)C)=O)C2)=O)cccc2nccn12 58399,C1(C(=O)NC2(CNC(CC3C(C)C3)=O)CCCCCC2)CCn2cnnc2C1 58400,N1(C(CC2N(C(c3n(C)ccc3)=O)CCC2)=O)CCC2(CNC(=O)N2)C1 58401,N1(C(C(COCC)C)=O)CCC2(CCC(CNC(c3ccc(C)n3C)=O)O2)CC1 58402,C1(C)(CNC(C2(F)CN(C(c3c(C)scn3)=O)C2)=O)CCCC1O 58403,Cc1ccc(Cl)cc1NNC(=O)NCC1COc2ccccc2O1 58404,c1(C(=O)NCCC(=C)CNC(=O)C(C)S(N)(=O)=O)cnc2sc(C)nc2c1 58405,C(CCCC(C)NC(c1ccc(C2CCCO2)[nH]1)=O)NC(C1(C)CC(C)C1)=O 58406,c1(C(N2CCN(C(=O)OC(C)(C)C)CC2)=O)cc(Br)c(N)cc1[N+](=O)[O-] 58407,c1(C(=O)NCCCN(C(c2cccc(C)c2C)=O)C(C)C)ccc2nc[nH]c2n1 58408,N1(C(c2ccc(CO)o2)=O)CCC2(CC(C(=O)NCc3ccsc3)C2)C1 58409,C(c1ccc2c(c1)OCCO2)=CC(=O)OC(c1ncc(C)[nH]1)C1CC1 58410,C(CC(C(C)(C)C)NC(=O)CSS(C)(=O)=O)N(C)C(C1CN(C)CCN1C)=O 58411,C1(CNC(C(N2CCOCC2)C)=O)CN(C(C23CC2COC3(C)C)=O)CCCO1 58412,Cc1noc(C)c1S(=O)(=O)N(C1CC2CC1CN2)C(C)CO 58413,C(=O)(CCC(CF)CF)N(C(C)CNC(C1CCOC1)=O)C 58414,CC(CC(F)(F)F)C(=O)N1CCCCC(N(C)C(c2snnc2C2CCC2)=O)C1 58415,c1(C(c2nnnn2C)C2(c3ccc(OC)c(OC)c3)CC2)c(N)cccc1F.CN 58416,CC(C)CC(O)C(=O)N1CC(CNC(C23CC(C2)C(C)O3)=O)C1 58417,c1(NC(C2N(Cc3cc(C)cc(C)c3)CCOC2)=O)csc2nccnc12 58418,N1(C(C2CCCOC2)=O)CCC2C(CCCN2C(c2ncoc2Br)=O)C1 58419,C12(NC(C3CC3C(F)(F)F)=O)CCC(C(N3CCC(CC4CC4)C3)=O)(CC1)C2 58420,c1(N2CCC(C)(COC)C2)nc(N2CCC(F)(CF)C2)c2ccc(C)cc2n1 58421,c1(C(=O)NCC(=C)C)cnc2ccc(-c3cc(OC)cc(C)c3)cc2c1Cl 58422,Cc1ccc([N+](=O)[O-])cc1C(=O)NCC1CN(C(=O)CCOCC(F)F)CC1O 58423,C1(NC(CC(=O)OCC)=O)CCN(C2CCN(C(=O)CSC(F)(F)F)C2)CC1 58424,CC1CN(C(c2ccnc(Cl)c2)=O)CC1NC(c1cc(O)no1)=O 58425,N1(C(C(CC)(C)CO)=O)CC2(CC(NC(c3ncccc3Br)=O)CO2)C1 58426,N1(C(COC)=O)CCC(F)(F)C(CNC(c2cnccc2C(C)(C)C)=O)C1 58427,N1(C(CC(=O)NCC#C)=O)CCC(F)(C(N2CCCC(C(C)C)CC2)=O)CC1 58428,C(C(=O)N1CCCCO1)(c1cn(C)nn1)NC(C(OCC)OCC)=O 58429,c1(C(N2C(C(N(C(C3CCOCC3)C)C)=O)CCC2)=O)ccc2c(ccn2C)c1 58430,N#Cc1ccc(C(F)(F)F)c(N2CCC(CCC#N)CC2)c1 58431,Cc1c(C(=O)NC(CO)C(=O)NCC(c2cnn(C)c2)C)cccc1C#N 58432,C(C(=O)Nn1cnn(C)c1=S)C1CC(C)N(C(c2cncn2C)=O)C1 58433,CC(CNC(c1n[nH]c(=N)[nH]1)=O)CC(=O)N(C(C)C(C)(C)O)C 58434,N1(C(c2c(COC)cco2)=O)CCC(C)C1CNC(=O)CCOc1ccccc1 58435,C1(C)(OCC(=O)Nc2conc2C2CCC2)CCOCC1.CN1CCNC1=O 58436,c1(C(N2CCC(n3cccn3)C2)C(=O)NC(C)C)cc(F)cc(F)c1Br 58437,C1(NC(c2c(CC)nns2)=O)CC(CNC(=O)CCc2c[nH]c(=N)[nH]2)C12CCC2 58438,C1(n2cc(CCCC(C)O)nn2)CCCCN(C)C1=O.C12(C)CCCN1c1nnnn12 58439,N1(C(COCCC(C)C)=O)CCCCC(NC(=O)CCCC(C)O)C1 58440,N1(C(c2cc(C)n(C)n2)=O)CCC(C)C(NC(c2csc(C3CCCO3)n2)=O)C1 58441,Cc1cc(C(=O)NC2CCN(C(C3CC3C3(C)COC3)=O)C2)cc2c1CCC2 58442,CCC(C(F)(F)F)NCC1CC(CC)(CC)CO1 58443,C(c1cccc(Cl)c1Cl)=CC(=O)NCCC(C)NC(=O)CC1NC(=O)NC1=O 58444,CC(C)C(C)(CNC(c1nscc1Br)=O)NC(C1C=CCC1)=O 58445,c1(C(N2CC3CC(NC(C4(O)CC(C)(C)C4)=O)C3C2)=O)cncc2ccsc12 58446,CC(C)(C)C#CC(=O)N1CC(NC(C2CS(=O)(=O)C2)=O)C(c2ccc(F)cc2)C1 58447,c1(OC)ccc2cccnc2c1C(=O)NC1CCC2(CCN(C(C)=O)CC2)C1 58448,N1(C(c2c(CCC)n[nH]c2)=O)CCCCC(C(=O)NCCC(CCC)C2CC2)C1 58449,c1(C(C2C=C(C)CCC2)NC(=O)CN(C)C)ccccc1[N+](=O)[O-] 58450,c1(C(=O)NC(C#C)Cc2ccccc2)nc(S(C)(=O)=O)ccc1Cl 58451,Cn1cnnc1CNC(c1n[nH]cc1CNC(C1(F)CCOC1)=O)=O 58452,CC1OC(C)C(C(=O)NCC2(C)CCCN2C(c2ccc(C(N)=O)s2)=O)C1C 58453,C1(NC(C(c2n(C)cnc2)O)=O)CCN(C(=O)CCN2CCCC2=O)CC1 58454,N1(C(C(C)OCC2CC2)=O)CC2(CCC2NC(c2cc(C(C)(C)C)nn2C)=O)C1 58455,CC(O)CCCNC(=O)CCNC(C1(C(C)(F)F)CC1)=O 58456,CC(C)(O)C(F)(F)C(=O)N1CC(C(N)=O)(CNC(C2CCCC(C(F)(F)F)C2)=O)C1 58457,C1(CN(C(C(C)CF)=O)C)CCCN(C(=O)CN2CSCC2=O)C1 58458,c1(C(=O)NC2C(CC)CN(C(c3cnn(C)c3N)=O)C2)cc(SC)cc(Cl)c1 58459,C1(NC(Cc2cc(C)no2)=O)CC2C1CCN2C(C1CC2CCCCC12)=O 58460,N1(C(C(=O)NC(Cc2cccc(C)c2)C)=O)CCC2(CCO2)CC1 58461,CCC(F)(F)C(C)(C)C(=O)N1CCN(C(c2ccc(CO)o2)=O)CC1C 58462,C1(C(C)C)CCOCCN1C(=O)COC1(C)CN(C(=O)C(C)Cn2ccnc2)C1 58463,c1(OC)ccc(C(N2CC(CO)(NC(=O)CC(=O)N(C)C)C2)=O)cc1S(C)(=O)=O 58464,CN1CCN(C(=O)C(C)(C)CC2CCC2)CC1CNC(C1Cc2nccn2C1)=O 58465,NS(=O)(=O)c1nc(C(N2CCC(NC(=O)CCF)C(CO)C2)=O)n2ccccc12 58466,CN1C(=O)c2ccccc2C1C(=O)N1CCCCC1CCNC(C1CC1(C)C)=O 58467,CC#CCCCC(=O)NCCCC1(C)CN(C)CCO1.C1CCC(C#N)CC1 58468,O=C1Cc2ccc(CC(N3CCCC3c3c(F)cccc3Cl)=O)cc2N1 58469,S(=O)(=O)(c1cccc(C(=O)O)c1)N1C(C(=O)NCCC#CC)CCC1C 58470,N1(c2cc(CC)ncn2)CCCC(CO)(NC(=O)C=Cc2ccc(C)o2)C1 58471,C1(NC(C(C)(N(C(=O)CSCC(F)F)C)C2CC2)=O)CCOC(C)(C)C1 58472,c1(C(N(C2CN(C(C(F)OC)=O)C2)C)=O)n[nH]c(C)c1C 58473,N1(C(COCCSC)=O)CCCC1CC(=O)NCCC12CC(CO1)C2.O 58474,N1(C(COCCOC)=O)CC2C3CCC(C2C1)N(C(C1CCC(C)S1)=O)C3 58475,CON1CCC(C(N2CC(NC(C3CCN(C)C(C)C3)=O)CC(F)C2)=O)CC1 58476,C12(NC(C(CSC)OC)=O)CCC(CN(C(c3cc(CO)on3)=O)C1)C2 58477,c1(-n2cc(CC3(O)CN(C(C(C)NC(C4CCC4)=O)=O)C3)nn2)ccc(Cl)cc1 58478,N1(CC=C(C)C)CCCC(C(=O)NC(CC2CC2)CO)C1 58479,c1(NC(CC(C)c2cnn(C)c2)=O)ccc2c(=O)n(C3CCCC3)sc2c1 58480,c1(OC)cc(C(=O)NC2CCCCC2NC(=O)C2=CCCO2)c2c(c1)CCO2 58481,c1(C(=O)OCC(=O)N(C2CCOC2=O)C)coc2cccc(F)c12 58482,N1(C(C=CC(C)(C)SC)=O)CC=CC(C(=O)N(C)Cc2sccc2C)C1 58483,C(=O)(C(COC)CC)NCC1N(C(CCOCC)=O)CC1 58484,c1(OCC)cncc(C(=O)NC2(CN(C)C(c3cc(C#N)c[nH]3)=O)CC2)c1 58485,C(C)(CCC(=O)NC1CCC1C(=O)NCC(O)Cn1cccn1)OC 58486,C(=O)(CC(COC)COC)N1CC(O)(C(C(=O)NCCS(CC)(=O)=O)F)C1 58487,n1(C(CC)C)ncc(C(=O)N(CCCN(C)C(c2snnc2C2CC2)=O)C)c1C 58488,N1(C(c2c(OC)nsc2OC)=O)CCC(C)C(NC(C2CSCCS2)=O)C1 58489,CC(C)(CF)C(=O)NC1CCCCC1NC(=O)CSCc1ccncc1 58490,CCC(CN(C)C)CC(=O)NC1CN(C(c2cc(C(C)=O)on2)=O)C(C)(C)C1 58491,c1(C(=O)NC2CC(NC(c3ncncc3Cl)=O)C23CCC3)cccc2sccc12 58492,N1(C(C2CCC(N(C)C)C2)=O)CCC(NC(=O)C#CC2(C(F)(F)F)CC2)C1(C)C 58493,N1(C(C2(C)CS(=O)(=O)C2)=O)CC(CNC(c2ccc(F)s2)=O)C2(CC2)C1 58494,C1(CC)CC(O)CN1C(c1ccc(OCCO)cc1)C(=O)Nc1ccccc1C 58495,N1(C(c2c(C)nc(C)o2)=O)CC2CCN(C(c3cnc4scc(C)n34)=O)C(C2)C1 58496,c1(C(=O)NC2C(C)CN(C(C3(C)CCC3)=O)CC2)cnc2[nH]ccc2n1 58497,N1(C(CC(C)(C)C)=O)C2CCC1C1CC1(NC(C1CC3CCC1O3)=O)C2 58498,C1(CNC(CCOC)=O)CN(C(=O)CCNC(=O)CC(C)C)CC(C)(C)C1 58499,C1(C(N2CCC(O)(CCNC(C3CC3(F)F)=O)C2)=O)CC(C2CC2)=NO1 58500,C=CC(CCC)CC(=O)N1CC(C(O)C(=O)NC(C2CC2C(=O)OC)C)C1 58501,C1(C(N(C)CC2(CO)CCC2)=O)(NC(=O)Cc2csnn2)CC(F)(F)C1 58502,C(=O)(C#CC1(C)CC1)NCC1(OC)CCN(C(c2ccc(CN(C)C)o2)=O)C1 58503,Cc1cc(C(=O)NCC2CCC(NC(C3CC4CCCC34)=O)C2)c(N)c(F)c1 58504,Cc1ccc(C)c(C(=O)NCC(C2CCN(C(c3ccn(C)n3)=O)CC2)C)c1 58505,c1(OC(C)(C)C)cccn2ncnc12.N12CCCC1c1ocnc1CNC2=O 58506,C1(C(N2CC(CCC#C)C2)=O)CC(NC(=O)Cn2ncnn2)CCO1 58507,C(=O)(C(C(C)C)C(C)C)NC1CC(CNC(C(C(C)(C)C)NC(C)=O)=O)C1 58508,c1(CO)ccc(NCC2(c3cccc(Cl)c3)CCC2)c([N+](=O)[O-])c1 58509,c1(-c2cccc(C)c2C)cc(C(N2CCC(CO)C(F)(F)C2)=O)cc2[nH]ncc12 58510,N1(C(C(CCCCCC)F)=O)CCOC2(CCCN(C(=O)CCC3CC3)C2)C1 58511,CN=c1nc(C(N2CCCC(O)(CNC(C3CC3Br)=O)C2)=O)cc(C)[nH]1 58512,c1(C(=O)NCCNC(=O)Cc2sccc2Br)c(F)cccc1[N+](=O)[O-] 58513,C1(C(N(C)CC2CC(=C)C2)=O)CC2CCC1N2C(=O)Cn1nnc(C)n1 58514,c1(C(=O)NC(C)CN(C)C(c2ncc(F)cc2F)=O)cc(F)cc(Br)c1F 58515,c1(CNC(C)Cc2ccco2)cc(Br)c(F)cn1 58516,C(=O)(CS(=O)(=O)CC(=O)NCC1CC(O)CN1C(=O)C(c1ccc(C)s1)C)OC 58517,C1(CN(C(C(OC)OC)=O)C)CCN(C(C2(Br)CC2)=O)C1 58518,C1(NC(C(N2CCCCCC2)C)=O)CCN(c2ccncc2C#N)CC1O 58519,C1(C(=O)NCC2(C(C)NC(c3ccc(N)cn3)=O)CC2)(CC)CNC(=O)C1 58520,C1(C(=O)NC(CNC(CC(CC)C2CCC2)=O)(C)C2CCC2)CC(=O)NC(=O)C1 58521,Cc1cc(O)ccc1CC(=O)NCC1COC(CNC(C2CC(C)(C)CO2)=O)C1 58522,c1(CC)nn(C)c(Cl)c1C(N1CC(CNC(=O)C(C)(O)C2CCC2)C(C)(C)C1)=O 58523,CCCCCCC(CC)NC(C1CC(CCNC(=O)CC(C)n2cccc2)C1)=O 58524,Cc1cc(C(N2CCC(C3CC3)C2CNC(=O)CC(C)(C)O)=O)cc2nc[nH]c12 58525,C=CCCC(C(=O)N(CC(=O)NC)CC)NC(c1ccc(C)cn1)=O 58526,N1(CC(CN)(C)C)CCN(C)CC1.Cc1cc(C(c2nnnn2C)NC2(C)CC2)cs1 58527,c1(C(N(C(CCNC(c2cccc(CC)c2)=O)C)C)=O)cc(C)cc(C)c1O 58528,C1(C(N(C2CN(C(C3CCN(C)CC3)=O)C2)C)=O)CCc2nn[nH]c2C1 58529,c1(C(=O)NCCNC(c2c(C(N)=O)cccc2)=O)cnc2nccn2c1 58530,c1(C(=O)NC2CC(CNC(CCC3CC(C)C3)=O)CC2O)ccc(F)cc1C#N 58531,C1(N(C(=O)CN2C(=O)CNC2=O)C)CCCN(C(c2cc(=O)n(C)cn2)=O)CC1 58532,c1(C(N2CC(CNC(c3nc(CC)oc3)=O)C3C2C3)=O)cc(C)ccc1[N+](=O)[O-] 58533,c1(C(N2CCC(NC(C=CCN(C)CC)=O)C2)=O)cncc2c[nH]nc12 58534,N1(C(c2cocn2)=O)CCCCC1CCC1CCCN1C(C1CC=CC(O)C1)=O 58535,N1(c2nc(OC)c(F)c(C)n2)CCC2(CC1)OCCC2NC(=O)C1=C(C)OCC1 58536,C1(C(N(C2CC(NC(CCSC)=O)C2)C)=O)CCOCC1C 58537,c1(OCC)c(F)c(C(=O)NC2CC(NCc3cc(Cl)ccc3O)C2)cc(F)c1F 58538,N1(C(CC(C)(C)O)=O)CCN(C(=O)CCc2nccs2)C(CO)C1 58539,c1(CCC(N2C(CN(C(C(C)SC(F)(F)F)=O)C)CCC2)=O)ccccc1Cl 58540,n1(CC(N2CC(C)(CNC(c3c(OC)nn(C)c3)=O)C2)=O)cc(C)c(O)nc1=O 58541,c1(CC(=O)NC2C(NC(c3n(CC)c(O)nc3)=O)CCC2)n[nH]c2c1CCCC2 58542,c1(OC)cc(C(=O)NC2CC3(C2)CC(NC(=O)C(C)CS(C)=O)C3)ccc1C 58543,C1(CN(C(Cc2c(C)nc[nH]2)=O)C)CCN(C(c2ncc(Br)cn2)=O)CC1 58544,C1(NC(CC=C)=O)CCC(CCNC(c2cn(C(C)C)nn2)=O)C1 58545,C1(C(=O)NCC(=O)NCC)CCC(O)CN1C(c1cn(CC)nc1C)=O 58546,N1(C(C(CC)NC(N)=O)=O)CCC(COC)(NC(c2nccc(C)n2)=O)C1 58547,N(C(=NCCCNS(C)(=O)=O)NC1CCC12CCCCC2)CCN(C)C(=O)NC.CO 58548,C1(CC=C)(NC(C2C=CCC2)=O)CCN(C(c2ccc(C(N)=O)cn2)=O)C1 58549,c1(C(N2CCC(C(C)(C)C)(CNC(C3N(CC)CC3)=O)C2)=O)sc(C)c(C)c1C 58550,N1(CC2CN(C(C=CC=CCC)=O)C2)CCN(C(c2cnsn2)=O)CC1 58551,C1(NC(C(C)OC)=O)COC2(C1)CN(C(c1cc(C)c(C)nc1C)=O)C2 58552,N1(C(C=CC=CC)=O)CCCCC1CCN(C)C(c1ccnn1CCC)=O 58553,c1(-n2ncc(C(=O)NCCNC(C3(C)CC3C(F)(F)F)=O)c2)cccc(O)c1 58554,n1(CC)ncc(Cl)c1C(=O)NCC(C)CNC(=O)Cc1cc(C)[nH]n1 58555,C1(N(C(CNS(NC)(=O)=O)=O)C)CCN(C(=O)CC2CCCCN2C(C)=O)CC1 58556,C1(C(=O)NCC(CNC(c2cc(O)ccc2F)=O)O)CCC2(CCC2)O1 58557,C(C(F)(F)C(=O)NC(c1ccccc1F)CNC(C1CS(=O)(=O)C1)=O)N(C)C 58558,N1(C(CCC)=O)CCC(C)(C(=O)NCc2ccsc2)C1 58559,C1(C(N2CC(C(C)OC)C2)=O)CCC=CC1NC(C1CCCN(C)C1)=O 58560,n1(-c2c(C(=O)NCCN(C)C(C3(C)C=CCC3)=O)cccc2)ccc([N+](=O)[O-])n1 58561,c1(NC(NOCCC#C)=O)ccc(OCCc2ccccc2)cc1 58562,Cc1ccnc(C(C)NC(=O)N(C2CC2c2ccccc2)CCN2CCCCC2)n1 58563,c1(C(C)NC(=O)CC2CSC2)nocc1C(=O)NCC1CCC(C)C1 58564,C=CCN(CC=C)N1CCC(CC(=O)N(CCCO)C)CC1 58565,CC(C)(C#Cc1cn(Cc2cscn2)nn1)NC(C1CCN2CCCC12)=O 58566,C#CCCC(O)C(=O)NCCC1CCN(C(C2CCS(=O)(=O)N2)=O)CC1 58567,Cc1nc(NCCS(=O)C(C)(C)C)cc(NCCCc2ncco2)n1 58568,C#CC1(O)CCN(C(C2CC(C)CN(C(C3(C#C)CC3)=O)C2)=O)CC1 58569,C1(C#CC(=O)NC2CCOCC2NC(=O)C(=O)NCCSC)(CC)CC1 58570,Cc1ncn2ccc(C(N3CC(CNC(=O)C=C4CCCC4)C4(CC4)C3)=O)cc12 58571,c1(C(N2CC3(CC(CNC(COCC)=O)C3)C2)=O)cc(C)cc(Br)c1F 58572,CC(CC(=O)NC1(C)CCCN(C(c2cccc3cnsc23)=O)C1)CC(C)(C)C 58573,CCCN=C(NCCCOCCS(C)(=O)=O)NCc1ccccc1.C1(C)(O)CCCC1 58574,n1(CCC)nc(C)cc1C(=O)NCC1CC(NC(C2(F)CC=CCC2)=O)C1 58575,C(CC(C)(C)C(=O)NCC1(F)CCN(C(C2(C)CC(C#N)C2)=O)CC1)OC 58576,c1(NC(CC2(N(C(c3c(CC)onc3C)=O)C)CC2)=O)ccc(=O)n(CC)c1 58577,C(=O)(CCC(C)(C)NC(=O)C1=COCCC1)NCCc1nc(C)sc1 58578,C(=O)(C(C)CN(C(=O)C(C1CCOCC1)O)C)NC(COC)CO 58579,C(=O)(C(C)CC(F)F)NC(CC)(CNC(=O)CCOCCCOC)CC 58580,c1(C(C)=O)cc(C(=O)N(C(C)CCNC(=O)C#CC(=O)N(C)C)C)oc1C 58581,c1(C(C(=O)NCC(O)CNC(C2(O)CCC2)=O)N(C)C)c(F)cccc1Cl 58582,C1(C(N(C2CCN(CC)CC2)C)=O)CC(C)CN(C(=O)CN2CC=CC2)C1 58583,N1(C(C(C)OCCCC)=O)CC2CCC2(CNC(=O)C=Cc2cnc(C)s2)C1 58584,c1(CC(=O)NCC(CC)NC(=O)COCC2CCC2)cn(C)nc1C 58585,C1(COC)(CNC(=O)C=Cc2ccnn2C)CCN(C(=O)CCF)CC1 58586,c1(C(N2C(C(N(CC(F)(F)F)C)=O)CC(F)(F)C2)=O)cc2ccc(Br)cc2s1 58587,N1(C(CC=C=C)=O)CCC2(NC(=O)CCc3ccc(OCC)cc3)CCCC12 58588,C=CC1(CC(=O)NCCNC(c2ccoc2)=O)CN(C(=O)CC2CC3C=CC2C3)C1 58589,C=CCC(CC(C)C)C(=O)N(C1CCN(C(C2CC3(CC(OC)C3)C2)=O)C1)C 58590,C1(CNC(C2(C#N)CC(C)C2)=O)CCN(C(c2cnnc(Cl)c2)=O)C1(C)C 58591,C(=O)(C(F)(F)CCn1ccnn1)N1CC(OCCNC(c2ccnc(OC)n2)=O)C1 58592,C=CC1(CO)CCN(C(c2cnc3c(c2)CCC3)=O)CC1 58593,Cc1cc(OCC(=O)NCC(CO)NC(c2coc(C3CC3)n2)=O)cc(C)c1Cl 58594,C#Cc1ccc(OCC(=O)NCCN(CCC)C(c2conc2CC)=O)cc1 58595,Cc1cc(C(N2CCN(C3CC3)CC2C)C(=O)NCCC2(C)CC2)cnc1C 58596,C(=O)(C(C)CNC(c1cnc(O)o1)=O)N(CCC)C1CC1 58597,n1(CC)ncc(Cl)c1C(=O)NC1CC1CNC(C1(O)CC(F)(F)C1)=O 58598,c1(OC)cc(C(=O)NC2CCCCC2NC(=O)CCC2CC2C)cc(C)n1 58599,C1(C(=O)NCC(CO)C(F)(F)F)CC2CCC(C1)N2C(C1(F)CCCCC1)=O 58600,N1(C(C2(C)CC2Br)=O)CCc2nc[nH]c2C12CCN(C(C1CCCCS1)=O)C2 58601,c1(C(=O)NC(CC)CN(C(=O)C(C)C2=CCCC2)C)oc2ccc(C)cc2c1C 58602,c1(C(=O)NCCCN(CCCNC(C2CC(O)C2)=O)C)n[nH]c2c1CCCC2 58603,CC1CCC=C1C(=O)N1CCCCC1CCNC(=O)C(=Cc1cn(C)cn1)F 58604,CC1CN(C(C(=O)NCCN2CCOCC2)C(C)CC2CC(F)(F)C2)CC(=O)N1 58605,c1(C(=O)NC)ccc(CC(=O)NC(CNC(=O)C(O)CN(C)C)C2CCC2)cc1 58606,C12(c3cn(CC(CC)C)nn3)COC(CN1C(c1nocc1Br)=O)C2 58607,c1(C(N(C2CN(C(=O)CCCN3C(=O)CNC3=O)C2)C)=O)n[nH]c2ccccc12 58608,N1(C(CC(C(C)OC)NC(C(C)OCCOC)=O)=O)CCCC(O)(C2CC2)C1 58609,c1(C(=O)NCCOCCNC(CS(CC)(=O)=O)=O)cc2sc(=O)n(C)c2s1 58610,C12(CCC)CCCN1C2=O.C1(c2ccccc2)(C(=O)OC)CC(F)(F)C1 58611,Cc1ccc(Cl)c(O)c1C(=O)NC1CCN(C(=O)CC(F)(F)F)CC1C 58612,C(C)(CNC(C1CC(=O)N(c2ccc(C)cc2)C1)=O)(C(C)C)NC(CCSC)=O 58613,C(=O)(C(C(C)(C)C)NC(=O)OC)N1CCC(F)(CNC(c2cn(CC)nc2)=O)C1 58614,CC1(C)OCC2CC12NC(C1(NC(c2cc(Cl)n[nH]2)=O)CC(F)(F)C1)=O 58615,C1(C(=O)O)(CCCCNC(CCNC(CCOCCOCC)=O)=O)CCCC1.OC 58616,CC(C)CC(C)CC(=O)NC1CCN(C(=O)CCc2cnc[nH]2)CC1 58617,c1(C(=O)OC)ccc(CNC2CC2C(=O)NC(C)CC#N)c(Br)c1 58618,c1(OC)ccc(C(c2nnnn2C(C)(C)C)NCC2CC(C)C2)cc1OC 58619,Cc1ccc(O)c(C)c1NC(C1CCC(CNC(=O)COCC2CC2)C1)=O 58620,c1(C(N(CCNC(=O)CC2CN(C)CC2O)CC)=O)ccc2c(c1)OC(C)(C)C2 58621,N1(Cc2c(C(=O)OC)c(C)sc2)CC2CS(=O)(=O)CC2(C#N)C1 58622,CNS(=O)(=O)NCC(=O)N(C1CN(C(=O)Cn2nnc(-c3cccs3)n2)C1)C 58623,C12(C(=O)NCCC(C)N(C(C(CC)C)=O)C)CCC(CC1)C(C)O2 58624,C1(NC(c2cccc(OCCF)c2)=O)CCN(C(c2ccoc2)=O)CC(O)C1 58625,N1(C(C(F)=CC)=O)CC(NC(=O)CCC(=O)c2ccncc2)C2CC12 58626,C(=O)(C(C)(CC1CCC1)OC)NC(CN(C(c1cc(CCC)[nH]n1)=O)C)C 58627,CC1(C)C2CCC1(CC(N1CC(CNC(C3SCCCS3)=O)C1)=O)CC2 58628,CC(C(=O)N(C)CC1CCN(C(C2CCCC2)=O)C1)C(C)(F)F 58629,CCCC(C(=O)OCC)N1CCN(C(=O)C(C2CCCCC2)N)CC1 58630,C1(NC(C2N(CCC)CCC2)=O)CC2CCC1(NC(c1cnn(CC)c1Cl)=O)C2 58631,c1(CN2CC(CC(=O)NC(C(=O)OCC)CO)C2)ncc(Br)cc1F 58632,c1(C(=O)Nc2cncc(Cl)n2)ccc(=O)n2c1COCC2 58633,C1(C)(CNC(C(CN(C)C)O)=O)CN(C(=O)C(C)(C)NS(C)(=O)=O)CCO1 58634,C=C(Cl)CC(C(=O)N1CC(CO)C2(CC2)C1)NC(c1cc[nH]c1)=O 58635,N1(C(CC2(C)CCCO2)=O)CCN(C(c2cc(Br)cnc2O)=O)CC2(CC2)C1 58636,C(=O)(C1=CCN(C(c2cn(C)c(=O)cn2)=O)C1)NC1CC2CC(OC)C2C1 58637,N1(C(CN(CCOC)C)=O)CCCC2CN(C(=O)C(CCSC)N(C)C)CCC12 58638,c1(C(C(=O)NCCN(C(=O)CCc2cnoc2)CC(C)O)O)ccc(Cl)cc1 58639,C1(CCSC)(COC)CCCN1C(=O)CNC(C)=O.C12CC(CN1C)CNC2=O 58640,N1(C(C=Cc2cnc(C)s2)=O)CC2OCCN(C(=O)COCCCN(C)C)C2C1 58641,c1(CC)nn(C2CC2)cc1C(=O)NCCNC(c1cncnc1)=O 58642,c1(OCC)ccc(C(=O)NC(CNC(c2cscc2CC)=O)CO)cc1C 58643,Cc1nc2ccccc2cc1C(=O)N(C1CCCC(N(C)C(C2COC2)=O)C1)C 58644,N1(C(C2(CS(C)(=O)=O)CCC2)=O)CC2CCC2(NC(C2COCCC2(F)F)=O)C1 58645,C=C(C)CCCC(=O)NC(C)C(C)NC(c1ccn(C(CC)CC)n1)=O 58646,Cc1ccc(C(=O)NCCC2(O)CCCN(C(c3nnc(S)n3C)=O)C2)c(N)n1 58647,N1(C(C(CCC)C)=O)CC(CO)C2(C1)CN(C(C1(S(N)(=O)=O)CCC1)=O)C2 58648,C1(C(N2CCC(COC)(CNC(c3cnc(O)o3)=O)C2)=O)CCC(C)=C(C)C1 58649,C(CCC(C)(C)C(=O)N1CCC(O)(C=C)C1)NC(c1ccc(C#C)o1)=O 58650,C1(c2nnnn2C2CCC2)(NC(c2ccc3c(c2)OCO3)C)CCCC(C2CC2)C1 58651,c1(C(=O)NC2CC3(C(NC(c4occ(C)c4)=O)C3)C2)ccc2c(c1)C(=O)CCC2 58652,CCC(CCC(=O)N1CCC(n2cccn2)C1)NC(c1cnnc(O)c1)=O 58653,N1(C(CCCC2C(C)C2)=O)C(C(=O)NC(C)(CO)C(C)(C)O)CCC12CC2 58654,C1(NC(C2(C(=O)NC)CC2)=O)CCCN(C(c2ccnc(C(C)C)n2)=O)C1C 58655,C=CC1CN(C(C2CC(OC)C2)=O)CC1NC(=O)C(C1CCCCCC1)C 58656,CC1(C)C=C(C(=O)NC2CCC(NC(C3(F)CCCCCC3)=O)CC2)C1 58657,C1(NC(=NCCC)NCC(c2ccccc2F)OC)CCc2cnn(CC)c2C1 58658,C(C)(c1ccc2ccccc2n1)=Cc1cc(C#N)cs1.CC=C 58659,C1(CNC(c2cn(CC=C)nn2)=O)CN(C(=O)C=CC(=O)NC2CC2)CCC1C 58660,C#CC1(C)CCCN(C(c2coc(CNC(C3CC3(F)Cl)=O)n2)=O)C1 58661,N1(C(C2(CCCC)CC2)=O)CCC2C(CCN2C(C2C=CCS2)=O)C1 58662,C1(C(N(C2CCN(C(c3cccc(O)n3)=O)CC2)C)=O)C2CCCOC12 58663,C=C(Br)CC(C)(C)C(=O)NCCC1CCC(NC(C2(OC)CC2)=O)C1 58664,C12(NC(=O)CC3CCC(O)C3)CC(C1)N(C(c1cccc(-c3cc[nH]n3)c1)=O)C2 58665,C(=O)(C1Cc2ccc(F)cc21)NCC1CC(N)(CC)C1 58666,C=CC(C)(CCOC)C(=O)NCC(C(=O)NCC(C)(C)CN=[N+]=[N-])OC 58667,N1(C(c2c(F)ccc(OC)n2)=O)CCCCCC(NC(c2cncc(F)c2)=O)C1 58668,c1(C(=O)Nc2ccc(C(=O)NCc3n(C)ccc3)cn2)c(F)cc(O)cc1F 58669,c1(NC(=O)NCC(C(C)O)C)nc2c(s1)C(=O)NCC(C)(C)C2 58670,Cc1nccn1CCCNC(c1nnnn1C1CCCC1)(CCCCO)C 58671,C12(CNC(=O)C(O)CC3CC3)CN(C(=O)Cn3cnnn3)CC1CCO2 58672,c1(C(=O)NCC(c2ccccc2)CNC(CC=C)=O)ccc2c(c1)C(=O)NC2=O 58673,N1(C(C(C)CO)=O)CCCC2(NC(C3(CN(C)C)CC3)=O)CC2C1 58674,FCCCN=C(NCC1(c2ccc(Cl)cc2)CC1)NCC1CC=CCC1 58675,C(=O)(C(C)C(C)NC(C1CN(C(c2cn(CCO)nn2)=O)CC1C)=O)OC 58676,C1(C(=O)NCC(=C)C(F)(F)F)CC(NC(=O)CCC#CC)C12CCC2 58677,c1(C(N(CC(CNC(c2c(C)coc2C2CC2)=O)C)C)=O)ccc2c(c1)CCN2 58678,c1(C(=O)NCCC(=O)N2CC(OCC(=O)NCC3CC3)C2)ncncc1Cl 58679,Cc1oc(CNC(C2CCCC(F)C2)=O)nc1C(=O)NC(c1ccc(O)cc1)C 58680,CC1(NC(C2CCNC(=O)C2)=O)CCCN(C(c2cnc3n2CCS3)=O)C1 58681,Cc1nc(N(C)CC2CCCN(C(c3ccco3)=O)C2)cc2nncn12 58682,C1(CC(=O)N(CC=C)CCO)(OC)CN(C(=O)CCc2nc(C)no2)C1 58683,c1(CC(=O)N(C(CN(C(C=CCC)=O)C)C)C)cccc(OC(C)C)c1 58684,C(=O)(CCCS(C)(=O)=O)NCCOC(C)(C)CNC(c1cc(C2CCC2)no1)=O 58685,N1(C(C=CCOC)=O)CC2C(CN(C)C(c3ccc(CC(C)(C)C)cc3)=O)C2C1 58686,C12(NC(C3C(CNC(COC(C)=O)=O)C3)=O)CC1COC2(C)C 58687,c1(C(=O)NC2C(C(=O)NC(CCCCC)C)OCC2)cc(C#N)n(C)n1 58688,NS(=O)(=O)c1cncc(C(=O)NC2CCCN(C(=O)C=C3CCCC3)C2)c1 58689,CC(CCCNC(=O)CNC(=O)C(C)(C)F)NC(=O)NCc1ccccc1 58690,C1(C(=O)NC(C=C)C)CCC(NC(c2csnn2)=O)CO1 58691,c1(C(N2CCOCC(CNC(C3(C)CCCCC3)=O)C2)=O)ccc(Cl)c(N)c1Cl 58692,N1(C(CC=CC)=O)CCCC(N(C(=O)C(=Cc2ccccc2)C)CCO)C1 58693,c1(C(=O)NC(CN(C(CS(=O)(=O)NCC)=O)C)(C)C)ccn2nccc2n1 58694,Cn1ncc(C#N)c1CNC(N1CCN(CCO)C(=O)C1)=O 58695,c1(C(N2CC(O)CC(NC(CSCC)=O)C2)=O)c(F)ccc(OC)c1OC 58696,N1(C(c2ncn(CC)c2)=O)CCCN(C(C2(C)CC2(C)C)=O)CC1C(C)C 58697,C12(NC(=O)C3=COCCC3)CCCCCC1N(C(C1C=CCC1)=O)CC2 58698,c1(C(=O)NCC2CCC(CNC(C3CC3CF)=O)CC2)c(O)cccc1Cl 58699,N1(C(c2c(C)cccc2)=O)CCN(C(C2(C(F)F)CCCO2)=O)CC1C(F)F 58700,C1(F)(CNC(C2(CSC)CC2)=O)CCCN(C(=O)C(C)O)CC1 58701,Nc1cncc(C(=O)NC2CCOCC2NC(C2COCCO2)=O)c1 58702,c1(OC)ccc(CCNC(C2CCC(n3cc(-c4ccc(Cl)s4)nn3)C2)=O)cc1 58703,CC(C)CCCCC(=O)N1CCC(C2CCCN2C(c2cc(Br)n[nH]2)=O)C1 58704,C1(C)(NC(Cc2cc(C)sc2C)=O)CCCN(C(C2CCCCC2(F)F)=O)C1 58705,c1(C(N2C3CC(CNC(CSCCOC)=O)C(C3)C2)=O)cc2ccccn2c1 58706,c1(CC(N2CCC(F)(CNC(c3ncc(F)cn3)=O)C2)=O)cn2ccsc2n1 58707,Cn1nc(C(=O)NCC2CC(F)CN2C(=O)CC2(O)CCCCC2)c(Cl)c1Cl 58708,C(=O)(CC(C)(C)C(F)F)N1CC2(COC)CC1(CNC(=O)C#CC(C)C)C2 58709,C1(NC(C2C3(CC3)C23CC3)=O)CC2CC(NC(C3CCSCC3)=O)C1C2 58710,c1(CC(N2C(CNC(c3ccoc3Cl)=O)CC2)=O)noc2cc(F)ccc12 58711,N1(Cc2nc(CCOCC)sc2)CC2C(=O)N(C)C(=O)C2C1 58712,Cc1[nH]nc(C(F)(F)F)c1C(=O)NCC1CN(C(=O)CC2CC2C2CC2)CCO1 58713,c1(CC(=O)NCC2(C)C(C)CN(C(C3C(C)C3C)=O)C2)cccc2c1CCC2 58714,c1(CSC)ccnc(F)c1.c12ccccc1NC2c1nnnn1Cc1cccs1 58715,C12(CC)COC(=O)N1CCN(C(C1CC13CCN(C(C)CC1(C)CC1)CC3)=O)C2 58716,C1(NC(C(CCO)N(C)C)=O)CCN(C(C2CCCS2)=O)CC1O 58717,N1(C(Cc2c(CC)cccc2)=O)CC2CC1CCC2NC(c1cnsc1)=O 58718,C1(NC(C(F)=CCC)=O)(COC)CCN(C(=O)C(C)Cc2cnc[nH]2)C1 58719,C(C1CCCCC1)=CC(=O)NC1C(NC(CCc2cc(C)[nH]n2)=O)CC1 58720,c1(Cc2onc(C(=O)NCCC(C)NC(=O)CCCF)n2)ccc(Cl)cc1 58721,N(C(=NCCC(C)(C)C)NCC(F)F)CC1CC(C)OC(C)C1 58722,c1(C(=O)NC(C)CC(N2CCCCC2CO)=O)ccc(S(C)(=O)=O)o1 58723,C1(N(C(=O)CC2(SC)CC2)CC)CCN(C(c2c(C(F)(F)F)coc2C)=O)CC1 58724,CCCCC(F)C(=O)N1CC(OCCC(=O)Nc2cccc(COC)n2)C1 58725,S(=O)(=O)(c1ccc(NC2CCOC3(CCCC3)C2)c(F)c1)NCC(C)CO 58726,CC1CC2(CC(C(=O)NCC3(C)CC3C(=O)NOCCCN(C)C)C2)C1 58727,C1(NC(c2cc(C)sc2C)=O)CCC12CCN(C(c1ccc(O)cc1)=O)CC2 58728,C1(NC(c2c(CNC(C(=Cc3ccco3)C)=O)occ2)=O)COC2(CCC2)C1 58729,CC1(C)CCCC(O)(C(N2CCC2CNC(=O)CC2CC2(C)C)=O)CC1 58730,CC1(C)C(CC(=O)NCCOCCNC(=O)Cc2ccco2)CC1O 58731,CC1(C)COC(C(=O)NC2CCCC(CNC(c3cc(Cl)ccc3Cl)=O)C2)CO1 58732,C1(C(=O)NC(C2CN(C(c3cccc(O)n3)=O)C2)C)C2CCC1(c1ccco1)C2 58733,C12(NC(C3C(C=C)CC3)=O)CC(C1)N(C(=O)Cc1sc(S)nc1C)C2 58734,Cc1[nH]c(C#N)cc1C(=O)NCCCC(C)NC(=O)CCCc1ccc(F)cc1 58735,C(CCNC(=O)CCc1cc(C)no1)(C(C)C)NC(COC(CC)(C)C)=O 58736,C(=O)(CC(CC1CCC1)NC(=O)C(C)n1cncn1)N(C1C(C)CC1)C 58737,C(=O)(C(C)CC(F)(F)F)NCCCN(CCCNC(=O)C(c1ccnn1C)O)C 58738,C(CCC(O)C(=O)NCc1ncco1)NC(c1cc(CC)nn1C)=O 58739,C(=O)(CCCC(=O)N1CC(N(C)C(C2CCC(C)O2)=O)C(O)C1)N(CC)CC 58740,CN1CC(C)(C)CC1C(=O)NC1CCCC1CNC(c1cc(Cl)cs1)=O 58741,c1(OC)cc(OCC(N)=O)ccc1NC(C1CC(SC)C1N)=O 58742,N1(C(C2CC(SC)C2)=O)CCC(NC(C2CN3CCC2CC3)=O)C(O)C1 58743,N1(C(c2c(C#C)cnn2C)=O)CCC2(CCCN2C(C23CCCC2CCC3)=O)C1 58744,C1(O)(C(=O)NCC2N(C(c3cnc(Cl)s3)=O)CC(C)(C)OC2)CN2CCC1CC2 58745,c1(NC(C(C)N(C)C(=O)OC(C)(C)C)=O)c(O)nn(C)c1C(F)(F)F 58746,c1(OC)cc(CN2CCCC2C(=O)Nc2cc(C#N)cnc2Cl)cc(I)c1OC 58747,C1(CC(=O)NC2CCC(NC(CC3CN(C)C3)=O)C2)CCC(C(F)(F)F)CC1 58748,c1(C(c2n(C(CC)C)nnn2)NCCc2nccs2)cc(Cl)ccn1 58749,C1(C(=O)NC2(CCNC(C3(CC(C)C)CC3)=O)CC2)CC(=O)N(C2CN(C)C2)C1 58750,CCCC(C#N)C(=O)NC(C(=O)NOC(C)(C)C(=O)OC)C1(C)CC1 58751,c1(N2CCCC(OCC=C)C2)nc(=N)[nH]c(=NCCc2ccc(CSC)cc2)[nH]1 58752,CC1CC=C(C(=O)N2CCC(F)CC2C(=O)NOCCF)CC1 58753,C(=O)(C(CC(C)C)C(C)C)NC(CC)CNC(c1nnn2c1CSCC2)=O 58754,C1(NC(c2c(CC)n(C)nn2)=O)CN(C(c2cnn(C)c2F)=O)CC12CC2 58755,C#Cc1ccc(C(=O)NC2CC3CCC(C2)N3C(=O)CC2CCOC2)cc1F 58756,C1(F)(C(=O)NCCN(C)C(c2cncc(-n3cncn3)n2)=O)CCOCC1 58757,Cc1ccc(C(=O)N(CCC(=O)NC(C)CCC2CCCO2)C(C)C)c(O)c1 58758,N1(C(C2C(CC)C2)=O)CC2(CC)CC1(CNC(=O)CNC(c1cnccn1)=O)C2 58759,C1(CNC(C2(CCOC)CCC2)=O)C(C)CCN1C(C1CC1C)=O 58760,C1(NC(CCOCC(C)C)=O)CN(C(=O)CN2CC3CC3C2)C2(CCC2)C1 58761,Cc1cccc2c1CC(C(=O)NC1COCCN(C(=O)C(F)=C3CCCC3)C1)O2 58762,N1(CC)CCCC1CC(=O)N(CC(C)(C)CNC(=O)C=Cc1ncc[nH]1)C 58763,C(=O)(CCC(=O)N1CC(c2ocnc2CNC(=O)CCC2COCCO2)C1)OC 58764,c1(OC)coc(C(=O)NCC2(C)CCCN2C(=O)COCCN(C)C)cc1=O 58765,C1(OC)CCCCC1C(=O)NC1(CO)CN(C(C2CC(=O)N(C)C2)=O)C1 58766,C1(NC(C23C(CN(C(=O)C=Cc4cc[nH]c4)C2)C3)=O)CC2(CCCO2)C1 58767,C1(O)(CCNC(c2c(C)nsc2)=O)CCN(C(=O)C(C)Cc2cnc[nH]2)CC1 58768,C(=O)(CCCC(C)(C)C#N)N1CCN(C(C(OCC)OCC)=O)CC1CO 58769,c1(OC)ccc(C(=O)NC2CCN(C(C3CC3(F)F)=O)C2C2CC2)c(O)c1 58770,C1(CC(=O)NCC2CC(NC(c3cc(C)[nH]n3)=O)C2)CCC2(CCOCC2)CO1 58771,C1(C(=O)NC(C)CCN(C)C(c2ccc(C(C)(C)C)cn2)=O)CC2(C1)CC21CC1 58772,N1(C(C(CSC)C)=O)CCN(C(C2CCC(=O)N2C(C)C)=O)CC1c1cn[nH]c1 58773,C12(CNC(=O)NCCCC3CCCCO3)CCC(CO1)C2 58774,N1(C(C(C2(O)CN(C(C3(N(C)C)CCCC3)=O)C2)F)=O)CCC2(CC1)OCCO2 58775,c1(C(N2CCC(O)(CNC(COCCOCC)=O)C2)=O)ccc(C2CC2)cc1F 58776,C1(C(=O)OC)CC(Oc2ccc3cc2-3)C12CCOCC2.C(C)(C)(C)OC 58777,C1(c2ccccc2)(CCNC2C(F)(Br)C2)CCCC1 58778,N1(C(C(C)(C)CO)=O)CC2CCN(C(c3conc3C3CC3)=O)CCC2C1 58779,C1(CN2CCC(NC(COC(CC)C)=O)C2)CCOC(C)C1 58780,c1(C(=O)NCC2CC(NC(C3C(CCC)CCC3)=O)C2)ccc(N)cc1 58781,c1(SCC)nccnc1C(=O)NCC1(CSC2CC(CC(C)(C)C)C2)CCCO1 58782,c1(OC)ccc(SCCC(N2CC3CC3(NC(C34CCC(C3)C4)=O)C2)=O)cc1 58783,CC1(CNC(C2CC2C)=O)CCN(Cc2cccnc2Cl)CC1 58784,C#Cc1ccccc1CC(=O)NCC1C2CC1N(C(=O)C(C)(Cl)Cl)C2 58785,c1(N(c2ccccc2F)CCNC(C(CC)N(C)C)=O)nc(C2CC2)nc(=N)[nH]1 58786,c1(N2CC(c3c4occ(C)c4ccc3)OCC2)ccn2ncc(S(=O)(=O)NC)c2n1 58787,N1(C(c2cc(F)ccc2CO)=O)CCC2C(CCN2C(=O)CN2CCSCC2)C1 58788,C1(=CC(=O)NC2CCN(C(c3ccc(F)s3)=O)C2)CN2CCC1CC2 58789,C12(CNC(c3ccn(CCNC(C(CCC)F)=O)c3)=O)CCCN(CC1)C2 58790,Cc1nn(CC(=O)NC2CCN(C(=O)CSC(C)(C)C)C2C)c(C)c1Cl 58791,CC1CC(NC(=O)C(=O)NCC2CC2)CN1C(c1cnc(C(F)F)nc1)=O 58792,CC(C)C(C(F)(F)F)NC(C1CC=CCN1C(c1ccc(Cl)s1)=O)=O 58793,N1(C(c2ncn(-c3ccn(C)n3)c2)=O)CC2CCN(C(c3csc(=N)[nH]3)=O)CC12 58794,c1(C(N2C(CCN(C(=O)CC(C)(C)O)C)CCCC2)=O)cc(Cl)c2c(c1)OCO2 58795,N1(C2CCCN(C(CSCC=C)=O)C2)CCN(C(C2CC(N(C)C)C2)=O)CC1=O 58796,N1(C(C(Cc2ccoc2)NC(c2ncc(F)cc2F)=O)=O)CC2CC1CC2O 58797,C1(F)(C(=O)NCCOCC(=C)C)CCN(C(C23CCN(CC2)CC3)=O)CC1 58798,N(C1CCCc2cc(F)ccc21)C(N1C(CCC)(CCC)CCC1)=O 58799,C1(C(=O)NCc2c(C)non2)CCCN(C(=O)C(F)CC2CCCC2)C1 58800,c1(C(=O)NCC2CC(NC(C(C(CC)C)C)=O)C2)c(C)ccc2ncccc12 58801,Cc1nnc(CCCC(=O)N(CC(O)CNC(c2ccc(CO)cn2)=O)C)n1C 58802,Cc1nc(CC(=O)NC(Cn2cncn2)C(=O)NC2CC(CCC(N)=O)C2)n[nH]1 58803,C(=O)(CC(C)C(=O)NCCOCCN(C(=O)Cc1ccc(C)c(C)c1)C)OCC 58804,CN1CCC(n2cc(NC(C3CC3NC(C3CCC=CC3)=O)=O)cn2)CC1.C(=O)O 58805,N1(C(C2CNC(=O)N2)=O)CC(NC(c2csc3cncn23)=O)C2CCCCC12 58806,C(=O)(CC(C)(C)C(C)(F)F)NCCNC(C1N(C(C)C)CCC1)=O 58807,c1(C(N(CCOCCCNC(Cc2scc(C)c2)=O)C)=O)ccc2ncnn2c1 58808,c1(C(=O)NC2(CCNC(CC)=O)CCC2)cnn2cc(OC)ccc12 58809,N1(C(c2nc(CC)sc2)=O)CC(N(C(=O)CN=S(C)(C)=O)C)C2(CC2)C1 58810,C1(CC(=O)OC(C)(C)C)CCCCN1.C1(N(C(=O)CO)C)CN(C(=O)C2CC2)C1 58811,C(=O)(C#CC1CCC1)NCC1(C)N(C(C(CC)CC2CCCC2)=O)CCC1 58812,C1(CCN(C(Cc2cc(C)[nH]n2)=O)CC2CC2)CCN(c2nnc(CO)s2)CC1 58813,c1(C(N(CC(O)CN(C)C(C2CCC2)=O)C)=O)ccc2nn[nH]c2c1 58814,CC(CC(C)NC(=O)Cc1csc(C(F)(F)F)n1)NC(=O)C(F)(F)C1CCCC1 58815,N1(C(c2ccc(C=C)cc2)C(=O)NCCC)c2ccccc2C(C)C1C 58816,C(CNC(=O)Cc1ccc(F)cc1F)(CC(F)(F)F)NC(c1c(C)[nH][nH]c1=N)=O 58817,C1(CNC(CSCC)=O)CCCCCN1C(c1oc(CC2CC2)nc1C)=O 58818,N1(C(CCCCCN(C)C)=O)CC2CC(NC(=O)CCc3cnccn3)CC1C2 58819,c1(N2CCC(NC(C3C(=C)C3)=O)C2)nc(C(C)CC)ccc1C#N 58820,C1(C(=O)NCCOC2CCCC2)CCC2CCC1N2C(=O)Cc1ccccn1 58821,C1(C(C)NC(=O)C=CC2CCC2)CN(C(C2(C(F)F)CC2)=O)CCO1 58822,c1(CN(C(=O)CC(n2cc(C3CC3)nn2)C2CC2)CCOCC)ccc(Cl)cc1 58823,c1(NC(C2(CNC(C=Cc3ccc(C)s3)=O)CC2)=O)ccc(C)c(Cl)c1 58824,C(=O)(C(CNC1CC1)Cc1ccc(Cl)cc1)OC.c12ncc(s1)c(=O)[nH]2 58825,N1(C(C2(COC)CCCC2)=O)CCC(CNC(C2C=CCCC2)=O)(OC)C1 58826,c1(NS(C)(=O)=O)cc(NC(=O)NCCCn2cnnc2)ccc1F 58827,N1(C(C2N(CC)CCC2)=O)CCC(CC(=O)NC2CCC(=O)N(C)C2)C1(C)C 58828,CN1CC(C(=O)NCCC2CN(C(c3cnn(C(F)F)c3)=O)C2)CC1=O 58829,N1(C(=O)OCCNC(C)(C)C)CCOC(CN2CCCC2)C1.c1(NC)ccc(Cl)cc1 58830,CSC1=C(C(=O)NC2CCC(CNC(=O)CN3CCCC3)C2)CCCC1 58831,Cc1occc1CC(=O)NCC(C)(F)CNC(C1(c2ccn(C)n2)CC1)=O 58832,C1(C(=O)NCCc2n[nH]cc2C(=O)NC(C)C(C)SC2CC2)(CC)CCOC1 58833,C(=O)(C(C(C)NC(c1ncncc1Cl)=O)C(C)C)NCc1nccc(C)c1F 58834,N1(C(CC2CCC(C)CC2)=O)CC2(CCC2NC(=O)C=Cc2cn(C)cn2)C1 58835,Cc1cccc(O)c1C(N1CC(N(C(=O)C(C2CCOCC2)C)C)C(C)(C)C1)=O 58836,S(=O)(=O)(c1ccc(NCCc2cc(C(F)(F)F)co2)c(Cl)c1)NC1CC(C)C1 58837,C(CC(=O)N(C)CCNC(=O)C(C1(C)CC1)NC(=O)C(C)C)OCC=C 58838,C1(O)(CNC(c2n(C(C)C)ncc2)=O)CCN(C(=O)CN2C(=O)CCC2=O)C1 58839,N1(C(C(C(C)C)SC)=O)CCC(C2CCN(C(=O)COC(C)C)C2)CC1 58840,C12C3CC1N(C3)C2=O.O=C(C(F)CC1CCCCC1)N1CC(N2CCCCC2)C1 58841,CC(CN(C)C)C(=O)NC1CCC(CNC(C2(C)CC2Br)=O)C1 58842,C1(C(=O)NCC(CCNC(c2cnc(C3CC3)[nH]2)=O)OC)C(C#N)C1(C)C 58843,Cc1c(N(CCCN2CCN(C)CC2)C)ncnc1N1CCCC2(CC2)C1 58844,c1(C(=O)NCC(CC)(C)NC(=O)C=CSC)ccc(C(C)C(F)(F)F)cc1 58845,c1(C(N(C)CC2CN(C(=O)C(C)(C)C3CC3)CCO2)=O)ccc2scnc2c1 58846,C1(C(=O)NC(c2cnc(C)s2)C)(COC)CCN(C(=O)CCOC(C)C)CC1 58847,N1(C(C(C)OC)=O)CCCCC2(CCN(C(c3cnn4ccncc34)=O)C2)C1 58848,c1(C(C(=O)N(CC(C)O)CCNC(C2(OC)CC2)=O)OC)ccccc1 58849,Cc1ncccc1C=CC(=O)NCCC1CN(C(=O)COC2CC2)CC(C)O1 58850,C1(CN(C)C(C2(Cl)CC2(C)C)=O)CCN(C(c2c[nH]cc2Br)=O)CC1 58851,C(=O)(C(F)n1ccnc1)NCCCN(C(C1CCSC1)=O)CC 58852,C#CCC(C)(CC)C(=O)NCCC1CCN(C(=O)Cn2[nH]cnc2=N)CC1 58853,CCC(CC(=O)N1CC(F)(CNC(C23CC2COC32CCC2)=O)C1)CC(C)C 58854,c1(C(N(CC(CC)NC(=O)CC(C)C2CC2)C)=O)cc(O)ccc1OC(F)F 58855,Cc1cnc(F)c(CNC(C23CC(NC(=O)C(F)(F)CN(C)C)(C2)C3)=O)c1 58856,C1(NC(C(COCc2ccccc2)OC)=O)(CO)CCN(C(=O)CSC)C1 58857,C#CCC(C)(C)C(=O)NCC1(C(N2CCCCC(N(C)C)C2)=O)CC1 58858,C1(OCC)CC2(C1)CC2C(=O)NCCCNC(=O)CCc1ncc(C(C)(C)C)o1 58859,Cc1c(F)cccc1S(=O)(=O)N1CC(NC(=O)Cc2ccccc2I)C(C#N)C1 58860,Cc1csc(CCCC(=O)OCCNC(C2CC(OC3(C)CCOC3)C2)=O)n1 58861,C1(C(N2CC(NC(Cn3ncc(C#C)c3)=O)CC(C)C2)=O)(OC)CCC(C)(C)C1 58862,C1(C(=O)NC2(C)C(C)CCC2)CCOCCN1C(=O)CC1(N(C)C)CCC1 58863,N1(C(C=CCOC)=O)CCC(CCNC(C2CCC2(C)C)=O)C1 58864,c1(C(=O)NCCC2N(C(CC(C=C)C)=O)CCCC2)cccc(C)c1Br 58865,N1(CC(=O)NC(C#C)(C)C2CC2)CCC(C(=O)O)C(c2cnn(C)c2)C1 58866,C(=O)(C1=CCCOC1)N1CCC(COC)(NC(=O)CC2CCCN2C)C1 58867,c1(-c2ccn(CC)n2)cnc(NC(c2ccsc2C(C)C)=O)c(O)c1 58868,C(CNC(C1CCC(N(C)C)CC1)=O)(CC(F)(F)F)NC(C=C(CCC)C)=O 58869,CCC(C)C(O)C(=O)NCCC1(NC(=O)CCCN(C)C(C)C)CCOCC1 58870,c1(CC(N2C(CN(C(Cc3nnc(C)s3)=O)C)CCC2)=O)cc(F)c(F)cc1F 58871,C12(CCNC(CCCC#N)=O)CCC1CN(C(c1cnc(O)o1)=O)C2 58872,c1(NC(=O)C=CC(=O)OCC)ccc(C(N2CCC(CCC=C)C2)=O)cn1 58873,c1(COC)nc(N2CCCC2C2(NC(c3cnc(C)o3)=O)CCC2)cc(C)n1 58874,c1(CNC(C2CCC(NCc3cscc3Br)CC2)=O)cc(F)cc(F)c1F 58875,c1(NCC2C(C)CCN(C(C3CCCSC3)=O)C2)cccc(F)c1[N+](=O)[O-] 58876,CC(N=c1[nH]c(N2CCOC(C3CCCC3)C2)nc2c1SCC2)c1ccncc1 58877,C1(NC(c2c(C)cno2)=O)CN(C(=O)C(C)(O)CC(C)C)CC12CCOCC2 58878,C1(OCCC)CCCN(C(C2(C(C)NC(c3cnc(C)o3)=O)CC2)=O)C1 58879,c1(C(c2nnnn2CC)NCC(=C)F)ccc2ccccc2c1Br 58880,CC(C1=CCCCC1)n1ccnc1-c1ccc(-c2ccc(O)nc2)cc1 58881,CC1(C)CN(C(=O)NC2CCCC3CC23)Cc2cccc(OC)c2O1 58882,C1(C(=O)Nc2cc(C(=O)OC)no2)CCC2CCC1N2C(=O)CCSC 58883,C1(C(=O)NCC(C)NC2CC2C2CCCC2)CN(C(=O)OC(C)(C)C)CCN1C 58884,C1(CNC(C(COC)O)=O)CCCC12CCN(C(c1cn(C)ccc1=O)=O)CC2 58885,C(C(C(=O)N(CC(=O)NC)C)C(C)C)NC(COCCCC#C)=O 58886,C1(CCc2n(CC=C)nc(-c3ccccc3Cl)n2)CC(OCC)C12CCC2 58887,c1(-n2cc(C3N(C(C(C)OCC(C)C)=O)CCC3)nn2)c(F)cccc1Cl 58888,Cc1nc[nH]c1C(=O)N(C)CCOCCN(C)C(C1CS(=O)(=O)C1)=O 58889,c1(C(=O)NC(CC)CN(C(=O)C=CC(F)(F)F)C)c(C)cc(C)nc1C 58890,C1(C)(C(N(CCNC(CC2N(C)CCCC2)=O)C)=O)CCC2CC2C1 58891,N1(CC(N2CCS(=O)(=O)C3CCCC23)=O)C(=O)c2cccnc2C1=O 58892,C1(NC(c2cn(CCN(C)C)nn2)=O)CC(CNC(C2C=CCCC2)=O)C(O)C1 58893,c1(C(N2C(CNC(c3ccc(OC)nc3)=O)C=CC2)=O)cnn2c1OCCC2 58894,C(CNC(c1nc(C)oc1C)=O)(C(C)C(C)C)NC(CCCC)=O 58895,C1(CNC(C=C(CC)C)=O)CC2CCC(C1)N2C(=O)Cc1csc(Br)c1 58896,C1(CNCCc2c(C)c(Cl)ccc2)CCC2(CCCOC2)O1 58897,C1(O)(CN(C(C(C)c2cc[nH]n2)=O)C)CCN(C(=O)CCn2ncn(C)c2=O)C1 58898,N1(C(CC=CC=C)=O)CCCC2CN(C(c3cc(Br)ccn3)=O)CCCC12 58899,Cc1ccnc(C)c1C(=O)NC1CCCCC1NC(C1(C(F)F)CCCO1)=O 58900,N1(C(=O)NCC)CCC(C(N2CCC(OCc3conc3C3CCC3)C2)=O)C1 58901,CC(C(=O)NC1CN(C(c2ccc([N+](=O)[O-])c(O)c2)=O)CC1O)C(F)(F)C(F)F 58902,Cc1cn2cccc(C(=O)N(C)CC3(NC(c4cnoc4C4CC4)=O)CC3)c2n1 58903,c1(C(c2n(C(CC)(C)C)nnn2)NC2C=CCCC2)ccc2scnc2c1 58904,C1(CC(N2C(C)(CCC)CC2)=O)CN(C(c2cc(F)ccc2O)=O)CC12CC2 58905,CC(CC(C)(F)F)C(=O)NC1COCC1NC(c1cccc2c1COC2)=O 58906,C(=O)(CCC(C)(C)[N+](=O)[O-])N(C1CCCN(C(=O)C=C2CCC2)C1)CC 58907,Cc1cccnc1CC(=O)N(C(CCSC)C(=O)NC1(CCF)CC(O)C1)C 58908,N1(C(c2c(C)nc[nH]2)=O)CCC(C2CCN(C(C34CSC(C3)C4)=O)CC2)CC1 58909,c1(C(N2CCN(C(c3cnc(SC)s3)=O)C3C2C3)=O)cc2ncccn2n1 58910,N1(C(C)=O)CCC(NC(=O)CN(C)C(c2coc(C(C)C)n2)=O)CC1 58911,CCC(C)CC(C(=O)N(CC(C)(C)COC)C)NC(=O)C1=C(Cl)CCOC1 58912,N1(C(COc2cccc(C)c2C)=O)CCC(C2CC2NC(=O)CC(C)(C)F)CC1 58913,C12(C(N3CC(NC(COCCOC)=O)C3)=O)CC(c3ccccc3)(C1)C2F 58914,C1(C2CCN(C(=O)CCC3C(c4ccn(C)c4)C3)CC2)(C(=O)CCF)CCC1 58915,C1(CCNC(c2c(COC)non2)=O)CCCN(C(c2scnc2C(C)C)=O)C1 58916,N1(C(COCCN(C)C)=O)CCCC1CN(C)C(c1csc(C2CCCO2)n1)=O 58917,C1(C(=O)NC(CCC(=O)N(C)CC)C)CC(=O)C12CCC2 58918,C1(OC)CC(C(N2CCC(c3cnccn3)CC2)=O)N(Cc2ccccc2Cl)C1 58919,C1(C(=O)NCC2(F)CN(C(c3ccccc3CO)=O)C2)CCCCC1C1CC1 58920,N1(C(C(Cn2cccn2)OC)=O)CC(C(N2CCC(O)C2)=O)C(C(C)C)C1 58921,c1(C(=O)NCC(C)(C2CC2)NC(C(C)SC)=O)cc(Br)c(C)o1 58922,CC1(F)CN(C(c2cnc3[nH]ccc3n2)=O)CCN(C(C2CC3CCC2O3)=O)C1 58923,CCC(C)C(C(=O)N1CCCC(CN=c2[nH]nc(C3CCCC3)s2)(CC)C1)OC 58924,C1(C(N2C(C)(COC)CC2)=O)CSCCN1C(c1ccc(CO)o1)=O 58925,N1(C(C(c2cc(C)oc2C)C)=O)CCC(CNC(c2cccc(N)c2)=O)CC1C 58926,N1(C(CP(C)(C)=O)=O)CCOCC(CNC(C2CC(n3ccnn3)C2)=O)C1 58927,c1(C(C)C)cccc(C(=O)N(C2CCN(C(C3CC3(C)C(F)F)=O)C2)CCO)c1 58928,CC1(CN)CCCN(C(=O)CCc2ccc(Br)c(Cl)c2)C1 58929,CC1CC(c2cn(-c3ccncc3)nn2)CCN1C(=O)CSC1CC1 58930,C(=O)(CCC(C)C#N)N1CCC(N(C(c2sc(CCC)c(CC)c2)=O)CC)CC1 58931,CC1CN(C(c2ccn(Cc3cccc(C(F)(F)F)c3F)n2)=O)CC(=O)N1 58932,CC1(C)CC(NC(c2cc3c[nH]nc3s2)=O)CN(C(C2CCS(=O)(=O)C2)=O)C1 58933,c1(OC)cc(F)c(NC(C2(C)CCN2C(=O)Cc2ncccn2)=O)c(F)c1 58934,C1(NC(C(C)OCC(C)C)=O)CC2CCC(C1)N2C(c1cc2c([nH]1)CCOC2)=O 58935,c1(NC(C2(F)CCN(Cc3nc(C)sc3)C2)=O)cncc(Br)c1C 58936,c1(C(=O)NC(C(C)NC(c2nc(C#C)sc2)=O)C)ccc(C(C)C)cc1O 58937,N1(C(CN(C(C)=O)C)=O)CCCCC1C1CCN(C(=O)C(C)CC2CC2)CC1 58938,N1(C(C(F)=C(C)C)=O)CC(NC(=O)Cc2[nH]cnc2C)C(C2CC2)C1 58939,C1(NC(C2C(NC(C(C(C)O)N(C)C)=O)CC=CC2)=O)CCCC(O)C1O 58940,C12(C(N3CCC(CNC(C(C)SCC)=O)C3)=O)COCC1CS(=O)(=O)C2 58941,N1(C(c2cn(CCC)nn2)=O)CCC(NC(c2cn(C)cc2C)=O)CC1C1CC1 58942,C12(C(N3CC4C(NC(c5cccc(C)c5F)=O)C4C3)=O)CCCCC1OCC2 58943,Cc1oc(C)c(C(=O)NCCCOCCNC(C2CC3CC3C2)=O)c1Br 58944,C(=O)(C#CC1CCCCO1)NC1CCC(NC(c2sc(C)c(Br)c2)=O)CC1 58945,c1(C(=O)NCc2c(C(=O)NC3CC(C)OC3=O)cccn2)ccn2ccccc12 58946,S(=O)(=O)(c1ccc(Br)cc1F)N1C2CCN(C(c3ncccc3Cl)=O)C2CCC1 58947,CCC(F)(F)CC(=O)NCC1CN(C(c2coc(CC3CC3)n2)=O)CCCO1 58948,c1(C(N2C(CNC(C(C)P(C)(C)=O)=O)CCCC2)=O)cc(=O)n2nccc2[nH]1 58949,CC(CC(=O)NCC(CNC(=O)C=CC=C(Cl)Cl)CO)c1cnn(C)c1 58950,c1(N2CC3CC(NC(C=C(C)c4ccco4)=O)C3C2)ncc2c(n1)CCCC2 58951,N1(C(C(C)OC)=O)CCCC(O)(CNC(=O)CSC(C)(C)C)CC1 58952,c1(C(N2CCN(C(C3(CC)CCC3)=O)CC2C2CC2)=O)ccc2c(c1)CCC=C2 58953,C12CCCC(C1)C(=O)NC1(C)CN(C1)C(=O)C2.Cc1nc[nH]c1CC(=O)N(C)C 58954,c1(C(N2CC3C(CNC(c4ccc(NC=O)cc4)=O)(C3)C2)=O)cccc(O)c1F 58955,C(C(C)C)(C(O)C(=O)N1CCCCCC1C(N1CC([N+](=O)[O-])C1)=O)OC 58956,C1(CNC(c2ncn(C(C)C)n2)=O)CC(C)CCN1C(=O)CP(C)(C)=O 58957,C(=O)(CC(C(F)(F)F)NC(=O)CC(C)C1CC1)NCCN(CCOC)C 58958,Cc1cc(C(=O)N(C(CNC(=O)Cc2cnnn2C)C2CC2)C)cn1C(C)C 58959,C1(C(N(C2CCCN(C(c3ccsc3)=O)CC2)C)=O)CC(F)(F)C12CCC2 58960,CCC(CN(C)C)CC(=O)N(CCCC(=O)NCC1(C)CC1(F)F)C 58961,c1(CNc2c(F)cc(C(F)(F)F)cn2)ccc2ncc(Br)cc2c1 58962,c1(C(CO)NC(C(C)C#N)=O)ccc(F)c(Cl)c1 58963,N1(C(CC=CC)=O)C2CCC1C1CC1(NC(C1COCCN1CC(F)(F)F)=O)C2 58964,C(=O)(C(C)(CO)NC(C1CC(n2cnnc2)C1)=O)OC 58965,C1(CC(=O)NCC(C2(O)CN(C(C(C=CC)O)=O)C2)(C)C)CCCC12CC2 58966,C(=O)(C(O)CC(=O)OC)NCCCOCCN(C(COCC#C)=O)C 58967,N1(C(C2(CC3CCC3)CC2)=O)CCCC(O)(CNC(C2(F)CCS(=O)(=O)C2)=O)C1 58968,c1(-c2cc(-c3nc(CCCCCC)nn3CCOC)ncc2)cc(F)cc(Cl)c1 58969,C=CCC(CC(F)F)NC(=O)C(COC)NC(c1cccn1C)=O 58970,C1(N(C(C2C(C(C)NC(=O)Cn3ccnn3)C2)=O)C)CCCCCC1O 58971,N1(C(C2C(C)C2)=O)CCS(=O)(=O)C(CCNC(=O)CCc2cn[nH]c2)C1 58972,CCC(CC)(CCNC(c1nnn(-c2ccc(Cl)cc2F)c1C(F)F)=O)OC 58973,n1(CC)ccc(C(=O)NCCCCCCNC(c2csc3nnsc23)=O)cc1=O 58974,C1(C(N(CCC(=O)NCC(C#C)CC2CC2)CC=C)=O)C2CCCCCC12 58975,N1(C(c2n(CC)ccc2)=O)CC(C)OC2(CCN(C(=O)C(=O)CC(C)CC)C2)C1 58976,CCCC(C)(C)CC(=O)NC1CC(C(F)C(N2CC3(CC(CO)CO3)C2)=O)C1 58977,N1(C(C2(CNC(CCN(C)C)=O)CCCO2)=O)CCSC(C)(C)C1 58978,C1(OC)CCC12CC(C(=O)NC1CC1NC(c1c(C)noc1C(F)F)=O)C2 58979,c1(OCCC(=O)N(C2(O)CCN(C(C3(SCC)CC3)=O)C2)C)ccc(C)c(C)c1 58980,c1(OC)cc(C(N2CC3CC2CCC3NC(=O)CCS(N)(=O)=O)=O)c(O)c(Cl)c1 58981,C1(NC(C(C)N(C(c2cnn(CCO)c2)=O)CC)=O)CCCCCCC1 58982,c1(C(=O)NCC(CN(C(CCC(=O)NC)=O)C)O)ccc(OC)c(S(N)(=O)=O)c1 58983,C1(NC(c2c(OC)cncc2)=O)CCN(Cc2ccc(Br)[nH]2)CC1O 58984,C1(C(=O)NC(CNC(c2c(C)nn(CC(C)C)c2Cl)=O)(C)C)CN(CP(C)(C)=O)C1 58985,C#Cc1ccc(C(N2CCC3CN(C(=O)COCC=C)C3C2)=O)cc1C 58986,c1(C(N2CCCCC(NC(C(C)(C)c3cnsc3)=O)C2)=O)cn2c(n1)COCC2 58987,c1(C(=O)NCCC2(CNC(CCC(C)OC)=O)CC2)cnn2ccncc12 58988,c1(C(=O)NC2(CCNC(C(CC#C)C3CC3)=O)CC2)ccc(C)cc1C 58989,C1(CNC(C2CC(SC)C2)=O)CCCCN(C(c2c[nH]c(=N)s2)=O)C1 58990,C1(C(C)(C)C)(CNC(C2(C)CCCS2)=O)CCN(C(c2ccncc2)=O)C1 58991,C12(CC3CCC1CC3)C(=O)NC2.N1(C(CN(C2CCCC2)C)=O)CCOCC1 58992,CC(=O)CC(C)(C)CC(=O)NCC(C)N(C(=O)C#CC1(C)CCCO1)C 58993,CON(CC1CC1)C(=O)C(F)(CNC(=O)C1CCc2nccn21)C(C)C 58994,Cc1ccc(C(=O)NCC2CCC(NC(c3cnns3)=O)C2)cc1C 58995,N1(C(C=C)=O)CC(C)(C)CC1NC(C1CCC(C(F)(F)F)O1)=O 58996,C1(C2CC2)(C(=O)NC(CNC(C(C=C)O)=O)Cc2ccccc2)CCC1 58997,c1(C(N2CCN(C(C)=O)CC2c2cccc(F)c2)=O)cccc2ccn(C)c12 58998,Oc1c(CN2CCC(O)(CO)C2)cc(Br)cc1Cl 58999,N1(C(C(CC2CCCC2)NC(c2cc(CC)oc2C)=O)=O)CCC2(CC1)CSC2 59000,C1(C(=O)NCCNC(c2cc(CC)no2)=O)CC1C1CCC1 59001,C=CCN=C(NCCc1nccc(C(F)F)n1)NCc1nc(C)cs1 59002,c1(C(=O)NCCOC2CCN(C(C3CC(C)N(C)C3)=O)C2)c(F)cc(F)cc1Cl 59003,c1(C(=O)OC)c(C)[nH]c(C(=O)NC2CC(NC(C3C=CCC3)=O)C2)c1C 59004,N#CC1(CC(=O)N(C2(C(=O)NC(C3CCCO3)CO)CCC2)C2CC2)CCC1 59005,Cc1cc(NC(=O)C(Cn2cncn2)NC(=O)CC2CSCCO2)cs1 59006,C1(NC(c2nc(OC(C)C)oc2)=O)CCN(CCC2CCCCO2)CC1O 59007,c1(N(CC(C)NC(c2cn(C(C)C)nc2)=O)C)nc(O)c2ccc(Cl)cc2n1 59008,Cc1nocc1CC(N1CC=CC1CNC(=O)CCn1ccnc1C)=O 59009,C(CC(C)CC)(C(=O)NCCn1nc(C)cc1C)NC(CC(=O)OCC)=O 59010,C(C(COC)CC(=O)N1CCOC(C(C)NC(=O)C=Cc2scnc2C)C1)OC 59011,N1(C(C=CC(CC)C)=O)CC(C2CC2)(C(=O)NCc2ccc(CO)o2)C1 59012,C(=O)(C(CCC1CC1)NC(=O)C=CC1CC1)NCC 59013,N1(C(C(CN(C)C(c2ccccc2O)=O)O)=O)CC(F)CC1C(N)=O 59014,CC(C(=O)NCCCNC(C1CC1(c1c(F)cccc1F)C)=O)C1=CCCC1 59015,CCC(CC)CC(F)C(=O)N1CCC(CC(N2CCC3(C=CCO3)C2)=O)CC1 59016,c1(C2CN(C(=O)CNC(C3(c4nc[nH]n4)CC3)=O)C2)cccc(O)c1 59017,C1(NC(c2n(C)nnn2)(CSC)C2CC2c2ccc(I)cc2)CCC2(CCC2)O1 59018,C(C(F)(C(=O)N1CCC(F)(CO)C1)C(C)C)NC(C1CCC(=C)CC1)=O 59019,CC(C)C(C(=O)N1CCC(N(CC(=O)O)CCO)CC1)c1cccc(Cl)c1 59020,c1(C(=O)NC(C2(C(=O)N(C3COCC3O)C)CC2)C)cn(C)cn1 59021,Cc1cccc(C(=O)N(C2CCCCC2NC(C2OCCCO2)=O)C)c1 59022,N1(C(C(C2CCC2)OC)C(=O)NC2CCOC2)C2CCC1CC(=O)NC2 59023,C1(CC(=O)OC)CCC(NC(C2CN(C(c3ncccc3SC)=O)C2)=O)CC1 59024,N1(C(=O)CCSCc2ccccc2)CC2(CCN(C(=O)C3=CCCOCC3)C2)C1 59025,N1(C(c2ccn(CC)c2C)=O)CCN(C(c2ccc(O)c(C)c2)=O)CC1C 59026,CN(NC(=O)C(F)n1cncn1)C(N)=O 59027,c1(CNC(C(N2CC(C)C(F)(F)C2)c2nc(CC)[nH]n2)=O)ccc(F)c(F)c1 59028,c1(C(=O)NCCCN(C(CCOCC#C)=O)C)c(C)nc2sc(C)nn12 59029,c1(OC(C)=O)ccc(OCCC2CCCN(C(C)C)C2)cc1C 59030,C1(CC(=O)NCC(C(C)(C)C)NC(=O)CCC2CCCCC2)CC2CCC(C1)C2 59031,C1(C(=O)NC(CC=C)C(=O)NCC2CCCC(=O)N2)CC2(C1)CC21CC1 59032,c1(C(=O)NC(CNC(CSC)=O)(C)C2CC2)nc(O)[nH]c(=O)n1 59033,CCCCCC(O)C(=O)N1CCC2CCCC12C(=O)N(CCC1CC1)CC 59034,c1(C(=O)NC(C(=O)NC(CC#C)C(=O)NC)CCSC)cccc(F)c1F 59035,n1(C(CC)C)ccc(=NC(=O)C(CC(N)=O)NC(c2cc(C(C)=O)c[nH]2)=O)[nH]1 59036,C1(NC(C2N(C)CC(O)C2)=O)C2CC3C(C2)C13C(N1CC(F)(C#N)C1)=O 59037,C1(C(=O)NC2C(OC)CN(C(c3ccnc(OC)n3)=O)C2)CCc2ncncc2C1 59038,c1(SC)ccc(F)c(C(=O)N(C2CCN(C(c3cn[nH]c3)=O)CC2)CCO)c1 59039,C1(OC)CC2CN(C(c3ccc(Cl)s3)CSc3ccc(F)c(F)c3)CCN2C1 59040,CCCCCC(=O)NCC(COC)NC(=O)CC1CCCOC1 59041,Cc1nc(C(=O)OCC(F)(F)CCC(C)(C)C)oc1-c1ccccc1 59042,C1(NC(C(CC)c2cccnc2)=O)(NC(=O)CN2CCCNC2=O)CCCCC1 59043,C1(CNC(C(F)=CC)=O)CCCC1C(=O)NCCSC 59044,CC1CN(C(=O)CCC(C)(F)F)CCC1NCc1ncccn1 59045,C1(C(=O)NCCC2CC(F)(F)C2)(OC)CN(C(=O)CC2CCSC2)C1 59046,CC(C)C(CNC(=O)CC(O)CN(C)C)C(=O)NCCCSC(F)F 59047,CC1c2cccc(F)c2CCN1C(CCCCC1CCCC1)C(=O)NCC1CC1 59048,n1(CC)cncc1CNC(=O)C(C)(C1CCC1)NC(C1CC(CC2CC2)C1)=O 59049,CCC(CCOC)C(=O)NCc1cnn(C)c1C(=O)NC1(C(=O)OC)CCCC1 59050,c1(CC(=O)NC2C(C)N(C(=O)C=C3CN4CCC3CC4)CC2)cc(Cl)ccc1Cl 59051,c1(CN2CC(NC(C(C)Oc3ccccc3)=O)C(C#N)C2)cccc([N+](=O)[O-])c1 59052,NC(=O)CC(c1ccccc1)NC(C1CCC(Oc2ccncc2)C1)=O 59053,N1(C(C(C)(C)CF)=O)CC(CNC(c2ccncn2)=O)C(F)(F)C1 59054,Cc1cccc(CNC(C23CCC(NC(C4CCC(CO)O4)=O)(CC2)C3)=O)c1F 59055,c1(C(=O)NC(c2cn(Cc3cnoc3)nn2)C)ccoc1-c1ccccc1 59056,N1(C(CCCCSC)=O)CCC2(CC1)CC2C(=O)NC1(CC2CC2)CCC1 59057,CC1CCC(C(=O)NCC2(C(N)=O)CCCC2)CN1C(=O)Cc1cncn1C 59058,CC#CCC(C(=O)O)NC(=O)C(C)(C)C1CCO1 59059,c1(-c2ccc(N3CCCC(C=C)C3)c(N)c2)ccc(C#N)cc1F 59060,CC1CCC(C(=O)N(C(CNC(=O)CCCNC(=O)C(C)(C)C)C2CC2)C)C1 59061,C1(CN(C2CCN(Cc3ccnn3C)C2)C)CC(=O)N(CCc2ccccc2)C1 59062,Cc1cnc2c(C(=O)N(C(C)CCNC(=O)C(O)CN(C)C)C)cnn2c1 59063,C(C(F)(C(=O)NCC(C)C=O)C(C)C)OC.C12CCC3(CC13)C(=O)N2.OC 59064,C1(C(N(CCCCN(C)C(=O)OC(C)(C)C)C)=O)CC(C)(Nc2cn[nH]c2)C1 59065,CCCC(C)(C)C(=O)NCCc1ocnc1CNC(=O)COc1ccc(Cl)c(C)c1 59066,N1(C(c2nc(CC)sc2)=O)CCCC(O)(CNC(c2ccnc(Cl)c2OC)=O)C1 59067,n1(CC(=O)NCCNC(C2CN(C(C3CCC(C)O3)=O)C2)=O)ncn(C)c1=O 59068,c1(NC(N(CC(O)C(F)(F)F)CCOC)=O)scnc1C#N 59069,O=C(C1=COCCC1)NC1CCN(C(c2cnn(CCO)c2)=O)C(C2CC2)C1 59070,c1(C(=O)OCCC(C(=O)OC)C2CCCCC2)csc2c1CCOC2 59071,C12(COC)CN(C(c3ccnc(O)c3)=O)C(CNC(=O)C3=CCSC3)(C1)C2 59072,c1(C(=O)NCC2C(NC(C=CC=CC)=O)CC2)cc2c(=O)cc[nH]c2s1 59073,Cn1nc(CC(=O)NC(CCN)C(F)F)cc1Cl 59074,c1(C(=O)NCCN(C(c2cc(C)cc(Cl)c2)=O)CC)ccc2nccnc2n1 59075,N1(C(Cc2nc(CC)sc2)=O)CCC(C(C)NC(c2cccnn2)=O)CC1 59076,C1(NC(c2cc(F)cc(F)c2)=O)CC2CN(C(=O)CC3CCSCC3)CC12 59077,N1(C(c2c(OC)n[nH]c2)=O)CC2CCCC2(NC(c2nc(SC)ncc2N)=O)C1 59078,C1(CNC(C(=Cc2cccs2)C)=O)(Nc2ncn(C(C)(C)C)n2)CCCCC1C 59079,c1(C(=O)NC2CCC(N(C(C(C)NC(CC)=O)=O)C)CC2)cc([N+](=O)[O-])ccn1 59080,CN=c1nc(N2CCC(C)(N(C)C)C2)[nH]c(=NCCc2ccccn2)[nH]1 59081,c1(C(N2CCCC(N(C(C(CC=CC)C)=O)CCF)C2)=O)cc(C)cc(C)c1O 59082,c1(C(=O)NC(CC)CNC(C2CCCC(F)C2)=O)c(OC)cccc1O 59083,c1(C(=O)NC(CNC(Cc2cn(CC)nn2)=O)C(C)(C)C)c(C)cc(C)nc1O 59084,C(=O)(C(O)CCCNC(=O)CC1(O)CCCOC1)N1CCC(C(C)OC)CC1 59085,c1(N(C)Cc2ccc(CO)cc2)ccc(S(=O)(=O)NC2CSC2)cc1Br 59086,C(c1cc(Cl)cc(Cl)c1)=CC(=O)NCC(CNC(C1CC(CC)C1)=O)(C)O 59087,C12(C(=O)NCC3(C)ON=C(C)C3)CC(CN(C(=O)CS(C)(=O)=O)C1)C2 59088,CCC(CC)C(C)C(=O)N1CCOCC(NC(=O)C(n2cc(Cl)cn2)C)C1 59089,C(CC(C)C)(C(=O)NCC1CN(C(c2cccnc2O)=O)CCCO1)NC(C)=O 59090,C1(NC(COCCCCC)=O)CC2CCC1N2C(c1cnns1)=O 59091,C1(C(=O)NC(C2CCS(=O)(=O)C2)(C)C)CC2(CCC2=O)C1 59092,C(=O)(CCCC(=O)OC(C)(C)C)NC(CC1CCN(C(CCCCOC)=O)CC1)C 59093,Cc1ncc(C(N2CCC(C)(C(=O)Nc3cnc(N(C)C)nc3)CC2)=O)c(C)n1 59094,C1(C(=O)NCCC2(C(=O)NCc3ncc(C)cn3)CC2)CC2CCC1CC2 59095,C(=O)(C1=CCN(C(C2CC2OC(C)=O)=O)C1)N1CCC(=C)CC1 59096,Cc1ncsc1C=CC(=O)N(CC(O)CN(C)C(c1cnn(C)n1)=O)C 59097,c1(C(N2CCOCC(NC(=O)CCCN3CCCC3)C2)=O)cn2ccncc2n1 59098,C(C)(CCC(=O)NC1CCN(C(=O)C(F)(F)c2cnn(C)c2)C1)SC 59099,C(=O)(C(O)CC(F)F)NCC(c1ccc(F)cc1)NC(CN(CC)CC)=O 59100,C1(CNC(C=C=C(C)C)=O)CCN(C(=O)Cc2ccoc2)CC1C 59101,CCC(COC)(CC)C(=O)NCC(O)C(=O)OCC1CN(C(C)=O)CCO1 59102,C1(CC=C)(NC(=O)CCN2CCCCC2)CCN(C(C2(C(=O)NC)CC2)=O)C1 59103,C1(C2CCCCC2)(NC(C)CCNS(=O)(=O)Cc2ccccc2)CC1 59104,C1(NC(C(C)Cc2ccccc2)=O)CC12CC(NC(=O)CCCn1ccnn1)C2 59105,CCC(C)C(C)C(=O)N1CC(N(C(=O)CCc2c(C)nn(C(C)C)c2C)C)C1 59106,c1(C(N2CCC(CCNC(c3ccc(COC)[nH]3)=O)C2)=O)cc(N)c(O)c(F)c1 59107,N1(C(C2CCN(C(C)=O)CC2)=O)CC2(CCC2NC(=O)CC2CCCCCC2)C1 59108,C1(C(=O)NCC2CCN(C(C)C)C2)CCN(C(C2(F)CCCCC2)=O)CC1C 59109,C(c1cccc(F)c1F)=CC(N1CC(NC(c2onc(C)c2C)=O)C(O)CC1)=O 59110,c1(C(N2CCC(N(C(=O)C(C)CC3CC3)CC#C)CC2)=O)ccc(=O)n(CC)n1 59111,CCS(=O)CC(=O)NCC(C)(C1CC1)NC(=O)CC1CC(C)(C)C1 59112,c1(C(C(=O)NCCCC(=O)NC)NC(=O)CSCC(N)=O)c(C)cccc1Br 59113,C1(C)(NC(C(n2cc(Br)cn2)C)=O)CCCN(C(C2(O)COC2)=O)C1 59114,c1(N(S(=O)(=O)c2cc(Br)cc(Br)c2)CC)ccc2c(c1)CCC(=O)N2 59115,C(=O)(C(C)CS(=O)(=O)c1ccc(F)cc1)NCC1=CCN(C(C=CCC)=O)CC1 59116,C1(C)(C(N(C)CC2CCN(C(c3ccon3)=O)C2)=O)CCCN1C 59117,CC(C)CC(O)CNc1nccc(N2CCN(CCN3CCOCC3)CC2)n1 59118,n1(CC)cc(Br)c(C(=O)NCC(O)CCNC(c2[nH]c(O)nc2C)=O)n1 59119,CC(CCS(=O)(=O)N1CCOC(C(=O)N(C)C)C1)C(F)F 59120,c1(C(CC)C(=O)NC(C)(C)CCNC(=O)CSc2nc[nH]n2)cccc(Cl)c1 59121,N1(C(c2ncn(C)n2)=O)CC2CC(NC(=O)C=Cc3cccs3)CC(C2)C1 59122,C1(N(C(CN(CC#C)C(C2CCSC2)=O)=O)C)CCCOC1 59123,C12(C(=O)NC(C)C(=O)NC(C)(C)C)CC(CCO1)N(C(=O)C(C)N(C)C)C2 59124,C1(C(N2CC(C)(NC(c3cncc(-n4ccnc4)n3)=O)C2)=O)CCC2CC1CO2 59125,C1(CNC(C(C)OCC#C)=O)(CO)CC12CCN(C(=O)CC1CC(=C)C1)CC2 59126,Cc1nc(C(N2CCSCC2C(=O)NCc2ccncc2)=O)ccc1Br 59127,N1(C(C2C(=C)CC2)=O)CCC2(CCC2CNC(=O)C2=CCOCC2)CC1 59128,C=CCC(C(=O)NC1CCCCN(C(=O)C(C)(C)C(=O)OCC)CC1)C(C)C 59129,c1(C(N2CC(NC(C3(CC)CCNC3=O)=O)C2)=O)ccc2ncn(C)c2n1 59130,CC1CCCc2cc(C(=O)NCCCN(C)C(C3CCC4(CCC4)OC3)=O)nn21 59131,N1(C(C(C)N2CCC2)=O)Cc2nccn2CC(NC(=O)Cc2cnccc2Cl)C1 59132,N1(C(c2ccc(C)c(F)c2F)C(=O)NCCOC)CC(C)OC2CCCCC12 59133,Cc1n[nH]c(C)c1CCCNC(=O)COC(c1coc(-c2ccccc2)n1)=O 59134,C1(CN(C)C(C23CC(F)C2C3)=O)CCN(C(C2CC3CC3C2)=O)CC1 59135,c1(C(N2CCC(F)(CNC(c3cn(C)nc3Cl)=O)C2)=O)coc2ccc(F)cc12 59136,c1(C(N2C(CNC(C3CC34CC4)=O)C=CC2)=O)cc([N+](=O)[O-])ncc1Br 59137,c1(OC)ccc(Cl)c(CN2CCCC(C(=O)Nc3ncc(F)cc3Br)C2)c1 59138,c1(C(=O)NC2CCN(C(C3(C#N)CC4CC4C3)=O)CC2)ccnc2ccccc12 59139,C1(C(N2C(CCNC(c3ccoc3Br)=O)CCC2)=O)CC12CCOC2 59140,C1(CC(=O)N(CCCOCc2ccccc2)C)CCc2ccccc2C1 59141,C(C(CO)(CO)NC(=O)C(C)Cc1cnc[nH]1)N(C(C(C)OC)=O)C 59142,CCCCCC=CCCNC(c1[nH]ccc1CNC(=O)CC1CC(C)C1)=O 59143,N1(C(C(C(C)NC(C(=O)NCC)=O)C)=O)CC2CCC(C1)O2 59144,N1(C(CC2N(C(CCC(CC)C)=O)CC(F)C2)=O)CC(C2CC2(F)F)C1 59145,N1(C(CCOC(C)=O)=O)CC=CC1C(=O)NC(C)CN1CCCCC1 59146,N1(CC(=O)N(CC(c2ccccc2)C)C)C(=O)C=CC1=O 59147,N1(C(c2csc(Br)n2)=O)CCC2(CCC(N3CCc4nocc4C3)CC2)C1 59148,C1(C)(C(N(CCCO)C)=O)CC12CCN(CC1CC3CCC1O3)CC2 59149,CC1CN(C(C2CCN(C)C2=O)=O)CC(C)CN1C(c1cc(O)cs1)=O 59150,CCCC(CCC)CC(=O)NCC(O)CNC(c1sccc1CC)=O 59151,c1(C(=O)NC(CNC(C2CC(OCC)C2)=O)(C)C)cc(Cl)c(Cl)cc1OC 59152,CN1CCC(C(=O)NCCC2(O)CCN(C(=O)CCC3CC3(C)C)C2)CC1 59153,c1(NC(C2(c3cc(F)cc(F)c3)CC(O)C2)=O)cc(F)c(CO)c(F)c1 59154,CC1(CNC(=O)C=CC(=O)NC2CC2)CCCN(C(=O)CC(F)(F)Cl)C1 59155,C(N=c1[nH]c(=NC2CC3CC4C(C3)C24)c2ncccc2[nH]1)c1cc(C)c(F)cc1 59156,O=C(C1CCNc2ccccc21)NCC1CCN(C(C2CCC3CC3CC2)=O)C1 59157,S(=O)(=O)(c1ccc(=NCCn2cccnc2=O)[nH]c1)NC(c1ccccc1)C 59158,C(=O)(C1=CC2CCC(C1)C2)NC1C(NC(c2ccc(C)c(C#N)c2)=O)C1 59159,c1(C(=O)NCC2CN(C(C3C(CCC)C3)=O)CC2O)cn(C)c(=O)nc1O 59160,c1(CC)ccc(C(=O)Nc2ccc(NC(=O)NC3(O)CN(CC)C3)cc2)cc1 59161,C1(NC(c2cc3ccsc3[nH]2)=O)CC2CC(C1)N(C(C1Cc3nccn3C1)=O)C2 59162,C(c1ccc(S(C)(=O)=O)o1)=CC(=O)NC1CC(CCNC(C(C(C=C)C)C)=O)C1 59163,c1(C(=O)NC2CC(NC(=O)COc3ccc(F)cc3)C2)ccc(Br)c(Cl)n1 59164,C(=O)(C(CC)C(C)(C)CC)NC1CCC(CNC(c2ccc(C#C)o2)=O)CC1 59165,C1(NC(CC(C)n2cccn2)=O)C2CCC1CN(C(=O)C(=O)NCC(F)F)C2 59166,C1(C(=O)NC(CCCNC(Cc2cc(C)ns2)=O)C)CCN(C)C(=O)C1 59167,Cc1c(C(=O)NCC#CCNC(=O)CC2CCCC2(F)F)sc2ccccc12 59168,c1(C(c2ccc(OC)nc2OC)N(CC(=C)C)C=O)ncc(Cl)cc1Cl 59169,C12(NC(c3cccc(Cl)c3)=O)CCCCC1N(C(c1ccncc1)=O)CC2 59170,O=C1CC(NC(c2ccc(-c3ccncc3)cc2)=O)CCN1 59171,Cn1nc(Cl)c(C(=O)NC2CCN(C(=O)CCC(C)(C)C)C(C3CC3)C2)c1Cl 59172,C#Cc1cc(F)ccc1CN1CCC(O)(C(=O)Nc2ncc(C)cc2O)C1 59173,c1(CNC(=O)Cn2cccc2)csc(CNC(c2cc(F)cs2)=O)n1 59174,c1(NC2(CNC(C(C3CCCOC3)OC)=O)CCOCC2)ncc(Cl)c(O)n1 59175,N1(C(COC)=O)CCC2(NC(c3cncc(C(=O)OC)c3)=O)CC2C1 59176,C1(CCNC(c2csc(C)c2C)=O)C(C)CCCN1C(=O)COc1cnn(C)c1 59177,c1(C(=O)NC2CCCC(NC(c3c(C(C)C)nn(C)c3)=O)C2)nccc(Cl)c1O 59178,C1(NC(c2cc(C)sn2)=O)Cc2ccccc2N(C(c2oncc2C)=O)C1 59179,c1(C(N(C)CCN(C)C(c2cncs2)=O)=O)ccc(F)c(S(=O)(=O)NCC#N)c1 59180,N#CC1CCN(C(C2(NC(c3ccoc3)=O)CCOCC2)=O)C1 59181,n1(CCCC)nnnc1C(C1CC1C1CC1)NCc1noc(CC)n1 59182,C1(C#N)(C(N(CCCNC(C2(CC(F)(F)F)CC2)=O)CC)=O)CC2CCC1C2 59183,C1(N(C(=O)CC2CSC2)C)CN(C(=O)Cc2cnn(C3CC3)c2)CC12CC2 59184,C1(N(C(=O)C(=O)NC(Cc2cccc(OC)c2)C2CC2)CCC)CCS(=O)(=O)C1 59185,N1(C(C(C)N(C)C)=O)CCN(C(=O)CC(C)(C)c2ccccc2)C(CO)C1 59186,CC1(C)CCCC(CC(=O)NCCC2CCCN2C(=O)CN=S(C)(C)=O)O1 59187,N1(C(c2ccn(C(C)C)n2)=O)CC(C)CN(C(=O)CS(=O)(=O)C(C)(C)C)C(C)C1 59188,c1(CNC(=O)C(=O)NCC2CC3(CC3)C2)nnc2c(Cl)cc(C(F)(F)F)cn12 59189,C1(NC(CNC(C)=O)=O)CC(NC(c2cnc(C3CC3)s2)=O)C12CCC2 59190,N#CC1(C(=O)NCC2CC(O)CN2C(c2cnc[nH]2)=O)CCCO1 59191,C1(NC(CCOC)=O)CS(=O)(=O)C2CN(C(=O)CC3(OC)CCCC3)CC12 59192,C#CC1(OCC(=O)NC2CN(C(=O)CCOCCNC(C)=O)C2)COC1 59193,c1(-c2cn(CC3CC(NC(C4CC(=O)C4)=O)C3)nn2)cc(F)ncc1Cl 59194,C1(NC(c2c(C)[nH]cc2)=O)CCCCC1N(C(=O)Cc1ccc(Cl)s1)C 59195,c1(NCC)ncc(C(=O)N(C)CCN(C(=O)C(C2(O)CCCC2)F)C)cc1Cl 59196,n1(CC)cnc(C(=O)NC2CCC2NC(C2(F)CC2)=O)n1 59197,C12(CNC(C3CCC3)=O)CCCCC1CN(C(c1ccc3c(c1)OCCO3)=O)C2 59198,S(=O)(=O)(c1ccc(NC2CCCC3(CCCCC3)C2)c(C#N)c1)NCC(CC)C 59199,c1(C(N2CCSC(C(C)C)C2)C(=O)NC)oc(C(=O)OC)cc1Br 59200,c1(C(C(=O)NC2CCC2)N(CCC2=CCCCC2)C)cc2cc(Cl)ncc2o1 59201,N1(Cc2c(OC)nsc2)CCN(CC(=O)NCCc2ccc(Cl)s2)CC1 59202,n1(CC(N2C3CC(CNC(C(CC=CC)C)=O)C2CC3)=O)cnc2ccccc12 59203,c1(-c2ccnc(C)c2Cl)cc(Br)c(F)cc1C#N 59204,C(C(CC(C)C)C(=O)NCC(C)(C)C1(O)CCC1)NC(C(CCOC)C)=O 59205,C(=O)(C(O)CN(C)C)N(CC(CC)NC(=O)C(n1cc(C)cn1)C)C 59206,N1(C(Cc2ccc(OC)nc2)=O)CCC(C)C(NC(C2(OC)CCSCC2)=O)C1 59207,CCCCCCC(C)C(=O)N1C2CCC1CC(N(C)C(c1nc(C)oc1C)=O)C2 59208,c1(Cc2nc(CC(C)OC)nn2-c2ccn(C)n2)ccc(Cl)c(Br)c1 59209,N1(C(CC2C(C)C2)=O)CC2CC2(NC(c2ccc(OCC3CC3)nc2)=O)C1 59210,C(C(CC1CCCC1)C(=O)NC1CCC(O)C1)NC(=O)C1CC1CO 59211,c1(C(N2CCC(CNC(C3C(C)OCC3)=O)C2)=O)cnn2ccn(C)c12 59212,C12(C(N(CCCC)C)=O)CCC(n3cc(C4CCCO4)nn3)(CC1)C2 59213,CCS(=O)CC(=O)N(CC(C)CNC(=O)CCCSC(C)(C)C)C 59214,CC1CN(C(=O)Cc2ccnn2C2CCOCC2)CC1NC(=O)Cn1ncnn1 59215,c1(N(C)C)cc(-c2ccc(C(=O)NCC3COCCO3)nn2)cc(C#N)c1 59216,C1CC(C(=O)NC(COC(F)F)CO)N1.C1(CC(=O)OC)CC(OC)C1 59217,S(=O)(=O)(c1cccc(C(=O)NCC2(C)CCC(NC(=O)C(F)CC)C2)c1)NCC 59218,c1(C(=O)NC2CC(CCNC(=O)CN3C(=O)CNC3=O)C2)nnn2c1CCCC2 59219,C(N=c1[nH]c(=N)[nH]c(=NCCS(=O)(=O)c2cnn(C)c2)[nH]1)C1C(C)CSC1 59220,S(=O)(=O)(CCC(F)(F)F)N1CCC(CNC(c2cnc(Cl)cc2I)=O)C1 59221,N1(Cc2cccc(OC)c2F)Cc2ccccc2C1C(=O)N1CCOC(CO)C1 59222,c1(C(=O)NC2CN(C(C3N(CCC)CCCC3)=O)CC2C)cc(C)c(Cl)cn1 59223,c1(CCCC)cc(C(=O)NCC2(NC(=O)C=Cc3cocn3)CCOC2)c(C)o1 59224,c1(OC)ccc2occ(CCNC(=O)NC3CCSC3C)c2c1 59225,C1(C(N(C2CCN(C(C)=O)C2)CC)=O)(C)CCCCC1.C12(C(=O)N)CCC1CC2 59226,C(=O)(CCCS(C)(=O)=O)NC1CCCC(NC(CCCCOC)=O)C1 59227,c1(C(=O)NCCN(C(=O)C(F)(F)CO)CCC)ccc(=O)n2c1COCC2 59228,c1(C(=O)NCCC(C)N(C(Cc2cc(C)no2)=O)C)c(C(C)C)cnn1C 59229,C(C(C(=O)NCC(C)(O)CN(C)C)N(C)C)NC(C(C)NC(=O)CC)=O 59230,N1(C(CS(=O)(=O)NC)=O)CCCC12CCN(C(c1ccccc1COC)=O)C2 59231,C(=O)(CC(F)(F)CC(=O)N1CCN(C)CC1CNC(=O)CC(C)(C)OC)OC 59232,c1(C(N2CC(NC(C(C(C)C)(C)C)=O)C(C(F)(F)F)C2)=O)ccc2nccn2n1 59233,C12(C(=O)NC3C(NC(c4cccc(OC)n4)=O)CCC3)CCCCC(OC)(C1)C2 59234,C1(C(=O)NCCC(CC)(CC)NC(=O)Cc2ccco2)CNC(=O)CC12CCC2 59235,N1(C(C(C)OCCC#C)=O)CCCC(NC(C2(C(C)(F)F)CC2)=O)CC1 59236,C(=O)(CCC(F)(F)F)NC1C=CCN(C(C(CC#C)C2CC2)=O)C1 59237,C1(NC(C2C3(CC3)C23CC3)=O)CCN(C(=O)CN2CCOC2=O)CC(O)C1 59238,N1(C(CN(CCOC)C)=O)C2CCC(C2)C1CNC(=O)Cn1nc(C)oc1=O 59239,C12(CNCC3(N)CCC3)CC3CC(CC(C3)C1)C2 59240,C1(NC(c2nc(CCC)sc2)=O)CN(C(=O)COc2cccnc2)CC(C)(C)C1 59241,Cc1ccc(Br)c(CNC2CC(C)CN(C(c3cc(O)ccc3C)=O)C2)c1F 59242,C(=O)(C1=NOC2COCC12)N1C(C(=O)NCCC2=CCOCC2)C=CC1 59243,Cn1nc(C(N2CCC(C(N3CC(c4ccccc4)C3)=O)C23CC3)=O)cc1C#N 59244,C(=O)(C(C)(C)CNC(C1CC(C)N1C(=O)CCc1cnco1)=O)OC 59245,N1(C(c2cc(CC)c(CC)o2)=O)CC(C2CN(C(=O)C(C)(O)CC)C2)C1 59246,c1(C(=O)NC2CN(C(CC3CC(CC)C3)=O)CC2C)c(C)nn(C(C)(C)C)c1C 59247,C(=O)(C1=NOCC1)NCCC(CNC(C(CSC)OC)=O)O 59248,C(c1ccc(Cl)cc1)=CC(=O)NCC(CN(C(CC(=O)N(C)C)=O)C)(C)C 59249,C(CCCCC(=O)NC(CC1CC1)CO)NC(c1cc(OC)ns1)=O 59250,Cc1cc(C(N2CC(NC(c3cnc(C)n3C)=O)C(C)C2)=O)c2c(C)noc2n1 59251,C1(NC(CCC=C)=O)CN(C(=O)C(C)CN(C)C)CC1OCC 59252,Cn1c(O)nc2cc(C(N3CCC(CCNC(=O)CCCC#N)C3)=O)ccc12 59253,Cc1ccc(C)n1CC(N1CCCC1CCC(N1CCCC(F)C1)=O)=O 59254,C1(C)(CNC(CCOCCOC)=O)CCC(C(=O)N(CCCN(C)C(C)=O)C)O1 59255,c1(N2CC3CC(C)(C)C3C2)nc(=NCCc2cccc(F)c2)[nH]c2c1COCC2 59256,c1(C(=O)NC(CNC(C=CC(C)(C)SC)=O)CCOC)cc2n(n1)CCO2.C(C)(=O)O 59257,C(=O)(C(c1ccccc1)=C(C)C)NC12C(CN(C(CCCOCC)=O)C1)C2 59258,c1(N(CCCN2CCOCC2)Cc2ccc(C)o2)ccc(F)cc1C#N 59259,C1(C(=O)NCCC(=O)NC(C)=O)CC(C)N1C(c1ncn(C)n1)=O 59260,CC(CC(N)=O)C(=O)NC(C)CCN(C)C(c1cc(OC(F)(F)F)ccc1F)=O 59261,Cc1ccc(Cl)cc1-c1cn(CCCNC(=O)CCNC(N)=O)nn1 59262,c1(C(N2C(CC=C)CCCC2)C(=O)NC2CCCCCC2)c(C)cccc1C 59263,N1(C2CCN(C(CCCOCC=C)=O)C2)CCN(C(c2ccc(Br)o2)=O)CC1 59264,C(=O)(C(F)C(C)(F)F)NCC(=O)NCC(F)F.C1C(N(C)C)C(=O)N1 59265,C12(NC(c3nc(C(C)C)oc3)=O)CCCC1CN(C(=O)CN1CC3CC3C1)C2 59266,c1(CC)nccnc1C(=O)NCC(C)(CO)NC(c1c[nH]c(C#N)c1)=O 59267,S(=O)(=O)(c1cccc(F)c1Cl)Nc1ccc(C=C)cc1 59268,c1(C(N2C(CNC(C3(C=C)CCC3)=O)C(C)CCC2)=O)ccc2c(n1)CCCC2 59269,c1(CN2C(C(=O)Nc3c(C(C)=O)cccn3)CC3CC32)c(C)cc(Br)cc1C 59270,c1(C(=O)COCCCSC(F)F)ccc(Br)cc1F 59271,c1(C(N2CC(NC(c3ccco3)=O)C(F)C2)=O)ccc(Cl)c(F)c1F 59272,c1(COC(C)C(=O)N(C)CC2CCS2(=O)=O)cn(CCCC(=O)O)nn1 59273,C(=O)(CC1CCc2ccccc21)NCCC1CN(C(c2c(C)onc2)=O)CC1C 59274,c1(OC(C)C)ncc(C(=O)NC(C)CN(C)C(C2(C)CCCC2)=O)cc1Cl 59275,C(C#Cc1ncccn1)N1CCC(OC(C)(C)C)C1 59276,C(CCC1CCC1)(C(=O)N(C)Cc1ncnn1C)NC(CCn1c(C)ncc1)=O 59277,CCC(C)CC(C(=O)N1CCCC1CNC(N)=O)NC(C1CC(=O)CC(=O)C1)=O 59278,C=C(C)CC(C(=O)N1CCC(C(CC)CC)C1)NC(=O)C(C1CCOCC1)F 59279,c1(CC(=O)NCCOCCCNC(C=C(C)CN2CCCC2)=O)nonc1C 59280,N1(C(c2cc(C)no2)=O)CCCC(CN(C2CN(C3COC3)C2)C)C1 59281,C1(N2CCC(C(=O)OCC)C2)CCCCN(C(c2cccc(C(N)=O)c2)=O)C1=O 59282,C1(C(N2C(CCC(C)(C)NC(C(C=C)C)=O)CCCC2)=O)CCC(=O)N(C)C1 59283,C(=O)(C1=NN(C)C(=O)CC1)N1CCC(N(C(c2c(C)nns2)=O)C)C1 59284,N1(C(C(C=CC)O)=O)CCC(NC(=O)C=Cc2cccc(OC)c2)C(CO)C1 59285,c1(C(N2CCC(C(=O)OC)C2C)=O)n[nH]c2c1CN(C(=O)CCC1OCCO1)C2 59286,N1(C(c2coc(C3CC3)n2)C(=O)NC(C)C)CCCN(C(C)C(=O)N(C)C)CC1 59287,c1(C(=O)NC(CC)CN(C)C(C2CCOC(C)(C)C2)=O)ccc(=O)n2c1CCC2 59288,N1(Cc2c(OC)cccc2Br)CCC2(CC1)CC2C(N1CCOCC1C(C)C)=O 59289,N1(C(CCC2N(C(CCN=[N+]=[N-])=O)CCCC2)=O)CC(C2CCCOC2)C1 59290,Cc1occc1C1CC1C(=O)NCCNC(=O)C(C)n1cccn1 59291,C1(NC(c2c(C)sc(Br)c2)=O)CC2CCCC(C1)N2C(C1CC1(F)F)=O 59292,C12(CNC(C3CCN(C4CCCCC4)C3)=O)CCC1CN(C(=O)CC1CCC1)C2 59293,Cc1ccc(C(=O)NCCC(=O)NC2CCCN(C(C3(CO)CC3)=O)C2)c(O)c1 59294,Cc1nc(C(=O)NC2CCCC2(C)CN(C(=O)C(O)CC(C)C)C)cc(O)n1 59295,N1(C(C2CC(NC(c3c(C)nc[nH]3)=O)C2)=O)CCC2(CCOC2)C1 59296,N1(C(CSCC=C)=O)CCSCC1C(=O)NCCOCCCC 59297,N1(C(c2[nH]cc(C(N)=O)c2)=O)CCN(C(C2CC3CCCCC23)=O)C(CF)C1 59298,C(CS(=O)(=O)c1ccc(C(=O)NC2CC2NC(=O)CCSC)cc1)OC 59299,C(C)(CCC(=O)NCc1nn(C)cc1C)NC(c1n(CC)ccc1)=O 59300,C1(C(=O)NC2C(CC=C)COC2)CCC2(CC2)N1C(=O)CC1(C)CC1 59301,N1(C(C2N(CC)CC2)=O)CC(C)CN(C(c2cnoc2-c2cnccn2)=O)CC1C 59302,CC1=C(C(=O)NCC2CCCN(C(c3coc(C(F)F)n3)=O)C2)COCC1 59303,C1(C(C)NC(c2nc(Cl)cs2)=O)CCCN(C(=O)CC23CCC(CC2)C3)C1 59304,c1(OC)cc(Br)c(NC(=O)C=Cc2ccc(C)cc2OC)c(Br)c1 59305,N1(C(C2C(CC)CCO2)=O)CCC(C(=O)NC(CN(C)C)C(C)(C)C)C12CCC2 59306,C(=O)(C1=CC2C=CC(C1)C2)NC(CCC=C)C(=O)OC 59307,Cc1nc(CC(C)C)c(C(=O)NCC2C3CN(C(=O)Cc4ccnn4C)CC23)s1 59308,C1(C(=O)NCC(c2ncc[nH]2)C)(CNC(=O)CCc2ccco2)CCC1 59309,c1(CC)ncc(C(=O)NC(C2CCCN2C(=O)COCC(N2CCCC2)C)C)s1 59310,N1(C(c2c(C)ocn2)=O)CCC2CN(Cc3ccc(OC4CCCC4)cc3)CC12 59311,c1(C(=O)NCC2(F)CC(NC(C(C)NC(C)=O)=O)C2)ccc(C)c(S(C)(=O)=O)c1 59312,N1(C(CC(C)N(C)C)=O)CCCCC1CC(=O)NCC1COCCO1 59313,c1(C(N2CCc3ccccc3C2)=O)ccc2nnc(S)n2c1 59314,C1(C(N(c2cnn(CCF)c2)C)=O)CN(C(C2CC(F)C2)=O)CCC1(C)C 59315,C1(NC(C=Cc2c(OC)cccc2)=O)C2CCN(C(=O)C3=CCCOC3)CCC12 59316,C1(C(=O)NC2COCC2O)CC(O)C(O)CC1CNC(C1(CO)CCCO1)=O 59317,c1(NC(C2CC(O)(CNC(c3cocn3)=O)C2)=O)ccc(Cl)cc1O 59318,N1(C(c2n(CC)nnc2)=O)CCC2(NC(=O)Cc3cc(Cl)sc3Cl)CC2C1 59319,N(C(=NCC1CCN(C)C1=O)Nc1nc(CSC)cs1)CC1C(OCC)CCC1 59320,C1(NC(CC2CCC(=O)NC2)=O)CCN(C(=O)CC2C=CCCC2)C12CCC2 59321,C#CCCC(C(=O)NC(CCC)C(=O)NC)NC(=O)C(F)C(F)(F)F 59322,N1(C(C2(C)CC=CCC2)=O)CCC2(CC(C(=O)N3CCCCC3C(N)=O)=NO2)C1 59323,C1(C(=O)NCC2(OC)CN(C(c3cc(C)c(C)nn3)=O)C2)CCc2ncsc2C1 59324,c1(C(=O)Nc2cccnc2Cl)cnc2c(-c3c(F)cc(F)cc3F)cccc2c1 59325,C1(=CC(=O)NCC2CCN(C(c3ccc(C(C)=O)[nH]3)=O)C2)CC2CCC(C1)N2C 59326,C1(NC(C2CCN(C)C2)=O)CC2(C1)CC1(CC(NC(=O)CC3(C)CCCO3)C1)C2 59327,C(=O)(C1=Cc2ccccc2C1)NCC(C(=O)NCCC#CCC)(F)C(C)C 59328,N1(C(C2CCCC3(CC3)C2)=O)CCC2(CC1)CN(C(=O)C(O)C1CCC1)C2 59329,c1(OC)cc(-c2ccc(F)cc2F)c(OC)cc1CN1CCCC(CC(C)C)C1 59330,C1(c2ccccc2)(C(=O)NCC2C(NC(C3(C(C)C)CC3)=O)CC2)CC1(C)C 59331,C#Cc1ccc(OCC(N2CCC(NC(c3scc(C)c3Cl)=O)C(C)C2)=O)cc1 59332,C(=O)(C1=CCCOCC1)N1CC(C(C)Nc2nc(C(=O)OC)c(Cl)cn2)OCC1 59333,CC1CCN(C(c2ccnn2CC(F)F)=O)CC1NC(c1cn(C)c(=O)n1C)=O 59334,N1(C(CC=C)=O)CC2(CCN(C(=O)C(C)CC(C)(C)C)CC2)CC1C 59335,N1(CC(=O)NC2CN(C(C3(CO)CCCCO3)=O)CC2O)CCS(=O)(=O)CC1 59336,C1(NC(CC2CCN(C)C2)=O)CCOCC1NC(C1CCS(=O)CC1)=O 59337,c1(C(=O)NCC2(OC)CN(c3cc(C(=O)OC)ncn3)C2)cc(F)ccc1F 59338,C1(C)(C(=O)NC(C#C)C)CCN(C(c2n[nH]cc2I)=O)C1 59339,C1(C(N2CC(C)(NC(C(C)SC)=O)C2)=O)CCCCN1CC(F)F 59340,c1(OCC)ccc(C(C)NC(=O)NC2c3noc2n3)cc1OC.C(=O)OC.OC 59341,C1(OC)C(NC(C2OCCC2CNC(=O)CC2CC2)=O)CC1O 59342,C1(NC(=O)Nc2cn(C(C)C)nc2)COC2(COC2)C1 59343,C1(NC(CCc2c(C)cccn2)=O)C(C)CCN(C(c2ccc(C#N)s2)=O)C1C 59344,C12(C(N3CC(CC)OCCC3)=O)CCC(CC1)N(C(c1ncncc1Cl)=O)C2 59345,c1(C(CC)NC(=O)NCC(C)(CO)c2ccccc2)cnc(C)cn1 59346,C1(C(C)OC(c2ccc(C(CCC)=O)cc2)=O)NC(=O)CNC1=O 59347,CC(C)CC(C(=O)NC1CC1(C)C(F)F)NC(c1cnn[nH]1)=O 59348,O=C1CCCC(CC(=O)NC2CC(NC(=O)CCc3cocn3)C(O)C2)N1 59349,C1(CC(=O)NCC2(CN(C(=O)C(F)CC3CCC3)C)CC2)CC(F)(F)C1 59350,N1(C2C(C)OCC2)CCN(C(c2ccc(CNc3cccnc3N)cc2)=O)CC1 59351,c1(CNC(C2(CNC(C3(C4CCCO4)CC3)=O)CCCC2)=O)ccncc1Br 59352,Cc1nc(C(=O)NCC2CC(C(=O)NC3CNC(=O)C34CC4)CO2)cc(O)n1 59353,c1(C(N2C3CC(CNC(CC(C)C(F)F)=O)(OC3)C2)=O)ccc2nn[nH]c2c1 59354,c1(C(=O)NCCN(c2ccnc(C(CC)C)n2)CCOC)cc2cnccc2[nH]1 59355,Cc1cc(Cl)c(NC(C2CCN(S(=O)(=O)CC3CC3)C2)=O)cc1O 59356,c1(OCC(N2CC(NC(CC(=C)Br)=O)C3C2C3)=O)ccc2c(c1)CCC2=O 59357,N1(C(C(N2CCN(C)CC2)C)=O)CCN(C(c2ccc(N)c(N)n2)=O)C(C)C1 59358,c1(-c2cnc(NC(c3ccc(OC)cc3F)=O)nc2)cnc(C#N)c(F)c1 59359,C1(NC(C(c2ccc(F)c(F)c2)C)=O)CCN(C(c2ccccc2)=O)C1(C)C 59360,C(CC(=O)N1CC2(CC(O)C2)C1)(C(F)(F)F)NC(CCC=C(C)C)=O 59361,C1(N(C)C(c2cnc(S)[nH]2)=O)CCCN(C(c2cc(O)n(C)n2)=O)C1 59362,C12(NC(c3cn(C=C)nc3)=O)CCC(C(N3CC4CCC3C4)=O)(CC1)CC2 59363,N1(C(c2ccc(OC)nn2)=O)CC(C)C(C)(C(=O)NC2(C)CCCCCC2)C1 59364,C12(CNC(C(CC)(C)C#N)=O)CC(NC(c3cc(C)oc3C)=O)(C1)C1(CCC1)O2 59365,C(=O)(C=C1SCC(=O)N1C)N(C1CCCC(NC(COCC#C)=O)C1)C 59366,C1(C(N2CC(c3c(CNCC)nco3)C2)=O)(NC(COCC#C)=O)CCCCC1 59367,C12(CONC(c3cn(CCNC(=O)OC(C)(C)C)nc3)=O)CCC(CO1)C2 59368,CC1CCc2c(C(N3CC(C)(C)CC3CNC(=O)CC3CC34CC4)=O)csc2C1 59369,C1(CCC)CN(C(=O)CC(C)COC)CCN1C(c1cn(C)nn1)=O 59370,c1(OC)cc(C(N2CC(NC(=O)CCc3n[nH]c(=N)s3)CC(O)C2)=O)cc(C)c1 59371,C=CCCCC(F)F.c1(CCNC)ccc(F)c(C)c1 59372,N1(C(c2n(CC)cc(Cl)c2)=O)CCCC(O)(CNC(C2C(C)(C)C2(F)F)=O)CC1 59373,c1(NC(C2(C#N)CCNC2)=O)cccc2c1OCCC(=O)N2 59374,N1(CC)N=C(C(=O)NCC2C=CC(NC(c3ncc(Cl)cc3Cl)=O)C2)CCC1=O 59375,C(CCCCC(=O)N1CCN(C(c2cc(C(F)(F)F)c[nH]2)=O)C(C)C1)=CC 59376,N1(C(C(C)P(C)(C)=O)=O)CCOC2(C1)CN(C(C1CC13CC(O)C3)=O)C2 59377,C1(NC(C2Cc3nncn3C2)=O)CN(C(c2ccsc2Cl)=O)CC2(CC2)C1 59378,c1(C(C(=O)NCC2CCOC2)N(C)Cc2n(CC)cnn2)ccc(F)c(C)c1Cl 59379,C1(OC)CCN(C(c2cc(CF)on2)=O)C1CNC(=O)OC(C)(C)C 59380,C(=O)(C1CCCc2sc(=N)[nH]c21)NCC(C)CNC(=O)C(F)(F)c1cccnc1 59381,C(C(=O)NCC1(CNC(=O)CCNC(=O)C(C)(C)C)CC1(F)F)(C(C)C)SC 59382,Cc1cc(Cl)c(C(=O)NCC2CCCN(C(=O)NCc3nc(C)c(C)s3)C2)s1 59383,c1(C(N2C3CCN(C(c4c(CC)nc[nH]4)=O)CC3C2)=O)cn2ccc(F)cc2n1 59384,c1(C(N2CCN(C(C3CCN3CC(F)(F)F)=O)CC2)=O)cc(F)cc(Cl)c1 59385,c1(C(=O)NC(C)CNC(C2CC(n3ccnn3)C2)=O)[nH]nnc1-c1ccccc1 59386,C(=O)(CCC(C)CC)N1CCC(CC=C)(C(N2CC(CS(C)=O)C2)=O)C1 59387,C1(CC(=O)N(C(C)CNC(c2c[nH]c(C(F)(F)F)c2)=O)C)CCCC(C2CC2)O1 59388,O(P(C)(=O)CNC(C1CC=CCN1C(=O)CC1CCCOCC1)=O)CC 59389,CCCCCCCCOCC(=O)NCC1CCCN1C(c1cc(N)nc(Cl)c1)=O 59390,N1(C(CC(SC)Cc2cccc(C)c2)=O)CCCN(CCNC(=O)C2CC2)CC1 59391,C12(CNC(c3c(C)nsc3)=O)CCCC1N(C(=O)C(C)C1CCOC1)CCC2 59392,C1(CN(C(C(C=CC)O)=O)C)CN(C(=O)CC(CC)c2ccccc2)CCO1 59393,N1(C(C(=O)NC2CC(C(=O)OC)C2)CCC2CC2C)CCCC2(CCCOC2)C1 59394,c1(C(N(CCNC(C(CC)(CC)OC)=O)CC2CC2)=O)cnc2[nH]nnc2c1 59395,C1(CNC(c2nc(COC)oc2)=O)CCN(C(C2CC3(CC3)C2)=O)CC1O 59396,C1(C(=O)Nc2cn(CCC#C)nc2)CSCCN1C(c1cc(CC)[nH]n1)=O 59397,C(=O)(C(C(C)(C)C)NC(N)=O)NC1C(CNC(c2c(C)cno2)=O)C1 59398,CCC(C(=O)OC)C(=O)NC1CC2(C1)CN(C(=O)CSc1nnnn1C1CC1)C2 59399,Cc1ccc(C(=O)NCC2CN(C(C3CCC3C(C)(C)C)=O)CCO2)c(F)c1Cl 59400,C(=O)(CCCCNC(C1C(NC(=O)CC2CC(C)(C)CO2)C1(C)C)=O)OCC 59401,c1(C(=O)NC2CCC(NC(c3ccnn3CC3CC3)=O)C2)ccn2ccnc2c1 59402,C1(CN(C(C2CC(C(F)F)(OC)C2)=O)C)CCN(C(C2CC(O)C2)=O)CC1 59403,C(N=c1nc(OC)c2ccccc2[nH]1)C1(CNC(CS(CC)=O)=O)CC1 59404,C1(C(=O)NC2CC(OC)CN(C(=O)C(C)(C)C#N)C2)CS(=O)(=O)CC(=O)N1 59405,N1(C(C=CCOC)=O)CC(O)CC1C(N1CCCC1C1(C)CC1)=O 59406,c12ccccc1CNC2.C1(CNC(C2CC(c3nn[nH]n3)C2)=O)CCCCO1 59407,N1(C(c2cnc(CC)o2)=O)CCC(CC)C1CNC(c1ccsn1)=O 59408,C1(Br)(C(=O)NCCOCCN(C(C2(C)C(C)C2)=O)C)CC1(F)F 59409,N1(C(c2cn(C)nc2Cl)=O)CC2CC(C1)C(CO)C2NC(c1cccc[n+]1[O-])=O 59410,N1(C(COC)=O)CCC(C)(C(=O)OCC(C(C)C)N2CCCC2=O)CC1=O 59411,c1(C(CC)CN(C2CC2)C(c2nc[nH]n2)C)ccccc1 59412,CCCC(C)CC(=O)N1CC(CCO)(NC(C2COCCN2CC)=O)C1 59413,CC1(NC(C2CN(C(N)=O)C2)=O)CCN(C(=O)C2=CCCS2)CC1 59414,N1(C(C(CC)F)=O)CCC(N(C)C(c2ccn(C3CCC3)n2)=O)C2(CC2)C1 59415,CC(C)CC(O)C(=O)NC1CN(C(c2cccc(SC(F)(F)F)n2)=O)CC1C 59416,CC1CC(N=c2c(Br)c[nH]cc2[N+](=O)[O-])CN1C(c1nc[nH]c2nccc1-2)=O 59417,C(CC(C)CCNC(c1cc(C(C)(C)C)no1)=O)NC(CCCOCC)=O 59418,c1(OC)ccc(C(=O)NC2CCCC2NC(=O)CC2CCOCC2OC)c(OC)c1 59419,C(=O)(C(CCOCC)NC(=O)C(C)C1CCCC1)N(CC=C)CCOC 59420,CC1(C)CCCC(CS(N2CCC(N3CCCCCC3)CC2)(=O)=O)O1 59421,c1(C(=O)NCC(C)(C2CC2)NC(CC(C)OC)=O)c(Cl)c2ccccc2n1C 59422,C1(C(N2C(C3CN(C(c4c(C(C)C)ccs4)=O)C3)CCC2)=O)CCC(CO)CC1 59423,C(=O)(C(C)CC(F)F)NC1C(NC(CCc2cccc(C)c2)=O)CCCC1 59424,c1(C(=O)OCC)cccc(S(=O)(=O)NC(c2cnsc2)C)c1 59425,C(=O)(C#CC(C)(C)C)NCc1c(C(=O)NCC2(O)CCN(C)C2)nco1 59426,C(=O)(C(C)(C)CC#N)N1C(C)CC(CNC(=O)C=CCOCc2ccccc2)C1 59427,N1(C(C2(C(C)C)COC2)=O)CCOC2(CCS(=N)(=O)CC2)C1 59428,C1(C2(O)CCOC2)(C(N2CCC(F)(CNC(c3ncc[nH]c3=O)=O)CC2)=O)CC1 59429,n1(CC(=O)NC2CC(CNC(=O)C(O)C3CC3)C2)cc(Br)cn1 59430,c1(C(=O)OC)cc(CO)[nH]c(=NCC(CC(C)O)c2ccccc2)n1 59431,Cc1nc(C2CCCO2)sc1C(=O)N(C)CC1CCN(C(=O)CC2(O)CCC2)C1 59432,C1(c2nnnn2C)(NC(c2cccc(N(C)C)c2)CC)CCN(C2CC2)CC1 59433,n1(CC)cccc1C(=O)NCCOCCN.c1(S)ccccc1.C1(=O)CC2C1C2 59434,C1(NC(=O)NCc2nc(C(C)C)on2)CCCC(O)CC1 59435,C1(C(N2CC(CC(=O)OCC)C2)=O)C(C)OCCN1C(c1c[nH]c(=NC)o1)=O 59436,C1(CNC(CC)=O)CCCN(C2CCc3ccc(Cl)cc32)C1 59437,CC1(CCCO)CCCN1C(c1ccoc1CNC(c1cnn(C2CC2)c1)=O)=O 59438,C1(N(C(=O)CCc2cnn(C)c2C)CC)CCN(C(C2CC(C)OC2=O)=O)CC1 59439,C1(NC(c2sc(N(C)C)nc2C)c2n(CCCC)nnn2)CC(O)CC(C)(C)C1 59440,C(=O)(CC(C)(C)CNC(c1ccoc1Cl)=O)NC(c1nccs1)CC 59441,C1(c2ncc(C(=O)OC)s2)CCN(C(=O)N(C)C)CC1.C(CCO)SCO 59442,C(=O)(C(C)C(C)COC)NCC#CC(=O)NC(CC#C)C 59443,N1(C(=O)CCc2cscn2)CC(NC(C23CC(c4ccccc4)C2C3)=O)C(O)C1 59444,c1(C(=O)NCCC2(CNC(CC(COC)O)=O)CC2)cc(C)cc(Cl)n1 59445,C(CCCCC(=O)N1CCCC(CC(=O)NC(C)(C)CCCO)CC1)=CC 59446,C1(NC(C(CC)(C)OC)=O)CC=C(C(=O)NCC(C)(C)CO)C1 59447,N1(C(C2(CC=C)COC2)=O)CCN(CC(C)NC(=O)C(C)CC=CC)CC1 59448,C1(C(=O)NCC(C)N(C(c2sc(C)c(Br)n2)=O)C)CNC(=O)C(C)(C)C1 59449,c1(C(=O)NCC(CC)NC(=O)CCc2ccnn2C)cn(CCC(C)C)nn1 59450,N1(C(C(C)CC(C)(C)C)=O)CCC2CCN(C(=O)Cc3cc[nH]n3)C2C1 59451,C1(NC(CC2C(C)(C)C(O)C2)=O)CCN(C(c2cc[n+]([O-])cc2)=O)C12CCCC2 59452,c1(-c2cn(C)nc2)cccc(NC(=O)NC2CCN(CC3CC3)C2)c1 59453,C(C)(CNC(=O)CC1CCOCC1)(C(C)C)NC(C(c1ccccc1F)C)=O 59454,c1(C(=O)NCC(CCC)NC(=O)Cc2cc(C)nn2C)ccc2ncnn2n1 59455,c1(NC(CC2CN(C(CC(C)=C(C)C)=O)CC23CC3)=O)cccc2occc12 59456,CC1(C)CCN(C(C23CC2COC3(C)C)=O)CC1CNC(=O)C=CBr 59457,C1(C(N(C(C(C)C)CO)C)=O)(CO)CCN(C(c2ccc(CO)s2)=O)C1 59458,c1(C(=O)OC)ncc(NC2(CNC(=O)CC(C)(O)c3ccccc3)CCCC2)nc1C 59459,C(=O)(C1=CCCN(C(=O)Cc2cc(C)cs2)C1)NCCCCC#CC 59460,Cc1[nH]c(C#N)cc1C(=O)NC1CCCCN(C(=O)CC2CC3CCC2CC3)C1 59461,CCCCC(C)C(=O)NCCOC1CN(C(c2ccn(C)c2)=O)C1 59462,CCCCC(C(=O)NCCN1CC(CF)C1)NC(C1CCOC(C)(C)C1)=O 59463,C12(NC(c3cnc(C4CC4)o3)=O)CCCC1N(C(c1ncccn1)=O)CCC2 59464,C1(C(=O)NC(c2nccs2)CC)CCCCC1(C)NC(=O)C=CC=C(C)C 59465,c1(CC(=O)NCCC(C)(C)NC(=O)CO)ccnc(-c2nn[nH]n2)c1 59466,c1(C(=O)NC2CC(C(=O)Nc3c(OC)nc(Br)cn3)C2)ccc(C#N)cc1Cl 59467,Cc1ccc2c(c1)N(C(=O)C(CNC(=O)Cc1ccc(O)cn1)C(C)C)CC2 59468,CC(C)CCCC(=O)N1CCC(C=CC(=O)NC(CO)CC(C)C)CC1 59469,C1(C(=O)NCCc2nc(CC)on2)CN(C(c2ccccn2)=O)CCN1 59470,c1(OC)cc(Cl)ncc1C(N1CCN(C(c2oncc2C)=O)CC1CC#N)=O 59471,Cc1ncn(C)c1C(=O)NC(C)CN(C)C(c1cnn(C(C)(C)C)c1)=O 59472,n1(C(C)(C)C)nccc1C(=O)NC1CCCC1NC(C1(N(C)C)CC1)=O 59473,C1(NC(c2cc(CO)[nH]n2)=O)CCN(C(c2ccccn2)=O)C12CCCC2 59474,c1(OC)cnc(C(N2CCC(N(C(=O)C(c3ccc(F)cc3)F)C)C2)=O)c(F)c1 59475,c1(C(N2CCCCCC2CCO)=O)cnc2c(Br)cccn12 59476,N1(C(C=CC2N(C)CCC2)=O)CCC(NC(=O)Cn2ccnn2)C2(CCC2)C1 59477,C1(C(N(C)CCNC(c2n[nH]cc2Cl)=O)=O)C2CC3C(C2)C13 59478,c1(OC)cc(NC(C2CCCC(NC(c3cnnc(O)c3)=O)CC2)=O)ccc1O 59479,C(=O)(C(CCC(C)C)OC)N1CCC(CNC(C2(C(CC)=O)CC2)=O)(COC)CC1 59480,C(CN(C)C(C1CC1F)=O)(CO)(CO)NC(C(c1cccs1)SC)=O 59481,Cc1cc(-c2cn(C3CC(C(=O)Nc4ncccc4F)C3)nn2)cc(F)c1 59482,Cc1nc(Cl)[nH]c(=NC2CN(C(c3ccc(N(C)C)cn3)=O)CC23CCC3)c1F 59483,C(=O)(C(=O)C(C)(C)C)NC1(CNC(c2n[nH]c(C)c2C)=O)CC1 59484,N1(C(c2c(C)noc2)=O)CCCN(CCCCNC(C2CC3CCC2O3)=O)CC1 59485,c1(C(=O)NC2CC(N(C(c3sc(C)c(Br)c3)=O)C)C2)cccc(F)c1N 59486,CN=c1[nH]nc(CC(=O)N(C)CCNC(C2(CC(C)C)CCCC2)=O)s1 59487,N1(C(C2(COC)CC2)=O)CCCC(C(C)NC(=O)C(F)=CC2CC2)C1 59488,C1(N(C(=O)CC2(CO)CC2)CC)CCCN(C(=O)C=Cc2ccncc2)CC1 59489,N1(CC(=O)NC(C(=O)Nc2c(OC)nsc2)C)CCN(C)CC1 59490,c1(CC(CNC(COC2CN(C(C)=O)C2)=O)NC(c2cnc[nH]2)=O)ccccc1 59491,c1(N)[nH]c(=NCC2(C)CSC(C)=N2)nc2ncn(CC)c12.CCCCCCO 59492,c1(C(N2CC(NC(CCC(C)(C)OC)=O)CC2(C)C)=O)ccc2c(c1)OCCC2 59493,Cc1cc(C(=O)NC(CNC(c2c(C3CCC3)cnn2C)=O)CO)cc(F)c1 59494,n1(CC(=O)NC(C2CCOC2)CNC(C2(CO)CC2)=O)ncc(O)nc1=O 59495,C1(S(N)(=O)=O)(C(=O)NCC(C)(C)Cn2cc(C3CCOCC3)nn2)CCC1 59496,CCC(C)(C)C(O)C(=O)NCC1(OC)CN(C(=O)C(C)(F)c2ccccc2)C1 59497,C(C(C)(C)C(=O)N1CCC(CNC(c2cnc(C(C)(C)C)s2)=O)C1)OCC 59498,CC1(F)CC(C(=O)NCC(CNC(=O)CNC=O)CO)C1 59499,N1(C(CCN(C)CC)=O)CC2CN(C(=O)C=Cc3cccnc3)CC2(C)C1 59500,C1(CC(=O)NC2C(CCC)CN(C(=O)COCP(C)(C)=O)C2)CC(C)(C)CCO1 59501,c1(C(N2CCC(N(C(CN(C)CC)=O)CCO)C2)=O)ccc(C(C)(C)C)cc1C 59502,N1(C(C(CC(C)(C)C)F)=O)CCC2C(CCN2C(c2ccnn2CCF)=O)C1 59503,C(=O)(CCCOC1CC(NC(=O)CNC(C2CC2C)=O)C1)OC 59504,C(=O)(C(C)C(F)(F)C(F)F)N(CCNC(c1coc(C2CC2)n1)=O)CC 59505,C1(C(N2C(CCNC(C(C)(C)CO)=O)CCC2)=O)Cc2ccc(Cl)cc2C(=O)O1 59506,CC1(C(=O)NCC2(CO)CCN(C(=O)COc3cccnc3)C2)CCC(O)CC1 59507,Cn1cnc2c1CCN(C(=O)C(F)C(F)(F)F)C21CCN(C(=O)CC2(C)CC2)C1 59508,c1(C(=O)NC2(C3CCCN3C(=O)C(F)=C3CCCC3)CC2)cc(C(F)F)c[nH]1 59509,C1(C(=O)NC(CC2CCC3(C(C=C)C3)CC(=O)N2)C)CCOC2(CCCCC2)C1 59510,Cc1[nH]nc2cc(NC(=O)Cc3cccc4c3OCCC4)ccc12 59511,C12(CC(=O)NCC3CCCN(C(C(CC#C)C)=O)CC3)CCC(CC1)C2(C)C 59512,C1(C(=O)NCC2(C(F)F)CCN(C(Cc3c(C)ccs3)=O)C2)CCC2(CCC2)C1 59513,C1(N(C)C(C)C)CCN(C(=O)CC(=O)Nc2ncc(C(=O)OCC)s2)CC1 59514,c1(C(N2CC(O)(CNC(C(CC)(C)C#N)=O)C2)=O)cn2ccc(C)cc2n1 59515,c1(C(N2CCC(CN(C(CCC=CC)=O)C)C2)=O)csc(Br)c1C 59516,c1(C(=O)NC(C(C)NC(C(CC)(C)CC)=O)C)cccc(F)c1C#N 59517,C=CCCCC(C(=O)N(CCCC(CC)CC)C)NC(=O)C(OC)OC 59518,c1(COC)ccc(C(=O)NC2CCCC(C(N3CCSCC3)=O)C2)cc1 59519,C1(C)(C(N2CC(CN(C(C(CC)(C)C)=O)C)OCC2)=O)CC(=O)N(C)C1 59520,CN1CCC(C(=O)NCC2CC2NC(C2CC(NS(C)(=O)=O)C2)=O)C1=O 59521,C1(CC)CN(C(c2cc(Cl)ncc2F)C(=O)NC(C)(C)C)CC(=O)N1 59522,N1(C(c2ccc(C)o2)=O)CCC(CNC(c2nc(Cl)cs2)=O)C(O)C1 59523,CC1(C)CCCC(O)(CNC(=O)Cn2cc(C3(C)CCCO3)nn2)CC1 59524,C(=O)(C(CO)C(F)(F)F)N1C(C(=O)NCc2n(CCC)cnc2)CCOCC1 59525,C=CC(C)(C)CC(=O)NC1CC(F)(F)CC1NC(=O)Cc1cccc(F)c1F 59526,C1(CC(N2CCC(c3cnco3)CC2)=O)CNCCS1(=O)=O 59527,C1(C(=O)NC2CCN(C(c3cc(C(C)=O)[nH]n3)=O)C2)CC12CC(C)(C)C2 59528,C(C(CNC(c1cncc(N)n1)=O)C(F)(F)F)NC(c1c(C)ccs1)=O 59529,c1(C(=O)NCCNC(c2ccc(C)cc2Cl)=O)cc(Br)cc2c1OCC2 59530,c1(CC(=O)NC(C2CCN(C(C3CCC3(C)C)=O)C2)C)coc2ccccc12 59531,Cc1nn(CCO)cc1C(=O)N(C)CC1CCCN1C(c1ccccn1)=O 59532,CCC(C)C(C)C(=O)N(C(C)CNC(=O)Cc1csc(C(=O)OC)c1)C 59533,CC1CN(C(C2CC2c2ccnn2C)=O)CC1NC(c1cnsn1)=O 59534,Cc1cc(C(=O)N(CCN(C(=O)C(N2C(C)CCC2C)C)C)C(C)C)cc(C)n1 59535,C12(C(N(C3CCCCC3)CCNC(c3c(C)noc3)=O)=O)CSCC1C2(F)F 59536,CC1CN(C(=O)CCCCCN(C)C)CC(C)C1NC(=O)Cn1cccnc1=O 59537,O=C1NCC2(CCN(C(C3C=CCN(C(=O)C(O)CC(F)(F)F)C3)=O)C2)O1 59538,C1(C(=O)NC(COC(C)=O)CO)(COC)C=CCN1C(=O)C(n1ccnc1C)C 59539,CC1(C)CN(C(=O)CC(CNC(C2(C)CC3CC3C2)=O)C2CCC2)CCCO1 59540,C1(C(=O)NC2CC3CN(c4c(C)cncn4)CC32)CCc2ccc(F)cc2O1 59541,C1(C(=O)OC)COCC1NC(=O)C(CN(C)C)NC(=O)C(C)=C(C)C 59542,Cc1cc(S(N)(=O)=O)cc(C(=O)NOCC2C(C)CC2C)c1C 59543,C(=O)(CCC(F)(F)F)N(C)CC1CCCN1C(C1CC(CC(F)F)C1)=O 59544,C12(C(N3CCCC(C)C3CNC(=O)Cn3cc[n+](C)c3)=O)CC=CCN1CCC2 59545,N1(CC(=O)NC(=O)NCC)CCCN(C(C2CCCC(OC)C2)=O)CC1 59546,Cn1nc(I)c2c1CN(N(CC1CCC1)Cc1ccncc1)CC2 59547,c1(C(=O)NCCN(C(=O)CCc2ncc(C(C)(C)C)o2)CC)cc(SC)oc1C 59548,C(C)(CCC(=O)Nc1ccc(C(=O)NOCC=CCl)o1)OCC 59549,c1(NC(c2c(CCCN)ccs2)=O)nccc(CCCN2CCCC2)n1 59550,c1(C(=O)NC2CCCCCN(C(C(CC)(C)CO)=O)C2)cc(F)c(Cl)c(N)c1Cl 59551,CCC(C)CC(C)C(=O)NCC1CCN1Cc1ccccc1Cl 59552,C1(NC(C(C(C)C)C#N)=O)CC2CCC1C(NC(C1(C(=O)N(C)C)CC1)=O)C2 59553,C12(C(=O)NCCC(C)NC(C3(C#C)CCCC3)=O)CCC(C)(C(=O)O1)C2(C)C 59554,C1(CNC(C(CC=C)NC(c2cc(O)n(C)n2)=O)=O)CC2(CCC2O)C1 59555,c1(C(N2CCCC(N(C(C(C)=C(C)C)=O)C)C2)=O)ccc2cnnc(O)c2c1 59556,C=CC(C)(C)C(=O)NCC(C1CCCN1C(=O)CCN1CCC1)(C)C 59557,N1(C(=O)CC2CC(F)CN2C(=O)Cc2nc(Cl)cs2)Cc2cccc(F)c2C1 59558,c1(CC)ccc(C(N2CCCC(NC(=O)CC3CCC(C)(C)O3)CC2)=O)cc1F 59559,C(=O)(CCCCC(F)(F)F)NCC(C(C)C)NC(CC(CC)C)=O 59560,c1(C(N2CCC(NC(CC(CC)O)=O)CC2C)=O)c(C)nn2cccnc12 59561,N1(C=O)CCC2CCC(C1)N2c1nnc(C2CCCC2)s1.c1(C(C)=O)cccnn1 59562,c1(CC)nc(C)c(NC(=O)CNC(C)(CNC(=O)OC(=O)C(C)(C)C)C(C)C)s1 59563,C1(C)(c2cn(CC3(C)CCC3)nn2)COCCN1C(=O)CC1CC(F)(F)CO1 59564,N1(C(c2ccon2)=O)CCC2(CCCN2C(c2ccn(CC(F)F)n2)=O)CC1 59565,N1(C(c2cc(OC)cc(F)c2)C(=O)NCC(F)F)CC2CCCCCC2(C#N)C1 59566,c1(C(N(C(CNC(c2cnsn2)=O)C2CC2)C)=O)ccc(=O)n2c1COCC2 59567,C(CCS(C)(=O)=O)(C(N)=O)NC(C(C)CCO)=O 59568,Cc1c(C(=O)NC2CCC(CNC(c3n[nH]cc3C(C)C)=O)C2)sc2nccn12 59569,Cc1cn2cc(CC(N3CCC(O)(C(C)NC(=O)C(C)C)CC3)=O)nc2s1 59570,C(N=c1[nH]nc(O)s1)C1CCCN(C(c2c(C)nn(CCO)c2)=O)C1 59571,N1(C(c2c(CCC)nns2)=O)CCCC(C)C1CCNC(c1ccnc(S)c1)=O 59572,N1(C(C(N)c2ccco2)=O)CC2COCC2(C(N2CC(O)C(F)C2)=O)C1 59573,C(CCN=C(NCC(=C1CCCC1)F)NCC1(C)CCS(=O)(=O)N1C)OCC 59574,N1(C(C(CC2CCC2)NC(COC(CC)(C)C)=O)=O)CCCN(C2CC2)CC1 59575,c1(CC)cc(C(=O)NCC(C)(C)CN(C)C(C2(CSC)CCOCC2)=O)ncn1 59576,c1(C(N2CCCC(O)(CNC(C3C=CC=CC=C3)=O)C2)=O)ccc2nncn2c1 59577,C1(N(C)C(c2cn(C)nc2O)=O)CC2CCC(C1)N2C(=O)C(N)=O 59578,N1(CC(c2cccc(N(CC(=O)O)CCOC)c2)=O)CC2CCC(CC2)C1 59579,C1(CC(=O)NCC2N(C(C(c3cnn(C)c3)C)=O)CC2)CC2(CC2)CO1 59580,c1(CN(C(Cn2c(C)ncc2)C)C=O)cccc(Cl)n1 59581,C1(COCCO)(NCC2CCOCO2)CCCSC1 59582,c1(C(N(C)CCNC(=O)CNc2cc(F)ccc2F)=O)occ2c1CCCC2 59583,N1(C(C2CC(=O)NC(=O)N2)=O)CC2(NC(=O)C3CC3)CCCC2(F)C1 59584,N1(C(COCCSC)=O)CCCN(C(c2cccc(F)c2N)=O)C(C)C1 59585,Cc1nc2ncnn2cc1C(=O)N(CC(O)CN(C(=O)CO)C)C 59586,c1(OC)cc(OC)c(NC(C2CC(F)CN2C(c2cccc(O)c2)=O)=O)cc1Cl 59587,c1(C(CC(=O)NCC2CCCN2C(C2(C3CC3)CC2)=O)O)ccc(Cl)cc1 59588,c1(C(N2CCCC(CNC(c3cccc(C)c3I)=O)C2)=O)cnc2snnc2c1 59589,c1(C(=O)NC2CC(C)(NC(CC3CCCC(C)(C)C3)=O)C2)ccc2nnnn2c1 59590,N1(C(C(C)(C)OC)=O)CCC(C)(CCNC(C2CC2C2CC2)=O)C1 59591,C(=O)(CCCCCc1ccccc1)NC1C(CNC(c2ccc(SC)s2)=O)C1 59592,CC1CC(=O)NC1C(=O)NCCOCCN(C)C(c1coc(C(F)F)n1)=O 59593,c1(C(C(=O)NC2(CS(N)(=O)=O)CCC2)C2CCCO2)ccc(Br)cc1 59594,c1(N2CCC3(C(C(=O)Nc4cc(N(C)C)cc(F)c4)C3)C2)ncnc2occc12 59595,Cc1nc(C)n(CC(=O)NC(c2ccc(F)cc2)CNC(=O)C=CC(F)(F)F)n1 59596,c1(OC)ccccc1OCCN(C(=O)NC)C(c1ccccn1)c1nncs1.SC 59597,c1(C(=O)NCCC2N(CC(=O)NCC(F)(F)F)CCC2)cc2ccccn2n1 59598,c1(CC)cc(C(=O)NCCCCC(C)NC(=O)CCCc2ccccn2)ccn1 59599,N1(C(C(CNC(CC(CC)(C)C)=O)O)=O)CCN2CC(C)CC2C1 59600,N1(C(Cn2nnc(C3(C)C(C)OCC3)n2)=O)CCC(CO)C(F)C1 59601,CCCCC(C(=O)N1CC(C)C1C(=O)NCCOCCOC)N(C)C 59602,c1(C(N2CCC(NC(N)=O)CC2)C(=O)NCC(=C)C)cc(-c2cccs2)oc1C 59603,CC1=NOC(C(N2CC(C)(OCC(=O)NC(C3CC=CCC3)CO)C2)=O)C1 59604,C(=O)(CCCN=[N+]=[N-])NC1CCC(C(=O)OC(C)(C)C)C1.C12CCC1CC(=O)N2 59605,Cc1ccc(C)c(C(N2CC(O)CCC2C(=O)NCCCSC(F)F)=O)n1 59606,c1(C(N)=O)ccc(N2CCC(NC(c3nccc(Cl)c3O)=O)C2)c([N+](=O)[O-])c1 59607,C(=O)(CCCCC1CC1)N(C1CCN(C(=O)CC2C(=O)NN=C2C)CC1)CC 59608,C1(C(=O)NCC(C)N(C)C(C2CCCN2c2cnccn2)=O)CCCC12CC2 59609,c1(C(N2CCC(OC)(CNC(=O)C(C)c3ccco3)C2)=O)ccc(F)c(F)c1N 59610,C(=O)(C#CC1CCCC1)NC(CC)CNC(=O)C(C1CCOCC1)OC 59611,c1(OCC)ccc(CC(=O)NC2CC(F)(CNC(=O)CC3CS(=O)(=O)C3)C2)cc1 59612,CC1(C)CCCC(C(=O)NC2CCN(CCCNC(=O)Cc3ccon3)C2)C1 59613,c1(CC(=O)NC2C(NC(c3c(CC)con3)=O)CC2)ccc(C)cc1F 59614,C(=O)(C1OCCn2ccnc21)NCC(CNC(c1c(NC)ccc(F)c1)=O)CO 59615,C=C(Cl)CN=C(NCC1(C)CCCCCCC1)NC1CCC1C 59616,CC1ON=C(C(=O)N2CCN(C(=O)CS(=O)(=O)N(C)C)CC2CO)C1C 59617,CCCCCCc1ccc(C(=O)NCC2CCN(C(C3CCS3(=O)=O)=O)C2)s1 59618,CC1CN(C)CC1C(N1CC(C)(NC(C2CCN(C(=O)N(C)C)CC2)=O)C1)=O 59619,CCC(CC(=O)N1C2CCC1CC(CNC(C1CCOC1)=O)C2)C(C)C 59620,N1(CC)N=C(C(=O)NCC2CC(O)(CNC(=O)Cn3nccc3C)C2)CCC1=O 59621,Cc1ccc(C(=O)NCC2C(C)CCN2C(=O)CCc2ccnc(Cl)c2)n1C 59622,N1(C(CN(C)C(N)=O)=O)CC(CO)C2(C1)CN(C(c1cccc(=O)n1C)=O)C2 59623,c1(OC)c(F)ccc(NC(=O)C(C)N(S(C)(=O)=O)C)c1F 59624,Cc1ccc(O)cc1C(=O)NCc1nocc1C(=O)Nc1ccc(O)c(Cl)c1 59625,Cc1nc2cccc(C(=O)Nc3[nH]nnc3C3CCN(C(=O)OC(C)(C)C)C3)c2s1 59626,C1(NC(C(c2ccn(C)n2)C)=O)CC=C(C(=O)Nn2cncn2)C1 59627,c1(CNC(COCC(=C)C)=O)occc1C(=O)NC1CC=CCC1 59628,C(=O)(C1OCCc2ccccc21)NC(c1cn(CCOC)nn1)(C)C 59629,C1(CNC(c2c(NC)cccc2)=O)CN(C(c2ccc([N+](=O)[O-])o2)=O)CC1(C)C 59630,CCCC(C(=O)NCc1cccc(CNC(C2(C)C=CCC2)=O)c1)OCC 59631,c1(CC(C)C)ccc(C(N2CCCC2CN(C)C(C2CNC(=O)N2)=O)=O)s1 59632,Cc1cc(Cl)ccc1C(=O)NC(C)C(C)NC(=O)C(C)(C)C 59633,C(C)(C(CC(=O)N(CCO)CCN(C)C)NC(C1CC2COCC2C1)=O)OC 59634,C1(C)(C(N(CCOC)CCF)=O)C=CCN1C(C1CCOCC1OC)=O 59635,N1(C(c2cc(C(C)=O)sc2)=O)CCCC2(CCN(C(C3CN(C(C)C)C3)=O)C2)C1 59636,c1(OC)ncc(-c2noc(-c3ccc(OCC(F)F)cc3F)n2)c(C)n1 59637,c1(N2C(=O)CC(C(=O)NC3CCC(O)(C(F)(F)F)CC3)C2)cc2ccccc2o1 59638,C1(CNC(c2c(CC)con2)=O)(COC)CCN(C(C2CC(C)CO2)=O)CC1 59639,CCCC(F)(F)C(=O)N(CC(CC)NC(=O)C(O)CN(C)C)CC 59640,c1(OCC)cnccc1C(=O)NC(CO)C(C)NC(=O)COc1ccc(C)cc1 59641,C(CCC(=O)NCC(CO)NC(c1cnc(C2OCCO2)s1)=O)NC(N)=O 59642,CC1CC(C(=O)NCC2(C)CCOCC2)CN(C(=O)COCCCN(C)C)C1 59643,C(=O)(C1=CC2C=CC(C1)C2)NCCC(C)NC(c1c(OC)c(C)sc1)=O 59644,N1(C(C(C)N2CCC2)=O)CCCC2(CNC(c3cccnc3Cl)=O)CCCC12 59645,CCCC(C)CC(=O)N(C(C)C(=O)NOCC1CCC1)C 59646,c1(C(=O)OCCC2CCC(F)(F)CC2)cc(C2CC2)nc2ccnn12 59647,C=CC1CN(C(C2CN(C(c3cnncc3OC)=O)CC23CC3)=O)CCO1 59648,C(C)(C(C)COC)(c1nnnn1-c1ccccc1C)NCCC(=O)OC 59649,c1(C(N2CCOCC2CC2CCC2)C(=O)NC)ccc(C(=O)OC)nc1 59650,c1(C(=O)NC23CC(NC(c4ccc(Cl)cc4Cl)=O)(C2)C3)ccc(Cl)c2[nH]ccc12 59651,C=CC(C)CC(=O)N1CCCC1CCNC(C12CC1CN(C(=O)NCCC)C2)=O 59652,N1(CC(=O)NCC2CCN(C(c3cn(CCC)nn3)=O)C2)CCN(C)CC1 59653,c1(OC(C)C)ccc(C(=O)NC2(C)CN(C(=O)CC3CC(C(F)F)C3)C2)cn1 59654,C=CCC(C(=O)NCC1CCCC1NC(=O)CCCOCC)c1ccccc1 59655,c1(C(=O)NCCCCCNC(C2N(CC)CC2)=O)cc(C)c(C(=O)OC)o1 59656,c1(C(=O)NC2CCCC(NC(C(C)SCCCC)=O)C2)nc(C)ccc1O 59657,c1(C(=O)NC2CCCN(C(C3(CC(=O)OC)CC3)=O)C2)cccc2c1COC2 59658,Nc1ccc(C(=O)NC2CCCC2NC(c2ncoc2C(F)(F)F)=O)cc1Cl 59659,N1(C(c2cccc(CCC)c2)=O)CC2(CC(NC(C3(C)CCC(=O)N3)=O)CO2)C1 59660,c1(C(=O)NC2CC(CC)(CC)N(C(=O)C3=NOC(C)C3)C2)c(C)ccc(C)c1O 59661,N1(C(C2N(C(c3ccc(C(C)=O)[nH]3)=O)CC=CC2)=O)CCOC(C)(C)CC1 59662,c1(NC(CNC(C(Br)=C(C)C)=O)C(C)C(C)C)ncnc2cc(F)c(F)cc12 59663,Cc1cnc(NCC(=O)NCCC2(NC(=O)CCCOc3cccnc3)CC2)o1 59664,C1(NC(CCN(C)C(=O)OC(C)(C)C)=O)C2CC3CN(C(=O)C4CC4)C1C3C2 59665,N1(C(C(CCC)N(C)C)=O)CCC2(C1)CN(C(C1CC1(C)C)=O)C2 59666,N1(C(CCC2(C)CN(C(CNC(C3C(C)C3)=O)=O)C2)=O)CC2CC(O)CC1C2 59667,C1(C(N2C(C(=O)NC)CC(O)C2)=O)CN(C(=O)CC2C=CCCC2)CCC1(C)C 59668,O=C1NCc2c1ccnc2C(N1CC(CNC(C2CC(O)C2)=O)C(O)C1)=O 59669,C1(C(N2C(C)(C(=O)NCCC3CCN(C)C3)C=CC2)=O)CCCC(C#N)C1 59670,C(C(C)(C)CC(=O)NC1CN(C(=O)CC2(C#N)CCCCC2)CC1(C)C)N(C)C 59671,c1(CC(=O)N(C(C2CCCC2C)C)C(=O)OC2CCC2)cccc(Br)c1 59672,Cc1cccc(NC(C2CCN(C(=O)Cc3cc(F)ccc3Br)C2)=O)c1[N+](=O)[O-] 59673,C1(C)(CNC(=O)OC(C)(C)C)CCC(NC(=O)C(=O)NCCN2CCCC2=O)C1 59674,N1(C(c2cn(CC)nn2)=O)CCC(CNC(=O)CC2CCCC(OC)C2)(OC)C1 59675,N1(C(c2cccc(OC)n2)=O)CC2CCN(C(=O)Cc3cccc(O)c3)CC2C1 59676,c1(C(=O)NC2C(NC(CCC=C)=O)CCC2)nc2ncccn2n1 59677,C1(C(=O)NCC(=O)OCC#C)(NC(C2CC2(Cl)Cl)=O)CSC1 59678,c1(NC)cccc(C(N2CCC(CN(C)C(C3CC(C)(F)C3)=O)C2)=O)n1 59679,Cc1sc2ncc(C(=O)NC3CC3CNC(c3ncoc3C(C)(C)C)=O)n2c1C 59680,Cc1cc(-c2ccc(CNC(c3cnn(C4CC4)c3)=O)cn2)cc2c[nH]nc12 59681,c1(COCC(=O)NCC(CNC(CCNS(CC)(=O)=O)=O)O)ncc(C)o1 59682,n1(C(C)C)cc(C(=O)NCCC2CCN(C(=O)CCN3CCC3)C2)c(Br)n1 59683,C=CCC(C)(C)CC(=O)NCc1cncc(C(=O)NC2CN(C(N)=O)C2)c1 59684,C1(CC(=O)NC(CC(=O)NCCC(C)(C)O)C2CC2)CC2(CC2)CO1 59685,Cc1ccc(F)c(O)c1C(N1CCC2(CC(NC(C3CC(C)CO3)=O)C2)C1)=O 59686,C1(C(N2CCOC(CC)C2)=O)(CNC(C(COCC)C)=O)CC12CCC2 59687,c1(C(N2CCN(CC(=O)NCC3N(CC)CCC3)CC2)=O)cc(F)cnc1O 59688,c1(C(C(=O)NCC(C)OC)NC(=O)OC(C)(C)C)cn(C)nn1 59689,CC(C)C(C(=O)NC(C)Cc1ccncc1)NC(=O)CCc1cccnc1 59690,c1(C2C(C(=O)OC(c3nc(CC)[nH]n3)C)C2)ccc(OC)cc1 59691,c1(OC)cccc2sc(C(=O)NCC(O)CNC(=O)C(C)n3cccn3)cc12 59692,c1(C(=O)NC2C(NC(C3C(C)C3)=O)CCC2)cnn(C)c1Cl 59693,C1(N(C(CC(=C)I)=O)C)CCC(n2cc(-c3ccc(OC)s3)nn2)CC1 59694,C(=O)(N=c1nc2cccc(OC)n2[nH]1)C1CC(=C)CN1C(c1cc(C)n(C)n1)=O 59695,C1(COC)C=CCCN1C(=O)CC(O)CNC(=O)C(C)(C)n1cccn1 59696,c1(OC)cc([N+](=O)[O-])ccc1C(=O)NC1C2CC1CN(C(=O)C(C)C1CC1)C2 59697,C1(NC(COCCC#C)=O)(CO)CCN(C(=O)CCC2CCCCN2C)C1 59698,c1(C(=O)NC2C(CNC(=O)CC3CCOC3)C2)c[nH]c2cc(Cl)ccc12 59699,CC1CC(CNC(C2CC3CC3C2)=O)CCN1C(=O)CCOC1CCOCC1 59700,C1(C)(CNC(CCC(=C)C)=O)CC(F)(F)CN1C(C1CC1C(F)F)=O 59701,c1(C(=O)NC(C(CCc2ccccc2)NC(CC=C=C)=O)C)cnc2sccn12 59702,c1(OC)cc(C(=O)Nc2cc(C)cc(C)c2Br)c(N)cc1Cl 59703,c1(C(N2CCCC(N(C(=O)CCN3C(=O)CCC3=O)C)C2)=O)cccc(F)c1N 59704,C(CC(=O)N1CC(C)(C)C12CCC2)(CC(C)C)NC(CC(COC)(C)O)=O 59705,C1(C(=O)NCCCN(C)C(c2ccc(Cl)c(O)c2)=O)COc2ccccc2C1 59706,N1(C(C2CC(=O)CN2C(C2(C(F)(F)F)CC2)=O)=O)CC2(CCNC2=O)C1 59707,c1(C(=O)NC(C2CCCC2)CNC(C2CC2F)=O)cnn(CC2CC2)c1 59708,C=CC(C)CC(=O)NC(C1CN(C(=O)CCc2cncnc2)C1)C 59709,C1(NC(=O)NCC2(CCO)CN(C(=O)OC(C)(C)C)C2)CCc2ccnn2C1 59710,c1(C(N2C3CC(NC(CNC(C4C(C)C4)=O)=O)(C3)C2)=O)cccc2c1OCC2 59711,N1(C(c2cc(SC)nn2C)=O)CCC(N)c2ccc(F)cc21 59712,c1(C(N2CC3C(N(C(=O)CC4(C)CC4(Cl)Cl)C)C3C2)=O)cncn(C)c1=O 59713,c1(C(=O)NCCCN(C(CSCC=C)=O)C(C)C)ccc(Cl)c(OC)c1 59714,Cc1ccc(C(=O)NC2CC2C(=O)N(CCO)C2CC2)cc1[N+](=O)[O-] 59715,c1(C(N2CCC(NC(CCCN(C)C)=O)C2C(C)(C)C)=O)nccc2cc[nH]c12 59716,C(CC(=O)NCc1cc(C(N)=O)no1)(C(F)F)NC(CNC(C1C(C)C1)=O)=O 59717,N1(C(CCC2(C)CCCN2C(=O)C(O)C2CC2)=O)CCCCCCCC1 59718,Cc1nc2ccc(NC(C3CCCN3C(c3cc(Cl)c(Cl)s3)=O)=O)cc2o1 59719,Cc1n[nH]c(C)c1CC(C)C(=O)NC(C)CC(C)NC(=O)C(C)O 59720,C(=O)(C(CNC(=O)CC(C)(F)F)CC1CC1)NCc1ccc(CC)o1 59721,C1(CCNC(c2ccc(C(F)F)s2)=O)CCCCN1C(C12CCC1C2)=O 59722,c1(C(N(CCNC(c2cc(C)oc2)=O)CCOCCO)=O)c[nH]ccc1=O 59723,CCCC(F)C(=O)NC1(CCCNC(=O)CCCNC(=O)OC)CC1 59724,CC(C)(C)C(=O)C(=O)N1CCN(C(c2sccc2F)=O)CC1CC1CC1 59725,CON1CCC(CC(=O)NC2CC(F)(CNC(C3CCN3S(C)(=O)=O)=O)C2)CC1 59726,C1(NC(c2nccc(OC)c2)=O)CCCC12CN(c1ccncn1)C2 59727,C1(CC=C)(NC(C2CC2c2ccccc2F)=O)CCN(C(=O)C(F)(F)COC)C1 59728,C1(c2c(Cl)cccc2Cl)CCCN1N1CCC(n2cccn2)CC1 59729,C1(CCCC)CCC(N=c2[nH]c(N3CCOC(C)C3)nc3c(F)cc(F)cc23)C1 59730,CC(C)(C)C#CC(=O)N1CCN(C(=O)CC2CCS(=O)(=O)CC2)C(CF)C1 59731,C1(OC)CN2CC1Nc1c(cccc1)C2=O.c1(CCCN)nc(O)n[nH]1.C(C)(C)O 59732,C(CCC(=O)NC(CSCC)C(=O)NC1CCN(C(N)=O)C1)OCC=C 59733,Nc1ccc(C=CC(=O)NCC2CCCN(C(C3CCCOCC3)=O)C2)cc1N 59734,CCC(C)C(O)C(=O)NC1CC(CNC(c2cc(-c3ccccc3)ccn2)=O)C1 59735,C(CC(C(C)(C)C)NC(=O)Cn1cnnc1)N(C(c1c(C)nccc1)=O)C 59736,CCC(CC)(CCNC(=O)C(C)Cn1ccnc1)NC(c1cc(F)n(C)n1)=O 59737,Cc1c(Cl)c(C(N2CCC(C)(NC(C3CC34CCCC4)=O)C2)=O)nn1C 59738,N1(C(C(=O)NC(C(=O)N(CC)CC)C)=O)CCCC2(C=CCO2)C1 59739,C12(NC(C(C)NC(C)=O)=O)CC1CN(C(c1ccc(N(C)C)nn1)=O)C2 59740,C1(C(N2CC(O)(C(C)NC(=O)Cn3cnc(C(N)=O)n3)C2)=O)(COC)CC1(F)F 59741,CC(C)(C)CC(N)CCN1CCC(C)(C)C1=O 59742,N1(C(COCCCCC)=O)CCCC1CN(C(C1CCC1c1nc[nH]n1)=O)CC 59743,N1(C(Cc2n(C)nnc2)=O)CC2(C(=O)NC3CC(CO)C34CCC4)CCC1CC2 59744,c1(CNC(N(C2CCCOC2)CCC)=O)cnc(COC)s1 59745,c1(OC)nccc(C(N2CC=CCC2C(=O)NCC2C(C)C2(F)F)=O)n1 59746,CC1(F)CCN(C(=O)C(C2CC2)NC(=O)CC2CC(F)(F)C2)C1 59747,CC(C)CC(C(=O)N1CC2CC(NC(C3(C(N)=O)CC3)=O)CC1C2)C(N)=O 59748,c1(SC)c(C(=O)N(c2cccn(C)c2=O)C)cccc1Br 59749,N1(C(C(CC(C)C)O)=O)CCC2(CC(NC(c3cc(C4CC4)ccc3F)=O)C2)C1 59750,C1(C(=O)NCCOC2CCN(C(C3(C)CC3(F)Cl)=O)C2)CN2CCCN1CC2 59751,c1(C(N2CC(NC(C=COCC)=O)C3(C2)CCC3)=O)ccc2c(c1)C=CS2(=O)=O 59752,C1(CNC(c2n(C(CC)C)ncc2)=O)CCCN(C(=O)C(C)(C)CC)C1 59753,C1(C)(CNC(c2ccc(CCC)s2)=O)CCC(NC(C2(CF)CC2)=O)CC1 59754,C(=O)(C(F)C(F)(F)C(F)(F)F)N1CC(CNC(=O)C2=NNC(=O)C2)CC(C)(C)C1 59755,C(CCCCC(=O)NC(C)C(C)(C)C)N(C(C(C)C1CCCO1)=O)C 59756,n1(CC)cnc2c(NCc3cnc(C)o3)nc(N3CCOC(C)(C4CC4)C3)nc12 59757,C(C)(C)(C(=O)NC1CCC1CNC(C1CCN(C(=O)OC)C1)=O)NC(CC)=O 59758,C1(Cl)(C(=O)NCC2(NC(c3nc(CC(C)C)sc3)=O)CCOC2)CC12CCC2 59759,c1(C(=O)NC(CC)CN(C(=O)COCC2CCCC2)C)cc(C(F)F)ncn1 59760,c1(C(=O)NCCC2(CNC(C(C)=C3CC3)=O)CC2)ccc2nc(S)oc2c1 59761,C(CNC(=O)CC1(N(C)C)CC1)(C(C)(C)C)NC(C(C=C)C)=O 59762,c1(C(C(=O)NCC)N(CC(C)OC(C)(C)C)CC)cc(C)c(C)c([N+](=O)[O-])c1C 59763,[N-]=[N+]=Nc1ccc(C(=O)NCC2CCCN2C(C2CCC3CCCCN23)=O)cc1 59764,C1(C(N(C2CC=CC2)C)=O)CC1C1CN(C(c2cc(Cl)cs2)=O)C1 59765,C1(CNC(c2n(C)ncc2)=O)CN(C(c2cc(F)n(C)n2)=O)CCN1C 59766,C1(CC(=O)NC(CC#C)C)CN(C(C2(O)CC(CF)C2)=O)CCO1 59767,c1(CCNC(C)=O)cn(CC2CCN2Cc2ccc(-c3cccs3)[nH]2)nn1 59768,N1(CCCCNC(CC(C)OC)=O)CCCN(C(=O)C=CC2(C)COC2)CC1 59769,C12(C(=O)NC(CNC(CCC=C(C)C)=O)CO)CCC(C)(C1)OC2 59770,n1(CC)nc(COC(=O)C(c2cnn(C)c2)=O)c2c1CCOC2 59771,N1(C(c2c(CC)n[nH]c2)C(=O)Nc2ccccc2C)CCC(O)CC1(C)C 59772,O=C(CC(C(F)F)c1ccccc1)Nc1ccc(N2CCC(CO)C2)cc1 59773,C1(NC(C=CC(C)C)=O)(CNC(c2cc[nH]c2C2CCCC2)=O)CCOC1 59774,c1(CC(=O)NC)ccc(C(=O)NCC2C=CCN2C(C2CC2(C)C)=O)cc1 59775,N1(C(c2c(CC)cns2)=O)CCN(C(=O)CCc2cncc(F)c2)CC1CCO 59776,C1(C)(COC)CC(NC(=O)CSc2nnnn2C)CN1C(c1cc(O)n(C)n1)=O 59777,C1(NC(C2(C)C=CCN2)=O)CCCC12CCCC2 59778,N1(C(C(CSCC)NC(c2ccsc2)=O)=O)CCC2(CCC(OC)C2)C1 59779,C1(c2cnc(C)[nH]2)NC(=S)N(C2CC2)C2=C1C(=O)NC(C)C2 59780,C1(C)(C(=O)NCCN(C(=O)CSCC2CCCO2)CCC)CCC(C)=C(C)C1 59781,C1(NC(c2cc(C)sc2C)=O)CC(NC(=O)CCCNC(N)=O)C12CCOCC2 59782,c1(C(NN)=O)ccnc(CNC(C2CC=CCC2NCC2OC3CCC2C3)=O)c1 59783,CCC(N=c1[nH]nc(-c2cccnc2)cc1C(F)(F)F)C(C)COC 59784,N1(C(CCOC(C)C)=O)C2CCC(C2)C1CNC(=O)Cc1cc[nH]n1 59785,C#CCC(C)(C)C(=O)N1CC2(CC(CC(=O)NCc3cc(C)cc(C)n3)C2)C1 59786,N1(C(Cc2c(OC)ccc(C)c2)=O)CC(C2CN(C(C3CC(C)CCO3)=O)C2)C1 59787,CC1CCN(C(c2cnn(C)n2)=O)C1CNC(=O)CCCN1CCCCC1 59788,C1(NC(CSC(C)(C)C)=O)CC(N=c2[nH]ncs2)C12CCOCC2 59789,Cc1ccc(OCC(=O)NC2CC3CCC2(NC(c2cncnc2)=O)C3)cc1C 59790,C=CC1CN(C(c2cccc(COC)n2)=O)CC1NC(C12CC(F)(C1)C2)=O 59791,N1(C(C(CCC)CNC(C2CC(=O)NC2(C)C)=O)=O)CCC(O)C12CCC2 59792,C1(C(C)C)CCc2c(sc(NC(c3cc(C4CC4)ns3)=O)c2C#N)C1 59793,C(=O)(CCS(C)(=O)=O)NC(C)C(C)C(=O)NC1(C(N)=O)CC1 59794,c1(N2CC(OCCNC(c3ncc(OCC)nc3)=O)C2)ncc2ncnc-2[nH]1 59795,c1(NC(Cn2cc(CCCS(C)(=O)=O)nn2)=O)cccc2c1CCNC2=O 59796,C(=O)(CS(C)(=O)=O)N(CC(=O)NCC(COC)(C)O)CC(C)C 59797,c1(C(N(C(CCNC(c2c(C)noc2C2CC2)=O)C)C)=O)cn2c(n1)CCC2 59798,N1(C(c2ccc(SC)o2)=O)CCC(C)CC1C(=O)NCC12CC(CO)(CO1)C2 59799,CC(C)(CC(=O)N1CCN(C(c2ccc(N)c(F)n2)=O)CC1)C(F)F 59800,C1(C(=O)N(C2(C(=O)OC)CCOCC2)CCC=C)CCCN(C(C)C(C)(C)C)CC1 59801,c1(C(=O)NC2CN(C(c3c(C)n(C)cc3)=O)C(C)C2)c(F)cccc1Br 59802,C#CCCN=C(NCC(c1ccccc1)CO)NCC1(C)CCCCO1 59803,c1(C(N(C)CC2CCN(C(c3c(C(C)C)csc3)=O)C2)=O)ncc(N(C)C)cn1 59804,c1(C(=O)NC2C(CNC(C(C)(C)N3CCCC3)=O)CCC2)cnc2n1CCCC2 59805,CC(C)CN=C(NCc1cnnn1C)NCC1(S(C)=O)CC1 59806,c1(C(N(C2CCN(C(C3(SC)CC3)=O)C2)CC)=O)ccc(Cl)c(C(=O)NC)c1 59807,C(CC(F)F)(C(=O)NCC1(C)CC(C)(C)C1)NC(c1cn(C)nn1)=O 59808,C1(NC(=O)CCn2cnnn2)CC(F)(CNC(C2CC2CF)=O)C1 59809,c1(C(N2CCC3C(NC(CCCC(=C)C)=O)C32)=O)cc2c(C3CC3)cccc2[nH]1 59810,c1(C(N2CC(NC(C(C)(C)OCC)=O)C(C)C2)=O)cnc(OC(F)(F)F)c(F)c1 59811,N1(C(C(COC)C)=O)CC2(C)CN(C(c3ccn(CC4CC4)c3C)=O)CC2(C)C1 59812,CCCCCC(O)C(=O)N1CCC(C(C)(C)NC(c2ccc(CC)c(C)c2)=O)C1 59813,c1(C(=O)NCCCCc2cn(-c3ccc(Br)cc3Cl)nn2)ccc2ncsc2c1 59814,C12(C(=O)NCC3(NC(CCC=C=C)=O)CCCC3)CCCCC1C2(F)F 59815,Cn1cc2cccc(C(=O)NC(=O)CCC3(C)CN(C(=O)CNC4CC4)C3)c2n1 59816,N1(C(c2cc(N)cc(F)c2)=O)CCCC2CN(Cc3ccc(F)cn3)CCC12 59817,n1(C(c2nnnn2C)NC(CCC)Cc2ccccc2)nc2ccccn2c1=O 59818,C=CCC(C)(C)CC(C(=O)NCCC1(C)CC1)N1CCC(C)(F)C1 59819,Cn1ncc2nc(O)c(C(N3CC(CNC(=O)Cc4cccs4)C3)=O)cc12 59820,C1(CC)CN(C(C2CC(C#N)(OC)C2)=O)CCN1C(=O)CCc1cccc(C)n1 59821,Cc1cc(CC(=O)NCCCN(C(=O)C(C2CC(C(C)(C)C)C2)C)C2CC2)n(C)n1 59822,C(CNC(c1nn(C)cc1Cl)=O)(C(C)C(C)C)NC(C1CCC(CC)CC1)=O 59823,c1(CC(=O)NC2CCN(C(c3cc[nH]c3)=O)CC2F)cccc2sccc12 59824,N1(C(C2C3(CC(OCC)C3)C2)=O)CCC(NC(=O)C=C(Cl)Cl)C2(CCC2)C1 59825,C(=O)(C(C)C(CC)CC)NCC(CC)NC(=O)CCCC1CCOCC1 59826,c1(CCC)cc(C(=O)NC(CNC(=O)C(C)CN2CCCCC2)CC)n(C)n1 59827,CC(O)C(C)C(=O)NCCOC1CN(C(c2nccnc2-n2ccnc2)=O)C1 59828,CCC(C)C(C(=O)NC1(CO)CC2CCCC12)NC(=O)C=CC(F)(F)F 59829,c1(-c2ccc(F)cc2)ccc(=NCCc2cnc3n2CCCC3)[nH]c1Cl 59830,Cc1cnc2c(cnn2CC(=O)N(CC(C)NC(=O)CC2CCOC2)C)c1 59831,C12(NC(CCCOC)=O)CCC1CN(C(=O)CCN1CCCS1(=O)=O)C2 59832,N#CC1CN(Cc2ccccc2)CC1NC(=O)NCCc1ccccc1Br 59833,C(=O)(C1=C(Cl)CCCC1)N1CCCC(C)(C(=O)NC(c2nc(C)on2)C)C1 59834,C1(N(C(C(CC#C)C)=O)C)CCCCN(C(c2onc(CC)c2C)=O)C1 59835,C1(C(N(C)CC2(O)CN(C(C(C)NS(C)(=O)=O)=O)C2)=O)Cc2ccccc2CO1 59836,CN1CCC(O)C(NC(N2CCN(CC3CCCCC3)CC2)=O)C1 59837,N1(C(c2c(C)nc(COC)s2)=O)CC2CCN(C(=O)CCC3CC3(Cl)Cl)C2C1 59838,CC1(C)CC(C)(C(=O)NCC2CCCCC2NC(C2CCCS2)=O)C1 59839,c1(CC(=O)NC2CCC(NC(c3c(C)cco3)=O)C2)sc2ccccc2c1C 59840,Cc1ccc(C(=O)N(C2(C(=O)NC(C3CCCO3)(C)C)CC2)C)c(F)c1 59841,C(=O)(C1=NNC(=O)C1)NC1CCCC(NC(C(N2CCCC(C)C2)=O)=O)C1 59842,c1(C(N2C3C(N(C(C=C(C)C)=O)C)CC(C3)C2)=O)cc([N+](=O)[O-])cn1C 59843,c1(CCC(=O)NC(C)CNC(=O)C2CC2)ccc(Br)cc1 59844,Cc1ccc(-c2ccc(CNC(c3cccn4c(O)nnc34)=O)nc2)c2cn[nH]c12 59845,CCCCCCCC(F)C(=O)NCC1CCN(C(C2(C)CCCC2)=O)C1 59846,N1(C(CCCN(C(C(C)(C)C)=O)C(C)C)=O)CCN(C(C2CCCC23CC3)=O)CC1 59847,N1(C(C2CC3(CC(C)C3)C2)=O)CCN(C(c2cnc(C3CC3)[nH]2)=O)C2COCC12 59848,C1(COC)CCN(C(=O)Cn2c([N+](=O)[O-])cnc2C)CC1(F)F 59849,N1(CCCC(CC)=O)CCN(Cc2ccncc2)C2CC12 59850,N1(C(C2N(C)CCC2)=O)CC2CC1C2NC(C1CCN(CC(F)(F)F)C1)=O 59851,c1(C(N2CC(OC)(CNC(C3(CCF)CC3)=O)C2)=O)ccnc(F)c1 59852,C1(NCC)CCCC(N=c2cc(C)[nH]c(=NCc3nc(C)c(C)nc3C)[nH]2)C1 59853,C1(CN(C)C(C2CC2F)=O)CN(C(=O)CCOC2CC2)CC12CC2 59854,c1(C(=O)NC2CN(C(CCC=CC)=O)CC(F)(F)C2)cccc2ncc(C)n12 59855,C1(NC(c2c(NCC)scn2)=O)CCCC12CN(C(c1cc(C#N)[nH]c1C)=O)C2 59856,N1(C(C(C)N(C)C)=O)CCCC(C)(CNC(=O)CCN(C)Cc2ccccc2)C1 59857,C1(CC(=O)NCCN(CCCN(C)C)C(=O)C=C(C2CC2)C2CC2)NC(=O)NC1=O 59858,N1(C(CSC(C)C)=O)CC(NC(C23CCC(F)(CC2)C3)=O)C2CCCCC12 59859,c1(C(C)C(=O)NC(C)(C)CNC(=O)Cc2nccn2C)ccc(Cl)cc1 59860,C(=O)(C#CC(C)(C)C)NCCN(C(c1snnc1C(C)C)=O)CC 59861,Cc1ccc(Cl)cc1C(=O)NCCN(C)C(C1COCC(=O)N1C(C)C)=O 59862,N1(C(C(CSC)OC)=O)CCCCCC(NC(c2cncc(OC(C)C)c2)=O)C1 59863,S(=O)(=O)(c1cnc(NCC(c2nccs2)C)c(Cl)c1)N1CCn2c(C)ncc2C1 59864,CCC(C)C(O)C(=O)N1C2CCC1(CNC(C1(C)CCC1)=O)CC2 59865,c1(C(=O)NC2C3CC2CN(C(C2CC(O)C2)=O)C3)cc2scc(Br)c2[nH]1 59866,C1(CCO)(C(=O)CC)CCN(C(C)=O)CC1O.C1(CCOCC)CCCC1 59867,C(CNC(=O)Cc1cnnn1C)(CC(F)(F)F)NC(C(C)SC)=O 59868,C12CCCCN(C1)C(=O)CC2.C1(NC2(c3ccn(C)n3)CC2)CCCC12CCC2 59869,c1(OCC(N2C(C(C)NC(c3n(C=C)nnc3)=O)CCC2)=O)ccc(F)cc1O 59870,Cc1nc2cc(C(=O)NC3(CNC(=O)CC4COC5CC4C5)CC3)[nH]c2s1 59871,c1(N2C(C(=O)Nc3nccc(C(=O)NCC)c3)COCC2)nc(OC)ncc1F 59872,N1(C(C(C)OCC#C)=O)CCN(C(c2c(C)noc2C)=O)CC1c1ccccc1 59873,N1(CC)CC(NC(=O)C(CC2CCCC2)NC(=O)C(C2CCOCC2)=O)C(C)C1 59874,N1(C(C2(C(=O)OC)CCCC2)=O)CCCC(C)(NC(C2CC(OC)C2)=O)C1 59875,CCC(C)C(O)CC(=O)NC1(CNC(c2n[nH]c3ccccc23)=O)CC1 59876,N1(C(COCC(=O)OC)=O)CC2C(N(C)C(C3CN(C(C)C)CCO3)=O)C2C1 59877,N1(C(C2(C#C)CN(C(=O)CN3C(=O)CCCC3=O)C2)=O)CC2(CC2)CC1CO 59878,C(=O)(CS(=O)(=O)C1CC1)NCC(C(C)C)NC(C1(CC(=O)OC)CCCC1)=O 59879,C(=O)(C(CCC(C)(C)C)N(c1ccccc1C(C)C)C)NC1CC(C(=O)OC)C1 59880,C(c1ccccc1Cl)=CC(=O)NC1CCCN(C(=O)CC2COCCO2)CC1 59881,C(c1ccncn1)=CC(=O)NC(C(C)NC(c1cscc1F)=O)C 59882,C1(CC(=O)NCCN(CC(C)O)C(c2cc3sccc3[nH]2)=O)CC(C)(C)OC1=O 59883,C1(c2c(F)cccc2)CC1N=c1ccnc(NC2CCN(C3CC3)C2)[nH]1 59884,c1(-n2c(C)nc(C3CN(C)CCO3)n2)ccc(C)c(Cl)c1.n1(CC)nnnc1C(C)C 59885,c1(N2CCC(C)SCC2)ccncc1S(=O)(=O)N1CC(C)(C)OCC1CO 59886,c1(C(=O)NC2CC(NC(C(C=C=C)C)=O)CC2O)cc(O)nc(C)n1 59887,c1(C(N2CC(O)(CCNC(C3(COC)C=CCC3)=O)C2)=O)[nH]c(O)nc1C 59888,CCCC(C(=O)N1CCOC(CCNC(=O)C(F)=C(C)C)C1)N(C)C 59889,N1(C(CCNC(=O)OC)=O)CCC(NC(=O)CC2COCCN2C)C1C(C)(C)C 59890,C1(C(=O)NCCC(C)CCO)(OC)CCN(C(=O)OC(C)(C)C)C1 59891,c1(-n2cc(C3CN(CC(c4cccnc4)OC)C3)nn2)ccc(Cl)cn1 59892,N#Cc1cc(C(N2CCC(CC(=O)Nc3ccc(F)c(F)c3Cl)C2)=O)ccc1F 59893,C1(NC(CCNC(c2c(C)csc2C)=O)=O)CCOC12CCOC2 59894,N1(C(=O)NCc2ccncc2)CCC2CCC12c1ccncc1 59895,N1(C(C=C(C)C)=O)CCCC(NC(c2ccc(CN=[N+]=[N-])cc2)=O)CC1 59896,C1(C)(C(=O)NCC(C(=O)OC)(C)C)CCCN(Cc2cccc(O)c2)C1 59897,CC(C)CC(C)N(C(=O)CONC(c1coc(C(F)F)c1)=O)C 59898,C(=O)(C(F)C(C)CNC(c1cc(C)c(N)cn1)=O)N1CCC(C(=O)OCC)C1 59899,C(=O)(CC1C(=O)Nc2ccccc21)N1CC(C)C(NC(C2CSCC(=O)N2)=O)C1 59900,C(CCN=c1cc(C)[nH]c(=NCC2CCN(C)C2C)[nH]1)OC=C 59901,C(=O)(C1CNc2ccccc21)NCC1CN(C(CC2C(C)(C)CCCO2)=O)C1 59902,C12(NC(=O)CCn3ccnn3)CC(C1)N(C(C1CC3C=CC1C3)=O)C2 59903,c1(C(=O)NC(C2CC(NC(C3(Cl)CC3(C)C)=O)C2)C)cc(-c2cnn(C)c2)[nH]n1 59904,CC1CN(C(=O)C(=O)C2CCCC2)CC(C)CN1C(c1cc(C(N)=O)co1)=O 59905,c1(C(=O)Nc2ncc(CO)cc2Br)cc(Cl)cc(Cl)c1F 59906,Cn1cc(C(=O)NC(C)(CNC(c2csc(C(F)F)c2)=O)C2CCC2)nc1O 59907,c1(C(=O)NC(CN(C(=O)C(CC)OC)CC)C)ccnn1C(C)(C)C 59908,C1(C(N2CCCCC2C2CC2)=O)C2CC(O)C(C2)N1C(=O)C(O)CC(F)(F)F 59909,CC1=NN(C)C(=O)C1CC(N1CCC(NC(c2ccnn2C(C)C)=O)C1)=O 59910,C1(O)(C(=O)NCC(N(C(c2ncn(CC)n2)=O)C)C2CC2)CCC(C)CC1 59911,c1(OCCCN(CC(O)CN(C)C(=O)C2CC2)C(C)C)ccc(F)cc1Cl 59912,c1(C(=O)NC(C(C)NC(=O)CCN2CCCC2)C)coc(C(N)=O)c1 59913,N1(CC(=O)NCC(C)NC(c2c(CC)c(C)sc2)=O)CCCCCCC1=O 59914,C(=O)(CC(C(F)(F)F)NC(=O)COCCF)NC1(CC#C)CC1 59915,N1(C(C2CCC(CC)O2)=O)CC=CC(NC(c2csc(CO)n2)=O)C1 59916,c1(C(=O)NC2C(CNC(c3ccnnc3O)=O)CCC2)cccc2[nH]nc(O)c12 59917,C#Cc1cncc(C(N2CCCC2C2CCN(CCN3CCNC3=O)CC2)=O)c1 59918,C(=O)(CCC(C)(F)F)N(CC(C)C(=O)NCc1cncc(C#N)c1)C 59919,c1(OC2(C(N(CCCNC(c3conc3C(F)F)=O)C)=O)CC2)ccccc1F 59920,C(=O)(C(C(C)C)NC(C)=O)N(CC(CN(C(CCN(S(CC)(=O)=O)C)=O)C)O)C 59921,c1(OC)ccccc1OC(C)C(=O)OC1C2CC1N(C(=O)OC(C)(C)C)C2 59922,c1(CC(C(=O)OC)NC(=O)NCc2cn(CC(O)COC)nn2)ccc(I)cc1 59923,C1(NC(C2C(C)(C)C2)=O)CC12CCN(C(c1ccn(CCF)n1)=O)CC2 59924,c1(N(C)CCC2CCN(C(=O)C=CCOc3ncccn3)CC2)ccccc1F 59925,C12(C(N(CC(c3nn[nH]n3)C)Cc3ccc(C)cc3)=O)CC=CCN1CCC2 59926,c1(N(CCCNC(C)=O)C)ncc(S(=O)(=O)N2CCS(=O)(=O)CC2C)cc1Cl 59927,Cc1cccc(Cl)c1C(N1CCC(OCCNC(=O)Cc2ccsc2)CC1)=O 59928,C(CC(=O)NCc1cnns1)(C(F)(F)F)NC(CC(C=C)(C)O)=O 59929,c1(C(N2CC(n3ccnn3)C(O)C2)C(=O)NCC)ccc2c(c1)sc(=O)n2C 59930,CC(C)CC(C)(CN=c1[nH]c(Cl)ncc1Br)NC(c1cn2c(n1)CC(C)CC2)=O 59931,C1(c2onc(-c3cc(F)c(O)c(F)c3)n2)CCC2(CCOCC2)CO1 59932,c1(CN2CCCC(C)(C(=O)NC3(CC#N)CCCC3)C2)cc(F)c(Cl)cc1O 59933,Cn1cnc2c(NC3CCN(Cc4ccc(Br)c(Cl)c4Cl)C3)ncnc12 59934,C1(C(=O)OC)CCC(C(=O)NCC2CCCN(C(C3(C(C)(F)F)CC3)=O)C2)CC1 59935,C12CCCN(C1)C2=O.C1(c2nnnn2C(C)C)(NCC=C(C)C)CCCC1 59936,C1(CN(C)C(C2CCC(=O)N2C2CC2)=O)CCCN(C(=O)C=Cc2cc[nH]n2)C1 59937,c1(C(=O)ONCC(C)N(C)C(c2ccco2)=O)ccn(CC(=O)N(C)C)n1 59938,S(=O)(=O)(CC(=O)NCC1CN(C(c2cnc(Cl)n2C)=O)CC1O)NCC 59939,C1(C)(CNC(C(C)CN2CCOCC2)=O)CN(C(=O)C(=O)N(C)C)CCO1 59940,C12(CCCN1C(c1cccc[n+]1[O-])=O)C(=O)NC2C1(O)CCCCC1.C(=O)(CO)OC 59941,CCCC(CCC)C(=O)N1CCCN(C(=O)Cn2cccc(N)c2=O)C(C)C1 59942,C1(C(=O)Nc2cc(O)ncn2)CN(C(c2ccc(O)nc2)=O)CCC1O 59943,S(=O)(=O)(C1CCCN(C(c2ccccc2OC)=O)C1)N1CC(C(C#C)C)C1 59944,N1(C(c2cn(CCNC(c3c(COC)noc3)=O)nc2)=O)CCC(CO)C(O)C1 59945,N1(C(C(C)CO)=O)CC2(C1)CN(C(c1cn(C)cc1C(F)(F)F)=O)C2 59946,C1(C(=O)NCCOC)CC12CCN(C(c1ccsn1)=O)C2 59947,C1(c2n(C(C)C)nnn2)(NCCc2ccncn2)CC2CC1CC2O 59948,c1(C(=O)NC2C(NC(CCC(c3ccc(C)cc3)=O)=O)C2)cc(F)ccc1Cl 59949,C(CNC(=O)CC1CC=CC1)(C(C)C(C)C)NC(c1c(NC(C)=O)cccn1)=O 59950,N1(C(C(N2CCNC2=O)C)=O)CCCC(N(C(=O)Cc2n[nH]c(=N)s2)CC2CC2)C1 59951,N1(C(C2CC(Cl)(Cl)C2)=O)CC2CN(C(C3CC(CF)C3)=O)CC2C1 59952,c1(C(=O)NC2CCC(C(N3CCC(O)CC3)=O)C2)ccc2occc2c1 59953,C12(CC(=O)NC3CN(C(=O)CCc4nc[nH]n4)CC3O)CCC(CC1)C2 59954,c1(NC(C2CC3C(C2)C3(F)F)=O)nc(Cl)cc(Cl)n1 59955,CCC1=C(C(=O)N2CCCCC2CCNC(=O)CC(O)CN(C)C)CCCO1 59956,N1(C(C(c2ccn(C)c2)C)=O)CCCC1CC(N1CC(F)C1)=O 59957,C(=O)(C(C(C)(C)C)NC(c1ccccn1)=O)N1CCN(C(CC)=O)CC1 59958,C1(C(=O)NC(CNC(c2c(C)ocn2)=O)(C)C2CC2)CCn2cnnc2C1 59959,c1(C(c2cnc(N(C)C)nc2)(F)F)ccc(N=c2ncnc3[nH][nH]c(Br)c2-3)c(F)c1 59960,C1(C(N(CCC=C)CC)=O)CC2(CC2)CN1C(c1cn(CCO)nn1)=O 59961,C1(NC(c2nc(C(C)C)sc2)=O)CC2(CCCCN2C(C2(O)CCC2)=O)C1 59962,C(=O)(C(F)(F)c1cncs1)NCC(C)NC(=O)C(c1ccc(Cl)s1)C 59963,N1(CC(N2C(c3ccc(C)cc3)CCC2)=O)C(=O)CN(C)C1=O 59964,Cc1nc(N2CCCC2C(=O)Nc2cccc(S(=O)(=O)O)c2)nc2ccccc12 59965,C1(O)(C(=O)NCC2(F)CC(NC(C(C)(C)NC(C)=O)=O)C2)CN2CCC1CC2 59966,C#CCCN=C(NCCc1ccccc1C#N)NCc1ccn(C)c1 59967,CC1C(C)N(C(=O)CSc2nnnn2C)CCN1C(=O)C(=O)C(C)(C)C 59968,N1(C(COC(C)=O)=O)CC(NC(C2(C)CC=CC2)=O)CC12CCC2 59969,C(CC(C(=O)N1CCCCC1CCNC(=O)CCCn1ccnc1C)OC)OC 59970,c1(C(N2CC3CN(Cc4ccc(Br)cc4I)C3C2)=O)nc2ccccn2n1 59971,c1(-c2cn(C3CCN(C(=O)NC4CC(O)C(F)C4)C3)nn2)ccc(F)c(F)c1 59972,N1(C(CC2CC(OC)C2)=O)CC(C(=O)Nc2cc(C)cnc2O)CC(C)C1 59973,C(=O)(C1=CCCCO1)NCCCCCCNC(CCC1CCCN(C)C1)=O 59974,c1(C(=O)NC(CCN(C)C(C23CC4CC2C3C4)=O)(C)C)ccc2c(n1)CCCN2 59975,C(C1C(C(=O)N(CC(C)NC(=O)CCC2CCCO2)C)C1(C)C)=C(C)C 59976,CC1(C)CNC(=O)C1NC(=O)C(=O)N(C1CCC1)C(c1ccc(F)cn1)=O 59977,c1(C2(C(=O)NCC=CCNC(CCC(C)OC)=O)CC2)ccccc1C#N 59978,C1(NC(C=COCC)=O)C2CCCC1CC(NC(=O)C(O)CCSC)C2 59979,c1(C(N2CC(CNC(C(c3ccccc3)NC(N)=O)=O)C2)=O)cc[n+]([O-])cc1 59980,C1(O)(CNC(c2c(C)cno2)=O)CCCN(C(C2(N3CCOCC3=O)CC2)=O)CC1 59981,C1(NC(C(CNC(c2c(NC)scn2)=O)(C)C)=O)CN(C)C(C)(C)C1 59982,Cc1ccc(C)c(CCCC(=O)NC2(CN(C(=O)COCC(C)(C)C)C)CC2)c1 59983,C#CC1(NC(=O)C=CCC2(NC(=O)CCc3ncccn3)CCC2)CCC(C)(C)C1 59984,c1(C(COCC(=O)NC2CCC(NC(C3(SCC)CC3)=O)C2)C)ccc(Cl)cc1 59985,C(C(=O)NC(C(=O)NOCCc1ccccc1)c1cnn(C)c1)(C(C)C)SC 59986,C(=O)(C(C)(C)C)NCC(C)(C)O.C(C(=O)N(CC#N)C1CC1)N(C)CC=C(C)C 59987,c1(C(=O)NCC2(O)CCN(C(C(C)OCC)=O)C2)coc2cccc(O)c12 59988,C(=O)(C1=C(Cl)CCOC1)N1CCC(CC)CC1C(N1CCC1(C)C)=O 59989,C12(C(=O)NCC(CCC)C)CCCC1CCN2C(c1cncc(C)c1)=O 59990,CC1(C)CCCN(C(c2cscn2)=O)C1CNC(=O)CSCc1ccccc1 59991,C1(C(=O)NC2CC(OCC(=O)NCCC(O)C3CCC3)C2)CCCC(F)C1 59992,C=C(C)CCC(=O)NC(CN(C(=O)C(C)(c1ccccc1)OC)C)(CO)CO 59993,CC1(C)Cc2cc(Br)ccc2C1NC(=O)C(N1CCC(C)(C)C1C)=O 59994,N1(C(=O)CC2COC(=O)C2)CCCN(C(=O)C(=O)NCC(F)(F)F)CC1 59995,C1(F)(C(=O)NCCCC(C)NC(C2(c3ccnn3C)CC2)=O)CCCN(C)C1 59996,C(C(O)CC(=O)NCc1nonc1C)NC(c1cc(C(C)=O)on1)=O 59997,c1(CCN(CCc2ccc(C=C)cc2)C2CC2)ccc2c(c1)CCO2 59998,C1(OC)(CNC(=O)CSCC(F)F)CCN(C(=O)Cc2cnc(C)[nH]2)C1 59999,N1(C(c2ncn(C)c2)=O)CC2ON=C(CNC(c3ccc(NC=O)cc3)=O)C2C1 60000,c1(NC(C(c2csc(Cl)n2)N(CC(=O)OC)C(C)C)=O)ccc(C(=O)OC)cc1 60001,c1(OC)ccc(CN2CC3CC3(C(=O)Nc3cc(Cl)ncc3Cl)C2)cc1Br 60002,C1(CC(=O)NC2(C(N(C(C)C(N)=O)C)=O)CC2(C)C)C(C)(C)C1(C)C 60003,Cc1nc(C)c(CC(=O)NCC(C)(C)CNC(c2cc(C3CCCC3)no2)=O)s1 60004,C1(NC(CC=C)=O)CCN(C(c2ccnc(OC(C)C)c2)=O)C(C)C1 60005,N1(C(CC=C(C)C)=O)CC2CC(NC(=O)C(C(C)C)n3ccnc3)C1C2 60006,N1(C(c2scc(OC)c2)=O)CCCC(F)(C(N2CCC(C#N)C2)=O)C1 60007,Cc1c(F)ccc(C(=O)NCc2c(O)cccc2Cl)c1C 60008,c1(C(N(CCCCCC)CCNC(=O)C(C)(O)COC)=O)cc(F)c(F)c(Cl)c1F 60009,c1(C(N2CC(C(=O)Nc3nnc(C)o3)C(O)CC2)=O)cc2cccc(O)c2[nH]1 60010,Cc1cc(F)ccc1Cn1nnnc1N.C1(N2CCOCC2)(C)CCCOC1 60011,CC1=C(C(=O)NCCCN2CCC(NC(=O)CC3CCOC3=O)C2)CCO1 60012,c1(CC(=O)NC2(C)CN(C(CCCOC)=O)C2)c[nH]c2cc(OC)ccc12 60013,CC1(C(=O)NCc2cc(F)cc(Cl)c2)CCN(c2ccc(Cl)nn2)CC1 60014,C1(CC(N2CC(O)(CN(C(c3cc(C(C)=O)oc3)=O)C)C2)=O)COCCOC1 60015,N1(C(c2ncc(OC)nc2)=O)CC2=C(C1)CN(C(=O)C(C)c1cccs1)C2 60016,C(=O)(C(F)(F)C(F)F)NCC(CN(C(C1CCCC1C(F)F)=O)CC)(C)C 60017,C(C(CNC(C1(Cc2cnn[nH]2)CCCC1)=O)CO)NC(c1cscn1)=O 60018,N1(C(C(C2CC2)OC)=O)CCC(CNC(c2cnn(C(C)C)n2)=O)C(F)(F)CC1 60019,c1(N2CCC(C3N(C(CCCC(C)=O)=O)CCC3)C2)nc2cccnc2s1 60020,Cc1sc(Br)c(C(=O)NC2CC(F)CN(C(=O)C(C)CC(C)C)C2)c1C 60021,CC1CN(C(C2(C#N)CC2)=O)CCN1C(=O)C(C)C(F)(F)F 60022,Cc1cccc2cc(C(=O)NC(C)CNC(=O)C(c3ccc(C#N)cc3)C)nn12 60023,C1(C)(C(=O)NC(CNC(c2nn(CC)c(O)c2)=O)CO)CC(C(F)(F)F)=NO1 60024,N1(C(Cc2ncc(CC)[nH]2)=O)CCCC(NC(c2c(C)nc(C)n2O)=O)CC1 60025,Cc1ccc(C=CCC(=O)NC2(CCNC(C3CC3F)=O)CC2)cc1 60026,Cc1c(C(=O)NC2(C)CC(NC(=O)C(O)C(F)(F)F)C2)sc2nnc(S)n12 60027,N1(C(c2c(C)coc2C)=O)CCC(NC(c2cnn(C)c2C(F)(F)F)=O)C(F)C1 60028,c1(C(=O)NC(C2CCCN(C(c3cc(C(C)=O)on3)=O)C2)C)cccc(Cl)c1F 60029,c1(CC(=O)N(CC(CC)NC(C2CC2(C)C)=O)CC)cc(=O)n(-c2ccccn2)[nH]1 60030,C1(NC(C2C(OC)C2)=O)CN(C(=O)CC2CC2)CC1c1ccnn1C 60031,N1(C(C2C(C=C)C2)=O)C(CNC(c2c[nH]nc2C(F)F)=O)CC2CCCC12 60032,CCC(C(=O)NCC1(C2(O)CN(C(=O)C(C3(O)CCCC3)F)C2)CC1)C(C)(F)F 60033,n1(CC(N2C(CN(C(c3n(C(CC)C)ncc3)=O)C)CCC2)=O)cccnc1=O 60034,c1(CC(=O)N(CC(C)NC(c2cccc(OC(F)F)c2)=O)C)ccc(O)cc1 60035,O=C1CC(C2(C(N3CCCC(N4CCOCC4)C3)=O)CC2)C(=O)N1 60036,C=C1CCCN(S(=O)(=O)CC)C1.C1C(C)C(=O)N1C(N)=O 60037,N1(C(c2c(NC)cccc2OC)=O)CC2(CC(N)C(O)C2)C1C(=O)OC 60038,CCC(C)(COC)C(=O)NCC1CCCC1NC(=O)Cn1cc(C(=O)OC)nn1 60039,C1(F)(CNC(C=CCOC)=O)CCCN(C(c2ncc(C)cc2C)=O)C1 60040,N1(C(C=CC(C)NC(C(C)OCCOCC)=O)=O)CC(F)(C(N)=O)C1 60041,Cc1cc(NC(=O)C(N2CCCC2CC(c2ccccc2)O)=O)c(C)s1 60042,N(C(=NCCc1ccc(F)cc1C)NCCF)CC1(OCC)CCSC1 60043,C(CCC(C)C(=O)N1CC(C)(C(=O)NCC2CCC(=O)NC2C)C1)OC 60044,N1(C(c2cccc(OC)n2)=O)C2CCC1C(CNC(c1cc(C)cc(Cl)n1)=O)C2 60045,c1(C(=O)NC(C(C)(C)NC(C(C)SCCCC)=O)C)cc(F)ccc1F 60046,O=C(CCN=c1[nH]ccs1)NC1CC(NC(c2ccn(C3CCCCC3)n2)=O)C1 60047,N1(C(C23CCC(N=[N+]=[N-])C2C3)=O)C2CCCC1CN(C(=O)C=C1CCC1)C2 60048,C1(CNC(c2csc3nnsc23)=O)CC2CCC(C1)N2C(c1cscn1)=O 60049,c1(NC2CC(CC#N)C2)cc(Br)ccc1S(=O)(=O)N1CCSC(C)(C)C1 60050,c1(C(N2CCC(Cc3cn(CCC(C)C)nn3)C2)=O)ncc(Br)cc1Cl 60051,O=CN1CCCC1C(N1CCC(CNC(=O)Cc2cnco2)C1)=O 60052,c1(NC(c2ccc(-n3cncn3)cc2)C)nc2c(F)cccc2n1C 60053,Cc1ccc2ncnc(N(C(=O)CCC3CCC3)CC3CNCCO3)c2c1 60054,c1(C(N2CCCC(N(C(=O)Cc3n[nH]c(=N)s3)C)CC2)=O)cnc2[nH]cncc1-2 60055,C1(CNC(CC2C(C)CC2)=O)(NC(=O)CCCN2CCCC2)CCCC1 60056,N1(C(C2C(C3(C)COC3)C2)=O)C2CCC(C(N3CCCC(F)(CO)C3)=O)C1CC2 60057,C(=O)(C(O)CC(F)(F)F)N1C(CC)C(C(=O)NCC(C)Cc2cn[nH]c2)CC1 60058,c1(CNC(CC2=CCN(C)CC2)=O)cccc2c1CCN(C(c1cnns1)=O)C2 60059,Cc1nc(C2CC2)ncc1C(=O)NCC1CCCCCN1C(=O)CNC=O 60060,c1(C(N(C2CCCNC2)CC)=O)ccc2c(c1)C=CC(C)(C)O2 60061,CN1CCN(C(=O)CC2CCCC(=O)N2)C(CNC(c2nccc(Cl)c2O)=O)C1 60062,C12(NC(c3ccc(OCC=C)cc3)=O)CCC(CC1NC(=O)CNC(N)=O)C2 60063,c1(CC)ccccc1C(C(=O)NC1CCCC1)N(n1ccnc1C)CCOC 60064,c1(OCC)cc(C(=O)NCC(CNC(C2(CC)CC2(F)F)=O)CO)ccn1 60065,c1(C(N2CCC(N(C(=O)COCC(F)F)CC)C2)=O)c(C)ccc(C)c1O 60066,C(CNC(C1CC1c1ccn(C)n1)=O)(CC(C)C)NC(c1nc(OCC)sn1)=O 60067,CC(C(=O)NCCC1(NC(c2ccc(C(C)(C)C)cn2)=O)CCC1)S(N)(=O)=O 60068,c1(C(=O)NC2CC(CNC(C3(COC)COC3)=O)C2)sc(C)c(C)c1C 60069,C(=O)(CCC(C)(C)NC(C12CSCC1C2)=O)NC(c1cn(C)cn1)C 60070,C1(NC(CCNC(C(COCC)(C)C)=O)=O)COC2(CCCC2)C1 60071,C1(NC(C2CCC3C(C2)C3(F)F)=O)CC2CCC(C1)N2c1nnc(C(F)(F)F)s1 60072,CC1CN(C(=O)CC2OCCC2C)CC(C)C1N=c1[nH]c(Cl)ncc1F 60073,N1(C(=O)COCC2CC2)CC2CCC1(CC1(F)CC1)C2 60074,N1(C(CN(C)CC)=O)CCC2CC1CN(C(=O)CCc1cnc3n1CCCC3)C2 60075,CC1(C)OCCN(Cc2ccncc2Br)C1c1ccccc1 60076,Cc1cc(=NCC2C(C)CCCN2C(c2cccc(O)n2)=O)[nH]c(CO)n1 60077,Cc1nc(N(CC(F)(F)F)CCC#N)cc(N2CC3CCC(C2)O3)n1 60078,N1(C(c2ccc(CC)[nH]2)=O)CCOCCC1C(=O)NC(c1cc(C)on1)C 60079,c1(C(C(=O)NCC2N(CCc3nc(C)sc3)CCC2)(C)C)cc(F)cc(F)c1 60080,c1(CC)ccccc1CC(=O)NCC12CC1CN(C(C1CC(SC)C1)=O)C2 60081,C12(CNC(=O)C3=CCCCCC3)CCCC1N(C(c1cccc(O)n1)=O)CCC2 60082,c1(C(=O)NCC(CNC(C(C)=C2CCC2)=O)O)cnc2nc(C)ccc2c1O 60083,c1(C(N2CCC(CC(C)(C)C)C2)C(=O)NCC)cncn1C 60084,C1(CNC(COC2CCN(C(c3c(OC)scc3)=O)C2)=O)C(C)(C)C1(F)F 60085,CN1CC2CC1CN2C(=O)CC1CN(Cc2cc(Br)ccn2)CCO1 60086,C1(C(C(=O)NC(C)C)N(CC(C)(C)S(C)(=O)=O)C)CC2(CCC2)CO1 60087,C1(C(N2CC(SC(C)C)C2)=O)(COC)CN(C(=O)CC23CCCC2C3)C1 60088,C12(NC(c3nc(CC)sc3N)=O)CCC(CNC(=O)C(C)CSC)(CC1)OC2 60089,C(=O)(C1(C)CCn2ccnc21)NCCN(C(CCCCC=C)=O)CCC 60090,C(=O)(CC(C)C(F)(F)F)NC1(C(N2CC(CC)C(O)C2)=O)CC1 60091,C(CC)(CC(=O)N(C)CP(C)(C)=O)N(C(CN(CCC)C)=O)C 60092,C1(F)(CNC(c2ccon2)=O)COCCN(C(c2ccc(Cl)s2)=O)C1 60093,N1(C(C(C)CC(F)F)=O)CC2(CCCC2NC(c2cc(-c3ccco3)c[nH]2)=O)C1 60094,c1(C(C)C)scnc1C(=O)NCC(O)CNC(c1ncc(C(F)F)s1)=O 60095,C=C(C)CC(C(=O)NC1C2CCC1CC2)NC(C1CCN1CC)=O 60096,c1(C(=O)NC2CC(NC(CC(C)(C)OC)=O)C2)ccc(N(C)C)cc1F 60097,n1(CC(=O)NCC2C3CN(C(CC(=C)C)=O)CC32)cc(P(C)(C)=O)cn1 60098,Cc1ccc(C(N2CC(F)CC2C(N2CC3C(CN(C)C)C3C2)=O)=O)nc1C 60099,c1(CNC(CCOCCN(C(CC(C)CN(C)C)=O)C)=O)cccc2c1OCC2 60100,CC1CCCCC1(CNC(C1(C2CCCO2)CCC1)=O)NC(c1csc(O)n1)=O 60101,c1(C(CCC)N(C)C(=O)NCCc2nccn2CC)ccc(Br)cc1 60102,S(=O)(=O)(c1cnn(C2CCCC2)c1)NCCOCC=C 60103,N1(S(Cc2cccc(C)c2)(=O)=O)Cc2ccc(C(=O)Nc3cncc(Cl)n3)cc2C1 60104,C1(C(=O)NC2(CC=C)CN(C(C3CC4CCC3CC4)=O)C2)CC2CCC1CC2 60105,c1(C(=O)NC(C(C)NC(=O)CCN2CCOCC2=O)CO)nc(O)nc(O)c1F 60106,c1(NCC2CC(OC)C2)nccc(=NCC2CCN(C3CC3)C2)[nH]1 60107,N1(C(CC)C(=O)NC2CC3CC2N(C(=O)CSC2CC2)C3)CCc2ccccc21 60108,C(=O)(C(CCF)NC(=O)CCOC(C)C)N1C(C(=O)OC)CC1C 60109,N1(C(c2ccc(SC)cc2)=O)CC(NC(c2cc(Br)ncc2F)=O)C(F)(F)C1 60110,CC1(C)CCCC1(C)NC(c1cnc(CNC(=O)CC2COCCO2)nc1)=O 60111,c1(C(C)(C)C)nc[nH]c1S(=O)(=O)NC12CC1CS(=O)(=O)C2 60112,c1(CNC2CCCC(C)C2)cc(Cl)c(Br)cc1F 60113,c1(N2CCC(SC)C2)nc(N(C)CC2CN(C)C2)nc2cc(C)ccc12 60114,C1(C(=O)NCCCCNC(COCCSC)=O)(N(C)C)CCCSC1 60115,c1(N2CCCC(CCCC)C2)nc(=NC)nc(N2CCOC(C(C)(C)C)C2)[nH]1 60116,N1(C(CCCn2cnc(C#N)n2)=O)CCC2CCN(C(=O)COC3CC3)C2C1 60117,C(=O)(C(F)C(F)(F)C(F)(F)F)N1CCCC(NC(c2ccc(COC)[nH]2)=O)CC1 60118,C(=O)(C(CCC(C)C)N=C1NS(=O)(=O)c2ccccc21)NCCNC(=O)NC 60119,c1(OC)cc(C(=O)NC2CCC(NC(c3c[nH]c(Br)c3)=O)CC2)c2c(c1)CCO2 60120,c1(C(=O)NC2CC(CNC(CCC3C(C)=NNC3=O)=O)C2)cncc(Cl)c1Cl 60121,N1(C(CC(C)SC)=O)CC2(C1)OC1(C)CC2(NC(=O)C(C)Oc2ccccn2)C1 60122,C1(NC(C2(OCC)CCOCC2)=O)CCC(C)N(c2ncc(Br)c(C)n2)C1 60123,N1(C(CCCNC(C)=O)=O)CCC(C)(C)CC1C(=O)NC1(C)CC(C)C1 60124,CC1(C)OC(=O)c2cc(C(N3CC(O)(CNC(C4CC4(F)F)=O)C3)=O)ccc21 60125,C(=O)(C(CC)CCCCC)N1CCCC(O)(CNC(C(CC=C)(C)C)=O)CC1 60126,C1(C(=O)NC(C2CCN(C(c3conc3C(C)(C)C)=O)CC2)C)CCS(=O)(=O)C1 60127,c1(OC)ccc2c(=NC(C)CCF)[nH]c(=NCc3ccc(C)c(N)c3)[nH]c2c1 60128,Cc1cc(OCCC(=O)NCC2(F)CCCN(C(=O)CCC(F)F)C2)cc(C)c1 60129,C#CCC(C)(CNC(=O)CCCN(C)C(C1CC2CC2C1)=O)CO 60130,CC1SCCC1N=c1nc(N2CCCC(F)C2)c2c([nH]1)COC2 60131,Cc1ncc(C=CC(=O)NCC2COCCN2C(=O)COC2CC=CC2)s1 60132,c1(OC)c(C)ccnc1NC(N1CCC(N2CCC(F)CC2)C1)=O 60133,C(=O)(CC(=O)NC1C=CC(CNC(=O)C(F)CC2CCC2)C1)OC 60134,N1(C(c2cnc(CC)s2)=O)CCCN(C(c2cnc(O)c(C)c2)=O)CCC1 60135,c1(C(=O)NCC(C)F)cc(O)nc2c1CN(C(C1CC1(Cl)Cl)=O)CC2 60136,C1(N(CCCC)C)CCCN(N2CCC(OCC3CC3)C2)C1 60137,C1(C(=O)NC(C(=O)NCCOCC#C)c2ccoc2)CCS(=O)CC1 60138,C=CCC(C(=O)NC1CCN(C(=O)C=C2SCC(=O)N2C)CC1F)C(C)(C)C 60139,C=CC1(O)CN(C(=O)C(C)N(C(=O)CC2CC3C=CC2C3)C2CC2)C1 60140,Cc1nc2ccc(C(=O)NC(C)CNC(c3cc4ncc(C)cn4n3)=O)cn2n1 60141,C1(CC=C)CCN(C(c2nc(C)cs2)C(=O)NCCCSC)C1 60142,C(CCC(N)=O)(C(=O)NCc1ccnn1C)n1cc(CC(C(=O)OC)C)nn1 60143,C1(F)(CNC(C=CCCC)=O)CCCN(C(=O)CCn2c(C)c(C)sc2=O)C1 60144,Cc1ccc(C(=O)NC2CCC(CCNC(=O)CCC3CCCC(=O)N3)C2)nn1 60145,C12(CCCO1)C(=O)OC2.c1(C(=O)NC2CCCC2)ccns1 60146,C(=O)(CC(C)(C)C(F)(F)F)NCC1N(C(CCOC)=O)CCC1C1CC1 60147,c1(SC)ccc(C(=O)NC2CN(C(=O)CC3COC(C(F)(F)F)C3)C2)cc1 60148,CC(C)(C(=O)NCCC1CCCN1C(C1(F)CCOC1)=O)C(F)(F)F 60149,Cc1cc(C(=O)N(C)CCN(C(=O)C2=NOCC2)C)c2[nH]cnc2c1 60150,N1(C(COCCOCCOC)=O)CC2CCC(NC(C3CCC3C(F)F)=O)(C2)C1 60151,CCC(CC)C(F)C(=O)NCC1(C)CN(C(C2CCCN2CC(C)C)=O)CCO1 60152,Cc1cc(C)c(C)c(C(N2CC(F)(CNC(=O)Cn3nnnc3C)C2)=O)c1C 60153,C1(COC)CC2CC1(CNC(c1oc(C)nc1C(F)(F)F)=O)C2 60154,C1(NC(Cc2cc(C)sc2)=O)CC(O)CN(C(c2c(O)cccc2F)=O)C1 60155,c1(CNCC(=O)NC23CC2C3)cccc(OCCF)c1 60156,C1(C)(C(N(C(c2ccco2)C)C)=O)CCCN(C(=O)CCc2cncn2C)C1 60157,c1(OC)nc(OC)nc(N2CCC(C(N3CC4CCCC4C3)=O)C2)n1 60158,c1(C(N2CCC(C(=O)O)(COC)C2)=O)ccc(Br)c2cccnc12 60159,C(CCSC)(C(N)=O)NC(C(C)N(CCC)C(c1ccc(Cl)cc1)=O)=O.C(C)=O 60160,C1(C(N2CCC(=C)CC2)=O)CN(C)CCN1C(=O)Cn1ccnn1 60161,c1(C(N)=O)cccc(C(N2CCOCC2CNC(=O)C=C2CCC2)=O)c1N 60162,C1(C(=O)NC2(C)CN(C(CC3(CC)CCC3)=O)C2)COc2c(OC)cccc2C1 60163,CCC(CC(=O)NCC=CCN(C(=O)CC1OCCC1C)C)CCOC 60164,c1(CN2CC(O)(c3ccccn3)C2)cc2c(O)cccc2s1 60165,C(CC(C)CCO)NC(c1cncc(C(C)(C)C)c1)c1n(CC(=C)C)nnn1 60166,N1(C(C(C2CCCC2)OCC)=O)CCN(C(=O)CS(=O)CC)CC12CC2 60167,c1(SCC)nc(C)c(C(CC)C(=O)NC2CC(C)(NC(=O)CC3CC3COC)C2)s1 60168,C=C(C)CCC(=O)NC(C1CCN(C(=O)C(C)N(CC(F)(F)F)C)CC1)C 60169,N1(C(C(C)OCOC)=O)CCC2CN(C(=O)COC3CC3)CC2C1 60170,c1(C2(C(=O)NCC(C)(CO)NC(c3cnc(OC)s3)=O)CCC2)cccc(Cl)c1 60171,C1(CC)CCC(C)CN1C(C1CC2CC2N1C(=O)C(C)C(C)COC)=O 60172,C1(N(C(c2n(CC)ncc2)=O)C)CN(C(c2cn(C)nc2COC)=O)CCC1O 60173,C1(NC(C2C=CCC2)=O)CC2(C1)CC2C(=O)Nc1ccc(Cl)cc1 60174,c1(CCC)cc(C(=O)NCC2COC(CNC(=O)CN3CCOCC3)C2)c(C)o1 60175,CC12CSCC1CN(c1ncncc1Br)C2 60176,c1(C(=O)NCC2CCCN(C(C=CC3(C)COC3)=O)C2)ccc2ccsc2c1 60177,c1(C(=O)OCC)nnc2n1CCN(C(C(C)=Cc1ccccc1)C(=O)NC)C2 60178,C1(C)(C(=O)NC2CN(C(C=C(CCC)C)=O)CC2O)CCS(=O)(=O)CC1 60179,c1(C(N(C(C2CCCC2)C)C)=O)ncccc1NC(=O)Nc1ccco1 60180,c1(OCCC)cccc(C(=O)NCC(O)CNC(=O)CCc2ccc(C)nc2)c1 60181,C1(CCCN(C(=O)CN2CC3CC3C2)C(C2COCC2NC2CC2F)=O)CCCCCC1 60182,C12(CNC(C3CCCO3)=O)CCCC1N(C(c1cc3sccc3s1)=O)CCC2 60183,C1(CNC(C2CC(CF)C2)=O)C2CN(C(=O)CCc3ncc[nH]3)CC12 60184,C(C)(C)(C#CCCC)NC(C1CC(CCNC(C(C=C)(C)O)=O)C1)=O 60185,C(C(C)(CO)Nc1csc(CCP(C)(C)=O)n1)NC(C=CC(=O)N(C)C)=O 60186,C(=O)(C(C)(C)CN1CCCC1)N(C)CC1CCN(C(C2C(C)C2C)=O)C1 60187,C12(C(=O)NC(CC(=O)NC)C3CC3)CC1CN(C(=O)CCc1cn(C)nn1)C2 60188,N1(C(C(COC)C)=O)CCN(C(=O)Cc2ccc(Br)s2)C(CO)C1 60189,C(=O)(C(F)C(C)CNC(=O)CCC(C)(C)OC)N1CCC(OC)C1C(C)C 60190,C1(C)(C(=O)NC(C)CCNC(=O)Cc2cnoc2)CC1(F)Cl 60191,c1(OC)ncnc(C(=O)NCC2CC2NC(c2ccc(C(C)C)cc2)=O)c1F 60192,c1(C(=O)NC(CC)CNC(c2cc(Cl)n(C)n2)=O)c(O)nnc2c1CCC2 60193,c1(C(=O)NC2C(NC(c3ccc(C(N)=O)cc3)=O)C2)cccn2ccnc12 60194,Cc1cc(O)ccc1C(N1CCC(NC(c2cnsc2C)=O)CC1C1CC1)=O 60195,C1(NC(C(C)OC)=O)CN(C(=O)CCS(=O)(=O)N(C)C)C(C)(C)C1 60196,C(=O)(CCCn1cc(CCC(N)=O)nn1)NCC(=O)NC(C)(C)C 60197,C(CC(=O)N1CCOC(CCC)C1)(C(C)C)NC(CCC=C)=O 60198,C1(NC(C=C(CCC)CCC)=O)CCC2CN(c3ncc(C)c(SC)n3)CC2C1 60199,C(C(CC(C)C)C(=O)NC1CC(CNC(C23CCC(N=[N+]=[N-])C2C3)=O)C1)OC 60200,CC(C)C(S(=O)(=O)Nc1ccc(I)c(Cl)c1)c1ccccc1 60201,N1(C(c2cc(CC)n(C)n2)=O)CC2CC1CN(C(c1cnn3cccnc13)=O)C2 60202,c1(C(=O)NC(C(CO)NC(c2cc(C)cc(C)c2)=O)C)cc2n(n1)CCCC2O 60203,CCCCC(C(=O)NC(c1cncnc1)C)NC(=O)CSC(F)(F)F 60204,CCC(C)(COC)C(=O)N1CCN(CCNC(=O)C=CS(C)=O)CC1 60205,N1(C(CCC#C)=O)CC=C(C(C)(C)C(=O)N(C(C)COC)C)C1 60206,C(CNC(c1cnc(C)n1C)=O)(CC(=O)NCCN(C)C1CC1)OC 60207,C1(CCNC(c2c(COC)ccs2)=O)COCCN1C(=O)CC1CCC(C)(C)C1 60208,c1(C(N(CC(C)NC(c2c(O)ccc(C)n2)=O)C)=O)cnc2c(c1)OCC(=O)N2 60209,C(CNC(C1CC2CC2C1)=O)(C(=O)N=c1cc2n([nH]1)CCCC2)N(C)C 60210,C(C(=O)N(CC(O)CN(C)C(c1nncs1)=O)C)(C1CCOC1)OCC 60211,CC(C)CC(C(=O)NCC1CCOC1(C)C)NC(=O)CCC(F)(F)F 60212,CC1(C)OC(=O)CC1C(N1CC(C(O)C(=O)NCCC2NC(=O)NC2=O)C1)=O 60213,C1(C(C)C)CN(C(c2ccns2)=O)CCN1C(c1c[nH]c(=S)cn1)=O 60214,N1(C(c2cnn(CC)n2)=O)CCC(C2CC2NC(=O)C(C(C)C)OC)CC1 60215,C(C(C)(C)C(=O)NC1CCC(CNC(=O)CC2CC2(C)C)C1)N(C)C 60216,C1(C2CC2)(C(=O)NC2C(NC(c3ccc(COC)o3)=O)CC2)CC=CC1 60217,c1(CC(N2CCC(NC(C(COC)C)=O)C23CC3)=O)cnc2n1CCOC2 60218,CC1C(NC(C2CC23CCC3)=O)CCN1CC(N1CCC(O)CC1)=O 60219,C(=O)(CCCC(C)(C)C#N)N1C(C(=O)NCc2c(CC)onc2C)C(CC)CC1 60220,c1(C2(N(C(CC(=O)NCCOCC#C)=O)CCC3CC3)CC2)ccccc1Cl 60221,O=C(C1CCSc2ccccc21)NC1CCCN(C(=O)Cc2cnccn2)CC1 60222,c1(C(=O)NCCCN(C(c2cncc3nc[nH]c23)=O)CC)n[nH]c2c1NCCC2 60223,N1(C(CCC(C)C#N)=O)CC2(C1)OC1(C)CC2(NC(c2c(Cl)cnn2C)=O)C1 60224,CC1(C(=O)NCCCN(C(=O)Cn2ccnn2)CCO)CCCS1(=O)=O 60225,Cc1cnc2nc(C(=O)N(CC(C)(C)CNC(=O)C=CC3CCCO3)C)nn2c1 60226,N1(CC=C)CC2CC2(C=O)C1.c1(C(=O)NCC=CCN(C)C)cn(C2CC2)cn1 60227,C1(C)(CC)C=C(C(=O)NCC(C)CC(=O)N2CC(N(C)C)C(C)C2)C1 60228,CC1NC(=O)OC12CN(C(=O)CCOCCCNC(=O)CCc1ccccn1)C2 60229,N1(C(CCCCOCC)=O)CCC2(CC(NC(=O)C(C)NC(C)=O)C2)C1 60230,c1(C(=O)Nc2c(C)c(Cl)ncc2)cc2cc(-c3ccc(N(C)C)nc3)cnc2[nH]1 60231,c1(C(N(C(Cc2cn(C(C)C)nn2)C)C)=O)cc(C(F)F)ccn1 60232,C1(C(=O)NCC(CNC(c2cc(Cl)ccc2O)=O)O)CC12CCOCC2 60233,c1(OC)ccnc(F)c1C(N1CCC(O)(C(=O)NCc2nccnc2Cl)C1)=O 60234,CCC(CC)(CO)C(=O)N1CC(C)(NC(=O)CC2CCCCC2F)C1 60235,CCCC(CC)C(=O)N(C1CCCN(C(c2cc(O)nn2C)=O)C1)CCO 60236,N1(C(CCc2c[nH]c(=N)[nH]2)=O)CCCC(NC(C2CCNC2=O)=O)CCC1 60237,O=C1CCC2(CCCN(C(=O)Nc3cccc(CCO)c3)C2)CN1 60238,O=C(CCCCCCNC(C1CCCC1)=O)NCC1CCC2(CC2)CO1 60239,N1(C(C(C(C)C)C2CCC2)=O)CC(C(N2CC(N(C)C)C(C)C2)=O)C(F)(F)C1 60240,CC1CN(C(c2c(C(F)F)cnn2C)=O)CCCN1C(C1CNC(=O)N1C)=O 60241,C1(NC(C2N(CC)CC2)=O)CCC(N(C)C(C2(C)CC(C)=NO2)=O)CC1 60242,N1(C(c2c(O)nc(=N)[nH]c2)=O)CCCC(C2(NC(=O)COCCO)CC2)C1 60243,C(C(C)C(=O)N(C1CCC1)CCO)N(C(C(C)C)=O)C 60244,C1(NC(C(C(C)(C)O)NC(C2C=C(C)CS2)=O)=O)CCN2CCCCC12 60245,c1(N2CC3(CCN(C(c4cnn(C)n4)=O)C3)C2)nc2ccccc2cc1C1CC1 60246,c1(CC)cc(C(=O)N(C)CCN(C(C2CCOC(CC)C2)=O)C(C)C)ncn1 60247,CC1CN(C(c2cc(Cl)no2)=O)CCC1N(C(=O)CNC(S(=O)(=O)C1CC1)=O)C 60248,C1(C)(OC)CCC(NC(C2CN(C(C3CCC3C)=O)CC2(F)F)=O)CC1 60249,c1(C(=O)NC2CCC(N(C(=O)CCC3CCCCC3)C)C2)ccn2nccc2n1 60250,c1(CC)c(C(N2CCCC2CNC(=O)CN2C(=O)CNC2=O)=O)cnn1C 60251,C1(F)(C(N(CCN(C(C(C)SCC)=O)C(C)C)C)=O)CCOC1 60252,N1(C(CC2(OC)CN(C(c3cn(C)c(C)n3)=O)C2)=O)CC2(CCC(=O)N2)C1 60253,c1(CC(C)C(=O)NCCCCNC(C2CCOC2C(F)(F)F)=O)cccc(Cl)c1 60254,C1(C(c2n(CCC)nnn2)NCC(C)(C2CC2)OC)CCC(C)(C)CC1 60255,C1(CN(C)C(C23CCC2CC3)=O)CCCN(C(c2cnccc2Br)=O)C1 60256,c1(NC(c2c(-c3cc(C)cc(F)c3)cncc2F)=O)ccc(S(C)(=O)=O)cc1F 60257,C(=O)(C1=CS(=O)CCC1)N1CC(NC(c2cc(CC)nc(O)c2)=O)C(CO)CC1 60258,C1(CNC(c2cc(CF)on2)=O)CN(C(C2(O)CCSCC2)=O)CC12CCC2 60259,C1(CNC(=O)CCCF)CCCCN(C(c2cc(Cl)cc(C(F)(F)F)n2)=O)C1 60260,C1(CNC(CN(C2CC2)CC)=O)CN(C(=O)CCC#N)CC(C(F)(F)F)O1 60261,c1(C(=O)NC2CC(C(C(=O)NCCCCSC)F)C2)nocc1Cl 60262,c1(C(=O)NC(C)CCN(C)C)n[nH]cc1-c1ccccc1 60263,c1(C(=O)NC(c2cccnn2)C)csc(CCN)n1 60264,c1(C(=O)NCC2(F)CC(CNC(C(C)N(C)C)=O)C2)ccc(SC(F)(F)F)nc1 60265,C1(NC(=O)COCCF)CN(C(=O)CCCn2cncn2)C2(CCC2)C1 60266,N1(C(CCOCCNC(c2ccc(C)s2)=O)=O)CC=C(C(C)(C)C)CC1 60267,C(=O)(C(C)CCCCCC)NCc1c(C(N2C(C)(CCC)CC2)=O)con1 60268,C1(CNC(c2c(SC)cccc2)=O)CCCN(C(=O)Cn2nc(C)cc2C)CC1 60269,c1(C(N2CCCC(N(C(c3cnc(COC)s3)=O)C)C2)=O)coc(S(C)(=O)=O)c1 60270,C1(C(C)C)CCCCC1C(=O)N(C1CC(F)CN1C)CCN1CC(O)(C(F)F)C1 60271,N#Cc1ccc(CN2CCC(C(=O)Nc3nc(C4CC4)c(Br)s3)C(O)C2)c(Cl)c1 60272,N1(CC(N2CC(N(C(CC(C=C)C)=O)C)C2)=O)CCCCC(O)C1=O 60273,C(=O)(CC(C)(C)CC(F)(F)F)NC1(CO)CN(C(Cc2ccc(C)s2)=O)C1 60274,c1(OC)ccc(C(=O)NC2CC(NC(c3cnc(O)s3)=O)C(O)C2)c(N)c1 60275,C#CCC(C)(C(=O)NC(CO)CCC=C)NC(=O)C(C)C#N 60276,c1(NCc2c(NC(=O)Nc3c(C)cccc3)cnn2C)c[nH]c2cc(F)ccc12 60277,c1(C(N2C(CN(C(C(C)SC(C)C)=O)C)COCC2)=O)cnn2ccnc(N)c12 60278,S(=O)(=O)(c1ccccc1Cl)N1CC(CN(C(C(N2C(C)CCC2C)C)=O)CCO)C1 60279,CC(C)C(C(=O)N1CCCC(CC(=O)NCc2ncccn2)C1)N(C)C 60280,n1(C(c2nc(C3CC3C)no2)C)ncc2ccccc12.N12CCC(CC1)C2 60281,c1(C(=O)OC)ccc(NC(C2(C)CS(=O)(=O)C2)=O)c(I)c1 60282,C(=O)(CC1=CCOCC1)NC1C(CNC(CCOc2cc(C)cc(C)c2)=O)CC1 60283,c1(OC)ccc2c(=NC3CCCN(C)C3C)[nH]c(=NCCCCC#N)[nH]c2c1 60284,C1(C(N2CCC(N(C(=O)CC3CC=CC3)C)C2)=O)CCC(=O)N(C2CC2)C1 60285,Cc1cccc(C(N2CC(CC(=O)NC3(CC4CCC4)CC3)CC2C)=O)c1 60286,CC(C)(CC#N)C(=O)NC1COCCN(C(c2c[nH]nc2Br)=O)C1 60287,c1(C(=O)NCC2(C(N)=O)CN(C(C(=O)N(C)C)=O)C2)ccc(C2CCC2)nc1 60288,C1(C(=O)NCC(C)NC(C2(CO)CCC2)=O)CC2(CC(=O)C2)C1 60289,CCCCCCC(F)C(=O)N(C)CC1(O)CN(C(=O)CC(C)(C)c2cccs2)C1 60290,CC(C(=O)NCC12CCC(CC1)N2C(=O)CN1CCCCC1)C(C)S(C)(=O)=O 60291,CC1(F)CC2(CN(C(C3CCCN3C(=O)C(CO)C(C)(C)C)=O)C2)C1 60292,C1(C(=O)NC(C)CCCNC(=O)C(C)CF)(C(=O)OC(C)(C)C)CCCCC1 60293,C1(CNC(C(=O)NCCNS(C)(=O)=O)=O)CC2(CCNC2)CO1 60294,C1(F)(C(N(C)CCNC(C2CC23CCC3)=O)=O)CCCN(C(=O)OC(C)(C)C)C1 60295,Cc1cc(N(C2CCN(C(=O)C(O)CCc3ccccc3)C2)C)nc(C)c1C#N 60296,C12(NC(CN3CC(C)(C)C3)=O)CCC(CC1NC(c1cnn[nH]1)=O)C2 60297,C1(N(c2nnc(CC)o2)C)CCCN(C(c2snnc2C)=O)C1 60298,c1(C(N2CC(C#N)C(NC(c3cc(Cl)cnc3F)=O)C2)=O)c(F)ccc(I)c1F 60299,C(CCCOC)(C(=O)NCC(C)(C)CSC)NC(C(C1CCC1)OCC)=O 60300,CCCC(C)(C)C(=O)NC1CN(C(c2ccc(CC(C)C)s2)=O)C(C)(CC)C1 60301,C(CCCN(C(=O)C(C)c1ccon1)C)NC(C1(CC=C)CC1)=O 60302,c1(C(N(C2CCCN(C(c3n[nH]cc3[N+](=O)[O-])=O)C2)C)=O)ccc(S(C)=O)cc1 60303,c1(-c2cncc(C(N3CCCC(CN(C)CC4CC4)C3)=O)n2)ccc(O)cc1 60304,c1(C(N2CCCC(O)CC2)C(=O)NC(C)C)n[nH]c2cc(Br)ccc12 60305,n1(C(C)C)cc(C(=O)NCC(C(C)(C)C)NC(c2cn(CO)nn2)=O)ccc1=O 60306,CC1(C)CC(C(=O)NCC2(C)CCCN(C(C3CCC(C)CC3)=O)C2)CNC1=O 60307,S(=O)(=O)(c1cn(C(=O)OC)nc1C)CC1CC1.N12CCC(CC1)N(CC)CC2=O 60308,N#Cc1ccc2c(c1)CC(NC(C1CNCC(F)(F)C1)=O)C2 60309,C#CCC(CC(F)F)C(=O)N1CCC(N(C(c2cnc3cccnn23)=O)CC)C1 60310,c1(C(N2CC3C(CNC(c4c(C)n[nH]c4)=O)(C3)C2)=O)cnc2snc(C)c2c1 60311,N1(C(CSCC#C)=O)CC(C[N+](C(C2CCCN2CCC)=O)([O-])NC)CC1(C)C 60312,N1(C(C2C(C(C)C)OCC2)=O)CCCC2(C1)CN(C(c1ccnc(Cl)c1N)=O)C2 60313,C(CCCCC(=O)N(C)CCN(C)C(c1occc1C1CC1)=O)(OC)OC 60314,c1(OC)cc(-c2noc(COC(C3CCC3)=O)n2)cc(Cl)c1OC 60315,N1(C(C2(COC(C)C)CC2)=O)CC2CCC(C1)N2C(C1Cc2nncn2C1)=O 60316,c1(CCC(=O)N(C(C)C(=O)N(CCCCOCC)C)CCC)nccn1C 60317,O=C1CC2OCCC2(C(=O)NC2CCCC2NC(c2cnc(S)nc2)=O)CN1 60318,c1(C(C(=O)NC(C(CO)NC(CC(=C=C)C)=O)C)(C)C)ccc(Br)c(C)c1 60319,CC1CCN(C(=O)Cn2ccc(=N)[nH]2)C1CNC(=O)CCN1CCCCCC1 60320,c1(OC)noc(C)c1NC(=O)NCC(C1CCCC12CC2)(C)O 60321,N1(C(CC(=O)NCC)=O)CCC2(CC1)CC2NC(C1C=CCS1)=O 60322,C(=O)(C1CCCn2cncc21)NCC1(CNC(C(CCCC)O)=O)CCC1 60323,C1(C)(C(=O)OC(C(=O)NC)C)CC(C(C)C)=NO1 60324,C(C)(CCCCNC(C1CCOC1(C)C)=O)NC(c1ccc(CCCCCC)s1)=O 60325,N1(C(C)C(=O)NC(C)C(=O)Nc2ccc(Cl)cc2)Cc2ccccc2C1=O 60326,CN1CCC(C(=O)NCC2(F)CCN(C(c3ncncc3Cl)=O)CC2)S1(=O)=O 60327,N1(C(C2OCCN(C(C(CC=C)C(C)C)=O)CC2)=O)CCC2(CNC(=O)C2)C1 60328,C1(NC(C2N(C(c3cccc(C)n3)=O)C3(CC2)CC3)=O)CCc2ncnn2C1 60329,C1(CNC(c2cc(C(C)(C)C)n[nH]2)=O)C2CN(C(C3CC34CC(O)C4)=O)CC12 60330,C12(CNC(C=CCCC)=O)CC(NC(=O)C(C)C(F)(F)F)(C1)C1(CCOCC1)O2 60331,c1(CNCC2(C(N3CC(C(=O)OC)C(F)C3)=O)CC2)cc(I)ccc1Cl 60332,c1(C(N(C(C)CNC(C2(O)CCSC2)=O)C)=O)cnc2[nH]nnc2c1 60333,CCC(CNC(=O)CCP(C)(C)=O)(CC)C(=O)NC1CCC1(C)C 60334,C1(NC(c2n(CC)ncc2Cl)=O)CN(C(c2c(Br)n[nH]c2C)=O)CC12CC2 60335,N1(C(C2(OC)CCCC2)=O)CCC(C2(NC(=O)CCC(C)N(C)C)CC2)CC1 60336,N1(C2CCCN(C(C=CSC)=O)C2)CCN(C(=O)C(C)OCC(C)C)CC1=O 60337,N1(C(CC2OCCN(C(C3CCN(CC)C3)=O)C2)=O)CCOC(CC)(CC)C1 60338,C(=O)(C(CC)CCCCCC)N1CCC(CC=C)(NC(c2ncncc2I)=O)CC1 60339,c1(C(=O)NCC2C(C)CN(C(C3CC(O)C3)=O)CC2)c(F)ccc2cnn(C)c12 60340,N1(C(c2cc(OCC)c(C)cc2)=O)CC2CC(C)N(C(C3CCC4CC34)=O)C2C1 60341,C#Cc1ccc(CC(=O)NCC2(NC(=O)CC3(CO)CCCCC3)CC2)cc1 60342,C1(NC(CC2N(C(CC(CN(C)C)O)=O)CC2)=O)CC2(C1)CC(C#N)C2 60343,c1(OC(COC(C)=O)C(=O)NC(C2CCC(=O)NC2)=O)cc(C)cc(C)c1C 60344,N1(C(C2(CNC(C(CCC)C(C)C)=O)CCCO2)=O)CCc2nnnn2CC1 60345,C1(C(N2C(CNC(C(CC(C)C)(C)C)=O)C=CC2)=O)CCc2ccccc2CC1 60346,c1(OC)cc(Cl)c(CN2CCNCC2C(=O)NC(c2ccsc2)C)c(Cl)c1 60347,N1(C(C(CC)(C)C)=O)CCC2(CC1)CC(NC(c1cc(SC(F)(F)F)c[nH]1)=O)C2 60348,C(C(COC)CC(=O)N1CCC(CC(=O)NC(C)CS(C)=O)C1)OC 60349,c1(C(N(CC(C)(C)NC(CNC(CNC(C)=O)=O)=O)C)=O)cc(C#N)ccc1O 60350,c1(NC(C2CC(F)CN(Cc3cc(Br)ccc3I)C2)=O)cnc2ccc(F)cn12 60351,CCC(C(=O)N1CCC(CNC(c2csc(CC(C)C)n2)=O)C12CC2)C(F)(F)F 60352,c1(C(C)(C)C)ccc(C(=O)NCCOC2CN(C(=O)CCC3CC3(C)C)C2)[nH]1 60353,c1(C(N(c2ccc(C)c(F)c2)C)=O)cc2c(nc1N)CCC2 60354,C1(CC(=O)NC(C)CCNC(=O)CCn2ccnn2)C2CC3CC(C2)CC1C3 60355,C1(CNC(c2scc(C)c2C)=O)CN(C)CCN1C(=O)CNC(N1CCCC1)=O 60356,N1(C(C2(CC#C)CCCC2)=O)CC2CC1CN2C(=O)C(C1CCS(=O)(=O)CC1)O 60357,C(C)(C(=O)NCCN(C(=O)CCC1CC1(Cl)Cl)C)NC(=O)NC 60358,C1(OC)C2CC3CC1CC(C(N1CCC(NC(=O)CC4(OC)CC4)C(F)C1)=O)(C3)C2 60359,c1(OCC)c(CC(N2CC(OC)C(NC(=O)C(C)CC(N)=O)C2)=O)cccc1Cl 60360,C#CC1(C(N2CCN(C(C)CNC(=O)CC(C)F)CC2)=O)CCCCC1 60361,C1(N(C(=O)C(O)CC2CC2)C)CCN(C(=O)C(C)(C)c2cscc2Cl)CC1 60362,c1(CCC)cnnc(C(=O)N(CCN(C(c2cc(OC)ns2)=O)CC)CC)c1 60363,c1(C(=O)NC(CCC)CNC(=O)C(N2CCCC2)C2CC2)cn(CC)nc1C 60364,C1(OC)NC(C(=O)NCCn2cc(CN3CCNC3=O)nn2)CCC1Br 60365,N1(Cc2c(OC)ccs2)Cc2[nH][nH]c(=NC(=O)c3ccc(F)c(C#N)c3)c2C1 60366,N1(C(C(C=C)(C)CCOC)=O)CCC2(CC1)OCCC2NC(C1(CCF)CC1)=O 60367,N1(C(C=CCC)=O)CC2CC1CN(C(=O)Cc1cc(C)[nH]n1)C2 60368,N1(C(C(C)COc2ccccc2)=O)CCC2CCC(C1)N2C(=O)CCC(F)F 60369,N1(C(CC2CN(C(c3cc(CC)[nH]n3)=O)C(C)C2)=O)CCC(C)(C2CC2)C1 60370,CCC(C)CCC(=O)NC(CNC(=O)CC12CNC(=O)C(C1)C2)CC 60371,N1(C(C(CCCC)NC(N)=O)=O)CCN(C(=O)C=Cc2ccsc2)CCC1C 60372,Cc1cc(Cl)cc(C(=O)N(C)CCNC(c2ncc(Cl)cc2Cl)=O)c1N 60373,C(=O)(C(C)C(C)S(C)(=O)=O)NCC1(CNC(CCOCCC)=O)CCCC1 60374,Cc1nccnc1C(=O)NC1COCC1NC(C1CC(C)(C)CO1)=O 60375,C(C)(C(O)C(=O)N(CCCNC(=O)C(N)=O)CC1CCCC1)SC 60376,c1(C(c2n(C(CC)C)nnn2)Nc2cccc(C(C)F)c2)cc(Cl)c(Br)cc1F 60377,c1(OC)ncc(Br)cc1CN1CCCN(C(c2ccn(C(F)F)n2)=O)CC1 60378,N1(C(c2ncc(C)nc2)=O)CCC2(CC1)CC2(CO)CNC(c1cocn1)=O 60379,C1(C(=O)NCC(CNC(c2c(CC)scc2)=O)(C)C)CCC(N(C)C)CC1 60380,C(=O)(CCS(=O)(=O)C(F)(F)F)NC(C)C(C)NC(c1cnc2[nH]ncc2c1)=O 60381,c1(OCCC)cccc(C(=O)NCCc2cnsn2)c1 60382,C1(C(=O)NC(C(C)(O)CN(C)C)C)CCCN1C(C1(c2ccccc2)CC1)=O 60383,c1(C(N2CC=CC2C(=O)O)=O)ccccc1Br.c12csc(c1)CNC2=O 60384,C1CCCNC(=O)C2CC2C(=O)N1C.C(=O)(C=CC(=O)N(C)C)NC1CC1 60385,C(=O)(CC(C)(C)CC(F)F)N(C1CC2N(C(C(C=C)(C)O)=O)C(CC2)C1)C 60386,N1(C(c2cn(CCOC)c3c2cccc3)=O)CC(C)(C)OC2(CCOC2)C1 60387,C1(CCCNC(c2c(C)occ2)=O)CN(C(=O)CN2CCOC2=O)CCO1 60388,c1(C(N(c2cccnn2)CCC)C2CC2)cc(CO)ccc1Cl 60389,Cc1ncc(C(=O)NCCCCNC(C2C3CCC2CC3)=O)cc1C#N 60390,C1(CN2CC(NC)C(O)C2)CC2(CCCO2)C1 60391,N1(c2nccc(OCCC)n2)CC2(CCC(NC(c3ccc(O)cc3)=O)CC2)C1 60392,N1(C(CS(=O)(=O)NC)=O)CC2CCCC(NC(=O)C(O)C3CCCC3)C2C1 60393,N1(C(c2c(C)ccs2)=O)CC2CCN(C(=O)C(c3ccc(Cl)cc3)O)CCC2C1 60394,CS(=O)(=O)c1cccc(-c2nc(-c3n[nH]cc3Cl)n(CC3CC3)n2)c1 60395,C1(CNC(C(C)(C)OC)=O)C2CC2CN1C(c1cncc(Cl)c1)=O 60396,c1(OC)ccc(O)c(NC(C2(C)C=CCN2C(=O)CCCC(=O)N(C)C)=O)c1 60397,C1(CC)C(C(=O)NCCSCCC(F)(F)F)CCN1C(=O)CSC 60398,c1(OC)cc(F)c(Br)cc1C(=O)NCC(O)CNC(=O)C=Cc1cnc[nH]1 60399,Cc1c(C(N2CC(O)(CC(N3CC(N(CC(C)C)C)C3)=O)C2)=O)ccn1C 60400,N1(C(Cc2c(C)non2)=O)CC(C(N2CCN(C)CC2)=O)C(C2CC2)C1 60401,CC1CCN(CCC(=O)N(CC(C)(C)C)C(C)(C)C2(C3CCCN3C(N)=O)CC2)CC1 60402,C1(C)(CNC(c2cn(CCC(C)C)nn2)=O)CCCN1C(=O)C(C)C(C)C 60403,C=CCN=C(NCC(=C)Cl)NCc1csc(C(C)OCC)n1 60404,CC1CCN(C(c2c(C#N)ncn2C)=O)CC1CC(=O)N(C)CCO 60405,C(=O)(C1=C(C2CC2)N(C2CC2)C(=S)NC1c1cn2ccsc2n1)OC 60406,c1(C(N(CCNC(C(C(CC)O)C)=O)CC)=O)cc2ccc(Cl)cc2[nH]1 60407,c1(CC)ccc(C(=O)NC(C2CN(C(C3CC(C)CO3)=O)C2)C)o1 60408,N1(C(c2c(CC)cno2)=O)CC2CCC(NC(=O)Cn3nccc3C)CC2C1 60409,C=CC1(CC(N2CC(CSC)C2)=O)CN(C(C2(C)CCOC2)=O)C1 60410,C(N=c1nc2sccc2c(N2CC3CCC3(C)C2)[nH]1)CCc1ccn(C)c(=O)c1 60411,Nc1c(C(N2CCCC(CNC(c3cc(Cl)nnc3Cl)=O)C2)=O)nc(O)nc1O 60412,C1(NC(C=CCN(C)CC)=O)CCC(C(=O)NC2(CO)CC(F)C2)CC1 60413,Cc1c(C=CC(N2CCC(C)C(NC(=O)C(C)(C)N3CCCC3)C2)=O)cnn1C 60414,c1(C(=O)NCCC(C(C)C)NC(C(C=CC)O)=O)ccc(Cl)c(F)c1 60415,c1(CC)[nH]nc(C(=O)NC2CCCCCC2NC(=O)CC(C)C)c1[N+](=O)[O-] 60416,C(CCN(C)OC)NC(C1(C)CN(C(C(CC2CC2)OC)=O)C1)=O 60417,CN1CCN(C(c2cnc[nH]c2=N)=O)CC1C(=O)NC1(C)CCCC1O 60418,c1(C(=O)NC(C)C(=O)N(C)C)ccc(SCCOC2CCOC2)cc1 60419,c1(CNC(CCCC#CC)=O)ccc2c(c1)CN(C(c1cccc(Cl)c1C)=O)C2 60420,C1(C)(C(N(CC)Cc2ccoc2)=O)CC(O)CN1C(=O)CC1CCCC2CC12 60421,CCC(Cc1ccccc1)CC(=O)NC(CNC(=O)CC1(O)CCOCC1)CC 60422,C1(C(=O)NCC(c2ccccc2)NC(C(C)Nc2csc(F)c2)=O)SCCCS1 60423,c1(C2CC(c3n(C)nnn3)(NCC3CC(F)(F)CO3)C2)cc(Br)ccc1Cl 60424,c1(C(=O)NCCOCCN(C(C2(CCO)CC2)=O)C)cc(Cl)ccc1C.CC(=O)N 60425,c1(C(=O)NC2CN(C(C3N(CC)CC3)=O)C(CO)C2)coc(=O)c2ccccc12 60426,N1(C(c2c(C)cccn2)=O)CCC2(CCN(C(C3OCCN(C)C3=O)=O)C2)C1 60427,C(=O)(C1CCCc2ncccc21)NCC(CNC(c1cn(CC(N)=O)nn1)=O)F 60428,c1(C(=O)NCC2CCN(C(C(C)OCC#C)=O)C2)ccc(C(=O)CC)cc1 60429,Cc1c(C(N2CC=CC2CNC(c2c[nH]nc2C(F)(F)F)=O)=O)cccc1C#N 60430,C1(NC(=O)C2=CCCOC2)CC2(CCN(C(C3(C4CCCCO4)CC3)=O)CC2)C1 60431,C=CCCCC(C)NC(C1(NC(=O)C=CC(=O)N(C)C)CC1)=O 60432,C(C(C)(C)CNC(C1(O)CCCC1)=O)N(C(=O)CC(C)NC(C1CCCC1)=O)CC 60433,N1(C(c2cc(C)sn2)=O)CC(C(=O)NCC2(C)CC=CCC2)C2(CC2)C1 60434,C12(NC(=O)Cc3ccc(Cl)s3)CCCC1CN(C(c1cccc3c[nH]nc13)=O)C2 60435,c1(COC(N(CCCC(=O)NCC(CCC)C)C)=O)ccc(F)cc1 60436,N1(C(c2ccc(CC)[nH]2)=O)CC(NC(=O)Cn2nc(C)cc2C)CC(O)C1 60437,c1(C(N2C(C)CCC(NC(c3cc(F)c[nH]3)=O)C2)=O)ccc2c(c1)CCC2(C)C 60438,N1(C(C=NOC)=O)CCC2(CC1)OCCC2NC(C1CC1c1ccccc1)=O 60439,c1(C(=O)NCCCN(C)C(C2CC3CCC2O3)=O)cccc2c1CCO2 60440,c1(C(=O)NCCCC(C)NC(CC2(C=C)CCCCC2)=O)coc(S(N)(=O)=O)c1 60441,C1(CC)CCCCCCN1C(C1CCN1CC)=O.C12OCCC1NC2=O 60442,c1(C(N(CC(CNC(C(C)C#N)=O)O)C)=O)nn(C)c2ccccc2c1=O 60443,c1(CNC(C2CC(F)CN(C(c3ccc(I)c(Cl)c3)=O)C2)=O)cccc(F)c1Cl 60444,C(C(=O)N1CCCC(CC(=O)N(CCCO)CCO)C1)(C(C)C)OC 60445,CC(C)CCC(=O)NCC(=O)NC1CCC(NC(c2nc(C3CC3)cs2)=O)C1 60446,CC1(CNC(=O)CCC(N)=O)CCN(C(=O)C(c2ccccc2)O)C1 60447,c1(C(N2CCCC(NC(C(C)OCCC=C)=O)C2CC)=O)cnc2n1CCCC2 60448,n1(CC)nc(C(=O)NC2CCN(C(c3cnc(N(C)C)s3)=O)C2C)c(C)n1 60449,Cc1nc(C(N2CCCC(C)(C)C2CNC(C2CCCCS2)=O)=O)c(=O)[nH]c1C 60450,C(=O)(CS(C)(=O)=O)NCC1CC(CNC(C2(C)CC2)=O)C1 60451,N1(C(C(C)(C2CCC2)NC(=O)Cc2ccsc2)=O)CC2CC(O)CC2C1 60452,CN1N=C(CC(=O)NC2(C)CCN(Cc3ccncc3Cl)C2)CC1=O 60453,c1(CC)ccc(C(=O)NC2(CNC(c3ccoc3Br)=O)CCOC2)s1 60454,C1(C(=O)NC2(C)CN(C(C(COC)(F)F)=O)C2)CC2(CCC2OC)C1 60455,C1(NC(c2[nH]cc(CC)n2)=O)CCCN(C(c2cc[nH]c2C2CC2)=O)C1C 60456,CCCC(C)C(C)NCC1CC1C(=O)OC(C)(C)C 60457,C1(C(N(CC(=O)NCC(CCC)C(=O)NC)C)=O)C2CCCCCCC12.C(C)=O 60458,Nc1cnc(C(=O)NC2CCC2NC(c2cccn2C2CCCC2)=O)cn1 60459,c1(C(N2CC3CC2C3C(N2CCC2(CO)CO)=O)=O)ccc2[nH]nc(Cl)c2c1 60460,c1(C(N2CC(OCCNC(c3cc(CCC)n(C)n3)=O)C2)=O)cnc(N)c(Cl)c1 60461,C1(CNC(c2c(C)snn2)=O)(OCCNC(C2CCC3(CC3)C2)=O)CCOCC1 60462,c1(C(C(=O)NCCC(=C)CNC(c2ccnc(OC)c2)=O)O)ccc(Cl)c(Cl)c1 60463,N1(C(c2cnc(C(C)OCC)s2)=O)CCC(NC(c2ccc(C)o2)=O)CC1C 60464,N1(C(C2C(=C)C2)=O)CC(NC(=O)Cc2cccc(C(N)=O)c2)CC1(C)C 60465,C(=O)(CC(C(F)(F)F)NC(=O)CCOC1COC1)N(C(c1cnnn1C)C)C 60466,C=CCC(CNC(c1ccncc1Cl)=O)C(=O)N1CCC(C(F)F)CC1 60467,c1(CC)ncc(C(=O)NC(C2CC(NC(=O)C(N3CCNC3=O)C)C2)C)c(C)n1 60468,Cc1cn2ccc(C(=O)NC(CNC(=O)C(C)(C)N(C)C)C(C)C)cc2n1 60469,c1(C(=O)NC2C(CC(=O)NC(CC#C)CC)C(O)C2)nccnc1C 60470,c1(N(CCOCCNC(C(C)NS(C)(=O)=O)=O)C)cnn2ccncc12 60471,c1ccc2c(N3CCC(OCC4CCCC4)CC3)nsc2c1 60472,C(c1ccsc1)=CC(=O)NCC=CCNC(C1CC(=C2CC2)C1)=O 60473,CC=C=CCCN=c1nc(N2CCN(C)CC(C)C2)c2ncccc2[nH]1 60474,c1(C(=O)NC2C(CNC(C3CC(=C)C3)=O)C2)cc2c(N(C)C)cccc2s1 60475,c1(C(N2CCC(c3nc(C)c(C)s3)CC2)=O)nc2ccsc2s1 60476,N1(C(c2c(CC)[nH]cc2)=O)CCCC(O)(CNC(C2(CO)CCOCC2)=O)CC1 60477,c1(C(=O)NCC2CN(C(c3ncc(C(F)(F)F)s3)=O)C2)ccc2ccccc2c1O 60478,c1(C(N2CC(NC(C=CC)=O)C(C(F)F)C2)=O)nc(OC(C)C)ccc1Cl 60479,c1(C(=O)NC(C2CCCN2C(=O)C#CC2CCOC2)C)ccc2c(n1)CCCC2 60480,c1(C(=O)NCC2CC(NC(C(C)(C)c3cc[nH]n3)=O)C2)cc(O)cc(Cl)c1Cl 60481,N#CC1(C(=O)NCc2ccoc2)CCC1.C12CC(C1)C(=O)N(C1CC1)CC2 60482,c1(C(c2c(C)cccc2)Sc2ccccn2)ccc(S(N)(=O)=O)cc1Cl 60483,CS(=O)(=O)CCCNC(=O)CC1CC(C(=O)NCc2cccc(N3CCCC3)c2)C1 60484,N1(C(C=Cc2nc(C)sc2)=O)CC(F)(F)CC1C(=O)NC1(C)CCCC1(C)C 60485,C1(CC(=O)NCC(C)(C2CC2)NC(C(C)C2CCCO2)=O)CCC=CCC1 60486,c1(N(C)CC2CCC2)nc(=NC2COCC2C2CC2)[nH]c2c1CSC2 60487,c1(C(=O)NC2C(CNC(c3cccc(C)c3Cl)=O)CCC2)cn2ncccc2n1 60488,N1(C(C2(CCCC)CC2)=O)CCC2(CC1)C(NC(=O)CCNC(=O)NC)CS2(=O)=O 60489,C1(CNC(c2ccc(CF)cc2)=O)CC2CCC(C1)N2c1nncs1 60490,c1(Oc2c(C(N3CCC(O)(C(=O)OCC)C3)=O)cnn2C)cn2nc(C)sc2n1 60491,N1(C(Cc2cc(C)on2)=O)CCC(NC(=O)Cc2c(C)n[nH]c2C)C(CO)CC1 60492,S(=O)(=O)(c1ccc(Br)cc1C(=O)O)NCC(c1cc(C)cc(C)c1)(C)C 60493,CC(C)(C)C(=O)C(=O)NC1CCC(C(C(=O)NCCCCCCF)N(C)C)CC1 60494,C1(NC(C(=O)Nc2cc(C)c(I)cc2)=O)(CO)CC(O)C12CCC2 60495,C1(CCNC(C2(C)CC(F)C2)=O)CCCN(CC(=O)N)C1.c1(CN)ccccc1 60496,c1(C(=O)NC2(CC(=O)Nc3ccc(C)cc3O)CCC2)ccc2ccn(C)c2c1 60497,C1(C(=O)NCC(C(F)(F)F)OC)CNC2(CC2)CO1 60498,c1(CC)ncc(C(=O)NC(C)CCNC(c2sc(=N)[nH]c2CC)=O)cn1 60499,N1(C(C(C)O)=O)CCc2[nH]nc(CNC(=O)CCC3CCOC3)c2C1 60500,S(=O)(=O)(c1csc2ccccc12)NC1CN(C(c2nc(Cl)ccc2F)=O)CC1O 60501,C(=O)(CCC(C)C)NCC(CCOC)NC(C1(C(F)F)CC(O)C1)=O 60502,CC(C)C(CCC(=O)N1CC2CC3CC2C1C3)NC(C1OCCC1(C)C)=O 60503,C(CS(=O)(=O)CC(=O)NCC1CCCCN(C(=O)CCCC(C)(C)C)C1)OC 60504,CC1(Cc2cc(F)ccc2F)CCCN1N1CCCC2(CC1)NC(=O)NC2=O 60505,N1(C(c2ccc(OC(C)C)nn2)=O)CCC(NC(c2coc(Br)n2)=O)C(O)C1 60506,C12(NC(C(=O)NC3CC3)=O)CCC(CC1)N(C(c1ccncc1)=O)C2 60507,C1CC(=O)N1C.C1(NNC(=O)OC(C)(C)C)CC(CSC)C1 60508,CC(C(=O)OCC1CN(CCCOC(=O)OC(C)(C)C)C1)c1cccs1 60509,N1(C(C(C=C)OC)=O)CC(C2CCCN(C(C3(C4CC4)CC3)=O)C2)C1 60510,C1(CC(c2nnnn2CCCF)NC(C)C(=O)NO)CCC(C)(C)CC1 60511,c1(CC)cc(C(N2CCC(NC(=O)CCc3nc(O)n[nH]3)CC2C)=O)cc(C)c1 60512,C1(CN(C(=O)CN2CCCC2CO)C)CCCN(C(c2cccc(O)c2)=O)C1 60513,N1(C(CONC(C(C)C2CC2)=O)=O)CC2(C1)CC(C)(C)C2 60514,c1(C(N2C(CNC(=O)CCc3ccon3)C=CC2)=O)cccc(F)c1Cl 60515,n1(C2CCN(C(N(C3CCC(=O)NC3=O)CC)=O)CC2)ncc2ccccc12 60516,CC1(C(=O)NCC2C=CCN2C(=O)CCc2ccco2)CC(F)C1 60517,N1(C(C2C(C)(CC)C2)=O)CCOC(CNC(=O)CCCCN2CCOCC2)C1 60518,C(=O)(NN1CCN(C(=O)Cc2ccccc2)CC1)c1scc(-c2c(C)n[nH]c2)n1 60519,N1(CC)CCC(NC(=O)CN(C(=O)CCc2ccc(C)[nH]2)CC)C(C)C1 60520,c1(OC)csc(C(=O)NC(C)CC(C)NC(=O)CC2(OC)CCC2)c1 60521,c1(C(N2CCC(C)C2CNC(=O)CC2(C)CC2(Cl)Cl)=O)cc[nH]c2nccc1-2 60522,C1(C(=O)NC2CC(O)(CN(C3CCC3)Cc3c(C)nc[nH]3)C2)CCCC(=O)N1C 60523,c1(C(N(CCN(C(c2cccc(OC)c2)=O)C(C)C)C)=O)ccc2c[nH]nc2n1 60524,N1(C(c2nc(N(C)C)oc2)=O)CCOC2(CCN(C(C3CCCC(F)C3)=O)C2)C1 60525,Cc1c(CN)cccc1F.C(C)(CCC(C)C)N(CC=O)C(c1cccs1)=O 60526,c1(C(N(C)CC2N(C(CC(C(C)C)O)=O)CCC2)=O)ccn2ccnc2c1 60527,C1(C(=O)NCCC2(CNC(C(CSC)O)=O)CC2)CC(=O)N(c2nccs2)C1 60528,c1(NC(C(c2cn(C)nn2)NC(CSCC=C)=O)=O)ccccc1F 60529,c1(C(=O)NC(CNC(CCC(C)C)=O)C2CCC2)c(C)oc2ncnc(O)c12 60530,C1(CC(=O)NC)CN(C(C2CCN(CCO)C(=O)C2)=O)CCN1C(=O)CC1CC1 60531,c1(C(=O)NC(CCC)CNC(=O)C(C)=C(C)C)cc(Cl)nn1C 60532,C(=O)(C1CC(=O)Nc2ncccc21)NC(C)(C)CCCNC(C1CCCOC1)=O 60533,c1(C(=O)NCC(C)(C)NC(=O)CSc2ccccn2)cccnc1O 60534,c1(C(=O)NCCN(CCCCCC)C(c2ccsn2)=O)ncc(N)cc1Cl 60535,c1(CCN(C2CCN(C(=O)CCC3CC(F)(F)C3)C2)C)cc(F)ccc1F 60536,C(=O)(C1=NOC2(CCN(C(=O)OC)C2)C1)N(c1cc2ccccn2n1)C1CCC1 60537,C(=O)(C(C(C)(C)C)N1CCNC1=O)NCC(C)CNC(=O)Cc1ccco1 60538,C(=O)(C(CC(C)C)OC)NCC(CC)N(C)C(C1COCCN1C)=O 60539,C1(c2c(C(=O)OC)nccc2)C2CCCC1CN(C(c1cccc(C)c1C)=O)C2 60540,Cc1cc(=O)oc(C)c1C(N1CCC(CN(C)C(C23CCCN(CC2)C3)=O)C1)=O 60541,c1(C(F)(F)F)cccc(C#CCNCc2cc(Cl)c(Br)cc2C(F)(F)F)c1 60542,C1(NC(C2(OCC)CCC2)=O)CCN(CCCNC(=O)CC2C=CCC2)C1 60543,C1(C(=O)NCC(CN(C)C(c2ncccc2O)=O)(C)C)Cc2cccnc2C1 60544,CCC(CNC(c1conc1CNC(C1CNC(=O)N1)=O)=O)CC(C)C 60545,C1(C(=O)NCCN(C(CC2(C=C)CC2)=O)CCc2ccccc2)CN(C)CCO1 60546,CCCC(C(=O)NC1CC1CNC(=O)Cn1cc(Cl)cn1)c1ccc(Cl)cc1 60547,CC(=O)CCCC(=O)N1CCN(C(C23CC(C(F)F)(C2)C3)=O)CC1C 60548,c12ccc(F)c(c1)-c1c[nH]nc1C(=O)N2.CC(C)CCSCCC(C)C 60549,N1(CC(=O)NCC(C)N(C(=O)CCc2ccccc2Cl)C)CCCC(C(N)=O)C1 60550,c1(C(C)NC(C(c2cnn(C)c2)NC(COCCOC)=O)=O)nocc1C(=O)O 60551,c1(CC(=O)NC2C(NC(C3C=CCCC3)=O)CCC2)cccnc1C(F)(F)F 60552,c1(C(c2nnnn2C)NCCc2nc(C(=O)OCC)sc2)c[nH]c2cccc(F)c12 60553,c1(NC(CN2C(CCC)CC2)=O)cc(Br)ccc1C 60554,C1(CCCC)CN(C(c2n[nH]c(C)c2Br)=O)CCN1C(=O)CC(C)F 60555,C=C(F)C1(CC(=O)NCC2(NC(C3CC4(CCC4)CO3)=O)CCC2)CCOCC1 60556,S(=O)(=O)(c1ccc(F)cc1F)N(C1CC2CC1CN2)C(c1c(CC)onc1)=O 60557,c1(C(C)OCC)noc(CN(C)C(C2(C)CCCS2)=O)n1 60558,c1(C(=O)NC2CC(NC(Cc3nc(C)sc3)=O)C2)ncnc2sccc12 60559,C1(CCNC(C2(C(N)=O)CC2)=O)CCC(NC(=O)CO)C1 60560,CCC(C)C(C)(O)CNC(C1CCCC1NC(c1cncc(O)c1)=O)=O 60561,CC(C)C(CC(=O)N1CCC(C)(CN(C)C)C1)NC(=O)CC1CC(C)(C)CO1 60562,N1(C(C(CC(C)(C)NC(c2cn(CCC)nn2)=O)F)=O)CCC2(CC=CCO2)C1 60563,c1(C(=O)NCC2(C)CCCN(C(C3=CCCCC3C)=O)C2)cnc2ncnn2n1 60564,CN1CC(=O)N(CCCC(=O)NCCCCCNC(C2CCCS2)=O)C1=O 60565,O=S(=O)(c1cnc(NCC(C(F)(F)F)SC)c(Cl)c1)NCC1CC2CCCC(C1)C2 60566,c1(COC(N(CC(CC)C(=O)OC(C)(C)C)C)=O)ccc2c(c1)CCN(C)C2 60567,c1(C(N2CC(CNC(Cc3ccc(OC)cc3)=O)C2)=O)ccc(P(C)(C)=O)s1 60568,C1(CC)CN(Cc2ccccc2N(C)C)CCN1C(=O)Cc1ccsc1 60569,C1(C(=O)NCC(C2CC2)SC)CC2CN(C(=O)Cn3nnc(C)n3)CC2C1 60570,c1(OCC#C)ccc(C(=O)NCC(CO)NC(=O)C(c2ccccc2)F)cc1 60571,CCCC(C)(C)CC(=O)N(CCC(=O)N(CC(O)C1CCC1)C)C1CC1 60572,C1(CC)(CNC(C2(NC(c3cc(OC)no3)=O)CC(O)C2)=O)CCOC1 60573,c1(CC)cc(C)nc(N2CCCC2CCCNC(C2(C3CC3)CCCO2)=O)n1 60574,Cc1ccc(C(=O)NC2(CS(N)(=O)=O)CC2)nc1C 60575,C(=O)(C(C)(CSC)NC(=O)C=Cc1ccoc1)NC(C#C)C 60576,C1(NC(=O)NC)CC(C)(C)CN1C(=O)CCn1cc(-c2cnc(C)n2C)nn1 60577,C(C(C)(C)CNC(c1ncoc1C1CCC1)=O)N(C)C(c1coc(Br)n1)=O 60578,CC1C2CCCCC2CN1C(=O)C(Cn1cncn1)NC(C1CCC(=O)O1)=O 60579,c1(CSCCC(=O)NCCC2CCN(C(CC(=O)OCC)=O)C2)ccc(F)cc1 60580,N1(C(c2ccc(C#C)cc2OC)=O)CCC2C(CCCN2C(=O)CC(C)(C)C)C1 60581,C=CC1(C(=O)N(C)Cc2ncn(C)n2)CCN(C(=O)CCc2cccs2)C1 60582,CC1(C#CC(=O)NC2CC3CCC2N3C(c2cc(Cl)c(Cl)s2)=O)CC1 60583,C1(C(=O)NC2CCN(C(C)=O)CC2)CCC2(CN(C(=O)C(O)C(C)C)C2)O1 60584,C1(NC(Cc2c(C)non2)=O)CN(C(C23CC2COC3(C)C)=O)C2(CCC2)C1 60585,c1(C(NOC(C(C(=O)N2C(C(=O)OCC)CCC2)(C)C)=O)=O)nccc(Cl)c1C 60586,CCC(C)CC(C)C(=O)NC(C)(C)C=CC(=O)Nc1cc(CO)cc(C)c1 60587,CC(CC(=O)N1CCC1C1CCOCC1)N(C(=O)COc1cnn(C)c1)C1CC1 60588,C=CCC(CC(=O)N1CCC(COC)CC1)NC(=O)C(CC=C)OC 60589,C1(CCC(=O)N(c2ccccc2F)C)CCCN(C(C2CC=CC(O)C2)=O)C1 60590,CC(CC(=O)NC(C1(O)CCCCC1)C(N1CC=CC(O)C1)=O)C(F)(F)F 60591,C(CCCCC(=O)NCc1nccn1C)N(C)C(C1(F)CCOCC1)=O 60592,c1(NC(C2(O)CCN(S(=O)(=O)c3cn[nH]c3)C2)=O)nc(C(F)(F)F)ccc1Cl 60593,C1(C(=O)NCCCC(C)NC(C2CCC3(CC3)C2)=O)C2CC3C(C2)C13 60594,CC1(C)CCCN(C(=O)C=CBr)C1CNCc1nnc2ccccn12 60595,C1(NC(C(C=C=C)C)=O)CCCCN(C(c2cnc(OC)s2)=O)C1 60596,CC1(NC(=O)CC2CCCC23CC3)CCN(C(=O)Cn2nnc(=N)[nH]2)CC1 60597,CC#CCCCC(C)N(c1ccc(N(C)C)cc1)CCC#N 60598,c1(OC)ccc(F)c(C(=O)NCC(C)(C)CN(C)C(C2CCCC2(C)C)=O)c1N 60599,C(C(C)C(C)C(=O)N1CCCC1CN(C(=O)CCNC(c1ccco1)=O)C)OC 60600,CC1CC(NC(=O)C(C)OC(F)F)CCO1 60601,C12(CNC(c3n(C)c(=O)ccc3)=O)CCC(CN(C(C3CCCC3(F)F)=O)C1)C2 60602,C1(CNC(c2cncc(OC)c2)=O)CCN(C(=O)CC(C)N(C)C)C12CCC2 60603,C1(NC(CC2(OC)CCCCC2)=O)CC(C)CN(C(=O)CCc2csc(=N)[nH]2)C1 60604,C1(CCC)(NC(=O)CCc2cnoc2)CCN(C(c2ccc([N+](=O)[O-])s2)=O)CC1 60605,C1(C(=O)NCCC2CCN(C(C(c3n(C)ccn3)(F)F)=O)C2)CCC(F)(F)CC1 60606,N1(C(c2cn(CCC=C)nn2)=O)CCN(CC(C)NC(c2n[nH]cc2Cl)=O)CC1 60607,CCC(C)(CN(C(=O)CN1CC2CC2C1)CCOC)C(=O)N1OC2CCC1CC2 60608,C#CC1CCN(C(C2COCCN2C(=O)C(C)=C2CCCC2)=O)CC1 60609,CC1(C(=O)NC2CN(C(c3cccc[n+]3[O-])=O)CC2CO)CCC(O)CC1 60610,c1(C(=O)Nc2nc(C)c(-c3nn[nH]n3)s2)n[nH]c2cc(Br)ccc12 60611,c1(CNC(C2CCN(c3ncc(C#N)nc3)CC2)=O)nnn2c1COCC2 60612,C12(NC(CC(COC)NC(=O)Cn3nc(C)nc3C)=O)CCC(C1)OC2C 60613,C1(NC(CNC(CC)=O)=O)(CC)CCN(C(C2CC2Cl)=O)CC1 60614,C=Cc1cccc(CN2CCCC(NC(=O)CCc3ccccc3)C2)c1 60615,C1(NC(C(C)(CO)OC)=O)CN(C(c2cc(C)cc(Br)c2)=O)CC1N=[N+]=[N-] 60616,c1(C(C(=O)NC(C(=O)OC)C)N(C(C)CCO)C)ccc(OC)c(Br)c1 60617,CCCCC(O)C(C)C(=O)NCC(C)=CC(=O)NCC(O)CCC1CC1 60618,c1(C(=O)NCCN(C(C(c2cnn(C)c2)OC)=O)C)nc(C)n2ccccc12 60619,CC(CC(C)(C)C)C(=O)NCC(C)(CO)NC(=O)CCCn1cncn1 60620,c1(C(=O)NCC2N(C(C(C)=C(C)C)=O)CC(F)C2)cccc(=S)n1O 60621,c1(OC)ccccc1NCC(N1CCCC(N(C(=O)CCF)CCO)C1)=O 60622,Nc1cccnc1S(=O)(=O)NC1CC(=O)N(CC(F)(F)F)C1 60623,c1(C(N(C2C3CN(C(C(C(C)(C)C)OC)=O)CC32)C)=O)cccc2c1OCCC2 60624,c1(C(N2CC(C)C(NC(=O)C(C)(C)N3CCCC3)C2)=O)cc(N)c(Br)c(F)c1 60625,N1(C(C(C)SC2CCCN(C)C2)=O)CC2CCC(C(=O)NC3CCCCC3)(C2)C1 60626,C=C(C)C1OCCCC1C(N1CCC2(C1)CN(C(c1cc(O)ncn1)=O)C2)=O 60627,C1(NC(C=C(C)c2ccsc2)=O)CC2CCC(C1)N2C(=O)C(C)S(C)(=O)=O 60628,CN1CCNC(=O)C12CCCN(Cc1cnc3ccc(Cl)cn13)C2 60629,C1(C(=O)NCC2(CO)CCCC2)CC2(CCC2)CN1C(c1ccnc(O)c1F)=O 60630,C(c1ccc(C)cc1)=C(C(N1CCC(O)(CCNC(C(CCC)OC)=O)C1)=O)C 60631,C1(NC(=O)CC2CC3C=CC2C3)CC2CC1N(C(C1CCCCC1)=O)C2 60632,c1(C(N2C(C(N3CC(CC)C3)=O)CNC(=O)C2)=O)ccc2[nH]ccc2n1 60633,C1(OC)CCC2(C(=O)N(CC(C)C(=O)N(C)Cc3cnco3)C)CC12 60634,Cc1cc(Br)cnc1C(=O)NCCCC(C)NC(=O)C(C)N1CCC1 60635,C(CN=c1nc2c(ncn2C)c(NC2CCN(C)C(C)C2)[nH]1)OCCOCCC 60636,c1(C(=O)NCC(CC(F)(F)F)NC(=O)C(O)C2CCC2)cc2ccc(F)cc2[nH]1 60637,C1(NC(c2c(CC)nc[nH]2)=O)CC2(CCN(C(=O)C(C)CCCOC)C2)C1 60638,C(CCC(O)C(=O)NC1CCOC(C)(C)C1)NC(C1(OC)CC(C)C1)=O 60639,N1(C(C2CC(=O)N(C)C(=O)N2)=O)CCC2(NC(c3cnc[nH]3)=O)CCCCCC12 60640,N1(C(CCCCN(C)C)=O)CC2CCN(C(c3snc(Cl)c3Cl)=O)CC2C1 60641,Cc1cnc(C)c(C(=O)NCC(C)CNC(=O)CSc2ccc(F)cc2F)c1 60642,c1(C(=O)NC2C(NC(C(CC)(C)C#N)=O)CC2)cc2c(cc1F)OCC(=O)N2 60643,N1(C(CC)=O)CCCC(C(=O)NC(C)(CNC(=O)C2=COCC2)C(C)C)C1 60644,c1(SC)cc(C)c(CNC(=O)CSC2(C(C)(C)C)CCN(C(C3(O)CC3)=O)C2)s1 60645,C(=O)(C(C)C(C)(C)C)NC(C(=O)NCC(C#C)C(C)C)Cn1ccnn1 60646,c1(C(N(C)CCOCC2(O)CCOC2)=O)ncc(C(C)(C)O)cn1 60647,c1(OC)cnc(Cl)nc1N1CCCC(C(C)NC(c2cnn(C)c2C2CC2)=O)C1 60648,C1(NC(c2n(C)cnc2)=O)COC2(CCCN(C(C3(CO)CCOCC3)=O)C2)C1 60649,c1(-c2cc(CCN(C)C)on2)nc(C2CCCCC2)nn1CCS(C)(=O)=O 60650,c1(OC)ccc(CCCNC(=O)Cn2cc(CC3CCCC3)nn2)cc1.C1CC1 60651,Cc1ncnc(C)c1C(=O)N(CCCNC(=O)C1=NOC(C)C1)C 60652,C1(C(N2CCC(N(C(C3(C4CC4)CC=CC3)=O)CC)C2)=O)(OC)CCS(=O)(=O)C1 60653,c1(-c2nc(-c3ccc(C)o3)nn2C2CC2)cc(C(F)(F)F)nc(Cl)c1 60654,N1(C(COCC)=O)CCC(C(=O)NC2(CO)CC(F)(F)C2)C1CC 60655,N1(C(C(CO)N(C)C)=O)CCC(C2CCN(C(=O)Cc3cnns3)CC2)C1 60656,N1(C(C=CC(C)(C)SC)=O)CCCC2C1CCCN2C(c1ccoc1C1CC1)=O 60657,C1(CCN2CCC(C)CC2)CCC2(CCN(C(=O)CSC(F)F)C2)O1 60658,C(C(C(=O)NCC(O)C1(Cl)CC1)NC(C1C(C)C1C)=O)OCC 60659,c1(NC(C2CCCC2CON)=O)cncc(C(F)(F)F)c1.c12csc(n1)NC2=O 60660,C1(CNC(CCCOC)=O)CC2CN(C(=O)C(C)(COC)CC)CC12 60661,c1(OCC)ccc(C=CC(=O)NCCn2cccc2)cc1OC 60662,C(CC)(CC)(CCNC(=O)CCCCC#N)NC(c1ncc(CC)nc1)=O 60663,c1(C(N(CCN(C(C)C)C(C2CCC(C)S2)=O)C)=O)c[nH]c2c(C#N)cccc12 60664,C12(NC(C(Cc3c(C)n[nH]c3C)C)=O)CCCC(CN(C(=O)C#CC3CC3)C1)C2 60665,CCC(C)(F)C(=O)NCCC1CCC(NC(c2ccccc2NC(N)=O)=O)C1 60666,C#CCC(CC(F)F)C(=O)NC1CC=C(C(=O)NC2(CO)CC(F)(F)C2)C1 60667,C1(CC(=O)NC2CC(=O)NC2)C2CCCC2N1C(C1(F)CCCC1)=O 60668,c1(C(N(CCN(C(=O)C(O)C(C)C)CC)CC)=O)sc2cc(C)ccc2c1Cl 60669,Cc1ccc2[nH]c(C)c(CC(N3CCC(NCC(C)N)CC3C)=O)c2c1 60670,N1(C(c2ccc(C(C)C)s2)=O)CCC(C)(CNC(=O)CC2C(C)C2(F)F)C1 60671,c1(C(=O)NC2CN(C(C(CC=C)C(C)C)=O)C2)[nH]c2c(F)cc(F)cc2c1C 60672,CCC(C)C(O)C(C)C(=O)N1CCC(C(N2CCC3(CCSC3)C2)=O)(C(C)C)C1 60673,C1(NC(CCOCCSC)=O)CN(C(c2snc(C)c2N)=O)CC1O 60674,C1(C(=O)NCCNC(C2CC(C)(CC)C2)=O)CCC(=O)N(c2cnn(C)c2)C1 60675,C1(NC(C(C=C)CC)=O)CN(C(=O)CCC(C)OCC)CC1C1CC1 60676,Cc1c(C(=O)NCC2CCCCC2NC(=O)COc2cnn(C)c2)cccc1O 60677,c1(CC(=O)NCCOCCn2cc(-c3ccc(C(F)(F)F)s3)nn2)cncnc1 60678,N1(C(C2CCC(OC)CC2)=O)CCN(C(c2ncn3c2CCC3)=O)C2CCCC12 60679,N1(C(C2CC(OC)C2)=O)CCOCC(CNC(=O)COC2CCC(F)(F)CC2)C1 60680,N1(C(C(C)OCC)=O)CCC2CN(C(=O)C(O)C(C)c3ccccc3)CC2CC1 60681,c1(CN2C(C)CCC2)ccc(-n2cc(C(=O)NCc3ccc(Cl)cc3)nn2)cc1 60682,C(C(O)CN=c1[nH]nco1)NC(C(CCCC)ON=C(C)C)=O 60683,C=CCC(C)(C)CSc1ccc(NC(C2(CO)CCCC2)=O)cc1 60684,N1(c2n(CCC(=O)NC)c(-c3c[nH]nc3C)nn2)CC(COC)C2(CCCC2)C1 60685,C(c1ccc(Cl)cc1F)=CC(=O)NC1CC(F)(CNC(C23CC(C)C2C3)=O)C1 60686,N1(C(CC2(C)CCCC2)=O)CC(CNC(c2cccc(F)c2Cl)=O)CC12CCC2 60687,N1(C(CC2(N(C)C)CCC2)=O)CCCC1C=CC(=O)NCC1(O)CCN(C)C1 60688,c1(C(=O)NC2C(NC(C3CCC(C)(C)C3)=O)CC2)ccc2nc(O)[nH]c2n1 60689,c1(C(N2CCC(O)(C(C)NC(c3ccncn3)=O)C2)=O)nccc2n[nH]cc12 60690,c1(CC(=O)NCC2CCC(NC(c3cnc(OC)s3)=O)C2)cc(C)ccc1OC 60691,N1(C(C(CCC)C)=O)CC2(C1)CN(C(C1CCC(F)(F)C1)=O)CC2C(=O)O 60692,C1(NC(CCNC(=O)NC)=O)CCC(O)CN(C(c2cn(C)c(O)n2)=O)C1 60693,N1(C(CC2CC(=C)C2)=O)CCN(C(c2ccc(N)cc2OCC)=O)CC(C)(C)C1 60694,Cc1nc(O)c2c(n1)CN(c1cc(C3CC3)nc(S(C)(=O)=O)n1)CC2 60695,N1(C(C(N2CCCCC2)C)=O)CCOC(CCCNC(=O)CP(C)(C)=O)C1 60696,C(=O)(C(=O)N=S(C)(C)=O)NC1C(C)CN(C(c2ccc([N+](=O)[O-])s2)=O)CC1 60697,C1(O)(C(N(CCC)C)=O)CCN(C(c2nnc(C)s2)=O)CC1 60698,c1(C(N2C(CCCNC(CSC)=O)CCC2)=O)ccc(F)cc1N 60699,CN1CC=C(CC(=O)NC(C)(CNC(C23CCCC2OCC3)=O)C2CCC2)CC1 60700,c1(C(N(CC2CCN(C(C=CC(=O)OCC)=O)C2)CC)=O)cn2c(n1)SCC2 60701,N1(C(C)C(N2CCCC2c2ccc(Cl)cc2)=O)CCCCC1C#N 60702,C12CCCN(CC1)C2=O.C1(CC(=O)NC2C(=C)C2)(OC(C)=O)CCCC1 60703,C(N=c1nc(C)[nH]s1)C1(C)CCN(C(c2c(CC)ccs2)=O)C1 60704,N1(C(C2CC(C#C)(O)C2)=O)CCC(CNC(c2ccc(Cl)nc2C)=O)C12CC2 60705,c1(C(N(CC(CC)NC(=O)CC2CCC(=O)O2)C)=O)ccc(C)c(C(C)(C)C)c1 60706,c1(CCC(c2nnnn2C2CC2)NCCOCCC(C)C)ccccc1F 60707,N1(C(c2n[nH]c(CC)c2C)=O)CC(C)N(C(c2cccs2)=O)CC1C 60708,C1(CC(=O)NC(=O)OC(C)(C)C)CC(c2ccccc2)=NO1.C1CC(C)C(=O)N1C 60709,C1(CCNC(=O)C=CC2CCOC2)(OC)CN(C(=O)CCOCCOC)C1 60710,c1(CC)c(C(N2CCCC(N(C(=O)CN(C)C(C)=O)C)C2)=O)oc2ccccc12 60711,c1(C(=O)NCC2(O)CCCN(C(C(CC=C)OC)=O)C2)cc2ccccn2c1 60712,c1(CC)[nH]nc(C(N2CCCC2CCC2CCCCN2C(=O)CNC=O)=O)c1C 60713,C(CN=c1[nH]c(=NCC2(F)CCCCC2)c2c(F)cccc2[nH]1)C1C(C)C1 60714,C1(CCC)CN(C(=O)COc2cc(C)on2)CC1NC(C1CCSC1)=O 60715,CC(c1ccsc1)=CC(=O)NCC(CC(C)C)NC(=O)CC12CC(C1)C2 60716,N1(C(C2C(C=C)C2)=O)C(CNC(=O)Cc2ccc(OC)c(F)c2)CC2CCCC12 60717,CON1CCC(C(=O)NC(C(C)NC(c2ccc(N(C)C)cc2)=O)C(C)C)CC1 60718,Cc1ccnc(O)c1C(N1CCN(C2CN(C(c3c[nH]c(=O)cn3)=O)C2)CC1)=O 60719,C1(NC(C2(C)CCN(C)C2)=O)CN(C(c2cn3c(n2)SCC3)=O)C(C)(C)C1 60720,n1(CC(C)C(=O)NC2CCSC23CN(C(=O)C(Cl)=CCl)C3)cnc2ccccc12 60721,C1(c2cn(CCC(=O)Nc3cccc(NCC4CC4)c3)nn2)CC2CCC1CC2 60722,C1(CNC(CCC=C=C)=O)CN(C(c2cnc(C)[nH]c2=N)=O)C2(CCC2)C1 60723,Cc1nn(CC(N2CCC(NC(C3C=CCC3)=O)C(C)C2)=O)c2ncccc12 60724,c1(C(=O)NCCNC(C2CCC(=O)NC2)=O)coc2c(F)c(Cl)ccc12 60725,c1(C(=O)NCC2(C)CCCN2C(C23COCC2C3)=O)ccc(F)c2cccnc12 60726,c1(CNC(c2cn(CCC)nc2)=O)cnn2c1CN(c1nnc(C)c(C)n1)CC2 60727,C1(NC(CSCCOC)=O)CCCC(NC(=O)Cc2n[nH]c(C)n2)C1 60728,n1(C(C(=O)NC(CC)CNC(C2(N(C)C)CC2)=O)C)ncc2c1CCCC2 60729,N1(C(C(C)NC(COC)=O)=O)CCN(C)CC1CNC(c1scnc1C)=O 60730,Cc1ccc(F)cc1C1(C(=O)NCC(C)CNC(C23CCCC(C2)OC3)=O)CC1 60731,C1(C(=O)NCC2ON=C(C)C2)CCN(C(c2cnn(C3CC3)c2)=O)C12CC2 60732,C(=O)(C(C#N)C(C)(C)C)OCCCC=CC(=O)NCC(CC(C)(C)O)=O 60733,CS(=O)CCC(O)C(=O)NCCCNC(c1cc(O)cc(Cl)c1Cl)=O 60734,N1(C(CCC(C)(C)OC)=O)CCC2CCCC12C(=O)NCC1(N(C)C)CCCC1 60735,C1(C(N2CCN(C(CN(C(C3CC(OC)C3)=O)C)=O)CC2)=O)CC(F)C(=O)N1C 60736,Cc1cnc(C)c(C(=O)NC2(C)CCN(C(=O)CCC3CCCN(C)C3)C2)c1 60737,c1(C(=O)NCCC(CNC(C(CCC)(C)C)=O)O)cn2cc(C)sc2n1 60738,CC1=C(C(=O)NC2CC(C(c3ccccc3)=O)(NC(C34CSCC3C4)=O)C2)CCO1 60739,N1(C(c2c(C)cnnc2)=O)CC2OCC(NC(=O)C(N3CCSCC3)C)C2C1 60740,CCC(COC)C(=O)NC(c1ccnn1C)C(=O)N(C)Cc1cccc(C)n1 60741,c1(OC)ccc(S(=O)(=O)N2Cc3ccc(C(=O)N=c4cnc(I)c[nH]4)cc3C2)cc1 60742,N1(C(C2CC23CCOC3)C(=O)NCC)CC(N(C)CC)Cc2cc(OC)ccc21 60743,c1(C(N2CCCC(CNC(C3CCC4CC34)=O)C2)=O)cc(Cl)cc2c1CCC2 60744,N1(C(c2ccn(C)c2)=O)CCC(C)(CC(=O)Nc2cnc(F)nc2)C1 60745,c1(C(=O)NC2(C)CN(C(=O)Cn3[nH]cnc3=N)C2)cc(=NS(C)(=O)=O)cc[nH]1 60746,Cc1nc(-c2ccsc2)ccc1-c1nc(-c2ccco2)nn1C1CCC(C)(C)C1 60747,N1(C(=O)COCC2CCOC2)CCCCC(C(=O)Nc2cncnc2O)C1 60748,N1(C(C2ON=C(C)C2)=O)CCC(C)C1CNC(c1ccnn1C(C)C)=O 60749,c1(C(=O)NCC(C)(C2CCC2)NC(C(CC#C)O)=O)cc([N+](=O)[O-])n[nH]1 60750,C1(NC(C2CCCN(C(C)C)C2)=O)CCN(C(C2(CCF)CC2)=O)C12CCCC2 60751,N1(C(C=CCC)=O)CC(NC(c2cc(F)cc3nccnc23)=O)C2CCCCC12 60752,C12(CNC(CN(C(C)C)C)=O)CCCC1CN(C(C13CCC(CC1)CC3)=O)C2 60753,N1(C(c2cc(C)c(C)[nH]2)=O)CCC(CNC(c2coc(Br)c2)=O)C12CC2 60754,Cc1nnc(COCC(=O)NC(C)C(CO)NC(=O)CC2CCCO2)s1 60755,C1(N(C)C)(CNC(=O)C(CC2CCC2)NC(C2(O)CCOC2)=O)CCCC1 60756,C1(SC)CN(C(c2ccc(F)cn2)=O)CC1n1cc(CCCC(C)=O)nn1 60757,N1(C(CCc2n(C)ncc2)=O)CCC(F)(CNC(=O)CCCCNC(N)=O)C1 60758,c1(OC)c(Cl)ccc(Cl)c1CNc1cnnc(Br)c1 60759,CCC(CC(=O)NC1CCCCCC1NC(c1ccc(C(C)(C)C)[nH]1)=O)C(C)C 60760,C1(S(C)(=O)=O)(C(=O)NC2CCN(C(c3cnc(CCC)s3)=O)C2C)CCOCC1 60761,c1(C(CNC(=O)CCCCN(C)C)NC(CCOC)=O)ccc(F)cc1 60762,C12(C(=O)NC(CC#C)C(N)=O)CCC(CC1)N(C(C1CCC3(CCC3)O1)=O)C2 60763,C1(C)(C(N2C(CNC(CC3ON=C(C)C3)=O)CCC2)=O)CS(=O)(=O)C1 60764,N1(C(c2c(Cl)ccc(CC)c2)=O)CC(CO)C2(C1)CN(C(c1coc(Cl)n1)=O)C2 60765,O=C(C1=CCSC1)NCC(c1ccccc1)CNC(c1cccnc1C1CC1)=O 60766,C1(CC)(NC(c2ncccc2O)=O)CCN(C(c2cccc(OC)c2F)=O)CC1 60767,n1(C(C)C)cnc2c(NCC3CC4C=CC3O4)[nH]c(=NC3CC(C)(CO)C3)nc12 60768,C1(C2(O)CCCOC2)(C(=O)Nc2ccc(SCCN3CCCC3)cc2)CC1 60769,C(=O)(C(CC1CCC1)NC(=O)COC1CCCOC1)NC1CC(CN(C)C)C1 60770,CC1(C)CC(NC(c2cc(CO)ccn2)=O)CN1C(C1CC12CCSCC2)=O 60771,CC1CCSC1C(N1CC(CNC(c2cnn(-c3nccs3)c2)=O)C1)=O 60772,C(C)(CNC(c1ncccc1Cl)=O)(CC(C)C)NC(C(CC)OC)=O 60773,C1(NC(C=CC)=O)COC2C(NC(c3c(Cl)ccc(F)c3F)=O)COC12 60774,N1(C(C2CC(CC)C2)=O)CCC(C(=O)NCC2(Cl)CCC2)C1C 60775,N1(C(C(n2c(C)ccn2)C)=O)CC(F)(F)CC1C(=O)NCC1CSCCO1 60776,C1(CN(C(=O)CCc2ccnc(Cl)c2)CC)CCN(C(=O)C(C)C2CCC2)CC1 60777,c1(C(CNC(C2(COC)CCCC2)=O)NC(=O)C(O)C2CCC2)ccccc1F 60778,N1(C(C(c2cccs2)NC(Cc2c(C)nccc2)=O)=O)CC(=O)N2CCCC2C1 60779,C1(C(N2CCN(C(CC)=O)CC2C)=O)CN2CCCN1CC2 60780,N1(C(c2ccc(F)c(F)c2)=O)CC(C(N2CCC=C(Cl)C2)=O)C(C2CC2)C1 60781,N1(C(c2cn(CC)nc2)=O)CCCC(N(C)C(c2cc(CO)[nH]n2)=O)CC1 60782,n1(CCCC)nnnc1C(c1ccccn1)NCC(C)(C)SC 60783,CC(CCC(C)(C)C)NC(=O)CN(C(c1cc(F)cnc1O)=O)C1CC1 60784,c1(CN(CC(N2CC(N(C)C(=O)NC(C)(C)C)C2)=O)C)ccc(C#N)cc1F 60785,c1(N(CCOCC=C)C)nc(=NC(C)c2ccc(F)c(Cl)c2)[nH]c2c1CSC2 60786,C1(C(=O)NC23C(CN(C(C(C)(C)OC(C)C)=O)C2)C3)CCOC(=O)CC1 60787,O=S1CCC(NCCOc2cccnc2)c2cccc(F)c21 60788,c1(C(N(C)CC2CN(C(=O)CC(C)(O)C3CC3)CCO2)=O)cc(O)nc(O)n1 60789,C1(CCC2N(C(c3c(OC)ocn3)=O)CCC2)CCCCN1C(C)=O 60790,Cc1ccc(C=CC(N2CCC(NC(=O)C(C)Oc3cccc(Cl)c3)C2)=O)cn1 60791,N1(C(C2CC=C(C)CC2)=O)CCCC2(NC(c3ccc(Cl)nc3Cl)=O)CC2C1 60792,Cc1ccc(OCCCC(=O)N(C)CCN(C(=O)C(C)N2CC(C)C2)C)cc1 60793,c1(C(=O)NCCN(C(=O)CCC(C)OCC)CCC)c[nH]c2c(CC)cccc12 60794,c1(C(N2CC(CCNC(C=NOC)=O)C2)=O)ccc(C(N)=O)cc1 60795,CC1(C)CC(CC(=O)NCCCCNC(c2conc2C2(C)COC2)=O)CO1 60796,N1(CC(=O)NCC(CCCC)NC(=O)Cc2occc2C)C(=O)CN(C)C1=O 60797,CCCCCCN(C(=O)Cn1cccn1)CCN(C(C1CCCC1C)=O)CC 60798,Cc1cc(NC(c2ccc(S(C)(=O)=O)s2)c2nnnn2C(C)(C)C)cc(C)c1F 60799,c1(C(=O)NCCC2(NC(C3C(C(=O)OC)C3)=O)CC2)sc(Cl)c(Cl)c1C 60800,C1(C(=O)NC(CCNC(C(c2ccc(C)cc2)=O)=O)C)CC12CCSCC2 60801,c1(C(=O)NC2CC3CC(NC(C(F)=CC)=O)C3C2)c[nH]c2ccc(Cl)cc12 60802,c1(C(N2CCCC(CCNC(CC3OCC(C)(C)C3)=O)C2)=O)cc(Cl)ccc1Cl 60803,c1(C(=O)NCC(CO)NC(=O)CCC2CCOC2)cnn(CC2CCCCC2)c1 60804,C(CCC(=O)NC1(c2ccccc2)CC(NC(C2CC23CC3)=O)C1)OC 60805,C(=O)(C#CC1(C)CC1)N1C(C(C)NC(c2cn(C)nc2O)=O)CCC1 60806,CCCCCC(C)CC(=O)N1CCC(C)C(CNC(c2cc(SC)oc2C)=O)C1 60807,Cc1cc(C(=O)NC(c2nocc2C(N2CCCCC2CC(C)C)=O)C)sc1C 60808,c1(C(C)(C(=O)NC2CC(F)(F)C2)N(C2CC2)Cc2ccccc2)ccc(Br)cn1 60809,c1(CCCC(=O)NC2C(OC)CN(C(c3cnoc3C)=O)C2)ccc(F)c(F)c1 60810,c1(C(=O)NC2CC(C)CN(C(=O)CCC3CC3)C2)ccc2nc3n(c2c1)CCC3 60811,c1(CNC(c2n(CC)nc(C)c2)=O)ccc(CNC(=O)C(C)NC(C)=O)cc1F 60812,CC1=C(C)CC(C(=O)NCC2CCC(C(N3CCCC(CN=[N+]=[N-])C3)=O)C2)CC1 60813,C1(C(N2CCC(C(=O)NCC3(CC)CC3)C2)=O)CCC(=O)N1C 60814,C1(C)(NC(C2N(C(C(C)C)=O)CCC2)=O)CCS(=O)(=O)C1 60815,CCC(F)(F)CC(=O)N1CCCC(C2CCCCN2C(C23CSCC2C3)=O)C1 60816,C1(NC(CCN(CC)CC)=O)CC2CN(C(c3cc4cc(C)sc4[nH]3)=O)CC2C1 60817,N1(C(C2(C)CC(C)C2)=O)CCC(NC(=O)C=CSc2nc[nH]n2)C(O)C1 60818,CC1(C)C(CC(N2CCOC3(CC3)C2)=O)CCN1C(=O)Cn1cnnc1 60819,C1(CC)CN(C(c2cnc(Cl)cc2I)=O)CCN1Cc1ccnc(OC)c1 60820,c1(C(N(C)CC2CCCN(C(C3CCC3(F)F)=O)C2)=O)cc2nc[nH]c2cc1F 60821,CC1(CNC(C2C=CCN(C(c3nc(Cl)cs3)=O)C2)=O)CC2CCC1C2 60822,N1(C(c2c(NC(CCC(N)=O)=O)nc(Cl)cc2)=O)CCc2ncncc2C1 60823,c1(C(C)(F)F)cccc(C(=O)NC2CC2NC(=O)CC2C=CS(=O)(=O)C2)c1 60824,N1(C(c2cc(C)c(C)[nH]2)=O)CC=C(CC(=O)NCc2cccc(F)c2)CC1 60825,N1(C(C2CC23CC3)=O)CCN(C(=O)C(F)CC2CC2)C2(CC2)C1 60826,c1(CC(=O)NC2CCN(C(C=C(C)C3CC3)=O)C2C)cc(C(F)(F)F)c(O)nn1 60827,C(CCCCC(=O)NCC1(F)CCC(NC(=O)C=Cc2ccco2)C1)=CC 60828,N1(c2nnc(OCC)s2)CCC(C)C(NC(c2cnn(C)c2C)=O)C1C 60829,N1(C(=O)C=C2CC2)CCOC2(C1)CN(C(=O)Cc1ccc(Cl)cc1O)C2 60830,Cn1cc2c(n1)CCCC2C(=O)N1CCCCC1CNC(=O)CC#N 60831,C(N=c1[nH]c2c(c(=NC(C)c3c[nH]nc3C)[nH]1)CCC2)C1(CSC)CCOCC1 60832,C1(CN(C)C(c2ccnc(C3CC3)c2)=O)CCCCN1C(c1cccn1C)=O 60833,C1(NC(C(C)Cc2ccccn2)=O)CC2CC1N(C(=O)Cc1csnn1)C2 60834,N1(C(C(C(CC)C)N(C(=O)CC2(C)OCCO2)C)=O)CC2CCCCC2C1C 60835,CCCC(C(O)C(=O)NC1CCN(C2CC2)C1)NC(C1(n2cccc2)CC1)=O 60836,c1(C(C)Cc2nc(-c3cccc(F)n3)no2)ccc(S(C)(=O)=O)cc1 60837,C(C1c2ccccc2CN1C(C1C2(CC2)C12CC2)=O)NC(C(C)OCC(C)C)=O 60838,N(C1CCCn2ncnc21)C(C(C)N(C(=O)CC(C)C(F)(F)F)CCC)=O 60839,Cc1nc(C(=O)NC2CC(NC(C3CCCN3C3CCCCC3)=O)C2)cc(O)n1 60840,C=CCCCC(C(=O)NC1(C)CC2(CC2)C1)NC(=O)C(F)CCC 60841,C1(NC(C(CC)(F)F)=O)CCCC12CN(c1nc(Cl)nc(C)c1F)C2 60842,C1(C)(C(=O)NC(CC)CN(C(c2cc(-c3ccoc3)on2)=O)CC)C=CCCC1 60843,N1(C(C(=O)NC(C)C)=O)CCC2(CCN(C(c3cccnc3NC(C)C)=O)C2)C1 60844,c1(C(=O)Nc2ncc(Br)cc2I)cc2c(s1)CCN(Cc1cc(Cl)cc(I)c1)C2 60845,CON1CCC(C(=O)NC2CC(C)N(C3CC3)C2)CC1.c12csc(c1)CNC2=O 60846,C1(N(C(C(C)=C2CC2)=O)C)CC2CCC(C1)N2C(=O)COc1ccsn1 60847,C1(CC(C)NC(c2ccc(N)cn2)=O)CCN(C(=O)Cc2cncs2)CC1 60848,CC(C)(C)C(=O)C(=O)N1CC2(CCC2NC(=O)CNC(C2CCC2)=O)C1 60849,c1(NCCC(C)(C)OC)cnn(C)c(=O)c1Cl 60850,c1(C(=O)NCC(C)N(C(=O)C(C)CF)CC)ccccc1NC(N)=O 60851,c1(OC)cccc(-c2nc(CC(=O)Nc3c[nH]nc3C#N)cs2)c1OC 60852,c1(CC(N2CC3C(C(N4CCC(CC)C4)=O)(C3)C2)=O)cccc(C#N)c1 60853,N1(C(C)=O)CCCCC1C(=O)NCC1CCC(F)C1 60854,N1(C(C(C2CCCO2)NC(c2c(C)nsc2)=O)=O)CCCN(C2CC2)CC1 60855,CC(C)CCCC(=O)NCCNC(c1scnc1C(C)C)=O 60856,C1(CC(=O)NC2CC(CNC(C3CC4CCC3C4)=O)C2)CCC(F)(F)C1 60857,N(C(=NCCCF)NCC1C(F)(F)C12CCC2)Cc1c(C)nn(C)c1 60858,C1(C(N)=O)(OC)CN(C(=O)C(C2CCCC2)NC(c2csc(C3CC3)n2)=O)C1 60859,c1(N(C)C)ccc(C(CNC(=O)CSC2CCOC2=O)NC(=O)C(N)=O)cc1 60860,CC1CN(C(c2cnn[nH]2)=O)CCC1C(=O)NCC1CC(C2CC2)C1 60861,C=C(C)CC(C)C(=O)NCC(C)(C)NC(c1ccsc1C)=O 60862,c1(CC)ccc(C(=O)N(C2CN(C(=O)C#CC3(C)CC3)CC2(C)C)C)c(O)c1 60863,N1(CC(=O)N(C(C)CN(C)C(c2cc(O)ccc2F)=O)C)Cc2ccccc2C1 60864,N1(C(Cc2ccc(C)cc2)=O)CCC(O)C(N(C(=O)C(O)C2CCC2)C)C1 60865,N1(C(c2ccc(C(=O)OC)o2)=O)CC2CCC(NC(C34CSCC3C4)=O)(C2)C1 60866,N1(C(C2CN(C(N)=O)C2)=O)CC2CC(NC(=O)CCC3CC3(F)F)CC(C2)C1 60867,Cc1ccc(CCC(N2CC(O)(CCNC(C3CC3(C)C(F)F)=O)C2)=O)o1 60868,C1(c2c(C(=O)NC3C(C)C3C)c[nH]n2)CCCCN1C(c1cnnc(O)c1)=O 60869,c1(C(=O)NC(CCN(C(CC2(COC)CC2)=O)C)C(C)C)ncc(C)cc1F 60870,CC1C(NC(c2c[nH]cc(F)c2=O)=O)CCCN1C(=O)CCc1ccccc1F 60871,C1(CCC)(NC(=O)Cc2cncc(C)c2)CCCN(C(=O)C2=C(C)CCC2)C1 60872,c1(C(N2CCC(F)(C(=O)NCC3CCC(F)(F)C3)C2)=O)cn2cc(F)ccc2n1 60873,C(=O)(CCCS(N)(=O)=O)NCCNC(CCCNC(CSC)=O)c1ccccc1 60874,N1(C(C2N(C=O)CCC2)=O)CCC2C1CCCN2C(c1cnc(OCF)cn1)=O 60875,C(=O)(CC1OCCc2ccccc21)N1C2CC(NC(C3CC3F)=O)CC1CCC2 60876,C1(CC(=O)NC(C)CCCNC(=O)CNc2cnn(C)c2)SC(=N)NC1=O 60877,c1(C(=O)NCC(C)(CO)NC(C2CC(C)C2)=O)ccc2cccc([N+](=O)[O-])c2n1 60878,c1(OCC)ccc2ccccc2c1-c1cc(COc2cc(C)c(C)cc2Br)on1 60879,CC(C(C)C(=O)N1CC(C#N)C1)NC(c1ccnn1CCF)=O 60880,c1(C(=O)NC2(CO)CCN(C(CCC(=O)NCC)=O)C2)cnn2c1NCCC2 60881,N1(C(c2cc(C)[nH]n2)=O)CC2CS(=O)(=O)CC2(CNC(=O)CCC(C)(C)C#N)C1 60882,C1(NC(c2cc(C)[nH]n2)=O)CN(C(c2snc(O)c2Cl)=O)C2(CCCOC2)C1 60883,N1(C(COC2(C)CN(C(C3CSC3)=O)C2)=O)CC(CO)C(C)(C)C1 60884,N1(C(CC2ON=C(CC)C2)=O)CCC(C(=O)NC(CC(=O)NC)C2CC2)C(C)C1 60885,c1(C(N2CC(O)(C(=O)NC)C2)=O)cnccc1C(=O)OC(C)(C)C.C1(O)CCC(C)C1 60886,C(C(COC)C(=O)NCC1(COC)CCCN1C(=O)CC1CCCN1C)OC 60887,CC1CCCc2cc(C(=O)NCC3(NC(=O)CCN4CCCC4)CCOC3)nn21 60888,CC1(C2CCN(C(C3CCN(C(=O)COc4cccnc4)CC3)=O)C2)CC1 60889,c1(NC2C(OC)C(C)(C)C2)nc2cccnc2c(=NCc2ccncn2)[nH]1 60890,S(=O)(=O)(c1cc(Cl)c(Cl)cc1Cl)NCCC1(C2C(C)CCCC2)NC(=O)NC1=O 60891,c1(C(N2CCC(OCCNC(CC(CCC)O)=O)C2)=O)cnc(S(C)(=O)=O)s1 60892,c1(C(N2C(CN(C)C(c3ncoc3C3CCCO3)=O)CCC2)=O)nc(=O)n(C)[nH]1 60893,C12(CC)CCC(CC1)N(c1nc(C(F)(F)F)c(NC(C3CC3C(=O)OC)=O)s1)C2 60894,C1(C(N2CCN(C(CCCOC)=O)C(CCO)C2)=O)CCc2ccccc2O1 60895,C1(NC(CC2(C)CCN(C(C(C(C)C)OCC)=O)C2)=O)CC2CC1CC21CC1 60896,c1(C(=O)NC2CCN(C(c3c(C)csc3)=O)CC2C)cnn2c1CC(F)(F)C2 60897,c1(C(N(CCC)CCNC(=O)C(C2CCOCC2)F)=O)ccc(C)cc1O 60898,C1CCCCC(=O)O1.C1(COCC)CCCC1NC(=O)CNC(c1cccs1)=O 60899,C(=O)(CC(C)C(C)C)NCC1(CNC(C2N(CC)CCC2)=O)CCC1 60900,N1(C(CC2N(C(C(C)OCCCC)=O)CC(O)C2)=O)CCC(F)(C#N)C1 60901,c1(C(=O)NCCCC(c2ccccc2)NC(CC=C)=O)cccc(=O)o1 60902,C(CC(C)(C)CC(=O)NC(C1(O)CN(C(=O)CC(C)c2ccccc2)C1)C)OC 60903,C1(NC(=O)NCc2nnc(CC)o2)(CSC)CCCCCCC1 60904,N1(C(c2n[nH]c(CC)c2C)=O)CCC2CCCC12C(N1CCC(CC)C1)=O 60905,C1(SC)CN(C(=O)CC2CCC(=O)N2C)CC1NC(C1(C2CCCO2)CCC1)=O 60906,C=C(C)CC(C(=O)NCC1(C)CCCS1)NC(=O)CCOCCOC 60907,c1(C(N2C(C(N3CCCC(C)(O)C3)=O)C3CCC2C3)=O)n[nH]c2ccc(F)cc12 60908,CCC(CCC(=O)N1CCCCC1CN(C(=O)CN1CC(C)(OC)C1)C)OC 60909,N1(C(COC2CCN(C(c3n(COC)ncc3)=O)C2)=O)CCN(C)C(=O)C1CC 60910,CC1CN(C(c2c[nH]cc2C(C)(C)C)=O)CC1NC(C1CCC(=O)N1)=O 60911,c1(CC)ccc([N+](=O)[O-])cc1C(N1CC(O)(C(C)NC(C2CC2C(F)F)=O)C1)=O 60912,Cc1cc(C(=O)NC(C)C(C)(C)C(N2CC3CC(O)CC2C3)=O)ccc1C#N 60913,C(Cc1ccco1)(C(=O)N(C)Cc1cc(C)no1)NC(C=CC(CC)C)=O 60914,c1(C(N2CC(NC(C3(COC)CCC3)=O)CC2(C)C)=O)cc(Cl)c(OC)cc1Cl 60915,c1(COC)nc2n(n1)CC(NC(=NCCCF)NCC1(CO)CCN(C)CC1)CC2 60916,c1(CC)cc(C(=O)N(CC(C)NC(=O)C=Cc2nc(C)cs2)C)ccc1OC 60917,CC1CCN(C(=O)CCCCF)CC1CNC(=O)CNC(c1cc(F)cc(F)c1)=O 60918,CC(C)C(O)C(C)(C)C(=O)N1CCC(C(=O)NCC2(C)CCCCC2O)O1 60919,c1(C(=O)OCC)n[nH]c(=NC2CCN(C(c3cn(C)cc3C)=O)C(C)C2)s1 60920,N1(C(=O)OC(C)(C)C)CCN(c2ccnc(CNCC3CNC(=O)C3)n2)CC1 60921,C=CCCCC(C(=O)OC)NCc1cc(Br)c(F)cc1OC 60922,c1(CCCC(=O)N(C)CC2(NC(c3cnn(CC)n3)=O)CC2)ccccc1OC 60923,C1(C(=O)NC(C2CC(C(=O)NCCC(O)C3CCC3)C2)C)CCCN1C=O 60924,Cn1nnc2cc(C(N3CC4CCC4(NC(c4csc([N+](=O)[O-])c4)=O)C3)=O)sc12 60925,C1(C(=O)NC(CN(C(c2cnc(O)n2CC)=O)CC)C)CCCCC1(C)C 60926,C(C1c2ccsc2CCN1C(C1C(C)C1C)=O)NC(C(=O)NC(C)C)=O 60927,Cc1cc(C(N2CCCCC2CS(N)(=O)=O)=O)ccc1Br 60928,S(=O)(=O)(c1cc(C)cnc1Cl)N1CCC(C(=O)Nc2cccc(C(C)=O)c2)C1 60929,C(=O)(C(=O)CCC(C)C)NC1(CC=C)CN(C(C2CC=CCO2)=O)C1 60930,C#Cc1ccnc(C(=O)NCCOC2CCN(C(=O)CC(C=C)CC)CC2)c1 60931,Cc1cc(-n2nc(CCCN(C)C)nc2C(N2CCC(C)C2)C)ccc1Cl 60932,c1(OC)cccc(-c2cn(C3CCC(C(=O)NCC4CNC(=O)O4)C3)nn2)c1F 60933,c1(-c2onc(CN3CCC(O)(CO)C3)n2)cc2ccccc2c(O)n1 60934,C=CC1(C(=O)NCCCN2CC=CC2)CCN(C(=O)C(C2CCCCC2)C)CC1 60935,c1(C(=O)NC(CCCNC(c2c(NCC)scn2)=O)C)cnc2c(c1)CCOC2 60936,c1(SC)cnn(C)c1C(N1CC(NC(=O)CNS(N)(=O)=O)C(C)C1)=O 60937,c1(NC)c(C)csc1C(=O)N(C1CC(NC(=O)CCN(c2ccncc2)C)C1)C 60938,c1(-c2cc(OC)nnc2OC)cnc2[nH]cc(C(=O)N=c3nc[nH]s3)c2c1 60939,c1(C(=O)NC(C)Cc2ccc(CNC(C3CC3C)=O)cc2)ccc(N)cc1F 60940,C1(CNC(C(n2cc(Cl)cn2)C)=O)CC2(CCC2)CN1C(C1CCCC12CC2)=O 60941,Cc1ccc(O)c(NCCCc2ccccc2C(F)(F)F)c1 60942,CC1CN(C(=O)CNC(N)=O)CC1NC(c1cncc(C(C)(F)F)c1)=O 60943,CC(c1ccsc1)=CC(=O)NCCCC(C)NC(c1ccc(CO)s1)=O 60944,C(c1ccc(Br)cc1)=CCC(=O)NCC=CCNC(C1CCC(F)C1)=O 60945,c1(C(=O)NC2(CCNC(=O)CCn3cc(Cl)cn3)CC2)cc(O)nc(O)n1 60946,Cc1cc(C(=O)NC2CCC2NC(c2[nH]nnc2C2CC2)=O)cc(C)c1Cl 60947,C1(C(N2CC(NC(c3c(CC)ncs3)=O)(CO)C2)=O)CC(=O)N(C2CN(C)C2)C1 60948,C1(CNC(C(CC=C)NC(C)=O)=O)COCCN(C(=O)C(=O)NC(C)C)C1 60949,C1(CN(C(C(C)n2ccnn2)=O)C)CCCN1C(C1CCCN1C1CC1)=O 60950,C1(C(=O)NC(C2CCOC2)CC)(CNC(c2ccns2)=O)CCCC1 60951,c1(C(N2CCC3(CC(C)OC3)C2)=O)ccc2c(n1)CN(C(=O)CC1(C)CC1)CC2 60952,c1(NC(C)=O)cnccc1C(=O)N(CCNC(C1CC1(C)C(C)C)=O)C1CC1 60953,C#Cc1ccc(CC(=O)NCC=CC(=O)NCC(C)C)cc1 60954,c1(C(N2CCC(O)(CCNC(CSSC)=O)CC2)=O)ncnc2c(C)csc12 60955,Cc1ccc(C2CC2C(N2CCCC(N(C)C(c3cnccc3Cl)=O)C2)=O)cc1 60956,c1(C(=O)NCC2N(C(COC)=O)CC=C2)cccc(-n2cccn2)n1 60957,C1(C(N(C(C)C)C)=O)CC2(CCN1C(C1CCOCC1)=O)CC2 60958,C(c1cccc(Cl)c1)=CC(=O)N(C1CCN(C(c2c(C)coc2)=O)C1)CCO 60959,C1(CC(=O)NCCNC(C(C)n2cccn2)=O)CCN(CCF)CC1 60960,C1(C(N(CC(CNC(CN(C(C(C)C)=O)C)=O)C)C)=O)CN2CCN1C(C)C2 60961,C(N=c1cccc(S(=O)(=O)NCC=CBr)[nH]1)C1C(c2ccc(C)cc2)CCC1 60962,N1(C(C2(CCC)CC2)=O)CCC2(CO)CN(C(=O)CC3CCCCCC3)CC2C1 60963,Cc1nc(Cl)[nH]c(=NCC2C3CN(C(=O)C(C)Cc4ccc(F)cc4)CC23)c1F 60964,C(=O)(C(O)C(CCC)NC(=O)C(C#N)C(C)C)NCC1(C=C)CCC1 60965,C12(CNC(C(CC=C)(F)F)=O)CCC(CNC(C3(C)CC3(F)Cl)=O)(CC1)CO2 60966,c1(C(=O)NC23CC(NC(c4nccc(C=C)c4)=O)(C2)C3)cccn2ccnc12 60967,CC(C)CCCCC(=O)NC(CCN(C)C)C(=O)NCCC1CCC1 60968,N1(C(CC(F)(F)F)C=C(C)C)CC(n2cc(C3(C)CCCO3)nn2)C(O)C1 60969,C1(CS(=O)(=O)NCC(CCOC)O)CN2CCCCC2CO1 60970,C12(C(N(C(C)CNC(=O)Cc3ccnn3C)CC)=O)CC3CC(CC(C3)O1)C2 60971,N1(C(Cn2c(C)ccn2)=O)CC(C)CN(C(=O)C2=CSCCO2)C(C)C1 60972,[N-]=[N+]=NC1CC2(C(N3CC(O)(CNC(C4(Cl)CC45CCC5)=O)C3)=O)CC12 60973,N1(C(CC2(NC(C(C)C3CCCO3)=O)CC2)=O)CCC(CCF)CC1 60974,c1(C(C(=O)NCCCF)N(C)Cc2ccsc2)ccc(OCC#N)cc1 60975,C=Cc1ccc(CN2CC3(CN(C(c4ccccn4)=O)C3)C2)cc1 60976,C(=O)(C1CCCn2cnnc21)NCC1C2CN(C(=O)OC(C)(C)C)CC21 60977,O=CN1CCCC1C(N1CC(O)CC1CNC(=O)C(O)c1ccco1)=O 60978,Cc1nc(CCC(N2CCC(CNC(=O)CC3CSCCS3)C2)=O)cs1 60979,c1(OCC)ccc(S(=O)(=O)NC2CC(S(C)(=O)=O)C2)cc1-c1cccc(C)c1 60980,Cc1cnc(C)c(NC(C2CC(F)CN(C(=O)Cc3cccs3)C2)=O)n1 60981,C1(NC(c2cnc(C)o2)=O)CCN(C(C2CC23CCSCC3)=O)C1(C)C 60982,S(=O)(=O)(c1ccc(Br)cc1NCC(c1ncccn1)O)N(CCO)CC 60983,N1(C(C2C(C)C2(F)F)=O)CC(NC(c2cc(N)nc(Cl)c2)=O)CC(C)(C)C1 60984,c1(OC)ccc(CN2CC(CNC(c3ncoc3C)=O)C2)nc1Br 60985,C1(C(=O)NC(C)CCN(C(=O)CCc2ccco2)C)CC2(C1)CC2F 60986,C=CC(C)(O)C(=O)NC(C1CN(C(c2ccnc(SC)c2)=O)CCO1)C 60987,N1(C(C(=O)N(c2ccccn2)CC)=O)CC2CC1C2CNC(c1c(C)ccn1C)=O 60988,CN1CC2CCN(C(=O)CCN(CCCO)C(C3CCC(=O)N(C)C3)=O)CC2C1 60989,CN1CCCC(CCC(N2CC(NC(c3ocnc3C3CCC3)=O)C(O)C2)=O)C1 60990,c1(CC(=O)N(C2CCCCN(C(c3cnc(O)o3)=O)C2)C)cn2ccsc2n1 60991,c1(C(N(C)CCN(C(=O)C(O)CC(N)=O)C)=O)cc2cc(Cl)sc2[nH]1 60992,C1(NC(C2(CC)CCC2)=O)CCN(C(=O)CSCCN(C)C)CCC1CO 60993,N1(C(COCCCC)=O)CC(C(N2CCCC(C(C)(C)C)C2)=O)CC1(C)C 60994,CCCCS(=O)(=O)NC(C)C(=O)NCCCN(C(=O)CC1(CO)CC1)CCO 60995,c1(CNC(=O)NCc2c(CS(=O)(=O)NC)cccc2)cnc(Cl)cc1Cl 60996,c1(CC(=O)NCC(C)N(C(c2ccnnc2)=O)CC)cc(Br)cnc1OC 60997,C=Cc1cncc(C(N2CCC(C(=O)N(CCCO)CCC)C2C(C)C)=O)c1 60998,C1(CNC(C(C)OCCC=C)=O)CC(C(N2CC(N3CCCCC3)C2)=O)CO1 60999,c1(OCC(N2CCC(C)N(Cc3ccccc3)CC2)=O)ncnc2ccccc12 61000,CCC(C(=O)NC1CC(CN(C(=O)C(C)N(C)C)C)C1)C(C)(C)CC 61001,C(CC(C(=O)N(C1CC(C(=O)OC)C1)C)NC(c1cc(CO)oc1C)=O)=CC 61002,O=C(C1=CCCOCC1)NC(CNC(C1(F)CC1c1ccccc1)=O)CO 61003,CC1CCC(CNC(=O)Cc2cncnc2O)CN1C(c1cc(=O)n(C)cn1)=O 61004,CCC(C)C(O)C(C)C(=O)N1CC2CCC1CN2C(=O)CN1C(=O)CNC1=O 61005,Cc1nc2cccc(C(=O)NCC(CO)NC(C3(C)CCN(C)C3=O)=O)c2[nH]1 61006,N1(C(C(C)CC2CCCC2)=O)CC2CC1CC2NC(C1(C)COC1)=O 61007,C(=O)(C(=O)N=S(C)(C)=O)NCCC1CN(C(=O)C=Cc2ccsc2)CC(C)O1 61008,c1(CN2CC3N(C(C4CC4c4ccc(F)cc4)=O)C(C3)C2)cc(Br)cc(Cl)c1F 61009,C1(NC(c2n[nH]c(C3CC3)c2Br)=O)CCCCN(C(=O)CC2CCCC2)C1 61010,c1(OC)ccc(Br)c(C(N2CC(OCCCOC)C2)=O)c1C 61011,N1(C(=O)CCCF)CCCC2C1CCCN2C(=O)CSCC(F)(F)F 61012,C1(NC(=O)Cc2ccccc2C2CC2)CCS(=O)(=O)C12CN(C(=O)CC1CC1)C2 61013,CCC(CC(=O)NC1COCC1NC(c1ccnc(C2CC2)c1)=O)C(F)F 61014,N1(C(CC2(COC)CCCC2)=O)CCCC1(C)CNC(=O)CC12CCCC1C2 61015,c1(CCC(=O)NC(CC2CN(C(C(COC)OC)=O)C2)C)cccc(F)c1 61016,CCCCCC(O)CNC(c1ccc(OC(C)C)nc1)=O 61017,N1(C(C=C(CCC)C)=O)CC2CC(NC(=O)C=Cc3cccs3)CC(C2)C1 61018,C(C(=O)NNC(=O)C(F)(F)F)C(c1c(C)cc(C)c(C(C)=O)c1C)=O.N 61019,Cc1nc(C)n(CC(=O)NC2COCCC2C(=O)NCC2CCOC2)n1 61020,N#Cc1ccc(CCC(N2CCOCC2CC(C2CCCCC2)=O)=O)cc1 61021,C(=O)(C(C)(C)C(=O)NCC(C)NC(c1ccc(SC(F)(F)F)s1)=O)OCC 61022,c1(C(N2CC(CC)(NC(=O)CC3CC(=O)NC3=O)C2)=O)cncc(F)c1C 61023,N1(C(=O)CCN2CCC(O)CC2)CC2(C1)CN(C(c1ccc(O)cc1F)=O)C2 61024,Cc1cc(CCC(=O)NCC(C)(C)CN(C)C(C2CCN(C)C2)=O)nn1C 61025,C(=O)(C(F)CC(C)(C)NC(c1ccccc1)=O)N1C(C)(CC)CC1 61026,C(CC(C)(C)NC(c1cnoc1C1CC1)=O)N(C(C(c1cnn(C)c1)C)=O)C 61027,C1(NC(c2n(C)nc(Br)c2)=O)CCN(Cc2cccc(C(F)(F)F)c2O)CC1F 61028,C1(NC(=O)COCCCF)CN(C(c2cnc3ncccn23)=O)C2(CCCC2)C1 61029,C(=O)(C(C)(C)C)NC(C)C(=O)N(C)CCN(C)C(C1(CC2CC2)CCCO1)=O 61030,Cn1cnc2ccc(-c3cnc(F)c(F)c3)cc12 61031,c1(NC(N2CCN(Cc3ccccc3)C(c3cccs3)C2)=O)ccc(Br)cc1Br 61032,n1(CCOC)c(SCCc2nncs2)nnc1-c1ccccc1 61033,C1(NC(CS(=O)(=O)NC)=O)CCN(C(=O)C(n2cc(Cl)cn2)C)CC1O 61034,c1(CC(=O)NCC(CNC(Cn2c(C)c(Cl)cn2)=O)C)cc(C(C)C)cc(F)c1 61035,C1(NC(COCc2ncc(C)o2)=O)CCC(C)(CNC(=O)CCc2ccsc2)C1 61036,c1(C(=O)NC2C(CNC(c3cn(C(C)C)nc3)=O)CC2)cccc2c1CCCC2 61037,N1(C(=O)COC(F)F)CCN(CC(c2ccccc2)F)CC1.c1(N)ccccc1 61038,c1(C(=O)NC2CCCC(NC(C3CCCS3(=O)=O)=O)C2)cnc2ncc(Cl)cn12 61039,C1(C2CCN(C(=O)Cc3cc(Cl)ccc3Cl)CC2)(NC(C2CNC(=O)N2)=O)CC1 61040,C1(C(=O)NCCC2CCCCN2C(=O)COCCCF)CC2CC1CC2(F)F 61041,c1(OCCC)ccccc1C(N1CC(NC(C2CC(C(C)(C)C)C2)=O)C1)=O 61042,O=C(CC1COc2ccccc21)NC1CC(NC(=O)C(F)(F)c2cncs2)C1 61043,C(=O)(CC(CC)C(F)F)NC1CCC(CCC(=O)NCc2scc(CC)n2)C1 61044,c1(C(N2CCC(N(C(C(C)OCC=C)=O)CCO)CC2)=O)ccc(F)cc1C 61045,N1(S(CCC)(=O)=O)CCC(C(N2CCC2CNC(=O)CCC(C)OCC)=O)CC1 61046,C(=O)(C(O)C(F)(F)F)N(CCCNC(c1cnns1)=O)Cc1ccccc1 61047,CCC(CC(=O)N(CC(C)NC(C1(c2cc[nH]n2)CC1)=O)C)SC 61048,C1(C(N2CCC(COC)C2)=O)CCN(C(c2cscn2)=O)CC1 61049,N1(C(CNC(=O)NC)=O)CCC(CO)C(NC(=O)CN2CCC(C)(C)C2)C1 61050,Cc1cc(=NCc2cnccc2C)[nH]c(=NCc2ccn3ncnc3c2)[nH]1 61051,c1(OC)cc(C(=O)NCC2CCN(C(=O)CCN(C)CCO)C(C)C2)cc(C)c1 61052,c1(CC(=O)NCC2CC(NC(CC(C=C)C)=O)C2)cc(C)ccc1O 61053,C1(CSC)CC(OCC(=O)NC(C)C)C1(C)C.C1(=O)CN(C)CC(=O)NC1 61054,C(CC(C)C)(C(=O)N1CCC(CNC(c2nnn(C(C)(C)C)n2)=O)C1(C)C)OC 61055,CC(C)CCC(C)N=c1[nH]c(=NC(C)CN(C)C(C)C)[nH]c2cc[nH]c12 61056,CC1(C(=O)NCC(C2CCOC2)NC(c2cnc(N(C)C)cn2)=O)CCCCC1 61057,c1(NC(=O)CSCC(N2CCCOC2)=O)csc(=Nc2ccccc2)[nH]1 61058,C1(CC)CN(C(=O)Cn2ncnn2)CCN1C(=O)Cc1cc(O)ccc1Br 61059,C1(CNC(C=C(C)C)=O)(CNC(=O)Cn2cnc([N+](=O)[O-])n2)CC2CCCC2C1 61060,c1(OCC(CC)CNC(=O)C(n2cc(CCC(C)(C)O)nn2)C)cccc(C)c1 61061,C1(C(=O)NC(C(CO)NC(CCSCC(=O)OC)=O)C)CCc2ncc(C)n2C1 61062,c1(OC)csc(C(=O)NCC2CCC(NC(C3CC34CC4)=O)C2)c1 61063,C12(NC(CNC(C(C)(C)C3CCCCC3)=O)=O)CC1CS(=O)(=O)C2 61064,N#Cc1sc(=NCC2CCN(C(c3cc(Cl)no3)=O)C2)[nH]c1Cl 61065,C1(NC(C2OCCN(C)C2)=O)CC2(CCN(C(c3ccc(C#N)c(O)c3)=O)C2)C1 61066,c1(C(=O)NCC2C(CNC(=O)C(F)n3ccnc3)C2)cc(-n2ccnc2)ncn1 61067,N1(C(c2cnn(CC)c2C)=O)CC(CNC(=O)C=CS(C)=O)OC2CCCC12 61068,c1(C(N(C)CCNC(C2CCCN(C(=O)CNC=O)C2)=O)=O)ccccc1[N+](=O)[O-] 61069,CC(C)C(O)C(=O)N(CCCNC(=O)CCN1CCCCCC1)C(C)C 61070,c1(C(N2CCC(CNC(C(C(C)C)F)=O)C2(C)C)=O)nccc2cccnc12 61071,Cc1noc(-c2cn(CC(=O)NC3CC3CNC(c3ccoc3Br)=O)cn2)n1 61072,C1(CNC(CCCSC)=O)CSCCN1c1nccc(CC#N)n1 61073,CS(C)(=O)=Nc1ccc(C(N2CC3CCCC3(CNC(C3(F)CC3)=O)C2)=O)cc1 61074,Cn1cnc(NC(=O)NCC2(c3cccc(C(F)(F)F)c3)CC2)cc1=O 61075,N1(C(c2ccc(C)o2)C(=O)CC2(NC=O)CCC2)CCn2c(C)nnc2C1C 61076,C=CCC(C(=O)OCC)NC(=O)CCN(C(C1CCC1C)=O)CC1CC1 61077,C(=O)(CCC(C)C#N)NC1(C2N(C(c3c(C)cc(C(F)F)o3)=O)CCC2)CC1 61078,c1(C(=O)NCC2(OC)CCN(C(=O)C=Cc3cccnc3)C2)cc(C)c(C)cn1 61079,C(=O)(CC(C)(C)C(C)(F)F)NC(CCN(C(C1(OCC)CCC1)=O)C)C(C)(C)C 61080,Cc1[nH]nc2c(C(N3CCC(CO)(NC(C4CNC(=O)N4)=O)CC3)=O)cccc12 61081,N1(C(C2CN(C(CNC(N(C)C)=O)=O)CC(F)(F)C2)=O)CCC2(CCOC2)CC1 61082,C(N=c1[nH]c(=NCC(C)(F)c2ccccc2)c2[nH]ccc2[nH]1)C1C(C)(C)C1 61083,C(C1CCCN1C(c1cnn(C)c1N)=O)=CC(N1CCC(CN(C)C)C1)=O 61084,c1(OCC)ccc(CC(N2CCC(NC(=O)C=CSc3ccccc3)C2)=O)cc1 61085,N1(C(C(CC(CC)C)C)=O)CC2CCCN(C(=O)COC3CC3(C)C)C2C1 61086,C1(C(C(=O)NCCC(CNC(C(CSC)(C)C)=O)O)O)CCCCCCC1 61087,C1(NC(C2CN(CC)C(=O)C2)=O)CCC12CN(C(c1cn(CC(N)=O)nn1)=O)C2 61088,CC1(C)C(CN(C(=O)Cn2ncnn2)C2CC2)CCN1C(C1CC1c1ccco1)=O 61089,C12(NC(CCc3cnc(C)o3)=O)CCN(C(c3ccn(C)c3)=O)CC1C2 61090,c1(COC)cc(C(N2CC(NC(=O)CSCC)C(c3nccn3C)C2)=O)n(C)c1 61091,c1(C(=O)NCC(C)NC(=O)C(F)CC2CC2)ccc(Br)cc1 61092,c1(CC)nn(C)c(Cl)c1C(=O)NC1C2CN(C(C3(c4cc[nH]n4)CC3)=O)CC12 61093,Cc1nn(CC(F)F)c(C)c1C(N1CCC(c2ccnnc2)CC1)=O 61094,CC1CN(C(=O)NC2CC2C(F)(F)F)CCN1c1ccncc1 61095,c1(C(=O)NCC(C(=O)Nc2c(CC)cccc2)(C)CC)ccc2nccn2c1 61096,C1(NC(C(CC#C)(C)NC(c2c[nH]c(=NC)o2)=O)=O)CC2CC1CC21CC1 61097,C1(NC(C2N(C)CCCC2)=O)CN(Cc2ccnc(F)c2Cl)CC1C#N 61098,N1(CCN(CC)CC)CCCCC1C1(NC(=O)COCC(C)C)CC1 61099,N1(CCC#C)CCN(C(=O)NC2C3CCC(F)C23)CC1 61100,C(=O)(CS(=O)(=O)Cc1cncn1C)NC(c1ccc(Cl)cc1)C(C)C 61101,CC1CC(C)N(C(c2cn3c(Br)cccc3n2)=O)CCN1C(=O)COCCF 61102,N1(C(Cc2cccc(OCCC)c2)=O)CCN(C(=O)CCCF)CC1CSC 61103,C1(NC(C2CCC(C)O2)=O)CCC2CN(C(=O)C(c3ccccc3)C)CCC2C1 61104,c1(CC(N2CC(C(N)=O)(CNC(C3C(C)C3C)=O)C2)=O)cccc(Br)c1 61105,N1(C2CCC(NC(C)=O)C2)CCN(C(=O)CCN(CC(F)(F)F)C)CC1 61106,CC(C)=C=CC(=O)N(CCC(C(C)C)NC(c1ncoc1C1CCC1)=O)C 61107,C1(NC(C2NC(=O)OC2)=O)CCN(C(=O)CCSc2ccccn2)C12CC2 61108,N1(C(C(N)=O)=O)CC(NC(=O)CNC(=O)CC2CCCCC2)CC12CCC2 61109,C(=O)(C(C)S(C)(=O)=O)NC1C(CC)N(C(=O)CCn2ccnc2)CC1 61110,N(C1CCCc2cc(C#N)ccc21)c1nccc(N2CCN(C(C)(C)C)CC2)n1 61111,C(C(C)C(F)C(=O)NC(C)C(C)SC)NC(C1(C(=O)OC)CC1)=O.C(C)(=O)O 61112,C(=O)(C1=CC2CCCC12)N1CCCC(C)(NC(CC(c2c(C)noc2C)C)=O)C1 61113,Cc1onc(C(F)(F)F)c1C(=O)NC1CCN(C(=O)CN2C(C)CCC2C)CC1 61114,Cc1ccc(=O)n(CC(=O)NCCCCNC(=O)C(c2ccc(F)cc2)(C)F)n1 61115,CCC(C)(C)C(C)Cc1nc(-c2cccs2)nn1-c1cnnn1C 61116,C1(C(=O)NC(=O)OC)C(CC)CCN1C(=O)C(C)Sc1ccco1.c1ccccc1 61117,CC(CCN=c1[nH]c(=NCc2csc(N(C)C)n2)c2[nH]ccc2[nH]1)CC(C)(C)C 61118,CCCC(C)(O)CC(=O)N(C1CCC(CNC(=O)Cn2cnnn2)CC1)C 61119,C1(Cl)(C(=O)NCCNC(c2cnc(C(F)F)s2)=O)CC12CCOCC2 61120,C12(CNC(C3(CC)CC3)=O)CCCCC1CN(C(c1ccc(CSC)cc1)=O)C2 61121,Cc1nc(C=CC(=O)NC2CC23CC(NC(=O)CCNC(N)=O)C3)[nH]c1C 61122,c1(C(=O)NCC(C)CN(C)C(c2cnn(C(F)F)c2)=O)cc(C(F)(F)F)c[nH]1 61123,c1(C(N2C(C)CN(C(c3cc(SC)oc3)=O)C(C)C2)=O)ccc2c(c1)N(C)CC2 61124,C1(C(=O)N(CC(O)CN(C(=O)Cc2n[nH]cc2Br)C)C)(OC)CCCCC1 61125,C(=O)(N=c1[nH][nH]c2c1CN(C(c1c(F)cc(Br)c(F)c1F)=O)C2)C1C(C)(C)C1 61126,CCC(C)C(C(=O)NC1CC(F)(F)C1)N1CCC(C(=O)NCCC#N)CC1 61127,C1(C(=O)NCC2CCN(C(c3ccccc3O)=O)C2)CCC2C(CC1)C2(F)F 61128,C1(NC(Cc2c(C)ccs2)=O)CCCC(NC(=O)CC(=O)N(C)C)CC1 61129,C12(CNC(C(C(CC)C)OC)=O)CCC(CC1)N(C(=O)Cc1cccnc1F)C2 61130,c1(C(N(CCOC)CCNC(=O)C(O)C2CCC2)=O)cc(P(C)(C)=O)cs1 61131,c1(C(=O)NCC(C)N(C(c2c(NCC)scn2)=O)C)c[nH]c2ccc(F)cc12 61132,c1(C(N2CC(CNC(CC(CCC)O)=O)CC2(C)C)=O)ccc(N)cc1[N+](=O)[O-] 61133,C1(NC(C(C(C)C)O)=O)CCC(C)(CNC(c2nn(C)cc2Br)=O)CC1 61134,CC(C)C(C)C(=O)NCc1cc(C(=O)NOCC2CCOC2)on1 61135,Cc1ccc(C(=O)NCC(c2ccccc2)CNC(=O)CC#N)c(F)c1 61136,n1(CC)cc(Cl)c(C(=O)N(CCNC(C2(OC)CC(C)C2)=O)C(C)C)n1 61137,C1(CC(C(=O)NCCCF)N(C)CCn2cncn2)CCC(C)(C)O1 61138,Cc1ccccc1C=CC(=O)NC1CC(C(C)NC(c2ccoc2)=O)C1 61139,c1(C(=O)NC2CC(NC(C3(C)CCCCO3)=O)C2)cc2sc(Cl)cc2s1 61140,N1(C(C(CC)NC(N)=O)=O)CC(NC(=O)C#CC(C)C)C(C)C1 61141,C(c1cc[nH]n1)=CC(=O)NCCC1(N(C(C2CCCC2O)=O)C2CC2)CC1 61142,Cc1cccc2c1OCCC2NC(=NCCN1CCCC1C)NCC1CC1 61143,CC(C)(CS(C)(=O)=O)C(=O)NCC1COCCN1C(=O)CC1CCCNC(=O)C1 61144,C#CCC(C(=O)NCC(N1CCOCC1)=O)NC(=O)C(F)OC(F)(F)F 61145,C1(CC)CCN(C(c2cscc2Cl)=O)C1C(=O)NC1(CC(N)=O)CC1 61146,c1(CN2CC3C(CNC(c4c(C)ccc(C)c4)=O)C3C2)ccc2c(c1)CCC2 61147,CC1(C)OC2(CN3CCN(c4cncc5nccn45)C(CC#N)C3)CCC1C2 61148,C(=O)(C(CCC)C(C)C)N1CC(NC(CCC=CC)=O)C2(C1)CC2 61149,N1(C(C(CSCc2ccccc2)NC(C)=O)=O)CC2(CC(NC(=O)C(C)C)CO2)C1 61150,C(C)(CNC(c1cn(-c2ccn(C)n2)cn1)=O)(CO)NC(C=C(C)C)=O 61151,c1(OC)cccc(C(C)CC(=O)NCC2(NC(=O)C(c3ccnn3C)O)CC2)c1 61152,CCCC(C)(CC)C(=O)N1CCC(CN(C(=O)CSCC(=O)NC)C)C1 61153,CC1(C)CN(C(c2sc(C#N)cc2Cl)=O)CC(CNC(c2n[nH]cc2F)=O)O1 61154,Cc1c(C(=O)NCC2(NC(=O)C(C(C)C)NC(N)=O)CCOCC2)cnn1C 61155,C(CC(=O)N1CCC(CC(N)=O)C1)(C(C)(C)C)NC(Cc1ccc(C#C)cc1)=O 61156,N1(C(C=CCN(CC)CC)=O)CCOC(C(N2CC(C)(COC)C2)=O)C1 61157,Cc1cc2c(C(=O)N(C(C)CCNC(C3CCNC(=O)C3)=O)C)cccc2o1 61158,c1(NCC2CC(N(C)C)C2)cc2oc(-c3ccccc3)cc2[nH]1 61159,c1(C(=O)NC2CCN(C(C(C)(C)NC(=O)OC)=O)C2)cc(C)nc2cc(C)nn12 61160,C1(CNC(C2C(CNC(C(CC#C)O)=O)C2)=O)CCC2(CC2)CO1 61161,c1(C(=O)NC2C(NC(C(C(=O)OC)C)=O)CC2)cnc2cc[nH]c2c1 61162,C(=O)(C1=NOC(C)C1)NCCN(CCC)C(c1cccc(CNC(C)=O)n1)=O 61163,c1(C(N(C)CC2CCCN(C(CC(COC)C)=O)C2)=O)c(OC)cccc1F 61164,C#Cc1ccc(OC)c(C(N2CC(CNC(=O)C=CSC)CC23CCC3)=O)c1 61165,Cc1cc(C(=O)NCCCN(C(c2ccc(C(F)F)s2)=O)C2CC2)[nH]c1C 61166,C1(NC(C23CC(NC(C(CCC)Cl)=O)(C2)C3)=O)CC2(CCC2)CO1 61167,C1(NC(c2ccc(N(C)C)cc2)=O)CC2CC1CN(C(c1cc(Cl)no1)=O)C2 61168,c1(C(N2CC(NC(Cc3n(C)cnn3)=O)C2)=O)ncsc1S(N)(=O)=O 61169,CCS(=O)CC(=O)NCC1CCCC(CNC(C2(n3cnnn3)CC2)=O)C1 61170,C(=O)(C1CCc2cccnc21)NCC(CCNC(c1ncn(C)n1)=O)O 61171,C=C(Cl)CCC(=O)N1CCCC(N(C(=O)CC(=O)NCC=C)CC2CC2)C1 61172,N1(C(c2cc(C)n(C)c2)=O)CC2(CCN(C(c3ccc4occc4n3)=O)CC2)C1 61173,C#CCCCC(=O)N1CCN(c2ccccc2NC(C2CC(O)C2)=O)CC1 61174,Cc1ccc([N+](=O)[O-])cc1-c1cnc(C(=O)Nc2c(O)cccc2C#N)cn1 61175,c1(C(N2C3CC(NC(C=C(C)C)=O)C2CC3)=O)c(F)cc(F)cc1Br 61176,C(C)(CCC(=O)NC(CCC1CCC1)C(=O)NCCc1ncccc1F)OCC 61177,CC1(C)CC(CC(=O)NC2(CO)CCN(C(=O)C(=O)C(C)(C)C)C2)C(=O)O1 61178,c1(SC)ccc(C(N2CCCC(C)C2C(=O)OC)C(=O)NC(C)C)cc1SC 61179,c1oc2ccccc2c1C(N=S(C)(=O)CCN)=O.c1(C(=O)N)csc2ccc(Cl)cc12 61180,N1(C(CN2CCC(C)C2)=O)CCC2(CC2)CC1C(=O)Nc1cnc(Cl)nc1 61181,c1(C(=O)NC(CNC(C(CCCC#C)C)=O)C)cnc2[nH]c(C)nc2c1 61182,c1(COC(c2cc3[nH]nc(C(=O)OC)c3cc2)=O)nc2cc(C)cc(C)c2[nH]1 61183,CCC(CC)C(C(=O)N1CC2(C)CC1(C(N1CCCCC1CC(C)C)=O)C2)OC 61184,C=CC(C)(CC)C(=O)NCC1=CCN(C(=O)C(C)c2cncs2)CC1 61185,CCCCC(C(=O)NCC1(O)CCCN(C(c2cnn(CC)c2)=O)C1)N(C)C 61186,C1(NC(C(CCC)NC(N)=O)=O)CC2CC1CN(C(=O)CCCCC(C)C)C2 61187,CC1(C)C(c2cccc(F)c2)CCN1CC(=O)NCCSCc1cccnc1 61188,C=C(C)C(C)(C)C(=O)NCCC(O)CNC(=O)C(C)OCC1CC1 61189,CC(C)(CC1CCOCC1)C(=O)NCC(C1CCCC1)NC(C1CC(CF)C1)=O 61190,c1(CC2(C(=O)NCCNC(=O)C(F)(F)c3cnccn3)CC2)ccccc1Br 61191,C1(NC(CCc2cccc(OCC)c2)=O)CCCCN(C(C2CCN2CC)=O)C1 61192,CC1CN(C(=O)CC2(C)CCCCC2)CCC1CNC(C1(C)COC(=O)N1)=O 61193,C(=O)(C#CC(C)(C)CNC(=O)CC1(COC)CC1)NC(CCCC=C)C1CC1 61194,N1(C(C2(CCCC)CC2)=O)CCOCC(NC(=O)Cc2cnc(C)o2)C1 61195,N1(CCNC(C2CCCC23CC3)=O)CCN(C(=O)CN2CCCS2(=O)=O)CC1 61196,c1(C(N(C2CCCN(C(=O)CCc3ncc[nH]3)C2)C)=O)cnc2c(Cl)cccn12 61197,S(=O)(=O)(CCC(=O)NC1CCN(C(=O)Cn2cnc(Br)c2)C1)N(C)C 61198,c1(C(N2CCC(N(CCO)C(C3CCSC3)=O)C2)=O)ccc2c(c1)NS(=O)(=O)C2 61199,N1(C(Cc2c(C)cc(C)s2)=O)CCCC2(CCN(C(C3C(C)C3(F)F)=O)CC2)C1 61200,c1(C(N2CCC(NC(C3(C)CCCNC3=O)=O)C2)=O)cccc2c1OCCCO2 61201,N1(C(=O)CSc2nc[nH]n2)CCCC2(C1)CN(C(c1cnc(O)s1)=O)CCO2 61202,Cc1nc2c(C(=O)NC(C3(CNC(c4sncc4C)=O)CC3)C)cccc2o1 61203,N1(C(c2c(CC)n(-c3ccccc3)nn2)=O)CCC2(CC1)CC(O)(C(F)(F)F)C2 61204,CCC(CC(=O)O)N(C(=O)C(C)CN(C)C)C.C1(C(=O)O)CC(C(F)F)C1 61205,Cc1oc(C)c(C(=O)NCC23CC(CN2C(=O)Cn2cc(F)ccc2=O)C3)c1C 61206,Cc1cc(NC(=O)CCc2ccc(C(=O)NCC3(C)CCC3)[nH]2)ccc1[N+](=O)[O-] 61207,C(C)(CCC(=O)NC(C)(CNC(=O)CSCC(N1CCCCC1)=O)CO)OCC 61208,CCCCC(C)(F)C(=O)NC1CCN(C(c2ccc(COC)o2)=O)CC1CC 61209,C1(CCC(=O)NC(CNC(C2(COC)CCC2)=O)(C)C)C(=O)ON=C1C 61210,c1(C(=O)NCCCCCN(C(C2CN(CC(C)C)C2)=O)C)cc(F)ccc1O 61211,C(=O)(C1COc2ccccc21)NC(c1ccc(N(C)C)cc1)CNC(=O)CO 61212,C(=O)(C1=CCCCC1C)NC1(CNC(C2CCN(CC(C)C)C2)=O)CC(F)(F)C1 61213,C1(CCOC)CN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CCN1C(C12CCOCC1C2)=O 61214,CC(C)CC(CNC=O)CC(=O)NCC(C)N(C)C(c1cccc2nonc12)=O 61215,N1(C(c2c(OC)c(Cl)sc2)=O)CCCC2(NC(C3CN4CCC3CC4)=O)CC2C1 61216,Cc1nc(C2CC2)[nH]c1C(=O)NC(C(C)NC(c1sccc1C)=O)C(C)C 61217,C1(CNC(c2c(CC)cno2)=O)CC2(CC2)CN1C(c1ccc(Cl)c(OC)c1)=O 61218,C1(CC(=O)NCCN(CC(C)O)C(=O)C=Cc2cocn2)(OC)CCCCC1 61219,C12(NC(c3nccc(C)c3F)=O)CCCC1N(C(C1CC13CCCCC3)=O)CC2 61220,C1(NC(CCCOCC=C)=O)CCCCN(C(=O)Cn2cc(C)ccc2=O)CC1 61221,CCCCC(C(=O)NCC1(CC2CC2)CCC1)NC(=O)C1=CC(C)(C)C1 61222,c1(OC)ccc(C(N2CC(NC(C3CC(CN(C)C)C3)=O)CC2C)=O)nc1Cl 61223,Cc1ncc(Cl)cc1C(=O)NC1(CNC(C2(F)CCOC2)=O)CCCC1 61224,N1(C(c2ncc(C)o2)C)CCCC(C(N)=O)(NC(=O)CN2CCCCCC2=O)C1 61225,N1(C(c2c(NC)nccc2)=O)CC(CNC(=O)CC(C)(C)SC)CC(C)(C)C1 61226,Cc1ccnnc1C(N1CCC(Cn2cc(-c3csnc3C)nn2)C1)=O 61227,C(CC(=O)NCC(C)S(N)(=O)=O)(C(F)F)NC(C1N(C(C)=O)CCC1)=O 61228,C(=O)(CC(C(F)(F)F)NC(C1CCCN1C(N)=O)=O)NC1CC(C)OCC1 61229,CCC(C)CCC(=O)NCC1(OCC)CN(C(c2cc(=O)cc[nH]2)=O)C1 61230,N1(C(CCOCCCNC(C2CC(CC)OCC2)=O)=O)CC2(CCC(=O)N2)C1 61231,c1(C(=O)NCC2(COC)CN(C(CCC=C=C)=O)C2)cc(C(F)(F)F)ccc1Cl 61232,c12ccc(nc1)[nH]2.CC(C(=O)SC(F)(F)F)OCCN(C)C.C12(CC1)C(=O)N2 61233,C12(NC(c3nn(C)c(Cl)c3)=O)CCCC(NC(=O)C(=O)NCC(F)(F)F)(C1)C2 61234,C1(NC(C(C)=CC2CC2)=O)C2COCC1CN(C(c1nnc(O)nc1O)=O)C2 61235,N1(C(c2c(C)nc(Cl)cc2)=O)CCOC2(CCN(C(c3ccon3)=O)C2)C1 61236,CC(C)C(CNC(=O)Cc1ccc(F)nc1)C(=O)NC1CCCC(O)C1 61237,CCCCC(=O)C(=O)N(C(C)CCNC(C1(c2cccc(Cl)c2)CCCC1)=O)C 61238,CC1=C(C(=O)N2CCCCC(CNC(C3CCC3)=O)C2)CCC1 61239,C(=O)(C(N)CCCCC#N)N1CCCC(N(C)C)CC1 61240,C1(C(=O)NC2(CO)CN(C(c3c(OC)cc(C)s3)=O)C2)CCc2nnnn2C1 61241,n1(C(CC)C)ccc(=NC(=O)C23CC(CN2C(=O)C(C)(C)C(C)(C)C)C3)[nH]1 61242,Cc1noc(C)c1C(C)NC(=O)C(=O)NCc1cn(C)nc1OC 61243,Cc1conc1C1CN(C(=O)CCCC2CN(C(=O)Cc3cnsc3)C2)C1 61244,C1(CNC(Cc2ccc(C)cc2)=O)CCN(C(c2cc(Cl)ncc2N)=O)CC1C 61245,C1(NC(C2CCN(Cc3c(C)ccs3)CC2)=O)CCC2(CCC(=O)N2)CC1 61246,C1(C(N2CC3C(NC(C4N(C)C(=O)CC4)=O)(CC3)C2)=O)CC(C)(C)SC(C)(C)C1 61247,c1(OC)cc(OC)c(-c2nnc(N3CCCC3CF)n2CC2CCCO2)c(OC)c1 61248,c1(NS(CCC)(=O)=O)cccc(C(=O)NC(CNC(=O)CCSC)CSC)c1 61249,CC1(C)CCN(C(c2cc(C3CC3)no2)=O)C(C(=O)NCC2(C)CC2(C)C)C1 61250,c1(C(=O)NCCOC2CN(C(C(N3CCC(C)C3)=O)=O)C2)c(F)cccc1F 61251,c1(C(N2CCCC(CN(C(=O)C(O)COC)CC)C2)=O)cnc2cc(C)ccn12 61252,C(C(C(=O)NC1CN(C(N)=O)C1)NC(c1cocc1C(N)=O)=O)N(C)C 61253,C1(NC(C=CCN(CC)CC)=O)C=CCC(C(N2CC(N3CCOCC3)C2)=O)C1 61254,N1(C(C(=O)N(CCCNC(=O)NCC)CC)=O)CCOC(CSC)C1 61255,C=CC1(C(=O)NC(c2ccncc2)C)CCN(C(c2cnsc2C)=O)C1 61256,C(=O)(C(CCSC)OCc1ccccc1)NCCN(C(=O)CCC1(C)CC1)CC 61257,N1(C(c2n(CCC)ccc2)=O)CC(NC(=O)Cc2cnn(CC)c2)C(C)C1 61258,c1(C(N(CC(C)NC(c2nocc2Br)=O)C)=O)cccc(Cl)n1 61259,c1(CC)nc(C)n(C)c1C(=O)NC1C2CN(C(c3csnn3)=O)CC12 61260,C(=O)(CCC(=O)c1cccnc1)N1CC(CCCC(=O)O)(OC)C1 61261,c1(NC(C(=O)NCC(c2cn(C)nc2)(C)O)=O)c[nH]c2cccc(Br)c12 61262,C1(O)(CN(C)C(c2cc(Cl)cc(Cl)c2)=O)CCN(C(c2cn(C)nn2)=O)CC1 61263,c1(CC)cc(Cl)ccc1C(=O)NC(CN(C)C(C1CCOC1CC)=O)(CO)CO 61264,Cc1cc(C(N2CCCC3(C(=O)OC(C)(C)C)CC23)=O)cnc1-n1cccn1 61265,C1(C#N)(SCC)CN(C(=O)C=CC2CCCN2C(=O)CC2CCC(C)O2)C1 61266,N1(C(c2c(C)nsc2)=O)CCN(C(=O)C(CO)NC(=O)C(C)C)CC(C)(C)C1 61267,C1(O)(CNC(C(c2ccnn2C)C)=O)CCCN(C(C2CN(S(C)(=O)=O)C2)=O)C1 61268,C#CC1(C(=O)NC(C2CCCOC2)CC)CN(C(=O)CN2CCCC2=O)C1 61269,c1(C(=O)NC(CC)C(=O)Nc2ncc(C(F)(F)F)s2)cccc(CN(C)C)c1 61270,c1(CNC(c2c(NC(C)=O)ccs2)=O)cccc(N2CCCNC2=O)c1 61271,C1(NC(C2SCCS2)=O)COC2(C1)CN(C(c1occc1Br)=O)C2 61272,C(=O)(CC(C)P(C)(C)=O)NCC12N(C(c3c(C)cns3)=O)C(CC1)CC2 61273,c1(C(=O)NC2CCC(CN(C(CC(C)(C)OC)=O)C)CC2)ccc2c[nH]nc2c1 61274,CC1CC2(CCO1)CCN(C(=O)Cc1ccc([N+](=O)[O-])cc1C(=O)O)C2 61275,C1(O)(C(C)CNC(=O)C=CC(F)(F)F)CCN(C(c2cnc(S)n2C2CC2)=O)C1 61276,N1(C(c2c3cc(cc2)N3)=O)CC(=O)N2CCCC2C1.N1(CC)C2CCC1CC(O)C2 61277,CCC(CC)CC(=O)NC1CC(CNC(c2ccc(C)nc2N)=O)C1 61278,C1(C2CCCCC2)(C(=O)NC(CNC(C(COCC)(C)C)=O)C2CCC2)CC1 61279,c1(NCCCOCCNC(CC(C)C2CCCC2)=O)nccc(C(F)(F)F)n1 61280,C1(CCCNC(c2c(C)scc2)=O)CCCCN1C(=O)CCc1ccncc1 61281,C1(CNC(CN2CCC(N(C(CC)=O)CC)C2)=O)CCc2nn[nH]c2C1 61282,c1(C(N2CCC(N(C(CC=CCC)=O)C)C2)=O)cc(Cl)c(C)cn1 61283,c1(C(=O)NC(C2(O)CCN(C(CC=CC)=O)C2)C)cc(F)cc2cc[nH]c12 61284,N1(C(CSC(C)C)=O)CC2CC(NC(=O)C(c3ccnn3C)C)CC(C2)C1 61285,CC(C)C(C(C)NC(c1cn(C)nc1C(F)(F)F)=O)NC(=O)C1=CCCC1 61286,c1(C(N2CC(NC(C(C=CC)O)=O)CC2(C)C)=O)cc(S(=O)(=O)NC)c[nH]1 61287,C1(CN(C)C(C2CC2c2cncs2)=O)CN(C(c2c[nH]c(C(N)=O)c2)=O)CCO1 61288,C(c1ccccc1)=C(C)C(N1CCCC1CC(=O)NCc1[nH]cnc1C)=O 61289,C(CN=c1nc(N2CCC(C)C(C)(C)C2)c2c([nH]1)COC2)NC(=O)OCC 61290,C1(C(=O)OC)CCCC(C(=O)NCC2(NC(=O)C(=C3CCCCC3)F)CC2)C1 61291,c1(C(N2CCC(NC(C(C)NC(COC)=O)=O)C2CO)=O)cc(O)cc(N)c1Cl 61292,C(=O)(C(C)(C)C(F)c1ccccc1)N1CCC(C)(NC(c2c(Cl)cn(C)n2)=O)C1 61293,c1(C(N2CC(C)C(Cc3ccccc3)C2)=O)cnc(O)n(C2CC2)c1=O 61294,c1(C(N(CC(=O)OC)Cc2cn(CCCO)nn2)=O)cc(Br)cc2nc(O)[nH]c12 61295,CCC(O)CCc1cn(C(C)C(=O)N(CCN2CCCC2)CC)nn1.C1(=O)CN1 61296,c1(C(=O)NC(C(C)NC(C(C)NC(COC)=O)=O)CO)ccc(CC2CC2)cc1 61297,CC(c1ccc(F)cc1)=CC(=O)N(CCCNC(c1ccc(CC(C)C)s1)=O)C 61298,N1(C(C(CCC)C)=O)CCN(C(C2(CCF)CC2)=O)C(c2ccncc2)C1 61299,c1(C(N2C(CNC(C#CC3(SCC)CC3)=O)CC2)=O)cc(OC)c(OC)cc1N 61300,C1(C(N(C)CCc2cccnc2)=O)CC(O)CN1C(=O)Cn1cc(Cl)cn1 61301,C1(NC(Cc2c(CC)con2)=O)CCC(NC(=O)COCC(F)(F)F)CC1 61302,c1(OC)nscc1CNC(c1ccoc1CNC(=O)CCCC1CCC1)=O 61303,Cc1ccc(C2CC2)c(C(N2CC(O)(C(C)NC(c3conc3C)=O)C2)=O)c1 61304,N1(C(C2(COC)CC2)=O)CCC2(CCN(C(=O)Cc3ccsc3)CC2)C(C)C1 61305,N1(C(C(C)N=[N+]=[N-])=O)Cc2[nH]nc(C(=O)Nc3cccc(N(C)C)c3)c2C1 61306,CCC(C)(CNCc1nnnn1CC1CCOCC1)CC1CCCC1 61307,CC(C)(CN=c1cc(OC(F)(F)F)cn[nH]1)OCC1CCOC1 61308,C(CC(CNC)OC)NC(CN(CCC)C(C1CCC1C(C)(C)C)=O)=O 61309,C1(C(N2CCC(N(C(c3cnc(S)nc3)=O)CC)C2)=O)NC(=O)OC1(C)C 61310,c1(C(C)(C)C)cc(C(=O)NC2CCC(CCNC(=O)Cn3cnnc3O)C2)on1 61311,N1(C(C(c2cccc(C)c2)=O)=O)CC2CC1CCN2C(c1nncn1C1CC1)=O 61312,C(=O)(C(CC(C)C)OC)N1CC(CCC)C(C(N2CC(CC(=O)OC)C2)=O)C1 61313,c1(C(=O)NCC(CN(C)C(c2c[nH]cc2C(F)(F)F)=O)O)ccc(N)c(O)c1 61314,N1(C(CC(CCC)O)=O)CC2CCC1CN2C(=O)C(C)Cc1cccc(F)c1 61315,N1(C(C2CCC(CC)O2)=O)CCC(C(=O)NOCc2ccc(F)cc2)C(O)C1 61316,N1(C(C(c2ccccc2)NC(N)=O)=O)CC(CNC(=O)CCC=CBr)C(O)C1 61317,N1(C(c2cc(C(F)F)on2)C(=O)NC(C(=O)OC)C)c2ccccc2CC1C 61318,c1(CC)ccc(SC)cc1.C12C(C1(F)F)CC(=O)N(C)CC1(CC1)CNC2=O 61319,c1(-n2cc(CNC(c3cc(-c4ccccc4I)no3)=O)nn2)c(F)cccc1F 61320,CCCCCCC(CC)NC(C1CCCCC1(C)NC(=O)CCCCCSC)=O 61321,CC1(NC(c2n[nH]c3c2COC3)=O)CCC(NC(C2(C)CCCCO2)=O)CC1 61322,C(C(C)(C)CCNC(c1cnsn1)=O)NC(c1cc(C(=O)OC)no1)=O 61323,CC12COCC1CN(Cc1nnc(CC3CC3)o1)C2 61324,CCC(C(=O)NC1(c2cn(C3CCCC3O)nn2)CCCOC1)C(C)(C)CC 61325,C(=O)(C1=NN(C)C(=O)CC1)NC1CCC(NC(c2c(C)c(N)cnc2)=O)C1 61326,n1(CC)cnc2c(N(CCS(C)(=O)=O)C)[nH]c(=NCCC(N)=O)nc12 61327,C1(C(=O)NC(CCOC)CNC(c2ccc(Cl)s2)=O)CC2(C1)NC(=O)NC2=O 61328,c1(OC)cccc(-n2nc(-c3ccco3)nc2CC(=O)N(C)C)c1 61329,C1(NC(CC=CCNC(C2CN(C(C)C)C2)=O)=O)(CO)CC2CCCC12 61330,C1(F)(CNC(C(C2CCCO2)OC)=O)CC(CNC(=O)COCC(F)F)C1 61331,C(C)(CCN=c1[nH]c(=NCC(C)(C)N(C)C)[nH]c2ccc(Cl)cc12)OC 61332,N1(C(c2c(Cl)ccnc2Cl)=O)CCC2C(CCN2C(=O)Cc2cccc(Cl)c2)C1 61333,C1(C)(CNC(C(C)S(C)(=O)=O)=O)CN(C(c2ncc3ccccn23)=O)C(C)(C)C1 61334,N1(C(CC=C=C)=O)CCC(C)(C)C1C(=O)NC1CC2OCCCC12 61335,N1(C(C(C)OC)=O)CC=C(CNC(c2ncccc2Cl)=O)CC1 61336,c1(CNC(C2CCC(CNC(=O)C=CCO)C2)=O)cnccc1Cl 61337,N1(C(C2CC(C)SCC2)=O)C2CCC1CC(CNC(c1cc(O)no1)=O)C2 61338,Cc1cccc(C(=O)N(CCCNC(=O)C(c2cnccn2)C)C2CC2)c1Cl 61339,c1(CC(=O)NC2CC(NC(Cc3c(C)n[nH]c3C)=O)C2)c(F)cccc1Br 61340,C(CC(C)C)(C(=O)N(C)CCOCCCN(C)C(c1ncc(C)cc1F)=O)OC 61341,N1(CCNC(CC2C(C)CCC2)=O)CCN(C(=O)C(C)(C)N(C)CCO)CC1 61342,c1(C(=O)NCCCNC(N(C(C)C)C)=O)cccc(Br)c1 61343,C(=O)(CC(C(C)C)NC(c1cnncc1C)=O)N1CCC(CC)(CC)C1 61344,c1(CCCC)ccc(NC(=O)NC2(C(=O)NC)CC2(C)C)c(C#N)c1 61345,N(C1CCc2cc(CNC(c3csnc3C)=O)ccc21)C(c1cnc(C)[nH]1)=O 61346,c1(C(=O)NC(CNC(c2cnc(OC)s2)=O)C)sc(F)cc1Cl 61347,C1(CC)CC(OCc2ccccc2)CN(C(C)C(=O)OCC(C)CC)C1 61348,N1(C(c2nccc(OC)c2OC)=O)CCC(NC(C2CCC2)=O)C(C)(C)C1 61349,N1(C(c2cnn(CC)c2Cl)=O)CCN(C(=O)CCc2ccoc2)CC1CO 61350,c1(C(N(CC(C)NC(C(C2CCOCC2)OCC)=O)C)=O)[nH]cnc1C#N 61351,N1(C(c2c(C)nsc2C)=O)C2CCC1C(C)C(NC(C1CC(C)(C)CN1C)=O)C2 61352,N1(C(c2n(C)c(Cl)nc2)C(=O)NC2CC2)CCN(Cc2ccccc2Cl)C(=O)C1 61353,C1(N(C(c2nnc(C)n2C)COC)C(C2CCC(OC)C2)=O)CC2CCC1C2 61354,c1(NC(=O)C(N2CCN(C3CCOC34CCOC4)CC2)=O)c[nH]c2cccnc12 61355,c1(C(C(=O)N2CCC2c2cccnc2)NC(C)=O)cccc([N+](=O)[O-])c1 61356,N1(C(C(CC#C)CC#C)=O)CC2CCCC(C1)N2C(=O)CC1(C(F)F)CC1 61357,Cc1cc(=NC(=O)N2CC(C)CC3(CC3)C2)[nH]n1Cc1ccc(Cl)cc1 61358,C1(OC(C)C(N2CC(O)(CCNC(C3(C#N)CCC3)=O)C2)=O)CCOCC1 61359,CC(C)CC(C)C(=O)N(C1CCCN(C(=O)COC2CCCCC2)C1)CCF 61360,C1(NC(c2nn(CC)nc2C)=O)CCN(C(=O)CCc2cscn2)C12CCC2 61361,n1(CCC(=O)NCC(CNC(C2(Cl)CC2(C)C)=O)OC)cc(C)cn1 61362,c1(C(N2C(CC(=O)N(CC(C(=O)OC)C)C)CC2)=O)cc(C)n(C)n1 61363,c1(C(N2CC3CCN(C(CC(C)SC)=O)C3C2)=O)ccnc2ncccc12 61364,C1(NC(c2ccc(CCF)cc2)=O)CCC2CN(C(C3CCCO3)=O)CC2C1 61365,c1(OC)cc(C(N2CCCC2C=CC(=O)NCC2CC2(C)C)=O)ncn1 61366,C(N=c1[nH]nc(CC)s1)C1C2CN(C(C3(CCCC)CC3)=O)CC21 61367,CCC(CCC(=O)Nc1ccc(C(C)C)nc1)NC(=O)C(C)c1cccs1 61368,C1(C(=O)N(C)CCN(C)C(C2CC=CCC2)=O)(NC(C)=O)CCC(C)CC1 61369,c1(C(=O)NC23CC(NC(C4CCC(CC)O4)=O)(C2)C3)n[nH]c2c1CN(C)CC2 61370,CCCC(C)(O)C(=O)N1CCOCC(NC(=O)C(C(C)C)c2ccccc2)C1 61371,C1(NC(C=CC)=O)CC2CCC1N(C(c1cnn(CC(F)F)n1)=O)C2 61372,CC(C)C(CC(=O)NC1(C)CCN(C(c2cc(C#N)on2)=O)C1)c1ccccc1 61373,c1(C(N2CC(C)C(NC(=O)C=CCN(C)C)CC2)=O)ccc2c(c1)C(=O)NCC2 61374,C1(C(N2CC(O)(CNC(C=C(c3ccn(C)n3)F)=O)C2)=O)CCc2ccnn2C1 61375,C1(CC#C)(C(=O)NCCN(C(C23CCC2C3)=O)C(C)C)CCOC1 61376,C1(CCNC(C(CO)OC)=O)CCN(C(C2C3COCC23)=O)CC1(F)F 61377,CC1CC(C(=O)NCCN2CCN(CC(F)(F)F)CC2)CCS1 61378,C1(C(N(CC(=O)O)Cc2cn(C3C(C)(O)CCC3)nn2)=O)CC2(CC(=O)C2)C1 61379,C(C(C)(C)C(=O)NC1CCC(CCNC(c2cc(Br)oc2C)=O)C1)OC 61380,N1(C(C(C)SC(C)C)=O)CCC2CN(C(c3ccnc4c3ccn4C)=O)CCC12 61381,Cc1cc(NC(C2(C)CN(C(=O)CCC3CC(C)C3)CC2C)=O)cnc1F 61382,c1(C(=O)NC2C(C(=O)NCC(c3cccc(O)c3)O)CCC2)cccc(F)c1F 61383,C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CN(C(=O)C=Cc1ccccc1Cl)C)(C)C 61384,C(=O)(C1CN(C(=O)CN2c3ccccc3CS2(=O)=O)c2c(C)cccc21)OC 61385,N(C(=NCC1CC1(F)F)NCC1CCCO1)C1CC(OCC(=O)NC(C)=O)C1 61386,N1(C(=O)NCCCCC(OC)OC(=O)NCCN=[N+]=[N-])CC2(C1)OC(=O)NC2C 61387,C1(NC(C(CC)=CCCC)=O)CC(CNC(c2sccc2C(=O)NC)=O)C(O)C1 61388,N1(C(c2nncc(OC)c2)=O)CC(O)CCC1C(=O)NCC1(Cl)CC1(F)F 61389,Cc1oc(C(N2CCCCC2CNC(c2ccc(C(F)(F)F)[nH]2)=O)=O)cc1Br 61390,Cc1cnc(C(N2CC3CC2C3NC(=O)CCc2cc(Cl)cs2)=O)nc1 61391,N1(C(C(F)=CCC)=O)CCN(C(C2CCCCC2(C)C)=O)CC1CS(C)(=O)=O 61392,c1(SCC(=O)NC(CC)(C)CNC(=O)Cn2nnc(C3CC3)n2)ccnc(Cl)c1 61393,C(=O)(C1=C(Cl)CCC(C)C1)NCC(CCCC)NC(c1ccc(Cl)o1)=O 61394,c1(CNC(c2c(C)coc2C)=O)cc(O)nc(CNC(=O)CC(O)C(C)C)n1 61395,c1(OC)ccc(-c2ccc(N)cc2CNC)cc1COC1CC(C)C1 61396,C(C(F)(F)C(=O)NCC1(NC(=O)C(n2cc(C)cn2)C)CCCCC1)OC 61397,CC(C)CC(CNC(=O)C(C)C(F)(F)F)C(=O)Nc1ccc2nc[nH]c2c1 61398,CCC(C)(C(=O)NCC1(F)CCN(C(C2(C)COCCO2)=O)CC1)C(F)F 61399,c1(OC)cc[n+]([O-])c(C(=O)NCC(O)CCNC(=O)C2=NNC(=O)C2)c1 61400,N1(C(c2c(C)ccc(C(F)(F)F)c2)=O)CC(NC(=O)CC(F)(F)F)CCC1(C)C 61401,C(=O)(CC1=Cc2ccccc2C1)N1CC(CCC)N(C(C2CCNC2=O)=O)CC1 61402,C=C(C)CCCC(=O)N(C(CNC(c1ccc(OCCC)c(N)c1)=O)C1CC1)C 61403,C#Cc1ccc(C(N2CC(C3(NC(=O)C(CC4CCCC4)CC)CC3)C2)=O)cn1 61404,N1(C(C2=C(C)OCCS2)=O)CC(NC(=O)C(C)c2cncs2)CC2(CCC2)C1 61405,Cc1cn2cc(C(=O)NCCC3(O)CN(C(C4(O)CCOCC4)=O)C3)sc2n1 61406,N1(C(=O)NC(c2cnccn2)C2CC2)CC2CCC(CO)(C2)C1 61407,N1(C(C(C=C)O)=O)CCC(CC)(NC(=O)CC(C(N)=O)NC(C)=O)CC1 61408,N1(C(C2C(C(C)C)C2)=O)CCC2CN(C(c3cn(CC4CCOC4)nn3)=O)C2C1 61409,C#Cc1nc(C(N2CCN(CCNC(C3SCCC3C)=O)CC2)=O)cs1 61410,C(=O)(C1=CCC(C)(C)CC1)NCC1CCN(C(COC(CC)C)=O)C1(C)C 61411,C1(NC(C(C(C)C)C#N)=O)CN(C(=O)CC2CC3(CCC3)C2)CC2(CCC2)C1 61412,c1(OC)ncc(OC)c(=NCC2CCN2)[nH]1 61413,C(C)(C(O)C(=O)NC(C1CCN(C(c2ccc(CSC)cc2)=O)CC1)(C)C)SC 61414,C(CCCCCN(C(=O)C=CCOCCOC)C)NC(c1c(CC)cco1)=O 61415,C(=O)(C(Cc1ccccc1)NC(C)COc1ccccc1)NC 61416,C1(CNC(c2c(COC)cco2)=O)CC2CCC1N2C(c1cc(OC)ns1)=O 61417,N1(C(CCNC(=O)NC)=O)CCN(CCNC(C2CC2CF)=O)CC1 61418,N1(C(C(C)SC(C)C)=O)CCC(C(O)CNC(=O)C(C)n2cncn2)CC1 61419,c1(C(N2CC3N(C(C(=O)NC(C)C)=O)C(CC3)C2)=O)cnc2ccc(F)cc2c1 61420,CC(C)CC(O)C(=O)NCC(Cc1ccccc1)N(C)C(C1CC1F)=O 61421,C1(C(N2CCC(O)C2)=O)CC2CC2N1Cc1ccccc1COc1ccccc1 61422,N1(C(C(CO)N(C)C)=O)CCCCC1CNC(c1ccc(-c2ccncc2)s1)=O 61423,c1(OC)ccnc(F)c1C(=O)NCC12CC(CN1C(=O)C(C)OC)C2 61424,C1(n2cc(CCNC(C)=O)nn2)CCCN(C(c2csc(C(F)(F)F)c2)=O)C1 61425,c1(C(=O)NCC2CN(C(c3c(Cl)nc(OC)s3)=O)CC2C)cc2ncccn2n1 61426,Cc1ccc(C(N2CCCC(NC(C3(C4CCCO4)CC3)=O)C2)=O)c(F)c1C 61427,c1(C(=O)NC2CN(C(CCc3ccnc(C)n3)=O)CC2C)ccc(=N)[nH]c1Cl 61428,Cc1cc2c(C(=O)NCCCCCCN(C)C(C3CCCC3O)=O)cccc2o1 61429,C(CN=c1[nH]c(=NCCN2CC3CCCC3C2)[nH]c2c1COC2)n1c(=O)cccc1 61430,CCC(C)(C)C(=O)N1CCC(C(=O)NCCN=[N+]=[N-])O1 61431,C#CCCC(O)C(=O)N1CCCC1CN(C(=O)CCC(=O)NC1CCCC1)C 61432,CC(C)C(C(=O)NCC1CCCS1)n1cc(CCCNS(N)(=O)=O)nn1 61433,Cc1ccc(C(=O)NCC(C)(C)C(N2CCCC(CO)C2C)=O)cc1C 61434,C1(C(N(CCNC(=O)Cn2nnc(=O)[nH]2)CC)=O)CC2CCC1NC2=O 61435,Cc1nc(CC(N2CC(OCCNC(c3cc(CO)[nH]n3)=O)C2)=O)co1 61436,CCC(C)(C(=O)NCC1CC(NC(C2CC2c2cccnc2)=O)C1)C(F)F 61437,CC(C)CC(F)(F)C(=O)NC1CCCCC1CNC(=O)CCC1CCCCN1C 61438,n1(CCC)nnnc1C(c1nc(C)cs1)NC(c1nnc(C)s1)C 61439,c1(C(=O)NC2CCCC(NC(C(COC)(F)F)=O)C2)cccc2c1NC(=O)CC2 61440,C1(NC(c2ccc(CC)[nH]2)=O)CCSC12CN(C(C1(C)CC1(Cl)Cl)=O)C2 61441,c1(C(=O)NC(C(C)(C)NC(C(COCC)C)=O)C)cc(C)n(C(C)C)n1 61442,Cc1c(C(=O)NCC(C)CN(C(=O)C=C2CCC(C)C2)C)ncn1C 61443,C(=O)(CCC(=O)NC1CCCCC1CNC(=O)CN1CSCC1=O)NC 61444,C1(C(=O)NCCCCCCC)CC2(CCN1C(C1CN(C(C)=O)C1)=O)CC2 61445,c1(CC)ncncc1C(=O)NC1CN(C(=O)Cc2ccc(Cl)s2)CC1O 61446,Cc1nc(C)c(S(=O)(=O)NC(CS(C)(=O)=O)c2ccccc2)o1 61447,C1(C(=O)Nc2ccc(C#C)nc2)CCN(C(=O)CC(CN(C)C)CC)C(C)(C)C1 61448,N1(C(c2cc3sccc3[nH]2)=O)CC2CCN(C(=O)CC34CCC(CC3)C4)C2C1 61449,c1(C(=O)NC(C)CN(C)C(c2n[nH]c(C3CC3)n2)=O)cc(Cl)c(Cl)cc1N 61450,C1(CC)CCCC(NC(=O)CC(C)NC(c2cn(C(C)C)nn2)=O)C1 61451,C(CCCCCNC(=O)C(F)n1ccnc1)NC(=O)CCCn1ccnc1 61452,C12(CNC(CC(C)NC(C3C(C(=O)OC)CC3)=O)=O)CCCC(CO1)C2 61453,Cc1nc(C#N)c(NNC(=O)N2CCSC3CCC23)o1 61454,C1(CC(=O)NC2CC(OCC(=O)NC(CO)C3CC3)C2)CCC(=O)N1 61455,c1(C(N(CC)CC2CCCN2C(C2CCC2)=O)=O)ccc2cccc(F)c2n1 61456,N1(C(CC(=O)N(C)C)=O)CC2(CCCC(CNC(c3n[nH]c4c3CCC4)=O)O2)C1 61457,CC(C(=O)N1CC=CC1CNC(c1ccc(Cn2ccnn2)o1)=O)C(C)(C)C 61458,c1(C(=O)NCCC(C)CCNC(C2CCCOC2C)=O)ccc2c(c1)C(=O)NC2 61459,Cc1ncc(C(=O)NC(C2(CNC(=O)CCN3CCCCC3C)CC2)C)c(=N)[nH]1 61460,CCC(CC)CCC(=O)N1CC2CC1CC2NC(c1sc(C)nc1C)=O 61461,N1(C(=O)CCN(CCO)CCO)CC=CC1Cn1cc(C(C2CC2)N(C)C)nn1 61462,c1(OC(C)C)nc(C(=O)NCC2CCN2C(c2cncc(C#N)c2)=O)cc(O)n1 61463,C(=O)(C1=C(Cl)CCOC1)N1CCC(N(C(=O)CSCc2ccccc2)C)CC1 61464,C1(NC(C2C(C)C2)=O)CCN(C(c2ccccc2Sc2ccccc2)=O)CC1F 61465,N1(C(c2cnc(C)[nH]2)=O)CC(NC(c2cc(C(C)(C)C)nn2C)=O)C(C)C1 61466,C(=O)(N1CC(O)CCO1)c1cc(CNC(C(=CC2CCCC2)C)=O)nn1C 61467,N1(C=O)CCN(C(c2cnc(C)[nH]2)=O)CC1C.c1(NC(=O)NC)cccc(C)c1 61468,C1(C(=O)NCc2cscn2)CC12CCN(C(c1cnc(Cl)cc1Cl)=O)C2 61469,C1(NC(CC(C)OCc2ccccc2)=O)CN(C(=O)C(Cl)=CCl)CCC1(C)C 61470,N1(C(C2(CC(C)C)CCC2)=O)CC2CC1CN2C(=O)CCC(C)N(C)C 61471,C(CCC(CC)CC)NC(=NCC=C)NCC(C)(C)C(=O)OC 61472,N(C(=NCC(F)(F)COCC)NC(C)C)C1CCCC(OCC)C1 61473,C1(N(C(C=CC)=O)C)CCCN(C(=O)NC2CC2c2ccncc2F)C1 61474,c1(C(=O)NCC2CCN(C(c3c(OC)scc3)=O)CC2C)cnc2ccoc2c1 61475,N1(C(C)C)CCC(CC(=O)N(CCNC(=O)CC2CCCCC2F)C2CC2)CC1 61476,c1(C2(C)CC2)ccccc1NC(=O)C=CCNC(=O)CC1COCCOC1 61477,N1(C(=O)Cc2cc(C3CC3)on2)CC2CN(C(C3(F)CCC3)=O)CCC12 61478,c1(C(N2CCC(NC(CN(c3ccncc3)C)=O)C2)=O)ccnc(Cl)c1O 61479,c1(C(N2CCC(Cn3cc(CN)nn3)C2)=O)c[nH]c2c(C)c(Cl)ccc2c1=O 61480,c1(C(N(C(C)CNC(=O)CSCC(F)(F)F)C)=O)csc(C(F)(F)F)n1 61481,C1(C(N2CCC(NC(c3c(C(C)(C)C)con3)=O)C2)=O)CC2(C1)CC(F)C2 61482,C(c1cnn(C)c1C)=CC(=O)NCCN(CCC)C(c1cc(OC)ccc1Cl)=O 61483,n1(CC(=O)NCCC2=CCN(C(=O)C=C(Cl)Cl)CC2)nc2n(c1=O)CCCC2 61484,CC1CCCCCN1C(c1c[nH]nc1CCNC(C1COCC1(C)C)=O)=O 61485,C=CCC(C(=O)OCC)NC(=O)CC1C=CC(NC(=O)C(C)C=C)C1 61486,c1(C(=O)NC(C2CN(C(CCNC(C)=O)=O)C2)C)ccnc(S)c1 61487,C1(CC)CN(C(=O)CCOCCOC)CC1NC(c1sccc1-n1cnnn1)=O 61488,CCC(C(=O)NC1(C)CCCN(C(c2ccn(C)c2C2CC2)=O)C1)C(C)(C)CC 61489,N1(C(CCCC(N)=O)=O)C2CCCC1CN(C(=O)CCOC1CC1)CC2 61490,Cc1cc(CNC(N2CCC(C)CC2C(C)O)=O)cnc1C 61491,C(=O)(C(C)(O)CC(C)C)N1CC(N(C(c2[nH]cc(C)c2)=O)C)C(C)(C)C1 61492,N1(C(CC2CCC(NC(=O)C(c3ccccc3)O)C2)=O)CCCCCC1CCO 61493,c1(C(N(CCN(C(=O)Cn2cnnc2O)C(C)C)C)=O)ccc(C(F)(F)F)cc1 61494,C1(C2CCOCC2)(C(N2C(CNC(C=C(CC)CC)=O)CC2)=O)CC1 61495,n1(CC(=O)N(C(C)C(=O)NC(CC)C(C)O)CCC)ccc(C)n1 61496,Cc1nsc(C)c1NC(C1(NC(=O)CC(=O)N(C)C)CC(F)C1)=O 61497,N1(C(C2CC(C)(F)C2)=O)CCC2C(C1)NC(=O)CN2C(c1ccc(O)c(Cl)n1)=O 61498,c1(C(=O)NCC=CCNC(c2c(C)nco2)=O)cnc(S)nc1 61499,C1(CC(N2CC(NC(C(C3CC3)OCC)=O)C(C)C2)=O)C(=O)N(C)N=C1C 61500,C1(C(=O)NC(CCNC(c2c(CC=C)cccc2)=O)(C)C)CS(=O)(=O)CCO1 61501,N1(C(CC2(COC)CC2)=O)C(C)CN(C(=O)C#CC(C)(C)O)CC1C 61502,CC1(CNC(=O)C=Cc2ccccc2)CCC(NC(=O)CNC(=O)C(C)(C)C)CC1 61503,N1(C(c2c(NCC)ccc(Cl)c2)=O)CCC(C)(C)C(NC(=O)CCC2CC2C)C1 61504,N1(C(CCC)=O)CC2CCC(NC(=O)CCC(C)c3ccccc3)CC2C1 61505,C1(NC(C2CCCN(C(C)C)C2)=O)CCN(C(C2(C)CC2)=O)CCC1CO 61506,N1(C(Cc2c(C)ccs2)=O)CCC(NC(C2CCOC2C)=O)C(F)C1 61507,c1(C(=O)NC2CN(C(CCCC)=O)CC(O)C2)ccc2c(c1)nc(C)n2C1CC1 61508,C(=O)C1CCCc2nc[nH]c21.Cc1c(NC)cnn1-c1cc(-n2cccn2)ncn1 61509,N1(C(C(CC)(F)F)=O)CCC12CN(C(=O)CCC(C)c1ccccc1)C2 61510,CC(C)(C)CCCCNC(C1C(CNC(=O)CCc2ccccn2)C1(C)C)=O 61511,C(=O)(C(O)P(C)(C)=O)N1CC(c2cn(C)nn2)C1.C1(COC)CCCC1 61512,Cc1c(C(N2CC(CNC(=O)C(F)C3CCC3)C(F)(F)C2)=O)[nH]ccc1=O 61513,c1(CS(=O)(=O)NC(C2CCC3(CCNCC3)O2)=O)ccc2ccccc2c1Br 61514,c1(C(=O)NCC(CNC(C(C=C=C)C)=O)(C)O)c(F)cc(Br)c(F)c1F 61515,NS(=O)(=O)C1(C(=O)NCCN(C2CCCCC2)C(C2CC(F)(F)CS2)=O)CC1 61516,C(=O)(C(F)C(C)(C)O)NCC(c1ccc(F)cc1)NC(CC1(C=C)CC1)=O 61517,CC(CCCCNC(C1CCC(=O)N1C)=O)NC(c1ccn(CCF)n1)=O 61518,c1(C(N2CCOC(c3ccco3)C2)C(=O)NCC=C)ccc2cc(Br)ccc2c1 61519,C(=O)(C(C1CCCO1)NC(=O)CCOCC(N1CC(OC2CC2)C1)=O)NC 61520,Cc1cccn(CC(=O)NC2CC(F)CN(C(=O)Cc3ccc(Cl)nc3)C2)c1=O 61521,N1(C(=O)C(C2CC2)NC(C23CSCC2C3)=O)CC2(CCOC2)C1 61522,C(=O)(CCCCC(=O)NCCC1(O)CCN(C(=O)CCCc2nccs2)C1)NC 61523,C12(C(N(CCOCCN(C(CC(C(C)C)O)=O)C)C)=O)CCCC(C)(C1)OC2 61524,Cc1cc(=NCCCCC#N)[nH]cc1S(=O)(=O)N1CCC(C)C1C 61525,c1(NC(c2n(CCCSCC)nnn2)(C)CC2CCC2)ccc2cnn(C)c2c1 61526,c1(C(N2CCC(CNC(C3(CCC=C)CC3)=O)C2)=O)nc(C)ccc1C 61527,CC1(C)COC(CCNc2ccc(C3(C)CC3(F)F)cc2)CO1 61528,c1(COC)nc(C(=O)NCC(C2CCCC2)NC(C2CC23CCC3)=O)cs1 61529,N1(C(CSCCOC)=O)CCC(C(C)(C)C(=O)NCCC(=O)NC(C)C)C1 61530,N1(C(C2C(C=C)CC2)=O)CCc2nc(CNC(C3(C)CC(C)=NO3)=O)sc2C1 61531,C(=O)(C(C)(C)CS(C)(=O)=O)N(CCNC(c1c(C)ncn1O)=O)C 61532,N1(C(C(CCC)OCC)=O)CCC(C2CC2)C1C(=O)NC1CCCC1CN(C)C 61533,C1(CN(CCC)C(c2cccc(-c3nn[nH]n3)c2)C)CC2CCC1O2 61534,C1(NC(=O)Cc2cc3sccc3[nH]2)CC2CN(C(=O)C3CC3)CCN2C1=O 61535,C1(CC(N2CC(C(N)=O)(CNC(CC(C)(C)SC)=O)C2)=O)COC(C)(C)CO1 61536,N1(C(C)=O)CCC(C)(NC(=O)C(N2CCN(C3CC4CCC3C4)CC2)=O)CC1 61537,N1(C(Cc2c(C)scc2)=O)CCOCC1CCNC(C12CC(C(F)F)(CO1)C2)=O 61538,C1(CNC(c2cnn(CC)n2)=O)CC(C)N(C(=O)CCCN(C)C(C)=O)C1 61539,C1(C2CCCO2)(C(=O)NCC2(CNC(c3nsnc3O)=O)CC2)CCCC1 61540,c1(CNC(=O)C(c2ccccc2)Nc2ccccc2)ccc(S(F)(F)(F)(F)F)cc1 61541,N1(C(C(CC)(CC)CO)=O)CCC2(CCC2NC(c2cnc[nH]2)=O)CC1 61542,c1(CN(C(=O)CCn2cc(-c3cccc(NC)c3)nn2)C)cccc([N+](=O)[O-])c1 61543,C12(C(=O)NOCC(F)F)CCC(CC1)N(C(c1cccc3[nH]ncc13)=O)C2 61544,C1(C(C)NC(COCC=C)=O)CCCN1C(c1csc(C(F)(F)F)n1)=O 61545,C(=O)(C(C)(C)S(C)(=O)=O)NC1C(c2n(C)ncc2)CN(C(C2CCOC2)=O)C1 61546,CC(C)(C)C(O)C(=O)NC1CC(F)CN(C(c2ccc(-n3cccc3)cc2)=O)C1 61547,C(=O)(C1=CCCC1C)NC(C1(C(N(C)Cc2cn(CC)nn2)=O)CC1)C 61548,c1(C(=O)NCc2cnc(CC)[nH]2)cc(Cl)cc(Cl)c1F 61549,C(=O)(CCCCN(C(=O)C(C1CC1)OC)C)NC(c1cccnc1)CC 61550,N1(C(c2cc(CC)ncn2)=O)CCCN(C(=O)C=CCF)C(C(C)C)C1 61551,Cc1cc(F)c(N)cc1C(=O)NCC(CC(C)C)NC(=O)CC=C(Cl)Cl 61552,N1(C(C(CC#C)NC(C)=O)=O)CCC(C2CC2)C1 61553,c1(OC)cccc(F)c1CNC(C1CCN1C(c1ccc(Br)s1)=O)=O 61554,c1(OC)ccccc1CSCCNc1ncnc(CN)n1 61555,N(C1c2ccccc2OCC1F)C(N(c1ccc(S(N)(=O)=O)cc1)C1CC1)=O 61556,C#CCCCC(=O)NCCCC(C)NC(=O)C(O)Cc1[nH]cnc1C 61557,N1(C(c2ccc(CC)c(N)c2)=O)CC2CCN(C(c3ccc(CO)nc3)=O)CC12 61558,N1(C(CC(C)O)=O)CC2(CCCC2)C1C(N(C)C[Si](C)(C)C)=O 61559,C(N=c1nc(N2CCC(CCO)C2)cc(C)[nH]1)C1(CCC=C)CCCC1 61560,C1(CNC(c2c(C)n[nH]c2C)=O)CC2(CC2)CN1C(=O)C=CCF 61561,CCCCCC(F)C(=O)N1CCC=CC1C(=O)N(CC1CCCCC1)OC 61562,C1(NC(c2cccc(CC)c2)=O)CS(=O)(=O)CC1NC(=O)C(C)=C1CC1 61563,C12(C(=O)OCC)CNCC1(C(=O)NC(C)C(N)=O)C2 61564,c1(C(C)C)c(N2CCC(CNC(=O)C(=O)Nc3ccc(Cl)cc3)C2)ncnc1Cl 61565,c1(C(=O)NC2CN(C(c3cn(CC)nn3)=O)C3C2C3)cc2occc2n1C 61566,C1(Nc2nc(C)nc(C#N)c2)CCC2(CC1)CN(C(C1CC1(C)Br)=O)CCO2 61567,c1(C(N(CC(O)CN(C)C(c2cc(O)ncn2)=O)C)=O)cc2c(=O)cc[nH]c2s1 61568,n1(CC(N2CCC(CN(C)C(C3CCOC3)=O)C2)=O)cc(Br)c(O)nc1=O 61569,C1(c2n(C(c3ccccc3)C)nnn2)(OCNc2ncc(CO)s2)CCC(=O)NC1 61570,C(=O)(C1=NOC2(CCC2)C1)N1C(CN(C(=O)C(CO)N(C)C)C)CCC1 61571,C(=O)(CCCCC(N)=O)NC(C1CCCN1C(c1cc(CN(C)C)on1)=O)C 61572,N1(C(C(CCO)N(C)C)=O)CCC(NC(C2CN3CCN2CC3)=O)C(O)C1 61573,N1(C(C(C)O)=O)CCN(C(=O)CCc2n[nH]c(=N)s2)C(C(F)F)C1 61574,CC(C)CC(C)(O)C(=O)NC(CNC(c1ccccc1SC(F)(F)F)=O)C(C)C 61575,C1(C(C)NC(COC(C)C)=O)CCN(C(=O)Cc2cnn(C)c2)CC1 61576,C(C)(CNC(=O)Cc1ccc(C)cn1)(CC(C)C)NC(C(C)OCC=C)=O 61577,Cc1c(C(=O)NC2(C)CN(C(=O)CC3CC4CCC3C4)C2)cncc1Cl 61578,C12(OC)CCC(C(=O)NC3CCN(C(C4CC45CCCC5)=O)C3)(CC1)C2 61579,C(C(C)(C)CNC(c1ccc(F)s1)=O)N(C(=O)C(C)(C)c1ccnn1C)C 61580,C1(NC(CCc2c(OC)cccc2)=O)CCN(C(=O)Cc2ncoc2C)C12CC2 61581,C=CCC(CNC(=O)CCCF)C(=O)N(C)CCn1cccn1 61582,Cc1cc(C(=O)NC2CN(C(c3cccc4c3OCO4)=O)C2)c2c(C)noc2n1 61583,N1(C(CC(C)C2CC2)=O)CCCCC1CCC(C)(C)NC(=O)CC1(O)CCC1 61584,N1(C(C2(C)CCN(C)C2=O)=O)CC2CCC1C(CNC(=O)C=Cc1ccoc1)C2 61585,c1(C(=O)NCC2C3CN(C(CCC)=O)C2C3)cc(Cl)c(Cl)c(Cl)c1 61586,C(CN=C(NCC(F)(F)C1CCCC1)N1CCC(F)(c2ccc(F)cc2)C1)OC 61587,c1(C(NOCC(=O)NCC2(CC3CC3)CC2)=O)ccncc1F 61588,C(c1nc(C)c(C)[nH]1)=CC(=O)NC(C(C(C)C)NC(C=CCCC)=O)C 61589,N1(C(CCC)=O)CCCN(C(c2cccc(N3CC=CC3)c2)=O)CC1CO 61590,n1(C2CC(C(N(CC=C)C)=O)C2)cc(-c2ncoc2C)nn1 61591,c1(C(N2CC(CCNC(CCC(=C)Cl)=O)(OC)C2)=O)coc2ccc(Cl)cc12 61592,N1(C(c2nc(OC)c(Br)cc2)=O)CC2CN(C(=O)C(O)C3CC3)CC2C1 61593,C(=O)(C(O)CC(F)(F)F)NC1CC(C(=O)NC(C2CCCCC2)C#C)C1(C)C 61594,C(C1=CCCN(C(C2CCCCC2O)=O)C1)NC(=O)Cc1ccnc(O)c1 61595,n1(CC(C)C)nccc1NC(=O)C(=O)NCCc1ccncc1 61596,n1(CC(=O)NC(CNC(C(C)Oc2ccc(C)cc2)=O)C)c([N+](=O)[O-])cnc1C 61597,C1(CNC(C(CO)N(C)C)=O)CC2(CC2)CN1C(=O)Cc1cccc(C(F)F)c1 61598,C1(C(=O)NC2CC(CNC(c3cnn(CCF)c3)=O)C2)C2CC3C(C2)C13 61599,c1(SC)ccc([N+](=O)[O-])[nH]1.C12CCN(C1)C(=O)C1CCCN1N(C(C)C)C2=O 61600,c1(C(N2C(C(=O)NCc3cc(C)nn3C)COCC2)=O)ccc(Br)c2nsnc12 61601,c1(CCCC)ccc(C(=O)NC(C)C(C#N)CC)cc1CCCC 61602,c1(C(=O)NCC(CNC(C2(CC#C)CCOC2)=O)O)cc(O)cc(F)c1F 61603,c1(C(N2CC(NC(c3ncc(C)cn3)=O)C(C)CC2)=O)cccc2scnc12 61604,C1(CC)CN(C(=O)CC2COCC2(C)C)CCC1NC(C1CSC1)=O 61605,Cc1nc2c(NCC3CC(CNC(=O)Cn4ccnn4)CO3)ncnc2s1 61606,Cc1c(C(N2CC(CNC(c3c(F)ccc(F)c3O)=O)C2)=O)nn2c1OCCC2 61607,C(=O)(CCCC(C)(C)CC)NC1CN(C(c2c(CC)noc2)=O)CC1C(F)(F)F 61608,c1(OC)cc(F)c(CNC2CC2C(=O)Nc2cc(Br)c(F)cc2Br)cc1F 61609,N1(C(C2CCCOC2)CC)CCC(O)C(F)(F)C1 61610,c1(C(=O)NC2(C(=O)NC(C#C)C)CSC2)cc(C)nnc1C 61611,C1(CNC(c2n(C(C)C)ncc2)=O)CN(C(=O)C2=CCCC2)CCC1C 61612,n1(CC(=O)NCC(C2CCC2)NC(C(CC=C)(F)F)=O)cc([N+](=O)[O-])nc1C 61613,Cc1nnccc1C(N1CC2CC1(C(=O)NCCn1ccnn1)C2)=O 61614,c1(CC)cc(C(=O)NC(C)CC(C)NC(C2CCC(=O)N(C)C2)=O)ccc1O 61615,c1(C(=O)NC2C(CNC(c3cncc(C)c3Cl)=O)CC2)noc2c1CCCC2 61616,N(C(=NCCF)NCC(CC)C(=O)OC)C(c1cccc(Br)c1)C#C 61617,C1(C(N2CC(C#N)C2)=O)CC(F)(F)CN1C(c1cccc(O)n1)=O 61618,c1(CN(C)C(C2C=CCCC2)=O)cnn2c1CN(C(c1cc(CF)on1)=O)CC2 61619,c1(C(=O)NC2CCCN(C(c3c(C)cccc3O)=O)CC2)ccc2ccsc2c1 61620,CC(C)C(C)CC(=O)NC1CCCC(NC(c2ccoc2C2CC2)=O)C1 61621,c1(OC)cccc(C(N2CCN(C(=O)Cc3cccc(C)c3)C3CC23)=O)c1C 61622,C1(NC(c2ccnc(Br)c2F)=O)COC2(CCC2)C1 61623,c1(OC)ccc2[nH]cc(-c3ccc(Nc4nc(C5CC5)ncc4Cl)nc3)c2c1 61624,c1(N2C(C)C(NC(=O)C(C)(C)F)CC2)nc(Cl)nc2ccc(Cl)nc12 61625,CON=Cc1ccc(C(=O)N(CCC(C)NC(C2(C(F)F)CC2)=O)C)cc1 61626,C#CCC(CC#C)C(=O)N1CCC2(C1)CN(C(C1CC(O)(C#C)C1)=O)C2 61627,N1(C(C(C=C)(F)F)=O)CCC2(CC1)OC1(CO)CC2(NC(c2cncn2C)=O)C1 61628,c1(C2(C(N(CC(CNC(Cn3ccc(C)n3)=O)O)C)=O)CC2)ccccc1Cl 61629,C(=O)(C1=NOC(CNC(c2cc(CO)c(C)o2)=O)C1)N(C1CCC(=O)NC1)CC 61630,c1(OC)cnnc(C(N2CC(CCCCNC(C3(O)CCSC3)=O)C2)=O)c1 61631,CC1CN(C(=O)CSc2cnn(C)c2)CCC1CNC(=O)CN1CCNC(=O)C1 61632,C(C)(C)(CC(=O)NC(C)C(C)CC)N(C(C1C(=C)C1C(=O)OC)=O)C 61633,N1(C(C(c2ccccn2)OC(=O)CC(C)O)=O)CC(OCC)C(C)(C)C1.C=CC 61634,c1(OCC)ccccc1C(=O)NC(CNC(C1CCCO1)=O)C(C)C 61635,Cc1nnc2c(C(N3CC(C)(NC(=O)Cc4cc(C(C)C)no4)C3)=O)cccn12 61636,C1(CC(=O)NC(CNC(CC(C)C)=O)C(C)C)CCCCCO1 61637,CCC(C)CC(=O)NC1CCC1CNC(C1CCN(c2ccc(Cl)nn2)CC1)=O 61638,c1(C(=O)NCC2(NC(CNC=O)=O)CCCC2)cc(Cl)sc1S(N)(=O)=O 61639,C1(CNC(C(=C(C)C2CC2)F)=O)CN(C)CCN1C(c1ccoc1)=O 61640,[N-]=[N+]=NCC(F)CCNC(=O)C(O)CCCNC(c1cnc2n1CCC2)=O 61641,Cc1oc(C(F)(F)F)nc1C(=O)NCC(C)CNC(C1CC1(Cl)Cl)=O 61642,c1(CN2CC(CNC(Cc3cncc(C)c3)=O)C2)c[nH]c2cc(Br)ccc12 61643,O(NC(=O)C(CCF)Nc1c(C(=O)N(C)C)ccnc1)CCCN(C)C 61644,CC1CN(C(c2ncc(F)cc2F)=O)CCC1NC(c1nn[nH]c1Cl)=O 61645,C1(C(=O)NCC(CC)NC(c2cc(CCO)on2)=O)CCC(O)CN1C 61646,Cc1ccc(NC(N2CCCC(C(C)(C)C)CC2)=O)c(O)n1 61647,N1(C(C2N(C(C(N3CCSCC3)C)=O)CSC2)=O)C2CCC1CC(CO)C2 61648,C1(C(N2CC3(NC(C(CC)C)=O)CC2(COC)C3)=O)CCc2nc[nH]c2C1 61649,Cc1nccnc1C(C(=O)NC1CN(C(=O)OC(C)(C)C)C1)N(C)C1CC1 61650,C1(N(C(CCCc2ncc(C)o2)=O)C)CCC(NC(C2CC2C2CC2)=O)CC1 61651,C1(C(N2C(CNC(=O)CC(=O)Nc3nccs3)CC2)=O)CC12CCc1ccccc12 61652,C(=O)(C1=CCCOC1)NCC(C1CCN(C(c2c[nH]cc2C2CC2)=O)CC1)C 61653,CC1CC(NC(c2ccccc2Cl)=O)CN1C(=O)Cc1csc(S)n1 61654,C1(CCC(=O)NC(CC2CC2)CO)CCCN(C(=O)CC2CCOC2=O)C1 61655,c1(C(=O)NC(C)CCCCNC(c2ccco2)=O)n[nH]cc1[N+](=O)[O-] 61656,CC(CC1CCCO1)C(=O)NCCOCCOCCNC(=O)C(c1ccc(Cl)s1)=O 61657,c1(N(CC(=O)NCC(C)NC(=O)C(F)(F)c2nccs2)C)ccccc1 61658,C#Cc1cncc(C(=O)NC2CC(N(C(=O)CCSCc3ccccc3)C)C2)c1 61659,CCC(C)C(CC(=O)NC1CC(C2CC2)C1)NC(=O)COCC(=O)NC 61660,c1(C2CCCN(C(C(=O)NCCCSC)c3ccns3)C2)ccccc1C#N 61661,CC(Cc1ccccc1)C(=O)N(CC(O)CNC(C1CCCC1)=O)C 61662,N1(C(C(C)(C2CC2)NC(C)=O)=O)CCC(CN(C(=O)C(C)CC2CCC2)C)CC1 61663,c1(N(C)Cc2csc(Br)n2)nc(=N)nc(NCCCc2ccccc2)[nH]1 61664,C(CC(C(=O)N1CCCC(OCC)C1)NC(=O)CCCSC)OCC 61665,N1(C(CC=C)=O)CC2CCCC(CNC(C3CCCC3OC)=O)C2C1 61666,C1(C(=O)NCCCC(C)C)CC(NC(=O)CCC2(C)CC2)CCO1 61667,C1(C(N(CCCNC(C(C)(C)OCC)=O)C)=O)CC(N=[N+]=[N-])C1 61668,C1(NC(CC=CC=C)=O)CC(NC(C2CCC(CCCCC)CC2)=O)CC1O 61669,C#CCC(CC(=O)N(C1(c2nn[nH]n2)CCOC1)C1CC1)c1ccccc1 61670,C#Cc1ccc(C(=O)NC2CC(C)CN(C(c3cnc(O)o3)=O)C2)c(OC)c1 61671,n1(CC)cc(CNC(=NCCF)NCc2ccccc2Cl)c(O)nc1=O 61672,Cc1ccc(F)c(C(=O)NCC(C(=O)N2CCC(C(C)C)CC2)C(C)C)c1 61673,N1(C(C2C(CCOC)C2)=O)CCC(F)C(NC(c2cscc2C)=O)C1 61674,C1(CC=C)(NC(C2CCCO2)=O)CCN(C(c2ccc(F)c(CO)c2)=O)CC1 61675,C(=O)(CC(=O)NCCn1cc(CC(C)O)nn1)OC 61676,C1(C)(SCC2CCCN(C(=O)NCCn3c(C)csc3=O)C2)NC(=O)NC1=O 61677,Cc1cc(CSC2CCC(F)C2)ncc1S(=O)(=O)N(C1(c2ccccc2)CC1)C 61678,CC1(C)CCC(C)(C(=O)NCCOCCNC(=O)Cc2ccccc2O)CC1 61679,CCCCCC(O)C(=O)NCCN(C(=O)CC1CC(=O)NC1=O)C 61680,C(=O)(CCCC(=O)NCCC1CCCN(C(C2CC3C=CC2C3)=O)C1)N(C)C 61681,c1(C(=O)NC(CN(C(C(COC)(C)O)=O)C)C)coc2c(F)cccc12 61682,c1(C(N2CCC(O)(C(C)NC(C=C(C)C(C)C)=O)CC2)=O)cccn2nccc12 61683,N1(C(C(=O)NCc2cccc(OC)c2)c2ccns2)CCSC2COCCC12 61684,c1(CC(=O)NC)ccc(C(=O)NCC2CCN2C(=O)CCn2cncn2)cc1 61685,C12(CNC(CC3(N(C(CS(CC)=O)=O)C)CC3)=O)CC=CC(C1)OC2 61686,c1(C(N2CCC(OCCNC(C(C)S(N)(=O)=O)=O)C2)=O)cc2cc[nH]c2cn1 61687,c1(C(=O)NC2CC(CNC(c3ncn(CC)c3)=O)C2)c[nH]c2ccccc2c1=N 61688,N1(C(C2(CCC)CC2)=O)CCC2CCCN(C(c3ccsc3)=O)C2C1 61689,c1(CC)nc(C)cc(=NCC2CN(C(c3cnn(CC(F)F)c3)=O)CC2C)[nH]1 61690,c1(C(C(=O)NC(CC=C)C)NC(=O)CC(C)C2CC2)cccc(F)c1 61691,CC1COCCN1Cc1cccc(C(=O)NCCC#N)c1 61692,C(=O)(C1=CC(O)C(NC(c2ccc(C)cc2C)=O)C1)NCCOCC(=O)OC 61693,C(=O)(C1=CCCCCC1)N1CC(O)(CNC(=O)CCN2C(=O)CCC2=O)C1 61694,C1(C)(CNC(CC2(C)C=CCC2)=O)CCN(C(c2ccc(OC3CC3)cc2)=O)C1 61695,N1(C(=O)COCc2cc[nH]n2)CC2CC1CN2C(c1ccc(OCF)cc1)=O 61696,N1(C(C(C)O)=O)CCCC(NC(C2CC3C=CC2C3)=O)CC1 61697,c1(OC)ccc2c(ccn2CC(=O)NCC(CNC(=O)Cc2ccsn2)OC)c1 61698,Cc1cc(CC(=O)NC(C2(O)CN(C(=O)C(F)CC3CCOC3)C2)C)n(C)n1 61699,c1(OCC(=O)N(C2(OC)CCOCC2)CCC)ccc(C(F)(F)F)cc1Br 61700,c1(OCC)cnc(C(=O)NC2(C)CCC(NC(C3CCCN3C)=O)CC2)c(Cl)c1 61701,Cc1cc(N2CCC(Nc3oc(C4CC4)nc3C#N)C2=O)ccc1Br 61702,C1(NC(C2CC(SC)C2)=O)CCCCCCC1NC(=O)CC(C)C(F)F 61703,C1(CCNC(C2(OC(C)C)CCOC2)=O)CN(C(c2cccn2C)=O)CC1C 61704,N1(Cc2ccc(-c3ccc(C(C)(C)C)cc3)o2)C(=O)C2C(O)CCN2C1=O 61705,C1(C(=O)NCC2N(C(C(c3ccc(C)o3)C)=O)CC=C2)CC(S(C)(=O)=O)C1 61706,c1(NCCN(C(C)C)C)cccc(S(=O)(=O)N(C2CC2C)C)n1 61707,C(=O)(C(F)CC(C)(C)NC(=O)CCC(C)(C)N(C)C)N1CCN(CCC#C)CC1 61708,c1(C(C)C(=O)NCCCNC(=O)CN(C2CCSC2)C)c(F)cccc1F 61709,N1(C(CC(C=C)CC)=O)CC2=C(C1)CN(C(C1CC(OC)C1)=O)C2 61710,C(C)(CC(C(=O)NC1CCN(C(C)=O)CC1)N1CCC(OCCC(C)C)C1)SC 61711,N(C(=NCCN(C)C1CC1)NCC(C)C)C1C(OCC)C1 61712,c1(C(C(=O)NCCCSCC)N(CC(C)C)CC)cc(Cl)cc(Cl)c1 61713,C#Cc1cccc(NC(=O)Cc2nc(SC)ns2)c1 61714,CC(C)CC(C(=O)N1CC(NC(=O)CCOCC2CC2)C1)C(C)C 61715,CC(C)C(C)C(=O)N(C)CC1(O)CN(C(c2ccnc(-n3cccc3)c2)=O)C1 61716,N1(C(C(CCCNC(c2c(F)ccc(C)n2)=O)(C)C)=O)CCC2CCC(O)C1C2 61717,C1(NC(COCCOC)=O)CC2(CCCN(C(=O)CC3CCC(F)(F)CO3)C2)C1 61718,CCC(O)C(C)C(=O)NCC1CC(NC(=O)C=Cc2cccs2)C1 61719,c1(C(=O)NCC(CC)(C)NC(C2CCN(C)CC2)=O)nc(OC)cc(OC)n1 61720,C=CCCC(C(=O)NCC(C)(C)C=C)NC(=O)CCCCNC(N)=O 61721,n1(CCOC)nccc1C(=O)NCC1(F)CN(C(=O)C(O)CC2CCCCC2)C1 61722,C1(C(=O)OCC)CCC(C(=O)NCC2CCN(C(c3[nH]ccc3C3CC3)=O)C2)C1 61723,C1(CNC(C2CCS2(=O)=O)=O)CCN(C(=O)C=CCN2CCCC2)C12CC2 61724,c1(C(=O)NC(CN(C)C(C2COC(=O)C2)=O)Cc2ccccc2)ccc(F)cn1 61725,N1(C(C23OCC(C(=O)OC)(C2)C3)=O)CCC2(C1)CN(C(=O)C(C)O)C2 61726,Cn1cnc([N+](=O)[O-])c1NC(=O)C(N1CCC(CCCN2CCOCC2)CC1)=O 61727,CC1CC(CO)CN(C(c2ccn(C3CC3(F)F)n2)C(=O)NCC(F)F)C1 61728,C1(NCC=CC=O)C2CC3C(C2)C13CO.N1(OC(C)(C)C)CCC1C(F)(F)F 61729,Cc1noc(C)c1C(=O)NCC1(F)CCC(NC(C2(CO)CCC2)=O)C1 61730,c1(C(N2CCCC(C)(CNC(C(C(C)C)F)=O)C2)=O)cc2cc(Cl)c(Cl)cc2[nH]1 61731,N1(C(CC2N(C)C(=O)CC2)=O)CCC(F)(CNC(C2C(F)(F)C23CC3)=O)CC1 61732,C1(CCNC(C=C(C)Cl)=O)CN(C(=O)CCCc2ccsc2)CCS1(=O)=O 61733,c1(C(=O)NC(CCNC(C2CC(C)C2)=O)C)cccc(S(C)=O)c1 61734,c1(C(C(=O)NC2(CC(=O)NC(CSC)C)CCC2)F)ccccc1 61735,N1(C2CCN(C(C3(NC(C)=O)CC3)=O)C2)CCN(CC2CC(C)(C)CO2)CC1 61736,c1(-c2ccc(C3(O)CCC3)cc2)cccc2snnc12 61737,CC1CCCC(C)N(C(C2CCC(CNC(=O)Cn3ccnn3)O2)=O)C1 61738,c1(C(=O)NC(C(C)NC(C2CCCS(=O)(=O)C2)=O)CO)ccc2ncccc2c1 61739,CN1CCN(C)C(C(N2CC(N(C)C(c3ccc(N)c(N)n3)=O)C2)=O)C1 61740,CC(C)C(Cc1ccccc1)C(=O)N1CC(CCNC(C2CCNC2=O)=O)C1 61741,C1(NC(C(C)C(C)O)=O)CN(C(=O)Cc2cccc(O)c2F)CCC12CCC2 61742,Cc1ccc(C(=O)N(CCCNC(=O)CC2(C)CC2(F)Cl)C(C)C)c(O)c1 61743,Cc1nn(C)cc1C(N1CC(CN(C(=O)C=C(Cl)Cl)C)C1)=O 61744,n1(C(C)C)nccc1-c1cn(CC2CCN(C(C3(CC4CC4)CCC3)=O)C2)nn1 61745,CC(=O)C(C)CC(C)C(=O)N1CCCCCC(NC(=O)CC(C)(C)CN(C)C)C1 61746,Cc1nn(C)c(C)c1CNC(C1CCC(C)CN1C(=O)C=Cc1ccccc1)=O 61747,CCC(C(=O)NC(CCCNC(=O)Cc1cnns1)c1ccccc1)SC 61748,c1(CC)ncc(C(=O)NC2CCC(CCNC(=O)CC3CC(F)(F)C3)C2)[nH]1 61749,Cc1ccc(C(N2CC(NC(c3cc(C)c(C)s3)=O)C3CC23)=O)cc1C 61750,c1(C(=O)NCCC2CC(OC)CN2C(C2CCNC2=O)=O)c(C)ncn(C)c1=O 61751,C(=O)(CCCC(=O)NCC1(C)CC(NC(c2cc(OC)ccc2N)=O)C1)NC 61752,C(=O)(C1Cc2ccccc21)Nc1ncc(Cc2cc(C(=O)O)c(F)cc2)s1 61753,c1(CN2CC(=O)N2C)cc(Cl)ccc1O.Cc1ccc(Cn2ccnc2)cc1 61754,C(=O)(CN=c1cc[nH]cc1)N1C(C(C)(C)NC(C2C(C)SCCC2)=O)CCC1 61755,C1(CNCCCC(c2ccccc2)NC(c2c(C)ccnc2)=O)CCC(C)(C)CO1 61756,C(CC(C)N=c1nc(COC)[nH]s1)NC(C(CC)CCOC)=O 61757,N1(C(C2(C)CCCN(C(=O)CCC3CCCC3)C2)=O)CC2CCNCC2C1 61758,C=CCC(CC)C(=O)NC1(c2ccccc2)CN(C(=O)CC(C)C(F)F)C1 61759,CC1CC(Nc2ncncc2Cl)CCN1C(=O)C(O)C1CC1 61760,N1(CC)CC(C(=O)N(C)Cc2nccn2C)c2ccccc21 61761,CC#CCCCC(=O)N1CCC(C(=O)NC2(CSC)CC2)C1 61762,C(CN=c1cc(C)nc(N2CCC(NS(C)(=O)=O)C2)[nH]1)(C1CCC1)OC 61763,C1(CNC(C2(OC)CCCC2)=O)CN(C(=O)CCC2CC(C)(C)CO2)CCO1 61764,N1(C(CC(C)(F)F)=O)CCCC1C1CCCCN1C(c1cn(C2CC2)cn1)=O 61765,S(=O)(=O)(c1cccc(F)c1)N(C1CC2CNC1C2)CCCc1cccc(C)n1 61766,C(=O)(CP(C)(C)=O)NCC(C)CN(C(=O)C(C)(C)Oc1ccc(Cl)cc1)C 61767,CCCC(O)C(CO)NC(C1CCCCCC1NC(c1ccc(CO)cn1)=O)=O 61768,C(=O)(N=c1[nH]nc(CC2CC2)s1)C1(CC=C)CCCCN1Cc1ccc(Cl)cc1 61769,n1(CCC(=O)NCC(C)NC(c2ncc(CC)cn2)=O)cnc(C)cc1=O 61770,c1(C(N(c2ccc(Cl)cc2)C)=O)cc(S(=O)(=O)N(C)C)cn1C 61771,c1(C(=O)NCCN(C(c2ccc(C(C)C)cc2)=O)C(C)C)cncc2c1CCC2 61772,C1(NC(C)=O)(CO)CCN(C(c2cccn(C3CCC3)c2=O)=O)CC1 61773,CC1(C)CCN(c2nc(Cl)ncc2C2CC2)CC1CNC(c1ccc(F)cn1)=O 61774,c1(CC(N2CCC(NC(c3ccn(C)c3)=O)C2C2CC2)=O)ccc(O)c(Cl)c1 61775,c1(CC)ncnc(NC(CNC(=O)CN2C(=O)CCC2=O)CC)c1F 61776,C1(F)(CNC(C2(C)CCC2)=O)CCCN(C(=O)CC2(C)CCOCC2)C1 61777,C1(NC(CCOC(C)C)=O)CC2CC1CN(C(c1ncccc1Br)=O)C2 61778,C1(C(N(C2CCN(Cc3nc(CC)on3)CC2)C)=O)CCCN(CP(C)(C)=O)C1 61779,c1(C(N2C(COC)CN(C(C3(C)CCCN3C)=O)CC2)=O)cc(C)c(C)nc1C 61780,C1(O)(CC(=O)OCC)CCN(S(=O)(=O)Cc2[nH]ccc2CC)C1 61781,c1(C(N2C(C(N3CC(OC)C(F)C3)=O)C(O)CC2)=O)cnn2ccncc12 61782,C(=O)(C(CCCC(=O)OC(C)(C)C)N1CCC2C(O)C(C)(C)C12)NCCCC 61783,C1(F)(C(=O)NC(c2c(C)nccc2)C)CCN(C(=O)C(C)CC(N)=O)CC1 61784,S(=O)(=O)(c1nc(Br)cs1)Nc1c(OCC)c(F)ccc1 61785,CC(C)(CC1CCC1)C(=O)NCCCCNC(C1CCCCC1n1cccc1)=O 61786,N1(C(c2cc(CCC)[nH]n2)=O)CCN(C)C(C(=O)NC2CCC3CC2CO3)C1 61787,c1(C(=O)NC2C(CNC(c3cnc(OCC)s3)=O)C2)ccccc1C(N)=O 61788,c1(OC)noc(C)c1C(=O)NCCC1(O)CCN(C(=O)C(c2nc(C)cs2)C)C1 61789,Cc1ccc(CCC(=O)N(C(C)CCNC(=O)C(C(C)C)NC=O)C)cn1 61790,C1(C(N2CCC(C(C)=O)CC2)=O)CC(=O)OC1(C)C 61791,c1(CC)n[nH]c(COC(C)(C)C)n1.c1(C2C(C)NC(=O)N2)ccccc1 61792,C1(COC)CN(C(c2cnn(C)c2C)=O)CCN1C(c1ncccc1Br)=O 61793,c1(OC)cc(CNCc2ccncc2C(F)(F)F)cc2cc(C)oc12 61794,c1(CC)nc(C(=O)N(C2CCCC2C(=O)NOC2CCCCC2)C)co1 61795,N1(C(CCSCC=C)=O)CCCC(NC(=O)CCNC(=O)NC)C1 61796,C1(CNC(C2(CNC(c3cncn3C)=O)CC(=C)C2)=O)COCC(C)O1 61797,C(=O)(C(C)CC(C)C)N1CC(C(=O)N(C)Cc2cnccn2)(COC)C1 61798,C(C(=O)N1CC(O)(CCNC(C2CCSC2)=O)C1)(C(C)(C)C)NC(C)=O 61799,C12(C(N3CC(C)(NC(c4ccn(C(C)(C)C)n4)=O)C3)=O)CCCC1CS(=O)(=O)C2 61800,C(=O)(CCC(C)(C)C(=O)OC)NCC(CC)NC(C1(C)CC2CC2C1)=O 61801,C(=O)(C(F)(F)C(C12CC3CC1C2C3)OC)NC1CC(CC)(CC)NC1 61802,N1(C(C(N2CCCS2(=O)=O)C)=O)CCCCC1CCCNC(c1ccncc1)=O 61803,c1(-c2cc(C(=O)NCC(CNC(C3CCS3(=O)=O)=O)OC)n[nH]2)ccccc1O 61804,CN1CCN(C(=O)C(C(C)(C)C)NC(=O)Cc2cscn2)CC1(C)C 61805,c1(OC)cc(C(N2CC(NC(C3CCOC3(C)C)=O)C(O)C2)=O)cc(N)c1O 61806,Cc1ccncc1-c1ccc(C(N2CCC2C)=O)nc1 61807,c1(SCC(=O)NCCN(C(C2C(C)(COC)C2)=O)CCSC)cc(F)cc(Cl)c1 61808,N1(C(C(N2CC(C)(CO)C2)=O)=O)CCCOCC1 61809,c1(CN(c2ccc(OCCC(=O)OC(C)(C)C)cc2)C)cccc(F)c1F 61810,N1(C(C(C)C(C)(C)C)=O)CCC2(CCCN(C(=O)CC3CCS(=O)(=O)C3)C2)C1 61811,c1(-c2n(-c3cc(CC)c(F)cc3)nc(COC)n2)cc2c(OC)c(F)ccc2[nH]1 61812,S(=O)(=O)(c1ccn(C2CC2(F)F)n1)NCC1(C)CNCCC1O 61813,C1(CCC#C)CCCN(C(C2(NC(=O)CCC(C)C)CC(CO)C2)=O)C1 61814,N1(C(C(C)NC(=O)C(O)CN(C)C)=O)CCC(O)C12CCCC2 61815,n1(CC)nnc(C)c1CNC(C1(CCCO)CCCC1)=O 61816,C12(C(=O)NCC(CN(C)C(C3(CCF)CCC3)=O)O)COCC1C2(F)F 61817,c1(NC(=O)NCC)cccc(C(=O)NC(C2(O)CCN(C(=O)CCOC)C2)C)c1 61818,c1(NC(C(C)C)=O)ccccc1C(=O)NC1CCC(NC(c2ncccn2)=O)C1 61819,C1(O)(C(CNC(C2(OC)CC2)=O)C)CCN(C(=O)C(C)(C)c2ccnn2C)C1 61820,N1(C(C2CCC(OC)CC2)=O)CC2CC1CN2C(=O)COCC(C)(C)C 61821,c1(C(=O)NCC2C(C(=O)NCC(COC)C)CCO2)nccc2cc[nH]c12 61822,C(=O)(C(F)C(CC)CC)NC(CN(C(C(C)OCC=C)=O)C)C 61823,N1(C(C(C2CCC(=O)N2)C)=O)CCC(C)(NC(c2ncccc2N)=O)CC1 61824,C1(C(=O)NCC2CN(C(C(CC=C)C)=O)C(C)(C)C2)CC2CCC1C21CC1 61825,Cc1ncc(C(N2CCCCC(CNC(C3CC3C3CCCO3)=O)C2)=O)cc1N 61826,C1(C(=O)OC)(C(=O)NCCCN(C)C(C2CC(F)(CSC)C2)=O)CCCCO1 61827,C1(NC(C2C(OCC)C2)=O)CCC12CN(Cc1ccc(NC(=O)C(C)C)cc1)C2 61828,c1(SC)cc(C(N2CCCC2CC(=O)NC(CO)CC(C)C)=O)ccn1 61829,C1(CNC(C2COCOC2)=O)CCCCN(C(=O)C(F)=CC2CC2)C1 61830,C1(NC(c2c(C)c(O)ccc2)=O)CC2CC(NC(c3ncccc3F)=O)CC2C1 61831,C1(CCNC(C=COCC)=O)CN(C(=O)CCc2scnc2C)CCCO1 61832,c1(OC)cc(Sc2ccnc(O)c2)ccc1C(C)NC(N1CCCC1)=O 61833,N1(C(C(C)(C)O)=O)CCC(c2ccccc2)C(NC(C2(S(C)(=O)=O)CC2)=O)C1 61834,CCC(F)(F)CC(=O)N1CC2CC1C2CNC(=O)C1=C(C)OCC1 61835,c1(C(=O)NCC(C2(O)CCN(C(CC3(C=C)CC3)=O)C2)C)cc(OC)cc(Cl)c1 61836,c1(C(=O)NC2C(NC(c3occ(C)c3C)=O)CCC2)cc2c(ncn2C)s1 61837,C1(C(=O)NCC(CNC(C(CCC)(C)C)=O)(C)OC)CCc2cnnn2C1 61838,c1(C(=O)NCC)ccc(C(=O)NCC2CC(C(F)(F)F)(OC)C2)s1 61839,c1(OCC)ccc(C(=O)NCCCN(C(=O)CCn2ncn(C)c2=O)CC)cc1 61840,C1(N(C)C(C2CCCN2S(C)(=O)=O)=O)CC2CC1N(Cc1ccc(Cl)c(F)c1)C2 61841,CC1(C)CC1(C)C(N1CCC(NC(=O)CCc2ccon2)C1)=O 61842,C(C(C)C(=O)NCC(C)N(C(=O)Cc1[nH]cnc1C)C)OCC 61843,c1(C(N2C3C(NC(c4cccc(C)n4)=O)CC(C3)C2)=O)coc2c1C(O)CCC2 61844,S(=O)(=O)(c1c[nH]c(C(N2CCN(C(C3(C#N)CCCO3)=O)CCC2C)=O)c1)NC 61845,N1(C(c2nnn(CC)c2C)=O)CCN(C(=O)C=CSC)CC1CF 61846,c1(N(C(=O)NCC2(C(C)C)N=N2)CCO)cccc(Br)n1 61847,N(C1CC2CCC(C)(C)c3cccc1c32)C(c1c(F)ccc(OC)c1N)=O 61848,C1(CN=[N+]=[N-])CCN(C(c2cn(CCNC(c3c[nH]c(=S)cn3)=O)nn2)=O)CC1 61849,C(C)(CNC(c1cnc(S)nc1)=O)(CC(C)C)NC(CC(=O)NCC)=O 61850,c1(CC)ccc(C(=O)N(C(C)CNC(=O)COc2cc(C)on2)CC)[nH]1 61851,C(=O)(C(C)CCCC(C)C)NC1C(CC)CN(C(c2cc(C(C)C)[nH]n2)=O)CC1 61852,C1(N(C(C2C(CC)CC2)=O)CC)CCC(NC(=O)C(CC2CC2)OC)CC1 61853,c1(NC(C(C)C)=O)ccc(C(=O)OC2COCC2F)cc1 61854,Cc1cc(NC(=O)CCCCCN(C(=O)C(C)S(C)(=O)=O)C)cc(Cl)c1 61855,C1(NC(CC2N(C)C(=O)CC2)=O)CC2(C1)CN(C(=O)C=Cc1ccccc1F)C2 61856,CC1CCCn2ncc(C(=O)NC3C4CN(C(C5CC6(C5)CC6(F)F)=O)CC34)c21 61857,c1(C(N(C)CC2(NC(C(c3ccc(Cl)cc3)C)=O)CC2)=O)csc2c1CCCC2 61858,C1(C(C(=O)OC(C)(C)C)O)CCCCN1C(C(C)CCc1ccccc1Cl)=O 61859,c1(CCC(N2CCN(C(CN(CC(C)C)C(=O)CO)=O)CC2)=O)nnc(S)nc1O 61860,C(=O)(C1=NOC(C)(C)C1)NC1N(C(C23CCCC2(C(N)=O)C3)=O)CCC(C)C1 61861,C1(C(N2CC(C)N(C(C)C)C(C)C2)C(=O)NCC=C)CCc2nnc(C)n2C1 61862,C1(CC(=O)Nc2cn(C(C)C)nc2)CCCN(C(C2(O)CCSC2)=O)C1 61863,N1(C(CC(C(C)C)C)=O)C2CCC1C(C)C(NC(C13CC(CC(F)F)(C1)C3)=O)C2 61864,C1(NC(COCCOCC)=O)C2CC3CN(C(=O)CC45CCCC4C5)C1C3C2 61865,c1(OC)cc(C(=O)NC(C)C(C)NC(c2cnc(C(C)C)o2)=O)cc(F)c1F 61866,c1(OCC)cc[nH]c(=NCCC(C)NC(=O)C=Cc2cncs2)n1 61867,N1(C(=O)COc2ccc(Cl)cc2Cl)CCC2OCCN(C(C3CC=CC3)=O)C2C1 61868,c1(CNC(c2csc(Cl)n2)=O)ccc(CNC(C2CC3CC2CO3)=O)c(F)c1 61869,C1(CCC(=O)NC(CC)CC2CC2)CCCCC1 61870,c1(OC)cc(N)c(F)cc1C(=O)N(C)CCC1CCN(C(=O)CC(C)OC)CC1 61871,c1(CC(N2C(Cn3cc(CCSC)nn3)CCC2)=O)ccc(O)cc1C 61872,C1(C(=O)NC2CN(C(c3ncccc3Br)=O)CC2O)CC2(CCCC2)CO1 61873,C1(C)(C(N(C(C)(C)CC(=O)NC2CN(C)NC2=O)C)=O)COCCO1 61874,C1(=CC(=O)N(CC(CC)NC(C(C)OCC)=O)CC)CCC(C(C)(C)C)CC1 61875,C(C(CC(C)C)C(=O)NCC(C)(O)CC(C)C)NC(c1n[nH]c(CC)c1C)=O 61876,C1(NC(Cc2n(C)ccn2)=O)CC2(CCN(C(=O)C#CC3CCCCO3)CC2)C1 61877,N1(C(c2cc(OCC)ns2)C(=O)NC(C)(C)C)Cc2cccc(F)c2C1 61878,c1(C(=O)NC2CC(NC(c3c(C)c(C#N)ccc3)=O)C2)cncc(P(C)(C)=O)c1 61879,Cc1cnc(C(=O)NCC(C)(O)CNC(c2c[nH]c(=N)s2)=O)cc1Br 61880,C1(F)(C(=O)NCCOCCC)CCN(C(=O)Cn2cccn2)C1 61881,C(C(CC1CCCC1)C(=O)N1CCC(C(N)=O)C1)NC(C(OC)OC)=O 61882,c1(CC)ccc(C(N2CC(NC(=O)CC(F)(F)F)C3CC23)=O)cc1[N+](=O)[O-] 61883,CCN=c1cc(-c2nc(Cc3cc(C)c(F)c(F)c3)n(C(C)C)n2)cc[nH]1 61884,C(c1ccccc1C)=CC(N1CCC(CC(=O)N(C2CCN(C)C2)CC)CC1)=O 61885,n1(CC(=O)NCC(C2CCOC2)NC(=O)Cc2cccs2)cc(Cl)cn1 61886,c1(OCCCC(=O)NCCN(CCC)C(C2(C)CC2C)=O)ccc(Cl)cc1C 61887,c1(CNC(c2cc(C)no2)=O)ccc(CNC(=O)C(F)C(F)(F)F)cc1F 61888,c1(N2CC(C)CN(C)CC2)[nH]c(=NCCS(C)=O)nc2scnc12 61889,C1(SC)CCCC1C(=O)NC1(C(N2CCC(N3CCOCC3)C2)=O)CCCC1 61890,C(=O)(CCC(F)(F)C(F)F)NCCCCC(C)NC(CC(C)OC)=O 61891,C(=O)(C1=CC2CCCC12)NCCOCCCN(C)C(c1cnn(C)c1Cl)=O 61892,N1(C(C(C)N(C(C(C)OCC)=O)C)=O)CCC(CC(=O)N(C)OC)CC1 61893,C1(NC(CCCC)=O)CN(C(C2CCn3c(cnc3C)C2)=O)C2(CCCCC2)C1 61894,c1(C(=O)NC(CC)(C)CNC(=O)Cc2cncs2)cnc(C)c(C#N)c1 61895,C12(CNC(c3c(C)nn(C)c3)=O)CCC(C1)N(C(C1CCC3CC1CO3)=O)C2 61896,c1(C(=O)NCC(C)N(C)C(c2c[nH]c(=O)cn2)=O)cnc(C(F)F)cn1 61897,C1(NC(c2c(CC)csc2)=O)CC=C(C(=O)NCCc2ccon2)C1 61898,n1(CC)cnc2c(NCc3cn(CC)nn3)[nH]c(=NCC(C(C)(C)C)SC)nc12 61899,C12(NC(C(C=C)CC)=O)CCCC1N(C(c1oc(C3CC3)nc1C)=O)CCC2 61900,CC1(NC(C2CCCC3CC23)=O)CCN(C(c2ccccc2F)=O)C1 61901,C12(C(N3CC(CNC(c4cccc(CC)n4)=O)OCC3)=O)CCCC1CCC2 61902,N1(C(c2noc(CC)c2C)=O)CCC2CCN(C(c3nc(C)nn3C)=O)CC12 61903,CC1(C)CC(NC(c2snnc2C2CC2)=O)CCN(C(=O)Cc2ccsc2)C1 61904,C#Cc1ccc(CC(N2CC(NC(=O)CCC3CCCOC3)C(CC)C2)=O)cc1 61905,n1(CCC(N2C(C(C)(F)F)CCC2)=O)nc(O)c2c1CCCC2 61906,c1(CN(C(C(=O)NC(CCCCC)C)=O)C)cc(F)ccc1C 61907,c1(NC(C)CC(N)=O)nc2ccccc2nc1N1CC2C(C1)C2(F)F 61908,C1(C(N2C(CC)CC2)=O)CCN(C(=O)Cc2nccn2C)C1(C)C 61909,c1(CNCC(CC2CN(C(CSC)=O)C2)(C)C)cccc2c1oc1ccccc21 61910,Cn1c(O)nc2cc(C(N3C4CCC3CC(CNC(C3CCC3)=O)C4)=O)ccc12 61911,CN(CCCC(=O)NCC1(F)CCN(C(=O)CCNc2ncccn2)C1)N=O 61912,c1(NC(C)CCO)[nH]c(=NCc2nc(Br)n(C)n2)nc2c1cnn2C 61913,N1(C(CCCOCC=C)=O)CCN(C(=O)C(C)c2ccco2)CC1c1cn[nH]c1 61914,C(c1cccnc1)=CCNC(N1CCC(NC(COCc2onc(C)n2)=O)C1)=O 61915,N1(C(C2CC3CCCC3C2)=O)CC2CCCN(C(=O)CSC(F)(F)F)C2C1 61916,C(CS(=O)(=O)CC(=O)N1CCC(C2CC2)C1CNC(c1c[nH]nc1C)=O)OC 61917,C1(N(C(C2(OC)CCCOC2)=O)C)CCCN(c2ccnc(C(F)(F)F)n2)CC1 61918,C1(CNC(C=CCCC)=O)CCCCC1NC(c1cc(CC)c(C)s1)=O 61919,C(=O)(N1CC(C)(O)CO1)C1CN(C(C(CC)N(C)C)=O)CC1C 61920,C(CC(O)CNC(=O)C(C)N(C(=O)CN1CCNC1=O)C1CC1)OC 61921,c1(CN2CCC(NC(C(c3ccccc3)OC)=O)C2)cc(Cl)c(O)c(Cl)c1 61922,N(C)(C1CCc2c(F)cccc21)C(C(C)C(C)c1ccccc1Cl)=O 61923,C1(C(=O)NCC(CNC(C2C(C(C)(C)C)C2)=O)(C)O)CCCCC(=O)N1 61924,CC1(C)C(NC(=O)CC2CCCCC2)CCN1C(=O)CC(F)(F)Cl 61925,N1(C(C)=O)CC(NS(=O)(=O)CC)C(C)(C)C1.C(=O)(CCO)NCC(C1CCCC1)OC 61926,C1(CNC(c2c(O)ccc(OC)c2)=O)(CO)COCC2CCCCN12 61927,c1(C(=O)NCC(c2ccco2)OC)n[nH]c2c1CN(C(=O)C(C)CC1CC1)C2 61928,C1(NC(C(CCC)OCC)=O)COC2(C1)CN(C(c1cc3c([nH]1)CCCC3)=O)C2 61929,c1(C(N2CC(C)C(CNC(C3CCC=CO3)=O)C2)=O)cccc(Cl)c1N 61930,c1(C(=O)OC)ccc(CC(N2CCN(C(c3nncn3C)C)CC2)=O)cc1F 61931,CC(CN=c1nc(-c2cccs2)[nH]c2ccccc12)N(C(=O)C(N)=O)C 61932,C1(CNC(C2CCCC3CC23)=O)CCN(C(c2nnc(O)nc2O)=O)C12CC2 61933,c1(NC(CCC(C)(C)NC(=O)CCN=[N+]=[N-])=O)cncc2ccccc12 61934,c1(C(N(C2CCCC2)CC#CC)=O)ccc(NC(=O)CC(C)n2ccnc2)s1 61935,c1(C(=O)NC2CC(C)N(C(=O)C(C)n3cccn3)C2)nc(F)ccc1Cl 61936,C1(C(=O)NCCC(=C)CNC(=O)C=Cc2cnc[nH]2)CCCC(=O)N1 61937,c1(CC)nc2ccccc2c(C(=O)NCC2(NC)CCOC2)c1C 61938,C(=O)(C(C)(C)CN=c1[nH]c(=NCCS(=O)(=O)CCO)c2cccc(F)c2[nH]1)NCC 61939,C1(NC(=O)COCc2ccncc2)C2CN(CC(=O)NCCC3CCOC3)CC12 61940,C1(C(=O)NCCC2CCC(CO)CC2)CC(C2CCC2)C1 61941,Cc1c(CC(=O)NCC2CC2NC(=O)C2=CC(C)(C)C2)c(O)nc2[nH]nc(O)c12 61942,CON(C)S(=O)(=O)c1cccc(C(N2CC3CC2C3NC(C2CC(F)C2)=O)=O)c1 61943,Cc1cc(C(=O)NCc2cccc(C(=O)NC(C)C(F)(F)CO)n2)c(C)s1 61944,CC1(C)CCN(C(C2CSCCS2)=O)CC1NC(c1coc(Cl)n1)=O 61945,CC(C)(O)C(c1ccccc1)NC(N1CC(OCCO)C1)=O 61946,C(N=c1ccc(C#N)c[nH]1)C1OCC(CNC(c2c(Cl)cn(CC)n2)=O)C1 61947,Fc1ccc2c(c1)C(NCCOCC1CCCC1)CCCO2 61948,Cc1ccc(-c2nc(C)c(C(=O)NC3CCC(CNC(=O)C(C)C)C3)s2)c(F)c1 61949,c1(CC(=O)NCC(CCNC(CCC=CC)=O)(C)C)coc2c(F)c(F)ccc12 61950,C(C(C)C(F)(F)F)N(C(C(C)NC(C(C=C)OC)=O)=O)C 61951,c1(C(=O)NCC(C2CCOC2)NC(=O)C=CCO)cnsc1 61952,CCN=C(NCCS(=O)(=O)c1ccccc1C)N1CCC2(CCCC2)C1 61953,CCC(C)C(C(=O)NC1CN(C(=O)Cc2ccnc(OC)c2)CC1C)N(C)C 61954,CN1CCN(C(C2CNC(=O)N2)=O)CC1CNC(c1ccc(-c2ccco2)o1)=O 61955,Cc1oc(S(N)(=O)=O)cc1C(N1CCN(C(C2CCC3(CCC3)O2)=O)C(C)C1)=O 61956,CCS(=O)(=O)c1cnc(O)c(C(=O)NCCC(C)CCNC(C2(C#N)CC2)=O)c1 61957,C(=O)(C(O)CC(C)(C)C)NCCN(CCC)C(C1CNC(=O)C1)=O 61958,C#CCC(C)(C(=O)N1CCCC(CC2CC2)C1)NC(=O)Cc1cnccc1C 61959,c1(C(=O)NC23CCCC(NC(CCCC(=C)C)=O)(C2)C3)cc(F)c(F)c(C#N)c1 61960,c1(C(=O)NC2(CO)CN(C(CC3CNC(=O)O3)=O)C2)cc2n(n1)CCO2 61961,S(=O)(=O)(CC(C)(C)C(C)C)NCC(n1cc(CCCC=C)nn1)C 61962,c1(N(C2CC(c3ccccc3)(NC(=O)CP(C)(C)=O)C2)C(C)=O)ccc(F)c(F)c1 61963,c1(OC)cccc(C2(C(=O)NCCN(C)C(C3CC=CCC3C)=O)CC2)n1 61964,c1(C(C)C)ncc(-c2nc(-c3ccc(N4CCN(C)CC4)cc3)no2)cn1 61965,C1(C(=O)NC2(C)CN(C(C(C)SC(F)(F)F)=O)C2)CCN(C(=O)C(N)=O)CC1 61966,c1(C(N2CC(CNC(c3cccc(SC)c3Cl)=O)C2)=O)ccc2c(c1)CNC2=O 61967,CCC(CC(=O)NC1CCC(O)CN(C(=O)Cc2cccc(OC)c2)C1)C(C)C 61968,c1(OC)cncc(C=CC(N2CCC23CN(C(c2c(OC)noc2C)=O)C3)=O)c1 61969,C1(C(C)C(=O)NCC(C2CC2)NC(C2CCC2CF)=O)CCCCC1 61970,CCCCC(C(=O)N(C1CC1)CC1CCCCN1C(=O)CSCCC)C(C)C 61971,c1(C(=O)NCC(C)NC(=O)C(C)CC2CCCCC2)nc(Br)n2ccccc12 61972,N1(C(CN(CCOC)C)=O)CC2CCC2(CCNC(c2c(C)ccnc2O)=O)C1 61973,C1(C(=O)NC)(N(C)CC)CCCN(C(c2ccc(OC)nn2)=O)C1.C1(CC)CCC1OC 61974,C1(OC)CC(CNC(=O)C2=CCOC2)N(C(=O)CC2(C)CCCCC2)C1 61975,n1(CC(=O)NCC2CC(CC(=O)OC)C2(C)C)nc(O)c2ccccc2c1=O 61976,N1(C(c2ccnc(C(=O)OC)c2)C(=O)NCCOC)CCCC(O)(C(C)C)C1 61977,N#Cc1cc(C(N2CC(NC(C3CCCOC3)=O)CC(F)C2)=O)ccc1F 61978,n1(CC(=O)NCC2CN(C(=O)C(O)CC3CCOCC3)CCO2)ncccc1=O 61979,CC1(C)CCOC1C(=O)NCC1(C(=O)Nc2cncc(Cl)c2)CC1 61980,C(CCCC(CO)NC(=O)C(O)Cc1cc(Cl)sc1Cl)NC(=O)COC1CC1 61981,N1(C(C23C(CN(Cc4ccc(C(C)(C)C)cc4Br)C2)C3)=O)CCn2cncc2C1 61982,c1(CC(=O)NCC2(C(=O)NCC3CCCC3(F)F)CCCC2)ccc(F)cc1Cl 61983,N1(C(=O)Nc2cccc(OCC)c2)CC(=O)Nc2ccc(C#N)cc21 61984,c1(C(=O)NC(C)CCN(C(=O)CCn2cc(Br)cn2)C)cccnc1O 61985,C(=O)(C(O)C1=CCCCC1)NC(C(=O)NCC(C#C)OC)CC(=C)Cl 61986,c1(CCC)ncoc1C(=O)NCCCN(C)C(c1cnn(CC(F)(F)F)n1)=O 61987,CC(CC(C)NC(=O)Cc1cnn2ccccc12)N=c1[nH]c(Cl)nc2c1SCC2 61988,CC(C)C(C)CC(=O)NC1(C2CCCN2C(=O)CN2C(=O)CCCC2=O)CC1 61989,c1(NCC2CCCN(C)C2)ccc(S(=O)(=O)NCCOC2CC2(F)F)c(Cl)c1 61990,C1(C)(COC)CN(N2CCCC(n3cccn3)C2)CCO1 61991,C(C(C)(C)CNC(=O)CN1CCCC1CO)N(C(CN(C1CC1)CC)=O)C 61992,C1(OC)CCC(C(=O)NCCC2CC2)CC1.N12CCCC1c1csc(n1)C2=O 61993,c1(C(N2CCC(NC(=O)C=Cc3ccccc3)C2)=O)cc(NC2CC2)ncc1Cl 61994,C12(NC(c3c(CC)csc3)=O)CCCC1CN(C(=O)C(C1CC1)C1CC1)C2 61995,N1(C(C(C(CC)C)N)=O)CCC2CN(C(=O)Cc3cccc([N+](=O)[O-])c3)CC12 61996,C1(SC)CN(C(=O)CNC(c2ccoc2)=O)CC1NC(=O)CC1CC(=O)N(C)C1 61997,C=C(Br)CN=C(NCC(=O)NC1CCCCO1)NCC(=O)NCC(F)F 61998,N1(Cc2ccc(C)o2)CCCC(O)(CNC(=O)C(=O)C(C)C)C1 61999,c1(OC)ccc(CN(C(c2ccccc2OC)C(=O)NC2CCCC2)C)nn1 62000,CCC(C(=O)OC)C(=O)NCC(C)CNC(c1cn(C(C)(C)C)nn1)=O 62001,c1(C2CN(C(C=CC(C)(C)SC)=O)C2)cc(O)n[nH]1.C1(N2C(C)C2=O)CC(C#N)C1 62002,O(NC(=O)CCCN(C)C(C1CC(C)(C)CN1C)=O)CC(=C)C 62003,N1(C(c2c(N)ccc(C)c2)=O)CCC2(CCN(C(C3(C(N)=O)CC3)=O)C2)C1 62004,C1(C2(NC(C3(C(=O)OC)C=CCC3)=O)CC2)CCCCN1C(c1ncncc1Cl)=O 62005,CC1=C(C(=O)NC2C=CCN(C(c3sccc3Cl)=O)C2)C(C)n2nnnc2N1C 62006,c1(CCOC(c2occ(C(=O)OC)c2)=O)c(C)nc(SC)nc1O 62007,C1(C)(NC(C2CC(=C)C2)=O)CCN(C(=O)CCn2c(-c3cccs3)nnc2S)CC1 62008,n1(CC)nc(-c2ccoc2)nc1CCSc1noc(CC(C)C)n1 62009,CC(C)CC(C(=O)N1CCC(CCN(C)C(C2(C)C=CCCC2)=O)CC1)N(C)C 62010,CC1N(C(c2ccc(CNC(c3cc(C#N)cs3)=O)o2)=O)CCCC1(C)C 62011,C=C(C)C(CC(=O)N1CCC(NC(=O)CN2CCC(CC)C2C)CC1C)OCC 62012,c1(C(N2CCC(CCN(C)C(C3(C4CC4)CC3)=O)CC2)=O)cccc2sccc12 62013,C1(C)(OCC(=O)N(C(C#C)C)CC)CN(C(=O)Cc2sccc2C)C1 62014,N1(C(=O)Cc2cc[nH]c2)CC(C2CCCN(C(=O)C(O)C3CCC3)C2)C1 62015,Cc1cc2n(n1)CCN(C(c1nccc3occc13)=O)C2 62016,C(C(CNC(C1C2(CC2)C12CC2)=O)S(C)(=O)=O)NC(C(c1c(C)cccc1)C)=O 62017,c1(CN2C(C(=O)Nc3c(C(C)C)scn3)CC3CC32)ccc(O)c(Cl)c1 62018,N1(C(c2cc3cccnc3s2)C(=O)NCC=C)CCNC(=O)C(F)(F)C1 62019,C1(CC)(CC)CC(NC(=O)Cc2nonc2C)CN1C(c1ccc(C)s1)=O 62020,c1(C(N(CC(O)CNC(=O)C=Cc2cn[nH]c2)C)=O)cccc(F)c1[N+](=O)[O-] 62021,C1(C(=O)NC(CNC(C2CC2C2CCC2)=O)CC2CCCCC2)Cc2nncn2C1 62022,N1(C(c2occ(C)c2)=O)CC=C(CC(=O)N(C2CCN(C(C)C)C2)C)CC1 62023,c1(-c2n(CC=C)nc(CC3CCC3)n2)cc2cc(OC)ccc2s1 62024,C1(O)(C(C)NC(c2cc(Cl)n[nH]2)=O)CCN(C(=O)CN2CCCC2)C1 62025,C1(C(N2CCC(C(=O)NC)CC2)=O)CN(C(c2ccno2)=O)Cc2cccn2C1 62026,O=C(C(F)(F)C(F)c1ccccc1)NC(c1ccc(F)cc1)c1ccc(Cl)cc1 62027,c1(C(C)N(C(N)=O)CC2CCCCO2)ccc(CNC(=O)CCc2cnc[nH]2)cc1 62028,CC(O)C(F)(F)C(=O)N1CC=CC(NC(=O)CCc2ccc(Br)s2)C1 62029,c1(CC(=O)NCC2CCC2NC(C2CC3CC3C2)=O)c[nH]c2cccc(F)c12 62030,c1(N2CCC(C=C)C2)nc(N2CCC3(CCC(O)C3)C2)nc2ccsc12 62031,c1(C(=O)NCCOCCCN(C(c2cc(CC)[nH]n2)=O)C)cc(F)ncc1OC 62032,C12(C(N3CCC(CN(C(c4c(OC)cccn4)=O)C)CC3)=O)CCCC1OCC2 62033,c1(NCC2(F)CC(CNC(C(=O)N(C)C)=O)C2)ncnn2cccc12 62034,c12c[nH]c(c1)C(=O)NCCC1(CC1)NC(=O)CC2.C1(C(N)=O)(N)CC1.CC 62035,c1(C(=O)NC2CCCN(c3nc(O)n[nH]3)C2)c(Cl)cc(F)cc1Br 62036,Cc1nsc(N(C)CCOCCNC(C2CCC(C)O2)=O)c1C#N 62037,N1(C(=O)Cc2cn[nH]c2)CCC(OCCNC(=O)CCCC2CCC2)C1 62038,c1(SCC)ccc(C(N2CCC(F)(C(=O)N(C)C)C2)=O)cc1 62039,CC1CC(=O)NCC1C(N1CCCN(C(=O)CCN2CCC(O)CC2)CC1)=O 62040,C1(C(=O)NCCCC(=C)Cl)CCN(C(C2CCN(C)C(=O)C2)=O)CCO1 62041,N1(C(c2ccccn2)=O)CC2(C1)CN(C(=O)CNC1C(C(C)(C)O)C1)CC2CO 62042,N1(C(Cc2cn(CC)nc2)=O)CCCC(C(N2CCC(NC)CC2)=O)C1 62043,N1(C(C(C)SC)=O)CCCC(C)(C)C1C(=O)N(C)CCC1CCCN1C 62044,CN1C(=O)CCC(C(=O)NC2CC2c2cn[nH]c2)C1=O 62045,c1(C(N2CC3(CC(NC(c4c(N)cc(F)cn4)=O)C3)C2)=O)c(F)ccc(F)c1Cl 62046,CCCCCCC(=O)NC(C1CCCC1)CNC(c1ccncc1C(F)F)=O 62047,Cc1cc(C(N2CCC(NC(C3CC4(C3)CC(C)(C)C4)=O)C2)=O)c(N)cc1F 62048,C(=O)(C1=CCS(=O)(=O)C1)NCCOC1CCN(C(c2nn(C)c(=O)cc2)=O)C1 62049,C(=O)(C1=CCCC1)NCC(CNC(C=C(CC)CC)=O)OC 62050,c1(C(=O)NCC2C(NC(C(C(C)C)(C)O)=O)CCC2)cccc2cc[nH]c12 62051,C1(C(N2C(C3(NC(Cc4n(C)cnc4)=O)CC3)CCC2)=O)OCCOC12CCC2 62052,C1(CC(N2CC(C)(NC(c3c(C)nccn3)=O)C2)=O)Oc2ccccc2NC1=O 62053,N1(C(C2(N)CC(=C)C2)=O)CC2(C)CC1CCO2 62054,c1(OC)cc(C(=O)NCC(C(C)C)NC(C23CCC(F)(CO2)C3)=O)cnc1OC 62055,c1(CC)c(NCC2CCN(CC(CSc3nccnc3Cl)O)CC2)csc1C 62056,c1(CC(C)NC(c2c(F)cccc2F)CCOC)ccc(OC)c(F)c1 62057,C1(C)(C(C)C)CCN(C(CCc2cnn(C)c2)C(=O)NCCCOCC2CC2)C1 62058,N1(C(C2CCC(Nc3ncnc4ccccc34)CC2)=O)CCC2(CCCOC2)C1 62059,CN1CCN(C(C(=O)N(CC)CC2CCCO2)c2ccco2)C(c2ncc[nH]2)C1 62060,C(=O)(CCCCC(C)(C)C)N(C1C2CCCC1COC2)C 62061,C1(C)(C(=O)NCC(=C2CN(C(CC(C)C3CCCO3)=O)C2)F)CCOC(C)C1 62062,Cn1cnc2[nH]c(C(=O)NC(CNC(=O)C(C)(C)S(C)(=O)=O)C3CC3)cc12 62063,c1(C(=O)NC(C(C)NC(c2ccn(CCF)n2)=O)C)cccc2cncn12 62064,N1(C(=O)CCN2C(=O)CCC2=O)CCC2CCN(C(c3cncc(Cl)c3)=O)C2C1 62065,C(=O)(C#CC1(C)CC1)N1CCC(C)(CCNC(C2CN(C)C2)=O)C1 62066,c1(CCC(=O)NCC2CC2NC(=O)CC2CNC(=O)C2)cccnc1Br 62067,CCCCCCCCC(=O)OCCOC(c1cccc(S(=O)(=O)NC)c1)=O 62068,C(=O)(CC(C(F)(F)F)NC(=O)Cc1cccnc1O)NCCSCC#C 62069,C#CCC(C)(C(=O)NCCCC(C)CO)NC(=O)Cc1cccn1C 62070,C1(C(=O)NCC(CN(C(C(C#C)(C)C)=O)C)(C)C)CC(c2cnn(C)c2)=NO1 62071,c1(COC(c2ccoc2C(=O)OCC(CC)(C)CC)=O)ccc(C)c(F)c1F 62072,Cc1cccc2c(C(=O)NCC3(C)CCCN(C(c4ccnnc4)=O)C3)coc12 62073,C(C(C)(O)C(=O)N1CC(CC(F)C(=O)NC)C1)C(=O)OC 62074,C1(OC)CC(NCC(=O)NC(c2cccc(Cl)c2)=O)C12CCC2 62075,N1(C(CC(COC)NC(=O)CCc2nc[nH]n2)=O)CC2(CNC(=O)OC2)C1 62076,C1(C(C)C)CCc2sc(C(=O)OCCC3CN(C(=O)OC(C)(C)C)C3)cc2C1 62077,n1(C(C=C)C)nc(-c2ccsc2)nc1-c1nn(C)nc1Br 62078,C12CC(C1)CN(CCCC)CC(=O)N2.C(=O)(C(C)N(C)C(=O)OC)NC(C)(C)C 62079,C(c1ncc[nH]1)=CC(=O)N(C(CNC(=O)C=Cc1cscn1)C1CC1)C 62080,CC1CNC(=O)CN1C(C1(F)CCN(C(C2(CF)CCOCC2)=O)C1)=O 62081,Cc1cc(C)c2[nH]cc(C(N3CCC(S(C)(=N)=O)C3)=O)c(=O)c2c1 62082,N1(c2nccc(-n3c(C)cc(C)n3)n2)CCC(NC(c2cccnc2)=O)C(O)C1 62083,C(CCC(CCC)NC(=O)CC1CC(OC)C1)NC(C(F)=CC)=O 62084,CC1(C)COC(CC(=O)NC2CC(NC(=O)C=C3CCC3)C2)CO1 62085,C(=O)(C1=C(C#N)CCC1)N1C(C)CC(NC(C=Cc2c(C)cccc2)=O)C1 62086,CCC(C)(C)C(O)C(=O)N1CCC2CC1CN2C(c1cccc(F)c1Cl)=O 62087,N1(C(c2cc(C)cc(Cl)c2)=O)CCC2(CC1)CN(C(=O)C1=CCC1)CC(C)O2 62088,C1(CNCc2ccc(C)s2)COCCN1C(=O)Cc1ccc(NS(C)(=O)=O)cc1 62089,C1(C(N2CCC(O)(C(F)F)C2)=O)(NC(=O)C(O)CN2CCCC2)CC(F)(F)C1 62090,CC1(C)CC(C(N2CC(C)(C(N)=O)C2)=O)CC(C)(C)S1(=O)=O 62091,c1(CC)ncc(C(=O)NC(C)CCN(C(=O)Cc2cccc(O)c2F)C)c(C)n1 62092,N1(C(c2cccc(I)c2)C(=O)NCCC)CCN(C2CCCC2CO)CC1 62093,CCCCC(C(=O)N1CCN(C)CC1C(=O)NC(CCC)c1nn[nH]n1)C(C)C 62094,c1(C(N2CCC(N(C(C(C)NC(=O)OC)=O)C)C2)=O)ccc(O)nc1C 62095,C1(CNC(CC2CC(=O)NCC2)=O)CN(C(c2cc(O)ncc2F)=O)CCCO1 62096,N1(C(C2(SCC)CC2)=O)CCC(CN(C(C2SC3C=CC2C3)=O)CC)CC1 62097,C1(NC(CSCCC)=O)CN(C(=O)C=Cc2ccccc2C)C2CCCC12 62098,N1(C(C=COCC)=O)CCC2(CC1)CCN2C(c1cccc2[nH]ncc12)=O 62099,C1(C(=O)NCC(C2CCN(C(C(C)n3cccn3)=O)CC2)O)CC(=O)NC(=O)N1 62100,c1(C(=O)NC(C2CCN(C(=O)CN(C)C(c3cccs3)=O)C2)C)ncc(Cl)s1 62101,c1(C(=O)Nc2nc(C(=O)NCCC#C)n(C)c2)c(C)cc(OC)cc1C 62102,C(CC(CNC(c1cnnn1-c1ccccc1)=O)NC(=O)CC1(C)CCC1)OC 62103,Cc1cnc2cc(C(=O)NC3CC4CCC3CC4NC(=O)C=CSC)nn2c1 62104,Cc1nn(C(C)C)cc1C(=O)N(C1CC(NC(=O)C(C)(O)C2CCOCC2)C1)C 62105,O=C1NC(C(=O)NS(=O)(=O)CC(Cl)Cl)Cc2n[nH]cc21 62106,CC(C(=O)NCC1(C(N)=O)CN(C(=O)CC2CCCC(F)(F)C2)C1)S(C)(=O)=O 62107,Cc1csc2cc(CNC(=O)NC3CCC34CN(C(=O)OC(C)(C)C)C4)[nH]c12 62108,c1(C(c2cnn(C)c2)C(C)C)nc(Cc2ccccc2)nn1-c1cccc(Cl)c1 62109,Cc1cc(C)c(OC(=O)C(O)CC[S+](C)C)c(Br)c1 62110,Cc1cccc(N)c1C(=O)NCC1CCCN(C(c2csc(Cl)c2Cl)=O)C1 62111,C1(C(=O)OC)(OC)CCN(C(=O)Nc2cccc(C(F)(F)C(F)(F)F)c2)C1 62112,Cc1cccc(C)c1CCN=C(NCc1ncccc1Cl)NC1CCN(C(C)=O)C1 62113,c1(C(=O)NC23CC(NC(c4csc(C(F)F)c4)=O)(C2)C3)cc(Cl)c2n[nH]cc2c1 62114,c1(N(C)C)ccc(-c2nc(CCc3nccn3C)n(CC(C)(C)C)n2)cn1 62115,c1(C(=O)OCC)nc(=NC(C)CNC(=O)CC2CCC(O)C2)cc(C(C)(C)C)[nH]1 62116,c1(OC)cc(C(=O)NCCC(C)NC(C2CNC(=O)C2)=O)cc2c(C)c(C)[nH]c12 62117,N1(C(C(F)(F)C2(OC)CCC2)=O)CC(N(C)C(C2CC3(CC3)CO2)=O)C(F)C1 62118,c1(C(=O)OC)ccc(C(=O)NC2CC2NC(C23CCCC2C3(F)F)=O)c(C#N)c1 62119,CC1CN(C(=O)COc2ccon2)CC(C)N(C(c2cc3cccnc3[nH]2)=O)C1 62120,c1(C(=O)NC2C(C)CN(C(C3CC=CCC3)=O)C2)cn2c(n1)SCC2 62121,C#CCCCC(C)C(=O)NCCCOCCCNC(c1cc2cnccc2[nH]1)=O 62122,C12(CNC(C3N(C)CCC3)=O)CC1CN(C(=O)CCNC(=O)C=CCl)C2 62123,N#Cc1cccc(NC(=O)CC2(NS(=O)(=O)c3cn[nH]c3)CCC2)c1[N+](=O)[O-] 62124,N1(C(C(c2ccc(F)cc2)NCCC#C)=O)CCCCC1C1(CN)CC1 62125,Cn1cc(C(N2CCC(C(F)CNC(=O)CCS(C)=O)CC2)=O)c(Cl)n1 62126,c1(C(N2CCC(CC(=O)NC(c3nncn3C)C)C2)=O)cccc2cnccc12 62127,C(=O)(CCCCCC#N)NC(C)C(=O)NC(CCO)C(C)(C)C 62128,CC(C)(C)C(CC(=O)NCc1cccc(NC(=O)CC=CC(C)(C)C)c1)C(F)F 62129,Cc1ncc(Cl)c(C(=O)NC2CC23CCN(C(c2ccncn2)=O)C3)n1 62130,C1(C(=O)NC2C(NC(C3(C(=O)OCC)CC3)=O)C2)CC(=O)N(C)C(=O)N1 62131,Cc1cc(C(N2CCN(C(C3(c4ccc(O)cc4)CC3)=O)CC2C)=O)cnc1Cl 62132,Cc1cc(C)c(C(N2CC(CC(C)NC(=O)CC3SC(=N)NC3=O)C2)=O)[nH]1 62133,C1(C(N2C(CC(N3CC(C(F)(F)F)(OC)C3)=O)CC2)=O)C2CC3C(C2)C13 62134,c1(C(c2ccc(Cl)cc2)NC(c2nccc(=N)[nH]2)=O)ccc(F)c(Cl)c1 62135,C(=O)(C(C)S(C)(=O)=O)N(CC(C)CNC(=O)COc1nn(C)cc1Br)C 62136,C(=O)(CCCC(=O)NC(C1COCCO1)C1CC1)NC 62137,c1(C(=O)NC(C)(C)CCNC(=O)CCC#N)cc(C(F)F)cc(C(F)(F)F)c1 62138,c1(C(=O)NC(C(C)C)CNC(c2cccc(Cl)c2Cl)=O)nccc(C#N)c1F 62139,N1(C(COCCC=C)=O)CCC2CCN(C(=O)C(c3ncccc3C)(F)F)CC12 62140,CC(C)C(C(=O)NCCOC1CN(C(=O)C=CC2CCOC2)C1)C(C)C 62141,CCCCC(CNC(c1cncc(N)n1)=O)NC(=O)C(C(C)C)c1ccccc1 62142,C1(NC(C(C=C)O)=O)C2CC1N(C(C1(S(C)(=O)=O)CC1)=O)C2 62143,c1(C(=O)CC(F)F)cc(C(=O)NCC2CCCN(CC(F)(F)F)C2)cc(F)c1 62144,N1(C(C(CC2CCC2)OC)=O)CCOC(C)(CNC(c2ccncc2F)=O)C1 62145,c1(CNC(=O)NC2CCOCO2)ccc(N2N=CCC2=O)cc1 62146,c1(C(=O)NC(CCN(C(c2c(C)[nH]nc2Cl)=O)C)C)ccc(S(C)=O)cc1 62147,C1(CNC(c2nn(C)c(Br)c2)=O)CC2(CCC2)CN1C(=O)C(F)=C1CCC1 62148,C1(CC#C)(C(=O)NCCC(C)CCNC(c2c[nH]cc2C)=O)CCOCC1 62149,c1(CNC(C2(NC(=O)CSCC(N3CCOCC3)=O)CC2)=O)cncc(Cl)c1 62150,C(=O)(C(C)(O)C(F)(F)F)N1CCCC(CC(=O)NC(C(=O)OCC)(C)C)C1 62151,Cc1cc(C)c(C(=O)NCC2CCC(C)CN2C(c2coc(O)n2)=O)cc1N 62152,N1(C(CC(C)OC)=O)CCC(NC(=O)CSc2nnnn2CC(F)(F)F)C12CC2 62153,Cc1ccc(N)c(C(N2CC(O)(CCNC(C3CC(C)CC(=O)N3)=O)C2)=O)c1 62154,CCCC(C)(CCC)C(=O)NCCOC1CCN(C(=O)CC2CCC2(C)C)C1 62155,C#Cc1cc(C(=O)NC2CCCN(C(c3cc4c([nH]3)CCCC4)=O)C2)cc(F)c1 62156,C#CC12CC(CN1C(=O)CN1CCN(C(=O)C(C)CC(C)C)CC1)C2 62157,C(C(=O)Nn1nnc2c1CCCC2)C1N(C(Cc2c(C)n[nH]c2)=O)CC1 62158,C1(C(=O)NCC(C)N(C(=O)C=C2CCN(C)C2)CC)CCOC2(CCC2)C1 62159,c1(CNC(=O)CC2CCN(S(=O)(=O)CCCN3CCOCC3)C2)ccnc(F)c1 62160,c1(OC)cc(C=CC(N2CC(=CC(=O)O)C2)=O)sn1 62161,c1(C(N2C(C(=O)NC(CC)CC)CC(C)C2)=O)cc(OC)cc(C(F)(F)F)c1 62162,c1(OC)cc(C(=O)NC(c2ccc3c(c2)CCC3)C)nc2ccccc12 62163,C1(c2n(CC(=C)C)nnn2)(NCCCCO)CC2CCC(C1)N2CCC 62164,C1(NC(C=CCC(C)(C)NC(Cn2c(C)ncc2)=O)=O)CCSC(C)C1 62165,C1(NC(C2CN(C)C2)=O)CCN(C(c2cn(C)c(=O)cn2)=O)CC1O 62166,C1(C(=O)NCC(CC(C)C)NC(=O)C(C)n2cccn2)CC(S(C)(=O)=O)C1 62167,C1(F)(CNC(C(CC)c2ccccc2)=O)CCN(C(c2sccc2C)=O)C1 62168,N1(CCNC(c2c(CC)nccn2)=O)CCCN(C(c2cccs2)=O)CC1 62169,c1(CC(=O)OCC)ccc(NC(CNC(=O)COCCCC(C)C)CC)cc1 62170,C#CC1CCCN(S(=O)(=O)Cc2ccc(C(N3CC(C(=O)OC)C(F)C3)=O)cc2)C1 62171,c1(C(N(C2CCN(C(=O)CN(C)S(=O)(=O)N(C)C)CC2)C)=O)cc(F)ccc1O 62172,N1(C(C2C(C=C)OCC2)=O)CC(CNC(=O)CCc2cnc[nH]2)CC1(C)C 62173,c1(C(C(=O)NC)N(C(c2ccccc2F)C(C)C)C)cc(Cl)c2c(c1)OCCO2 62174,c1(C(C)=O)ccc(C(=O)NCCCC(C)NC(c2cc(-c3ccco3)no2)=O)o1 62175,N1(C(C2(C(=O)NC)CC2)=O)CC(CCNC(c2c(SC)cnn2C)=O)C(C)C1 62176,c1(C(N(CCC(F)(F)F)C(=O)C2CC2)=O)cccnc1SCC(=O)NCC 62177,C1(OC)CCCCN(CC(N2CC=CC23CCCC3)=O)C1=O.C(CO)N 62178,C(N=c1cc(-c2ccccc2)nc[nH]1)C1CCCC(NC(=O)COCC(F)F)C1 62179,c1(C(=O)NC2(CNC(c3c(C(C)C)cco3)=O)CCCC2)ccnn(C)c1=O 62180,CCCC(CNC(c1cn(C2CCOC2)cn1)=O)NC(C12CSCC1C2)=O 62181,c1(N(S(CCC(=O)OC)(=O)=O)C2CCNCC2(C)C)ncc(C#N)c(OC)n1 62182,Cc1cc(S(=O)(=O)NN2CCC(C(C)(C)F)C2)ccc1OCC(=O)O 62183,N1(C(c2cccc(-c3ccccc3)n2)=O)CC2CC1CN2C(C1CCOC1)=O 62184,C1(NC(C2CC(C)CN2C(c2ccc(C#N)o2)=O)=O)CC(C)N(C)CC1C 62185,CC(CCN=c1[nH]cnc2cc(F)c(F)cc12)NC(c1cc2ccccc2o1)=O 62186,CC1CCN(C(=O)Cc2cnccn2)C(C)C1NC(=O)CCCC1CCCCC1 62187,N1(C(C(=O)NC2CCOC2)C2C(C)C2)CCC(CC(N2CCCCCC2)=O)CC1 62188,C(CC(C(C)(C)C)NC(C1CCC(C)(C)C1)=O)N(C(C1(CCCC)CC1)=O)C 62189,c1(NC(=O)Nc2ccc(C(N(CC)CC)=O)cc2)cc(C)c2c[nH]nc2c1 62190,C(=O)(C(C)C(C)(C)C)N(C)CC1(NC(CC(=O)OCCC(C)C)=O)CC1 62191,N1(C(C(C(C)C)C)=O)CCN(C(c2ccc([N+](=O)[O-])s2)=O)CC(CO)C1 62192,C#Cc1ccc(C)c(NC(C2CC(C)(NC(=O)CC3CCC(=O)N3C)C2)=O)c1 62193,CC1CN(C)C(C)CC1NC(C1C(NC(=O)COCCF)C1(C)C)=O 62194,c1(C(N(C2CN(C(c3ncoc3C(C)(C)C)=O)C2)C)=O)cc2sccc2n1C 62195,Cc1[nH]nc(C(N2CCOCC2CN(C(=O)C(F)(F)c2nccn2C)C)=O)c1N 62196,C12(C(=O)NCC3(C(N4CCC(C(=O)OCC)C4)=O)CCCO3)CCN(CC1)CC2 62197,c1(NCCN(CCN(C)C)CC)ccc(S(=O)(=O)N(C)C2CC2)cc1C#N 62198,c1(C(=O)NC2(C(N)=O)CN(C(=O)CC3CC3)C2)sc(Cl)cc1Cl 62199,c1(C(=O)NCCN(C(c2ncc(C)c(Cl)c2)=O)C2CC2)cc2n(c1)CCSC2 62200,c1(C(=O)NCC2(CN(C(c3ccc(C)s3)=O)C)CC2)ccc(Cl)nc1N 62201,c1(CCC(=O)NC2CN(C(=O)C(O)CC3CC3)CCC2O)nc2ccccc2o1 62202,C1(NC(CCc2nc(C)sc2)=O)CCC(NC(C2C3COCC23)=O)CC1 62203,C1(C(=O)NC(C#C)C)(NC(=O)C(COC)N(C)C)CC1(C)C 62204,C1(CNC(c2cc(C)sn2)=O)CC2CCC1N2C(=O)CCCCc1cnc[nH]1 62205,C1(NC(=O)C(F)CC2CC2)CC(Nc2cc(O)ncn2)C12CCC2 62206,C1(C(=O)NC2(c3ccc(C(C)C)cc3)CC2C)COC2(CCC2)C1N 62207,C1(c2nnnn2CC2CCCO2)(NCc2nc(C)sc2)CCCCCC1F 62208,N1(C(C)C)CC(c2nnnn2C2CC2)(NCc2nc(C(F)F)n[nH]2)CCC1=O 62209,C1(C(N(C)CCNC(=O)CNC(N)=O)=O)CNC(=O)CC1(C)C 62210,C1(CNC(C(F)=CC)=O)CCCC1NC(c1cc(C(=O)NC)[nH]n1)=O 62211,C1(CNC(C(CC)CC)=O)CCN(C(C2CC3CC(=O)C2O3)=O)C12CCC2 62212,C(=O)(C(O)C(C)(C)C)NCC(C)(C(C)C)NC(C1(C(=O)OCC)CCC1)=O 62213,C(=O)(CCCC(C)C)NCCCCC1CN(C(C=C(C)C)=O)C1 62214,c1(CC)ccc(C(=O)NC2CC(N(C(=O)CCOC3CCOC3)C)C2)c(Cl)c1 62215,CC(C)(C)CC(=O)NCCCOCCC(N1CCC(CCC(N)=O)CC1)=O 62216,C(CCCOC)(C(=O)Nc1cc(F)ccc1OCC)NC(c1c(CC)[nH]cc1)=O 62217,N1(C(CCn2c(C)ncc2)=O)CCC2(CCCC2NC(=O)Cc2n[nH]c(=N)s2)C1 62218,CN1CCCC(NC(c2cn(CCNc3cncc(N4CCCC4)n3)nc2)=O)C1 62219,C(=O)(CCCC(C)(C)C#N)NCC(C)(C)NC(Cc1cc(OC)cc(OC)c1)=O 62220,N1(C(CSCC)=O)CC2COCCC2(NC(=O)CC(n2nc(C)cc2C)C)C1 62221,n1(CC(=O)NCC2C3N(C(C(COC)O)=O)C(CC3)C2)nc2ccccn2c1=O 62222,C1(C(=O)NC(C)(C)C=CC(=O)NC(C2CCOC2)CO)C2CCC(F)C12 62223,N1(C(COc2c(OC)cccc2)=O)CCC2(CCCN2C(=O)CCC2CC2)CC1 62224,c1(C(=O)NCC2N(C(C(C)c3cccs3)=O)CC2)cc(NC2CC2)ncc1Cl 62225,c1(CC)cc(C(=O)NC2C3CC2N(C(c2oc(C)nc2C)=O)C3)ccc1C 62226,CCC(CNC(=O)CC(C)CNC(c1nccnc1C(N)=O)=O)(CC)OC 62227,c1(CC)cc(C(=O)NCC(O)CNC(c2cnc(C(C)(C)C)o2)=O)nn1C 62228,N1(C(C(C)CF)=O)CCCC(N2CCN(C(c3n[nH]c(=N)s3)=O)CC2)C1 62229,c1(C(=O)NC2CC(NC(c3c(CC(N)=O)occ3)=O)C2)nc2n(c1Cl)CCCC2 62230,c1(C(=O)NC(CNC(C(C)C2CCCC2)=O)(C)CO)cc2c(s1)CC(C)(C)C2 62231,n1(CC)nc(C(=O)NC(C2CCN(C(C3CCCCS3)=O)CC2)C(C)C)cc1C 62232,c1(NC2(C)CC(C(=O)NC)C2)nc(NC(=O)OC(C)(C)C)ccn1 62233,C1(NC(c2c(CC)noc2)=O)CCN(C(c2ccccc2C(C)(C)C)=O)CC1C 62234,N1(C(c2ccnn2CC(F)F)=O)CCC(Nc2cccc(C(F)(F)F)c2)CC1 62235,c1(C(N2CC(CC)C(NC(c3nccn3C)=O)C2)=O)cc(C)nc(C)n1 62236,c1(CC(=O)NC(CC)CNC(C2CCCN2C)=O)ccccc1OC 62237,C(=O)(CCCC(=O)NCCCCNC(c1ccccc1N1CCCC1)=O)OCC 62238,C1(NC(C(CC=C)(C)O)=O)CCCC2CN(C(=O)C(O)C(F)(F)F)CC12 62239,CCN=C(NCCC1(C)CC1(F)F)N1CCc2c(Br)cccc2C1 62240,C1(O)(C(C)NC(=O)CC(C)c2ccco2)CCN(C(c2ccc[nH]2)=O)CC1 62241,c1(C(N(CC(C)CO)C)=O)coc(CNC(C2(O)CCOC2)=O)n1 62242,c1(NC)c(C(=O)NCC2CN(C(C3CC4CCCC34)=O)C2)cccc1N 62243,C(=O)(C(C)CCC(C)(C)C)N1C2CC(C(=O)NCc3c(C)noc3C)C1CC2 62244,C1(C)(CNC(C2N(CC)CC2)=O)CC(OC)CN1C(=O)CC(C)n1cccn1 62245,C1(NC(=O)C(O)Cc2ccccc2)CC2CC1CN(C(C1CCC3(CC3)C1)=O)C2 62246,C12(NC(COC3CN(C(C(C)OCC4CC4)=O)C3)=O)CCCN(CCC1)C2 62247,N1(C(C=C2CCN(C)CC2)=O)CCCN(C(c2ccc(Cl)nc2N)=O)CC1 62248,CN1CC(C)(C(=O)NCC2CC(NC(c3ccn(C4CC4)n3)=O)C2)CC1=O 62249,C1(NC(CCCCSC)=O)COC2(CCN(C(=O)Cn3ccc([N+](=O)[O-])n3)C2)C1 62250,c1(OCC)ccccc1OC(C)C(=O)N(C(C)C(C)=O)C 62251,N1(C(CN(CCC#C)C)=O)CCCC(F)(C(N2CCS(=O)C(C)C2)=O)C1 62252,c1(C(C(=O)NCCCCCC)N(C(C#N)C2(COC)CC2)C)cccc2c1CCO2 62253,c1(C(=O)NCC(CC)NC(c2ccon2)=O)ccc(Cc2nc[nH]n2)cc1 62254,Cc1cc(N)cnc1C(N1CC(CC(F)C(=O)NCC(CC(C)C)CF)C1)=O 62255,c1(C(=O)NC2CC(NS(=O)(=O)c3cccnc3)C2)cc(Cl)nc(Cl)c1F 62256,c1(CC(N2CCC(CC=C)(C(=O)O)C2)=O)c(Br)ccc(Cl)c1F 62257,n1(CC(=O)NCc2onc(-c3cccc(C)c3)n2)c(C(C)C)nc2ccccc12 62258,C1(CC)CC(C)CN(C(C2(C)CCCN2Cc2ccc(OC(C)C)cc2)=O)C1 62259,C1(C(=O)NC(C2CN(c3cnc(F)cn3)C2)C)CCC(N(C)C)CC1 62260,n1(CCC(=O)NCCCC2(NC(C(C)C#N)=O)CC2)cnc2sccc2c1=O 62261,c1(NC(=O)CC2CN(C(C3CN(C(C)(C)C)CCO3)=O)C2)ncc(Cl)nc1Cl 62262,C1(NC(C(CC)(C)O)=O)COC2(C1)CN(C(=O)C1=CCCOCC1)C2 62263,N1(C(CCc2n(C)ccn2)=O)CC2CC(NC(C3CCCC(C)(C)C3)=O)CC1C2 62264,C1(NC(C=CC(C)NC(c2n(CCC)ncc2)=O)=O)CCN(C)CC1C 62265,N1(C(C2CCCN(CCC)C2)=O)CCN(C(=O)C(C)S(N)(=O)=O)CC(C)(F)C1 62266,c1(C(=O)NC(C(C)NC(COc2c(F)ccc(C)c2)=O)C)cccc2scnc12 62267,c1(C(=O)NCC2N(C(c3cc(SC)oc3)=O)CCCC2C)n[nH]c2c1CSCC2 62268,CC1CCCC(C(N2CC3C(CNC(=O)C=Cc4cnn(C)c4)C3C2)=O)C1 62269,Cc1ccc([N+](=O)[O-])c(C(=O)NCC2CC3CCC2N(C(C2CCOC2)=O)C3)c1 62270,CC1CC(=O)NC(C(=O)NCc2cccc(NC(=O)C(F)(F)c3cncs3)c2)C1 62271,N1(C(CCC#CC)=O)CCCCC2(CCN(C(=O)C3=C(C)CCCC3)C2)C1 62272,CC(O)CCN=c1[nH]c(N2CCC(N3CCOC3=O)C2)nc2c1COC2 62273,c1(-c2ncc(NC(=O)C(F)(F)F)s2)ccccc1-n1cncn1 62274,c1(-n2c(C(CCCOC)C)nc(-c3ccc(F)cc3)n2)cc(F)c(F)cc1OC 62275,C12(CCN3CCN(C(c4ccc(OC)cn4)=O)CC3)CCC(CC1)C2(C)C 62276,c1(CCC(=O)N(CC(CC)NC(=O)C(C)Cc2cccnc2)C)c(C)noc1C 62277,C1(C(=O)NCC(CC=C)NC(=O)CC)C(C)(C)CCCC1(C)C 62278,Cc1nc(C(=O)NC2(C(N3CCC(CCF)CC3)=O)CCCC2C)c(C)o1 62279,C1(OC)CCC(CC(=O)NCC2(C)CCCN2C(c2occc2C)=O)CC1 62280,C(C(O)C(F)(F)F)NC(c1cncc(OCCN2CCCCC2)c1)=O 62281,N1(CC(C)NC(N)=O)CCN(C)C(=O)C1.N12CC(C1)C2=O 62282,C1(CC(=O)NC2CN(C(C(C)OCC3CCCO3)=O)C2)COCCOC1 62283,c1(C(c2nnnn2C)NC2(CO)CC(OC)C2)ccc(N2CCC2)cc1 62284,N1(C(C2(C)C(C)C2)=O)CC(NC(c2csc(-c3ccco3)n2)=O)C(O)C1 62285,C1(CNC(Cn2c(C(C)C)ncc2)=O)CN(C(=O)Cn2nnc(=O)[nH]2)CCCO1 62286,CC1CC2(CCN(C(=O)CCC3CC3)CC2)CN1C(c1ccc(S(C)=O)cc1)=O 62287,C=CC(C)(CCOC)C(=O)NC1CCN(C(=O)CCC(C)(C)OC)CC1CO 62288,c1(CNC(CC(=C=C)C)=O)cc2n(n1)CCN(C(c1c(C)cc(Cl)cc1N)=O)C2 62289,CC1(CNC(=O)C(C#N)C2CC2)CCCN1C(c1cnc(Br)s1)=O 62290,c1(C(=O)OC)sc2ccncc2c1NC(C1(CNC(c2cccnc2)=O)CC1)=O 62291,Cc1ccc(C(=O)NC(C)CCN(C(=O)CCc2cnn(C)c2)C)nc1 62292,N1(C(CCSC)=O)CCC2C(CCN2C(c2ccc(C(C)(C)C)[nH]2)=O)C1 62293,C1(NC(CC)=O)(CNC(=O)CNc2nc(C)cs2)CCCCC1C 62294,c1(NC(C2N(C(CC(C=C)(C)C)=O)C3(CC2)CC3)=O)cccc([N+](=O)[O-])c1 62295,C1(C(=O)NCCN(C(=O)C=CCO)CC)CCCC1N(C)C 62296,OCC(F)(F)CCN=C(NCC1CCC1)N1CCOC(C(F)(F)F)C1 62297,Cc1cc(Cl)ncc1NC(=O)C(C)C(C)NC(c1ccn(CCF)n1)=O 62298,C1(C(N2CCOCC2)=O)CC(C2CC2)C1.CC(C(F)F)=CC(=O)NC 62299,Cc1cc(=O)oc(C)c1C(=O)NC1CC1NC(c1cnc2n1CCCC2)=O 62300,C=CC(CCC)CC(=O)N1CCCC1CNC(c1cc2n(n1)CC(F)C2)=O 62301,Cc1nc(N(C)C)sc1C(N1CCC(C)C1CN(C(C12CC(C1)C2)=O)C1CC1)=O 62302,CCCCN=C(NCCc1cccc(F)c1F)NC1CN(C2CC2)C1 62303,C1(CNC(C2(CC#C)CCOC2)=O)CC2CCC1N2C(=O)C(C)(CC)CC 62304,C1(CC(=O)NC(CC(C)C)CNC(=O)COCC2CCCC2)CCCNC(=O)C1 62305,CCCC(C(=O)OC)C(=O)N1CC(C2(NC(C3CCS(=O)(=O)C3)=O)CC2)C1 62306,c1(N(CCCCO)CC)nnc(C2CCOC2)n1CC1CC=CCC1 62307,Cc1nc(C=CC(=O)NCC2(C)CC(NC(C3CCC3)=O)C2)[nH]c1C 62308,c1(CC)cc2c(N(C(C)CCNC(C34CCC(CC3)C4)=O)C)nc(C)nc2s1 62309,C#Cc1ccc(F)cc1C(=O)NC1C=CCN(C(c2ccc(F)cc2C#N)=O)C1 62310,N1(C(CC(C)(C)CNC(=O)C=CCN2CCCC2)=O)CCC(C2(O)CC2)CC1 62311,N1(C(=O)NCc2c(CSC)cc(F)cc2)CC(C)(C)C(O)C1(C)C 62312,C1(C)(C(=O)NCC(C)(C(C)C)NC(C(CCC)=CCC)=O)CCCCC1(F)F 62313,c1(N(CC(CN(C(C2N(CC#C)CCC2)=O)C)O)C)cc(C)c(C#N)cn1 62314,N1(C(CCC)=O)CCC(C(C)(C)OC(C2CCOCC2)C(=O)NC)C1 62315,C1(NC(c2c(O)ncc(C(C)C)c2)=O)CCC2CCN(C(=O)C=CCO)C1C2 62316,CCC(CC)C(=O)N(C)CC1CCN(C(c2cnn(CC3CCOC3)c2)=O)CC1 62317,N1(C(C=Cc2occ(C)n2)=O)CC2CN(C(=O)COC(F)F)CCC2(CO)C1 62318,C(C1CCC(c2nnnn2C(C)C)(Nc2cccc(F)c2)C1)=CC(=O)OC 62319,C(CCC(=O)NCCCOCCC(=O)NC(CN1CCC1)CC)=CC 62320,c1(C(N2C(C(=O)Nc3c(Br)ncc(OC)c3)CC(F)C2)=O)ccc(C#N)cc1O 62321,C(=O)(N=c1cccn[nH]1)C1(C)CCN(C(CC)=O)C1 62322,c1(NC(=O)NCCOc2ncccc2Cl)ccc2c(c1)CCOC2 62323,C1(C(=O)NCCN(c2ccn(C(C)C)c2C)CC)CN(CCOC)CCC1(F)F 62324,N1(CCOC)C(=O)NC2CN(C(=O)C(CN)CC(C)(C)C)CCC12 62325,N1(C(C(N2CCCCC2=O)C)=O)CC2CCC1C(CNC(=O)CO)C2 62326,N1(C(CC2(OCC)CC2)=O)CCCC1CN(C(=O)Cn1ccnc1C)C 62327,S(=O)(=O)(c1ccc2occc2c1)NC(C(OC)OC)C 62328,N1(C(c2c(COC)n(C)nc2)=O)CCC2(NC(=O)CCCC3CCC3)CC2C1 62329,CC1CCCN(c2ccc(Cl)cc2)N1C(=O)c1cc2ccc(F)cc2o1 62330,c1(C2CCN(C(c3[nH]nc(NC(=O)NC4CC4)n3)=O)C2)cc(Br)ccn1 62331,c1(C(N2C(CN(C(c3c(COC)nc[nH]3)=O)C)CCC2)=O)cnc(C(F)F)nc1 62332,C1(NC(C(CSCc2ccccc2)NC(C)=O)=O)CC2CCC1N(C(C)=O)C2 62333,c1(CC(=O)N(CCCNC(=O)CCN(C)CCO)CC)csc2ccc(Cl)cc12 62334,C(CC(CNC(=O)C(C1CC1)OCC)OC)NC(COCC#C)=O 62335,c1(C(=O)NCC(C)NC(C(C(CC)C)OC)=O)c(Cl)cc(CO)cc1Cl 62336,C(=O)(CCCCC(F)(F)F)NCC12CCC(NC(CC3(C)CCC3)=O)(C1)CO2 62337,CCCC(C(O)C(=O)Nc1ccc(O)c(OC)c1)NC(C1(COC)C=CCC1)=O 62338,n1(CC)c(C)nn(CC(=O)NCCCNC(c2ccc(C(N)=O)cc2)=O)c1=O 62339,C(=O)(C(F)(F)C(F)F)NCC1CN(C(c2c(CC)nns2)=O)C(C)C1 62340,CCC(CN1CC(=O)N(CC(C)CSC)C1=O)(CC)C(=O)OC 62341,N#Cc1c(CNC(N2CCC3CCCC23C(=O)OC(C)(C)C)=O)cccc1F 62342,Cc1nc2sc(C(N3CC(CNC(=O)C(C)N4CCC4)C3)=O)cn2c1Br 62343,C1(O)(N(C)CCNC(=O)C(C2(O)CN(C(=O)C3CC3)C2)F)CCSCC1 62344,C1(NC(=O)CCC2CC2(F)F)CCN(C(c2ccnnc2O)=O)CC12CCC2 62345,CC(C)CC(CC(=O)NC1(CO)CCC(C)C1)NC(C1CC2(CCC2)C1)=O 62346,c1(C(C)(C)C(=O)NC(CNC(=O)CC2CC=CCC2)CO)ccc2c(c1)OCO2 62347,CC1CCC(OCCNC(=O)C(O)C(C)c2ccccc2F)CC1 62348,c1(OC)ccc(C(=O)N(C)CCNC(C2(C)CCCC2(F)F)=O)c(N)c1F 62349,C1(CNC(C2CC(C)C(C)CC2)=O)C(C2CC2)CCN1C(c1cnc(N)cn1)=O 62350,c1(C(=O)NC2(C(=O)NCC(C3CC3)SC)CC(CO)C2)cc(Cl)cn1C 62351,N1(C(=O)CCOC2CC2)CCCN(C(C2(C(F)(F)F)CC3CC3C2)=O)CC1 62352,c1(CC(C)N(C(c2ncccc2C)C(=O)NCC)C2CC2)ccc(C)cc1 62353,N1(C(C=CCOC)=O)CCC2(NC(c3cc(CCO)on3)=O)CC2C1 62354,c1(N(CCCC)C)nc2ccccc2c(=NC2CCc3ncccc3C2)[nH]1 62355,N1(C(=O)COc2ccc(-n3ccnn3)cc2)CC2CCC1CO2 62356,C1(CCC)C(C)CCCN1CCCOc1cccc(C(F)(F)F)c1 62357,C1(CNC(CNC(CNC(=O)NC)=O)=O)C2CCCCC12 62358,CC(C)S(=O)(=O)C(C)C(=O)NC1(C)CC(NC(c2cc3c(nc2O)CCC3)=O)C1 62359,c1(C(=O)NC(C2CCN(C(C(COC)NC(C)=O)=O)C2)C)cc2oc(Cl)cc2[nH]1 62360,C1(C)(CC(=O)NCC(C(=O)NC(C)Cc2cnn(C)c2)O)CCCCC1 62361,c1(CC)cc(F)ccc1C(=O)NCCCCCCNC(=O)C=CCCCN=[N+]=[N-] 62362,C1(CNC(c2ccc(CSC)o2)=O)CN(C(=O)C(C)C2CC2)C2(CCC2)C1 62363,c1(NC(C2(O)CCN(C(=O)CC3C=CCCC3)C2)=O)cnc(Br)c(Cl)n1 62364,C1(CNC(C2(C3N(C(CNS(CC)(=O)=O)=O)CCC3)CC2)=O)C(C)(C)C1(F)F 62365,c1(OCCN)ccc(Cl)cc1.C(C(F)(F)F)OCCNC(=O)CNC(C1CNC1)=O 62366,C1(C2CCC2)(CNC(COC2CN(C(C(C)(C)OCCC)=O)C2)=O)CC1 62367,n1(CC(=O)NC2(COC)CN(C(=O)C(C)(C)F)C2)ccc(C)cc1=O 62368,c1(N2CCC(C3(NC(CC(C=C)(C)C)=O)CC3)CC2)cc2c(cn1)C(=O)CCC2 62369,c1(C(N(CCCCN(C(C(C)C2CCOC2)=O)C)C)=O)ncccc1N 62370,c1(-c2cn(CC(N3CCC(c4ccc(F)cc4)C3)=O)nn2)cc(F)c(F)c(F)c1 62371,Cc1cc(F)c(CC(=O)NCCCCCCNC(C2COCCC2C)=O)cc1F 62372,c1(CC(=O)NCC2(OC)CN(C(C=NOC)=O)C2)sc(C)cc1C 62373,c1(OC(COC)C)cc([N+](=O)[O-])ccc1C(=O)Nc1ccccc1-c1nn[nH]n1 62374,C1(CC)CN(C(=O)CCCC(=O)OC(C)(C)C)CCN1C(C1CCC1OC)=O 62375,c1(C(N(C(c2cn(C3CC(O)C3)nn2)(C)C)C)=O)ccnc(C(N)=O)c1 62376,CCC(CC(=O)NCCn1cc(C(=O)Nc2ccc(C)c(O)c2)nn1)C(C)C 62377,N(C1CS(=O)(=O)N(C)c2ccccc21)C(=O)NC(c1cccnc1)CC 62378,Cc1[nH]c2ccccc2c1NC(=O)Cc1ccc(CCC(=O)O)cc1C 62379,CC1(C)CC(C(N2CC=CC2CNC(=O)C=C2CCCCC2)=O)CCO1 62380,N1(C(CCCCSC)=O)CC(CNC(=O)C(C(C)(C)C)SC)C2(CC2)C1 62381,Cc1c(Cl)ccc(C(=O)NCC2CCN(Cc3ccnc(Cl)c3)CC2)c1F 62382,c1(C(=O)NC(C)CNC(=O)C(C)n2cncn2)cccc2c1OCCN2 62383,c1(C(=O)NC2C(CNC(c3ccccc3O)=O)CC2)ccc2nc(CO)[nH]c2c1 62384,C1(NC(C2CCCCO2)=O)CCN(C(=O)Cc2ccccc2Cl)C12CCCC2 62385,C1(C(N2CC(NC(c3c(C)cn(C)n3)=O)C(C)C2)=O)CC2CCC(C1)C2 62386,C(C1c2ccccc2CN1C(=O)OC(C)(C)C)N(C)C(C1(CCO)CN(C)C1)=O 62387,N1(C(C(F)=CCC)=O)CC(NC(c2c(OC)noc2C2CC2)=O)C(F)C1 62388,N1(C(CC(=O)NC2CC2)=O)CCc2nc(S)[nH]c2C1 62389,c1(SC)ncc(C(N2CCN(C(c3cnc(=N)[nH]c3)=O)C(CF)C2)=O)c(O)n1 62390,N1(C(C#CC(C)C)=O)CC2COCCC2(NC(c2nccnc2N)=O)C1 62391,C1(CNC(c2cccc(Cl)c2C(F)(F)F)=O)CC2CCC1N2C(c1ccoc1)=O 62392,CC(C)C(O)C(=O)N1CC(NC(=O)C=CC2CC2)C(c2ccccc2F)C1 62393,Cc1cc(C(=O)NCC(C)(C)CNC(=O)C(O)Cc2ccc(F)cc2)cc(C)c1 62394,C(=O)(C(C)(C)CCCF)NCC1CC(NC(C(c2n(C)ncc2)O)=O)C1 62395,C1(CCNC(C(C)SC)=O)CCN(C(=O)CSCC(C)C)C1 62396,c1(C(N2CCN(C(C(CC#C)O)=O)C(CO)C2)=O)cnc2c(cnn2C)c1O 62397,C1(NC(CNS(CC)(=O)=O)=O)CN(C(=O)C(CC)SC(C)C)Cc2nccn2C1 62398,CC1(C(=O)NC2CCC(NC(=O)CCc3nc(=N)[nH][nH]3)C2)CCC(=O)NC1 62399,c1(NC(C)=O)ccc(C(=O)NCC23CC2CN(C(c2cscc2C)=O)C3)c(Cl)c1 62400,Cc1ccc(C(=O)NCCC(C)NC(c2cnc(C(N)=O)s2)=O)c(N)c1F 62401,CC(CCCCNC(C1CCC(N(C)C)C1)=O)NC(C1CC1c1cnc[nH]1)=O 62402,CCCCS(=O)(=O)CC(=O)N1CCC(NC(c2n[nH]c(CC)c2F)=O)C1(C)C 62403,CC1(NC(=O)CC23CC(C2)C3)CCN(C(c2ccc(N3CCC3)nc2)=O)C1 62404,C(=O)(C(C)CCC(C)(C)C)NC(CC)(CNC(c1sccc1COC)=O)CC 62405,N1(C(C2CCCN(CCC)C2)=O)CC(CNC(=O)CCc2ccco2)C(C)(C)C1 62406,c1(NC(C23CC(C2)C(C(F)(F)F)O3)=O)ccccc1-n1ccccc1=O 62407,CN=c1nc(N2CCOC(C)CC2)[nH]c(=NCC2(c3cccs3)CCOCC2)[nH]1 62408,c1(OC)cc(C2CC2)ccc1C(=O)NC1(C)CC(NC(=O)Cc2ccon2)C1 62409,Cc1nn(CO)cc1C(=O)N(C)CCN(C)C(C1(Cc2cnn[nH]2)CCCC1)=O 62410,C1(C(=O)Nc2ncc(NCC(C)O)nc2)CC12CCN(C(=O)OC(C)(C)C)C2 62411,Cc1nc(=NC(=O)CC2CN(Cc3cccc(N4CCOCC4)c3)CCO2)s[nH]1 62412,Cn1ccnc1C(F)(F)C(=O)NC(CNC(C1(C2CCCO2)CC1)=O)CO 62413,c1(C(=O)NCCN(C(=O)C(C)=C2CC2)CCC)cc(C2CCCO2)n(C)n1 62414,C1(c2onc(-c3ccc(SCC)cc3)n2)COCC1S(=O)CCC(=O)N(C)CCN 62415,N1(C(c2ccc(C)c(C)c2)=O)CC(C2CN(C(c3cscc3C(F)(F)F)=O)C2)C1 62416,C1(C2CCN(N3CCC(S(=O)(=O)c4ccc(F)cc4)C3)CC2)(C(=O)OC)CCC1 62417,C1(C(N(C2CCSC2)C)=O)CSCN1C(C1(CO)CC1)=O 62418,c1(C(=O)NC2CC(CCNC(CN(C3CC3)CC)=O)C2)ccc2c(c1)ncn2C 62419,C1(CC(=O)NCC(C)(C2CC2)NC(=O)CCCC2CCCO2)CNC(=O)O1 62420,C1(C(=O)NC(CCC)(C)CC)N(C(c2cccc(F)c2F)=O)CC12CCCC2 62421,CCC(C)(C)CCCC(=O)NCCCCNC(C1CCCCO1)=O 62422,CN(C)NC(=O)CCC(=O)NCC12CC(NC(C3CC4C=CC3CC4)=O)(CO1)C2 62423,Cc1cnc(CC(=O)N(CCNC(=O)C(F)(Cl)c2ccccc2)CC2CC2)s1 62424,Cc1cc(C(N2CCC(NC(=O)Cc3ccco3)C23CC3)=O)cc([N+](=O)[O-])c1Cl 62425,N1(C(C2CCCN(C(=O)OCC)CC2)=O)CC2CCN(C)C2C1 62426,CC1CCC(NC(C2(C(=O)NC(N)=O)CC2)=O)CN1C(=O)CNc1ccccc1 62427,c1(N(CC(COC)(F)F)C)nc(NC2CC2F)c2c(n1)c(C)nn2C 62428,Cc1ccc(C(F)(F)F)cc1C(N1CC2CC1CC2CNC(=O)CCC#N)=O 62429,C1(NC(C2C(C)(C)C2(C)C)=O)CCC2CCN(C(c3cc(CCO)on3)=O)C1C2 62430,O=NN1CCCCC1C(=O)NCCc1ccc(CNC(=O)Cn2ccnn2)cc1 62431,N1(C(C(c2ccnn2C)NC(C(C)CC#N)=O)=O)CCC12CCCOCC2 62432,C1(C(F)(F)F)(C(=O)NC2C(NC(COCCN(C)C)=O)CC2)CC=CC1 62433,C1(C(=O)NCCC2N(C(Cc3c(C)nccc3)=O)CCSC2)CCn2cncc2C1 62434,C1(OC)CC(C)CN(C(C2CN(C(=O)CC3NC(=O)NC3=O)CCO2)=O)C1 62435,Cc1[nH]c2ccc(Cl)cc2c1C(N1CC(NC(C2CC=CC2)=O)CC(O)C1)=O 62436,N1(C(c2c(OC)nccc2)=O)CCC2CN(C(C3CCCCO3)=O)CC2C1 62437,CCCCC(CC)C(C(=O)Nc1ccc(F)cc1)N1CCCC1C1CCOCC1 62438,Cc1nc(Br)sc1C(=O)NC1CC(CNC(C2CCOC2)=O)C1 62439,C1(O)(CN(C(=O)C(O)CC2CCCC2)C)CCN(C(C2(C)CSC2)=O)C1 62440,N1(C(C2C(C)(NC(C=CC(=O)N(C)C)=O)CCCC2)=O)CCOC2(CCCC2)C1 62441,S(=O)(=O)(c1c(Cl)cc(Cl)cc1Cl)N1C(C(N=c2nc(C)[nH]s2)=O)CC(F)(F)C1 62442,C1(C(=O)NC(C(C)(C)C)CNC(=O)C=CSc2ccccc2)CCC2CC1CO2 62443,Cc1nsc2ncc(C(N3CC(CCNC(c4ccoc4)=O)C3)=O)cc12 62444,N1(C(C=CC(C)C)=O)CCC2(CCC2CNC(=O)CCNC(=O)C=CCl)CC1 62445,C1(NC(=O)CCF)CCCN(C(C2(C(=O)NCC3CC3)CCC2)=O)CC1F 62446,C1(CNC(c2ccc(CC)nc2C)=O)CC2COCC2N1C(c1nccn1C)=O 62447,C1(N(C(C2CC(CCC)C2)=O)CCNC(=O)C(C)c2ncco2)CCCCC1 62448,C1(C(=O)NCCC(=C)C)CC(F)(F)CN1C(c1ncsc1C)=O 62449,c1(C(N(CC(CC)NC(c2ccnnc2)=O)C)=O)ccc(C2CC2)o1 62450,C(=O)(C1=COCCC1)NCC(C(C)C)NC(C1(O)CCSC1)=O 62451,N1(C(=O)NCCCCl)CC2CC1CN2C(=O)Nc1ncccc1C(F)(F)F 62452,c1(NC(c2nnnn2C2CCNCC2)CCC)cc(=O)oc2cc(C)ccc12 62453,C1(C(N2CC(OCCNC(C3CC3(C)C)=O)C2)=O)(CC)CCOC1 62454,C=C(C)C(C)(O)C(=O)NCCN(C(c1ccc(N(C)C(C)=O)cc1)=O)CC 62455,C1(C(N2CC(CCC)C(OC)C2)=O)NCCOC1(C)C 62456,c1(C(=O)NC(CCNC(C(C)CO)=O)Cc2ccccc2)ncn2cccnc12 62457,CC1(CCC(=O)NCCOc2ccncc2)CN(C(c2cnco2)=O)C1 62458,c1(OC)c(C(=O)NCC(C)(C2CCC2)NC(c2ccc(CO)s2)=O)csc1C 62459,C1(CC(=O)N(CCC(=O)NCc2csc(COC)n2)CC=C)CC2(CC2)CO1 62460,N1(C(c2n[nH]c(C)c2Br)=O)CC2CCC2(CCNC(C2(C#N)CC2)=O)C1 62461,Cn1nc(C(N2CCCC(C(=O)NCC34CCC(CC3)OC4)C2)=O)cc1C#N 62462,C1(c2cn(Cc3c(C)cn(C)n3)nn2)CCN(C(=O)CCC(N)=O)C12CC2 62463,C1(C(=O)NC(C)Cn2cccn2)C=CCN(C(C2CCCC(=O)C2)=O)C1 62464,Cc1[nH]nc(C(F)F)c1C(N1CCCC1Cn1cc(CNC(=O)N(C)C)nn1)=O 62465,N1(C(C2(C)COC2)=O)CCN(C(C2CCCC2n2cccc2)=O)C(CC(F)F)C1 62466,c1(CC(=O)N(C)CCN(C)C(c2cocn2)=O)cccc2nonc12 62467,C(=O)(C1CCCc2nn[nH]c21)N1CC(O)(CCNC(c2nc(C)nc(O)c2)=O)C1 62468,N1(CC#N)CCN(C(=O)C(c2ccc(SC(F)(F)F)cc2)=O)CC1=O 62469,C1(CNC(C(C2CN(C(C3(C)C=CCCC3)=O)C2)OC)=O)CCCC(=O)C1 62470,N1(C(COCCOCC)=O)CC2(C1)CN(C(C1CCCS1(=O)=O)=O)CC(C)(C)O2 62471,CCCC(O)CC(=O)N1CCN(C(C2(c3ccccc3)CC2(F)F)=O)CC1 62472,CC(C(F)(F)C(F)(F)F)=CC(=O)NCC1C2CN(c3ccnc(Cl)n3)CC12 62473,C1(C(=O)NC(C2CCOC2)C#C)CN(C(=O)CCS(C)(=O)=O)CC(C)O1 62474,C1(C)(C(N2CC(CCCC)N(C(c3n[nH]cc3F)=O)CC2)=O)CCCNS1(=O)=O 62475,N1(C(CSCC#N)=O)CC(NC(C2CC3CCC2O3)=O)C2CCCCC12 62476,C1(C(N2CC(C)(C)C(c3cc[nH]n3)C2)=O)Cc2ccccc2C(=O)O1 62477,c1(C(=O)NC2C(C(=O)NCCC3(C)OCCO3)C2)ccc(Br)cc1F 62478,c1(CNC(CCCC)(C)c2nnnn2C2CCOCC2)cc(C(F)(F)F)cc(Cl)n1 62479,c1(C(N(CC(C)NC(Cc2c(CC)cccc2)=O)C)=O)cc2n(n1)CCC2 62480,N1(C(=O)C=C(Cl)Cl)CCCC2(CCN(C(C3(CC(F)F)CCC3)=O)C2)C1 62481,Cc1cc(Cl)c(C(N2CC(NC(=O)CC3CCCN3C(C)C)CC2C)=O)cc1C 62482,C(c1ccccc1)=CC=CC(=O)N(CC1(C)CC(NC(c2c(C)coc2)=O)C1)CC 62483,C1(COC)(NC(c2scnc2C)=O)CCN(C(=O)CC2(O)CCOCC2)C1 62484,N1(C(C)C(=O)Nc2ccc(CC(F)(F)F)cc2)CCC2CCCC12 62485,N1(C(COC(C)(C)C)=O)CCCN(C(=O)CS(=O)(=O)Cc2cccs2)CCC1 62486,C1(C(N2CC(C#C)(C(=O)NCc3ccc(C)c(O)c3)C2)=O)CCC(C)=C(C)C1 62487,CC1CCCC(n2cc(CN(C(C)C(=O)N(CCCC(=O)O)C)C)nn2)C1 62488,Cc1cc(C(=O)NCC(F)CNC(C2CC(C)(C)O2)=O)nc(C)n1 62489,c1(C(=O)Nc2c(C(=O)OCC)nc[nH]2)cc2cc(-c3cc(C)cs3)cnc2[nH]1 62490,c1(C(N(C(C)CN(C(=O)C(C)(C)N(C)C)C)C)=O)nn(C)c(Cl)c1Br 62491,c1(CC)cnc(C(N2CCC(CO)(NC(c3cc(C)n(CCO)n3)=O)C2)=O)nc1 62492,CC1(C)C(CN)CCN1C(=O)Cc1cc(Cl)cs1.c12cccc(c1)C(=O)NC2 62493,CC1C(NC(C2(C)CCNC2=O)=O)CCCN1C(=O)COc1cc(Cl)ccc1Cl 62494,c1(CC(C)C)cc(C(=O)NC2CC(F)(CNC(=O)COc3ccccc3)C2)n[nH]1 62495,C1(C(N(CC)OC)=O)CC2CCCC2N1C(c1ccc(Cl)s1)=O 62496,C1(C(N2CCC(NC(c3cncc(C)c3)=O)C2C)=O)CCOCC1(C)C 62497,c1(C(C)C)ccc(C(N2CCC(O)CC2C(=O)NC(C)CN(C)C)=O)cc1Br 62498,CC(C)(F)CCC(=O)NCCCNC(c1cc(-c2ccc(Cl)cc2)ns1)=O 62499,C(=O)(C(O)C(CCC)NC(c1cc(O)n(CC)n1)=O)NCCC(CCC)O 62500,c1(OC)ccc2[nH]c(C(N3CCSC(C(=O)NCC(C)O)C3)=O)cc2c1 62501,N1(C(CC2C=CC(NC(c3nc(C)c(C)s3)=O)C2)=O)CC2CC(CO)C(C2)C1 62502,N1(C(C(CCC)C(C)C)=O)CC(NC(=O)C(C)(C)CS(C)(=O)=O)CC12CCCC2 62503,C1(NC(CNC(C(C)(C)C)=O)=O)CCN(C(=O)CN2CCCC2)CC1(C)C 62504,C(=O)(CCC(F)(F)CN=[N+]=[N-])N1CCN(C(c2ncc(C)c(Cl)c2)=O)CC(O)C1 62505,O=C(CCCC(F)(F)F)NC1CC2CC(NC(c3c[nH]c4cccnc34)=O)C2C1 62506,c1(C(=O)NC2C(C)CN(C(=O)C(O)CC3CC3)C2)nc2ccc(Br)cn2n1 62507,C1(C(=O)NCC(C)(F)CNC(=O)C(C2CCCCCC2)O)CCc2nncn2C1 62508,c1(CNC(NN(CC)CCO)=O)nn(C)c2cccnc12 62509,CCCCC1C(=O)N2CCC(F)(C2)C(=O)N1.C(C(C)(C)C(=O)NC)OC 62510,C(=O)(CCCNC(c1cnn(CC2CC2)c1)=O)N1C(CN=[N+]=[N-])CC1 62511,N1(C(CNC(C2CCCN2C(=O)C2CC2)=O)=O)CC2C3CCC(C3)C12 62512,Nc1sc2c(c1C(=O)NC1CCCC1NC(=O)C(=C1CCCCC1)F)CCC2 62513,C(=O)(C(CCCC)N(C)C)N1C2C(NC(C(C=C)C)=O)C(C2)C1 62514,N1(C(=O)CSc2cccnc2)CCCCC1c1cn(C2CCCC=C2Br)nn1 62515,Cc1cccc(C)c1C(=O)NCc1ccoc1C(=O)NCC1COCC1N(C)C 62516,C1(CC#C)(C(=O)NCCN(C)C(c2ccccc2)C2C3CCCC23)CCCO1 62517,c1(C(=O)NC2CC(CNC(C3CCC4CC34)=O)C2)ccc(=NCC2CC2)[nH]c1 62518,Cc1cc(N)ccc1C(=O)NCCNC(C1CC2(C1)CC2F)=O 62519,N1(C(c2c(SC)cn(C)n2)=O)CCC(C)(C)C(CNC(=O)C(C)=CC2CC2)C1 62520,c1(C(=O)Nc2ccc(OC(C)C)cc2)cccc2oc(N(C)C)nc12 62521,N1(C(C(CCF)NC(c2n(CC)ccn2)=O)=O)CCSC(C)(C)C1 62522,C1(NC(c2cc(C3CC3)no2)=O)CCC(C(=O)NCc2ocnc2C2CC2)CC1 62523,c1(C(=O)Nc2ccc(OC(F)F)cn2)csc(=NCc2ncc(Br)cc2Br)[nH]1 62524,c1(C(=O)NC2CN(C(CSCCOC)=O)C2)cc(-c2cccn2C)[nH]n1 62525,c1(C(N2CC(NC(CC(CC)OC)=O)C(SC)C2)=O)cc(C)c(N)cc1Cl 62526,c1(OC)cccc(I)c1C(=O)OCCS(=O)(=O)C(F)(F)F 62527,c1(C(C)OC)nc(-c2csc(N3CCC(O)C3)n2)n(C)n1 62528,C(CCCCCC(=O)N1CC(COC)CC1C)NC(C1C(CC)OCC1)=O 62529,c1(C(=O)NCCCN(CCCCNC(C(COC(C)=O)C)=O)C)c(C)n[nH]c1C 62530,c1(SC(C)C(N2CCN(C(C3(O)COC3)=O)CC2CO)=O)ccc([N+](=O)[O-])cc1 62531,C(CC(C)C)(C(=O)N(C)C)NC(C1CCN(c2snc(CC)n2)CC1)=O 62532,C1(OCC#C)CCCN(C(=O)C=CC(C)(C)NC(=O)C=Cc2cnccn2)C1 62533,N1(C(c2cnc(CCCC)[nH]2)C(=O)NCC2CCCO2)CC2COCC2(CO)C1 62534,C1(c2c(C(=O)NCC(=O)NCC)c[nH]n2)CCCCN1C(=O)C(C)C1CCC1 62535,C1(C(N2CCC(C(c3cccc(OCC)c3)C)C2)=O)CCC(N)C(O)C1 62536,C1(CNC(c2cn(CC)nn2)=O)CC(F)(F)CN1C(=O)CC1(COC)CCCCC1 62537,c1(C(=O)NCCOC(C)(C)CNC(=O)Cc2ccon2)ccc2nccn2n1 62538,CC(C)(C)C(O)C(=O)N1CC(CCNC(=O)C(N)=O)C1 62539,C1(n2c(C3C(C)(C)CC3)nc(-c3cccc(SC)n3)n2)CC2CCC1(C)C2(C)C 62540,C1(CN(C)CCNS(C)(=O)=O)CC(O)(OC)C1(C)C 62541,c1(C(=O)NCC(CC)NC(c2nn(C)c(Cl)c2Cl)=O)cc(C)nc2ccccc12 62542,N1(C(C(CCSC)NC(=O)CCC2OCCO2)=O)CCOC(C#N)C1 62543,c1(-c2cn(C(CC)(Cc3ccccc3OC)OC)nn2)cn(C)nc1OC(F)F 62544,C(C(CC1CC1)C(=O)NCCCC1CCCCO1)NC(c1c(C)nns1)=O 62545,C1(C(N(C(C#C)C2CCC2)C)=O)(CC)CCN(C(C2COCCN2C)=O)CC1 62546,C1(C(N2CC(CC(=O)OC)C2)=O)C2CCC(C2)N1C(=O)Cn1ccnn1 62547,Cc1cc(CC(=O)NCCNC(c2c[nH]nc2C(F)(F)F)=O)no1 62548,N1(CCCNC(c2c[nH]c(=N)o2)=O)CCN(C(c2ccc(C(N)=O)o2)=O)CC1 62549,C1(CC(C)C)CN(C(=O)CC2(CNC(C3CCN3C(C)(C)C)=O)CC2)CCO1 62550,C(C)(C(C(=O)NCCCCCN=[N+]=[N-])C(C)C)NC(C(C)=NOCC#N)=O 62551,c1(C(N2CCC(C(C)NC(=O)CC3(C#N)CC3)C2)=O)ccc2c(c1)CC2 62552,C1(C(N2CCC(C(CNC(CSC)=O)(C)O)CC2)=O)CCCCN(C)C1=O 62553,C12(NC(CC3CCC(C)C3)=O)CCC(C(=O)NCC(C)(O)C3CCC3)(CC1)C2 62554,N1(C(C(C)Cn2cccn2)=O)C2CCC1CC(NC(c1cnn(C)c1F)=O)C2 62555,Cc1ccc(Br)c(CN2CC(NC(c3cnc(O)[nH]3)=O)C3(CC3)C2)c1F 62556,C1(OCC(=O)NCCN2CCN(C(C3CC3(F)Cl)=O)CC2)CCC(F)(F)CC1 62557,C1(NC(C2(C)COC2)=O)CCN(C(=O)CSc2ccncc2F)CC1(C)C 62558,Cc1cccc(C(CNC(c2cocn2)=O)NC(=O)CC23CCCC2C3)c1 62559,CCC(C)CC(C)C(=O)NCC1(C(N)=O)CN(C(c2ccc(OC)c(Cl)n2)=O)C1 62560,N(C1c2ccccc2CC12CCCC2)C(=O)NC(CSC)Cc1cccc(Br)c1 62561,C1(NC(c2cc(CCC)oc2C)=O)CCCN(C(c2nc(CC)no2)=O)C1C 62562,c1(C(N(C2CCCC2)CC=Cc2c(Br)ccc(C)c2)=O)ccc2c(c1)OCCO2 62563,N1(CC(=O)NCC(CNC(=O)CCc2n[nH]c(=N)s2)OC)CCS(=O)(=O)CC1 62564,Cc1ccc(-c2cnc(C(=O)NC(c3nnc4n3CCC4)C)c(F)c2)cc1Cl 62565,c1(-c2ccc(N(C3CCCNC3)S(CC)(=O)=O)s2)ncccc1OC(C)C 62566,C1(CNC(C2CC(C)SCC2)=O)CN(C)CCN1C(c1cccnc1N)=O 62567,C1(C)(C(N(CC(O)CO)C)=O)CCCN(C(=O)CC2NC(=O)NC2=O)C1 62568,c1(C(=O)NC(C(=O)NCCCC=C)CC2CC2)cc(O)ncn1 62569,CC1CN(C(=O)C(O)CC(N)=O)CCC1C(=O)NCCC1CCCC1O 62570,C(=O)(C(C)C(F)(F)F)N1CCC(CC=C)(NC(c2cn(CC3CCCO3)nn2)=O)C1 62571,C(=O)(C1=CCC(C)CC1)N1CCC(CCNC(C2CCCC(OC)C2)=O)CC1 62572,c1(CC)nc(C(=O)NC(C2CN(C(c3cnn[nH]3)=O)C2)C)n[nH]1 62573,C1(OC)CCC12CC(C(=O)N(C)CCN(C)C(C1CC3CCC1O3)=O)C2 62574,c1(NC(C2N(Cc3ccc(OC)cc3)CCC2)=O)cccc([N+](=O)[O-])c1 62575,n1(CCCOC)cc(CCC2CN(C(=O)CC(C)C3CCCO3)C2)nn1 62576,c1(CC(=O)NCC2(NC(C(C)n3cccn3)=O)CCCC2)cccc(C(F)F)c1 62577,Cc1[nH]c(C(=O)NCC2CN(C(C3CN(C)CCO3)=O)CCCO2)c(C)c1C 62578,Cc1csc(=NCC(=O)NCC2CC(C)N(C(c3cscc3F)=O)C2)[nH]1 62579,C1(NC(C(C)(C(C)C)OC)=O)CCC2(CCCN2C(=O)CS(=O)(=O)C2CC2)CC1 62580,CC1CCC(C(=O)NC(c2ncccn2)C)N1C(C12CC(C(=O)O)(C1)C2)=O 62581,C#CCC(C)(CNC(=O)C(CNC(=O)C(C)NC(=O)OC)CC=C)CO 62582,N1(C(C(CC=CC)CC)=O)C2CCC1C(F)C(NC(c1ccc(O)nn1)=O)C2 62583,c1(N(C(=O)NCCC(N2C(Cc3cnc(C)s3)CCC2)=O)C)ccccc1Cl 62584,c1(OC)ccc(C(=O)NCC2CCCCC2NC(c2n[nH]cc2F)=O)cc1F 62585,Cc1[nH]nc(C(=O)N(C(C)CNC(=O)C(C)CC2CCCC2)C)c1O 62586,N1(C(CC2(N(C)C)CCC2)=O)CC(C)(C)CC1CC(N1CCCC(C(F)F)C1)=O 62587,Cc1noc(Cl)c1CC(=O)NC1CCN(C(=O)CC2C=CS(=O)(=O)C2)C1C 62588,N#Cc1ccc(CN2CCC(CC(=O)NCC=Cc3cccnc3)C2)c(Cl)c1 62589,N1(C(C(C)N2CCCC2)=O)CC=C(CC(=O)NC2CCCC2C(N)=O)CC1 62590,O=C1CC2(C1)CC(C(=O)NCC(CC1CC1)C(=O)NCC(F)CO)C2 62591,CC1CC2(CO1)CN(C(=O)CCCN(C)C(C1(CO)CCCCO1)=O)C2 62592,C1(C(N(CC(C)N(C)C(C23CC(F)(C2)C3)=O)C)=O)CCCCS1 62593,c1(-c2nc(C(C)SCC)nn2C2CC(C)(C)OC2(C)C)ccnc2c1cnn2C 62594,N1(C(c2c(OCC)oc(C)n2)=O)CCC(NC(C2CCS(=O)(=O)N2)=O)C(C)C1 62595,C12(NC(c3c(F)ccc(C)c3)=O)CC(C)(C1)OC21CN(C(=O)CC(C)C)C1 62596,Cc1cc(CNC(=O)CCN(C(=O)CC2CCC3CC23)CCO)sn1 62597,N1(C(C(C2CCN(C(Cn3nc(C)oc3=O)=O)C2)(C)C)=O)CC(C)OCC1C 62598,N1(C(C2(C)CCCS2)=O)CCC2(CCC2NC(c2cnc[nH]2)=O)CC1 62599,C(=O)(CC1=CCCC1)NCCC1(NC(CCc2c(C)noc2C)=O)CCOCC1 62600,C1(OC)CC(NC(c2cscc2SC)=O)CN(C(=O)C(c2cnn(C)c2)OC)C1 62601,Cc1cc(=O)oc(C)c1C(=O)NCCC(O)CNC(C1CC2CC2C1)=O 62602,c1(C(=O)NCC23CC2CN(C(=O)CCCc2nccs2)C3)ncc2ccccn12 62603,N1(C(C(COC)C)=O)CC(NC(c2[nH]nc(C(F)(F)F)c2C)=O)C(O)C1 62604,c1(CNC(C2(OC)CCN(C(CC)=O)C2)=O)nn(C)c(=O)n1C 62605,c1(C(N2CCCC(CNC(c3cccc4occc34)=O)C2)=O)coc2c1COC2 62606,CCC(C)(CC(=O)NCC=CCNC(c1ccc(S(C)=O)cc1)=O)C(=O)OC 62607,N1(C(CSC)=O)CCC2CN(C(c3cc4c(Br)cccc4[nH]3)=O)CC2C1 62608,Cc1[nH]nc2c1CC(C(N1CCN(C(=O)C(C)(F)F)C(CC(C)(C)C)C1)=O)CC2 62609,c1(C(=O)NCCNC(C2(Cl)C(C(C)=O)C2)=O)ccc2c(c1)NCCC2=O 62610,C(CC(N)=O)(C(=O)NCc1cc(C(=O)O)n[nH]1)NC(C(CN(C)C)O)=O 62611,N1(C(c2n[nH]c(C)c2Br)C(=O)NCC=C)CCN(CC)CC1.C1CCC(=O)N1.OCC 62612,C1(CN(C)C(C2CCCCC2)=O)CCCN1C(=O)CCCc1nccs1 62613,c1(C(=O)NC2CCCC(NC(C3CCC(F)(F)C3)=O)C2)cc(F)ccc1C1CC1 62614,N1(C(CCOC)=O)CCC2(CC1)CCN(C(=O)C(C)CCC(C)(C)C)C2 62615,C1(=O)C(F)CC(C)(C)N1.CC(C)C(C)(O)CN1CC(N2CCNC2=O)C1 62616,Cc1ccc(C(=O)NC2C(C(=O)NCC3CC(=O)N(C)C3)C2(C)C)cc1F 62617,C1(CC(=O)NS(=O)(=O)CCCN2CCOC2=O)CCS(=O)(=O)CC1 62618,n1(C(C)C)ncc2c(NCCS(=O)(=O)CC)[nH]c(=NC(C)CC(C)C)nc12 62619,C1(C(=O)NCC(COC)NC(C2CC=CCC2C)=O)CCCCC12CCC2 62620,CCCCC(CNC(c1ccc(C#N)s1)=O)NC(=O)C(C)F 62621,c1(C(=O)NCc2occ(C(=O)NCC3C(C)OCC3)n2)ccc(O)nn1 62622,O=[N+]([O-])c1ccc(Sc2nc(C3CC4CCC3CC4)ns2)cc1 62623,c1(C(N2CCC(CN(C(C(CC#C)O)=O)C)CC2)=O)cccn2nnnc12 62624,CC(c1ccsc1)=CC(=O)NC(C)(C)C(C)NC(=O)CC(C)n1cccn1 62625,c1(COC)nc2cccc(C(N3CCSCC3C(=O)O)=O)c2[nH]1 62626,c1(C(=O)NCC(=C)CCNC(=O)C(F)C2CCOC2)nn(CC)cc1[N+](=O)[O-] 62627,Cc1cc(F)ccc1NC(=O)C(=O)NC(c1ccccc1F)C 62628,c1(C(=O)OC(C)C(=O)N(C)C)cc(Br)c2occc2c1.c12ccc(cc1)o2 62629,N1(C(c2n(CCC)ncc2)=O)CC2CC2(CNC(c2nn(C)cc2C)=O)C1 62630,c1(CC)cc(CN(CCCN2CCCC2=O)Cc2cnn(C)c2)ncn1 62631,c1(C(N(CCC(=O)NC(CC)C(=O)N(C)C)CC2CC2)=O)cnc(O)c(F)c1 62632,CC1CN(C(C2CC(n3cc(C45CCC(CC4)C5)nn3)C2)=O)CC1C(F)(F)F 62633,c1(CNC(CC=C=C)=O)ccc(CCNC(c2coc(C(=O)OC)n2)=O)cc1 62634,C1(CCC(=O)N(C)Cc2nncs2)CCCCN1C(=O)C=CC1CC1 62635,Cn1cc(C(=O)NCC2CCCC2NC(=O)Cc2cn(C)nn2)n(C)c1=O 62636,c1(C(=O)NCC(CNC(C2(CC)CCNC2=O)=O)(C)F)n[nH]c2c1COCC2 62637,N1(C(C(C)OCC)=O)CCn2cccc2C12CCCCC2 62638,C1(CNC(c2c(OCC)scc2)=O)CC(O)CN1C(=O)CC1(C)CCC1 62639,Cc1ccccc1-c1cc(C(=O)N(CCC#N)CCO)on1 62640,Cc1c(NC(C2CCC(C(C)C)N2C(c2c[nH]ccc2=O)=O)=O)cccc1CO 62641,c1(OC)cc(C)ccc1-c1cn(CC(C(=O)OC)NC(=O)C2=CCCC2)nn1 62642,Cc1ccc([N+](=O)[O-])c(OCCCC(=O)NCCNC(=O)C(C)C2CCOC2)c1 62643,C1(CC(=O)NCCC2(OCC)CCC2)CCCN(C(=O)Cc2cc(C)on2)CC1 62644,c1(CC)ccc(C(=O)NC2(C)CCN(C(c3c(OC)nsc3OC)=O)C2)nc1 62645,N1(C(C2N=C(C)SC2)=O)CCN(C)C(CNC(=O)C=Cc2ccccc2F)C1 62646,C1(NC(=O)CC2(CNC(c3scnc3Cl)=O)CC2)CCCCC1O 62647,C1(NC(C2(NC(c3c(CCC)cccc3)=O)CC2)=O)CN(C)CC12CC2 62648,O=S(=O)(c1ccccc1S(=O)(=O)NC1CCN(Cc2ccccn2)C1)C(F)F 62649,c1(C(=O)NC2CC(CNC(c3nc(C(C)=O)sc3)=O)C2)ccc2cncn2c1C 62650,N1(C(c2cccc(C)c2)C(=O)NCCCC)CC(O)CC2(CCCC2)C1 62651,C1(NC(C=CC(C)(C)NC(C(CSC)O)=O)=O)CCCCC12CC2 62652,c1(OC)cc(OC)nc(C(N2C3CCC2C(CNC(=O)CCCC(C)=O)C3)=O)n1 62653,c1(C(=O)NCC(C)N(C(c2ccc(OC)cc2)=O)CC)cccc2nncn12 62654,c1(C(=O)NCC(CCOC)NC(c2[nH]c(O)nc2C)=O)cc2occc2[nH]1 62655,C1(C(N2C(CC)(CO)CCC2)=O)CCC(C)(C)N(C(C2CC(=O)CCO2)=O)C1 62656,C1(NC(c2c(N)nccn2)=O)CC12CCN(C(c1ncccc1Cl)=O)CC2 62657,CCC(CC(F)F)C(=O)N(CCCOCCN(C)C(c1cc(C)cc(C)n1)=O)C 62658,CCCCCC(C(=O)NCCC1CN(C(=O)C=Cc2ncc[nH]2)CC1C)C(C)C 62659,C1(OCC(=O)NCC2(F)CCN(C(CNC=O)=O)C2)CCC(F)(F)CC1 62660,c1(CC)cc(C)c(C(N2CCC(CN(C(=O)Cc3csc(Cl)n3)C)C2)=O)o1 62661,Cn1nc(Br)c2ncnc(N3CC4(CN(C(c5c(F)cc(F)c(F)c5F)=O)C4)C3)c12 62662,c1(C(CC(=O)NCCCOC)NC(c2nccn2C)=O)ccc(C#N)cc1 62663,CC1CN(C(c2cnn(CC(F)(F)F)n2)C(=O)NCCC2CC2)CC2(CCC2)O1 62664,c1(C(N2C(CNC(CC3CC(CC)OCC3)=O)COCC2)=O)ccc(O)c(Cl)c1 62665,C(N=c1nc[nH]c(N2CC3CC2CS3=O)n1)C1(C(F)F)CCC1.N1CCOCC1 62666,C1(C(C)CO)CCN(C(C2(C(C)C)CCCN2C(=O)CC2CCC(=O)N2)=O)CC1 62667,C(=O)(CCC(=O)NN(C)C)NCCC(C)NC(c1nccc(COC)c1)=O 62668,C1(O)(CN(C(CSC)=O)C)CCCN(C(=O)C(C)(C)OC)C1 62669,c1(C(N2CC(O)(CCN(C(CC3C(C)C3)=O)C3CCN3)C2)=O)snc(Cl)c1Cl 62670,C1(NC(C(C(C)C)OC)=O)CCN(C(=O)CC(C)(O)C2CC2)CC1(C)C 62671,C1(OC)CC(CNC(C2(C(F)F)CC(O)C2)=O)N(C(c2cc[nH]c2)=O)C1 62672,c1(C(=O)NC(CC(C)C)CNC(C2(C#N)CCC2)=O)cc(Cl)cc2ccncc12 62673,N1(C(C2=C(C)CCC2)=O)CCC2CC2(C(N(C)C[Si](C)(C)C)=O)CC1 62674,C=C1CC2CCC(C1)N2C(C1CCC(CNC(=O)CCCSC)C1)=O 62675,N1(C(c2c(C)nc3ccccn32)=O)CCC(C2CCN(C(=O)C(C)C)C2)CC1 62676,C1(C(C)C)CCC(N(CC(O)Cc2cccc(Cl)c2)CCN2CCOCC2)C(=O)N1 62677,n1(CC)c(CNC(C2(SCCNC(=O)OC(C)(C)C)CC2)=O)nc2ccccc12 62678,C=CCS(=O)(=O)CCNC(=O)CSCc1nnc(-c2ccccc2Br)o1 62679,CC(CC(N)=O)C(=O)NCC(=C1CN(C(C2(CF)CC2)=O)C1)F 62680,C1(C(N2CCC(OC)CC2)=O)C(C)OCCN1C(C1CCC1C)=O 62681,C1(SC)CN(C(=O)NCCc2ncnn2C)CC1N(C)C 62682,CC(C)(C)C(CNC(c1cc(=N)[nH][nH]1)=O)NC(=O)Nc1ccccc1 62683,c1(C(=O)NCCC2CC(Nc3nc(SC)c(C)cn3)C2)cnn2c1C(=O)NCC2 62684,N1(C(CCCn2cc(-c3cncc(OC)c3)nn2)=O)CC(C)NC(=O)C2CC12 62685,c1(C(=O)NC(CCCC)CNC(=O)CC2CCC2)nc(OC)ccc1C 62686,C1(C(N2CCC(NC(C3CCCC3)=O)C2)=O)COc2ccc(F)cc2C1 62687,c1(CNC(=O)NCCCCCl)cc(O)nc(O)n1 62688,c1(C(N2CCC(NC(c3ccnnc3)=O)C2)=O)cnc(-c2nccs2)nc1O 62689,c1(C(=O)NCCOC2CCN(C(c3c(C)nn[nH]3)=O)C2)cnc(O)n(C)c1=O 62690,C1(NC(CCc2onc(C(C)OCC)n2)=O)CC2(C1)CC(NC(=O)CC1CSC1)C2 62691,Cc1cc(Br)cc(CN2CC3CC2C3C(=O)NCc2ccc3ccoc3c2)c1O 62692,Cc1nc[nH]c1C(=O)NC(Cc1nccs1)CO 62693,N1(C(c2c(C(C)(C)C)con2)=O)CCC2CCCC12C(=O)NC1CCNC1=O 62694,c1(C(N(C)CC2N(C(CC(C)C(F)F)=O)CC(F)C2)=O)ccc2c(c1)CCCC2 62695,CN1CCC(O)(C2(C(=O)NCC(C3CC3)N(C(=O)CS(C)(=O)=O)C)CC2)CC1 62696,Cc1nc(CNC(c2ccc(CNC(c3csc(F)c3)=O)nc2)=O)sc1C 62697,CC1CN(C(c2ccc(Cl)cn2)=O)CC2(CCN(C(c3ccnc(O)c3)=O)C2)O1 62698,N1(C(c2c(C)con2)=O)CCCC2C1CCCCN2C(C1CC(C(F)F)C1)=O 62699,C1(N(C(CSCC#C)=O)C)CCCCN(C(=O)CSCCC)C1 62700,C1(=O)C(CCS(C)(=O)=O)O1.N1(CC(=O)OC)CCC(N(C)C(=O)NC(C)(C)C)C1 62701,N1(C(C2CC(NC(=O)CN3CCOCC3)C2)=O)CCOCC1Cl 62702,N1(C(C(CC)N(C)C)=O)CCC12CN(C(c1nccc(Cl)c1C)=O)C2 62703,c1(OCC)ccc(C(=O)NC2(CCOC)CCN(C(=O)C(C(C)C)OC)C2)cn1 62704,N1(C(C2CCCC(=O)O2)=O)CCOC2CCN(C(c3cc(Cl)ccc3Cl)=O)CC12 62705,C1(O)(CNC(C(CC)OCC)=O)CCN(C(C2(c3ccnc(Cl)c3)CCC2)=O)C1 62706,C1(NC(c2nc(C)sc2)=O)CN(C(=O)CCNS(=O)(=O)c2cccs2)CC1(C)C 62707,c1(C(=O)NC(C)(C)CCNC(C2CCS2(=O)=O)=O)ccc(C(O)CF)cc1 62708,N1(C(C2(C#N)CCCC2)=O)CCN(C2CCCN(C(C3CC3(F)F)=O)C2)C(=O)C1 62709,S(=O)(=O)(c1cc(Br)cnc1N)N1CCN(C(C)C2CC2)CC1 62710,Cc1cc(F)cnc1C(N1CCCC(CNC(c2cn(C)ccc2=O)=O)CC1)=O 62711,CC1CC(CNC(=O)C(C)(C)c2ccccc2)CN1C(=O)CCOCC(F)(F)F 62712,c1(C(=O)NC2C(OC)CN(C(=O)C(C)c3ccco3)C2)cc(F)c(SC)cc1N 62713,C(CCCC(=O)N1C(CNC(C2CC2C)=O)CC2CC12)OCCC=C 62714,C1(NC(c2ccccc2)=O)CCCCC12CCCN(C(=O)COCC(F)F)C2 62715,c1(SC)ccc(C)c(C(=O)NCC2=CCN(C(c3c(F)cccc3F)=O)CC2)c1 62716,C#Cc1ccccc1CSC1CC1C.C1C(=O)OCCOCCNC(=O)N1 62717,N1(C(COC2(C)CCC2)=O)CC2C(NC(c3cc(C#N)cs3)=O)C2C1 62718,O=C1CCc2c(C(N3CCC(CCNC(C4CCCO4)=O)C3)=O)cccc2N1 62719,C(=O)(C(C)(O)CC(C)C)NCC1CCCN(CC=C)C1 62720,Cc1cc(C(=O)NC(C(C)NC(=O)Cc2c[nH]nc2O)C(C)C)c(O)nc1C 62721,C1(CCOC)(C(=O)NCc2cccs2)CCN(C(C2CC2C(F)F)=O)C1 62722,Cc1ccoc1CC(=O)NCC(C1CCN1C(c1ccnn1CCN(C)C)=O)C 62723,C(=O)(C(C)(C)CCF)NC(C1OCCN(C(COc2ccc(C)cc2)=O)C1)C 62724,c1(C(=O)NC2C(CNC(c3cnn(CC)n3)=O)CC2)ccc(Cl)cn1 62725,c1(OC)ccc(CC(C)C(=O)NCC(C)(C)CNC(C2(C)CC2(C)C)=O)cc1 62726,C(=O)(CCCS(C)(=O)=O)NCC12OCC(CNC(CC(CC)C3CC3)=O)(C1)C2 62727,N1(C(C2=NNC(=O)CC2)=O)CCC2C(CCN2C(=O)C(CC(F)F)C2CCC2)C1 62728,C1(NC(CNC(CC)=O)=O)CC12CCC(NC(=O)CC1COCC(C)(C)O1)CC2 62729,C1(C(=O)NCCCOCCCNC(C(n2ccc(C)n2)C)=O)CCCCCCC1 62730,c1(CC(=O)N(C(C)CNC(C2CCCCC2C)=O)CC)ccc(O)cc1 62731,c1(NC(C2CC(=C)CN2C(=O)CCc2ccc[nH]2)=O)ccc(OC)nc1Br 62732,n1(CCC)cc(C(=O)NCCCCCNC(=O)C(C2CCC2)OC)nn1 62733,c1(CC)c(NC(C2CCN(C(c3ccn(C4CCCC4)n3)=O)C2)C)ncnc1Cl 62734,N1(C(CC(CCC)O)=O)CC2CC1CCC2NC(=O)Cc1nnc(C)s1 62735,c1(CC)cccc(C(=O)NCCOC2CCN(C(c3cccc(C)n3)=O)C2)c1F 62736,C(=O)(C1=CCC(NC(C2(C)COC(=O)N2)=O)C1)NC(c1nnc(C)o1)C 62737,C=CCC(CNC(c1ccccn1)=O)C(=O)N1CCC(SC)C1 62738,C1(C(=O)NC2C(CC)N(C(=O)Cc3cncs3)CC2)CCc2nnn(C)c2C1 62739,c1(C(=O)NCCC(C(=O)NC2C3CCCCCC23)OC)ccnc2ccsc12 62740,N1(C(c2cccc(N(C)C)c2)=O)CC(NC(c2cncs2)=O)C2(CCC2)C1 62741,N1(CC2C(C)CCCC2)C(=O)CN(CCCn2cnnn2)C1=O 62742,N1(C(=O)NCC2(C#C)CCC2)CCCC(CC)C1 62743,c1(NC(C(C2CCCCC2)C)C)nc(CO)ns1 62744,N1(C(c2n(CC)nnc2)=O)CC2CCC(C(=O)N(c3csnc3C)C)(C2)C1 62745,CCC(O)C(F)(F)C(=O)NCC1C2CN(C(C3(C(=O)N(C)C(C)C)CC3)=O)CC12 62746,c1(C(=O)NC2(CNC(c3c(CC)nns3)=O)CCCC2)cc2c(cc1N)CCC2 62747,C1(C(=O)NC(CNC(C2(SC)CCC2)=O)CC(F)(F)F)CN2CCN1CC2C 62748,N1(C(C2C(C)(CC)C2)=O)CC=C(C(=O)N2CCCOCC2C)CC1 62749,N1(C(c2nc(C)c(C)s2)=O)CCC2C(CCCN2C(c2ccc(CO)nc2)=O)C1 62750,C=CCCCCCCC(=O)N1CCC(NC(=O)CC2(COC)CC2)CC1C 62751,C1(C(=O)NC2CCC(NC(CC3(C)CC3F)=O)CC2)CCCCCCC1 62752,C(=O)(CC1NC(=O)c2ccccc21)N(C1CCCN(C(C2(O)CCC2)=O)CC1)C 62753,CC1CN(C(c2cc(Br)co2)=O)CCC1SCC(=O)N(C)CCN(C)C 62754,c1(CC(=O)NCC(C)CNC(c2cc(O)cc(F)c2F)=O)csc(S(N)(=O)=O)c1 62755,S(=O)(=O)(c1c[nH]c(C(=O)NC2CCN(C(c3cc(Cl)cnc3O)=O)C2)c1)N(C)C 62756,C1(CNC(c2cn(C)nn2)=O)N(C(c2cccc([N+](=O)[O-])c2)=O)CCCC1(C)C 62757,N1(C(=O)Cc2cscn2)CCCC2(C1)CN(CC1CC(O)C13CCC3)CCO2 62758,S(=O)(=O)(c1ccc(N2CC(CO)C3(CCC3)C2)cc1Cl)NCC1(CC)CCCC1 62759,CC1CC(C#N)(C(N2CCC(CNC(=O)CC3CCN(C)C3=O)CC2)=O)C1 62760,c1(C(=O)OC)cc(=NCC2CCCCC2NC(c2cc(Br)ccc2Cl)=O)[nH]cn1 62761,Cc1ccc(Cl)c(C(N2CCC(CCNC(C3CCCCO3)=O)C2)=O)c1N 62762,C1(C2CCN(C(c3ccc4cncn4c3)=O)C2)(NC(C=CCC)=O)CC1 62763,C1(O)(CCNC(C2(CC)CC2)=O)CCN(C(=O)CN2CCCC2C)CC1 62764,c1(N2CC(CO)OCC2)[nH]c(=NCCC(O)C2CCC2)nc2sccc12 62765,C1(CNC(c2nccc(CC)c2)=O)COC(C)(C)CN1C(C1CC(F)C1)=O 62766,Cc1cc(C(=O)NCC(O)CNC(=O)C(C)n2cccn2)c2c(n1)CCCC2=O 62767,C1(CCNC(Cc2c(C)n[nH]c2)=O)CN(C(=O)CCCC(=O)N(C)C)CC(C)O1 62768,C1(C(=O)NCCC(C)(C)NC(c2cc(CC)nn2C)=O)CC2(CCC2)CO1 62769,c1(CNC(=O)NC(C2CC(OC)C2)C(=O)O)cc2cc(Cl)ccc2o1 62770,C(=O)(C(F)C(C)C)NC(C1N(C(c2nc(C(=O)NCC(=C)C)sc2)=O)CCC1)C 62771,CC1CCc2onc(CNCC(C)(C(=O)O)c3ccccc3)c2C1 62772,c1(CC(=O)N(CC(C)NC(c2cnc(O)c(F)c2)=O)CC)cnn2c1OCCC2 62773,CCC(CC)(CCNC(C1CC2(CCO1)CC2)=O)NC(C1C(C)(C)C1(F)F)=O 62774,S(=O)(=O)(c1ccncc1)NC1CCC(NC(c2ccccc2Cl)=O)C1 62775,C1(C#N)(NC(c2c(SC)cccc2)=O)CCN(Cc2ccnn2C)C1 62776,C1(C(N2CCC(CNC(=O)CSc3ccccc3)C2)=O)(CC)CCOC1 62777,N1(C(C(=O)NC)=O)CCCCC1C(=O)NCCOCC(F)F 62778,c1(C(=O)NCC23C(CN(C(C(CCC)C)=O)C2)C3)c(C)nn(C)c1-n1cncn1 62779,N1(C(C(C)Nc2nnnn2C)=O)CCC(C(=O)OC2CN(C(N)=O)C2)CC1 62780,C1(NC(c2cccc(C(N)=O)n2)=O)CC(F)CN(C(c2scnc2C(F)F)=O)C1 62781,c1(C(=O)NCCSCC(=O)N(C(CC)C2CC2)C)ccncc1Cl 62782,C(CCNC(=O)CC1CCCCO1)(C(=O)NC(C)(C)CCCO)OC 62783,N1(C(CC(C)OC)=O)CCC2(CC1)CC(NC(=O)C=C(C)C(C)C)C2 62784,N1(C(c2c(C)oc(CO)c2)=O)CC(O)CCC1C(=O)NCCSC(C)(C)C 62785,C(=O)(C1CCCc2nc[nH]c21)NCCCNC(c1c(C)n(C2CC2)cc1)=O 62786,c1(OCC)cnc(C(=O)NCCC2CN(C(=O)C(C)COC)CCO2)cn1 62787,CC1CCCCN1CC(=O)NCCCCNC(c1cccc(C(=O)C2CC2)c1)=O 62788,N1(C(C(CC=CC)C)=O)CCN(C(=O)COc2ccc(SC)cc2)CC1C(C)C 62789,Cc1nc(O)nc(O)c1CCC(=O)N(C(C)CNC(=O)CSCCC#N)C 62790,c1(C(N(CCNC(C(C)NC(CC)(C)C)=O)C(C)C)=O)sccc1Br 62791,c1(OC)ncc(C(=O)NCC(n2cc(-c3ccccc3N)nn2)C)c(C)c1Br 62792,c1(C(N(CC(=O)N(CC(=O)N(C)C)C)CC)=O)ccc(C#N)n1C 62793,N1(C(C2(C#C)CC2)=O)C2CCC(C2)C1CNC(C1(C#C)CCCC1)=O 62794,CC(C(=O)NN1CCCC1C(=O)N(C(CO)CO)C(C)C)=CC1CC1 62795,Cc1cc(C(=O)NC2CS(=O)(=O)CC2NC(=O)C(C)N2CCCC2)cc(C)n1 62796,CCCC(CCC)(c1ccccc1)NCCn1cnccc1=O 62797,CCCCCCC(=O)N1CCCCC1CNC(c1c(Cl)cncc1Cl)=O 62798,N1(C(C2C(C)CCN2C(=O)CNC(=O)C(F)(F)F)=O)CCC2C1CCCN2C 62799,c1(OC)ccc(C(=O)NC2CCCC2NC(=O)C2=COCC2)c(C)n1 62800,c1(CNC(=O)NCC2(C)C=CCCC2)cnc(O)c(F)c1 62801,CC(C)C(O)C(=O)NC(C)C(CO)NC(=O)C(c1ccccc1)C 62802,C1(C(=O)NCCN(C(c2cncc(OC)c2)=O)C(C)C)Cc2ccccc2C1 62803,CC(C)(C(=O)N1CCC(F)(F)C(F)C1)C1=CCN(C(c2ccns2)=O)C1 62804,N1(C(Cc2cccc(C)c2)=O)CCN(C(=O)C(C)C2CC2)C(CCO)C1 62805,N1(C(c2ccc[nH]2)=O)CCCC(C2CCN(C(C3CCC(F)(F)C3)=O)C2)C1 62806,c1(C(=O)NC2CCCC(C(N3C(C)CC3CO)=O)C2)cn2c(n1)CCC2 62807,C1(CC)(NC(=O)Cc2cnn(C)c2)CN(C(=O)C=CC(=O)N(C)C)C1 62808,CCC(CC)C(C)C(=O)NC1CCC(F)(CNC(c2n[nH]c(C)c2Cl)=O)C1 62809,C1(CCC)CCCCN1C(=O)CN(C(=O)CNC(=O)COCC(C)(C)C)C(C)C 62810,c1(C(N2CCOCC(C)(CNC(C(CC)C)=O)C2)=O)cc(C)c2nc(C)nn2c1 62811,NS(=O)(=O)c1ccccc1NC(=O)CC1(O)CCN(C(C2CC2F)=O)CC1 62812,C1(CNC(C(Br)=C(C)C)=O)CC(O)CN1C(C1CCCN1C(C)C)=O 62813,C#CC1(O)CCCN(C(C2CCCC(NC(=O)C3=CCCC3)CC2)=O)C1 62814,C1(NC(C(C)N2CCCC2)=O)CCCC12CCN(C(=O)C(=O)C(C)(C)C)CC2 62815,Cc1cnn(C)c1CC(=O)NC1(CNC(C2CC2C#N)=O)CCCC1 62816,C1(NC(c2cc(C)sn2)=O)C2CC1N(C(c1cccc(N)c1Br)=O)C2C 62817,C1(=CC(N2C(C)CCC(NC(CCN(CC)CC)=O)C2)=O)CCCCCC1(F)F 62818,C=CCCCC(C(=O)N1CCOCCC1CC)NC(C1SCC=C1C)=O 62819,N1(C(Cn2c(C)cc(C)n2)=O)CCN(C(c2cc(C)n(C(F)F)n2)=O)C2CCC12 62820,Cc1cc(C(=O)NCC=CCNC(=O)CC2CC(F)(F)C2)cc(S(C)(=O)=O)c1F 62821,N1(C(=O)CCC2CCOC2)CCN(C(=O)CSC2CC2)C(c2cccs2)C1 62822,N1(C(C2(CCCC)CCC2)=O)CCC(O)C(NC(c2ccc(C)c(OC)c2)=O)C1 62823,c1(C(N2CC(C)C(NC(c3c[nH]nc3C(F)(F)F)=O)C2)=O)ccc(Cl)c(F)c1 62824,C(CN=C(NCc1cnco1)NCC1CCCCC1(C)C)OCC 62825,C#Cc1ccc(C(N2CCCC(O)(C(F)F)C2)C(=O)NC(C)CC)cc1 62826,C(=O)(C(O)CC(C)C)N1C2CC(NC(c3n[nH]c(C)c3Cl)=O)(C2)C1 62827,c1(NC(c2cc(Br)ccc2Cl)c2n(C(CC)(C)C)nnn2)cc(C)cc(Br)c1C 62828,C(=O)(C1CCc2c[nH]nc21)NC1(C2CCN(C(CN(C3CCC3)C)=O)C2)CC1 62829,CCCCC(=O)C(=O)N1CC(CNC(C2(CO)CCOCC2)=O)C(C)(C)C1 62830,N1(C(C(C2CCCN(C(c3c(C)scn3)=O)C2)(C)C)=O)CC2C(C1)C2(C)C 62831,C1(NC(c2cnccc2Br)=O)C(CNC(=O)C(F)F)CCC12CCC2 62832,N1(C(C2(C)CCC(C)C2)=O)CC2CCC1CN2C(C1C=CCC1)=O 62833,N1(C(CC(C)(C)C#N)=O)C2CCC1CC(NC(C1CCn3nccc3C1)=O)C2 62834,C1(NC(c2c(CC)occ2)=O)CN(C(=O)C=CC2CCC2)CCC1C(F)(F)F 62835,C(C(=O)N1CCC(C(N2C3CCC2CC3)=O)O1)C1C(=C)C1 62836,c1(C(N2CC(C)(NC(C(C)=C(CC)C)=O)C2)=O)ccnc(C(N)=O)c1 62837,c1(C(N2CCC(CCC(=O)NCC3(CCC=C)CC3)C2)=O)cc(C)c(O)nn1 62838,c1(C(N2CC(C)CC(C(N(CCC)CC)=O)C2)=O)c[nH]c2ccccc12 62839,c1(-c2nc(C(=O)NC3CCNC3)on2)cccc(-c2cscn2)c1 62840,N1(C(C(C)CN2CCOCC2)=O)C(C)C2CC1C2NC(=O)COC(F)F 62841,CC(CC(=O)N1CCC(C2CCCN2C(c2ccc(CO)cn2)=O)C1)C(F)F 62842,C1(C(=O)OCC(=O)C(Cc2ccccc2F)N2CCCCC2)(CSC)CCCCC1 62843,CCC(CCCC(=O)N(CCCn1ccnc1)C)NC(=O)C(C)N1CCCC1 62844,n1(CCOC)nc(C)c(S(=O)(=O)Nc2ccccc2-n2nc(C)cc2C)c1C 62845,c1(CCC)nc(C(=O)N(CCC)C(C)C)cs1 62846,n1(CC)ncc(C(=O)NCC2CC(NC(C3CCCN3C)=O)C2)c1C 62847,C(C(C)(C)C(=O)NC1CN(C(c2cnnn2C(C)C)=O)CC1OC)OCC 62848,CC(CNC(=O)CCc1ccsc1)(C1CCC1)NC(=O)CCc1csnn1 62849,Cc1ccc(CC(=O)NC2(CNC(c3ccccc3OC(C)C)=O)CC2)c(F)c1 62850,S(=O)(=O)(c1cccs1)NC(C)C(=O)N1CCC1CNC(c1ccc(O)nn1)=O 62851,CCC(CC)C(C(=O)N(CC(=O)NC(c1ccc(C)s1)C)C(C)C)OC 62852,C(C(=O)N1CCC(C(=O)N(CC(CC)CO)CC)O1)N(CCC)C 62853,Cn1ccc2ccc(C(N3CC(NC(C4CCOCC4)=O)C3)=O)cc12 62854,C1(NC(C(CNC(c2c(CC)cns2)=O)N(C)C)=O)CC(C)N(C2CC2)C1 62855,c1(NC(c2cccc(Cl)c2)CC)ncnc2c1CCO2 62856,c1(-c2cn(CC3OCCN(C(C(=O)NCC)=O)C3)nn2)ccc2sccc2c1 62857,CS(=O)(=O)c1ccc(CN2CC3C(C(N4CCCCC4CCO)=O)C3C2)c(F)c1 62858,N1(C(CCNC(NC)=S)=O)CC2CCCC2(N=c2cncc(Cl)[nH]2)C1 62859,c1(C(N2CC(CC(=O)Nc3cccc(CO)c3)OCC2)=O)ccc2cccnn12 62860,Cc1oc(-c2ccccc2)nc1C(=O)NC1CCN(C(=O)CSC(C)(C)C)C1 62861,N1(CC)N=C(C(=O)NC2CCC(NC(=O)C=CC(C)(C)C)C2)CCC1=O 62862,c1(OC)cccnc1C(F)(F)C(=O)NCC1CCCN(C(=O)C(CO)N(C)C)C1 62863,N#Cc1cccc(C(=O)NCC(CNC(=O)CC2CCC(=O)N2)C(F)(F)F)c1 62864,c1(C(=O)NC2CC(NC(C3(C)CC(C)OCC3)=O)C2)cc2c(=O)cc[nH]c2s1 62865,C1(C(=O)NCCN(C(c2nocc2C(C)(C)C)=O)CC)CC=CCO1 62866,Cc1cc(CNCC2CN(c3nccc(-c4cccnc4)n3)CCO2)cc(C)n1 62867,c1(C(=O)NC(CC)CNC(=O)CN(C)CCO)c(C)c(Cl)cc(C)c1N 62868,C1(NC(c2cc(OC)no2)=O)CC2CC1CC2C(=O)N(c1cnn(C(C)C)c1)C 62869,N1(C(C2(CCOC)CC2)=O)CCCC(NC(=O)C(C)C2CCCC2)CC1 62870,N1(C(C=CC(CC)C)=O)CC(NC(=O)C=Cc2ccc(C(N)=O)cc2)C2(CC2)C1 62871,CCC(C)C(=O)NCC(=O)N(CCCCNC(=O)CCC1CCCC1)C 62872,C(=O)(C1CCOc2ccccc21)NC(C)C(C)(C)NC(c1scnc1Cl)=O 62873,C12(C(=O)NCC3(CN(C)C(C4CCCC45CCC5)=O)CC3)CCC(F)(CC1)CC2 62874,C1(C(=O)NC2C(CNC(CCN(CC(F)(F)F)C)=O)CC2)CC2CCC1O2 62875,N1(C(C(C)OCC)=O)CCC(CNC(=O)Cc2cccc(F)c2F)C(F)(F)CC1 62876,N1(C(C(C=C)(C)C)=O)CCN(C(c2cc(F)c(OC)c(Cl)c2)=O)CC12CC2 62877,C1(C(C)NC(=O)CN(C)C)CN(C(=O)CNc2cc(CO)on2)CCCO1 62878,C1(CC(=O)NCC)CN(C(=O)CN(C)Cc2ccnn2C)CCO1 62879,c1(-c2cc(C(=O)NCCCCNC(C(C)OCC)=O)on2)cccc(Cl)c1 62880,c1(C(=O)NC2COCCN(C(C3(CC(C)C)CCC3)=O)C2)cc(Cl)c(F)cc1Cl 62881,c1(C(N(C(C(=O)NCCC)C)CC2CCCO2)=O)ccc(CN(C)CCC)o1 62882,C1(N(C(C(c2cn(C)nc2)O)=O)CCO)CCCN(C(c2ccnc(S)c2)=O)C1 62883,N1(C(CSS(C)(=O)=O)=O)CCCC(NC(c2ncc(Cl)cc2F)=O)C(F)C1 62884,c1(C(=O)NCC2(NC(c3ccc(Cl)nc3O)=O)CC2)cc2nn[nH]c2cc1F 62885,C1(O)(CNC(C2CC2(F)F)=O)CCCN(Cc2cc(F)cc(Br)c2)C1 62886,C=CCC(C)C(=O)NCC(Cc1ccccc1)N(C)C(C1CC1(C)C)=O 62887,C=CCC(C(=O)NCCCCC(C)NC(c1ccc(COCC)o1)=O)OC 62888,N1(C(C(CCC)CC)=O)C(C)CC2CN(C(c3cc(Br)c(N)cc3C)=O)CC12 62889,C(N=c1[nH]c2ccc(Cl)cc2s1)C1(NC(=O)C(F)(F)C(F)(F)F)CCCC1 62890,c1(CNC2CCC(N(C(=O)Cc3ccc(Cl)nc3)CC)CC2)cnc(F)c(Cl)c1 62891,C1(NC(c2ccc(Cl)s2)=O)CCN(C(=O)C(C2CCOCC2)F)C1 62892,C(=O)(C(CNC(=O)C=C(C)C(C)C)CC(C)C)NCCC(CC)(C)O 62893,c1(C(=O)NC2CCC2NC(=O)C(O)Cc2ccc(F)cc2)coc2c1COC2 62894,c1(C(=O)OCC)nc(CNC(C2(OC)CN(C(=O)Cc3ccsc3)C2)=O)oc1C 62895,Cc1ccc2cccnc2c1C(=O)NC1CC(C)CN(C(=O)CC2CCC2)C1 62896,Cc1cc(NC(C2COC(CNC(C3CC4(CSC4)C3)=O)C2)=O)cc(C)c1C 62897,C1(NC(c2c(OC)nsc2)=O)CCN(C(=O)C=CCN(C)C)C1C 62898,N1(C(c2c(NC)nccc2)=O)C2CCC1CC(C(=O)NC1CC(C)(C)C13CC3)C2 62899,Cc1c(NC(C2CC2c2ccc(F)c(F)c2)=O)cccc1COCC(F)(F)F 62900,Cc1cnc(C(=O)NC2CC(CNC(=O)CN3CSCCSC3)C2)c(C)c1 62901,O=C(C(O)C(F)F)NCCC1CCCCN1C(=O)CCN(C1CCCCCC1)C 62902,Cc1[nH]nc2c(C(N3CC(NC(c4cn(C)c(O)n4)=O)CC3C)=O)cccc12 62903,c1(C(N(CC(C)NC(C2CC3CCC2C3)=O)C)=O)cnc2c(c1)N(C)CCO2 62904,C(=O)(C(C)C(=O)N1CCC=CC1C(=O)N(CC(O)CO)C)OC 62905,C1(NC(Cc2c(C)non2)=O)CCCCC1CNC(c1coc(Cl)c1)=O 62906,C(=O)(C(O)CC1CC1)NCCC1(C(N(CC(COC)C)C)=O)CCC1 62907,c1(C(N(C2CC(NC(C(COC)N(C)C)=O)C2)C)=O)cnn2c1C(C)CCC2 62908,C(C)(C(=O)N1CC(O)(CN(C(=O)C(C2CCOCC2)O)CC)C1)(C(C)C)NC(C)=O 62909,c1(C(N2CCC(CCC#N)CC2)=O)c(F)ccc(N)c1Br 62910,Cc1ccc(CC(=O)NC2COCCC2NC(c2cccnc2S)=O)c(Br)c1 62911,O=C1CNC(=O)C(CC(N2CC(NC(C34CCC(C3)C4)=O)C3(CC3)C2)=O)N1 62912,N1(C(C(CC=CC)C)=O)CCN(C(c2n[nH]cc2F)=O)CC1CCOC 62913,C1(NC(C(C(=C)Cl)(C)C)=O)COC2CN(C(=O)CCNc3ncccn3)CC12 62914,C1(C(N(CC(N2CCN(C(C(C=C)(F)F)=O)CC2)=O)C)=O)CCC2CCC(=O)N12 62915,c1(C(=O)NCC2OCCN(C(C=CC)=O)C2)cc(C(C)C)cc(Br)c1 62916,c1(C(=O)NCC2CCC(NC(C(CC)(C)F)=O)CC2)cc2cccc(OC)c2o1 62917,C(=O)(C(C)(C)C(C)(F)F)N(C)CC1N(C(CNC(=O)OCC=C)=O)CCOC1 62918,c1(CNC(NC(CC)CC)=NCc2ccc(C)c(Cl)c2)nc2ccccc2o1 62919,c1(OC)cc(NC(=O)NC2CCN(C(=O)Nc3cccc(C)c3)C2)cc(Cl)c1 62920,CCC(CC(=O)NCc1ccoc1C(N1CCC(OC2CC2)CC1)=O)OC 62921,c1(C(N2CC(C(=O)NC(CCCC)CO)C(O)CC2)=O)cc(F)c(F)c(F)c1 62922,c1(OCC2(NC(C(C)C(C3CCCCC3)C)=O)CC2)ccccc1 62923,c1(OC)cc2c(=O)c(C(N3CCC4(CCC(=O)NC4)C3)=O)c[nH]c2cc1Br 62924,N1(C(C2C(COC)C2)=O)CCCC1CCNC(=O)C(C)C1CCCC1 62925,c1(CC)ccc(F)cc1C(N1CC=C(CNC(=O)CNc2ncccn2)CC1)=O 62926,C(=O)(C(C)CC(C)(F)F)N1CCC(C(C)NC(c2ccc(-c3cccs3)[nH]2)=O)CC1 62927,CCC(C)CC(C)C(=O)NC1(C(N2CCN(CCO)CC2)=O)CCC1 62928,c1(NC(C2N(Cc3ncc(C)nc3)C(C)CC2)=O)c(F)cc(F)cc1Br 62929,N1(C(C2C(c3ccc(C)cc3F)C2)=O)CCCN(C(c2cscn2)=O)C(CO)C1 62930,CC1(NC(=O)C(F)C2CCOC2)CCCN(C(=O)C(F)F)C1 62931,N1(C(C(CC=C)NC(=O)Cc2ccoc2C)=O)CCS(=N)(=O)CC1 62932,N1(C(C2CN(C(C(C)NC(=O)OC)=O)CC2F)=O)CC2C3CCC(C3)C12 62933,C1(C(N(C(CC(=O)N(C)Cc2ccc(C)cn2)(C)C)C)=O)CC2(CCCO2)C1 62934,CC(O)CCCCCC(=O)N1CCCC1C(C)(C)NC(c1ncccc1Br)=O 62935,N1(C(c2ncc[nH]2)=O)CCCCC2(CCN(c3ncnc4c3COC4)C2)C1 62936,CC(C)(CCC(=O)NCC(c1ccccc1F)NC(c1cnsn1)=O)[N+](=O)[O-] 62937,c1(C(=O)NCC2CC(C)N(C(=O)C=Cc3cncs3)C2)cccc2sccc12 62938,c1(C(=O)NCC2(CNC(c3c(OCC)nccc3)=O)CC2)ncc(N)nc1C 62939,C1(C(=O)NC(CCOC)(C)C)CN(C(=O)C(C)C(C)(C)C)C2(CCC2)C1 62940,C1(NC(=O)Cn2ccc(C(F)F)n2)CCCCN(C(C2OCCCO2)=O)C1 62941,C(=O)(CCCC(=O)N(C)C)NCC(C)(CO)NC(C(COC(C)=O)C)=O 62942,N1(C(C(C)SCC)=O)CCC(NC(c2ccc3c(c2)CCC=C3)=O)C(F)(F)CC1 62943,C1(CN(C(=O)C(F)C2CCCC2)CC)CCCN(C(C2CC2C(C)C)=O)C1 62944,C(CCC(C)(C)C(=O)NCCc1ncn(C)n1)NC(CC(=O)OC)=O 62945,Cc1cc(C(N2CCC(CNC(=O)CCc3nnc(C)o3)C23CC3)=O)cc(N)c1 62946,c1(CNC(=NCCCN2C(=O)OCC2)NCC(F)F)cc2c(s1)CCCC2 62947,N1(C(C(C2N(C(C(CN(C)C)O)=O)CCC2)(C)C)=O)CC(O)C(O)C1 62948,c1(CC)ccc(NC(c2ccc(F)cn2)c2nnnn2CCOC)cn1 62949,C1(NC(c2c(C(C)=O)ccs2)=O)CN(C(C2(C3CCC3)CC2)=O)C2(CCOC2)C1 62950,Cc1ccc(C(F)(F)F)cc1C(=O)N(C1CN(C(=O)C(O)CNC(=O)CO)C1)C 62951,C1(NC(CN2C(C)CCCC2)=O)CCCC12CN(C(=O)Cc1cncn1C)C2 62952,C1(C(N(C)CC2OCCN(C(CSCC(C)C)=O)C2)=O)CCC(N=[N+]=[N-])CC1 62953,c1(C(N2CC3(CN(C(C=CS(CC)(=O)=O)=O)C3)C2)=O)cc2ccc(Cl)cc2s1 62954,c1(C(=O)NCC(C)CN(C(=O)C(C)NC(N)=O)C)cc2ccccc2nn1 62955,C1(NC(C2(C)CCN(C(c3cnn(C)n3)=O)C2)=O)CCOC12CCCC2 62956,c1(C(=O)NC2C(CC)CN(C(C3(C)CCCOC3)=O)C2)ccc(Cl)c(Cl)c1 62957,CCCCC#CC(C)(C)NC(C1CN(C(C2(C)CCCC2O)=O)CC1C)=O 62958,C1(C(N(CCCNC(=O)C#CC2CCCC2)CC)=O)CCCN1S(=N)(=O)N(C)C 62959,c1(C(=O)NC2CC3(CN(C(CCSCCC)=O)C3)C2)nccc(C#N)c1F 62960,C(=O)(C(CC)CCOC)NC1(CC=C)CCN(C(=O)C=CCOC)C1 62961,C(CC(C(C)(C)C)NC(C1(C)C=CCC1)=O)N(C(c1c(OC)scc1)=O)C 62962,C1(NC(C(CSC)c2ccccc2)=O)CN(C(c2ccc(=N)[nH]c2)=O)CC1(C)C 62963,Cc1ccc2c(c1)C=C(C(=O)N(CC(C)CNC(=O)CCCC(N)=O)C)CO2 62964,c1(CCC(=O)NCCNC(CNS(C)(=O)=O)=O)ccc(F)cc1Cl.N12CC(C1)C2 62965,C1(CNC(=O)NC2CCN(Cc3cccnc3)CC2)CC2C=CC1O2 62966,C(=O)(C(O)C(C)(C)C)NC(C)CC1CN(C(=O)C(F)=C2CCCC2)C1 62967,C1(C(=O)NCC(C2(O)CN(C(C=CCC)=O)C2)(C)C)CC2(CCCCC2)C1 62968,C1(CC)CN(C(C23CC4CC2C3C4)=O)CCC1NC(C1(C(F)F)CCOCC1)=O 62969,C(=O)(CCC(C)CN(C)C)NCC(c1cccc(C)c1)NC(CN(CCC)C)=O 62970,Cc1cccc(C(O)CN(C(=O)CC2CCCC(=O)N2)C)c1 62971,C(=O)(N1CCC(C(=O)NCC2CC3(CCC3)C2)O1)C1(C=C)CCC1 62972,C1(N(C)C(C2CCCS2)=O)CN(C(c2c[nH]c(C#N)c2)=O)CC12CC2 62973,N1(C(C2(OC)CCCC2)=O)CC(CNC(c2scnc2C(C)C)=O)OC(C)(C)C1 62974,C1(CNC(CC)=O)CC2CC1CN2C(=O)COCc1cccc(C)c1 62975,N1(C(Cc2c(C)noc2)=O)CC(C)N(C(=O)CN(C)C2CC2)CC1C 62976,C1(c2nnnn2CCCOCC(C)C)(NC2(CSC)CC2)CC2CCOC12 62977,c1(C(=O)NCC2(O)CCN(C(C3CC(SC)C3)=O)C2)cc(=O)n2nccc2[nH]1 62978,c1(CNc2c(OC)cc(F)cn2)cc2cccc(-c3cn[nH]c3)c2s1 62979,N1(C(C(C#C)(C)C)=O)CCC(C)(C)C(CNC(=O)COc2ccc(OC)cc2)C1 62980,C1(C(N2CCC(CCN(C)C)C2)=O)CC2(CCN1C(=O)C(Cl)Cl)CC2 62981,c1(CC(=O)N(C(C)CCNC(=O)CO)C)cc(F)c(N)cc1F 62982,C1(NC(C(C)SCC)=O)CCCCC12CCN(C(c1n[nH]cc1C1CC1)=O)CC2 62983,CC(C)(C)CC(O)C(=O)NC12CCCCC(NC(C3COCCO3)=O)(C1)C2 62984,O=C1NCCc2occ(C(N3CCCC(c4cn(C5CC(O)C5)nn4)C3)=O)c21 62985,Cc1nc2cccc(C(=O)N(CC3=CCCOC3)C)n2n1 62986,c1(C(=O)NC(COC)CNC(=O)CC2CCC(C)(C)C2)c(F)ccc(N)c1F 62987,C(=O)(C(CC)C(F)(F)F)N1CCC(n2cc(CNC(C(C=C)CC)=O)nn2)CC1 62988,CC(CC(F)F)C(=O)NC1(CNC(=O)CC2CN3CCN2CC3)CCCC1 62989,C1(CC(=O)NC(C)(CSC)C2CC2)CCCCC1NC(c1ccc(SC)o1)=O 62990,C(CCSC)(C(=O)N(CC(O)CNC(C1(c2cc[nH]n2)CC1)=O)C)OC 62991,N#CC1(CC(=O)NCC2CC2CC(=O)NCCSCCO)CC1 62992,C1(C(N(CCn2cc(C(c3ccccc3)C)nn2)CC)=O)CCn2ncnc2C1 62993,O=C(C#CC1CCOCC1)NCCN(C(c1ccc(CO)o1)=O)CC1CCCC1 62994,N1(C(C(C)OCC)=O)CC2(CNC(c3ccc(C)nc3O)=O)CCC1CC2 62995,N1(C(c2c(O)ccc(C)c2)=O)CCCN(C(c2sc(C)cc2C)=O)C(C)C1 62996,N1(C(C2(C#N)C(C)(C)C2)=O)CC2(CC(C(N3CCOC(C#N)C3)=O)CO2)C1 62997,c1(C(=O)NCC(C2CCC2)NC(C(C=C=C)C)=O)cnc(C)c(C)c1 62998,N1(C(c2c(OC)cncc2)=O)CC2CN(C(C3CC34CCCCCC4)=O)CC2C1 62999,C(=O)(C(C#N)C(C)C)NCCN(C(C(C)OC)=O)CCCN(C)C 63000,c1(OC)cc(NC(C2CC2NC(=O)Cc2ncccn2)=O)c(Br)cc1F 63001,C1(NC(CCOCC(C)C)=O)C2CC(O)C1N(C(C1(C)CC(=O)N(C)C1)=O)C2 63002,Cc1cc(NC(C2(CO)CCCO2)=O)ccc1NC(C1COC2(CCC2)C1)=O 63003,c1(CC)nc(=N)[nH]c(=NCC2CC3CCC2N(C(=O)Cn2ccnc2C)C3)[nH]1 63004,CC(C)CC(C)CC(=O)N1C(C(=O)NCCCC(O)CO)CC1C 63005,N1(C(C2CCN(C(c3c(C)nc(O)cc3)=O)C2(C)C)=O)CCCN(C)CCC1 63006,c1(C(=O)NC(CC)CNC(c2cc(COC)on2)=O)c(C)noc1CC 63007,CC(C)CC(C(=O)N(C)CCN1CCCCC1)N(C(=O)C(C)n1cccc1)C 63008,C1(CN2CCC(CNC(c3c(C)snn3)=O)C2)CCS(=O)(=O)CC1 63009,C(=O)(C1COc2ccccc21)NCC(CCNC(c1nc(Cl)cs1)=O)O 63010,S(=O)(=O)(CCC(=O)N(C(C(=O)NCC1(C)CNC(=O)O1)C1CC1)C)NC 63011,Cc1cc(CC(=O)NC2C=CC(CNC(=O)CC(C)(C)F)C2)cc(F)c1 63012,C=C(C)CCCC(=O)N1CC(C(O)C(=O)Nc2cscc2C)C1 63013,c1(C(=O)NC(CN(C)C)C(=O)NCc2ccnc(F)c2F)ncnc(O)c1F 63014,C1(CNC(C2N(CC)CC2)=O)CCC2(CN(C(c3oc(Br)cc3C)=O)C2)O1 63015,CC1(CNC(c2cnc(O)s2)=O)CCN(C(C2(N3CCCC3)CCC2)=O)CC1 63016,c1(C(C)C)cnc(O)c(C(N2CC(C(C)NC(C3CN(S(C)(=O)=O)C3)=O)C2)=O)c1 63017,C1(CNC(C(CC)C#N)=O)CN(C(c2cc(Br)no2)=O)C2(CCC2)C1 63018,C1(C(=O)NC2(C)CCN(C(Cc3cc(C)no3)=O)C2)CC(=O)NC1(C)C 63019,N1(C(c2c(C)nn[nH]2)=O)CC(C)CN(C(=O)CN2CCCOC2=O)CC1C 63020,c1(C(N2C(C(=O)Nc3cn(C(C)(C)C)nc3)CC3CC32)=O)cc(F)c(F)cc1I 63021,C(=O)(CC(O)CC(C)(C)C)NC1C(NC(C=Cc2c(C)cccc2)=O)C1 63022,C1(NC23CC(NC(c4nc(SC)oc4C)=O)(C2)C3)CS(=O)(=O)CC1C(F)(F)F 63023,c1(C(=O)NCC(C(C(C)C)C)NC(c2cccnn2)=O)cc2ccc(Cl)cc2o1 63024,N1(C(CCCOCC)=O)C2CCC(C2)C1C(=O)NCc1ccc(O)nn1 63025,N1(C(CCCCN(C(=O)Cc2cc[nH]c2)C)=O)Cc2cccc(F)c2C1 63026,c1(NC(c2cc(CNC(=O)CC3CCCCC3)ncc2)=O)cccc(F)c1F 63027,c1(C(=O)NCCCNC(=O)Cc2cccc(F)c2)nc2cc(F)ccc2s1 63028,C1(NC(NCC2CC(F)(F)C2)=S)CCC(F)(F)C1 63029,N1(C(CN2C(C)CC2)=O)C(C(NC(=O)CCn2cc(Cl)cn2)SC)CC2COCC12 63030,N1(C(C2N(C(C(C)(O)C3CC3)=O)C(C)C2)=O)CCc2cnccc2C1 63031,c1(C(N2CC(NC(c3c(C)scn3)=O)C(C)(C)C2)=O)cnc2c(c1)CCC2 63032,N1(C(c2ccc(C(C)(C)C)s2)=O)CC2CC1CN(C(=O)CC#N)C2 63033,C1(NC(CS(N)(=O)=O)=O)CCN(C(c2ccoc2Br)=O)CC12CCC2 63034,N1(C(=O)C=Cc2ccncn2)CC2CC(C1)CN(C(=O)Cc1ccno1)C2 63035,c1(C(=O)NC(CCNC(C(C)C#N)=O)(C)C)cc2c(ncn2C)s1 63036,c1(CNC(C(N2CCCC(C)C2)=O)=O)n[nH]c2c1CN(C(c1cnco1)=O)CC2 63037,CCCC(C(=O)N1CC2CC1C2NC(c1ccc(CN(C(C)=O)CC)o1)=O)N(C)C 63038,C1(C(=O)NC2(C(=O)Nc3c(CC)n(C)nc3)CCCCC2)CC(C)CC(C)C1 63039,C1(CCC)CCC(C(=O)NC2CCN(C(c3cc(Br)nn3C)=O)C2C)CC1 63040,C(CNC(=O)C(F)(F)c1ccnn1C)(CC)(CC)NC(c1ccc(CC)s1)=O 63041,c1(OC)cc(CC(=O)NC(C)CCCCNC(=O)CN2CCCC2C)ccn1 63042,c1(C(=O)NC(CNC(CNC(C)=O)=O)C2CC2)cc(=O)c2ccccc2[nH]1 63043,C1(C(N2CCSCC2)=O)(NC(C2C=CCCC2)=O)CCOCC1 63044,Cc1csc(C(=O)NC2CN(C(c3cnoc3C3CCC3)=O)C2)c1Br 63045,c1(C2(C(=O)NCC3(F)CC(CNC(C4C5COCC45)=O)C3)CC2)ccccc1F 63046,C1(NCC(COC2COCC2)(C)C)CCC(=O)N1C 63047,c1(C(=O)NCc2ccc(OC)nc2C)c(F)ccc2c1OCO2 63048,C1(C)(N(c2cc(-c3ccn(C(C)C)n3)[nH]n2)S(=O)(=O)C(C)C)CCS(=O)(=O)C1 63049,C#CCCCC(CC)OC(C1CC(C(=O)OC(C)(C)C)C1)=O 63050,C1(CNC(=O)CCc2cccnc2Cl)CC12CCN(C(C1CCC1(F)F)=O)CC2 63051,c1(CC(=O)OCc2ccc(C(=O)OC)cc2)cccc2ncccc12 63052,N#Cc1cnc(C(N2CC3CC(NC(C4CCC(=O)NC4)=O)CC3C2)=O)c(Cl)c1 63053,c1(C(=O)NCc2cc(Cl)cnc2Br)cc(Br)cc(F)c1O.C12CCCN(C1)C2 63054,CCC(C)CCC(=O)N1CCCCC1CCNC(c1cc(C)on1)=O 63055,c1(COC)nc(NC2(C3CC3)CCC2)cc(N(CC(O)CN(C)C)C)n1 63056,c1(C(=O)NC2CCCN(C(Cc3cc(C)[nH]n3)=O)C2C)ccc2c(c1)CCOC2 63057,c1(-c2cn(CC(CNC(C3C(OCC)CC3)=O)(F)F)nn2)ccccc1N(C)C 63058,C1(C(=O)NCc2c(C(=O)NC(C)(C)CCCF)n(C)nc2)CN2CCC1CC2 63059,c1(CNC(C(C(C)C2CC2)N2CCC(CC3CC3)C2)=O)csc2c(F)cccc12 63060,c1(OC)cc(C(N2CCC(c3cn(CC4COCCO4)nn3)C2)=O)cnc1Cl 63061,c1(C(N2CCC(C)(C(=O)NCC(N3CCCCC3)=O)C2)=O)cc(F)cc(I)c1 63062,C1(C2CN(NC(C(C(C)C)O)=O)C2)(CCn2cc(CN3CCCCC3=O)nn2)CC1 63063,C=CC1OCCC1C(=O)NCC(C1CCCC1)NC(C1(CO)CCCO1)=O 63064,c1(NC(C)=O)ccc(C(=O)NC23CC2CN(C(c2cc(=O)n(C)o2)=O)C3)cc1F 63065,C12CCCC3(CCN(CC3)C1=O)O2.C(CC(=O)NC(C1CC1)C1CC1)OC(C)C 63066,C1(C(N(CCN(C)C(c2ccc(CC(C)(C)O)s2)=O)C)=O)C(F)(F)C12CC2 63067,c1(C(C)(C)C(=O)NCC2(CNC(C3CCCOC3)=O)CC2(F)F)cccc(F)c1 63068,c1(C(=O)NC2CN(C(C#CC3(C)CC3)=O)CC2(C)C)ccc2ncccc2n1 63069,Cc1ccc(CC(N2CCC(F)C(NC(c3cc(Cl)c(Cl)cn3)=O)C2)=O)cc1C 63070,N1(CCCC)CC2CCC(NC(c3ccc4cc(C)cn4c3)=O)CC2C1 63071,C12(C(=O)NCCC(C)N(C(CC(CCC)(C)C)=O)C)CCCN(C1)S(=O)(=O)C2 63072,c1(C(=O)NC2CC(N(C(CCC(C)N(C)C)=O)C)C2)nn(C)c2ccc(F)cc12 63073,n1(CC(N2CC3C(N(C(C(C)NC(=O)NC)=O)C)C3C2)=O)ccc(=O)n(C)c1=O 63074,CCC(C(=O)OC)C(=O)NC1COCCC1NC(c1cnn(CC2CC2)c1)=O 63075,c1(NC(c2cnn(C)c2)CC)ccc(S(=O)(=O)NCCc2n[nH]c(=N)s2)c(Cl)c1 63076,Cc1c(C(=O)NCC2(O)CCN(C(C3(C)CCCOC3)=O)C2)ncn1C 63077,N1(C(c2c(Cl)cn(CC)n2)=O)CCC2C(CCN2C(=O)C(O)C2CCCC2)C1 63078,Cc1cnccc1C=CC(N1CC=CC(NC(C2CCNC(=O)C2)=O)C1)=O 63079,C(CC(Cc1ccco1)NC(C1(n2cc(CCCCO)nn2)CCC1)=O)OC 63080,N1(C(c2ccn(CC)n2)=O)CC(OC)CC1CNC(=O)C1=CCCS1 63081,N1(C(c2c(Cl)nc(N(C)C)s2)=O)CC(CNC(=O)C(C)(O)C(C)C)CC1(C)C 63082,C12(C(=O)NCCC(C)NC(=O)C=CCOC3CCOCC3)CCOC(C)(C1)C2 63083,c1(C(N2CCOCC2c2cn(Cc3csc(Br)n3)nn2)C)cccc(C(F)F)c1 63084,CC1Cc2cc(S(=O)(=O)N(c3ccc(Cl)cc3)CC3CCCCC3)cc(Cl)c2O1 63085,C1(C)(OC)C2CC1CN(N1CCC3(CCC3)C(O)C1)C2 63086,C1(NC(c2c(OCC)cncc2)=O)CN(Cc2ccc(O)c(F)c2)CC(F)(F)C1 63087,CC(CN(C)C)CCC(=O)NCC1CC(C)(C)CN1C(C12CSCC1C2)=O 63088,c1(C(N2CCC(NC(CCOCCC)=O)C23CCC3)=O)ccc(S(C)(=O)=O)cc1 63089,C(=O)(C(C)(COC)OC)NC(CN(C(C=NOC)=O)C)Cc1ccccc1 63090,c1(C(N2CC(NC(c3c(OC)ccs3)=O)C(F)C2)=O)ccc2c(c1)nc(C)n2C 63091,N1(C(C(CNC(C2CC(=C)C2)=O)O)=O)CCC2(CCCO2)C1 63092,C1(CC(=O)NC(C(C)C)(C)CNC(=O)CCc2nncs2)CCCCC1(C)C 63093,CC(CC(F)(F)F)C(=O)N1CC(C)(C)CC1CC(N1CC2C(C1)C2(F)F)=O 63094,C1(C(C(=O)NC(CC)(C)C)N(C(C)CC(N)=O)C)CCCC1O 63095,c1(C(=O)NC(C2(C)CC2)CO)csc(CNC(=O)CN2CCOCC2)c1 63096,C1(C(N(CC(COC)O)C)=O)(CO)CCCN(C(c2cc(C)co2)=O)C1 63097,Cc1nc(CN2CCCC(CN3CCCCC3)C2)c(Br)[nH]1 63098,C(C(O)C(=O)NC(C1(C(=O)N(C)CC2CCCN2C)CC1)C)SC 63099,c1(CN2CC3N(C(c4cc(C(C)C)[nH]n4)=O)C(C3)C2)ccc(N)c([N+](=O)[O-])c1 63100,N1(C(c2cc(CNC(C3CN4CCN3CC4)=O)ncc2)=O)CCCCCC1CO 63101,c1(OCCCC)ccc(C(=O)NCCC(C)CCNC(C2CCS2(=O)=O)=O)cc1 63102,C1(CCC(=O)N(C2CCN(C(=O)Cc3nncn3C)C2)CCC)CCCCO1 63103,c1(NC(C(CNC(C(C)C2CCCC2)=O)N(C)C)=O)cn(C)nc1C(N)=O 63104,N1(C(C(C)=CC(C)(C)C)=O)CCC(CC(N2CC(F)C2)=O)C1 63105,N1(C(c2c(C)con2)=O)CCCC1C1CCCN1C(c1cc(Cl)cc(F)c1N)=O 63106,c1(OC)ccc(CC(=O)N(CC(O)CNC(c2ocnc2C)=O)C)cc1F 63107,C1(F)(CNC(=O)Cc2cccc3sccc23)CC2CCC(C1)N2C(=O)CCF 63108,Fc1cc(F)c2nc(Cl)nc(N3CCC4(CC3)CC(N3CCCOCC3)C4)c2c1 63109,c1(CO)cccc(C2(CO)CC2)c1.c1(C(c2ccsc2)N)nnnn1CCC1CC1 63110,C1(CC=C)(NC(=O)Cn2nnc(SC)n2)CN(C(=O)CCNC(N)=O)C1 63111,C1(N(C)C)CCC2CN(C(c3ncc(F)cc3F)C(=O)NCC3CC3)CC12 63112,CC(C)C(CC(=O)NCC1(CO)CCCO1)NC(C1CC2(C1)CC2(F)F)=O 63113,Cc1ccc(C=CC(=O)NCCCCNC(c2nocc2C(C)C)=O)cc1Cl 63114,C1(C(N2CC(O)(CC=C)C2)=O)CC(F)CN1C(C1CC(C)=NO1)=O 63115,C(CC1=CCN(C(c2ncn3cccnc23)=O)CC1)NC(C1C(C)C1)=O 63116,C#CCCCC(=O)N(C)CCOCCCN(C)C(C1CCC(CCO)CC1)=O 63117,C12(C(N(CCC(C)NC(=O)CCc3nc[nH]n3)C)=O)CCCCN1CCC2 63118,CC1(C)CCC(C(N2CCC23CCCSC3)=O)CN1C(=O)Cn1cnnn1 63119,Cc1cc(CNC(C2COCCN(C(C3CCC=CCCC3)=O)C2)=O)nnc1C 63120,COn1cnc(C)c1C(=O)NCC(CC(C)C)NC(C1CC(CN(C)C)C1)=O 63121,C(CCCC(C)(c1nnnn1C1CCOC1)NCc1ncc(Br)s1)OC 63122,N1(C(CC2=NNC(=O)C2)=O)CC2C3CCC(C2C1)N(C(C1CCCOC1)=O)C3 63123,c12cccc(n1)C2.c1(C(=O)OC(C)(C)C)[nH]ccc1CNc1ncc(CO)s1.OC 63124,c1(C(=O)NC2CN(C(CCNC(C)=O)=O)C2)c(C)ccc(F)c1N 63125,C1(CNC(CC2(OC)CC2)=O)CC(NC(=O)Cc2sccc2C)C12CCC2 63126,c1(C(=O)NC2C(N(C(C(C)c3ccsc3)=O)C)CCCC2)cc2n(n1)CCCO2 63127,N1(C(CN(C)C(N)=O)=O)CCCCC(CNC(C23CCCC2C3)=O)CC1 63128,c1(CCC(=O)NC2CC(C(=O)NCC3(CCOCC)CC3)C2)ccc(F)c(Cl)c1 63129,C1(NC(C=C(C)C)=O)CN(C(=O)Cc2cccc3ncccc23)CCC12CCC2 63130,CC1(C)NC(=O)CC1C(=O)NC1CCCN(C(c2cnn(C(C)(C)C)c2)=O)CC1 63131,C1(C(N(C2CCNC2=O)CC)=O)CN(C(C2CC3CC(=O)C2C3)=O)CC1(F)F 63132,C1(CC)CN(C(C23CCC(CC2)C3)=O)CCN1C(c1ccc(C(O)CF)cc1)=O 63133,c1(COC)occc1C(=O)NC1CCC1CNC(c1cc(C(=O)OC)co1)=O 63134,N1(C(C2(C=C)CC2)=O)C(CNC(=O)C(C)Sc2ccc(F)cc2)CC2CC12 63135,c1(OC)cc(C(C(=O)NC2CC2)N(C2CCN(C(C)C)C2)C)ccc1OC 63136,CC(C)S(=O)(=O)C(C)C(=O)N(C)CC1(O)CN(C(C2C(F)(F)C23CCC3)=O)C1 63137,c1(C(N2CC(NS(C(C)C)(=O)=O)C2)=O)ccc2nc(Cl)sc2c1 63138,C=C(C)C(C)(C)C(=O)N1CCC(CO)C(NC(c2ccc(C(F)F)c(F)c2)=O)C1 63139,n1(C(C)C(=O)NC(C(=O)OC(C)(C)C)C2CCCC2)cc(C2CC2)nn1 63140,c1(C(=O)NCCCCNC(C2CC(C)(C)O2)=O)ccn2ccccc12 63141,N1(C(C2(OC)CCOC2)=O)CCCC(NC(=O)COCc2cc(C)on2)C1 63142,c1(SC)ccccc1C(=O)N(C1CN(C(=O)CCc2ccc(Cl)nc2)CC1O)C 63143,N=S1(=O)CCC2(CC1)CN(C(=O)C(N)Cc1ccco1)CCO2 63144,N1(C(CSCC(C)=O)=O)CCC(N(C(=O)CN2CC=CC2)CC2CC2)C1 63145,CCCC(CCC)C(=O)N(CC(C)NC(=O)CNC(c1cc2c(s1)CCC2)=O)C 63146,C=CCC(CN=c1[nH]c(=NC)[nH]c(=NCC(C)n2ccnn2)[nH]1)c1ccccc1 63147,C1(CNC(CCN(CC)CC)=O)CC2(CN1C(=O)CCC1CC1)CC2(F)F 63148,c1(CC(C)C)cc(C(=O)NC2CCCC2NC(c2ccc(Cl)o2)=O)n(C)n1 63149,C#CC1(N(C)C)CCN(C(C(=O)NCCCC)C2CC2(C)Br)CC1 63150,c1(C(N2CC3C(N(C(c4cn(CC)nc4C)=O)C)C3C2)=O)c(F)cc(N)cc1F 63151,c1(C(N2C(c3cn(C)nc3)C(C)(C)C2)C(=O)NC2CC2)cc2ccc(Cl)cc2o1 63152,c1(C(=O)NCC23N(C(c4c(C)nccn4)=O)CCC2CC3)cc(F)c(Cl)cc1F 63153,C1(C(N2CCC(C(C)(C)NC(c3c(C)noc3C)=O)C2)=O)CC2(COCCO2)C1 63154,C1(CNC(=NCC=C)NC(C)CC)CS(=O)(=O)c2ccccc2O1 63155,c1(C(=O)NC(CCCNC(c2c(CC)con2)=O)C)cc(O)c2ccccc2c1 63156,N1(C(CCCCOC)=O)CCCCC2(C1)CN(C(c1[nH]c(C)nc1C)=O)C2 63157,c1(C(=O)NN2CCCC2CNC(C2CC(CF)C2)=O)ccc(OC(F)(F)F)cc1 63158,c1(C(N2CCc3nc[nH]c3C2)=O)cn2cc(-c3cccc4cc[nH]c34)ccc2n1 63159,c1(C(=O)OC)nn(C)c(CC)c1N=c1cc[nH]c(C2CC2)n1 63160,CCCCCCC(C)CC(=O)NC(CNC(=O)C(=O)NC(C)C)C1CCC1 63161,c1(C(N2CCC(F)(CNC(C(CC)O)=O)C2)=O)cc2c(C)sc(C)c2s1 63162,C1(OC)(CNC(=O)C(F)CC(C)C)CCN(C(c2ccccc2C)=O)CC1 63163,C(=O)(C(CC(C)(C)C)OC)N(CCOC)CCNC(C1CCC(C#N)CC1)=O 63164,C1(CNC(c2c(C)sc(Cl)n2)=O)CN(C(c2n[nH]cc2C2CCC2)=O)CCN1C 63165,N12CCC(C(F)(F)CC1)CNC(=O)Nc1c(OC)ccnc1C2=O.C(C)(C)(C)OC 63166,c1(SC)cc(CN(C)C(=O)NCC2CCCN2C2CC2)cc(Cl)c1 63167,C1(C(=O)Nc2cn(CCC#C)nc2)CCCN(C(=O)C(C)=C2CCCC2)C1 63168,C(CNC(=O)CCn1ccnn1)(CCCC)NC(C1C(C#C)C1)=O 63169,N=c1nc(N2CCCC(c3nncs3)C2)[nH]c(=NCc2ccccc2C(F)F)[nH]1 63170,N1(C(C(CC(C)C)O)=O)CC(CNC(c2nc(=N)cc[nH]2)=O)CC12CCOCC2 63171,c1(N2CCC(CCOC)(NC(C3CN(C)CCO3)=O)C2)ncccc1[N+](=O)[O-] 63172,c1(C(N2CCN(C(=O)C(O)CN(C)C)C(CCO)C2)=O)c(F)cccc1F 63173,C1(CC)CCCC1C(=O)NCCC1(OC)CN(C(c2ccc(CO)s2)=O)C1 63174,c1(C2(C(=O)NC(C(C)NC(Cc3nnc(C)s3)=O)CO)CC2)cc(F)ccc1F 63175,c1(C(=O)NCC2CC(NC(C(C3CCCC3)OCC)=O)C2)ccn2nncc2c1 63176,c1(C(=O)NC2(C)CN(C(=O)C(C)(C)c3ccn(C)n3)C2)scc(Cl)c1Cl 63177,c1(C(=O)NC2C(C)CN(C(=O)CCC(F)F)C2)n[nH]c2c1CC(C(C)(C)C)CC2 63178,C(=O)(C(C)C(C)(C)c1ccccc1)NC(CNC(c1c(C)c[nH]n1)=O)CC(C)C 63179,C1(NC(CC=C=C)=O)CC(OC)CN(C(c2nc(-c3cnn(C)c3)oc2C)=O)C1 63180,C1(NC(C2C=C(C)CS2)=O)COC2(C1)CN(C(c1ccc(C3CC3)o1)=O)C2 63181,Cn1cc2cc(C(=O)NCCC(C)(C)CNC(c3c[nH]c(=N)o3)=O)ccc2n1 63182,C1(CNC(CC2(C=C)CC2)=O)C2CCC(C2)N1C(c1cccc(N(CC)CC)c1)=O 63183,c1(C(=O)NCCOC2CCN(C(C(COC)(C)O)=O)C2)cc(Cl)c(C)cn1 63184,C(=O)(CC1COc2ccccc21)N(C)CCOCCNC(c1ccc(O)nc1)=O 63185,c1(C(=O)NC(C(CCc2ccccc2)NC(COCC)=O)C)cc2sccc2s1 63186,C1(C(=O)NC(C(=O)NCC(C#C)OC)CC2CC2)CCCC(O)C1 63187,c1(C(N2CCC(N(C(=O)COCC3CCOCC3)C)C2)=O)c(Cl)nsc1Cl 63188,C#CCCCCCC(=O)NC1CCC(NC(=O)CC2CCN(C)C2=O)CC1 63189,c1(N2CCN(CC)CC2)nc(NC(c2nccn2C)C)nc2cc(C)ccc12 63190,N1(C(CC(CC)SC)=O)CC(NC(c2conc2C2CC2)=O)CC12CCOCC2 63191,N1(C(c2c[nH]c(=N)o2)=O)CCC2(C1)CN(C(c1cscc1Br)=O)CCO2 63192,N#Cc1c[nH]c(C(=O)NC2CN(C(C3CC34CC4)=O)CC2n2cccn2)c1 63193,Cc1ccc(C=CC(=O)NCC2(CCNC(C34COCC3C4)=O)CC2)cc1C 63194,N1(C(C(C(C)C)OC)=O)CC(C(=O)NCCc2ncccc2F)C(C2CC2)C1 63195,N1(C(CC(CC)(F)F)=O)CC2CCCCC2(CNC(=O)CCc2cnc[nH]2)C1 63196,CON(CCC(=O)NCC1CC2CCC1O2)C(=O)c1ncc2ccccn12 63197,C1(C(=O)OC)C2CCC(C2)N1C(=O)Cn1cc(F)ccc1=O 63198,Cc1ccc(C=CC(N2CCC(C(O)CNC(c3cnc[nH]3)=O)CC2)=O)o1 63199,C(CCCCC(=O)NCC1=CCCC1)N(C(=O)C(F)CC1CCOC1)C 63200,CCCC(C)(C)CC(=O)NC1CC=C(C(=O)NC(c2ccnn2C)CC)C1 63201,CCCCC(C)CCC(=O)NC(CCC)C(O)C(=O)Nc1cc(O)cc(F)c1 63202,C(C)(C(=O)N(O)Cc1cn(C2CC(O)C2)nn1)Oc1ccc(C)cc1 63203,c1(CNC(CCOCCC)=O)nc(C)c(C(N2CCSC(C)C2)=O)o1 63204,N1(C(c2c(C)nc(Br)o2)=O)CC2(CCN(C(c3cccc4[nH]ccc34)=O)CC2)C1 63205,c1(OC)cccc2c1C(C(=O)N1CC(OC(=O)C3CC3)C1)CC2.C1(F)CC2(CCC2)C1 63206,N1(C(C(C)Sc2nccn2C)=O)CCCC(O)(C(C)NC(c2cnn(C)n2)=O)C1 63207,C(=O)(CCCCO)NCC(=O)NCCCCC1CN(C(CSSC)=O)C1 63208,Cc1ccc(F)c(C(=O)NC2CC(C(F)F)(NC(c3cnc[nH]3)=O)C2)c1 63209,c1(OC)cnc(C(=O)NCC2CCN2C(C2CC(O)C2)=O)cn1 63210,CCC(C)(C)C(O)C(=O)NCCC1CCN(C(=O)C(C)CN2CCCCC2)CC1 63211,c1(OCC)cc(C(=O)NCC(C2CC2)N(C)C(c2ccsc2C)=O)ccc1C 63212,N1(C(C2(COC)CC=CCC2)=O)CCCC(N(C(=O)COC(F)F)C)CC1 63213,c1(C(=O)NCCn2cc(C(c3ccccc3)O)nn2)ccc2[nH]nc(O)c2c1 63214,C12(C(=O)NCCN(C)C(c3sc(N(C)C)nc3Cl)=O)CCC(F)(CC1)CC2 63215,c1(C(=O)NC2C(NC(CCNC(=O)C=CCl)=O)CCC2)nccc(Cl)c1Cl 63216,c1(OC)ccc(C(N2CC(C)CC2C(N2CC(NS(C)(=O)=O)C2)=O)=O)cn1 63217,C1(CC(C)C)CN(C)CCN1C(=O)NC1CCC(O)C(C)C1 63218,c1(OC)ccccc1CC(C(C)C)NC(=O)CCCn1cccc1 63219,c1(N2CCC(N(C)C(C3(Sc4ccccc4)CC3)=O)C2)ncccc1C#N 63220,N1(C(CCCC)=O)CC2ON=C(CNC(c3cn(-c4cncc(F)c4)nn3)=O)C2C1 63221,C1(NC(c2cc(C(C)=O)oc2)=O)CC2CC(C1)N(C(C1CC=CCC1)=O)C2 63222,O=C(C(F)C(F)(F)F)NC1CC2(C1)CN(C(=O)CCc1ccc(Cl)cc1)C2 63223,N12CC3CCCC3(C1)C2=O.Cc1ccc(NC(=O)C(F)C(F)(F)F)c(C)c1 63224,N1(C(C(C)(C2(C)CC2)OC)=O)CC2C(CNC(C3CCC=CCC3)=O)C2C1 63225,CC1N(C(=O)C(C2CCNCC2)F)CCCC1(C)C 63226,c1(SC)ncc(Br)c(=NC2CC2C(=O)NCCn2nc(C)nc2C)[nH]1 63227,N1(C(c2c(C)coc2)=O)CCC2(CC2)CC1C(=O)NC1CC2(CCC2)C1O 63228,Cc1cnc(C(=O)NC2(C)CCCN(C(C3CCOC(=O)CC3)=O)C2)c(Br)c1 63229,C1(OC)CC(NC(=O)CN(C)C(C)C)C12CCN(C(c1cccc(N)n1)=O)CC2 63230,C1(CCC(N2CCCC2Cc2cn(CCOCCO)nn2)=O)(OC)CCCC1 63231,N#Cc1cccc(C#N)c1N1CCC12CCCOCC2 63232,O=C(C1=CC2C=CC(C1)C2)NCCCC(O)C(=O)NCCCC(F)F 63233,Cc1cncc(C)c1C(=O)NCC(O)CNC(=O)C(c1ccccc1)F 63234,C12(CNC(C3C(C)CC3)=O)CCC(CC1)N(C(c1cnn3ncccc13)=O)C2 63235,C(CNC(c1cncc(OC)n1)=O)(CC(C)C)NC(COCCCC)=O 63236,C1(C)(C(N2CCC(C(=O)NCC(=O)N(C)CC)CC2)=O)CCC2CC2C1 63237,C(CCC)(C(=O)NC(C)(CNC(c1c(C)n[nH]c1C)=O)C1CC1)=CCC 63238,c1(C(=O)NC2(CNC(C(C)(C)OC)=O)CCCCC2C)nnc2ccccn12 63239,c1(CC)c(C(N2CC3CC3C2C(N2CCOC(C)C2)=O)=O)ccn1C 63240,c1(C(N(CCCNC(COCCOCC#C)=O)C)=O)ccncc1Br 63241,N1(C(CN(C(C)C)C)=O)CCN(C2CN(C(C3CC34CCC4)=O)C2)CC1 63242,N1(C(C(C(CC)C)O)=O)CC2CCC(NC(c3ccncc3C(F)(F)F)=O)C2C1 63243,CCN1C(=O)C(n2cnnc2-c2cccnc2)c2ccc([N+](=O)[O-])cc21 63244,N1(C(c2nc(CC)sc2)C(=O)NCCCSC)CCc2nnnn2CC1 63245,C1(C(=O)NC2(c3ncc[nH]3)CC2)CN(C(C2CC(F)(CF)C2)=O)CC1F 63246,C(=O)(C1COc2ccccc21)NC1CC2CC(NC(c3ccc[n+]([O-])c3)=O)C2C1 63247,C(=O)(C(F)C(C)CC(C)(C)C)NCC1CCC(CN(C(C=CCCC)=O)C)CC1 63248,Cc1ccc(C(C)NC(N2CCN(Cc3nc(-c4cccs4)n[nH]3)CC2)=O)cc1 63249,C(CNC(=O)CC1CC(F)(F)C1)(CC(=O)NCCN1CCCC1)OC 63250,c1(C(=O)NC2C(NC(C3(C)CC3(Cl)Cl)=O)CCC2)cnc(N)c(N)c1 63251,CC1CS(=O)CCN1C(=O)C(Cc1cnc[nH]1)NC(C1CCC(C)(O)CC1)=O 63252,N1(C(C(C)C)=O)CCCC1(C)C(=O)NCc1nncs1 63253,C1(C(=O)NCC(C)(C2CC2)NC(c2c(C)nc[nH]2)=O)CCC2(CCOCC2)C1 63254,C1(NC(C2(CF)CC2)=O)CC2CC(NC(C3CC(O)C3)=O)CC12 63255,Cc1nccc(C(=O)N(C)CCN(C(c2cc(CF)on2)=O)CC2CC2)c1C 63256,c1(CC(=O)NCC(CNC(CSCC)=O)O)c[nH]c2cc(OC)ccc12 63257,Cc1nc2ccccc2cc1C(=O)NCC(CO)NC(=O)C(O)CC[S+](C)C 63258,CC1(C(=O)O)CC(F)(F)CN1C(c1nc(C2CC2)n(-c2ccccc2)n1)=O 63259,C1(CC(N2CC(OCC(=O)NC)C2)=O)CCCCN1C(=O)C(F)SC 63260,C(=O)(C1CCCn2cc(C(C)(C)C)nc21)N(CCN(C)C(C1CC(Cl)(Cl)C1)=O)C 63261,Cc1cc(C2(c3noc(-c4sc(C)cc4Br)n3)CCC2)n(C)n1 63262,C1(OC)CC(C(N2CC3CCCC(C2)N3C(c2ccoc2)=O)=O)C12CCOCC2 63263,CC1CCC(C(N2CC(S(C)(=N)=O)C2)=O)CN1C(c1cc(C(N)=O)[nH]n1)=O 63264,c1(CN(C(=O)C(=O)NCc2ccc(I)s2)CC)ccc2nc(O)oc2c1 63265,C1(C(=O)NC2C=C(C)CCC2)C(C)OCCN1C(=O)Cc1cccnc1C 63266,c1(C(=O)NC(C(C(C)C)NC(CCCC#C)=O)C)ccc2c(c1)CC2 63267,c1(C(=O)NC2C(CNC(C(C)C#N)=O)COC2)cc(Cl)cc2c1CCC2 63268,N1(C(C2CCC(CNC(COC)=O)C2)=O)CC2OC(=O)N(C)C2C1 63269,C1(NC(CC=C=C)=O)CCN(C(=O)CN2CCCC2C)C12CC2 63270,C1(NC(C(CC)F)=O)CC(F)CN(C(c2ccccc2-c2nc[nH]n2)=O)C1 63271,CC(C)CC(O)C(=O)NC(C(=O)NCc1ncn(C(C)C)n1)C1CCCC1 63272,c1(CC)n[nH]c(CC)c1CC(=O)NC1CN(C(=O)COC2CCC2)CC1C(F)F 63273,C1(C(C)NC(c2cnn(CC3CCCC3)c2)=O)CN(c2cnc(F)cn2)CCO1 63274,N1(C(c2c(C)nc(COCC)s2)=O)CCC(NC(C2CC3(CCC3)C2)=O)C(F)C1 63275,C1(C(=O)NC(C)CNC(C2(CF)CC2)=O)CCC2(CCC2)CC1 63276,c1cccc(OCC)c1.C(CN=C(NCC1CC1)NC1CC1)c1scc(C(=O)OC)n1 63277,N1(C(CC(C)(C)OC)=O)Cc2nccn2CC(NC(C2(F)CCCOC2)=O)C1 63278,O=C1CC(C(=O)N2CCCC2CN(C(=O)CC2COCCO2)C2CC2)=NN1 63279,c1(C(=O)NCC2CCC(C(=O)NC3(CC)CCOC3)C2)ccnc(C)n1 63280,N1(C(=O)CC2CC3CCC2C3)CC2CCC1CN2C(c1cccc(C2CC2)n1)=O 63281,CC1(C)C(C(=O)N(CCCNC(C2CCOC2)=O)CCO)C1C#N 63282,Cn1c(-n2cc(C3CCCN3CC(F)(F)C(C)(C)O)nn2)nc2ccccc12 63283,c1(CC(=O)NC2(COC)CN(C(c3sc(N(C)C)nc3C)=O)C2)ccc(Cl)nc1 63284,C(=O)(CCCCC(F)F)N(CC(C)(C)NC(C1C(C2CC2)C1(F)F)=O)C 63285,C1(NC(C(c2ccc(C)s2)C)=O)C=CCN(C(=O)Cc2cnnn2C)C1 63286,C(C)(CNC(=O)C=C(Cl)Cl)(C(C)C)NC(CCc1cc(C)[nH]n1)=O 63287,CC1(C)C(NC(=O)CC2CCC=CCC2)CCN1C(=O)C(c1cc(F)ccc1F)=O 63288,c1(CCC(=O)N(C2CCCN(C(=O)CCC#N)C2)CC)cncnc1O 63289,c1(C(N2CCC(C(N(C)CC3(O)CCC3)=O)C2)=O)ncc(F)cc1N 63290,c1(C(N2CCC(COC)(NC(C3CC(=O)N(C)C3)=O)C2)=O)c(Cl)ccnc1C 63291,C1(C(=O)NCCC2OCCN(C(c3c(OC)cncn3)=O)C2)CC2(CCOC2)C1 63292,c1(CCC)nc(COC)ncc1C(=O)NCCN(C(=O)C(C1CCC(=O)N1)C)C 63293,N1(C(c2c(C(=O)OCC)c[nH]c2)=O)CCC(C)C(CNC(=O)CSC(F)F)C1 63294,c1(OC)cc(C(=O)NCC2CCN2C(C2CC(CF)C2)=O)cc([N+](=O)[O-])c1Cl 63295,Cc1c(N)ccc(C(=O)NCC(C)CNC(=O)CN2OC(C)(C)CC2=O)c1C 63296,c1(C(C)C)nc(NCC2CC2c2ccccc2C)cc(=NC(C)C2CCC2)[nH]1 63297,N1(C(C=CC(CC)=CC)=O)CC(c2ccccc2)CC1C 63298,c1(C(N2CCC(CCNC(c3c(CCC)occ3)=O)C2)=O)cccc(F)c1Br 63299,CCC(C)(C(=O)N1CCC(OC)CC1)OCC1CCN(C(=O)C(C)(F)F)C1 63300,C1(NC(C=CCOC)=O)CC2CC1N(C(=O)C(F)C(C)(C)O)C2 63301,N(C1CN(C(C2CC(F)C2)=O)Cc2ccccc21)C(C1C(CCC)C1)=O 63302,C#CC(C)(C)C(=O)NC(CNC(=O)CCCn1cc(C)cn1)C(C)C 63303,c1(OC)cc2cc(C(=O)Oc3ncnc(-c4ccccc4)n3)[nH]c2cc1OC 63304,C(=O)(CC1=NN(C)C(=O)C1)NCc1occ(C(N2CC(C)C(CO)CC2)=O)n1 63305,N1(C(C(C)CO)=O)CCCCC(C2CN(C(C3CC4(CC4)C3)=O)C2)C1 63306,C(CC(F)(F)C(=O)NC1CCC(=O)NC1)n1cc(CC(C)O)nn1 63307,N1(C(CC2C(C)(C)OCC2)=O)CC2(CCCC2)C1C(N1CCOC(CCO)C1)=O 63308,n1(CC)ncnc1C(=O)NC(CC(N)=O)c1ccccc1 63309,c1(C(=O)O)ncccc1CN1CCC(F)(C(=O)Nc2ccc(OC(F)F)nc2)C1 63310,c1(OCC(=O)NCC(C)NC(=O)CN(C2CCCC2O)C)ccc(Br)nc1 63311,CCCC(C)(CC)C(=O)N1CC(C(=O)O)C(CCO)C1 63312,C1(NC(C=CCC)=O)CC2CCC1N2C(c1c(C)nn(C)c1-n1cc(C)cn1)=O 63313,C(CC(C(=O)N1CCCCC1CNC(c1cc(C(C)=O)cs1)=O)N(C)C)SC 63314,N1(C(c2cc(OC)ncc2Cl)=O)CC2CN(C(c3cnc(O)o3)=O)CC2C1 63315,N1(C(c2c(C)scn2)=O)CCC2(C1)CN(C(c1nc(C3CC3)cs1)=O)CC(C)O2 63316,C#Cc1ccc(C(=O)N(C(C)C(N2CCCC(F)CC2)=O)CCC)cc1C 63317,CN(C)NC(=O)CCC(=O)N1CCC2(NC(c3c[nH]c(=N)o3)=O)CC2C1 63318,CN1CCC(C(=O)NCC2CC2NC(c2cc(C#N)c[nH]2)=O)CC1 63319,N1(C(c2cc(C3CC3)on2)=O)CC2CCN(C(C3CC3C3CCOCC3)=O)C2C1 63320,N1(C(CC(=O)NCC)=O)CCC(NC(=O)COCC)CC1 63321,Cc1cccc2cc(C(=O)NCCCN(C)C(C3(O)CCOCC3)=O)nnc12 63322,CCCCCC(CC)C(=O)N1CC(NC(=O)CC(F)(F)F)C(C)(C)C1 63323,C1(C(=O)NCC2CC(OC)C2(C)C)(CC)CCCN(C(=O)C(F)C(C)C)C1 63324,C1(C(N(CCCCNC(C2CC(OC)C2)=O)C)=O)CC2(C1)CC21CC1 63325,C1(NC(C(C)SC(C)C)=O)C2CC1N(C(C1CCCCC1c1nc[nH]n1)=O)C2 63326,c1(C(N2CC(CC(=O)NC3CC34CCCC4)C3(C2)CC3)=O)cc2ncccc2[nH]1 63327,CN(CCN1CCOCC1)N1CCCC(C(N2CCCC2)=O)C1 63328,CN1CC(C)(C)CC1C(N1CCC1CC(N1CCCC(CCF)C1)=O)=O 63329,c1(CNC(C2CC3CCC2N3C(C2C3CCCC23)=O)=O)cc(F)ccc1O 63330,CCCCCS(=O)(=O)CC(=O)N(CCC(C(C)(C)C)NC(=O)C(C)CSC)C 63331,c1(C(N2C(CC)CN(C(C3CN(C)C(=O)N3)=O)CC2)=O)ccc2c(c1)CCCO2 63332,c1(NC(CNC2CCCC(OC)C2)=O)c(C)nc(C)nc1O 63333,N1(C(=O)CCCn2cncn2)CC2CC(C1)N(C(=O)Cc1n[nH]cc1C1CC1)C2 63334,c1(CC(=O)NCC2CCC(NC(CN3C(C)CCC3)=O)C2)nc2ccccc2o1 63335,Cn1c(C(N2CC(NC(c3ccc(C(C)(F)F)cn3)=O)C2)=O)cnc1S 63336,N1(C(C(CN(C)C)(C)C)=O)C2CCCC1CC(NC(c1cc(N)c(F)cn1)=O)C2 63337,C(=O)(C(=O)NOCCOC(c1cccc(Br)c1)Oc1ccc(F)cc1)OC(C)(C)C 63338,C(=O)(CCCCCCn1cc(-c2ccc(CN)cc2)nn1)NC(CC)CC(C)O 63339,CC(C)CC(CC(=O)NC(c1ccccc1)CNC(=O)CC(C)N(C)C)CC(N)=O 63340,c1(C(N(CCCNC(C23CCC2C3)=O)C)=O)cc2c(s1)CCCCC2 63341,C(C)(C(=O)N(C)OC)Nc1cccc(C(c2n(CCOC)nnn2)NCCO)c1 63342,N1(C(c2ccc(NC(C)=O)s2)=O)CCC2CN(C(C3OCCC3C)=O)CC2C1 63343,O(NC(=O)CC1CCCC1)CCCN(C(=O)COCCC(C)C)CC 63344,N1(CCn2nc(C)c(C)c2C)CCCC2(CN(C(c3ccn(C)c3)=O)CCO2)C1 63345,c1(C(=O)NC2(C(=O)NCC(C)C(C)(F)F)CC2(C)C)n[nH]c2c1CCC2 63346,N1(C(C2CCC3N(C(c4c(C)ccnn4)=O)C2CC3)=O)CCc2ccncc2C1 63347,c1(C(=O)OCC)nn(C)c(C)c1COC(C1NC(=O)CC1C)=O 63348,C1(C(=O)NC(CCOC)(C)C)CC(C)CCN1C(C1CCC(F)CC1)=O 63349,N1(C(c2c(C(C)=O)cn(C)n2)=O)CC(CNC(=O)C(O)C(F)F)OC2(CCC2)C1 63350,C1(NC(C(C)Cc2ccccn2)=O)COCCN(C(=O)Cc2cnnn2C)C1 63351,C1(NC(C2CC(OC)C2)=O)(CO)CCN(C(c2cn(C(C)C)nc2Br)=O)C1 63352,Cc1[nH]nc(C(F)F)c1C(=O)N(CC(O)CN(C)C(C1CCS1(=O)=O)=O)C 63353,Cc1ccc(F)cc1C(N1CC(CNC(=O)Cc2cn(C)nc2C)CCC1C)=O 63354,N1(C(C(C)O)=O)CCN2CCOCC2(CNC(C2CCS(=O)(=O)CC2)=O)C1 63355,Cn1ncc([N+](=O)[O-])c1C(=O)NC1C2CN(C(=O)COC(C)(C)C)CC12 63356,N1(C(c2c(CNC(C3CC34CCOCC4)=O)n[nH]c2)=O)CC2CCCC(O)C2C1 63357,N1(C(c2cncc(OC)c2)=O)CCCC2(NC(=O)COC3CCC3)CC2C1 63358,C1(NC(c2csc(Br)c2Br)=O)CCCC(O)C1 63359,N1(C(CN(CC)CC)=O)CCC2(CCC(NC(=O)C(C(C)C)NC(C)=O)O2)CC1 63360,C12(C(=O)NC3CCN(C(=O)CCC=CBr)CC3)CCCC1CCC2 63361,CCCCCCC(C)(F)C(=O)N1CCN(CCn2cc(C3(O)COC3)nn2)CC1 63362,N1(C(=O)CC2CC23CC3)CC(C2CCCN(C(C3(F)CC4(CCC4)C3)=O)C2)C1 63363,C1(CNC(CCCSC)=O)CN(C(c2cc3cc[nH]c3cn2)=O)CC(C)(C)O1 63364,c1(C(N2C3CC(NC(C4CC(OCC)C4)=O)(C3)C2)=O)c(F)ccc(F)c1Cl 63365,Cc1ccc2c(c1)CC(C(=O)NCC(O)CNC(C1(C(F)F)CCC1)=O)O2 63366,C1(OCCOC)CC2CN(C(=O)C(c3ccco3)NC(=O)Cc3ccns3)CC12 63367,c1(OC)ccc(O)c(C(N2CCOC(CNC(=O)C(O)CC(N)=O)C2)=O)c1 63368,C(CN=c1cc(C)nc(-c2ccccn2)[nH]1)C1CN(C(C2C(C)(CC)C2)=O)C1 63369,c1(CC(N2CC(NC(Cn3c(C)ncc3)=O)C(C)(C)C2)=O)c[nH]c2ncccc12 63370,C1(C(N(C2CCCC(O)C2)C)=O)(NC(c2ccncc2N)=O)CCOCC1 63371,c1(CNCCC(C(C)(C)C)OC)cc(C(=O)OC)cc(C(C)(C)C)c1 63372,N(C1CCOc2c(Cl)cc(Cl)cc21)C(N1CCCN(c2c(C)cccc2)CC1)=O 63373,N1(C(C(CC)NC(=O)CCC(=O)NC)=O)CCC(C(=O)NC)C(C)(C)C1 63374,C1(C)(NC(C=C(C)CNC(=O)Cn2cnnn2)=O)CC2(CCC2)C1 63375,C(C(CC)(CC)C(=O)NC(c1noc(C)n1)CC)NC(C(=O)NCC)=O 63376,c1(C(=O)NCC2C(C)CN(C(c3ncc(F)cn3)=O)CC2)ccc(S(N)(=O)=O)[nH]1 63377,Cc1oc(Cl)nc1C(=O)NC1(C(=O)N(C)Cc2cnn(C)c2)CCSC1 63378,c1(C(=O)NCCN(C)C(C2CCOC2=O)=O)ccc2c(c1)CNC2=O 63379,N1(C(Cn2ccc(C)n2)=O)CCC(C(=O)NCCCC2(C)CC2)C1C(C)C 63380,N1(C(COC2(C)CCOCC2)=O)CC2COCC2(C(=O)NCC2CCCS2)C1 63381,N1(C(c2c(CC)[nH]nc2Cl)=O)CCCC2C1CCCN2C(=O)CSc1nncs1 63382,N1(C(c2ccc(NC)c(F)c2)=O)CC2CCC1CN2C(=O)CC(C)COC 63383,c1(CC(=O)NCCC2CCC(NC(CSC)=O)C2)ccccc1[N+](=O)[O-] 63384,c1(C(=O)NC(C2CN(C(C3(C#N)CCCO3)=O)C2)C)cc2nccnc2cc1F 63385,c1(CCC(N2C(CNC(C3CC3C(F)(F)F)=O)CC2)=O)ccc2c(c1)OCO2 63386,C1(c2ccccc2)(NC(C(F)=CC)=O)CCN(C(c2ocnc2CCC)=O)C1 63387,c1(CC(N2CC(CNC(C3COCCO3)=O)C(O)C2)=O)nc2ncccn2n1 63388,c1(C(=O)NC(C)CCNC(C23CC(CO)(C2)C3)=O)cccc2[nH]ccc12 63389,C(=O)(C1=C(Cl)CCOC1)NCC1CN(C(C2C(C)(C)C2CO)=O)C(CO)C1 63390,c1(NCC2N(CC)CCC2)nc(=NC2CC2CF)[nH]c2c(C)nn(C)c12 63391,c1(C(N(C(CNC(C2CCC(C)(C)O2)=O)C2CC2)C)=O)cc2ccc(Cl)cc2o1 63392,c1(C(=O)NC2(CC)CN(C(=O)C(c3ccc(Cl)cc3)O)C2)ccc(NC)cc1Cl 63393,C(C(CC(C)C)C(=O)NC(c1nnc(O)n1C)C)NC(CC(=O)NCC#C)=O 63394,N1(C(c2n(CCC)ncc2)=O)CC2CC1C2NC(c1ncccc1OC)=O 63395,C1(CNC(C=CCCC)=O)CC(OC)CN1C(c1cnc(O)o1)=O 63396,c1(OC)cnc(F)c(C(=O)NCC(C)NC(C2CC2c2nc[nH]n2)=O)c1 63397,N1(Cc2ccc(C(=O)OCC)[nH]2)CC(C(N2CCCC(C)CC2)=O)CC(F)(F)C1 63398,Cc1cnc(NCc2cc(C)no2)c(S(=O)(=O)NCC2(CO)CC(C)C2)c1 63399,CCCC(C)(O)C(=O)N1CC(CCNC(=O)C(c2ccccc2F)C)(OC)C1 63400,C#Cc1cc(C(=O)NC2CCC(NC(=O)C(C)O)CC2)cc(N)c1 63401,c1(C(=O)NC2CN(C(C3(C)N(C)CCC3)=O)CC2(C)C)c(Cl)nc2ccccn12 63402,C1(CC)CCN(C(=O)Cc2ccccc2C)C1C(=O)NC1CC(=O)N(O)C1 63403,c1(CN2C(C(=O)NC3(C#N)CCOCC3)CCC2)c[nH]c2nc(Cl)ccc12 63404,C(C(C(=O)NC1CN(C(c2cc(OC)ns2)=O)C1)C(C)(C)C)OCC=C 63405,Cc1cccc2[nH]c(=NCCN(C(=O)CC3CC3C)C)oc12 63406,N1(C(CN(C)C(N)=O)=O)CCC(NC(=O)C(C)(C)C(=O)NC)C(CO)CC1 63407,Cc1ccc(C(=O)NCC(N2CC=CC2C(=O)NCC2(Br)CCC2)=O)cc1 63408,c1(CNC(CC2N(C(CC=C)=O)CCOC2)=O)cc(F)c(Cl)cc1Cl 63409,c1(C(=O)NCC2N(C)CCN(C(c3ccoc3Cl)=O)C2)c2c(nn1C)CCC2 63410,C1(C(=O)NC(c2nc(CC)on2)C)CCCCCCN1C(=O)CC(C)O 63411,C(=O)(C(F)CCC(C)C)N1CC(N(C(c2[nH]cc(C)c2)=O)C)C(O)C1 63412,c1(C(=O)NC)ccc(N2CC(CNC(=O)NC(C)CN(C)C)C2)nc1 63413,N1(C(c2c(C)n[nH]c2)=O)CCCC(C(C)NC(=O)Cc2csc(S)n2)C1 63414,C(=O)(C1CCOc2ccccc21)NC(C)CN(C)C(c1c(Br)cnn1C)=O 63415,N1(C(C(CC)SC)=O)CCOCC(CNC(=O)CC2(N(C)C)CC2)C1 63416,CCC(C)C(O)CNC(c1ccc(OC2CC2)cc1)c1ccn(C)n1 63417,N1(C(CC(C(F)F)NC(C2CCCC23CCC3)=O)=O)CCCC2CNC(=O)C12 63418,C1(O)(CCNC(C2(CC#C)CCCC2)=O)CCN(C(c2ccnn2C(C)C)=O)C1 63419,C1(C#N)(C(N(CCC(C)NC(C(C)N2CCC2)=O)C)=O)CCSCC1 63420,N1(C(CCC2(C)N(C(c3c(C)c[nH]n3)=O)CCC2)=O)CCOCC2(CC2)C1 63421,Cc1cn2nc(C(=O)N(C3CN(C(c4cccc(CO)n4)=O)C3)C)cc2c(=O)[nH]1 63422,C1(C(=O)NCC(CCOC)NC(c2cnccn2)=O)CCN(C(C)C)CC1 63423,Cn1cnc(NC2CCC(NC(=O)CCc3ccncc3)CC2)cc1=O 63424,C1(CNC(C(CCC)OC)=O)CCN(Cc2nnc(Cn3cccn3)o2)CC1C 63425,N1(C(C)=O)CCCCC1C(N1CCC(CNC(=O)CCCc2csc(C)n2)C1)=O 63426,C(C1CCOC1)=CC(=O)NCCC(O)CNC(=O)C(F)(F)C1CCCC1 63427,CC(C)(CCCC(=O)NCC1CC(O)C1(C)C)NC(=O)CS(C)(=O)=O 63428,C(=O)(C(CC)CC=CC)N1CCCC(CCC(=O)NCC(=C)CC)C1 63429,C(CN=C(NCc1ccnc(F)c1)N(C)CC1CC=CCC1)OCCC 63430,C1(C(=O)NCCN(C(=O)CCCNC(=O)C2CC2)CC)NC(=O)CC1C(F)(F)F 63431,c1(C(c2nnnn2CC(F)F)NCc2cn(C)nc2Cl)cc(S(C)(=O)=O)cs1 63432,CC1OC2(C(=O)NCC3CCN(C(=O)CN4CCN(C)CC4)CC3)CCC1C2 63433,CCC1=C(C(=O)N2CC3CC2CCC3NC(c2ccnc(F)c2)=O)CCCO1 63434,C1(C2CCC2)(C(=O)NC(CC)CNC(=O)CC(C)(C)SC)CC1(F)F 63435,C1(C(=O)NCCNC(CC)=O)C2Cc3c(Br)cccc3C12 63436,c1(SCC(=O)NCC(CC)NC(c2cccs2)=O)ccccc1N=NN(C)C 63437,n1(CC)c(CNC(=O)CC(C)(C)NC(=O)C(C)=C2CC2)nnc1O 63438,C1(CNC(=O)CC2CC3C=CC2C3)CN(C(=O)C2CC2)CCC12CCOCC2 63439,C12(C(=O)NC3CN(C(Cn4c(C)ccn4)=O)CC3C(F)F)CC1COC2(C)C 63440,c1(C(N2C(C3CCN(C(=O)C(F)C4CCOC4)C3)CCC2)=O)cccc(F)c1O 63441,c1(C(=O)NC2CC(NC(c3ccccc3-n3ccnc3)=O)C2)cc(F)ccc1Cl 63442,c1(CCC(=O)N(CCC(C)NC(=O)C#CC2CCC2)CC)cc(F)c(F)c(F)c1 63443,Cc1cccc(C(N2CC3(NC(c4ccsn4)=O)CCC2C3)=O)c1Cl 63444,c1(CC(=O)NCC(C)NC(C2C(C(=O)OC)CC2)=O)coc2c(C)c(Cl)ccc12 63445,c1(C(=O)NCC(C)NC(C2N(CCC)C(=O)CC2)=O)cccc2cccc(O)c12 63446,N1(C(CN(C(COC)=O)C)=O)CC(NC(=O)C(C)(C)C2CCC2)C(O)C1 63447,N1(C(C(c2cncnc2)C)=O)CC(F)(F)CC1CNC(=O)Cc1cnco1 63448,N(C(=NCc1ccc(C(N)=O)cc1)NCC1CCCO1)C1C(C)(C)CC1 63449,C(CC(C)(C)C)(C(=O)N1CC(O)C(C2CC2)C1)NC(C(CC=C)OC)=O 63450,c1(OCC)nc(N2CC3CC3(NC(=O)C(O)C(C)CC)C2)ncc1OC 63451,C(=O)(C1=CCC(F)(F)CC1)N1CCC(CCNC(CCC(C)OC)=O)C(F)(F)C1 63452,N1(C(CC(CC)C)=O)C(CC(=O)NC2CCCCCC2C)C2CCCC12 63453,C1(CC)CCN(C(=O)CCc2cn(C)cn2)C1C(=O)NCC#CCOC 63454,C(=O)(CCC(C)CN(C)C)NCC1(F)CN(C(C(C)NC(C)=O)=O)C1 63455,C1(C(CNC(CCC)=O)Cc2ccccc2)CCN(C(c2ccoc2Cl)=O)CC1 63456,c1(C)cccc(C)c1.c1(C(=O)NC2C(CC)CCO2)cccc(C(F)(F)F)c1 63457,C=CC(CC)C(=O)N1CCC(=CNC(=O)CC)CC1 63458,N1(C(c2n(CC)ncn2)=O)CC2(CC(NC(=O)CC3(N(C)C)CC3)CO2)C1 63459,CC1=C(C)CC(C(=O)NCC(C(=O)N(CCCCO)C2CC2)C(C)C)CC1 63460,N1(C(CCC2CCCN(C)C2)=O)CCN(C)CC1CNC(=O)CCNC(=O)CO 63461,Cc1cc(CNC(C2COC(CNC(c3sccc3C)=O)C2)=O)cc(C)c1 63462,c1(C2(C(=O)NCC(C3N(C(C(COCC)C)=O)CCC3)(C)C)CC2)ccccc1F 63463,Cc1cccc(C(CNC(=O)CSc2nc[nH]n2)NC(=O)C(O)C(F)F)c1 63464,N1(C(C(CCC2CC2)NC(c2c(OC)ccs2)=O)=O)CC2COC(=O)C2C1 63465,C1(CCNC(C2(C)CCCC2)=O)CC(F)(F)CN1C(c1cc(CO)ccc1Cl)=O 63466,C1(NC(c2occ(C(=O)OC)c2)=O)CCC(C)N(C(C2CC3(C2)CC(F)C3)=O)C1 63467,c1(-c2cn(CC(N3CC(C)C3C(N3CCCC3)=O)=O)nn2)ccc2ccn(C)c2c1 63468,c1(CC)ccc(C)c(C(N2CCC(NC(=O)C(c3cccnc3)O)C2)=O)c1 63469,CC(CCCC(=O)NC(C)(C)CC1CCOC1)NC(c1cc(Cl)no1)=O 63470,c1(C(=O)NC(C2CN(C(=O)CC3(CO)CCC3)C2)C)ccc[n+]([O-])c1 63471,C1(C(=O)NCC(=C)Cl)CC2CC1CC2NC(=O)CC1CNC(=O)O1 63472,Cc1nc(C(=O)NC2CN(C(C3CCC3c3nc[nH]n3)=O)C2)cn(C)c1=O 63473,c1(C(=O)OCC)cc(C(=O)OC)c(NC(c2cncc(Br)c2)C)c(Cl)c1 63474,c1(CC(=O)NCC(CNC(C2CC(C(F)F)C2)=O)OC)ccc2c(c1)OCCO2 63475,c1(CNC(c2ccc(CC)o2)=O)c(C)nn2c1CN(C(C1(C)CC1F)=O)CC2 63476,N1(C(C23CCC(C(C)=O)(CC2)CC3)=O)CCc2ncc(Br)cc2C1 63477,c1(C(=O)NC(CNC(C(C(C)C)N(CC)CC)=O)CC(C)C)ccc(N)c(Cl)n1 63478,C=CCC(F)(F)C(=O)NCC1CC(C)N(C(=O)C#CC2CC2)C1 63479,O=S(=O)(CCO)CCNC1CCCCCCC1 63480,c1(C(N(C)CC2N(C(CCOCC)=O)CC(F)C2)=O)cc2n(n1)CCC2 63481,c1(C(=O)NC2CN(C(c3c(C)ocn3)=O)CC3C2C3)ccnc2ncccc12 63482,c1(OCC(N2C(CNC(=O)CCCF)CCC(C)C2)=O)cccc(S(C)(=O)=O)c1 63483,c1(C(N2CCN(C)C(CNC(=O)CCOC3CC3)C2)=O)cccn2nnnc12 63484,C1(NC(COCCCCC)=O)CCCCC1NC(=O)C(c1cccc(C)c1)C 63485,N1(CC(C)NC(c2cc(C(C)=O)on2)=O)CCN(C(=O)Cn2nnc(C)n2)CC1 63486,C12(C(=O)NCC3N(C(C4CCC(F)(F)C4)=O)CCN(C)C3)C3CC(CC13)C2(F)F 63487,C(=O)(C(C)CC)N(CC(=O)N(CC(CSC)O)C)CC1CC1 63488,c1(N2C(CNC(C3(C)CCC(=O)N3)=O)CC(F)(F)C2)ccc(S(C)(=O)=O)cn1 63489,C1(C(N(C)CCOCCNC(=O)Cc2cncc(O)c2)=O)CC2(CCC2O)C1 63490,CN=c1cc(C(=O)N(C(C)C(N2CCCC(C)(N(C)C)C2)=O)C)cc[nH]1 63491,c1(CC(=O)N(CC(C)NC(C2CCCS2)=O)C)cccc2c1CCC2 63492,CC(CCNC(c1cccc(N2CCCCC2)n1)=O)CCNC(C1CCCO1)=O 63493,c1(NCCCCSC)ncccc1S(=O)(=O)NC1COC2(CCC2)C1 63494,C(C(C)(C)C(=O)NCC[Si](C)(C)C)NC(C(N1CCOCC1)C)=O 63495,c1(C(N2CC(NC(CCC#C)=O)CC(F)(F)C2)=O)c(F)cc(OC)c(F)c1F 63496,C1(C(=O)NC2CN(C(c3c(CCC)nsc3N)=O)C2)CC2(CCCC2)CO1 63497,C1(NC(c2ccc(-c3ccccc3)nc2)=O)CN(C(C2CCO2)=O)CC(F)(F)C1 63498,C12(CNC(CN(CCOC)C)=O)CC(NC(=O)CCc3cccnc3)(C1)C2 63499,N#Cc1ccnc(C(N2CCC(NC(C3CCCC(F)(F)C3)=O)CC2)=O)c1F 63500,C(=O)(CCCCC(F)(F)F)NCCCCn1cc(CN(C(C)=O)C)nn1 63501,C=CC(C)(O)C(=O)N1CCC(CF)(NC(=O)C(C)(C)COC)C1 63502,C12(NC(Cc3n(C)ncc3)=O)CCN(C(c3cc4sccc4s3)=O)CC1C2 63503,N1(C(CCn2cnc(=N)[nH]2)=O)CCN(C(C23CCC(C2)C3)=O)CC1c1cn[nH]c1 63504,Cc1cc(C)c2[nH]c(C(=O)NC3CCC3NC(=O)CNS(=O)(=O)C3CC3)cc2c1 63505,c1(OC)cc(NC(=O)C(N2CC(C)C2c2cccs2)=O)cc(OC)c1OC 63506,Cc1cc(O)ncc1C(=O)NC1CC(O)CN(C(c2ccnc(C(C)C)n2)=O)C1 63507,N1(C(C(CNC(C2CC3(CC(C)C3)C2)=O)(C)C)=O)CCN(C)C(C)C1C 63508,Cc1csc(C(=O)NCCNC(c2c(C3CCCCC3)noc2C(C)C)=O)c1C 63509,C1(C(=O)NCC2CCC(C(=O)N(C34CC(C3)C4)C3CC3)C2)C2CCCC12 63510,C1(CC(=O)NCC2(CC)CC2)C2CCCC2N1C(C1(C)CCN(C)C1)=O 63511,c1(N2CC3C(NC(C(CC)C4CCOCC4)=O)C3C2)cc(S(C)(=O)=O)ncn1 63512,C1(NC(C(F)=C(C)C)=O)CCCCC1CNC(c1cnns1)=O 63513,Cc1cc(C(=O)N(C(C)CCNC(=O)C(F)(F)c2cnn(C)c2)C)c(C)cn1 63514,O=C(CCCCCNC(C1CCSC1)=O)NOCCc1ccccc1 63515,C1(C)(NC(CCC)=O)CCC(NC(c2ccc(C(F)(F)F)c(Cl)c2)=O)CC1 63516,CC(C)(F)CCC(=O)N1CC(F)CC1CNC(c1c(N)cccc1Cl)=O 63517,NS(=O)(=O)c1ccc(C(=O)NC2CCN(c3ccc(Cl)cc3)C2)nc1 63518,N1(C(Cc2cc(C)sc2)=O)CC(CNC(=O)CCOC2CCC2)C2(CC2)C1 63519,N1(C(C(C)SCCCC)=O)CCC(NC(c2cc(C(C)=O)cs2)=O)C(C)C1 63520,C1(CN(C(C(CC=C)N(C)C)=O)C)CCCN(C(C2CCCCCC2)=O)CC1 63521,c1(C(C(=O)NCC(O)CC2CCC2)NC(c2ccccn2)=O)ccccc1 63522,C(=O)(C(C(C)C)C(C)C)N1CCOCC(C(=O)NCC(COCC)O)C1 63523,C(=O)(C1CCc2nccn21)N1CCCC(O)(CNC(C2N(C)CC3(CC3)C2)=O)C1 63524,CCC(CC(C)C)C(=O)N(C(C)C(=O)NCC(CC)OC)C1CC1 63525,c1(C(=O)NCC2N(C(C(CCC)(C)C)=O)CCCC2)cc2n(n1)CC(C)NC2=O 63526,c1(C(N2CCCC(NC(c3cc(C)on3)=O)(CO)C2)=O)cc(S(N)(=O)=O)ccn1 63527,c1(C(=O)OC)ccc(C)nc1N1CCCCC(NC(=O)CCCCN(C)C)C1 63528,CC(CC(=O)NCCN(C(=O)Cc1ccccc1)C1CC1)n1ccnc1 63529,C12(C(=O)NC(C)C(F)F)CC(n3cc(CN4CCCC4)nn3)C1C2 63530,Cc1nc(C#N)ccc1C(N1CCCC(CCNC(C23CC(CO2)C3)=O)C1)=O 63531,Cc1c(Cn2cc(CSCCNC(c3ncccc3O)=O)nn2)cnn1C 63532,C1(C(=O)NC2CC(CCNC(c3c(CC)ocn3)=O)C2)CCCC(C)(C)O1 63533,CCC(F)(F)CC(=O)NCc1ncoc1CCNC(=O)C(C)(O)CCC 63534,C1(C)(c2onc(-c3c(C)cccc3)n2)CC2CCC1C2 63535,c1(OC)cc2nc(O)n(CN3CCCCC(CC(N)=O)C3)c(=O)c2cc1OC 63536,Cc1ccc(C(N2CCCC(C)(NC(=O)CC(C)c3ccncc3)C2)=O)c(N)c1 63537,C1(NC(C2(CC)CCCN2C(=O)C(F)C2CCCC2)=O)CCC2CC1CO2 63538,Cc1cc(C(=O)NCC(O)CNC(=O)CC(C)F)nn1-c1ccc(Br)cc1 63539,C1(C)(NC(CCCn2cc(CNC(CCC(=O)OC)=O)nn2)=O)CCCCC1C 63540,c1(C(N2C3CC(CN(C(C4COCCOC4)=O)C3)C2)=O)c(F)ccc2c1OCC2 63541,C(CC)(CC(=O)N1CC(C)(C(N)=O)C1)NC(c1n(CC#C)ccc1)=O 63542,C1(NC(c2c(CC)cno2)=O)CC2CC1CN(C(c1ccsc1C)=O)C2 63543,CC(CC(=O)NC1CCC1NC(=O)CC(=O)N(C)C)P(C)(C)=O 63544,Cc1ccc(C(N2CC3C(C2)N3c2ncncc2C#N)=O)c(F)c1 63545,C1(CNC(C(C2CCCO2)NC(C2CC=CC2)=O)=O)CC(C2CC2)=NO1 63546,c1(CC(N2C(CNC(C(CC#C)C)=O)CC3(CC3)C2)=O)cccc2c1CCC2 63547,C1(CC(=O)NCc2ccc(CCCC)cc2)COC2(CCC2)CN1 63548,CCCCCC(O)C(C)C(=O)N1CCCC(CCNC(C2CCN2CC)=O)CC1 63549,C(C1CCC(C)CC1)=C(C(=O)NCC1(C(C)=O)CN(c2ccc(C#N)nc2)C1)C 63550,CC1(C(=O)NC(C)(CNC(=O)Cn2ccc(C3CC3)n2)C2CCC2)CCCCO1 63551,C1(CC(=O)NCC(C)CNC(=O)C(F)(F)c2csc(=N)[nH]2)CC(=O)NC1=O 63552,C1(C(=O)NCC2(F)CC(NC(CCNC(C)=O)=O)C2)CCCC(O)C1 63553,CC1CN(C(c2ccc(Cl)o2)=O)CC1n1cc(C2(CCO)CC2)nn1 63554,C1(C)(C(=O)NC(CNC(C(CCCC)O)=O)CCOC)CCCCCCC1 63555,c1(CN2CC(C(=O)Nc3ncc(F)cc3Br)OCC2)ccc2ncnn2c1 63556,C(=O)(C(F)C(F)(F)F)NCCC1CC(NC(c2cc(C)n(C(C)C3CC3)n2)=O)C1 63557,CC1CC(C(=O)NCCn2cc(CNC(c3nnn(C)c3CO)=O)nn2)CCS1 63558,C12(CNC(c3c(N)cc(F)cc3)=O)CCC(CNC(C3CCCO3)=O)(CC1)CO2 63559,C1(NC(CCc2cn(C)nn2)=O)CN(C(C2(O)CCOC2)=O)CC(C)(C)C1 63560,N1(C(CSCC(=O)OC)=O)CCN(C(=O)CCc2cncn2C)CC1C1CCC1 63561,C1(NC(C2CC(C)C2)=O)CC(C)CN(C(=O)NCCC(=O)OC(C)(C)C)C1 63562,N1(C(C=CC(CC)=CC)=O)CCC(C)(C)C(CNC(C2CCCC3(CC3)C2)=O)C1 63563,N1(C(CCN(CC)CC)=O)CC(NC(c2cnn(C)c2C(C)(F)F)=O)CC1C 63564,CN1CCc2cc(C(=O)NC3COCC3NC(=O)C(O)CC(C)(C)C)ccc2C1 63565,C#CCCC(C(=O)NCCCC(O)CO)NC(=O)CCC=CCC=C 63566,C(CN=C(NCCc1ccc(Cl)cc1)NC1CC12CC2)c1ccc(C(C)C)cc1 63567,N1(C(COCCCCC)=O)CC(C)(CNC(c2cc(SC)c(C)o2)=O)CC1(C)C 63568,c1(C(=O)NCC=CCNC(CCC(C)C#N)=O)cc2n(n1)CCCN2 63569,C(=O)(CC1=CCN(C)CC1)NC1(CNC(C(CCC#C)O)=O)CC1 63570,C(N=c1[nH]c(Cl)nc2cccc(C#N)c12)c1cc(N(C)C)ncc1 63571,Cc1ccc(CNCCc2ccc(O)c(O)c2)cc1C.N1(O)CCOC(CC=O)C1 63572,c1(CC)nc(NN(C)C(=O)OC)cc(=NCC(c2cccs2)OC)[nH]1 63573,N1(C(CC(=C)C)=O)CCC(C2CCCN(C(=O)CC3CCCCCN3)C2)C1 63574,Cc1cc(=NCC2(C)CCC(C)(C)CC2)[nH]c(=NCCCC(C)O)[nH]1 63575,N1(C(=O)CN2CCN(CCF)CC2)CCN(C(C2(F)CC=CC2)=O)CC1C1CC1 63576,C1(C)(CC)CCC(C(N2CC(N(C)C(c3csnc3Cl)=O)C2)=O)O1 63577,C12(NC(C(CC(C)C)C)=O)CCCN(C(=O)COC3(C)CCCC3)CC1C2 63578,N1(C(C(COC)O)=O)CC(C2(NC(C3CCN(C(=O)CSC)CC3)=O)CC2)C1 63579,O=C1NC(=O)N2CCN(c3ncnc4c3ncn4CC3CCCN(C4CC4)C3)CC12 63580,N1(C(CN2CC(CC)C2)=O)CCN(C(=O)CC2CC2C2CC2)CC1 63581,C12(C(=O)OCC)CC(CC(N3CCCC3CN(C(=O)C(F)CC)C)=O)(C1)C2 63582,N1(C(C2(OC)CCC2)=O)CC(NC(=O)Cc2cc(Br)cs2)CC(F)(F)C1 63583,C1(O)(C(=O)NCC2CCCN(C(C(C)C3CCCO3)=O)CC2)CCC(C)(C)CC1 63584,C1(C2(O)CN(C(C3CCc4nn[nH]c4C3)=O)C2)(CNC(CCNC(N)=O)=O)CC1 63585,c1(-c2cn(C(C(=O)NC(COCC)C)C)nn2)[nH]nc(C(=O)OC)c1Br 63586,C#CCCCCCC(=O)N1CC(OC)C(NC(C2(C(C)C)CNC(=O)C2)=O)C1 63587,N1(C(COC(C)C)=O)CCCC(C)(C)C1C(=O)NC(CC1CCCC1)CO 63588,N1(C(C2(CNC(C(COCC)C)=O)CC=CC2)=O)CCCSCC1C 63589,c1(C(=O)OC)cnn2c1CC(NC(N1CCC(C)(C)CC1)=O)CC2 63590,C1(N(CCC)C(C2CC2CF)=O)CCN(C(=O)C(F)(F)C2(OC)CCC2)C1 63591,C12(C(=O)NCC3(O)CCN(C(=O)Cc4cnc[nH]4)C3)CC3CC(CC1C3)C2 63592,c1(C(=O)O)nnc(CNC(=O)C(O)CC2CCOCC2)s1 63593,C1(CC=C)(C(=O)O)CCCCN1C(=O)C(F)CC 63594,CC(CC(F)(F)F)C(=O)N(C1CN(C(C2CC(n3cnnc3)C2)=O)CCC1O)C 63595,Cc1csc(CNC(c2nnnn2C(c2ccccc2)C)c2cnc[nH]2)c1 63596,c1(NC(C(=O)NCC(C)C)=O)ccc(OC2CCOC2)c(S(=O)(=O)N(C)C)c1 63597,CCC(CC#N)N=c1ccc(Br)c(S(=O)(=O)NCCS(=O)(=O)NC(C)C)[nH]1 63598,C(C(=O)NCC(C)CN(C)C(c1c(NC(C)=O)c[nH]c1C)=O)(C(C)C)OC 63599,N1(C(Cc2ccc(OC)c(Cl)c2)=O)CCN(C(=O)C(C#N)C2CC2)CC(C)(F)C1 63600,N1(C(=O)C=Cc2ccco2)CCC2CCN(c3c(Cl)cncc3[N+](=O)[O-])CC2C1 63601,c1(C(N(C(CNC(C2(CCC=C)CCCC2)=O)C)C)=O)nccc(Cl)c1O 63602,c1(N(CCN(CC)CC)CC)cc(Cl)c(F)cc1S(N)(=O)=O 63603,CCCCC(CC)C(=O)NCC1CCCN(C(=O)CC2CCOC(C)(C)C2)C1 63604,N1(CC(=O)NC2CCOCC2NC(C2CC(=C3CCC3)C2)=O)C(=O)CCC1=O 63605,Cc1cc(C(F)(F)F)nc(C(=O)NC(c2nnc(C)s2)C)n1 63606,c1(C(=O)NCC2OCCN(C(c3c(C)nn(C)c3)=O)C2)ccc(F)cc1F 63607,C(=O)(CC(C)(C)C(=O)NC1CCC(NC(=O)CC2CCC(C)(C)O2)C1)OC 63608,C1(NC(CCC(=C)Cl)=O)CN(C(=O)COc2cc(Cl)ccc2C)CC12CCC2 63609,CC1CC=CCC1C(N1CCN(C2CN(C(C3(O)COC3)=O)C2)CC1)=O 63610,C1(NC(=O)OC(C)(C)C)CN(C(=O)c2cc([N+](=O)[O-])n[nH]2)NC1=O 63611,N1(C(CCC(C)OC)=O)CCCC2(NC(=O)C(N3C(C)CCC3C)C)CCCC12 63612,c1(C(=O)Nc2ccc(NC(C(CCC)CC)=O)cc2C)cnc2c(c1)NCC(=O)N2 63613,N1(C(CNS(NC)(=O)=O)=O)CCCN(C(C2CC(O)C2)=O)C(C(C)C)C1 63614,C1(C(=O)NCCN(C(=O)CC2COCCN2C=O)C(C)C)CCCCN(C)C1=O 63615,c1(C(C2C(C(=O)OC)C2)N(CCC(C)Sc2ccccc2)C)ncsc1Br 63616,C12(NC(c3ccn(C4CC4)n3)=O)COCCC1CN(C(c1nc(Cl)sc1Cl)=O)C2 63617,C1(C(=O)NC(C)CNC(=O)C(C)(C)n2cc(Cl)cn2)CCC(=O)NC1 63618,C1(C(N(CCCC(=O)NC)C)=O)CCC2(CC2)N1C(C1CCCN1C)=O 63619,Cn1c(C(=O)NCC23CC(CN2C(=O)C=CC(F)(F)F)C3)ccc1C(F)(F)F 63620,c1(OC)c(C(C(=O)NCCCF)N(C2CCOC(C)C2)C)ccnc1F 63621,C=C(CC(C(=O)OCCO)NC(=O)OC(C)(C)C)c1occc1C#N 63622,c1(C(N2C(C(=O)Nc3cc(C)c(Cl)cc3Cl)CC3CC32)=O)ccc2c(c1)C(=O)CC2 63623,N1(Cc2scc(C(=O)NC(Cn3c(C(C)C)nnn3)=O)n2)CCC(N(C)C)CC1 63624,N1(C(Cc2nc(C)sc2C)=O)CCC2(CC1)CC2CNC(C1(C#N)CCOC1)=O 63625,N1(C(C=C=C(C)C)=O)CCN(C(=O)CC(C)n2cccc2)C(CC(F)F)C1 63626,C(=O)(C(CC(C)C)ONC(c1cnsc1C)=O)NCc1nc(C(C)OCC)sc1 63627,CC1CCN(C(C2(CO)CC(F)(F)C2)=O)CCN1C(=O)Cc1cnns1 63628,Cc1nccn1CCCC(=O)NC1CCC(CC(N2CCC(O)C2)=O)C1 63629,C(=O)(CC(C)(O)C(F)(F)F)N1CCCC(CNC(C2(SC)CC2)=O)CC1 63630,c1(C(=O)NC(C(=O)N(CCC)C)C)cccc(OCCc2cccnc2Br)c1 63631,C1(NC(C=Cc2n(C)ncc2)=O)CN(C(=O)Cc2n[nH]c(=N)s2)CC1S(C)(=O)=O 63632,c1(C(N2CC3C(NC(CCCC#C)=O)C3C2)=O)cc(C)nc(N(C)C)n1 63633,CC1(C)CN(C(C2CN(C(N)=O)C(C)(C)C2)=O)CCC1NC(c1csc(Cl)n1)=O 63634,C(=O)(CCC(C)(C)C#N)NC1C(C(C)C)N(C(=O)C(O)Cn2cncn2)CC1 63635,c1(C(N2CC3C(C(=O)NC(c4n(C)cnn4)CO)C3C2)=O)cnn2cccc2c1 63636,C1(NC(CCOCC)CO)CC2CCC1O2 63637,C(=O)(C(F)CC(C)(C)N)NCc1nnc(C(=O)OC)s1 63638,N1(C(C(C)(C)OC)=O)CCN(C(c2ccc(C#N)c(F)c2)=O)CC(C)C1 63639,C(=O)(C(C)(O)C(C)(C)C)N(C1CCN(C(c2ccc(CCC)cc2)=O)CC1)CC 63640,C12(NC(c3ccc(Cl)cc3F)=O)COCCC1CN(C(c1ccns1)=O)C2 63641,c1(C(=O)NC(C)CCN(C)C(C2CC2C)=O)cc(-c2ccncc2)nn1C 63642,c1ccc(CN(C2CCNC2)CC2CCNCC2)cc1 63643,Cc1cncc(CCNC(=O)C(C2CCN(C(c3cnncc3O)=O)CC2)C)n1 63644,N1(CC)CCN(C(F)(F)F)C(=O)C1.c1(O)cnc(CNC(=O)C(=O)NC)nc1 63645,Cc1c(Cl)ccc(C(=O)NCCNC(=O)C2=CCCC2C)c1N 63646,c1(OC)ccc(-c2c[nH]nc2C)cc1S(=O)(=O)NCC1CCS(=O)(=O)C1 63647,C12(OC)CCC(CN(C3CCOC3)CCO)(CC1)C2 63648,c1(NC)ccc(C(N2CCCC(CCCCNC(=O)C3CC3)C2)=O)nc1 63649,c1(C(=O)NC2C(CNC(C3CCC(C)CC3)=O)CCC2)cccc2cncn12 63650,N1(C(Cc2c(C)scc2)=O)CCC(NC(=O)C=Cc2ccoc2)C(C)C1 63651,c1(OC)cc(C)c(C(=O)NCCN(C)C(c2nnn(C)c2C(F)F)=O)cc1Cl 63652,C(=O)(C(F)C(C)(F)F)NC(C(=O)NC(c1nc(CC)on1)C)(C)CSC 63653,c1(C(=O)NCC2C3CN(C(C4CC(C(=O)OC)C4)=O)CC32)c(Cl)cc(Cl)nc1N 63654,C(=O)(C(C)(C)CCCO)N(C)CC1CCCN1C(c1ccc(C(F)F)cc1)=O 63655,N1(CC(=O)NCC2CC2CC(N2CCC3CC23)=O)C(=O)CCC1=O 63656,c1(C(N(CCC(C(C)C)NC(C(CC(=O)OC)C)=O)C)=O)cc2cn[nH]c2cn1 63657,O=C(C1CCCc2scnc21)NC1CCN(C(=O)CCOCC(F)(F)F)CC1F 63658,C1(CC(=O)NCC2C(CNC(c3cc(C)oc3)=O)C2(F)F)CCCNC1=O 63659,C1(N(C(=O)COCP(C)(C)=O)C)CN(C(C2CCN(CC(F)(F)F)C2)=O)CC12CC2 63660,C12(C(=O)NC3C(NC(COC(C)=O)=O)CS(=O)(=O)C3)C3C4C1C1C2C3C41C(N)=O 63661,C1(NC(C2N(CC)CCOC2)=O)CCN(C(=O)Cc2cccs2)CC1C 63662,N1(C(C(CC)(C)O)=O)CCCCC(NC(c2ccsc2Br)=O)CC1 63663,Cc1c(C(N2CCCN(C(C3CCC(=O)N3)=O)C(C)C2)=O)[nH]c2cc(F)ccc12 63664,C(=O)(CCC(=O)N(CCCCNC(C1CCCC(F)C1)=O)CC)NCC 63665,C1(CNC(COCCCC#C)=O)CC(C)CN(C(c2occc2CC)=O)C1 63666,C1(NC(c2n(C)ccn2)=O)CN(C(C2CC2C(C)(F)F)=O)C(C)(C)C1 63667,c1(C(N(CCCNC(c2c(C)nc(CC)o2)=O)C2CC2)=O)ccc2c(n1)NCC2 63668,N1(C(c2n(CC)ccc2)=O)CCC(N(C(=O)Cc2c(C)noc2Cl)C)C2(CC2)C1 63669,C1(NC(c2n(C=C)nnc2)=O)(CC)CCN(C(=O)C(C2CCC(=O)N2C)C)CC1 63670,C1(NC(C2(C(N)=O)CCC2)=O)CCC(NC(c2cnc(Br)s2)=O)C1 63671,c1(CC)c(C(=O)NCCNC(=O)CCCc2nc(C)no2)cccc1Br 63672,c1(C(N2C(CNC(c3c(C)coc3)=O)CC2)=O)c(C)nn(CC(F)(F)F)c1Cl 63673,Cc1nsc(CNC(=O)C=CC(C)NC(C2(CO)CCOC2)=O)n1 63674,N1(C(C=CCNC(c2c(CC)n(C)nn2)=O)=O)CC(N(C)OC)C1 63675,C1(NC(c2nc(C)c(C)s2)=O)CCCN(C(=O)CN2C(C)CCC2C)CC1 63676,S(=O)(=O)(c1ccc(=NCCC2CCSC2)[nH]c1)NC1CC(C)(C)SCC1 63677,Cc1cc(C(=O)NCC2COC(CNC(=O)CCc3n[nH]c(C)n3)C2)nc(O)n1 63678,CC1N(Cc2cnn(C)c2C(=O)O)CCC1(C)C 63679,C=C(Cl)CCC(=O)NC(C1CC=CCC1)C(=O)NCC(C)(C)C1CCCC1 63680,N1(C(C(N2CCCCC2=O)C)=O)CCC(F)(CNC(c2cn(CCO)nn2)=O)C1 63681,c1(C(=O)OCC(=O)N(C(CC)CC)C2CC2)cc(Br)c(C)s1 63682,N1(C(C2(OC)CCC2)=O)CC(CNC(c2cc(OC)nc(OC)c2)=O)C(C)(C)C1 63683,c1(NC(C)=O)cccc(F)c1NC(=O)CNc1ccc(F)c(F)c1 63684,CC1(C)CCC(CNC(=O)C(CCF)NC(c2ccc(C(F)F)o2)=O)O1 63685,CC(C)C(O)C(=O)NC(C)(CNC(=O)C(C)(C)C1CCOCC1)C(C)C 63686,Cc1conc1N(C(=O)OC(C)(C)C)CC1CC1c1ccccc1 63687,CC(=O)CCCCC(=O)N1CC=CC1(C)C(=O)NCC(C)CC(F)(F)F 63688,C1(C)(C(N2CCC(O)(C(C)CNC(c3ccc(CO)o3)=O)C2)=O)CCC2CC2C1 63689,c1(CC(=O)NCC2(C)CCN(C(C3(CO)COC3)=O)C2)ccc(S(N)(=O)=O)cc1 63690,C1(OC)CC(C(=O)NC2COCCC2O)C12CCC2.N12CCC(CC1)C2=O 63691,C12(C(=O)NCC(C)(C)CNC(C3(C)CCOC3)=O)CCC(CC1)C2(C)C 63692,CC1CCC(O)CN1C(CC1CC1(Cl)Cl)C(=O)NCc1cccc(Cl)c1 63693,N1(C(C(CCSC)O)=O)CC(C(=O)NC2CCCC2N=[N+]=[N-])CC(C)(C)C1 63694,c1(C(N2C(C(=O)Nc3cc(OC)n[nH]3)CC3CC32)=O)cnc(Cl)cc1OC 63695,c1(C(N(C2CCCC(NC(CCC=CC(C)C)=O)C2)C)=O)cc(Cl)cc(F)c1F 63696,c1(CNC(C(=O)NC(c2nc(C3CCCCC3)no2)C)=O)cccc(F)c1 63697,N1(C(c2cnc(CC(C)(C)C)s2)=O)CCC2(CC1)CN(C(=O)C(O)P(C)(C)=O)C2 63698,C(C(C)(C)CC(=O)N1CCC(C)C(C)C1)NC(COCCCOC)=O 63699,N1(c2ccc(-c3ccc(CC)cc3)c(C)n2)CCC(CO)C(C)(C)C1 63700,CCCCCCCCC(C)CC(=O)N1CC(NC(=O)CCNC(=O)OC)C(C)C1 63701,CN1CCN(C(c2nc3c(s2)CCCC3)C(=O)NCCC2CC2)CCC1=O 63702,C1(=CC(=O)NCCC2CCC(NC(C(C=C)C)=O)C2)CCC(C)CC1 63703,C(CCCCCC(=O)N1CCCC1c1ccccc1CO)n1cc(C(=O)O)nn1 63704,N1(CC)CCCC(C(=O)NCC2CN(C(=O)COCP(C)(C)=O)CC2O)C1 63705,Cc1noc(C(C)C)c1C(=O)NCC(C)(C)CCNC(C1(N(C)C)CCC1)=O 63706,c1(C(=O)NC(c2ccccc2C(F)(F)F)C)ccc(I)c(OC(F)(F)F)c1 63707,c1(CC)ccc(Cl)c(C(N2CCC(CNC(C3(OC)CCCC3)=O)C(C)C2)=O)c1 63708,C1(C(=O)NCC(C(C)C)NC(CC(CC)CC)=O)CC2CCCCCC12 63709,N1(C(c2c(C)snc2)=O)C(C(=O)NCC2CCOC2(C)C)CC2CCCC12 63710,C1(CNC(c2occ(C)c2C)=O)CN(C(=O)COC2CCCOC2)CCC1(F)F 63711,Cc1cc(C(=O)NC(C)CNC(=O)CC2CCC(=O)CC2)n(C)n1 63712,N1(C(COC(C)(C)C)=O)CC2CC(C(=O)Nc3ncn4c3CCCC4)CC2C1 63713,C1(CCNC(N2C(C(=O)OC)CCC2c2ccccc2)=O)CCC(OC)CC1 63714,Cc1nc(=N)[nH]c(=NCCCCNC(=O)C=Cc2scnc2C)[nH]1 63715,c1(COCC)nc(N2CCC(NC(=O)Cn3nc(C)oc3=O)C(F)C2)cc(Cl)n1 63716,c1(N(C)C)cc(C(=O)NCC2CN(C(=O)Cn3ccc([N+](=O)[O-])n3)C2)ccc1F 63717,N1(C(C2C(C)(C)C2)=O)CC(C2CCCN(C(c3ncn4cc(Cl)ccc34)=O)C2)C1 63718,c1(CNC(C2CCN(C(c3scc(C(=O)OC)n3)=O)C2)C)cnc2[nH]cncc1-2 63719,C(=O)(C1=NOC2(CCOC2)C1)N1CCC(CN(C(=O)CNS(C)(=O)=O)C)C1 63720,CCCCCC(O)CNC(C1CCN1C(c1coc(C(C)C)n1)=O)=O 63721,c1(C(=O)NC2(COC)CN(C(C3COCC3(C)C)=O)C2)cnc(C(=O)O)nc1 63722,c1(C(N2C(CNC(C=C(CC)CC)=O)C(C)(C)CC2)=O)cccc2nccn12 63723,C1(CNC(c2cncs2)=O)CN(C(=O)CN2C(=O)CCC2=O)CCC12CCOC2 63724,CCC(CCNC(=O)CN(C(=O)C(n1ccnc1C)C)C1CC1)C(=O)OC 63725,c1(CCOC)nc(CC(CC(F)F)c2ccccc2)n(-c2ccc(Cl)cn2)n1 63726,C(=O)(C(F)(F)C(C)O)NCCC1(OC)CN(C(=O)C(C2CCOCC2)C)C1 63727,c1(OCC(N2CCC(N(C(=O)COCCCF)CC)CC2)=O)ccc(F)c(C)c1 63728,c1(OC)cccc2c1OC(C(=O)NC1C3CCC1N(C(C1(CF)CCC1)=O)C3)C2 63729,CCCC(CNC(C1CCCSC1)=O)NC(c1cnc(SC)[nH]1)=O 63730,C(=O)(C(C)C(C)(C)C)N1CCC(C(C(=O)NCc2n(CC)ccn2)(C)C)C1 63731,Cc1ncc(C(=O)NC2CC(C)(NC(=O)CCC(C)CN(C)C)C2)c(C(C)C)n1 63732,c12ccc(cc1)SC(C)(C)C(c1n(CCC)nnn1)NC2CCO.C1(CC)CC1 63733,C1(NC(C(CC2CC2)NC(=O)CCc2ccc[nH]2)=O)C2C3CCC(C3)C12 63734,S(=O)(=O)(c1cccc(N2CC3CC2CS3=O)n1)NCC(c1ncc(C)s1)C 63735,C1(NC(C2C(C)C2)=O)CC(F)(F)CC1NC(c1ccsc1Br)=O 63736,CC(C)C(CN(C)C)C(=O)N1CCCCC1C(C)(C)CNC(=O)CSCC(N)=O 63737,c1(NC(C2CN(C(C)(C)C)C(=O)C2)=O)scc(Cl)c1C#N 63738,C1(C(=O)NCC2(OC)CN(C(C(CC=C)(C)C)=O)C2)CC2COCC(C1)C2 63739,c1(OC)ccc(C(=O)NCC2(CNC(C3CCC(C(C)C)CC3)=O)CCC2)cc1 63740,C(=O)(C1=CCC(NC(=O)C(CO)NC(N)=O)C1)NCCCCC1C(C)C1 63741,N1(C(CCC#C)=O)CCC2(CC1)C(NC(=O)CN1CCC(C)C1)CS2(=O)=O 63742,C1(CSC)(CN2CCC(c3nnc(C)n3Cc3ccccc3)CC2)CC(F)(F)C1 63743,C1(COC)(NC(=O)CC2CCC(C)(C)C2)CCN(C(c2cscn2)=O)C1 63744,C1(C)(NC(C(C)c2cccs2)=O)CCCN(C(=O)C=CC(=O)N(C)C)C1 63745,C(c1cccc(F)c1)=CCC(=O)NCC(C(C)C)NC(C1CC(NC)C1)=O 63746,C1(NC(c2ncn(C(C)C)n2)=O)COCCN(C(=O)CN2CCCCCC2)C1 63747,Cc1cc(=O)c2cc(C(=O)NC3CN(C(=O)C4=CCCOC4)CC3C)ccc2[nH]1 63748,CC1(C#CC(=O)N2CC3CN(C(c4cncc(Cl)c4)=O)CCC23)CCCO1 63749,C1(C)(C(N(CC(C)(C)NC(C(Cn2ccc(C)n2)C)=O)C)=O)CCC(C)(C)CC1 63750,C1(CC)CCN(C(=O)CCCC2CCCO2)C1CNC(C1C2CCCCC12)=O 63751,C1(C(N(CCNC(c2ccc[nH]2)=O)CC2CC2)=O)CS(=O)(=O)CC1C(F)(F)F 63752,C1(CNC(CC2N(C)CCC2)=O)(CO)CCN(C(C23CCCC(CO2)C3)=O)CC1 63753,O=C(N=c1cc(Cl)nc(C(F)(F)F)[nH]1)C1COCCN1Cc1ccsc1Br 63754,Cc1cc(N)c(C(=O)NCC2CC2CNC(=O)C(C)CC2CCCC2)c(F)c1 63755,C1(CC(=O)NCC(N2C(C(=O)NC)CCC2)=O)CC(=O)NC1=O 63756,N1(C(C(c2ccccc2)C)=O)CC2(CCCCN2C(c2cnc(S)n2C)=O)C1 63757,C(CC(C)C(=O)NCC(C)CNC(c1ccc(C2CCCCC2)o1)=O)=CC 63758,c1(C(N2CCC(CCNC(CC(=C)Br)=O)C2)=O)nc2ncccn2n1 63759,C1(CNC(c2[nH]cc(C)c2)=O)CCN(C(C2CC(C)CCC2C(C)C)=O)C12CC2 63760,C1(NC(C2CCN(C3CC3)C2=O)=O)CC2CCC1N2C(=O)CNc1ncccn1 63761,C(=O)(CC(C)C(=O)N1CC=C(CNC(=O)C(C)NS(C)(=O)=O)CC1)OC 63762,CC1(C)CN(C(=O)CCN(C(=O)C(C2CCCCC2)O)C2CC2)CCC1O 63763,C(C(CC)(CC)C(N)=O)NC(CN(CC#C)C(c1cccnc1S)=O)=O 63764,C1(NC(C2CCCCC2)=O)CC2CCC1N(C(c1ccn(C3CC3)n1)=O)C2 63765,C(=O)(C(F)C(C)C(F)(F)F)NCC1(C)CCN(C(CCSCCCC)=O)C1 63766,N#Cc1ccc(F)cc1NC(C1CC(F)CN1C(c1c[nH]c2cnccc12)=O)=O 63767,c1(CC)cc(NC(=O)COCCCn2cc(NC(C)=O)nn2)ccc1O 63768,CON=C1CN(C(=O)Cn2ccccc2=O)C1 63769,C1(CC#C)CCCCN1C(=O)C(C)CNC(c1cc(Cl)no1)=O 63770,C1(NC(c2scnc2C(F)F)=O)CN(C(=O)CC2OCCCO2)Cc2nccn2C1 63771,C(=O)(C(C)CNC(=O)C(CNC(c1nc[nH]n1)=O)N(C)C)OC 63772,CC1C(C(=O)NCC2CC(F)(F)C2)CCN1C(=O)CCC1CCCC1 63773,C1(NC(C2CC(N3CCN(C)CC3)C2)=O)CCN(C(c2ccns2)=O)CC1F 63774,c1(OC)nc(NC(N(CC)Cc2ccc3[nH]ccc3c2)=O)c(Cl)cc1C 63775,CC1(C)CCc2c1n[nH]c2C(=O)NCC1CN(C(=O)CCn2ccnc2)CCO1 63776,C1(OC(C(C)C)=O)CCN(C(=O)C(=O)N2CC(Oc3ccc(C(N)=O)o3)C2)CC1 63777,C1(N(C(CS(=O)(=O)NC)=O)C)CCCCN(C(c2nnc(S)n2C)=O)C1 63778,CCC(CCCC(=O)NCCCC1CCOC1)NC(c1ncncc1C)=O 63779,C(CCCCC(=O)N1CC(NC(C2CC3COCC3C2)=O)C2(CC2)C1)OC 63780,c1(C(=O)OC)cc(C)sc1NC(C1CN(C(=O)C(C)Cc2c(C)noc2C)C1)=O 63781,C1(NC(C2CC23CCC3)=O)CCN(C(c2cc3c(s2)CCCC3)=O)C12CCC2 63782,N1(C(c2cnn(CC)c2Cl)=O)CCN(C(=O)C#CC2CC2)C(c2ccncc2)C1 63783,N1(C(CCN(C(C2(CCCC)CCCC2)=O)CC)=O)CC2(CNC(=O)N2C)C1 63784,CC(CC(=O)NC(CNC(=O)C(N)=O)CO)S(=O)(=O)c1ccc(F)cc1 63785,CCCCC(CNC(c1cncc(F)c1)=O)NC(=O)Cn1ccnn1 63786,CC(Cc1ccc(C#N)cc1)N=c1[nH]c(N2CCC3CCC(C3)C2)nc(=N)[nH]1 63787,C12(C(=O)NCC=CCNC(c3c(O)ccc(OC)c3)=O)CCCN1CC(OC)C2 63788,c1(CC(=O)N(CCN(C(=O)C(C)c2ccsn2)CC)CC)ccc2c(c1)CC2 63789,N#CC1CN(C(C2(C3CCCN3C(c3cnn(C4CC4)c3)=O)CC2)=O)CC12CCC2 63790,C(=O)(CC(C)CCC=C(C)C)NC1CC(N(C(c2c(O)ccc(OC)c2)=O)C)C1 63791,c1(C(=O)NCC(C)N(C)C(c2cc(C(F)(F)F)n[nH]2)=O)ccc(F)cc1C(F)F 63792,C1(C(=O)NCC2N(CC)CC2)CC(O)CCN1C(=O)C(C)CC#N 63793,CC1(C)CN(C2CCN(C(=O)Nc3cccc(F)c3I)CC2)C(=O)O1 63794,CCCS(=O)(=O)CC(=O)NCCC(O)CNC(c1cc(OC)cs1)=O 63795,c1(NC(C(=O)NCC2CCN(CCC)C2)=O)ccc(OC)c(C#N)c1 63796,N1(C(C(CCC)NC(N)=O)=O)CCC(NC(c2ccc(C)cc2F)=O)C12CC2 63797,N1(C(C2CC(C)(C)SC(C)(C)C2)=O)CCCCC(C2CCOCC2)C1 63798,c1(C(=O)NC2C(C)CN(C(c3ccncc3F)=O)C2)cc2c(F)ccc(F)c2[nH]1 63799,c1(C(C(=O)NC2CC2)N(C2C(OC)COC2)C2CCCC2)cc(C)c(C)cc1C 63800,CC(C(=O)N(C1(CC(=O)N(C)CC2CC2C)CC1)C)C1CCC1 63801,C(C(C)(O)C(=O)N1CCC(F)(C(=O)NCC2=CCCOC2)C1)OC 63802,c1(CC(N2CCC(C(C)NC(c3c(C)n[nH]c3)=O)C2)=O)ccn2cncc2c1 63803,c1(C(N(C2CCN(C(c3cccc4cc[nH]c34)=O)C2)C)=O)cccc([N+](=O)[O-])c1 63804,c1(NCC(CSC)OC)ncnc(N2CCOC(C)(c3ccccc3)C2)c1C 63805,c1(CC(C(N2CCC(NC(CN3CC(C)C3)=O)CC2)=O)O)c(F)cccc1Cl 63806,c1(C(=O)NCC2CN(C(C(C)O)=O)C(C)(C)C2)cccc2c1OCCCO2 63807,O=C(CCSC1CC1)NC(C1(CNC(C2(CCl)COC2)=O)CC1)=O 63808,c1(C(N2CC(c3nn[nH]n3)(CC=CC)C2)=O)cc(OC)cc(C(=O)OCC)n1 63809,C1(N(CCOCCN(C(CCOCCN(C)C)=O)C)C)CCN(C)CC1 63810,N1(C(c2cncc(C)n2)=O)CC(C)CN(C(=O)Cc2ccc(Cl)c(Cl)c2)CC1C 63811,C(=O)(C(CCC(N)=O)N(C)C)N1C(Cn2cc(-c3ccc(OC)nn3)nn2)CC1 63812,CC(C)(C)CCCC(=O)NCCC1(NC(=O)C(F)OC(F)(F)F)CCC1 63813,c1(CC(=O)NC2CCC(N(C(CC3(CSC)CC3)=O)C)C2)coc2ccccc12 63814,CCCCC(O)C(=O)NCC1(O)CCCN(C(=O)CCCNS(C)(=O)=O)C1 63815,N1(C(CC2(OC)CC2)=O)CC(NC(=O)Cn2nc(C)c(C)c2C)CC(F)C1 63816,C(=O)(C(=O)N=c1ncn(C(c2ccccc2)C)[nH]1)Nc1n(CC)ccc1 63817,N1(C(C(CC)CC)=O)CC(CNC(c2ccnc(C)c2C)=O)OC2(CCC2)C1 63818,N1C2c3ccccc3OCC2CCCCC(=O)Nc2ccc(OC)cc21.OC 63819,CCC(C(=O)N1CC2CCC(CNC(C34CCCC3CCC4)=O)C2C1)C(F)(F)F 63820,C1(NC(C(C)OCC#C)=O)CC2CCC(C1)N2C(c1cccnc1OCCO)=O 63821,n1(CC)cncc1C(=O)N(CCNC(C1(CN(C)C)CCC1)=O)C(C)C 63822,c1(CNCCN(C)C)csc(=NC(CCO)C2CC2)[nH]1 63823,N1(C(c2ccc(OC)c(I)c2)=O)CC(NC(c2cnsn2)=O)CC(F)(F)C1 63824,CC(CC(=O)NC1(C)CC(NC(c2cc(C(N)=O)cs2)=O)C1)C(F)F 63825,c1(OC)ncc(C(N2CC3CCC3(CCNC(=O)C(C)(C)CO)C2)=O)cc1C 63826,Cc1ccc2c(=NCCC3CC=CC3)[nH]c(=NC(C)c3ccccc3)[nH]c2c1 63827,C1(OC)CN(C(=O)C(C)=C(C)C)CCC1NC(=O)CN1CCCCC1C 63828,c1(CNC(C=CSC)=O)ccccc1CNC(c1coc(O)n1)=O 63829,Cc1cc(C(N2CC(C(N3CC(S(N)(=O)=O)C3)=O)CC(C)C2)=O)nnc1C 63830,c1(CC(=O)N(CCC(C)NC(C(C)(c2ccccc2)OC)=O)C)nnc(S)n1C 63831,N1(C(c2c(OC)oc(C)n2)=O)CC(NC(=O)CC2CCOC2(C)C)C2(CC2)C1 63832,N1(C(c2n(C)cnc2)=O)CCCC(C2CN(C(=O)CCCC3CCCO3)C2)C1 63833,CC(C)(O)C(F)(F)C(=O)NC1CC(C(F)C(=O)NCCCSC(F)F)C1 63834,c1(C(N2CC3C(CNC(C4C(C)OCCC4)=O)C3C2)=O)cccc2c1COCC2 63835,c1(NC)nc(Sc2cc(-c3cccc(CO)n3)ccn2)ncc1Br 63836,N1(C(CCC2N(C(C3N(C4(C)CC4)CC3)=O)CCC2)=O)CCC2(COC(=O)N2)C1 63837,C1(NC(CC2N(C(C)=O)CCC2)=O)CCC(CNC(c2cnnn2C)=O)CC1 63838,C1(CC)(NC(c2ccc(F)c(C(F)(F)F)c2)=O)CCCN(C(=O)C(C)(C)OC)C1 63839,c1(C(=O)NC2CCN(C(c3ccnc(OC)n3)=O)C2)cccn2ccnc12 63840,c1(NC(C2CCN(Cc3ccncc3O)CC2O)=O)cnc(Cl)cc1[N+](=O)[O-] 63841,C(CNC(c1n[nH]c2c1COC2)=O)(CC(F)(F)F)NC(CC(C)N(C)C)=O 63842,c1(C(=O)NCC2N(C(C(C)SC)=O)CC2)ccc(S(=O)(=O)N2CCCCC2)cc1 63843,c1(CC)csc(CNCC(c2ccccc2)C)n1.c1ccccc1 63844,CCC(C(=O)NCC#CC(=O)N(C)Cc1cncn1C)NC(C)=O 63845,C(=O)(CCCCCC#N)N1CC(CNC(C(C)(C)SC)=O)OCCC1 63846,C1(F)(C(=O)NC2CC(C)N(C(C3CN(C)C(=O)N3)=O)CC2)CCC(F)(F)CC1 63847,C(=O)(CC1CCOc2ccccc21)N1CC(C)C(NC(=O)C=CBr)C1 63848,Cc1cccc(CC(N2CCC(C)(CCNC(=O)CC(C)(C)O)C2)=O)c1F 63849,N1(C(C(C)OCC=C)=O)CCCC2CN(C(c3ccc(CC(C)(C)O)s3)=O)CC12 63850,Cc1ccc(C(=O)N(CCNC(c2ccc(F)cc2F)=O)C(C)C)cc1C(F)(F)F 63851,c1(C(N2CCC(c3cn(-c4ncc(Br)cn4)nn3)C2)=O)cccc2oc(O)nc12 63852,c1(CNC(c2c(C)nsc2)=O)ccc(C(=O)NC(c2ccccc2)C(N)=O)cn1 63853,N1(C(c2c(C(C)C)scn2)=O)CC(CNC(C2CCCN(C)C2)=O)C2(CCC2)C1 63854,S(=O)(=O)(CCC(=O)N1CC(N(C(=O)C(c2ccccc2)N(CC)CC)C)C1)NC 63855,c1(CN(CCNC(CSCC)=O)C(C2CC(C)=NO2)=O)cccc(Cl)c1 63856,C1(C(=O)NC2(CC)CC2)OCCC1NC(c1cnn(C(C)C)c1)=O 63857,C1(CC(=O)NCC(CC)(C)NC(c2c(Cl)n[nH]c2C)=O)CCCCC(=O)N1 63858,C1(C(N)=O)CN(C(=O)C(CCF)NC(=O)CC2CC(=O)NC2=O)CC12CC2 63859,C(CC(C)C(=O)NC(CNC(c1cc(-n2cccc2)ccn1)=O)(CC)CC)=CC 63860,CCCCCC(F)C(=O)N1CC(CNC(=O)CCN2CCOC2=O)CC(C)C1 63861,C1(NC(C(C)N(C(=O)CC2(O)CCOCC2)C)=O)CCOC(C2CC2)C1 63862,c1(CNC(C(c2ccc(Cl)c(Cl)c2)N)=O)cc(C(F)(F)F)ccc1Cl 63863,C1(C(N2CC3(CN(Cc4c(C)cc(C#N)cc4)C3)C2)=O)CCC2(CC1)OCCO2 63864,C12(NC(CC3N(CC)C(=O)CC3)=O)CCC(CC1)N(C(c1ccncc1)=O)C2 63865,Cc1nn(C)cc1C(=O)NC1CCCC1C(=O)NCC(O)C1(Cl)CC1 63866,C1(C(=O)NC(C(N2CCCC(CCC#C)C2)=O)CCC)CCC(O)CN1C 63867,C1(OC)CCC(C(N2CCCC(NC(c3cnn(C)c3C)=O)C2)=O)CC1 63868,CC1CCC(O)(C(N2CC3C(C(=O)NC(CC4CC4)CO)C3C2)=O)CC1 63869,C(C)(C(=O)N(C)Cc1cccnc1)(C1CCOCC1)OC 63870,Cc1cccn2c(CC(=O)NC(C)CCNC(=O)C(C3CC3)C3CC3)cnc12 63871,Cc1nc(NC(C)(C)CN(C(=O)CSC(F)F)C)cc(Cl)n1 63872,c1(C(=O)NC(CNC(COCC=C)=O)C(C)C(C)C)cc(Cl)cc(Cl)c1Cl 63873,Cc1cnc(C)c(NC(C2(F)CC=CC2)=O)c1 63874,C1(C(=O)NC(CC)C)CC2CCC1N2C(=O)C=C=C(C)C 63875,N1(C(CCC#C)=O)CC2CCCC(CNC(C3CCC(OC)CC3)=O)C2C1 63876,CCCCCCC(C)C(=O)NCC(C(C)C)NC(c1c(C)cnnc1O)=O 63877,c1(C(N2C(CNC(C(F)=CC)=O)CCC2)=O)ccc(Br)c(SCC)c1 63878,Cc1scc(C(=O)NC2CN(C(c3cc(CO)[nH]n3)=O)CC2CC(C)(C)C)c1C 63879,CC(C)C(C(=O)NC1(C)CC2(CCC2)C1)C(C)NC(c1cc(C#N)ccc1N)=O 63880,N1(C(C(COC(C)C)NC(C)=O)=O)CC(N(C(=O)CCn2cnnn2)C)C(O)C1 63881,C(=O)(C1=Cc2cc(Cl)ccc2OC1)N1C(CNC(C(C)O)=O)C2CCC1C2 63882,c1(OCC)cccc(CC(=O)NC2CC2CNC(=O)Cc2ccnc(OC)c2)c1 63883,N1(C(CSCCC)=O)CC2CCCCC2(CNC(=O)C=C2CCCCC2(C)C)C1 63884,c1(OC)cc(Cl)ccc1CN1CCC(O)C(C(=O)N(C)C)C1 63885,Cc1nccnc1C(N1CCC(C(F)C(=O)N(C)CCN2CCCC2)C1)=O 63886,C1(CC(NOCC#C)=O)CC(NC(C2CCN2CC)=O)C1(C)C 63887,C1(C(C(=O)NCCCOC=C)NC(=O)CCn2cccc2)CC=CCC1 63888,c1(CC(=O)NCC(CNC(COCC=C)=O)(C)C)cc(Cl)cc(Cl)c1 63889,C1(CC(N2CC(SC)C(NC(=O)Cc3cc[nH]n3)C2)=O)CSc2ccccc2O1 63890,N1(C(=O)Nc2c(C)cc(N3CCOCC3)cc2)CCN2CCOCC2C1 63891,Cc1ccsc1CC(=O)NCCC1CC(NC(c2nocc2C(C)C)=O)C1 63892,C1(C(NOC(C)(C)CO)=O)CCC(O)CN1C(=O)CC1CCOC1(C)C 63893,N1(C(c2n(CC)ncc2)=O)CC(C(=O)NCC(C)OCCO)CC12CCC2 63894,C1(C(F)(F)F)(C(=O)NCC(CC=C)NC(C2(n3cccn3)CC2)=O)CC(C)(C)C1 63895,c1(C(N2CCC3(CN(C(c4cc(C)ns4)=O)C3)C2)=O)cn2cccc(F)c2n1 63896,O=C(C1=Cc2ccc(Cl)cc2OC1)NC1CN(C(c2cc(CO)[nH]n2)=O)CC1F 63897,C(=O)(CC1CCOc2ccccc21)NC(C(C)NC(c1nc(C)nn1C)=O)CO 63898,C1(CC(=O)OC)(NC(c2ccc(-n3ccc(O)n3)cc2)=O)CS(=O)(=O)C1 63899,C(c1ccc(F)c(Cl)c1)=CC(N1CC(C)C(NC(=O)CN2CSCC2=O)C1)=O 63900,C(CCCCC(=O)N1C(C(=O)NC(CO)CCOC)CCC12CC2)OC 63901,CC1CC(C(=O)NC(c2cnn(C)c2)C(=O)NCCN2CCCNC2=O)CCS1 63902,CON(CCC(=O)N1CCCC(C)C1CO)C(=O)C(C)(C)C#N 63903,CN1CC(NC(N2CCCCC2c2ocnc2C(=O)O)=O)Cc2ccccc21 63904,CCC(C(=O)NC1(C)CCC(NC(C2(COC)CCC2)=O)CC1)C(C)(C)CC 63905,c1(CC)cc(=NCCC2CCC(NC(=O)CC3CCCCC3O)C2)[nH]cn1 63906,c1(OCC)cc(CNc2ccc(C(=O)NC(C)(C)C)o2)ccc1O 63907,c12ccc(cc1)s2.c1(CNCCN(C(C)C)C(C)C2CC2)nnnn1C 63908,S(=O)(=O)(C1CCNC(C)(C)C1)Nc1cc(C)cc(C(N)=O)c1 63909,N1(C(C=C(CC)CC)=O)CCC2CCCC12C(N1CCCC1CSC)=O 63910,C1(CC)CN(C(c2c(Cl)cccc2Cl)=O)CCN1Cc1cccc(Cl)n1 63911,C(=O)(CCCCCN(C)C(C1CC(C)(F)C1)=O)NCCCOCCCC 63912,c1(CC)ncccc1S(C)(=O)=NC(=O)C1(Cl)CC12CCC2 63913,C1(C)(C(N(CCC)Cc2ncc[nH]2)=O)CC12CCN(c1cccc(CC)n1)CC2 63914,Cc1c(C(N2CCC(F)(CNC(=O)C(C)n3cnnn3)C2)=O)ccc2n[nH]cc12 63915,c1(C(N2CC(NC(CCCOC(C)=O)=O)C(O)C2)=O)ccc(OC(F)F)nc1Cl 63916,CC1CN(C(C2CC23CCSCC3)=O)CCN1C(=O)CCCC1CCCCC1 63917,c1(-n2ccc(C(=O)O)n2)cccc(CO)c1.C12CCN(C1=O)c1ccccc1N2 63918,C1(N(C(=O)COC(F)(F)F)CC#C)CCN(C(C2CC2c2ccn(C)n2)=O)CC1 63919,N1(C(C2C(C(=O)OC)C2)=O)CC(C(=O)Nc2cc(C#N)ccc2O)C2(CCC2)C1 63920,C=CCCC(CC(C)C)C(=O)NCCOCCNC(=O)C(C(C)C)n1cnnn1 63921,C1(C(C)NC(=O)C(C)N(CC(F)(F)F)C)CCN(C(C2(F)CCC2)=O)CC1 63922,C1(NC(=O)CCC2CCC(=O)N2)CCN(C(=O)CC2(O)CCC2)C12CCC2 63923,Cc1n[nH]cc1C(=O)NC1(C(=O)NCC2CC2CO)CCC1 63924,C1(C(C)C)CN(C(c2cc(C3CC3)cnc2Cl)=O)CCN1C(=O)C(C)N1CCC1 63925,C(=O)(C1=CCNCCC1)N1C(CCCC)CCCC1 63926,c1(NC(CC)CSC)cc(=NCC(Cc2ccccc2F)CO)[nH]c(C)n1 63927,CC1CC(C)CN(C(=O)COC(=O)CCc2nc[nH]n2)C1 63928,C1(CNC(CN(C(C)=O)C)=O)CCCC2(CCN(C(=O)CC(C)C(C)C)CC2)O1 63929,n1(CC(=O)NC2C(C)CN(C(=O)CN3CC=CC3)C2)ccc([N+](=O)[O-])n1 63930,Cc1ccc(C(=O)NCCC(C)NC(c2cnn(CC(C)C)c2)=O)cc1F 63931,CN1CCC2(CCN2C(c2ccc(-c3cc[nH]n3)o2)C(=O)NC2CCOC2)C1 63932,N1(S(C)(=O)=O)Cc2ccccc2CC1C(=O)NCc1cc2c(s1)CCSC2 63933,Cc1cnc(C(=O)N(C2CCN(C(c3cc(Cl)ccc3Cl)=O)CC2C)C)c(C)c1 63934,CN1CCC(NC(=O)CC(C)(C)C)C12CCCN(C(C1(O)CCCCCC1)=O)C2 63935,C1(NC(CCNC(N)=O)=O)CCOC12CCN(C(=O)CC1CCC(=O)C1)CC2 63936,c1(N2CC3(C(NC(C4C(C)(Br)C4)=O)CCS3)C2)nc2cc(F)c(F)cc2s1 63937,N1(C(C2CCC(=C)CC2)=O)CC2(CCC2NC(c2cc(C(C)C)cnc2O)=O)C1 63938,c1(OC)ccc(F)cc1C(=O)N(C1CN(C(=O)Cn2ccnn2)CC1(C)C)C 63939,c1(C(N2CC(COC)(CNC(=O)CCCF)C2)=O)cnn2ccncc12 63940,CCC(C)(C)C(=O)NCC1CC(NC(c2nc(C(C)(F)F)cs2)=O)C1 63941,N1(C(C2(N(C)C)CCCC2)=O)CC(CNC(c2csc(=N)[nH]2)=O)C2(CC2)C1 63942,c1(OC)ccc2c(CC(N3CCC(CNC(=O)C(C)CN(C)C)C3)=O)coc2c1 63943,N1(C(C2(CCOCC)CCC2)=O)CC2CC1(C(=O)N(c1cncnc1)CC)C2 63944,c1(NCC2C(NC(c3cnn(C)c3C3CC3)=O)CCC2)ncc(Br)cc1[N+](=O)[O-] 63945,c1(CC(=O)NC2CN(C(C3CCCC4CC34)=O)C2)ccc2c(c1)OCCO2 63946,C1(NCc2scc(C(=O)OC)c2)CCN(C(c2ccc(OC)cc2F)=O)CC1O 63947,C(=O)(CCNC(=O)CCNC(=O)CN(C)C(N)=O)NC(COC(C)=O)C 63948,C=Cc1ccc(C(N2CCC(NC(c3ccccc3CC(C)C)=O)CC2)=O)cc1 63949,c1(CC(C(=O)N(CCCNC(C23CC(OC)C2C3)=O)C)O)ccc(Cl)cc1 63950,N1(C(c2cn(CCNC(=O)CCc3nc[nH]n3)nc2)=O)CC2CCC(O)C(O)C12 63951,C1(C)(CNC(CCOC(C)C)=O)CCCN1C(=O)Cc1cn(C)nn1 63952,c1(C(=O)NCC2N(C(c3c(OC)c[nH]n3)=O)CC2)[nH]c(-c2cccc(C)c2)nc1C 63953,C(c1ccc(F)c(F)c1)=CC(N1C2CN(C(c3cc(OC)ncc3)=O)C(C2)C1)=O 63954,N1(CC(CNC(=O)Cc2cc3c(s2)CCC3)O)CC2CCCC2C1c1nn[nH]n1 63955,N1(C(C(CCSC)OC)=O)CCC2(CC1)CCN(C(C1(CO)CCCC1)=O)CC2 63956,S(=O)(=O)(c1cc(F)ccc1C)N1CC2C(C(N3CC(OC)C(O)C3)=O)C2C1 63957,N1(C(C(C)S(N)(=O)=O)=O)Cc2ccccc2C1CNC(C1CC2(C1)CC(O)C2)=O 63958,N1(C(CC2N(C)CC2)=O)CCCC(c2cc(C(c3cccs3)=O)n[nH]2)C1 63959,C1(N(c2ccc(F)cc2)C(=O)C(F)CC2CN(C(C)=O)C2)C2CCC(C2)C1C 63960,c1(C(CO)CNCC(O)CC2CCOCC2)ccc2c(c1)OCCO2 63961,C12(C)CCCN(C1)C2=O.c1(OCC)cc(COC)on1.N12CC(C1)OC(C)(C)C2=O 63962,c1(NC(c2cnc(C)s2)=O)cnc2n1CCN(C(=O)COc1ccc(O)cc1)C2 63963,c1(NC(C2C(C)C2)=O)cnc(F)cc1C(N1CC2CC2C1C#N)=O 63964,C1(NC(CC(C=C)(C)C)=O)CC2(CCCCN2C(C2(F)CCC2)=O)C1 63965,C1(C(=O)NCCC2(O)CN(C(CCOC)=O)C2)CC2CC(C1)CC(F)(F)C2 63966,C1(C(=O)NC2CC(CNC(C3(c4ccn(C)n4)CC3)=O)C2)CC2(C1)CC2F 63967,N1(C(C(C)CC(N)=O)=O)CCC2(CCCC2CNC(=O)Cc2cccnc2)CC1 63968,CN1CCC(C(N2CCSCC2CO)=O)(NC(C23CC(C#N)(C2)C3)=O)C1 63969,CCC(CC(=O)NCCC1CCOC1(C)C)NC(=O)C(n1cc(C)cn1)C 63970,c1(CCNC(=O)NC2CN(C(C)=O)C2)ccc(-c2ccccc2)[nH]1 63971,N1(C(C2CN(CC)C(=O)C2)=O)CC2(CCC2)CC1CNC(C1C=CC=CC=C1)=O 63972,c1(C(=O)NCCC2(CNC(c3n(CC)ccn3)=O)CC2)cc2n(n1)CC(F)C2 63973,n1(CC(=O)NCCCC2N(C(C3CC(=O)C3)=O)CCC2)cnc([N+](=O)[O-])c1 63974,C(CC(CC)C(=O)N1CCC12CN(C(C1CCCC1c1nncn1C)=O)C2)=CC 63975,c1(C(C(=O)NC)N(C(c2ccccn2)COC(C)=O)C)cnc(COC)[nH]1 63976,CCCCC(C(=O)N(C(C)CC(C)C)C)NC(C1CS(=O)C1)=O 63977,c1(C(N2CCC(N(C(C(CC)O)=O)C)C3(C2)CC3)=O)cc2cccnc2cc1F 63978,N1(C(Cc2c(OC)cc(F)cc2)=O)CCCC12CN(Cc1cc(Cl)cnc1F)C2 63979,c1(C(=O)NCC2N(C(c3c(C)onc3)=O)CCC2)ccc2c(c1)CCC(C)N2 63980,Cc1ncc(C(N2CC3CC(NC(c4nccc(Cl)c4F)=O)C3C2)=O)c(O)n1 63981,c1(C(=O)NCCCN(C(=O)C(O)c2ccco2)C)c[nH]nc1S(N)(=O)=O 63982,N1(C(CC(n2c(CC)ncc2)C)=O)CCC2CN(C(=O)C(O)CCSC)C2C1 63983,c1(C(=O)NCC2OCCN(C(c3cccc(C)c3)=O)C2)cc(C)ccc1O 63984,CC1(C)CN(C(=O)Cc2ccccc2O)C(CNC(=O)CCc2ncc[nH]2)CO1 63985,C1(CNC(c2ccc(SC)s2)=O)CC(NC(c2nncn2CC2CC2)=O)C1(C)C 63986,N1(CN(C2CCN(C(C)C(=O)NC3CCCC3)C2)CCO)CCS(=O)(=O)CC1 63987,c1(C(N2C(CNC(c3nc(C)sc3C)=O)C3CCC2C3)=O)ccc2snnc2c1 63988,C1(C(=O)NCCCC(C)(C)NC(=O)C=Cc2cscn2)CCC2(CCOC2)O1 63989,C12(C(=O)NC(C3CN(c4nc(C5CCCC5)ns4)CCO3)C)CCC(CC1)CC2 63990,C(=O)(CC(C)C(F)F)NCC1(CCNC(COCCC#C)=O)CC1 63991,c1(CC(=O)NC(C(C)(C)NC(C(CC)C#N)=O)C)ccc(Br)c(OC)c1 63992,N1(C(C(C)=C2CC2)=O)CC2CCCC2(CNC(=O)C(c2ccccc2Cl)(C)C)C1 63993,c1(C(C)N(C(=O)CCCC(c2ccccc2)O)CCO)ccccc1Cl 63994,C=CC1(CC(=O)NC(C)CNC(=O)C(O)CSC)CCCCC1 63995,C1(C(=O)NC(C(C)C)(C)CNC(=O)CC(=O)N(C)C)CC2C(C1)C2(F)F 63996,C1(NC(c2cn(C3CC3)nn2)=O)CCCCN(C(C2C3CC4C(C3)C24)=O)C1 63997,C1(NC(CNC(N)=O)=O)C=CCC(C(=O)NCCOc2cccnc2)C1 63998,Cc1cn2cc(C(=O)NCCCNC(C3CCN(c4nc(=N)[nH][nH]4)C3)=O)sc2n1 63999,c1(C(N2CCN(C(C3(O)C(C)(C)C3)=O)CC2)=O)ccnc2[nH]c(O)nc12 64000,c1(-c2nc(CC(C)(C)CO)nn2CCCCO)cc2ccc(Cl)cc2s1 64001,N1(C(CCNC(=O)OC)=O)CCC(CO)(NC(c2ccc(OC)cc2)=O)C1 64002,C(=O)(CC(CC)C(C)C)N1CCCC(NC(=O)Nc2cncc(C#C)c2)(CC)C1 64003,C(=O)(CC(C)CC(C)(C)C)N1CC(C2N(C(c3sc(C)c(O)n3)=O)CCC2)(O)C1 64004,c1(CC)cc(N)ccc1C(=O)NCCN(C(C1CC2CC1C2)=O)C(C)C 64005,N1(C(CS(CC)(=O)=O)=O)CCC(C)N(C(=O)C(N2CCCCC2=O)C)CC1 64006,C1(NC(c2cc(-c3nc(C)sc3)sc2)=O)CCC(NC(c2ccn(C)c2)=O)CC1 64007,C1(NC(COCC=C)=O)CN(C(C2CCCC(O)C2)=O)CC2(CCC2)C1 64008,c1(NC(C(=O)NC(COCC)CO)=O)ccc(C)c(O)c1 64009,C#Cc1cccc(C(=O)NC2(c3cccc(Br)c3Cl)CC2)c1Cl 64010,C(=O)(C#CC1CCOCC1)NC(C1CN(C(C2CCc3nnnn3CC2)=O)C1)C 64011,c1(C(N2CC3(C(NC(c4cn5c(n4)CCC5)=O)CC3)C2)=O)c(F)ccc(F)c1Cl 64012,C1(CC(=O)N(CC)Cc2ccncc2)CCN(C(=O)CCC2(C)N=N2)C1(C)C 64013,C(C(C(=O)NCCCC(=O)OC)N1CCC(OC)CC1)(C1CC1)OCC 64014,c1(NCCOC)nc(OC2(C)CCOCC2)cc(=NCCN2CCCC2=O)[nH]1 64015,c1(C(=O)NCC(=C2CN(C(COCC)=O)C2)F)ccc2[nH]ccc2c1 64016,C#CCC(CC(=O)OC)NC(C1CCC(C(C)C)N1C(=O)C=CCSC)=O 64017,N1(C(C(CSCC)NC(=O)CC2CCCC(=O)N2)=O)CCc2ncn(C)c2C1 64018,C1(CNC(Cc2c(C)nc(S)s2)=O)COCCN(C(C23CCC2C3)=O)C1 64019,C1(CC(=O)NC2C(C(C)(C)C)C2)CCCNC(=O)C1.c12ccnc(n1)CS2 64020,c1(C(=O)NC2C(NC(c3c(C)ncs3)=O)CCC2)ccc(OC(C)C)nn1 64021,C1(CC=C)(C(N2CCN(C)CC2)=O)CCN(C(=O)C(=Cc2cnn(C)c2)C)C1 64022,N1(C(CN2CCN(C)CC2)=O)CC(CC(=O)NC2CCCC2N=[N+]=[N-])CC1(C)C 64023,C1(OCCCNC(CC2(C#N)CC2)=O)CCN(C(C23CCCCC2C3)=O)CC1 64024,c1(C(=O)NCC(C)CN(c2cnc(C#N)cn2)C)ccc(C2CC2)cc1F 64025,N1(C(C(=O)NCCCC)C)CC(C(C)OC)(OCCSCC)C1 64026,N1(C(C=C(CC)C)=O)CCC2CCC12CNC(c1ccnn1C)=O 64027,C1(NC(C(CC)O)=O)CC=C(C(=O)N2CCC3CC23)C1 64028,c1(CC(N2CC(NC(c3cc(C(N)=O)[nH]c3)=O)C(F)C2)=O)cccc(Cl)c1Cl 64029,c1(C(N2CCc3nc[nH]c3C2)=O)cccc2occc12.CCCC1CC(=O)N1 64030,CCC(F)(F)CC(=O)NC1CS(=O)(=O)CC1NC(c1ccc(N)c(N)n1)=O 64031,N1(C(C(CCC)CNC(c2cc(CO)on2)=O)=O)CCOCC(F)(F)C1 64032,C=CC(CC)CC(=O)N1C2CCC1C(NC(=O)CS(C)(=O)=O)C2 64033,C1(CC=C)(C(=O)NC(c2nc(C)no2)CO)CCN(C(=O)CNC(=O)CC)C1 64034,N#CC1CN(C(C2(c3ccc(F)cc3)CC2)=O)CC1NC(c1c(F)cccc1Cl)=O 64035,Cc1ccc(F)cc1C(=O)C(=O)N(C1CCN(C(C2(C#N)CC23CCC3)=O)C1)C 64036,CC1CCN(C(=O)C(=O)NCC(O)CCNC(=O)CSCCC#N)CC1 64037,c1(C(=O)NC(CNC(COCCOC)=O)C2CCC2)cc2c(s1)CC(C)(C)C2 64038,C1(C(=O)NC2C(NC(=O)C=CC3CC3)COC2)CCCOC1c1ncc[nH]1 64039,c1(CNC(N2C(CNC(C=CS(CC)(=O)=O)=O)CCC2)=O)ccn2cc(C)nc2c1 64040,c1(N(C)CC)ccc(CCCCNC(=O)NCc2ccccc2OC)cc1 64041,c1(C(=O)NC2CCCC(NC(c3c(C)ccnc3)=O)C2)c(C)cccc1F 64042,c1(C(N(C)CC2(NC(=O)COCc3nccn3C)CC2)=O)cc2nnn(C)c2s1 64043,N1(C(=O)NCCc2c(OC)ccc(Br)c2)CC2(CO)CCCC2(F)C1 64044,c1(C(N2CC(SC)C(NC(c3cccn3C)=O)C2)=O)n[nH]c2ccc(Cl)cc12 64045,C(=O)(C1=CC2C=CC1C2)N1CC(CCC(=O)N(CCOC)C(C)C2CC2)C(C)C1 64046,c1(COC)nc2n(n1)CC(NC(c1cccc(C(N)=O)n1)=O)CC2 64047,C(=O)(CC(C(C)C)c1ccon1)N1C(C2(NC(c3c(C)c[nH]n3)=O)CC2)CCC1 64048,N1(C(CN2CCC(OC)C2)=O)CC=C(C(=O)NCc2cscc2C)C1 64049,C1(C2(O)CCN(c3nc4cccc(F)c4o3)CC2)(NC(=O)COCC2CC2)CC1 64050,C12(C(=O)NCC3N(C(=O)CC4CC4)CC=C3)CC3CC(C1)CC(O)(C3)C2 64051,c1(CC(=O)NC(C2(O)CCN(C(=O)C3=CSCS3)C2)C)cn2cc(F)ccc2n1 64052,Cc1nc(-c2cccnc2)[nH]c1C(=O)NCC(C1CC1)NC(C1CCCN1C)=O 64053,c1(C(N(CCOC)CCNC(=O)C(C)SC(F)(F)F)=O)ccoc1Cl 64054,C(=O)(C1=CC2C=CC(C1)C2)N1C(C(=O)Nc2cccc(CC)c2)CC1 64055,C(=O)(CC1COc2cc(O)ccc21)N(CC(C)NC(=O)CCC(=O)NN(C)C)C 64056,N1(C(c2n(CC)nnc2)=O)CCC2(CC1)CCN(C(c1ccccc1)=O)CC2 64057,N1(C(CCc2cc(C(=O)OC)[nH]c2)=O)CCC2C(C1)CN2C(C1CC(OC)C1)=O 64058,c1(C(N2CC(CCO)(NC(CNC(C)=O)=O)C2)=O)ccn2cc(C)nc2c1 64059,N#CC1(CC(=O)NC2CCCCN(C(=O)C(F)CC3CCCC3)C2)CCOCC1 64060,c1(CC)ccc(O)c(C(=O)N(CCN(C(=O)C(C)OCCC(C)C)CC)CC)c1 64061,N1(C(c2ccn(CC)n2)=O)CCN2C(=O)C(NC(c3cc(O)ncn3)=O)CC2C1 64062,C1(C(=O)NCC(CC)(C)NC(c2csc(-c3ccccc3)n2)=O)CC2CCC1O2 64063,C=CC(CC)CC(=O)NCCC1CC(OC)CN1C(=O)Cc1cc[nH]c1 64064,N1(C(c2nc(CC)sc2C)=O)CCC(O)(C2(C(=O)O)CCC2)CC1 64065,CCC(C)C(C)CN=c1nc2sccc2c(N2CCC(C)(C)CC2)[nH]1 64066,C1(CN(C(=O)C(CC2CCOCC2)NC(C23CSCC2C3)=O)C)C(C)(C)C1(C)C 64067,Cc1cn2c(C(=O)NCC3CC3CC(=O)NC(c3ccccc3F)C)csc2n1 64068,CC1CN(C(=O)CC2CCC(=O)NC2)CCC1CNC(C1CC2(C1)CC(F)C2)=O 64069,Cc1cc(=NCC2CCN(C)CC2)[nH]cc1S(=O)(=O)NC1CC(CF)C1 64070,c1(C(N2CCC(NC(C(C=C)(C)O)=O)C2)=O)cc2ccc(C(C)C)cc2[nH]1 64071,N1(Cc2nc(C)on2)CC2C(C(=O)N(C(C)Cc3ccccc3F)C)C2C1 64072,C1(C)(OC)CCCN(C(=O)C(C)Cc2ccc(Cl)cc2)C1.C1C(=O)NCCS1 64073,c1(CC)nc(C)c(C(=O)NCC2CC(C)N(C(C3CC(OC(C)(C)C)C3)=O)C2)s1 64074,C1(C(=O)NCC(C)NC(C2(c3ccc(C)nc3)CC2)=O)CCC2(CCC2)O1 64075,c1(C(N(C)CC2(CNC(COC)=O)CC2)=O)nccs1 64076,N1(C(CC2(NC(CC(C(CC)C)O)=O)CCC2)=O)CCC2(CCOC2=O)C1 64077,c1(CN(CCNC(CC(C)c2ccco2)=O)CC2CC2)ccc(S(C)(=O)=O)cc1 64078,Cc1ccc(C)c(N(C(c2scnc2Cl)C(=O)NCC2CC2)C)c1 64079,CC(C)(C)CCCC(=O)NCC12CN(C(C3CCCN3C3CC3)=O)CC(F)(C1)C2 64080,CCC(CC)C(F)C(=O)N(C1CN(C(=O)CC(C)N(C)C)CC1(C)C)C 64081,C#Cc1cnc(NC2CCCCC2CNC(C2(CC)COC2)=O)nc1 64082,CCC(CC)CCC(=O)N1CC2CC1CN2C(=O)CNC(c1ccccc1)=O 64083,C1(NC(CN(C(=O)CCn2ccnn2)CCC)=O)CCC(C(C)O)CC1 64084,c1(CC)[nH]nc(Cl)c1C(=O)NCC1CN(C(=O)C(CN(C)C)c2ccccc2)C1 64085,N1(CC)C(=O)NC(c2cccc(C(=O)O)c2)C(C(=O)OC)=C1C(C(C)OC)OC 64086,C1(OC)CC(CNC(c2coc(O)n2)=O)N(C(C2CNC(=O)N2)=O)C1 64087,C1(NC(c2ccc(CC)s2)=O)(CO)CCN(C(c2ccnc(Cl)c2OC)=O)CC1 64088,N1(C(c2cc(COC)no2)=O)CCC2CN(C(=O)CC(F)(F)Cl)CCC2C1 64089,c1(C(N2C(C)CC(c3cn(C(C)CO)nn3)CC2)=O)cc(Cl)c2c(c1)OCO2 64090,N1(C(C2CC(C)N2C(c2cc(C(N)=O)[nH]n2)=O)=O)CCN2C(=O)OCC2C1 64091,C1(C(=O)NC2(C#C)CCCC2)CC2(CCC2)CN1C(=O)C(CCOCC)SC 64092,c1(C(N(CC(CNC(Cc2c(SCC)cccc2)=O)C)C)=O)cc(O)cc(O)c1 64093,C(C(=O)NOCC1CCC1)(C1CCCO1)NC(c1cc(C2CC2)on1)=O 64094,C1(CNC(C(C2CC2)OC)=O)CCN(C(=O)C(C)(C)N(C)C)C1 64095,Cc1cc(=NCc2ccns2)[nH]c(N2CCC(C(C)C#N)CC2)n1 64096,C1(NC(c2ccc(SC)s2)=O)CCN(C(=O)CN2CCC(C)C2)CC1(C)C 64097,CCCCC(F)(F)C(=O)N1CC2CCOC2(CNC(C2CCN(C)C2=O)=O)C1 64098,c1(NC(=O)Nc2ccc(C(C)NC(=O)OCC)o2)ccc(Cl)c(CC)c1 64099,C1(N)CCCC1(F)F.c1(CN(CC(C)(C)O)C(C2(C)CC2)=O)ccccc1 64100,C1(C(N2CC(CN(C(=O)Cc3ccn(C)n3)C)C2)=O)CCc2ccc(F)cc2O1 64101,CC(C(=O)NCCC1(O)CCN(C(=O)C(C2CCOCC2)F)CC1)C(F)(F)F 64102,N1(C(c2ccc(OC)c(Cl)n2)=O)CCCc2[nH]nc(CO)c21 64103,Cn1nc(Br)c2ncnc(NC3CCN(C(=O)Cc4nsc5ccccc45)C3)c12 64104,CC1Cc2cc(C(=O)NC3CC(F)(CNC(C4CC=CCC4)=O)C3)ccc2O1 64105,C1(CCNC(C(CCC)=CCC)=O)CCN(C(c2cc(C)nn2CC)=O)C(C)C1 64106,N1(C(C(C)OCCCC)=O)CC2(C1)C(=O)NC2.C(C)(C(=O)N1CCCC1)OC 64107,N1(C(C#C)C)CCN(C(c2ccc(N3CCC(O)CC3)cc2)=O)CC1 64108,C1(C(=O)NC(C2CCCCC2)CNC(C2CC(OC)C2)=O)CC=CCO1 64109,N1(C(CCCCCOC)=O)CC2CC(C(N3CCC(CC(F)F)C3)=O)C(C2)C1 64110,N1(C(CN(C(CCCCC)=O)CCCCCCOC)=O)CC(CC)CC(C)C1 64111,c1(C(N2C(C)CCC(C(=O)O)C2)=O)ccc2nc[nH]c2n1 64112,C1(CNC(C2(COC)CC2)=O)CN(C(=O)Cc2cnnn2C)CCC12CCOC2 64113,N1(C(Cc2nc(C)c(C)[nH]2)=O)CCC(C)C(CNC(c2c(C)nsc2N)=O)C1 64114,c1(OC)c(C)cc(C(=O)OC)cc1C.N12Cc3[nH]nc(c3C1)NC2=O 64115,Cc1nn(C)cc1CC(=O)NCCc1cn(Cc2ccco2)nn1 64116,N1(C(C(C)SCCOC)=O)CC2CC(C1)C2NC(=O)C(C)(C)NS(C)(=O)=O 64117,C(=O)(CCC(=O)C(C)(C)C)N1CCC(C)CC1C(=O)NC1CN(C2CCC2)C1 64118,C#CCC(O)C(=O)NCC(F)CNC(c1cccc(C)n1)=O 64119,CC(N=c1nc(-c2ccccc2)nc(N2CCCCCCC2)[nH]1)C1CCC1 64120,CCC(CNC(=O)CCc1cc(Cl)cs1)N=c1[nH]c(C(=O)OC)nc(=N)[nH]1 64121,N1(C(CCC(CC)NC(c2cnco2)=O)=O)CC(C)(C)C2CCCC12 64122,C1(CC(=O)N(CCOCC=C)C)CCN(C(C2CCCCC2O)=O)CC1 64123,C(=O)(C(C)(C)CNC(C1CCOC(CC)C1)=O)NC(c1ccnn1C)CC 64124,N1(C(C2N(CCC)CCC2)=O)CC2CC(C)N(C(=O)CN3CCCNC3=O)C2C1 64125,C(=O)(CC(C)(C)c1ccc(F)cc1)NCCN(C(=O)CCc1ccc(=N)[nH]c1)C 64126,C1(C(N(CC(C)NC(C23CCCC2(C(N)=O)C3)=O)CC)=O)CCC2(CCC2)CC1 64127,N1(C(c2c(C(N)=O)csc2)=O)CC2C(CNC(c3cc(Cl)c[nH]3)=O)C2C1 64128,CCC(CC(F)F)C(=O)NC(C)CN(c1cc(OC)nc(C2CCOCC2)n1)C 64129,N1(C(c2cc(C)ns2)=O)CCCC(F)(CNC(=O)CCc2cc(C)sc2C)C1 64130,C#CCCCC(C)C(=O)Nc1cccc(NC(=O)C(C)ON2CCCC2)c1 64131,c1(CC)cccc(F)c1C(=O)NC1CC(C)N(C(=O)C2=NOCC2)C1 64132,C12(CC(=O)N(C3CCN(C(C4(C)CCNC4=O)=O)C3)CCC)CCC(CC1)OC2 64133,C(=O)(C(C)(O)CC(C)C)N1CCC(O)(CCNC(C(CC)n2ccnc2)=O)CC1 64134,C12(OC)CCCCC(C(=O)NCCCNC(=O)CCC3COC(C)(C)O3)(C1)C2 64135,C(=O)(CCCCCCN=[N+]=[N-])NCC(CC)NC(c1ccc(Cl)c(Cl)c1O)=O 64136,C12(N(C(c3ccc(C(F)(F)Cl)cc3)=O)CCO)CC3CCC(N3)C1C2 64137,N1(C(c2n(C)nc(O)c2)=O)CC(C)(C)CC1CNC(=O)C=CC(N)=O 64138,N1(C(C=C(C)C)=O)C(C(=O)NC(c2ccc(Cl)cc2)C)CC2CCCCC12 64139,C=CC1OCCC1C(=O)NCC(CC)NC(=O)CCC(=O)N(CC)CC 64140,C1(=CC(N2C(C(=O)Nc3c(C(=O)OC)n[nH]c3)CCC2)=O)CCC(C)CC1 64141,N1(C(c2cc(C)[nH]n2)=O)CCCC2CN(Cc3ccnn3C)CC12 64142,CCC(C(=O)N(CC(C)N(C(=O)Cc1ccc(C)s1)C)C)Oc1ccccc1 64143,CC(C)(C)C(CNC(C12CC(C1)C2)=O)NC(C1CC12CC(O)C2)=O 64144,c1(C(N2CCC([N+](=O)[O-])CC2)=O)c(O)ncc2c1CCC2 64145,N1(C(C(CC#C)NC(=O)CN2CCC(=O)CC2)=O)CC2CCC=CC12 64146,N1(CC(=O)NC2CC(N(C(CC(C)C)=O)C)C2)CCP(C)(=O)CC1 64147,N1(C(c2cc(SC)oc2)=O)C(C(=O)NCC(C)(C)C(N)=O)CCC1C(C)C 64148,c1(C(N2CC(C(C)NC(C3CCCC3C)=O)OCC2)=O)csc([N+](=O)[O-])c1 64149,N1(C(CC2CCN(C)C2=O)=O)CC2CCC1C(NC(c1c[nH]cc(Cl)c1=O)=O)C2 64150,CCCCCC(F)C(=O)N1CC(CC(C)NC(C2(C)CC2(C)C)=O)C1 64151,C=CC(CCC)CC(=O)N1CC(CNC(=O)C(C)(C2CC2)OC)(OC)C1 64152,N1(C(CCN(C(=O)C(C)SC)CC#C)=O)CCC(CN(CC)CC)C1 64153,N1(C(CC2CCCC(C)O2)=O)CCCC2(CCCN2C(=O)CC2CCCC2O)C1 64154,C1(OC)CCCC(CC(N2CC(O)(CCNC(=O)COc3ccsn3)C2)=O)C1 64155,C1(N(C(c2sccc2S(=O)(=O)N2CCCC2)=O)CCO)CC[Si]2(CCCC2)CC1 64156,Cc1cc(CC(N2CC(NC(=O)CP(C)(C)=O)CCC2C)=O)cc(Br)c1 64157,C(N1CC(C)C1c1ccccc1)C1CCC1.O([Si](C)(C)C(C)(C)C)C(C)C1CC1 64158,c1(CSCC(=O)NC2C=CC(C(=O)NC(c3ccccc3)C)C2)ccc(Cl)cc1 64159,Cc1ncnc(N(C)CC2CCCCN2C(=O)C(F)CC2CCCCC2)c1F 64160,c1(OC)ccc(C(CN(C)C)NC(N2CCC(C3OCC3(F)F)CC2)=O)cc1 64161,N1(C(C2CCC(CCCCC)O2)=O)CC=C(CNC(=O)CC2CC2(C)C)CC1 64162,C1(NC(CSCC)=O)CC2CN(C(=O)C(c3ccccc3)F)CC2C1 64163,c1(C(=O)NC2CCN(C(c3cnc(O)s3)=O)C2)ccc(F)c(C2CC2)c1 64164,C1(NC(C2(CC(C)C)COC2)=O)CCN(C(C2(C(F)F)CCCC2)=O)CC1(C)C 64165,C1(c2nccc(C)c2)CCN(N2CC(CS(C)=O)C2)C1 64166,CCN=c1[nH]cc(C(=O)NCCOc2ccc(CC#N)cc2)s1 64167,C1(CC(=O)N(CCCNC(c2ccccc2SC)=O)CC)CC2(CCC2)CO1 64168,C(=O)(C#CC1CCCO1)NCC1(COC)CCN(C(C(CC)SC)=O)CC1 64169,CCCCCC(=O)NCC(=O)NCC(CC)NC(=O)CNC(=O)C(C)SC(C)C 64170,C=CCC(CC(F)F)NC(C1CC=CC(NC(=O)C(C)CCCC)C1)=O 64171,C(N=c1cc[nH]cc1C#N)C1C(C)CN(C(c2cnn(C3CCC3)c2)=O)C1 64172,N1(C(C(c2c(C)ccc(F)c2)(F)F)=O)CC2CCCC(CNC(=O)C(C)O)(C2)C1 64173,C1(NC(C(CC)OC)=O)CCOC12CCN(C(=O)Cc1nncs1)CC2 64174,c1(CC(=O)NC2(CC)CN(C(=O)CC3COCCO3)C2)cc(F)ccc1O 64175,N1(C(=O)CCSc2cccc(F)c2)CC2CC(NC(C34CC(CO3)C4)=O)CC1C2 64176,c1(C(N2CC(OC)C(NC(c3[nH]nnc3C)=O)C2)=O)cnc(C)c(C)c1 64177,CCCCC(F)C(=O)N1CC2CC1CN2C(c1ccn(C2CC2)n1)=O 64178,C1(O)(C(=O)NC(C(=O)N(CCC)CCN(C)C)c2cccs2)CCSC1 64179,c1(C(=O)NC(CNC(CCN(C)CC)=O)CCOC)cc2sccc2s1 64180,c1(C(N(C2CCN(C(c3cnc(F)c(F)c3)=O)CC2)C)=O)cccc(Cl)c1F 64181,C(=O)(C1COc2ccccc21)NCC1N(C(C(C(CC)C)O)=O)CC(C)(C)C1 64182,c1(C(=O)NC2CC3CN(C(c4cc(OC)ns4)=O)C2C3)ccc2nccn2c1 64183,c1(C(N(CC(CC)NC(=O)CCc2cscn2)C)=O)ncc(C)cn1 64184,c1(SC)ncc(C(N2CC(O)(CNC(C3C(F)(F)C34CC4)=O)C2)=O)c(O)n1 64185,C(CO)(C(=O)N1CCC(CCNC(=O)CC2(C3CC3)CC2)C1)N(C)C 64186,n1(CC(=O)NC2C(CNC(CCCOC(C)=O)=O)CCC2)cc(Br)ccc1=O 64187,N1(C(c2onc(COC)n2)=O)CCN(C(=O)C=CC2CCOC2)CC1 64188,N1(C(C(C)(N(C(CC2CC(SC)C2)=O)C)C2CC2)=O)CC(C)(C#N)C1 64189,S(=O)(=O)(c1ccc(C2CN(CCNC(c3cc(N)cnc3Cl)=O)CCO2)s1)NC 64190,N1(C(C)=O)CCCCC1C(=O)NCC(C)NC(c1cccnc1Br)=O 64191,c1(C(N(C)CCN2CCN(C(=O)CCc3cncs3)CC2)=O)cc(N)cc(O)c1 64192,C1(C(N2CC(C)N(C(=O)CCCN(C)C)CC2)=O)CC2(C1)C(F)(F)C21CC1 64193,CC(C)CC(O)C(C)C(=O)NC(C(=O)N1CC(n2cnnn2)C1)C1CC1 64194,c1(C(N2C(CCNC(c3c(C)ncs3)=O)C(C)CCC2)=O)ccc2ncnn2c1 64195,C1(N(C(C(Cn2ccc(C)n2)C)=O)C)CCCN(c2nccc(C#N)n2)CC1 64196,CC1(C)CC(NC(c2cc(F)cc(Br)c2)c2nnnn2CN2CCOCC2)CCO1 64197,c1(OC)cc(C(=O)NCC2CN(C(c3c(O)noc3C)=O)C2)ncn1 64198,Cc1cccc(C=CC(=O)NCC(C)(C)OCC(=O)NCCC(O)C(F)(F)F)c1 64199,Cn1nc(C(N2CCSCC2CCNC(C2CCC2(C)C)=O)=O)cc1C(F)F 64200,c1(C(N2C3CCC(NC(c4cc(OC)n(C)n4)=O)(C3)C2)=O)cccc2c1NCC2 64201,n1(CCOC)ncc(C(N2CCOCC2CCNC(C2CNC(=O)N2)=O)=O)c1C 64202,N1(C(C(C(C)C)N(C)C)=O)Cc2nccn2CC(NC(C2(C)CC2(F)F)=O)C1 64203,c1(C(N2CCC3(C(C(=O)Nc4n(C)nc(C)c4Cl)C3)C2)=O)cc(C#N)ccc1F 64204,c1(C(=O)NC(c2cc(C)cc(C)c2)C)cc(S(=O)(=O)N2CCOCC2)cn1C 64205,C1(C(=O)NCCCCN(C(CCC2CC(C)C2)=O)C)CCC2(CC1)CC(O)C2 64206,c1(C(N2CCC(C(C(=O)N(CC(=O)OC)CCC)C)C2)=O)cc(C)ccc1O 64207,N1(C(CC2C(C)C2)=O)CC(O)(CCNC(c2csc(N3CCCCC3)n2)=O)C1 64208,Cc1cc(=NC(=O)C(=O)C(C)(C)C)[nH]n1-c1ccccc1 64209,C1(CCF)(NCC(=O)NC(c2ccccc2)C(=O)NC2CCCOC2)CC(O)C1 64210,c1(CC(=O)NC(C)C(=O)NCc2nn(C)cc2CO)ncccc1F 64211,Cc1oc(C(C)C)cc1C(N1CCC(C(C)O)CC1)C(=O)Nc1ccccc1Cl 64212,c1(C(N2C(C)CCC(c3ccccc3)C2)=O)cc2ccccc2oc1=O 64213,c1(OC)ccc(O)cc1C(N1CCCCC(NC(=O)C2=CCCCC2)C1)=O 64214,c1(CCC(=O)N(C)CC2CN(C(=O)CC3CCCC3)C2)ccn(C)n1 64215,CC(O)CCCC(=O)NCC1CCN(C(C2CN3CCC2CC3)=O)C1 64216,C1(CCNC(c2ccc(CC)o2)=O)CN(C(=O)C(c2ccc(C)o2)C)CCCO1 64217,c1(CS(C)=O)cccc(C(=O)NC2CN(C(=O)CC3C=CCC3)C2)c1 64218,C1(NC(C2(COC)CN(C(c3cnsc3)=O)C2)=O)CC(=O)N(C)C1 64219,C1(O)(CNC(CN(C(=O)OCC)C)=O)CCN(C(=O)C(C(C)C)n2ccnc2)C1 64220,C1(CC)CN(C(c2c(C)nsc2C)=O)CC1C(=O)NC1(C)CC1(C)C 64221,Cc1cc(C(=O)NC2C3CCN(C(=O)Cc4ccc(O)c(C)c4)C23)ccc1F 64222,N1(C(C(=O)NCCOCCOC)=O)CCCCC(C(=O)Nc2nn(C)cc2Cl)C1 64223,N1(C(C(CC)NC(C)=O)=O)CCC12CN(C(C1CCC(C(F)(F)F)O1)=O)C2 64224,C1(CC(=O)OC)Cc2ccccc2CN1C(c1cnc2c(Cl)cccn12)=O 64225,C1(CC(=O)N(CCC)Cc2ncc(C3CC3)o2)Cc2cc(C(F)(F)F)ccc2O1 64226,c1(C(=O)NCCC2(OC)CN(C(=O)C=C(C)Cl)C2)cccc(S(N)(=O)=O)c1 64227,c1(C(N2C(CN(C(c3c(CC)n(C)cc3)=O)C)CCC2)=O)cnc2cc[nH]c2c1 64228,c1(C(N2CCC(CC=C)(NC(C3CCCC3O)=O)C2)=O)ccn2c(O)nnc2c1 64229,C1(N(C(c2csc(CO)n2)=O)CC)CCN(C(=O)COC(C)=O)CC1 64230,C(CNC(c1cc(C(N)=O)co1)=O)(CC(F)(F)F)NC(c1ccc(OC)nc1)=O 64231,C1(C(N(CCCNC(=O)Cc2cc(Cl)cs2)C)=O)CN2CCCCC2CO1 64232,Cc1cccc(C(=O)NC2(C)CCN(C(C3CC(=O)N3)=O)C2)c1N 64233,C=C(Cl)CC(C(=O)N1CCC2(CC1)N=N2)NC(c1cccnc1O)=O 64234,c1(NC)scnc1C(=O)NC(COC)C(=O)NCCCc1cccnc1 64235,C1(CNC(c2ccccc2N2CCOCC2)=O)CCCCN1C(=O)C=CCBr 64236,C(=O)(C(CC(C)C)NC(=O)C(C)CCOC)N(CC(CCC=C)O)C 64237,C1(NC(=O)CCc2cc(Cl)cs2)CC2(C1)CC2NC(c1cc(C2CC2)[nH]n1)=O 64238,C12(CNC(CC(C=C)C)=O)CN(C(c3cnc(C(C)(C)C)[nH]3)=O)CC(F)(C1)C2 64239,C1(S(N)(=O)=O)(C(=O)NC2CCC(NC(c3cnn(C)c3C(F)F)=O)C2)CCCC1 64240,N1(C(CC(C(C)(C)C)NC(c2c(C)oc(CO)c2)=O)=O)CCCC2(C=CCO2)C1 64241,c1(C(=O)NC(CC)CNC(c2ccc(C)cc2F)=O)cccc2cccc(Cl)c12 64242,c1(N(CC(=O)NC)C)nc2cc[nH]c2c(=NC(C)c2ncccc2Cl)[nH]1 64243,c1(CC)cc(Br)ccc1C(=O)NC1CCN(C(c2csc(NC(C)=O)n2)=O)C1 64244,N1(C(CC(CC(C)C)O)=O)CC2CCC1CN(C(=O)C(N1CCSCC1)C)C2 64245,C1(NC(CC(C)c2cccnc2)=O)CC12CCN(C(=O)C(C)(C)CCC#N)CC2 64246,C(=O)(CC1C(=O)Nc2c(F)cccc21)NCC1(NC(=O)CCF)CCOC1 64247,C1(CC)CN(C(C2CCC(C)CC2)=O)CCN1C(c1cccc(SCC#N)c1)=O 64248,C(=O)(CCCCCS(N)(=O)=O)N1CCC(C)C1CNC(c1cc([N+](=O)[O-])c[nH]1)=O 64249,C(=O)(C(C)CNC(=O)C(CC1CC1)NC(C1CC1C#N)=O)NC 64250,N1(C(CC2C(C)C2)=O)CC(NC(C2(C)CCCCO2)=O)C2CCCCC12 64251,N1(C(C(C=C)O)=O)CC2CCCC1(CNC(c1cccc(OC)c1F)=O)C2 64252,c1(OC)cc(CC(=O)NC2(CNC(C3CCC(C)(C)CO3)=O)CCC2)cc(F)c1 64253,CC(Cc1ccc(Cl)cc1)CC(=O)NC(C)(CNC(=O)C=Cc1nccs1)CO 64254,CC(CCC(C)(C)C)C(=O)N1CCN(CCN(C)C(c2cc(Cl)ccn2)=O)CC1 64255,N1(C(CCC=C)=O)CC2(CCN(C(c3ccccc3-c3ncc[nH]3)=O)C2)C1 64256,CC1CCCC(CNC(c2cc(CNC(c3cc(Cl)n[nH]3)=O)nn2C)=O)CC1 64257,C1(C(=O)NCc2cccnc2O)CSCCN1C(c1ccnc(Br)c1)=O 64258,C1(C(=O)NCCOC(C)=O)CCCCN1C(C1(C)C=CCCC1)=O 64259,c1(C(n2cc(C3(F)COC3)nn2)C)ccc(C(=O)CCOC(C)(C)C)c(Br)c1 64260,N1(C(CC(=O)OCC)=O)CCCC(C2CCCCN2C(c2cccn2CC)=O)C1 64261,CC1OCCC1CCNC(C1(CNC(c2sccc2CO)=O)CCC1)=O 64262,c1(C(C(N2CC(C)(NC(C3(c4cc(C)no4)CC3)=O)C2)=O)O)ccc(F)c(F)c1 64263,C(=O)(C(CCS(C)=O)N(C)C)NCCC(C)CCNC(c1cnnn1C)=O 64264,N1(CCC(=O)N(C2(O)CCCCC2)CC(C)CCO)CCOCC(C(=O)OC)C1 64265,Cc1nn(C)cc1S(=O)(=O)N(C)C.c12cc(ccc1Cl)CS2 64266,C12(NC(c3cc(O)ncn3)=O)COC(C1)C(NC(c1scnc1Cl)=O)C2 64267,N1(C(c2cc(OCC)ncc2)=O)CC2CC(Nc3nc4ccccc4s3)CC1C2 64268,C1(C)(CNC(COC(CC)C)=O)CCCN1C(=O)CN(C1CCC1)C 64269,C(=O)(C(C(F)(F)F)C(F)(F)F)NCC1(O)CN(C(CC2CCN(C)C2)=O)C1 64270,C1(CNC(=O)CCCC2CCCC2)CC2CCC1N(C(c1cccnn1)=O)C2 64271,C#CCCCCCNC(c1ccc(CNC(=O)CC2CCCOC2)nc1)=O 64272,c1(C(=O)NCC(CO)NC(c2n(CC)ccc2)=O)cnc(N)cn1 64273,c1(C(=O)NCC(C)N(C(c2n(CCC)ncc2)=O)C)ccc2c(c1)C(=O)CCN2 64274,N1(C(C)C)CC(NC(c2cc(CNC(C3CC3(F)Cl)=O)[nH]n2)=O)CC1=O 64275,C(CC(CC)CC)(c1n(CC=C)nnn1)Nc1cccc(C(C)CC)c1 64276,c1(C(=O)NCC2C(NC(C(CC)NC(C)=O)=O)CCCC2)ncc2[nH]ncc2n1 64277,N1(C(C(CC)N(C)CC)=O)CCC(C(=O)Nc2cc(C(=O)OC)nn2C)CC1 64278,C12(C(N3CCC(C(C)NC(C=C(C)Cl)=O)C3)=O)CC3CCC(CC(C3)C1)C2 64279,Cc1cccc2c(CN3CCC(NC(c4cnn(C)c4)=O)C(O)C3)c[nH]c12 64280,C(c1nc(C)c(C)[nH]1)=CC(=O)NCC(CC)NC(c1ncc(C)cc1O)=O 64281,C1(CNC(c2ncncc2Cl)=O)C2CCC(C2)N1C(C12CC3CC1C2C3O)=O 64282,Cc1cc(=NCCC2CCC(=O)N2)[nH]c(N2CCN(CC(C)C)CC2)n1 64283,CCCC(CCC)C(=O)NC1CCCC(NC(c2cc(C(F)(F)F)on2)=O)C1 64284,CC1CCCCC1(C)C(=O)NCCOCCN(C(=O)COc1cncc(Cl)n1)C 64285,c1(N2CCCC(NCc3cc(OCC)ncc3Br)CC2)ncnc2c1CC(=O)N2 64286,C1(CNC(C(CC)CC)=O)CN(C(c2ccnc(C3CC3)n2)=O)CC1(C)C 64287,N#Cc1cc(C(N2CCC3CN(C(c4cc([N+](=O)[O-])cs4)=O)CC23)=O)ccc1F 64288,c1(N2CC3CN(Cc4cc(C)nc(C)c4)C3C2)ncnc2n[nH]cc12 64289,c1(CC)cccc(C(=O)NC2(CNCc3ccc(CSC)o3)CCOCC2)c1C 64290,Nc1cc(C(N2CCN(C(=O)CCCN3CCCC3)CC2C2CC2)=O)cc(O)c1 64291,c1(C(=O)Nc2cccc(-n3cc(C(=O)OC)nn3)c2)ncc(Cl)nc1OC 64292,C1(NC(c2n[nH]c(C)c2C)=O)CCN(C(c2ccc(C(C)C)c(F)c2)=O)C(C)C1 64293,c1(CC(N2C(CCNC(c3c(C)cc[nH]3)=O)CCCC2)=O)c(F)cc(F)cc1F 64294,c1(C(=O)Nc2c(C)nccc2Br)c[nH]c2cc(-c3ccccn3)cnc12 64295,c1(CC(=O)NCC(CC=C)NC(c2cc(Cl)no2)=O)cn2ccsc2n1 64296,c1(C(N2CCC(N(C(CN(CC)CC)=O)C)C2)=O)nnc(O)c(Br)c1O 64297,C(=O)(C1=CCC(C)(C)CC1)NC1C(C)N(C(=O)CCNC(N)=O)CCC1 64298,C1(C(=O)NC2(C)CN(C(C(c3cscn3)N(C)C)=O)C2)CC2CCC(C1)C2O 64299,c1(C(=O)NC(CCN(C(C(CC=C)(F)F)=O)C)C)cnc2cccc(C)n12 64300,n1(CC)ccc(CC(=O)NCC(CNC(C2CC=CCC2)=O)OC)n1 64301,N1(C(CC=CCNC(C(C=C)C)=O)=O)CCN(CC)CC1 64302,Cc1cnn(C)c1CC(=O)NCC1CCC(NC(c2ccc(N(C)C)nn2)=O)C1 64303,c1(C(N2CCC(NC(C(C(C)(C)C)OCC)=O)(CF)C2)=O)cc(C)c(N)cc1Cl 64304,c1(NC2CC(CNC(CC(CC)C(C)C)=O)C2)ncnc2sc3c(c12)CCC3 64305,N1(C(C2CCN(C(C3CCC(CC)CC3)=O)C2)=O)CCCNC(=O)C12CC2 64306,c1(NC(C2(C)CCN(Cc3nccc(C(=O)OC)c3)C2)=O)cc(Cl)c(Cl)cc1O 64307,c1(C(N(C(C)CNC(C23CCC(CO2)C3)=O)C)=O)cc(C#N)ccc1F 64308,C(=O)(C(COC)COC)Nc1cc(N)no1.C(=O)(C1CO1)SCCOC 64309,C1(CCN(C(C2CCN(C(=O)NC)C2)=O)C)CCCCN1C(c1ccc(F)s1)=O 64310,C1(CNC(C2C(C(C)C)CCO2)=O)CCCCN1C(=O)CCN(S(C)(=O)=O)C 64311,N1(C(C(CSC)OC)=O)CCC2(CCC(NC(c3[nH]c(O)nc3C)=O)C2)CC1 64312,C(CCCC(C)(C)C)NC(CC(CNC(C1CC1(C)C)=O)OC)=O 64313,Cc1nn(C)c(C)c1C(=O)NC12CC1CN(C(=O)CC1CCC(C)(C)CO1)C2 64314,c1(COC)nc(NCc2cnn(CCF)c2)cc(=NC(C)C2CCCO2)[nH]1 64315,C(=O)(CC1=CCCCC1)NCCOC(C)(C)CNC(=O)CCNC(=O)CO 64316,C1(NC(c2cc3c([nH]2)CCCC3)=O)CCN(C(C2(O)COC2)=O)CC12CCC2 64317,C1(NC(COCCCC)=O)CC2CCC(C1C)N2C(c1cnn(CCF)c1)=O 64318,C(N=c1ccc(NC(c2cncc(Cl)c2)=O)c[nH]1)c1c(SC)cccc1 64319,CCC(CC(=O)NCC1C=CCN1C(c1cc(OC)cs1)=O)C(C)C 64320,Cc1nc(C(=O)N(C)CC2CCCCN2C(C2CC2c2cn[nH]c2)=O)c(C)s1 64321,C1(C(N2CCC(NC(C3CCOCC3)=O)C2)=O)(OCC)CCOCC1 64322,CCC(F)(F)CN(C(C=CC(C)NC(=O)CC1C=CCC1)=O)C.c12cc([nH]n1)S2 64323,c1(C(=O)NC2CCN(C(C3NC(=O)OCC3)=O)C2)ccc2nc(O)[nH]c2c1F 64324,Cc1cccc(Br)c1C(C(=O)NCC1(O)CCCOC1)NC(=O)CCC1(C)N=N1 64325,c1(C(=O)NCC2(CNC(CC3C(C)OCC3)=O)CC2)ccc(C(N)=O)cn1 64326,CC1(C)CCCN(C(=O)Cc2cnns2)C1C(=O)N=c1ccn(C2CC2)[nH]1 64327,CCC(CN(C)C)CC(=O)NC1(CO)CN(C(C2CC(OC3CC3)C2)=O)C1 64328,c1(CCC(=O)NCC2CCCC(NC(C=CCC)=O)C2)ccc2ccccc2c1 64329,C1(NC(C2(CC)COC2)=O)CCC2CCN(C(c3csc(=NC4CC4)[nH]3)=O)C1C2 64330,N1(C(C(C)CNC(C2CCCN2C2CC2)=O)=O)CCCCC(CO)C1 64331,N1(C(C(N2CCOC2=O)C)=O)CC2(CCCC2)C1C(=O)NC1CCC2CCC12 64332,C(c1ccc(OC)cc1OC)=CC(N1CCCC(NC(CCOC)=O)C1C)=O 64333,C(=O)(C(C)(C)COCC)N(CC(=O)NC(C=C)CO)CCOC 64334,C1(N(C(CCOCCOC)=O)C)CCN(C(c2cnn(C)c2N)=O)CC1C 64335,N1(C(=O)COCC2CCOC2)CC2(C1)CN(C(=O)C(F)C1CCC1)C2 64336,C1(NC(Cc2n(C)ncc2)=O)CC2CN(C(c3ccn(C(C)(C)C)n3)=O)CC12 64337,N1(C(C2N(C(CC)=O)CSC2)=O)CC2(CNC(=O)CCF)CC1(COC)C2 64338,C1(F)(CNC(C2N(C)CCC2)=O)CCN(C(c2ccc(-c3cccs3)o2)=O)C1 64339,C1(CNC(=O)CC2CCC3CC23)CC2COCC2N1C(=O)CCn1cncn1 64340,c1(C(N2CC(CNC(C(C=C)(C)O)=O)C(F)(F)CC2)=O)ccc2nc(O)[nH]c2c1 64341,N1(C(C)C)CCCCC1C(=O)NCCCN(C(=O)C(C1CCOCC1)C)C 64342,C(=O)(C(F)C(C)(F)F)NCCC1(C(N2C(C)(CCC)CC2)=O)CC1 64343,N1(C(c2cc(C)oc2C)=O)CCCOC(CNC(=O)Cc2cocn2)C1 64344,C(=O)(CC1=CCOCC1)N1C(CCNC(CCC(=O)N(C(C)C)C)=O)CSCC1 64345,CCC(CC)C(F)C(=O)NCCCC(O)C(=O)N(C1CC1)C(C)C1CC1 64346,C12(NC(C(C)CC3CC3)=O)CCCC1CN(C(c1csc(C3CC3)n1)=O)C2 64347,Cc1cc(C=CC(=O)NCC(C)(O)CNC(=O)C(C)Cc2ccco2)c[nH]c1=N 64348,C(=O)(C(O)CCNC(c1cc(C2CC2)on1)=O)N1C(C=C)CC1 64349,c1(C(N(C(CN(C(C2(OC)CCC2)=O)C)C)C)=O)ccccc1CC(C)(C)C 64350,CCC(CC(=O)N(CCCN(C)C(C1(C)CCNC1=O)=O)C)C(=O)OC(C)(C)C 64351,N1(C(Cc2scc(C)n2)=O)CCCC(C)C1CNC(=O)Cc1cnoc1 64352,c1(C(=O)NCC(C)NC(=O)NC(C(=O)N(CC)CC)C)cc(Cl)ccn1 64353,c1(C(N2CC3C(NC(C(C(C)(C)F)(C)F)=O)C3C2)=O)ccc(N)c([N+](=O)[O-])c1 64354,C(=O)(CC(CC)C(C)C)N1CCN(C(c2c(OC)nsc2)=O)C(CC(F)F)C1 64355,N(C1CC(C)n2ncnc21)CC(=O)N(C(=O)CCc1ccccc1)C 64356,C(CCCC(=O)NC1CCCC1NC(=O)Cc1ccc(C)o1)OC 64357,c1(SC)nc(N(C(C)CCNC(=O)C(CO)NC(N)=O)C)cc(Cl)n1 64358,CN1C(=O)OCC1C(=O)NCC12CC1CN(C(=O)CC1(O)CC1)C2 64359,C(C(CC(F)(F)F)NC(=O)CCc1nccs1)NC(=O)C=CCO 64360,C(c1cocn1)=CC(=O)N(CCOC)CCNC(=O)CC1(OC)CCC1 64361,c1(CC)cc(C(=O)N(C2CN(C(=O)CNc3cnn(C)c3)C2)C)c2c(c1)CCO2 64362,c1(C(CC)N(CCO)CC2CC2(F)F)ccccc1 64363,c1(C(=O)NC2C(C(C)(C)C)N(C(=O)C(=O)N(C)C)CC2)nnn2c1CCCC2 64364,C(N=c1ccnc(C2CCCC2)[nH]1)C1(NC(c2c(C(C)C)ocn2)=O)CC1 64365,c1(OC)cc(C)c(C(=O)NC2(CCNC(C34CCCC3C4(F)F)=O)CC2)cn1 64366,c1(OC)c(Br)cc(CN2C(C(=O)NC(c3ccc(I)cc3)C)CC3CC23)cc1Br 64367,C(C(C(C)C)NC(=O)C(C#N)=C1CCCC1)NC(C(C)OCCOC)=O 64368,CC(C)(C(=O)NCC1CCC(NC(=O)CN2CCCC2=O)C1)n1cc(Br)cn1 64369,c1(N2C(C(=O)NC(c3cnccn3)C)CNCC2)ncnc2c(F)cccc12 64370,c1(C(N2CCCC(C(C)NC(c3cc(C)sn3)=O)C2)=O)n[nH]c2cc(Cl)ccc12 64371,Cc1cnn(CCC(N2C(C(N3CC(OCCF)C3)=O)CC2C)=O)c1 64372,C1(OCC)CC(NC(=NCCC(=O)N(C)C)NCC2CC2)C12CCOCC2 64373,C1(CNC(C2C(=C)C2)=O)CN(C(=O)Cc2ccc(Cl)cn2)CC12CC2 64374,CC1(C)CCCN(C(c2nccc(Cl)c2O)=O)C1CNC(=O)Cc1c[nH]nc1O 64375,c1(C(N)=O)cccc(CC(=O)NCCOCCCNC(=O)C(O)C(F)F)c1 64376,C1(NC(c2nc(C)oc2C)=O)CCN(C(=O)C(C)Cc2cnn(C)c2)CC1F 64377,CCC(CC(=O)NCC1CN(C(c2ccoc2C)=O)C2COCC2O1)C(C)(C)C 64378,C(CO)(C(=O)N1CCCC1C(C)(C)NC(=O)C(C)OCC1CC1)OC 64379,c1(C(=O)NCCCS(C)(=O)=O)cn2c(n1)CN(C(C1CC(O)C1)=O)CC2 64380,Cn1cnc2c(C(=O)NCCC(O)CNC(C34CC(F)(C3)C4)=O)ccnc12 64381,C1(CNC(C(CC)n2cncn2)=O)CN(C(=O)Cc2csc(Cl)c2)CC1C 64382,C12(NC(C3C(C)OCC3)=O)CCOC(CNC(C3CC(=O)N(C)C3)=O)(C1)C2 64383,c1(C(N(CC(O)CNC(=O)COc2ccc(Cl)nc2)C)=O)cc(F)c(F)cc1F 64384,C1(CC(=O)NC2CCN(C(=O)CC34CCCC3C4)C2)(CC=C)CCCC1 64385,C1(NC(CCN(CC=C)C(c2cn(C)cn2)=O)=O)CCCCC1C 64386,C(=O)(CCC(C(=O)OC)NC(=O)C(N1CCC(SC(F)F)C1)C1CC(O)C1)OC 64387,N1(C(C2(NC(c3c(CC)c[nH]n3)=O)CCOCC2)=O)CC(OC)C2(CC2)C1 64388,O=C1NCC2(CCN(C(=O)NCCSCCO)CC2)N1 64389,C1(NC(CC2C(C)OCC2)=O)CCN(C(c2cccc(O)c2)=O)CC1C(N)=O 64390,c1(C(=O)NC23CCN(C2)C3=O)ccc(O)c(Cl)n1.C=CC(O)(CC)c1ccccc1 64391,C1(C(=O)NCC2CCCCN(C(Cc3c(C)noc3)=O)C2)Cc2ccncc2C1 64392,C1(C(C)(C)C)CCC(C(O)C(=O)OCCOCc2c(C(=O)OC)cccc2)CC1 64393,Cc1[nH]c(-c2ccco2)nc(=S)c1C(=O)NC1CCN(C(=O)CCCF)CC1F 64394,C#CCCCC(=O)NC(COC)C(=O)NC(c1nncn1C)CO 64395,C12(C(=O)NCC3(OC)CN(C(=O)C(F)C(C)C)C3)CC(C)(C1)OC21CCOCC1 64396,c1(C(C)C)nc(NCCC(=O)NC2CCCSCC2)cc(N(C)CC2CC2)n1 64397,C(N=c1[nH]c(=NC(CCO)C(F)F)[nH]c2c(F)cccc12)C1(OC)CCCC1 64398,N1(C(c2sc(CC)c(C)c2)=O)CCN(C(=O)C(C)Oc2ccccn2)C(C)C1C 64399,N1(C(C(CC)O)=O)CCN(C(CNC(c2cc(C(N)=O)[nH]n2)=O)C(F)(F)F)CC1 64400,C1(CNC(c2ccc(CC)[nH]2)=O)CC2(CCC2)CN1C(=O)CCc1ccon1 64401,c1(CCC(=O)NCC2(CNC(C(C)CO)=O)CC2)nc(=O)c2ccccc2n1C 64402,C(C(C)(CNC(c1nonc1CC)=O)OC)NC(C(C)OCC#C)=O 64403,C1(CNC(C2(CC=C)CC=CC2)=O)COCCN(C(C2CC3(CC(=O)N3)C2)=O)C1 64404,C(=O)(C(F)CCC(C)(C)C)N(C(C)CCNC(c1cccnc1O)=O)C 64405,c1(C(=O)NCC2(CNC(c3nc(C)oc3C)=O)CC2)cccn2cnnc12 64406,CCC(CC(C)C)C(=O)N1CC2C(CC(=O)NCC3CC3C(C)C)C2C1 64407,C12(C(=O)NCC3CC(F)CN3C(=O)CC34CCC(CC3)C4)CCN(CC1)C2 64408,N1(C(CC(C)(C)CC(F)F)=O)CC2CCN(C(c3nncs3)=O)CCC2C1 64409,N1(C2CC(C(=O)OC)C23CCC3)CC(NC(=O)OC(C)(C)C)CC(C)(C)C1 64410,C(=O)(C1=NOC2(CCC2)C1)Nc1c(C(=O)OCC)ncc(Cl)n1 64411,C1(CCNC(CSCC#C)=O)COCCN1C(c1cn(CC)cn1)=O 64412,c1(NCC(CNC(CC(CCC)C)=O)C(F)(F)F)ncccc1[N+](=O)[O-] 64413,c1(CC)onc(C)c1C(N1CCC(OCCNC(=O)C(C)=CCO)C1)=O 64414,C(=O)(CC(F)(F)CC(=O)OC)NC(CNC(c1c(CC)n(CC)nn1)=O)C1CC1 64415,Cc1ccc(C)n1CC(=O)NCCC(C)N(C)C(c1cccc(C(N)=O)c1)=O 64416,CN=c1[nH]nc(CC(=O)NCC2CC(NC(C3CC3c3ccc(F)nc3)=O)C2)s1 64417,c1(NC)ccc([N+](=O)[O-])cc1OC(F)F.C(Cl)(C(F)(F)F)N1CCC1 64418,c1(C(=O)NC2C(C=C)CN(C(=O)C(C)O)C2)cc(S(N)(=O)=O)ccc1F 64419,C1(NC(c2nc(COC)sc2)=O)CCN(C(=O)C(C)OC(C)(C)C)CC(C)(C)C1 64420,C(C)(c1cccnc1)=CC(=O)NC(CN(C(CCC#C)=O)C)CC 64421,c1(CNC(CNC(C2C(C)C2)=O)=O)ccnc(C(=O)NC2(C)CC2(C)C)c1 64422,CN=c1nc(N(C)CCNC(c2cc[nH]n2)=O)[nH]c(=NCC2CCC=CO2)[nH]1 64423,c1(C(=O)NCCN(C(c2cc(OCC)ncc2)=O)CC)cnn2c1CCCC2 64424,c1(OC)ccc2c(c1)CC(C(=O)NCC(O)CCNC(=O)CC1CCOCC1)O2 64425,C1(NC(CC)=O)CN(C(c2ccc(NC)cc2)=O)Cc2nccn2C1 64426,N1(C(c2cc(CC)nn2C)=O)CC2CCCC2C1C(N1CC(CO)CC(C)C1)=O 64427,C1(CC(N2CC(CNC(C3CCC(c4ccccc4)C3)=O)C2)=O)CCCC(O)C1 64428,c1(C(N2CCCC(C(=O)NCc3cc(OCC)no3)C2)=O)cnc(O)cc1OC 64429,c1(CNC(C(C)N(C(=O)C(C)SCC)CCC)=O)cc(O)ccc1C 64430,c1(C(N2CC=CC(C(=O)NCC=C=C)C2)=O)ccc(C)c(C)n1 64431,C1(NC(Cc2nc(C)sc2)=O)CN(C(C2CCC=CCC2)=O)C2(CCOCC2)C1 64432,N1(C(COC2(C#C)COC2)=O)CCOCC(C)(CNC(c2ccc(C)nn2)=O)C1 64433,c1(NC(C2(C)CN(C(C(CC)=CCCC)=O)C2)=O)ccc(O)c(CO)c1 64434,N12CCOCC(C1)N2Cc1nc(C)n(C)n1.c1(OCC)cccnc1.C=O 64435,N1(C(CCC=CCC=C)=O)CC(NC(=O)COCC(F)(F)F)CC12CCOC2 64436,C1(C)(C(=O)NC2CC(OC)CN(C(CC=CC)=O)C2)CCS(=O)(=O)CC1 64437,c1(C2(C(=O)NCC3(F)CN(C(C4CCCO4)=O)C3)CCCC2)ccc(F)cc1 64438,N1(C(C2CC(C)(C)N(C(C3CCC(O)CC3)=O)CC2)=O)CC2CCC(O)C(O)C12 64439,c1(C(=O)NCCN(C(=O)CCOC(C)CC(C)C)CCC)cc(C2CC2)n[nH]1 64440,c1(CC)ccc(C)cc1C(=O)NC1CCN(C(c2cc(COC)on2)=O)C(C)C1 64441,c1(N2C(C3(NC(CCC(=C)C)=O)CC3)CCC2)ncnc2c1COC2 64442,CC(=O)CCCC(=O)NCC1(O)CCN(C(=O)C(C)OC2CCCCCC2)CC1 64443,Cc1oc(C#N)cc1C(=O)N(C(C)CCNC(=O)C=CSc1ccccc1)C 64444,N1(C(C=C(C)CNC(c2cccc(CC#N)c2)=O)=O)CCC(C)C(O)C1 64445,CC(C)C(C(=O)NCC(CNC(=O)Cc1cscn1)CO)NC(N)=O 64446,N1(C(C(C=CC)O)=O)CCCCCC(NC(=O)C=Cc2c(C)nn(C)c2Cl)C1 64447,N1(C(C2CC(C)NC(=O)C2)=O)CCC2(CC1)CCN(C(=O)CC1OCCCO1)C2 64448,CC(CC(=O)N(CCCN(C)C(C1(Cc2ccccc2)CC1)=O)C)C(F)F 64449,N1(C(c2c(CCNC(C(C)OC(C)(C)C)=O)n[nH]c2)=O)CCC(C2CC2)C1 64450,C1(CN(C(COC(CC)C)=O)C)CC(F)CN1C(c1cnc(C(C)(C)C)s1)=O 64451,C1(NC(=O)Cc2csc(-c3ccsc3)n2)CCCCC1CNC(c1cscn1)=O 64452,N1(C(C(CC2CCCC2)NC(c2c(CC)[nH]cc2)=O)=O)C2CCC1CC2 64453,N1(C(c2csc(O)n2)=O)CCC2CCN(C(c3nc[nH]c3C(F)(F)F)=O)CC2C1 64454,N1(C(C(CC)NC(C)=O)=O)CC(O)CC1CC(=O)Nc1ccsc1 64455,C=CCC(C)(C)CC(=O)NC(c1ccc(F)cc1)CNC(=O)Cc1nccn1C 64456,c1(NC(C2(c3nn[nH]n3)CCCOC2)=O)cc(Cl)c2ccc(Br)cc2n1 64457,c1(OC)ncccc1CN1CC(F)CC1C(=O)NC(c1ccccc1)(C)C 64458,C1(CNC(C(=O)NCC)=O)CN(C(=O)CCC2C(=O)ON=C2C)C2(CCC2)C1 64459,c1(C(=O)NC2(C)CCCN(C(Cc3ccn(CC)n3)=O)C2)ccc2nsnc2c1 64460,C#Cc1ccc(C(=O)NC2CCOC(C(=O)N(C)C3CC3)C2)cc1C 64461,Cc1cccc(C=CC(N2CCC(O)CC2C(=O)N(C2(C3CC3)CC2)C)=O)c1 64462,c1(C(C(=O)N(C2CCC2)C(C)C)N(C(C=C)C2CC2)C)ccoc1C 64463,CS(=O)(=O)c1cnn(CC(N2CC(OCCNC(C3CC3C(F)(F)F)=O)C2)=O)c1 64464,c1(C(C(N2CC3C(CNC(C4(OC)CCCC4)=O)(C3)C2)=O)C)ccc(F)cc1F 64465,C12(C(=O)NC3(C)CC=CC3)CCC1CN(C(c1ccc(Cl)cc1)=O)C2 64466,C1(CNC(C(C)CN(C)C)=O)CC2COCC2N1C(=O)C(F)(F)c1cnnn1C 64467,c1(C(=O)NCCN(C(c2nc(CCCCC)sc2)=O)CC2CC2)ncccc1O 64468,N1(C(CCN(CC#C)C(c2cccc[n+]2[O-])=O)=O)CCC12CCC2 64469,c1(C(C)C)nc(CNC(=O)C=CCNC(=O)CCC2CC2(F)F)no1 64470,c1(CCN=C(NCC2NC(=O)OC2)NCC2CCCO2)ccc2c(c1)COC2 64471,C12(NC(CSCC=C)=O)CC3CCC(C1C2)N3C(=O)C(C(C)(C)C)NC(C)=O 64472,c1(C(=O)NC(CNC(c2ccc(OCC)nc2)=O)(C)C)[nH]nc([N+](=O)[O-])c1Cl 64473,C1(C(=O)NCC(=C)C(F)(F)F)CC2CC1CN(C(=O)C(C)(C(C)C)OC)C2 64474,Cc1ccc(OCCC(=O)NC(C)CCNC(c2c(C)cnn2C)=O)c(C)c1 64475,c1(-n2cc(NC(C(=O)NC(CCC=C)C(=O)O)=O)nn2)ccc2nonc2c1 64476,c1(CC(=O)NCC(C)CNC(=O)COc2cccc(F)c2F)c(F)cccc1Cl 64477,c1(CNC(c2c(CC)cc[nH]2)=O)cccc(C(=O)NCC(Cl)Cl)n1 64478,c1(C(N(CC2CCCN(C(CCCOC)=O)C2)CC)=O)cc(Cl)cnc1C 64479,c1(OC)ccc(NC(C2CC3CC3N2C(c2cnc(O)[nH]2)=O)=O)cc1F 64480,c1(C(=O)NC(C(=O)NC(C(C)O)CO)Cn2cncn2)ccccc1F 64481,Cc1ncnc(O)c1C(=O)NC1CCN(C(=O)C(n2cc(Cl)cn2)C)C1C 64482,C1(NC(C2C(C#C)C2)=O)CCCCCN(C(=O)COc2cccc(CC)c2)C1 64483,C1(C(N(CCCNC(CCCN(CCCC)CCCC)=O)C)=O)CC12CCOC2 64484,C12(C(=O)NC3C(C)CCN(C(c4c(C)nc[nH]4)=O)C3)CCC(CC1)C(C)O2 64485,C=CCC(C(=O)NC(C)CN(C(=O)CC(C)O)C)NC(C)=O 64486,c1(-c2c(OC)cc(OCC)cc2)cnc2c(C(=O)Nc3ncc(F)s3)cccn12 64487,n1(C(C)C)cc(C(N2CC(CNC(=O)C(C)(C)C(C)C)C3(CC3)C2)=O)ccc1=O 64488,C(=O)(C(C)(C)CC(C)(C)C)N1CCC(CC(N2C(C)CCCC2)=O)C1 64489,N1(C(C2C(=O)NCC2)=O)CC(NC(=O)C(C2CC2)C2CC2)CC12CCCCCC2 64490,c1(C(=O)NC(C(C)NC(CCOCC#C)=O)CO)c(Cl)cccc1Br 64491,C(CCC(=O)N(CC(C)CNC(c1csnc1C)=O)C)NC(=O)OCC 64492,C=CC(C)(CC)C(=O)N1CC(OC)C(NC(=O)C(F)(F)c2cscn2)C1 64493,O=C(CS(=O)(=O)N1CCCCC1)NCCC1CCCCN1C(C1CC=CC1)=O 64494,c1(C(=O)NC2CN(C(c3c(OC)nn(C)c3)=O)C3C2C3)cn(C)c(=O)cn1 64495,C(CCC1CCC1)(C(=O)N(CC(O)CO)CCO)SC.N12CC(C1)NC2=O 64496,Cc1cc(O)c(F)cc1C(N1CCOC(c2cn(CC3(O)CCC3)nn2)C1)=O 64497,C1(C)(C(=O)NCC(CC(=O)N(CCNC(C(C)C)=O)C)C)CCC(=O)NC1 64498,c1(C(N(C2CCN(CC3CCOCC3)CC2)CC#C)=O)csc2c1CCCC2 64499,C(=O)(N=c1ccc(Cl)n[nH]1)c1ccc(NC(C(CCC)(C)C)=O)cc1OC 64500,C#CCCCCC(=O)N1CC2CC2C1C(=O)NC1C2CCCCCC12 64501,C1(NC(CC(CCC)C)=O)COC2(C1)CN(C(c1cc(OC)ncc1Cl)=O)C2 64502,C1(NC(C=COCC)=O)CN(C(=O)C=CI)CC2(CCOCC2)C1 64503,C1(NC(C(C)C)=O)CN(C(=O)C(F)C2CCC2)C2(CCOCC2)C1 64504,CC1(C)NC(=O)N(CC(N2CC3(CC(NC(=O)C(F)C4CCC4)CO3)C2)=O)C1=O 64505,c1(C(=O)OC)cc2cc(CN(C3(C)COC3)C)ccc2o1 64506,CCC(C)CC(=O)C(=O)N1C(C(N2CCC(N3CC(O)C3)C2)=O)CC2CCCC12 64507,C1(C)(C(=O)NCCN(C(c2nnc(S)n2C)=O)CC)CC2(CCC2)C1 64508,CCC(C(=O)N1CCCC1C(C)(C)NC(c1ccc[nH]1)=O)N(C)C 64509,N1(C(N2CC(CNC(C3(OC)CCC3)=O)C2)=O)CCOC(CC2CCCC2)C1 64510,CN1CCN(C(C2CCC(O)C(C)(C)O2)=O)c2cc(-c3cccc(O)c3)ccc21 64511,c1(OCCC(=O)N(C)CCNC(c2coc(O)n2)=O)ccccc1Br 64512,C(C(CC)NC(=O)CCc1cc[nH]n1)N(C(C=CCOCCOC)=O)C 64513,C1(C)(C(N(CC(C)CNC(=O)CC(C)(C)F)C)=O)Cc2ccccc2C1 64514,c1(NC(c2n(C(CC)C)nnn2)CC2CCC2)cnc(C2CCC2)nc1 64515,C1(C(=O)NC(C(=O)N(CCCCO)C)CC2CCCC2)CCC2(CC1)CC2 64516,C1(NC(c2cc(S(=O)(=O)NC)oc2)=O)CC2(CCCCN2C(=O)C(C)CO)C1 64517,Cc1cc(C)c(C(=O)NCC(C)N(C(=O)C(C2CCOCC2)O)C)c(O)n1 64518,Cc1cnc2ccccc2c1C(=O)NC1CC1NC(=O)Cc1ccno1 64519,C1(CNC(C(C)(C)SC)=O)CN(C(=O)COc2cc(Cl)ccc2C)CC12CC2 64520,c1(-n2c(C3c4cc(on4)CN3)nnn2)cccc(OC)c1.C(C)(C(N)=O)SC 64521,C1(NC(CC2CC(C)(C)C2)=O)CN(C(C2(CC(F)(F)F)CC2)=O)CCC1(C)C 64522,N1(C(C(C)(F)F)=O)CC2CCC(CNC(C3C=CCC3)=O)C2C1 64523,C(=O)(C1CCc2ccccc21)NCC1(N(C(C2CC(C)C2)=O)C2CC2)CCC1 64524,CC1CCCCN1CCc1ccccc1NC(=O)NCc1cn(C(C)(C)C)nn1 64525,N1(C(c2ccc(OCC)cc2)=O)CCCC12CN(C(=O)C(n1cc(C)cn1)C)C2 64526,C1(C(N2C(C)C(NC(c3ncnn3C)=O)CCC2)=O)CCc2nncn2C1 64527,c1(OC)cccc2sc(C(=O)N(CCCCN(C(=O)CN(C)CCO)C)C)cc12 64528,c1(CC(=O)N(C2CCCN(C(C=CCC)=O)C2)CCO)c(Cl)cccc1Cl 64529,CCCC(C(=O)N1C2CCC1CN(C(c1nncn1CC)=O)C2)C(C)C 64530,c1(CC)ccc(C(=O)NC2CCC2C(N2CCOCC2c2ccccc2)=O)nc1 64531,CCCC(C)N=c1[nH]c(=NCc2nocc2C(C)(C)C)[nH]c2c1CCC2 64532,CC(C)(O)CCC(=O)NCCCCC(=O)NC1CC1 64533,N1(C(c2csc(C)c2C)=O)CC2CCN(C(c3cc(Br)c(Cl)cc3F)=O)C2C1 64534,CC1C(NC(c2cnn(C)c2N)=O)CCCN1C(=O)CNS(N)(=O)=O 64535,c1(C(=O)NC(C(=O)NC(COCC)C(C)C)c2ccoc2)cnc(O)c(F)c1 64536,Cc1cc(-c2cnc(NC(c3sccc3Cl)=O)c(O)c2)cc(O)c1F 64537,c1(CC)ccccc1OCCC(=O)NC1CCCN(C(=O)Cn2cc(C)cn2)C1 64538,Cc1ncncc1C(=O)NC1CCCC1C(=O)NCC1(CO)CC1(C)C 64539,C1(NC(C(C)SC)=O)CCOC12CCN(C(c1cc(Cl)c(F)cc1N)=O)CC2 64540,C(=O)(N=c1c(C)c[nH]cc1Br)c1cccc(NC(C2(CC=C)CC=CC2)=O)c1 64541,N1(C(CC2(C)CCCC2)=O)CC(NC(c2coc(Cl)n2)=O)CC(O)C1 64542,C1(NC(CSCCC)=O)CC(C)CN(C(=O)C(O)C(C)CC)C1 64543,Cc1ccc(CC(=O)NC2CN(Cc3ccon3)CCC2C)c(C)c1 64544,C12(CCNC(c3n[nH]cc3Cl)=O)CCC1CN(C(c1ccsc1Cl)=O)C2 64545,c1(C(N2CCC=C(F)C2)C(=O)NCCC#N)ccc2cccnc2n1 64546,c1(C(C)=O)ccc(C(=O)NC(C)C(C)NC(=O)C(CN(C)C)C(C)C)cc1C 64547,Cc1cnc(C(=O)NC2CCC(NC(=O)CCc3cn(C)nn3)C2)nc1 64548,c1(C(=O)NCc2c(C)n[nH]c2C)cc2ncccc2[nH]1 64549,N1(Cc2c(C)noc2)CCC(C2CCCN(C(c3coc(S(N)(=O)=O)c3)=O)C2)C1 64550,S(=O)(=O)(c1csc2ccccc12)N1C2CN(C(CCCN(C)C)=O)C(CC2)C1 64551,c1(C2(C(=O)O)CC2)ncc(C2CC(CNC(=O)OC(C)(C)C)C2)cn1 64552,C1(C#N)(NC(=O)NCc2c(F)cc(C)c(Cl)n2)CC2CCC(C2)C1 64553,C(=O)(CC(C(F)(F)F)N(C)C1CC1)N(C1CN(C(=O)CN2CC=CC2)CC12CC2)C 64554,Cc1ccc(NC(C2CN(C(=O)OC(C)(C)C)CC2(F)F)=O)c(C)c1 64555,Cn1ccc2cc(N3CCN(C(=O)CC4CCCNCC4)CC3)ccc12 64556,c1(NC(C2N(C(c3ccc(OC)c(Br)c3)=O)CC2)=O)cc(Cl)cc(Cl)c1O 64557,N1(c2n(CCOCC=C)c(CC(O)CF)nn2)CCc2ncnc(O)c2CC1 64558,C1(C(=O)NCC2N(C(C3=NOC(C(C)(C)C)C3)=O)CC2)CCC2(CCC2)CO1 64559,c1(C(=O)NCC(C)(C)NC(=O)Cc2ccc(Br)cn2)ncncc1Cl 64560,C1(NC(CC(=C=C)C)=O)CC2CN(C(C3CC(N(C)C)C3)=O)CC2C1 64561,C1(NC(CC2(C=C)CC2)=O)CC2CC1N(C(C1(CC)CC(C)(C)C1)=O)C2 64562,c1(CC)cc(C(=O)NC2CC(C)(NC(=O)CC3(NC(C)=O)CCC3)C2)c(C)nn1 64563,C(=O)(CC(C)CC(=O)OC)NC(CCC)C(=O)N1CC(C(C)CC)C1 64564,C1(C(=O)NC(C)CN(C)C(c2ncoc2C2CCCCC2)=O)C2CC3C(C2)C13 64565,N1(CCC(C)O)CCCN(C(=O)CCCCCc2nn[nH]n2)CC1 64566,c1(C(=O)OC)cncc(C(N2CC(F)CC2CNC(=O)CCC=C(C)C)=O)c1 64567,CCC(C(=O)NCC1(CCNC(c2sc(C)nc2C)=O)CC1)C(C)C 64568,C#CCCCCCCC(=O)N(CC(=O)N(C1CCOC(C)(C)C1)C)C(C)C 64569,N1(C(CC=C)=O)CCC2C(NC(c3cc(Cl)cnc3OC)=O)C2CC1 64570,c1(C(=O)NCCCCC(CO)NC(CSCC)=O)cnc2ccccc2c1 64571,c1(C(N2CCN(C(CS(=O)(=O)NCC)=O)C(C)C2)=O)cc(Cl)cc(C)c1N 64572,c1(C(N2CCCC(NC(CNC(CC)=O)=O)(CO)C2)=O)cc2c(C)cccn2c1 64573,C(=O)(CC(C)CC(C)(C)C)NCc1c(C)c(Br)ccc1 64574,C1(C)(C(=O)OC)CCCN1C(=O)CCc1ccccc1OCCN1CCOC1=O 64575,C=C1CCN(C(c2nocc2CC)=O)C(C(N2CCCC(O)C2C)=O)C1 64576,C(=O)(CC(F)(F)C(F)F)N(C1CCCN(C(c2cn(CCOC)nc2C)=O)C1)C 64577,N1(C(C2C(NC(CCCC3C(C)C3)=O)COC2)=O)CCCC(C2CCC2)C1 64578,Cn1cc(N)c(-c2nc(CS(C)(=O)=O)nn2-c2ccccc2OC(F)(F)F)n1 64579,c1(OC)ccc2c(c1)OCC(C(=O)NCCC1(NC(=O)C(F)C(F)(F)F)CC1)C2 64580,Cc1ccc(Br)c(NC(c2nc(-c3cnn(CCCO)c3)cs2)=O)n1 64581,C1(NC(c2cnc(Cl)[nH]2)=O)CCN(C(=O)CSCc2ccccc2)CC1 64582,C1(F)(C(=O)OC)CCCN(C(=O)NCC(c2ccc(O)cc2)O)C1 64583,c1(C(C)C)cc(C(N2CCC(CNC(c3ccnc(Cl)c3N)=O)C2)=O)cc(O)n1 64584,c1(OC)ccc(Cl)cc1C(=O)N(C)CCOCCCN(C(=O)C(C)C(C)C)C 64585,c1(NC)c(NC(C2(CCNC(C3CCCC(=O)N3C)=O)CC2)=O)cccc1F 64586,N1(Cc2cc(C)ncn2)CC(NC(=O)CCn2cccn2)CCC1C 64587,N#Cc1ccnc(N2CCN(C(=O)Nc3ccccc3N3CCCCC3=O)CC2)c1 64588,C(=O)(CC(CC)SC)NCC(C)N(C(C=CC)=O)CCC 64589,Cc1ccc(C=CC(=O)NC2(C)CCN(C(c3cc(C(C)(F)F)on3)=O)C2)nc1 64590,N1(C(c2cnc(CNC(=O)OC(C)(C)C)s2)=O)CCc2c(C(=O)O)cccc21 64591,c1(-c2c(C(F)(F)F)cn(C)n2)ncc2c(n1)C1CCC2C1 64592,C(=O)(C1=CCOCC1)NC1(C(N2CC(COC)C2)=O)CC(F)(F)C1 64593,N1(C(c2cc(CC(C)C)on2)=O)CC(CNC(c2nsnc2O)=O)CC1(C)C 64594,Cn1c(=O)n(C)c2cc(S(=O)(=O)NC(c3cccc(Br)c3)C3CCCO3)cnc12 64595,N1(C(CC(CC)C)=O)CC(C2CCCCN(C(c3cccc4ncoc34)=O)C2)C1 64596,CC1CC(C#N)CN1C(C12CC(c3nc(CC4CC5C(C4)C5(F)F)no3)(C1)C2)=O 64597,N1(C(c2c(COC)scc2)=O)CCCC12CCC(NC(=O)C(C)(C)C(C)C)CC2 64598,c1(C(=O)NC(C(C)(C)NC(c2nc(OC)oc2)=O)C)cncc(Cl)c1Cl 64599,C1(C(N(C2CCCC2)CC#C)=O)COC2(C1)CN(C(=O)C=CCO)C2 64600,C(CC(F)(F)F)N(C(=O)CC(C)NC(NOCCC#CC)=O)C1CCCC1 64601,C1(N(C(c2ccc(CC)s2)=O)CC)CCCN(C(=O)CCc2ccccn2)C1 64602,N1(C(C=C(C)C2CC2)=O)CCC2(CC1)CCN(C(c1c(C)cc(Cl)cc1N)=O)C2 64603,C1(C(=O)NCC2C(NC(c3c(CC)nco3)=O)CC2)CCCCN1N=O 64604,C(c1ccc(Cl)s1)=CC(=O)NCC(CN(C(=O)COCCCF)C1CC1)CO 64605,c1(CN(CCNc2ccc[n+]([O-])c2)CC)cccc2c[nH]nc12 64606,C1(NC(c2ccncc2F)=O)COC2CN(C(c3nccc4n[nH]cc34)=O)CC12 64607,c1(OC)ccccc1C(C)(C)C(=O)NCC1C=CCN1C(c1cc(Cl)cs1)=O 64608,CN1CCC(=CC(N2CC(NC(c3ncccc3C(F)(F)F)=O)C(O)C2)=O)CC1 64609,CC1(C)CC(C(=O)N2CCC(NC(c3ccc(C(F)(F)F)nn3)=O)C2)=NO1 64610,c1(N2CC(CO)C(CO)C2)nc2c(c(=NCC#CC3CC3)[nH]1)CCC2 64611,C1(c2nnnn2CCCSCC)(NC(CCCCC=C)C)CC2(CCCC2)C1 64612,Cc1nc(CCC(=O)NC2CCN(C(=O)CNC(C3CCC(=O)N3)=O)C2)[nH]c1C 64613,Cc1cc(Cl)cc(C)c1CN(CC(=O)NC1CCCCC1)CCC#N 64614,CCS(=O)CC(=O)NCC(N1CCN(C(C2(Br)CC2)=O)CC1)C 64615,N1(CC(=O)NC(CCCN(C(=O)C(C)(C)C)CCO)C)CCN(C(C)=O)CC1 64616,c1(CC)noc(CCCC(=O)NCCN(C(=O)CC#N)CC)n1 64617,CC1(C=CC(=O)NCC2CN(C(C3(CO)CCCO3)=O)CC2(F)F)CCOCC1 64618,CCCC(C(=O)N(C)CCOCCNC(c1cncc(OC)n1)=O)S(N)(=O)=O 64619,C(=O)(C(C1CC1)N(C(=O)CC1CCOC1)C)NCC(C1CCCC1)C 64620,N1(C(c2c(Cl)cn(CCC)n2)=O)CCCN(C(=O)CCOC(C)C)CC1C(C)C 64621,C(C1=CCN(C(=O)CN2CCC(O)CC2)CC1)NC(C(C(C)C)NC(C)=O)=O 64622,N1(C(C(CC)C)=O)CCCC(C)(NC(=O)CCc2cccnc2Cl)C1 64623,N1(S(CC)(=O)=O)CCc2cc(C(=O)NCc3ccccc3CO)ccc2C1 64624,C(=O)(CC(O)C(Cl)(Cl)Cl)NCCC(C)NC(CC(C(=C)C)O)=O 64625,C1(C(N(CC(CC)O)CC)=O)CCCCCC1NC(C1OC2CCC1C2)=O 64626,C1(C(N2CCC3C(CCN3Cc3nccnc3Cl)C2)=O)CCCC2CCCCC12 64627,c1(OC)ccc(C=CC(=O)NC2(C)CCN(C(C3C=CCCC3)=O)C2)cc1 64628,c1(C(N2CC(c3cn(CC=C)nn3)C(O)C2)=O)ccc2ccccc2n1 64629,c1(C(N2CCC(C)(NC(=O)Cc3ccns3)C2)=O)cnn2ccc(O)nc12 64630,C(=O)(C(C(C)C)C1CCC1)N(CCCNC(C1(CC)COC1)=O)C 64631,C1(C(N(C(CCNC(c2c(C)nn[nH]2)=O)C)C)=O)CN2CCCC1C2 64632,C1(N(C(=O)OC)C)CC(S(C)(=O)=NC(=O)c2cccc(CSC(C)(C)C)c2)C1 64633,CC1=C(C(=O)N2CC(NC(C3(O)CCCC3)=O)CC23CCC3)C(=O)OC1(C)C 64634,c1(C(=O)NC(CC)CNC(=O)CCNC(=O)COC)cc(C#N)[nH]c1C 64635,C(=O)(C1=CC2C=CC(C1)C2)N1CC(NC(c2n(C(C)C)ccn2)=O)C(N=[N+]=[N-])C1 64636,C12(NC(C(C)=C(C)C)=O)CCC1CN(C(=O)Cc1sc(C)nc1C)C2 64637,C(=O)(C(C)(C)C1=CCSCC1)NCC1N(C)CCN(C(c2csc(O)n2)=O)C1 64638,c1(C(=O)NCC2CCC(NC(c3c(SC)cnn3C)=O)C2)cc(C)c(O)c(N)c1 64639,Cc1nc2ncccn2c1C(N1CCC(C(=O)Nc2nccs2)CC1)=O 64640,c1(CC)cnoc1C(=O)N(CCC(C)NC(=O)Cc1cscc1Br)C 64641,c12ccc(cc1)CNC(=O)N2.C1(CCC)(OCC(F)F)CCNC1=O 64642,c1(OC)cccc(CC(=O)NCC2COCCN2Cc2cnco2)c1 64643,N1(C(CCc2onc(CSC)n2)=O)CC2CC(NC(C3(C)C=CCCC3)=O)C2C1 64644,N1(C(C(CC)NC(C2CCC(=O)N(C)C2)=O)=O)CCC12CCCSC2 64645,C(=O)(CC(C)(O)C(F)(F)F)NCCC(C)(C)NC(c1c(C)n(CC(C)C)nc1)=O 64646,N1(C(c2nnc(CC)s2)=O)CCC2(NC(c3c(Cl)n[nH]c3C)=O)CCCCCC12 64647,N1(CC(=O)NC2CCC2)CCN(Cc2cccc(Br)c2)CC1 64648,C1(CCOC)(NC(=O)C(C)c2cccs2)CCN(C(C2CN(C3CCC3)C2)=O)C1 64649,C1(NC(CCN(CC)CC)=O)CN(C(c2cc(CO)[nH]n2)=O)C2CCCC12 64650,CC1CC(C(=O)NCc2ccccc2-c2cccc(Cl)c2)C1(C)C 64651,C(=O)(CC(O)CC(C)C)N1C(C(=O)NC2(CCC)CC2)CC2(CC2)C1 64652,N1(C(c2cccc(SC)c2)=O)CC(C)CN(C(=O)C=Cc2cnc[nH]2)CC1C 64653,c1(N(CC(CN(C(C(c2ccccc2)SC)=O)C)O)C)ccc([N+](=O)[O-])c(C)c1 64654,C1(C(=O)NC2COCCN(C(=O)C3=CCCC3)C2)CCn2nnnc2C1 64655,CCCC(C)C(=O)NC(CN(C(=O)CSc1cccc(OC)c1)C)(CO)CO 64656,c1(OC)ccc(C(N2CC(OC)CC2CNC(=O)C(C)CC2CC2)=O)c(O)c1F 64657,CC(C)CC(CC(=O)O)NC(=O)Nc1cn(C2CCN(S(C)(=O)=O)CC2)nn1 64658,c1(NCC(=O)NC(CC)CNC(=O)CC2(N(C)C)CCC2)cc(C)ccc1C 64659,c1(C(=O)OC)sc(C)cc1NC(=O)C(=O)NCC1CC(C)CO1 64660,c1(C(=O)NCCN(C(=O)CSCC(N)=O)C)cc(OC)ccc1Br 64661,c1(C(N2CCC(C(C(=O)NC(n3ccnc3)C)C)CC2)=O)c(F)ccc(Cl)c1Cl 64662,c1(NC(N2CC(C)OC(C(F)(F)F)C2)=O)ncc(C#N)cc1F 64663,C1(C(=O)NCCC2CC3C=CC2C3)CC12CCN(C(C1CC(O)(CO)C1)=O)CC2 64664,O=C(C1=CC2CC(C1)CC2O)NCC1(F)CCN(C(=O)C(=Cc2c[nH]cn2)F)C1 64665,C1(C(C(=O)NC(c2ccncc2)C)(C)C)CCC(NC(=O)OC(C)(C)C)CC1.OC 64666,N1(C(C2N(Cc3c(OC)ccnc3)CCNC2)=O)CCc2cccnc2C1 64667,C1(NC(c2n(CC=C)ccc2)=O)CCC(NC(C2(C)CC=CCC2)=O)CC1 64668,C1(CC(=O)NCCOCC(=O)NCC2CCSCC2)CCCOCC1 64669,CC1CCC(C(=O)NC(C2CCN(C(=O)C3=CCOCC3)C2)(C)C)C(=O)N1 64670,c1(-c2cncc(COCC)c2)c[nH]c2ncc(C(=O)NCc3ccsc3)cc12 64671,C(=O)(CC(F)(F)F)NCC1(O)CC(NC(CCc2onc(C)n2)=O)C1 64672,C(=O)(CS(C)(=O)=O)NCC(C)(F)CNC(=O)C(C)(C)n1ccnn1 64673,CC(CCCNC(C1(Cl)CC1(F)F)=O)NC(=O)COCCCF 64674,c1(C(C)OC)nc(-c2ccnc(C)c2)n(-c2cccc(C(N)=O)c2)n1 64675,N(C1c2ccccc2CC1NC(=O)C=Cc1nccs1)C(CSCC(C)C)=O 64676,c1(C(N2CC(CNC(CC3N(C(C)=O)CCC3)=O)C2)=O)cc(F)cc([N+](=O)[O-])c1 64677,c1(C(CNC(c2ccsc2Cl)=O)NC(C2CC(C)(F)C2)=O)ccc(F)cc1 64678,N#Cc1ccc(C(=O)NC2COCC2NC(=O)CCc2ccncc2)cc1F 64679,c1(C(=O)NCC2CCN2C(c2cn(C3CC3)cn2)=O)c(F)cncc1Cl 64680,C1(=CC(=O)N(CC(CNC(CCn2c(C)ncc2)=O)(C)C)C)CCCCC1(C)C 64681,C1(CC(=O)N(CC(N2CC(N(C)C3CC3)C2)=O)C(C)C)CCC(C)C(C)C1 64682,C1(N(C(=O)CC(C)C2CC2)CC#C)CCN(C(C2CC(OC)C2)=O)CC1 64683,CCC(C)CC(C)C(=O)N1CC(CO)C2(C1)CN(C(c1cnn(C(F)F)c1)=O)C2 64684,N1(C(C2(CF)CCOCC2)=O)CCOC2(CCN(C(C34COCC3C4)=O)CC2)C1 64685,C1(C(N(C2CCC(NC(CC3C(CC)C3)=O)CC2)C)=O)CC2CCC(C1)C2=O 64686,N1(C(C=C(C)Cl)=O)CCN(CCNC(c2nn(C)nc2Br)=O)CC1 64687,c1(C(C(=O)NC)N(C)Cc2cccnc2OC)ccc(C(F)(F)C(F)(F)F)cc1 64688,c1(C(=O)NCC(C)(C)CNC(=O)COC2CCC2)cc2ccc(F)cc2nc1O 64689,c1(NC(CC2C(NC(COC(CC)C)=O)CC2O)=O)ccc2c(c1)CCO2 64690,c1(C(=O)NCC2C(NC(=O)CCC3CCOC3)CC2)cc(F)cc2nn[nH]c12 64691,n1(CC(N2CCN(C(CCCC=C)=O)CC2C(F)F)=O)ccc(=O)c([N+](=O)[O-])c1 64692,N1(C(C(=O)NC2CC(F)(CNC(C(C)n3ccnc3)=O)C2)C)CCC(O)CC1 64693,C1(OC)(CNC(C2CC3CC3C2)=O)CCN(C(C2CC2c2cncs2)=O)CC1 64694,c1(C(=O)NCC(CNC(C2NC(=O)OC2)=O)C(F)(F)F)cnc2c(c1)CCCO2 64695,C12(C(N(C3CCN(C(c4cnc(S)[nH]4)=O)C3)C)=O)CCCCC1C2Br 64696,c1(NCc2c(C)ccs2)ncccc1S(=O)(=O)NCc1c[nH]c(=N)s1 64697,C1(OC)CC(C(=O)NCC(O)CC2CCCC2)N(C(=O)CNC=O)C1 64698,CC1=CCC(NC(N2CCC2C(=O)Nc2cc(C)nn2-c2ccccc2)=O)CC1 64699,CCC(CN(C)C)CC(=O)NC1(CNC(C2CC23CCC3)=O)CCC1 64700,C(CCCCC)=CC(=O)NC(CN(C(=O)C=Cc1ccsc1)CC)C 64701,N1(C(c2ccc(C)s2)=O)CC2(CCOCC2)CC1CNC(=O)CC(C)C 64702,CCC(C)CCCC(=O)N1CC2C(NC(=O)Cc3cc(C(C)C)no3)C2C1 64703,C(=O)(C(C)CC(C)(F)F)NC(CCNC(C1(OC)CS(=O)(=O)C1)=O)C 64704,C1(N(CCOC)C(c2cn(C)nn2)=O)CCN(C(=O)C(c2cnccn2)C)CC1 64705,C1(C(=O)NCC23C(CN(C(c4cnc(C)n4C)=O)C2)C3)CCCC2(CCC2)O1 64706,C(=O)(C(O)C(C(C)C)OC)NC1CC(CCC(N2CC(COC)(OC)C2)=O)C1 64707,C(CO)(CCCCNC(c1cc[n+]([O-])cc1)=O)NC(c1c(CC=C)cccc1)=O 64708,C1(CCC#C)CCCN(C(=O)C(C2CN(C(=O)C(C)OCCCC)C2)OC)C1 64709,C(=O)(C1=C(C)C(C)(C)OC1=O)NCC(C(=O)OCC)(C)CC 64710,c1(OC)cnc(C(=O)NC2CCC(NC(=O)CC3CCC(C)(C)C3)C2)cn1 64711,c1(C(C(=O)NC2(CNC(C=CCC)=O)CCOC2)O)ccc(Cl)cc1Cl 64712,CCC(C)C(O)C(=O)N(C(C)CCNC(c1cc(-c2cccc(Cl)c2)ns1)=O)C 64713,N1(C(C(CSC)O)=O)CCC(C)(CNC(c2ccc(C)n2C)=O)C1 64714,C1(NC(c2c(COC)ncs2)=O)COC2(C1)CN(C(=O)C(C)C(C)COC)C2 64715,C(=O)(C(C(C)CC)N(C)C(c1coc(CCC)n1)=O)N(CCOCC=C)C 64716,c1(C(N2CC=CC(NC(C(CC)(C)COC)=O)C2)=O)sc2ncccc2c1N 64717,CCC(CNC(=O)C=NOC)(CC)C(=O)NC1CCNC(=O)CC1 64718,CC1(C)CC(CNC(c2cc(Cl)ccc2F)=O)CN(C(=O)C(C)(C)C#N)C1 64719,N1(C(C2(CC)CC2)=O)CC2(C1)CN(C(=O)Cc1nc(C3CC3)oc1C)CC2CO 64720,CC1CCCC=C1C(=O)NCCC1CCN(C(=O)CN(CC(C)(C)C)C)CC1 64721,c1(C(=O)NC(C)(CNC(C2(C(F)F)CC2)=O)C2CCC2)csc(O)n1 64722,c1(CCCC(=O)NCC(CC)NC(=O)C=Cc2cnn(C)c2)cccc(Cl)c1 64723,C1(NC(COCCCC)=O)CCC12CCN(C(=O)C(=O)Nc1cccc(C)c1)CC2 64724,c1(C(=O)NCC2CC2NC(c2csnn2)=O)cnc2ccccc2c1 64725,c1(OCCN(C(=O)CNC(c2nn[nH]n2)C2CC2)CC)cccc(F)c1 64726,CC1OCCN(C(C2CN(C(=O)C=CC3CCC3)CCN2C)=O)C1CO 64727,O=C(CCc1cccc(OCC(F)(F)F)c1)N=c1[nH]n(C2CC2)c2ccccc12 64728,C#CC1(O)CC(C(N2CCCC2CN(C(=O)C(c2ccncc2C)C)C)=O)C1 64729,C(=O)(C1=C(Cl)CCCC1)N1CC(C)CC(C(N(C)Cc2nc(C)on2)=O)C1 64730,C1(C(N2C(C)CN(C(=O)CCc3cccs3)CC2)=O)CCN2CCOCC12 64731,C(=O)(CC(C(C)C)OCC)NC1(C)CN(C(c2cc(CCC)c(C)s2)=O)C1 64732,CC(C(=O)N1CC(O)CC1CNC(=O)CC1CCC=CCC1)C(F)(F)F 64733,c1(C(=O)NC(C2CCCN2C(=O)CN(C)C(N)=O)C)cc2ccc(Cl)c(F)c2[nH]1 64734,C(C(=O)NC(C)C(CO)NC(C1CCN(C(=O)CC)C1)=O)(C(C)C)NC(C)=O 64735,C1(C)(NC(C2C(C)CCC2)=O)CCN(C(C2(c3ccccc3Br)CC2)=O)CC1 64736,C(C)(CO)(C(=O)N1CCC(OCCNC(=O)CNC=O)C1)OC 64737,C1(NC(=O)C(c2ccccc2)O)CC2CC1CN(C(C1(F)CCCC1)=O)C2 64738,C1(C)(CNC(CCNC(COC)=O)=O)CN(C(c2ccnc(C3CC3)n2)=O)CC1C 64739,n1(CC(N2CC(OC)C(NC(=O)C=C(C)C(C)C)C2)=O)ccc(=O)cc1C 64740,c1(CCC(=O)NC(CC)(C)CNC(C2(CF)CC2(F)F)=O)cccc(Cl)c1 64741,C1(NC(C(CSC)OC)=O)CCN(C(c2cc(-c3ccco3)on2)=O)C12CCC2 64742,N1(C(c2c(CNC(C3CC(=O)NCC3)=O)ocn2)=O)CC2COCC(C2)C1 64743,Cc1c(C(=O)OCC2(C(C)C)OCCO2)noc1C1CC1 64744,NS(=O)(=O)CCCCCCC(=O)NCC1CC1NC(c1cc(O)cs1)=O 64745,c1(SCNC(C(C2COC(C)C2)N(C2CC(F)(F)C2)C)=O)ccncc1Cl 64746,N1(C(CC2(OC)CCC2)=O)CCN(C(c2cnc(C(F)(F)F)s2)=O)C(C(F)F)C1 64747,c1(C(N(C2CC(NC(C3ON=C(CC)C3)=O)C2)C)=O)cc2c(Cl)cccc2s1 64748,Cc1scc(C(=O)N(CC(=O)NC(C(O)CO)C2CC2)C(C)C)c1C 64749,S(=O)(=O)(c1cccc(N2CCOCC(C(C)(C)C)C2)n1)N(CC=C)CCO 64750,N1(C(CCCOCC)=O)CCN(Cc2cn(CCOC3CCOC3)nn2)CC1 64751,Cc1n[nH]c(C)c1CC(=O)N(CC(O)CNC(=O)C(C)Sc1ccccc1)C 64752,C1(NC(CC(C)(C)NC(Cc2ccc(C)s2)=O)=O)C(O)C2CCOC12 64753,C12(C(=O)NC(CCOC)C)COC(C1)C(NC(=O)C=CC1CCCCC1)C2 64754,C1(CC(N2CC(C)CC(C)C2)=O)CCC2(CC1)CCN(C(=O)COCCO)CC2 64755,CCC(C)C(O)C(C)C(=O)NCC1CN(C(=O)CNC(=O)CC)C2CCN1C2 64756,c1(C(=O)NCC2N(C(c3cn(C)nn3)=O)CCC2)c(O)cccc1O 64757,N1(C(C(C=C)O)=O)CC(O)CC1CNC(=O)CNC(=O)NCC1CCCC1 64758,CC1CC(c2nc(-c3cc[nH]n3)nn2-c2ccc(C34CC(C3)C4)cc2)=NO1 64759,N1(C(CS(CC)(=O)=O)=O)C2CCC1C(C)C(NC(=O)C=CC=C(Cl)Cl)C2 64760,c1(C(N(C)CCOCCN(C)C(C2(Cl)CC2(F)F)=O)=O)cccn2[nH]c(=N)nc12 64761,c1(C(=O)NCCC(C(C)C)NC(C=CSC)=O)cc2cccc(F)c2o1 64762,CC1CCC(C(N2CCCCC2)=O)NC1.N12CC(CC1=O)NC(=O)N1CC2C1 64763,N1(C(=O)CCC2CC2)CCCCC1C1CCCN(CC2(O)CCC2)C1 64764,c1(C(C)NS(c2ccc(NC(=O)NCCC)s2)(=O)=O)sc2ccccc2c1C 64765,CCC(C)(CCC(C)C)C(=O)NC1CC(CCNC(c2c(Cl)ccnc2C)=O)C1 64766,c1(OCC(=O)NCC(C)N(C)C(c2ccc(N)c(N)c2)=O)ccc(F)c(F)c1 64767,N1(C(c2ccc(CNC(c3cc(OC)n[nH]3)=O)cn2)=O)CCC2C(C(N)=O)C2C1 64768,c1(C(=O)NC2CN(C(C=Cc3n(CC)ccn3)=O)CC2F)cnc2cccnn12 64769,CC1(C)CCCC(CNCC2CCCS2(=O)=O)C1 64770,CC(CCC(C)(C)C)C(=O)NC1CN(C(=O)CN2CSCC2=O)CCC1O 64771,c1(N(C)CC)ccc(-c2nc(C3CCCO3)n(-c3ccc(Br)cc3)n2)cc1 64772,c1(C(=O)OC)ccc(CNC(=O)N(C2CC2)Cc2ccco2)c([N+](=O)[O-])c1 64773,N1(C(C2COCCO2)=O)CCC2(CCCN(CC=Cc3ccccc3)C2)C1 64774,c1(COC)nc(C)c(C(=O)NCCCN(C(=O)Cc2csc(Cl)c2)CCO)s1 64775,N1(C(C2(CN(C)C)CC2)=O)CCOC2(C1)CN(C(c1ccnnc1O)=O)C2 64776,CC1CC(F)(F)CN1C(=O)C(=O)Nc1ccc(F)cc1-c1nc(C(C)(C)C)no1 64777,Cc1cnc2c(cnn2CC(=O)NC2CCCN(C(c3cccs3)=O)CC2)c1 64778,c1(CC(=O)N(CC(CNC(C2C(COC)C2)=O)O)C)cc(C)cc(F)c1 64779,c1(NC(=O)NC(CC)CNC(C2CC2C(=O)OC)=O)ccccc1C(F)(F)F 64780,c1(CCNC(N2CCC(CNC(CC)=O)C2)=O)ccc2c(c1)COC2 64781,C(c1cc(C)cc(C)c1)=CC(=O)NCCN(C(C(C(C=C)C)C)=O)CC 64782,C1(NC(c2oc(C)c(CO)c2)=O)C2CC3C1C3C2C(N1CCC(C)(CCO)C1)=O 64783,CCC(C)(CO)C(=O)N1CC(CNC(=O)CNC(=O)OC)C(F)C1 64784,C(CN=c1ccnc(N(C)Cc2cccc3ccccc23)[nH]1)C1C(C)C1 64785,c1(C(=O)NCC2C(NC(c3ncc(OC)nc3)=O)COC2)cc(C)ccc1Cl 64786,CC1(C)CC(NC(C2C(O)CCN2C(=O)CC#N)=O)C12CCC2 64787,Cc1ccc(CCC(=O)NCC2CCC2NC(=O)CCC(=O)N(C)C)cn1 64788,c1(C(N(C(CCNC(C(CC=C)N(C)C)=O)C)C)=O)ccc([N+](=O)[O-])cc1 64789,C(=O)(C1=NOCC1)N(C(CCNC(C1CC(CC)C1)=O)C)C 64790,N1(C(C2CC=CCC2)=O)CC2=C(C1)CN(C(C1(O)CC(F)(F)C1)=O)C2 64791,Cc1cc(C2CCC2)ncc1C(N1CCC(NC(C2CCC(C)(C)O2)=O)C1C)=O 64792,N1(C(COCCCC)=O)CC(NC(=O)C(C)(C)CF)C(C(F)F)C1 64793,c1(CC(N2CC(C)C(NC(c3ccn(CCF)n3)=O)C2)=O)nc2ccccc2s1 64794,C#CC(C)(C)C(=O)NCC=CCC(=O)NC1CN(C)NC1=O 64795,c1(C(=O)NCC2(O)CC(NC(C(C)OC)=O)C2)cc2c(nc1O)CCCC2 64796,c1(CC)[nH]c(C(=O)NC(C)(CNC(C2CCOC2)=O)c2cccs2)nc1Cl 64797,O=C1CC(C(=O)NCCc2ccncc2F)N(C(C2CC2Cl)=O)C1 64798,CCCCCCCNC(=O)C(C1CCCO1)NC(=O)C=C(CC)CC 64799,C1(NC(C2CCC(C(C)C)CC2)=O)CN(C(C2CC2(C)Br)=O)Cc2nccn2C1 64800,Cc1ccccc1C=CC(N1CC(C(C)NC(c2cccc(F)n2)=O)C1)=O 64801,C(CN=C(NCc1ccc(C2CC2)c(F)c1)N1CCC(C)C1C)OC 64802,C1(C(=O)NC(C(C)NC(c2cn[nH]c2)=O)C)CCc2cn(C)nc2C1 64803,C(=O)(CCCCC(N)=O)N1C(c2cn(-c3c(F)ccc(OC)c3)nn2)CCC1 64804,N1(C(C(C)C)=O)CCC(C2CCN(C(=O)C(F)C3CCC3)CC2)C1 64805,c1(C(N2CCNC(C(N3CCC(O)C(O)C3)=O)C2)=O)cc(I)ccc1F 64806,Cc1[nH]nc2c(C(N3CCC3CNC(c3ccc4cncn4c3)=O)=O)cccc12 64807,c1(C(N2CC(OC)C(NC(=O)CC3(C)CCCO3)C2)=O)cn2ccccc2n1 64808,C(CCCC(c1cn(-c2ccc(C(=O)O)nc2)nn1)NC(C1(SC)CC1)=O)OC 64809,C(=O)(CCCCCC(C)C)NCCCN(C(C=Cc1c(C)noc1C)=O)C1CC1 64810,C(=O)(C1c2ccccc2C2CC1C2)NC1CNCC(C)(C)C1 64811,C1(C(=O)OC(C)Cc2ccco2)CCN(C)C1 64812,CC1(C)CN(C(C2CCN(CCO)C(=O)C2)=O)CC1NC(=O)CCc1nc[nH]n1 64813,N1(C(c2ccc(C)o2)=O)CC(CNC(C2(C)CCCCCC2)=O)CC1(C)C 64814,c1(C(N2C(C)(C(N3CCN(C)CC3)=O)CC2)=O)cc(Cl)cc([N+](=O)[O-])c1 64815,Cc1cc(CN2CC3CC3(C(=O)Nc3cc(C(F)(F)F)c(Br)cn3)C2)ccc1Br 64816,c1(C(N(CCCCNC(CC2CCC(C)C2)=O)C)=O)cccc(F)c1Cl 64817,N1(C(c2sc(CO)nc2C(F)(F)F)=O)CC2CCCC(C1)C2O 64818,CC1CC2CC(C(=O)N(C3CN(C(=O)CCn4cccn4)C3)C)(C2)O1 64819,c1(OC)cncc(C(=O)NCCC(C)NC(=O)C(O)CCc2ccccc2)c1 64820,c1(CCC)c(C(=O)NCC2CC2CNC(=O)C=Cc2cccnc2)nnn1CC 64821,Cc1cccc(C(=O)NCCCCCNC(=O)C(c2cnn(C)c2)O)c1O 64822,N1(C(C(CC=C)CC)=O)CCCCCC(NC(c2onc(C)c2C)=O)C1 64823,Cc1ccc(C)n1CC(N1CC(O)(C(C)NC(c2cnn(C3CC3C)c2)=O)C1)=O 64824,Cc1ccc(C)c(C(N2CC(N(C(=O)C(C)NC(N)=O)C)C3(CC3)C2)=O)c1N 64825,C1(CNC(C2C(OC)CCC2)=O)(OC)CCN(C(=O)COCCSC)C1 64826,c1(C(=O)NC(CC#C)(C)C(=O)NCCCN=[N+]=[N-])ccc2cc[nH]c2n1 64827,N1(C(C(CCC#C)O)=O)C2CCC1CC(F)(CNC(c1cccc(CC)n1)=O)C2 64828,Cc1cc(C)[nH]c(=NCc2cn3ccc(-c4ccc5c(c4)OCO5)cc3n2)n1 64829,N1(C(c2n(C)cc(Cl)c2)=O)CC(NC(c2cn(C3COC3)nn2)=O)C(C2CC2)C1 64830,Cc1cc(=O)n(C)nc1C(N1CCCCC1CN(C)C(C1CC1(Cl)Cl)=O)=O 64831,C1(CN(C(=O)C(F)n2ccnc2)C)CCN(C(=O)C(F)(F)C2CC2)C1 64832,Cc1cc(Br)cc(C)c1C(=O)NC1CN(C(c2c(O)cncc2F)=O)C1 64833,Cc1ccc(O)c(C(N2CC3CC2CN3C(=O)Cc2ccc(Cl)s2)=O)c1 64834,C1(CC=C)(C(=O)NC(Cc2cnc[nH]2)CO)CCN(C(c2csnn2)=O)C1 64835,N1(C(=O)OC(C)(C)C)CCC(C(C)(C)C)CC1C(=O)OCCN1CCC1C 64836,C1(CNC(C23CC(C(=O)OC)(C2)C3)=O)(NC(=O)CC2CSCCS2)CCOCC1 64837,N1(C(c2cnc(CC)o2)=O)CCOCC1CN(C(=O)CCOCC(F)F)C 64838,C(CCCCC(=O)NC1CC(CNC(=O)CC2OCCOC2(C)C)C1)NC(C)=O 64839,C1(OCC)CC(NC(=NCCSC)NCc2ccccc2NCC)C12CCCC2 64840,CCCC(C)CC(=O)NCCC1CCN(C(c2cc(C)nc(OC)n2)=O)C1 64841,N1(C(c2cc(C(C)C)[nH]n2)=O)CC(NC(c2c(Br)cnn2C)=O)CC(C)C1 64842,Cc1cc(O)nc(C)c1C(=O)NCC(c1ccccc1)CNC(N)=O 64843,c1(CNc2c(CC(=O)NCc3ccc(F)cc3)cccc2)cnc(Cl)cc1F 64844,CC#CCC(C(=O)NCc1ccc(Cl)cn1)NC(c1cncc(NC)c1)=O 64845,C1(NC(=O)CC2CC3(CC3)C2)CCN(C(=O)CS(=O)(=O)Cc2cccs2)CC1F 64846,C(CC(C(=O)NCc1ccc(F)cc1)NC(C1C2CCC(F)C12)=O)SC 64847,C1(CC(=O)NC2C(C)CC=CC2)CCCN(C(C2(C)CCCCCC2)=O)CC1 64848,Cc1ccc(CCN=C(NCC(C)(C)C2CC2)NCC2CC2)c(O)c1.C(C)C 64849,c1(C(=O)NC(C2(O)CN(C(c3c(SC)cn(C)n3)=O)C2)C)nc2sccn2c1C 64850,c1(C(=O)NC2COCCN(C(C(C)c3ccsn3)=O)C2)cccc2cnsc12 64851,N1(C(CCSCc2nc(C)sc2)=O)CC(O)CC1CNC(=O)Cn1cnnc1O 64852,Cc1ccc(C(=O)NCC(C)NC(=O)C(C(C)C)NC(c2ccco2)=O)c(C)c1 64853,Cn1ncc2c1CN(C(C1CC3CC3N1Cc1cc(F)cnc1Cl)=O)C2 64854,C1(SC)CC(N(C(=O)CN(C)CC2CCCC2)C)C1.C12CC(C1)NC(=O)C2 64855,C1(C(=O)NC(c2ccc(F)cc2)CC)CC(O)CCN1C(c1sc(C)cc1C)=O 64856,C1(C(N(C(CCC(C)C)C)C)=O)CC1C1CN(C(C2(O)CCCOC2)=O)C1 64857,CCC(C(=O)NCCC1CCN(C(=O)CCc2ccsc2Cl)C1)SC 64858,c1(C(N2C(C)CN(C(C3(C)CC3(F)F)=O)CC2)=O)ccc2nc(CO)[nH]c2c1 64859,c1(C(N2C(C(C)(C)C(=O)NCc3ccccc3)CCC2)=O)cc2ncccc2[nH]1 64860,C1(C(N(C[Si](C)(C)C)C(C)(C)C)=O)CCCN(S(N)(=O)=O)C1 64861,CC1=C(C(=O)N(C2CCN(C(=O)CCC3CC(F)(F)C3)C2)C)CCO1 64862,N1(C(C=C(CC)CC)=O)CCC2CN(C(c3c(N)sc(C)c3C)=O)CCC2C1 64863,N1(C(C2CCCCC2n2cc(CCCCO)nn2)=O)CCC2(CCNC2=O)C1 64864,c1(CC(N2CCC(N(C)C(c3ccnc(C(F)F)c3)=O)C2)=O)cc(F)ccc1F 64865,N1(C(=O)CC=Cc2ccccc2)CCC2(CC2NC(=O)CC23CCCC2C3)C1 64866,c1(C(=O)Nc2cc(Cl)cc(F)c2F)noc2c1CCc1sccc1-2 64867,c1(C(=O)NC2C(NC(CNC(c3ccc(C)s3)=O)=O)C2)nccc(F)c1Cl 64868,C=C(F)C1(CC(N2CCSCC2C(=O)NCC#CC2CC2)=O)CCC1 64869,Cc1ncsc1COCCC(=O)NC1CCC(NC(=O)COC(C)C)C1.C1CS1 64870,N1(CCCc2c(C)ncs2)CCCC(NC(c2cc(C(C)C)nn2C)=O)C1C 64871,C(=O)(C(C)(C)C(=O)NCc1occc1C(N1CCSC2CCC12)=O)N(C)C 64872,c1(CC)sc(C(=O)NCC2CN(C(C3CC3C(F)(F)F)=O)C2)cc1Br 64873,c1(OCC)ccc([N+](=O)[O-])c(C(=O)NC2CCCC2NC(=O)Cc2cnoc2)c1 64874,C1(C(=O)NCC2(C(N)=O)CN(C(c3cc(C(C)C)on3)=O)C2)CCCC(F)C1 64875,CC(CC(=O)N1CC(F)(CF)C1)C(C)(C)NC(=O)C(c1ccccc1)F 64876,C1(CN(C(C=C(C)C(C)(C)C)=O)C)CC(F)CN1C(=O)COCC(F)F 64877,C1(C(N2CC(n3cc(CNC(c4ccccc4O)=O)nn3)C2)=O)CC1C1CCC1 64878,c1(C(c2ccccc2OC)C(=O)OCC(=O)NCC)ccc(C)cc1CC 64879,C1(CNC(C=Cc2ccc(CC)o2)=O)CC(F)(F)CN1C(=O)CC1CNC(=O)C1 64880,N1(C(CCCC(OC)OC)=O)CCCC12CCN(C(=O)C(CO)N(C)C)C2 64881,C(CC(=O)NC(C)(C)CCNC(=O)COc1ccc(Cl)c(F)c1)(C(F)(F)F)OC 64882,CCC(C)(C)C(=O)NCCN(C(=O)CCc1nc(O)n[nH]1)CC(C)O 64883,C(c1ccccn1)=C(C)C(=O)NC(C)(C)C(C)NC(c1cc(C)c(C)[nH]1)=O 64884,C1(C(N(CCN(C(=O)Cc2cn(C)nn2)CC)CC)=O)(OC)CCC(C)C1 64885,N1(C(C2(C)CC(C)C2)=O)CC(NC(c2c(C3CCC3)cnn2C)=O)CC2(CC2)C1 64886,c1(OC)n[nH]cc1C(=O)NCC(CNC(=O)Cc1ccsn1)CO 64887,c1(C(=O)NC(=O)C(C)N2CCCC2)csc(CN(CCNC(C(C)C)=O)C)c1.NC 64888,c1(COC)cccc(OC)n1.N12CC(C(CSC)C1)CNC(=O)C1(CC1)C2=O 64889,N1(C(C2C(NC(COC(C)=O)=O)CCOC2)=O)CC2(CNC(=O)N2)C1 64890,N1(c2nccc(N3CC(C)CC(C)C3)n2)CC2CCC(C1)C(=O)O2 64891,C1(C)(CNC(Cc2ncc(C)o2)=O)CCCN1C(c1csc(Cl)n1)=O 64892,C1(C(N2CCC(C(=O)NC)C2)=O)CCN(C(=O)CCC2CCCCC2)C(C)C1 64893,N1(C(c2c(C)n(C3CC3)nc2)=O)CCN(C(c2coc(C#N)c2)=O)CC1CF 64894,C(=O)(C(O)CC[S+](C)C)NCC1CC(NC(C(C)Cc2cccc(Cl)c2)=O)C1 64895,N1(C(C2C(C=C)C2)=O)CCc2c(CNC(=O)CCCc3nccs3)cccc2C1 64896,CON(CC1CCCC(C)C1)S(=O)(=O)c1ccc(F)c(F)c1F 64897,C1(CNC(C(=O)NC(c2ncco2)C)=O)(CO)CC2CC2C1 64898,C(=O)(C(C)(F)C(C)(C)F)NC1CC(CCNC(C(C(=C)C)(C)C)=O)C1 64899,C1(NC(CCOCCN(C)C)=O)CCCCCC1NC(C1CCSC1)=O 64900,Cc1ccc(-c2ccc(CN(CC(O)CO)C)cc2)cc1F 64901,C1(CN(C(C2CC(O)(CC#C)C2)=O)C)CCCCN1C(C1CCOC1C)=O 64902,c1(C(=O)NCCCCN(C(CC2C(OC)CC2)=O)C)cnn(CC(C)(C)O)c1C 64903,c1(CC)ccc(C(N2CCC(OCCNC(=O)C(C)C)C2)=O)cc1CC 64904,C1(N(C(C(C)SC)=O)C)CCC(CNC(c2sccc2Cl)=O)CC1 64905,n1(-c2scc(C)n2)c(C(N2CCN(C(=O)C(C)O)CC2C)=O)nc2ccccc12 64906,c1(CCNC(=O)NC2C(CN(C)C)CCC2)nccc(=O)n1C 64907,CC1CC=C(C(=O)N2CCC(F)(F)C(CNC(C3CCCO3)=O)C2)CC1 64908,N1(CCCN2C(C(=O)O)CCC(F)C2)C(=O)C(=O)N(Cc2ccccc2)C1=O 64909,CC1(C)CC(C)(CO)CN1C(C1CC(=O)CN1C(C1CCCC(=O)C1)=O)=O 64910,Cc1cn(C)c(C(c2nnnn2C2CCCC2)NCCCCCCN(C)C)n1 64911,C1(c2nccn2C)CCN(C(C=CSC)=O)CC1 64912,N1(c2snc(CCC)n2)CCC2CC(CNC(=O)C(=O)NCC(F)F)CCC2C1 64913,N1(C(CSCCC)=O)CC(NC(c2[nH]c(C)c(C(C)=O)c2C)=O)CC1(C)COC 64914,Cn1cc(Cl)c(C(=O)NCCc2ocnc2CNC(=O)CC2CCC3CC23)n1 64915,c1(CC(C)N(C(=O)C(=O)NC(C2(O)CCC2)CC(F)F)C)ccc(Cl)cc1 64916,Cc1ccc(NCC(CO)NC(=O)CC2CCCN(C(=O)OC(C)(C)C)C2)cc1 64917,C1(C(N(C)Cc2nc[nH]n2)=O)CCCCC1CNC(C1(C)CCN(C)C1)=O 64918,C1(C(=O)NCC(CC=C)(C)C)CCCN(C(C2CCC2(OC)OC)=O)CC1 64919,C(C)(c1cnn(C)c1)=CC(=O)NC(C(=O)OCC)Cc1ccc(OC)cc1 64920,c1(CNC(=O)NNC(=O)c2cc(I)n[nH]2)c(Br)cc(Br)c(O)c1Br 64921,CC(C(C)C(=O)NCC(O)CNC(=O)C=Cc1cccc(CO)c1)S(C)(=O)=O 64922,CC1(C(=O)NC2CC2NC(=O)CCc2nc(-c3cccs3)no2)C=CCC1 64923,c1(CC(=O)NCCC2N(C(c3c(OC)n[nH]c3)=O)CCC2)ccc(Cl)cc1F 64924,C1(C(=O)NCCCOC)CN(C(=O)CC2(O)CCOCC2)CC(C)O1 64925,C1(C(N2CCC(OCC3CC3)C2)=O)CN(C(=O)C=Cc2ccncc2)CCO1 64926,C(=O)(CC(C)CC(C)C)N1CCN(CC(C)NC(C=Cc2ccc(C)o2)=O)CC1 64927,Cc1c(C(N2CC(Oc3cccc(O)c3)C2)=O)cc(S(C)(=O)=O)cc1Br 64928,c12cc(ncn1)N1CCN(CC1)C(C)CN2C.c1(CSC)noc(C2CC2)n1 64929,c1(CC)nocc1CN(C(=O)C(=O)NCCn1cc(I)cn1)C 64930,n1(CC)cnc2nc(=NCC3CCCC(C)(C)O3)[nH]c(NCC(CO)OC)c12 64931,N1(C(C(C2CC2)OCC)=O)CCCC12CCN(C(c1c(C)cccc1O)=O)C2 64932,Cc1nc(CC(=O)N(C2CCCN(C(c3ccc(C)n3C)=O)C2)C)c(Cl)s1 64933,CC(=O)CC(C)(C)CC(=O)NCCC1CCCN(C(=O)C(F)(F)CC(C)C)C1 64934,Cc1cn2c(n1)CCC(NC(=O)NCc1ccnn1Cc1ccccc1)C2 64935,c1(C(=O)NC2CC(CNC(C(C#C)(C)C)=O)C23CCC3)cccc2sccc12 64936,c1(C(=O)NC(C=CC(=O)NC(CCC)(C)CC)C)ccc2cccnn12 64937,c1(NC2CC3(CC(C)C3)C2)nccc(=NCCCCc2cnc[nH]c2=N)[nH]1 64938,C1(NC(C(C(C)C)F)=O)CCC2(CC1)CCN(C(=O)C=C1CCOCC1)CC2 64939,N1(C(CCN(CCC)C)=O)CC(NC(c2cc(C)oc2C)=O)C2CCCCC12 64940,CC1CCC(CC(=O)NCCSCC(N2CCC(c3cnco3)C2)=O)C1 64941,c1(CC)conc1CC(=O)NCCOCCN(C)C(C1(OCC)CC(=O)C1)=O 64942,N1(C(c2c(C)n(-c3ccccn3)nc2)=O)CCCC(NC(=O)C2=CCSC2)CC1 64943,S(=O)(=O)(c1cccnc1N1CCC(OCCOC)C1)NCC1CCC(CC)CC1 64944,C1(NC(C2CC(NC(C=C(C)c3ccco3)=O)C2(C)C)=O)CC2CC1C(O)C2O 64945,O=CN1CCN(C(C2CC23CN(C(=O)CCc2ccc(Br)cc2F)C3)=O)CC1 64946,N1(C(C2C3(CCN(C(C4N(C)CC(F)C4)=O)C3)C2)=O)Cc2ccc(O)cc2C1 64947,CC(F)(F)C(C)(C)CS(=O)(=O)Nc1ccc2c(c1)NC(=O)CO2 64948,c1(C(=O)NC2C(CNC(c3cnn(CC)n3)=O)CCC2)cccc(OC)c1OC 64949,c1(C(C)=O)cc(C(=O)NC(CNC(c2cc(OC)nn2C)=O)C2CC2)oc1C 64950,c1(OCC)n[nH]c(C(N2CC(C)(C)C2c2cnn(C)c2)=O)c1Br 64951,Cc1nc(C)n(CCC(N2CCC(C(F)F)(CNC(c3c[nH]nc3C)=O)C2)=O)n1 64952,N1(C(Cn2cnc(=N)[nH]2)=O)CCCC(CNC(=O)CCc2ccc(O)nc2)CC1 64953,CC1CN(C(c2ccc(NC3CCOCC3)nc2)=O)Cc2nncn21 64954,CC1OC(C)CC1CC(=O)NC(C)CN(C(=O)CC1CCCS1(=O)=O)C 64955,c1(N(CC)CC2CCN(C(C3CC34CC4)=O)CC2)cc(C)nc(C(C)(C)C)n1 64956,Cc1ccc(C(=O)NC(C)CNC(c2cncc(C3CC3)c2)=O)c(C(C)C)n1 64957,C=CC(C)(O)CC(=O)NC1CCC(NC(=O)CS(=O)(=O)N(C)C)C1 64958,N1(C(C2(COCC)CC2)=O)C(C(=O)NCC2CC(C)C2)C2CC(O)C1C2 64959,N1(C(C(C(C)O)(C)C)=O)CC2(CC(C(N3CCOC(C#N)C3)=O)CO2)C1 64960,C1(CCNC(CC(C=C)C)=O)CCCN(C(=O)CSCc2csc(C)n2)CC1 64961,c1(C(N2CCN(C(Cc3cc(C)[nH]n3)=O)C3C2C3)=O)ccc2c(c1)C(=O)C(=O)N2 64962,N1(C(C2(OC)CCOC2)=O)C(C(=O)NCC2(O)CC3CCC2C3)C2CC(O)C1C2 64963,C1(C)(C(=O)NCc2cn(CC(=O)NCc3nc(C)sc3)nn2)CCC(C)C1 64964,Cc1cnc(C(=O)NC(CNC(c2cnc(=N)[nH]c2)=O)CO)c(F)c1 64965,c1(CNC(C(=O)N(CC(N)=O)C)=O)nc2ccc([N+](=O)[O-])cc2[nH]1 64966,N1(C(CN(C(C)C)C)=O)CCC(CNC(=O)COc2ccc(Br)cc2)C1(C)C 64967,c1(CNC2CCC(C(=O)NC(C3CCCCO3)C)C2)cc(C#N)ccn1 64968,c1(C(=O)OC)ccc2c(n1)CCCN2C(c1ccc(-c2cnnn2C)cc1)=O 64969,c1(C(=O)NCC2COC(CNC(=O)C(F)n3ccnc3)C2)ccnc2[nH]ncc12 64970,N1(C(c2cn(CC)nc2)=O)CCCOC(CCNC(C2CCCSC2)=O)C1 64971,N1(C(C(C)S(N)(=O)=O)=O)CC2(CCC(CNC(c3ccncc3C3CC3)=O)O2)C1 64972,c1(OC)c(Br)ccc(F)c1CN1CCC=C(C(=O)Nc2cnc(Cl)c(Br)c2)C1 64973,N1(C(c2ccc(C(C)=O)cn2)=O)CCC2(NC(=O)CC3CC3(C)C)CCCC12 64974,C(=O)(C(CO)C(C)(C)C)N1CCN(CCN(C(c2c(COC)cco2)=O)C)CC1 64975,O=C(C#CC1CCOC1)NCC1CC2CCC1N(C(=O)CC1CCOC1)C2 64976,c1(NC(c2n(C(CC)(C)C)nnn2)(C)C(C)OC)ccc2nncn2c1 64977,C(=O)(C#CC1CCCOC1)NC1CC(CNC(C2(SC)CC2)=O)OCC1 64978,c1(SC)cc(C(=O)NCCC(C)NC(=O)C(C)NC(c2cccs2)=O)ccc1F 64979,CC(CC(=O)N(C1(C(N2CCOC(C#N)C2)=O)CC1)C)C(F)F 64980,C(C)(CO)(CC(C)C)NC(c1c(CCNC(c2c(C)cccc2)=O)n[nH]c1)=O 64981,c1(NC2CC(OCC)C2)nccc(=NC(CC)CC#N)[nH]1 64982,C#CC1CN(C(=O)C(C)C2CCOC2)CCN1C(=O)CNC(=O)NC 64983,c1(C(N2CC(O)(CNC(C(C)SCc3ccccc3)=O)C2)=O)nc(=O)n(C)[nH]1 64984,c1(C(=O)NC2(C)CCN(C(CN(CC)CC)=O)C2)ccc2cc(C#N)ccc2c1 64985,CC(C(=O)N1CC(NC(=O)CC2CCCCCC2)C2(CC2)C1)C(C)(F)F 64986,c1(C(C(=O)NC)N(C)CC2(CC)CCC2)cccc(N2CCOC2=O)c1 64987,S(=O)(=O)(c1cccnc1NC(C)CCS(C)(=O)=O)NCC1(CC)CCC1 64988,N1(C(CC2CCC(=O)CC2)=O)CC2(CCC2)CC1CNC(C1CCS(=O)(=O)N1)=O 64989,CC(C)CCCC(=O)N1CCC(O)(CCNC(C2(O)CC2)=O)CC1 64990,c1(C(=O)NCC2(O)CN(C(C3C4C5CCC(C5)C34)=O)C2)cccc2c1CCCN2 64991,C#CCCCC(C)C(=O)NC1CC(CNC(=O)COc2ccc(F)cn2)C1 64992,c1(C(N(CCCNC(=O)CC(O)C2CC2)C(C)C)=O)ncccc1OC(F)F 64993,CC1(C)CC(CNC(=O)CN2C(=O)CNC2=O)CN1C(C1CCC1C#N)=O 64994,N1(C(C(C)(C)F)=O)CC2(CCN(C(c3cc(C(C)(C)C)ccc3N)=O)C2)C1 64995,C(=O)(CCN(OC)C(=O)C1CCc2nccn21)NCC(N(OC)C)=O 64996,CC1CCCC1C(=O)NCC1(Cn2cc(-c3nccn3C)nn2)CC1 64997,c1(C(=O)NC2(CO)CCN(C(C(C)=CC3CC3)=O)C2)nccc2ccsc12 64998,C#CCC(CC(=O)N1CCC(C)=C(C)C1)NC(C1(CCC)CC(=O)C1)=O 64999,C1(CCNC(CCN(CC)CC)=O)CCCN1C(=O)CSC1CC1 65000,C=CCCC(C(=O)NCC(O)CC(C)C)NC(c1cccnc1O)=O 65001,C1(F)(C(=O)NCC(C)(C)CNC(C2(c3ccccc3F)CCC2)=O)CCCOC1 65002,c1(C(=O)NC(CC=C)CNC(=O)Cc2cncn2C)cccnc1C(F)F 65003,N=c1[nH]c2cc(C(=O)NCC3C4CN(C(=O)CCc5cc[nH]n5)CC34)ccc2o1 65004,c1(OCCC(=O)NCC(C)NC(c2sc(F)cc2Cl)=O)c(F)cccc1Cl 65005,c1(NC(N(C2CCN(CCOC)C2)C)=O)csc2c1CCCC2 65006,C(C1=CCCCC1)(c1nnnn1CCCCCC)NCC(CC#C)(C)C 65007,c1(OCC(=O)NC2CC(C)(NC(c3ccn(C(C)(C)C)n3)=O)C2)cccc(F)c1 65008,CC1(NC(c2ccc(C3CC3)s2)=O)CCN(C(C2(C)CCOC2)=O)C1 65009,C1(NC(C(COC)N(C)C)=O)CC(F)CN(C(c2c(C3CCC3)cnn2C)=O)C1 65010,Cc1n[nH]c(C)c1CCCNC(=O)NC(c1ccc(F)cc1)C1CCOC1 65011,c1(C(C(=O)OC)OC(=O)CC(c2ccc(F)cc2)O)ccc(Br)cc1[N+](=O)[O-] 65012,C(CCN=c1[nH]c(=N)[nH]c(=NC2CCOC2C)[nH]1)(C1CCCC1)OCC 65013,c1(C(N2CC(NC(C3(C(N)=O)CC3)=O)C(F)C2)=O)cc(Cl)c(F)c(Cl)c1 65014,CC1CCN(C(c2cc(C(F)(F)F)on2)=O)CC1N(C(=O)CCC1OCCO1)C 65015,C(C(=O)N1CCC(CCNC(C2(CO)CCC2)=O)CC1)(C(C)C)OCC 65016,c1(CC(=O)NC2C(CNC(Cn3c(C)ncc3)=O)CC2)nc2c([nH]1)CCCC2 65017,C1(C(=O)NCCC(Cc2ccccc2)NC(=O)CNS(N)(=O)=O)C(CC)C1(F)F 65018,C1(C2CCCN(C(=O)C(C)C#N)C2)(NC(c2ccn(C(C)C)c(=O)c2)=O)CC1 65019,C(CN1C(=O)Cc2ccccc21)NC(c1cn(C)nn1)c1nnnn1C(C)(C)C 65020,C1(NC(C2CC(=O)N2)=O)CN(C(c2cnn(-c3ccc(F)cc3)c2)=O)CC1F 65021,Cc1oc(C)c(C(=O)N(C)CC2CCN(C(=O)Cc3nnc(O)s3)C2)c1C 65022,c1(NCC2C(NC(c3scc(C)c3Cl)=O)CCCC2)ncnc2c1cnn2C 65023,C1(CNC(c2c(CC)nc(C)[nH]2)=O)CC2(C1)CN(C(=O)Cn1nc(C)cc1C)C2 65024,C=CCN=C(NCC(=O)NCc1ccccc1)N1CN(C)C(=O)C1C 65025,N1(C(C=CCOC)=O)CCC(C2OCCC2NC(=O)Cn2ccnc2C)CC1 65026,CCC(C(O)C(C)C)NC(=O)NCC(c1ccc(Br)cc1)(C)C 65027,C1(O)(C(C)NC(CSCCCC)=O)CCN(C(=O)Cc2ccc(C(=O)OC)cc2)C1 65028,c1(C(N(CCN(C(C(C)OC(C)(C)C)=O)C)C(C)C)=O)ccc(Br)cc1 65029,C#CCC(CC(=O)NC1CCCC(CO)C1)NC(=O)C(F)(F)CC 65030,C=CCCCC(=O)N1CC2C(NC(c3c[nH]cc3C(C)(C)C)=O)C2C1 65031,N1(C(C(CC)n2cncn2)=O)CCCCC1CCCNC(c1c[nH]c(C#N)c1)=O 65032,C1(OC)CCC12CC(C(N1CCC(C(C)NC(=O)C3=COCCC3)CC1)=O)C2 65033,CN1CC(C(=O)NCC2CCC(C(=O)NCCOc3ccccc3)CC2)CC1=O 65034,c1(COC)nn(C)cc1C(=O)N(C1CCC(=O)N1)C 65035,CCC(C)C(C(=O)NCC1=CCN(C(c2ccc(NC)cc2Cl)=O)CC1)OC 65036,C1(C(=O)NC2CC(C)N2C(=O)C(C)(C)C(=O)N(C)C)CN(C)CC1(F)F 65037,c1(COC)cccc(CNC(=O)CC2CCN2C(c2ocnc2C)=O)c1 65038,c1(OC(=O)Cc2ccc(C(C)C)cc2)ccc(CN(C)CC)cc1C 65039,N1(C(C2(OC)CCC2)=O)CCOC(CCNC(C23CCCC2(C(N)=O)C3)=O)C1 65040,c1(C(N2CCN(C(c3c(C)ncc(C)c3)=O)CC2C)=O)cc(C)ccc1[N+](=O)[O-] 65041,c1(C(=O)NCCC(=C)CNC(c2c(C)nn(C)c2C)=O)sccc1S(=O)(=O)NC 65042,N1(C(C2C(C)C2)=O)CCCC(C)(CNC(=O)CCOc2ccccc2Br)C1 65043,n1(CC(=O)NCC(COC)NC(=O)Cc2cn(C)nc2C)cccc(C)c1=O 65044,C=CCC(CC)C(=O)NCCC1CC(NC(=O)Cc2cccc(NC(N)=O)c2)C1 65045,C(=O)(CCC(C)NC(C1(C#N)CC=CC1)=O)NCC(CSC)OC 65046,C1(c2ccc(F)cc2)(C(=O)NC(CC)CNC(=O)CSC2CC2)CCOCC1 65047,CCC1c2cc(Cl)cc(Cl)c2CCN1Cc1cnc(-c2ccccc2)o1 65048,C(CNC(=O)CCc1nc[nH]n1)(C(=O)N(C)C(C1(C)CC1)C)OC 65049,CC1(CNC(c2cc(CC(C)(C)C)on2)=O)CCN(C(C2CCCCS2)=O)C1 65050,C(C(C(=O)NC(C)CC(C)C)NC(=O)Cn1cc(C)cn1)OCC 65051,c1(CCC(=O)NC2C(C)(CC)C2)nc(C(C)OC)no1 65052,C1(CC)(CO)CCN(C(C2(C)CCCN2C(c2nccnc2N)=O)=O)CC1 65053,CC1Cc2ccccc2N1Cc1ccc(NC(=O)N(C)C(C)C)cc1 65054,CC(C)C(O)CC(=O)N1CCN(C)C(C(=O)NCC2(O)CCSC2)C1 65055,c1(CNC(CN(C(C)=O)C)=O)cnn(C)c1C(=O)NCCC1CCCC(C)C1 65056,N1(C(c2c(C)nc(O)cc2)=O)CCCCCCC1C(=O)NC1C2CCCC1CC2 65057,C1(NC(c2cc(C(C)C)no2)=O)CCCCCN(C(=O)C(=Cc2c[nH]cn2)F)C1 65058,c1(OC(C)C(=O)NC2CN(C(C3C4COCC34)=O)CCC2O)ccc(C#N)cc1 65059,c1(C(=O)NCC(CNC(=O)COc2ccccc2)O)cccc2cccc(O)c12 65060,C1(NC(COCC#C)=O)CC2(C1)CN(C(c1csc(C3CC3)n1)=O)C2 65061,S(=O)(=O)(c1c(F)cccc1F)NC1C(C(=O)Nc2cncc([N+](=O)[O-])c2)C1 65062,CS(=O)(=O)c1ccc(S(=O)(=O)NCCNC(=O)Nc2ccc(Cl)c(Cl)c2)cc1 65063,c1(C(=O)NCC2CCCCC2)ccc(NC2=NCCC2)cc1 65064,c1(NC(CC2C=CC(NC(c3c(CCC)nco3)=O)C2)=O)cnc(OC)cc1C 65065,C=CCC(CC(=O)Nc1cnc(C2CC2)nc1)NC(=O)CC1(O)CCOC1 65066,c1(C(=O)NC(C(CO)NC(C(CCCOC)C)=O)C)nnc(O)c2ccccc12 65067,C(=O)(CC(C)P(C)(C)=O)N1CCCC(CCNC(c2cc(C)cc(N)c2)=O)C1 65068,Cn1c(C(=O)NCC2(CO)CCN(C(=O)Cc3cn(C4CC4)cn3)C2)cnc1O 65069,C1(CN(C)C)CC(O)CN1C(c1n[nH]cc1CNC(=O)CC1CC(=O)C1)=O 65070,n1(CC)ncc(C(N2CCCCC2CNC(=O)Cc2csc(NC=O)n2)=O)c1Cl 65071,C1(CNC(CC(C=C)CC)=O)CC2(CCN(C(=O)C(C)C(C)CC)CC2)CO1 65072,COn1cnc(C)c1C(=O)NCC1CCC1NC(c1cc(F)ccc1C1CC1)=O 65073,c1(C(=O)NCCCN(C(C(C)OCCCC)=O)C(C)C)cc(S(C)(=O)=O)oc1C 65074,C#CCCCCC(=O)N1CCC(NC(=O)CCc2cccc(OC)n2)C(F)C1 65075,N1(C(c2c(CC)nco2)=O)CC(NC(C2CCCC2C(C)C)=O)C(O)C1 65076,c1(C(N(C2CCN(C(CCCC)=O)C2)CCO)=O)c(C)cccc1C 65077,c1(C(=O)NC(C2CCCN(C(C3(COCC)CC3)=O)C2)C)cc(Cl)ncc1O 65078,c1(C(=O)NCCCNC(c2cc(C(F)F)ccc2O)=O)cc(Cl)c2n[nH]cc2c1 65079,CCC(C)CC(=O)NCC1CC(NC(=O)Cc2sc(C)nc2C)C1 65080,C(=O)(CC1CCc2ccc(O)cc21)NCC(C)NC(c1cccc2cncn12)=O 65081,n1(CC)nc(C)cc1C(=O)NCC1CN(C(=O)C(C(C)C)NC=O)CC1O 65082,N1(C(Cc2c(C)cnn2C)=O)CCC2CC2(C(=O)NCC2(O)CC=CC2)CC1 65083,Cc1[nH][nH]c(=N)c1C(N1CCC(CN(C)C(c2cnc(CC(C)C)[nH]2)=O)C1)=O 65084,N1(C(C2(C#C)CN(C(C3CCC(F)(F)C3)=O)C2)=O)CCN(C)CC1C 65085,C1(C(=O)NCC2(O)CCCN(C(=O)C(C)C(C)C)C2)(CC)CCC(O)CC1 65086,C1(CN(C)C)CCCCN1C(=O)CC=CCNC(=O)CC(O)C1CCCC1 65087,c1(C(=O)NC2CC(NC(C3(c4ccc(F)cc4Cl)CC3)=O)C2)occ2c1CCOC2 65088,CCC(C(=O)NC(CC1CCC1)C(=O)NCCCCCSC)N(CC)CC 65089,c1(OC)cc(N(CCNC(c2nn(C)c(Cl)c2Cl)=O)C2CC2)c(Cl)cc1[N+](=O)[O-] 65090,C(CC(=O)NOCCCC1CC1)N(C(CCOCCCO)=O)C.C1CN1 65091,Cc1cc(C(=O)NCC(C)NC(=O)C(O)C2CC2)c(C)n1CC(F)(F)F 65092,n1(CC)nc(C(=O)NC2CN(C(=O)C(C3CC3)N(C)C)CC2C)cc1C(F)(F)F 65093,c1(CNC(C(C)OCC(C)C)=O)ccc(CCNC(=O)CNC(N)=O)cc1 65094,C(=O)(C#CC(C)(C)CNC(C1(C)CCCC1O)=O)NC(C(=O)N(C)CC)C 65095,C(=O)(C(C)C(F)(F)C(F)F)N1CCN(C(CC2CCC(C)CO2)=O)CC1CO 65096,C1(C(=O)NCC2CC(NC(C3CCS3(=O)=O)=O)C2)CCC([N+](=O)[O-])CC1 65097,c1(NC(C2CCC(C)(C(C)=O)C2(C)C)=O)cccc2c1COC(=O)N2 65098,c1(C(N2C(CC(C)C)CCCC2)C(=O)NC2COC2)cccn2ccnc12 65099,N1(C(C(CC)CN(C)C)=O)CC2(C)CC1(C(=O)NOCc1cncs1)C2 65100,N1(C(C(CCC)C)=O)CCN(C(=O)CSCC(C)C)CC1C 65101,N1(C(CSCCC(C)C)=O)CCN(C2CCN(C(C3COCCN3C)=O)C2)CC1 65102,C1(C(C)(C)O)(CNC(=O)C=CC2CCC2)CN(C(=O)CC2C=CCC2)C1 65103,N1(C(c2cc(CC)on2)=O)CCN(C(=O)C=Cc2ccc(SC)cc2)C(CF)C1 65104,c12ccc(cc1)C(=O)N1CCC(C1)N(C)C2=O.C1(F)(CC2CC2)CC1.C(CO)S 65105,c1(CN(CCNC(C2CCCN2C(=O)NC(C)C)=O)CC)ncccc1F 65106,N1(C(CCCN(CCC)CCC)=O)CCC2(CCCN2C(=O)C(C)SCC)C1 65107,Cc1cc(C(c2nnnn2-c2ccc(F)cc2)NC2(CCF)CC2)c(C)cc1Br 65108,Cn1cnc2ccc(C(N3CCN(C(c4ccon4)=O)C(C(F)(F)F)C3)=O)cc12 65109,CC1(NC(C2C3CC4C(C3NC(c3cnc(O)o3)=O)C24)=O)CCCCCC1 65110,C1(C)(COC)CC(NC(C2(C(N)=O)CCC2)=O)CN1C(=O)CCC(C)C 65111,Cc1cc(C(=O)NC(CCN(C)C)C(=O)NCC2=NOC(C)C2)c(C)nn1 65112,C1(O)(CN2CCN(C(C3C(OC)COCC3)=O)CC2)CCCCCC1 65113,C1(CC(=O)NCCOCCN(C(COCCCCCC)=O)C)COC(C)(C)C1 65114,c1(C(N2C(CCNC(C3CCN(C)C3)=O)CCC2)=O)cc(F)c2cn[nH]c2c1 65115,c1(C(C(=O)NCCSC)N(CC(F)F)C(C)C)ccc(C)c(F)c1F 65116,C1(C(N(CC(C)NC(C2(CC)CCC2)=O)C)=O)CCCN(c2ccnc(Cl)n2)C1 65117,C(C(F)(F)C(=O)NC(C)CN(C(c1cc(-c2ccco2)on1)=O)CC)OC 65118,C(CN=c1[nH]c2ccc(F)cc2s1)C1CC(NC(C(C(C)O)C)=O)C1 65119,C1(NC(C2C3CN(C(C(C)=C4CCCC4)=O)CC32)=O)CCCOC12CCC2 65120,c1(C(N2C(C)CCC(CNC(=O)Cc3cccs3)C2)=O)cncc2c1CCC2 65121,N1(C(C(C)=CC2CC2)=O)CCCC(CO)(NC(c2cncc(Cl)c2)=O)C1 65122,C#CC1CN(C(C23CC(CN(C(C4(F)CCC4)=O)C2)C3)=O)CCO1 65123,c1(C(=O)NC2CCCN(C(C(C)C(F)(F)F)=O)CC2)cc2c(F)c(Cl)ccc2[nH]1 65124,C1(NC(C2C(c3ccc(C)c(Br)c3)C2)=O)CC2(CCC(NC(C)C)CC2)C1 65125,C(CCC(C)(C)C(=O)N1CC(O)C(O)CO1)OC(c1c(OC)scc1)=O 65126,Cn1[nH]nnc1=NCC1(CNC(=O)CCn2cnnn2)CCC1 65127,N1(C(c2cnc3n2CCOC3)C(=O)NC(C)C)CCC2(COC(C)C2)C1 65128,N1(C(CCC2C(=O)NC(=O)N2)=O)CC2CCN(C(C3(F)CC3)=O)CCC2C1 65129,c1(CN2CCN(CCOC)CC2)ccc(-c2ccc(Cl)s2)cc1F 65130,c1(OC)cc(C(N2CC(O)CC2CNC(=O)CCCOC(C)=O)=O)c2c(c1)CCO2 65131,C1(NC(CNCC(=C)C)=O)CCOC12CCN(C(=O)CCNC(=O)COC)CC2 65132,N1(C(c2c(OC)cc(C)cc2)=O)CC2CC1CN(C(=O)CCC1(C)CC1)C2 65133,CCC(C(=O)NCC1CCN(C(C2CCN(CC)C2)=O)C1)n1cncn1 65134,c1(C(N(CC(=O)NC)CC)=O)ccc(C2COCCN2C(c2ccsc2Cl)=O)n1C 65135,C1(C(N2CC(NC(C3(CC)COC3)=O)C2)=O)CCOC(C)C1 65136,CN1CCOC(C(=O)NC2CN(C(c3cc(-c4ccccc4)ns3)=O)CC2O)C1 65137,N1(C(c2cccc(SC)c2Cl)=O)CCN(C(=O)C(=O)C(C)(C)C)CC(O)C1 65138,C1(CN(C2CCN(CCS(N)(=O)=O)CC2)C)CN(C(=O)OC(C)(C)C)CC1O 65139,c1(CC)occc1C(=O)NC(CNC(c1cnc(C)s1)=O)CCOC 65140,C1(C(=O)NCCCN(C(C2CC2)=O)CC2CCCC2)CCC2CC2C1.CCS 65141,N1(C(C)C)CCC(C(=O)NC(C)CC2CCN(C(=O)CC=C(Cl)Cl)CC2)CC1 65142,C(=O)(CC(O)Cc1ccccc1)N1CC(NC(C2CSC2)=O)C1 65143,n1(CCNC(NC(C2CCC2)C)=NCCC(C)F)nnc2ccccc2c1=O 65144,c1(C(=O)NC(CN(C(=O)C(C(C)C)OC)CC)C)cc2cc(Cl)ccc2n1C 65145,c1(N2C(CCNC(C3C(C)C3c3ccccc3)=O)CCC2)ncc(I)cn1 65146,c1(CC)cccc(C(N2CC(F)CC2CN(C)C(c2ccc(Cl)s2)=O)=O)c1O 65147,c1(C(=O)NC2CCN(C(C3(OC)CCOC3)=O)C2)cc2cccc(Cl)c2nc1C 65148,c1(OC(C)C(N2CCCCC2CCNC(=O)CP(C)(C)=O)=O)cccc(F)c1 65149,C1(CNC(C(C)(C)c2ccccn2)=O)CN(C(C2CCCS2)=O)CCC1(F)F 65150,c1(C(N2C(C)(C)C(O)CC2)=O)cc(Cl)cn2nccc12 65151,c1(C(=O)OCC)cc(C)sc1NCc1cn(-c2ccccc2OC)cn1 65152,C1(CNC(c2c(C)cn(C)c2)=O)CN(C(c2ocnc2C2CC2)=O)CC(C)(C)C1 65153,C(CCC(C)C(=O)N1CC(O)(CN(C(=O)Cc2cc(C(F)(F)F)n[nH]2)C)C1)OC 65154,C1(C(N(CCCN(C(=O)CCn2cnnn2)C)C)=O)CCCNC1=O 65155,C1(NC(C(C)OC)=O)C2CN(C(=O)CCC(=O)N(C)C)CC12 65156,c1(C(=O)NCC2CN(C(C(CC(C)C)OC)=O)CC2(F)F)scc2c1OCCO2 65157,c1(C(N2CC(C)N(C(=O)C=CC3CCOC3)CC2)=O)cc(Cl)c(F)c(Cl)c1 65158,CC1N(N2CCOC(c3ccc(F)c(F)c3)C2)C2(CCCC2)C1C(N)=O 65159,C12(NC(CC(CC)C3CC3)=O)CN(C(c3ccc(F)s3)=O)C(COC)(C1)C2 65160,C1(N(C)C(c2coc(CNC(C3CC(=C4CCC4)C3)=O)n2)=O)CCCC1C#N 65161,N1(C(CCC(N)=O)=O)CC2CCC1C(Nc1ncnc3c1COC3)C2 65162,C(C(CC)(CC)CC)(c1n(CCCOC)nnn1)NCC1CCCC12CCC2 65163,c1(C(=O)NC(C(=O)NCCc2cnc(C)[nH]2)Cc2ccoc2)cnc(Cl)n1C 65164,Cc1nnc(C(=O)N(C(C)CCNC(C2CC2(C)C(F)(F)F)=O)C)s1 65165,C1(C(=O)NCC2(N(C)C)CCC2)CCCCCN1C(=O)CCc1ccoc1 65166,Cc1ccc(C(N2CCN(C(=O)C(Cl)=CCl)C(CC(C)(C)C)C2)=O)c(=O)n1C 65167,N1(C(=O)CCc2ncc(F)cn2)CC2CCC1CN2C(=O)Cc1ccc(Cl)cc1 65168,N1(C(CCC)=O)CC2(NC(c3ccc(F)cc3CC)=O)CCC1C2 65169,Cc1ccc2c(=NCC(C)Cc3cn[nH]c3)[nH]c(=NC(CCO)C3CC3)[nH]c2c1 65170,c1(C(N2CCC(F)(CF)C2)C(=O)NCCC)cc(C(F)F)nc(C)n1 65171,C=CC1(C(=O)NCc2c(C)ccnc2C)CCN(C(=O)CCN(CC)CC)C1 65172,c1(C(N2CC(F)CC(NC(C(CC)C(C)C)=O)C2)=O)cccc2c(C)c(C)[nH]c12 65173,c1(C(=O)NCC2(COC)CCCN2C(=O)C(C)C(C)(C)C)cn2c(n1)CCC2 65174,N1(C(C(C2CC2)OCC)=O)CC(C)C(C)(CNC(c2ccc(N)c(O)c2)=O)C1 65175,c1(-c2cn(CC3N(CC(=O)Nc4ccc(Cl)nn4)CCC3)nn2)sc(O)nc1O 65176,C(=O)(C1CCc2nccn21)NCC1(NC(c2cn(C)nc2)=O)CCOC1 65177,C1(NC(c2cc(C)nn2C(F)F)=O)CC2CN(C(c3cnc(Cl)s3)=O)CC12 65178,c1(OC)c(C)cc(C(=O)NCCCCNC(=O)CC(C)C)cc1Cl 65179,c1(C(N)=O)cccc(C(=O)N(CCC(=O)NCc2ncccc2O)CC2CC2)n1 65180,N1(C(C(C)(C)C)=O)CC(NC(=O)CCOC(=O)NC(=O)C(C)(C)C)C(F)C1 65181,c1(CCNC(c2c(CCC(=O)OC)cccc2)=O)c(Cl)cc(Br)cc1Cl 65182,C1(CCOC)CCCCN1C(C1CCN(C(c2cc(C)no2)=O)C1)=O 65183,c1(C(=O)NC)cccc2c(Br)cccc12.c12nc(cs1)C(=O)N2.c1ccccc1 65184,N1(CC(=O)NC2(CO)CN(C(CC3CCC(C)C3)=O)C2)CCCNS1(=O)=O 65185,C(CC(C)(C)C(=O)NC1CC1NC(=O)Cc1cccc(OC)c1Cl)OC 65186,CN(C[Si](C)(C)C)C(=O)CC1CCCCN1C(=O)CCc1cnco1 65187,C(=O)(C1Cc2c(Cl)cccc21)N(CCCCN(C(CCC(=O)NC)=O)C)C 65188,c1(OC)ccc(C)nc1C(=O)NC1CCCC(NC(C2CC3(C2)CC(O)C3)=O)C1 65189,CC1CCCCC1OCC(=O)NCCC1CC(NC(C2(C(N)=O)CCC2)=O)C1 65190,Cc1cc([N+](=O)[O-])cnc1N1CC(CNC(C2(Cl)CC2)=O)OC2(CCC2)C1 65191,N1(C(C(C)SC(F)(F)F)=O)CCCC(CCNC(=O)C(c2ccccc2Cl)O)C1 65192,CC1(C)C(CNC(=O)Cc2cc(C(F)(F)F)co2)CCN1C(=O)CCc1ccsc1 65193,c1(NC(C2CC(F)(F)CO2)=O)cc(Cl)c(Cl)cc1CO 65194,C(CCCCCCCO)=CC(N1C(CNC(C2CCC2(C)C)=O)CC(C)(C)C1)=O 65195,N1(C(Cc2c(C)non2)=O)CCCC(CNC(c2cc(C(N)=O)no2)=O)C1 65196,C(CC(C)C(=O)NC(Cc1ccoc1)C(=O)NCC1CC(O)C1)=CCC 65197,N1(C(CCCC=C)=O)CCC(NC(=O)C(O)CCCCC)CC(C)(C)C1 65198,CC1(C)C(NC(c2ccn3nnnc3c2)=O)C(C)(C)C1NC(=O)C(F)=CCCF 65199,CC1(C)CCC=C1C(=O)NC1CCOCC1NC(C1Cc2cscc2C1)=O 65200,N(C(=NCc1ccccc1)N1CCC2(CCCC2)CC1)CC1CC(=O)NC1 65201,N1(C(C(C2CCN(C(c3cc(CC)[nH]n3)=O)C2)C)=O)CC(C)CC1C(=O)OC 65202,C#CCC(C)(C(=O)NC1CC(C)(C(N)=O)C1)NC(C1CC2(CC2)CO1)=O 65203,c1(NC(=O)NCc2cc(C3CCN(C(C)=O)CC3)no2)ccc(C(N)=O)c(Cl)c1 65204,CCC(CO)(C(=O)NC1CCOC1C(=O)NC1CC(CO)C12CCC2)OC 65205,C(=O)(C(C)=NOCC#N)NCC1(CC=CC(=O)NC(C(C2CC2)OC)C)CCC1 65206,C1(CNC(CCC#C)=O)CCN(C(=O)C=Cc2cncn2C)C(C)C1 65207,Cc1nnc(O)c(C(=O)NCC(CC(F)(F)F)NC(=O)CC(C)(F)F)c1C 65208,C1(C(=O)NC2C(NC(CC=CC=C)=O)COC2)CCCCN1C(=O)OC 65209,c1(C(N2CC3C(N(C(CC=C)=O)C)C3C2)=O)cc(C(F)(F)F)cc(N)c1 65210,C(=O)(C1=CCN(C(c2ccc(F)c(F)c2)=O)C1)NC1CCN(CC)C1 65211,c1(C(=O)NCCCNC(CCc2ccc(C)o2)=O)ccn(C2CC2)c1C 65212,Cc1ccnc(C(C)(C)C(=O)NC2CCCC2NC(C2CCCC2(C)C)=O)c1 65213,C1(C(C(C)OC(=O)Cc2nncn2C)=O)CCCC(C)(C)CC1 65214,c1(CC)ccc(C(N2CCC3(NC(c4cnn(C)c4C)=O)CC3C2)=O)c(O)c1 65215,C1(C)(CNC(C2C(C)(C)C2(C)C)=O)CCN(C(C2CC2C2CC2)=O)CC1 65216,C1(C(=O)NC2C(NC(c3ccsc3)=O)CCCC2)CC12CCCCCC2 65217,c1(OC)cc(CNC(=O)C(=O)NCC(C2CCCNC2)N)ccc1F 65218,O=C(C1=CCCSC1)NC1C2CN(C(=O)CC3CCCO3)CC12 65219,N1(C(c2c(C)noc2)=O)CCC2(CO)CN(C(=O)C=CC3CCC3)CC2C1 65220,C1(NC(COCC(=O)NC)=O)CC2CC1N(C(c1csc(CO)n1)=O)C2 65221,C1(CN(C(=O)C(C2CCN(C(=O)Cc3ccc[nH]3)C2)F)C)CCCC1(C)C 65222,Cc1cc(F)cnc1CNC(C1CC1c1ccccc1Cl)=O 65223,C1(CNC(C2(SC)CCC2)=O)(CO)CCN(C(c2c[nH]c(C#N)c2)=O)CC1 65224,c1(C(=O)NCC=CCC(=O)NC(C2CCOCC2)C)sccc1C#N 65225,N1(C(C(c2ccccc2)OCC)=O)CCN(C(=O)CS(=O)(=O)NC)CC1CC 65226,CC(CC(C)(C)C)C(c1nnnn1C)NC1CCS(=O)(=NC(=O)C2CCCC2)C1 65227,C1(NC(C(C)NS(CC)(=O)=O)=O)CC2CCC1N(C(c1c(C)nsc1N)=O)C2 65228,Cn1nc(C2CC2)cc1NC(=O)NCc1cnc(C(F)(F)F)cn1 65229,N1(C(c2c(OC)scc2)=O)CCN(C(=O)C(F)CC(C)C)CC(C)(C)C1 65230,c1(C(=O)NC2C3C(C)N(C(C4CCCCN4C)=O)C2C3)ccc2nc[nH]c2c1 65231,C1(C(=O)NC2CCN(CC(=O)NC(COC)C(C)C)CC2)CC2(C1)CC2(F)F 65232,c1(C(c2ccc(C)o2)NC(C2C(C(=O)OC)C2)=O)cc(CSC)cc(OC)n1 65233,C12(NC(Cc3cnc(C)s3)=O)CCCC1N(C(=O)CCCN(C)C(C)C)CCC2 65234,N1(C(=O)CCCC(F)(F)F)CC2C3CCC(C2C1)N(C(c1ccc(Br)cn1)=O)C3 65235,c1(C(=O)NC2CCC(N(C(CNC(CCCCC)=O)=O)C)C2)nnc(O)nc1O 65236,c1(OCCC)ccc(Cl)cc1C(=O)NC1CN(C(=O)C(C)(O)CC)CC1O 65237,C1(C(N2CCN(C(c3cnc(N)c(CO)c3)=O)CC2)=O)CC12CCS(=O)(=O)CC2 65238,C(C)(c1ccco1)=CC(=O)NC(C1C(CC(=O)NCC2C(=C)C2)CC1)=O 65239,c1(C(N2CCN(C(C=CC)=O)C(CCC)C2)=O)nnc2ccccc2n1 65240,N1(C(C2C(C=C)OCC2)=O)CC2(CC2)CC1C(=O)NCC1CC2CCC2C1 65241,N1(C(CSS(C)(=O)=O)=O)CC2(CCCC(CNC(C3CCS3(=O)=O)=O)O2)C1 65242,C(=O)(C(C)(CO)N(C)C)N(CCN(C(C=CCOC)=O)C)C 65243,C(=O)(CCC(=O)NCc1nc(C)c(C(=O)N(CCC(O)CO)C)o1)NCCC 65244,C1(C(=O)NCCC2(C)CCCO2)CCC(CNC(c2ccc[nH]2)=O)CC1 65245,C1(NC(C2C3(CC3)C23CC3)=O)CCCCC1CC(N1CC2CC1CO2)=O 65246,c1(OC)nc(C(N2CCC(OCCOC3CCOCC3)CC2)=O)ncc1F 65247,n1(CCC)nc(C)cc1C(=O)NC(C)CCN(C(=O)CCCn1cncn1)C 65248,N1(C(C2(CC=C)CCOC2)=O)CC(N(C(=O)CSC2CC2)C)C(O)C1 65249,c1(CC(=O)NC(CC)CN(C)C(C2C(CC3CC3)C2(F)F)=O)ccccc1F 65250,Cc1nc(O)ccc1C(N1CCC(CNC(=O)CCCSC(C)(C)C)C1)=O 65251,N(C(=NCCC1CC1(Cl)Cl)NC1CCOc2c(C)cccc21)CC(=C)C 65252,S(=O)(=O)(c1ccc(COC)s1)NC(CC)C(c1cc(C)ccc1C)O 65253,Cc1ncc(C(=O)NC2CCC(C(=O)NCC(c3ccccn3)O)C2)c(=N)[nH]1 65254,C1(O)(C(C(=O)N(CC(=O)NC(C)C)C)F)CN(C(C2(CO)CCC2)=O)C1 65255,C1(C(=O)NC(C(=O)NC(C)C)C)(CO)CCN(C(c2c[nH]c(=S)cn2)=O)C1 65256,C1(CNC(C(c2ccccc2)N(C)C)=O)CCCCN1C(=O)COC(F)(F)F 65257,C1(OC)CN(C(=O)Cc2cccn2C)CC1NC(=O)CCCN(C)C(C)C 65258,C1(C(=O)NCCCCNC(c2[nH]cc(C)c(=O)c2)=O)CCCC1S(C)(=O)=O 65259,C1(C(=O)NCCCOCCN(C(=O)CC2C=CCCC2)C)C2CCCCC12 65260,N1(C(CCNC(=O)OC)=O)CC(CNC(=O)CC2CCCSC2)OC(C)(C)C1 65261,N1(C(CC(CC=C)NC(c2coc(CO)c2)=O)=O)CC=CC12CCOCC2 65262,C1(C#N)(C(N2CCC(NC(c3cnc(SC)s3)=O)C(F)C2)=O)CCN(C)CC1 65263,N1(C(CCCOCCOC)=O)CCCC(C(C)NC(c2c(OC)noc2C)=O)C1 65264,C1(C(=O)NC2(CNC(CSCC#C)=O)CCOCC2)COC2(CO)CC1C2 65265,C1(CNC(C(CCCC)O)=O)CN(C(c2ccnn2C(F)F)=O)CCC12CCC2 65266,c1(C(N(CCC(C)NC(=O)CC2CCCOC2)C)=O)csc2c1CCCC2 65267,n1(CC(=O)NCC(C)C(=O)NC2CCC3CCC23)cc(C#N)cn1 65268,C1(C(=O)NCC2CCCN2C(=O)CCc2ncc(F)cn2)SC2C=CC1CC2 65269,c1(CCn2cc(COc3ccc(Cl)cc3)nn2)cccc2c1B(O)OC2 65270,c1(CN(C(C(C)=CCC)=O)C)ncc(-c2ccccc2)[nH]1 65271,c1(C(N2C(CNC(C3COCC(C)(C)O3)=O)CC(F)C2)=O)ccc(C#N)c(F)c1 65272,CC1(C)CN(C(C2CC3(CC(NC(C4CC4C4CC4)=O)C3)C2)=O)CCN1 65273,N=c1ccc(C(=O)NC(CC2CCOCC2)C(=O)NCC2C=CCCC2)n[nH]1 65274,C1(c2nnnn2CCCSC)(NC(N2CC(=CCOCC)C2)=O)CC(F)(F)C1 65275,C(=O)(C1CSc2ccccc21)NC1CCN(C(Cc2cc(C)[nH]n2)=O)C12CC2 65276,c1(SC)cc(Br)ccc1C(N1CCCC(C)(NC(=O)C(C)C2CC2)C1)=O 65277,c1(C(N=S(C)(=O)C2CCCC2)=O)c(CN)ccc2ccccc12 65278,C=CCC(CC=C)C(=O)NC1(C)CCN(C(C2(COC)CC=CC2)=O)C1 65279,CCCCC(C)CCC(=O)N1CC(CNC(c2cccc3ccnn23)=O)C1 65280,C1(NC(C2CCN(c3ccncc3)C2)=O)COC2(C1)CN(C(C1CC(O)C1)=O)C2 65281,C1(CC)(CC)CCCN(C(C2CCCSC2)C(=O)NC2CCOCC2)CC1 65282,C1(NC(CN2CC(=O)NCC2)=O)C2CC(NC(=O)CN3CCCCCC3)CC12 65283,C(=O)(C1SCCc2sccc21)N(CCC)CCNC(=O)CCc1ccsc1 65284,N1(CC(=O)NCCc2cc[nH]n2)CCN(C(C2CC23CCCC3)=O)CC1 65285,n1(CCC)ccc(C(N2CCC(CCNC(C3(c4n[nH]cc4C)CC3)=O)C2)=O)n1 65286,c1(CN(C2CCN(C(c3ccc(F)nc3)=O)CC2)CCOC)ccc(Br)cc1F 65287,c1(OC(=O)CSc2ncc(C=CC(=O)Nc3ccccc3)s2)cncc(Cl)c1 65288,Cc1ccc2snc(C(=O)NCC3(NC(C4C(F)(F)C45CCC5)=O)CC3)c2c1 65289,C12(CNC(CCC#C)=O)CCCC1N(C(c1ccc(NS(C)(=O)=O)nc1)=O)CC2 65290,N(C(=NCCCCl)NCC1CC1C(F)(F)F)CC(C1CCOCC1)(F)F 65291,Cc1cc(C(N2CC(CCNC(c3ccns3)=O)C(C)C2)=O)cc2cccnc12 65292,CC(C(C)(C)NC(S(=O)(=O)C1CC1)=O)NC(C1(n2cncn2)CC1)=O 65293,C(=O)(CC(C(F)(F)F)OC)NC(CCC)CCCNC(c1ccnnc1O)=O 65294,CC(C)CCC(C(=O)O)NC(=O)COCc1cn(CCCO)nn1 65295,c1(C(N(CC(C)N(C(=O)C(C)c2cc[nH]n2)C)C)=O)c(Cl)ccc(O)c1N 65296,S(=O)(=O)(c1cccc(Cl)c1F)N1CCN(C(c2n(CC)nc(C)c2)=O)C(C#N)C1 65297,C1(C(N2CCN(CCNC(C=CC(C)(C)C)=O)CC2)=O)CCCCC1C1CC1 65298,C(=O)(C1=C(C)N(C)c2ncnn2C1C)NC1CN(C(C=C(C)C(F)F)=O)CC1C 65299,n1(CC(=O)NC(C)C(=O)NCCC2(NC(=O)CO)CCC2)ncc2ccccc12 65300,c1(NC)cccc(C(=O)N(C2CC(C(=O)N(C34CC(C3)C4)C(C)=O)C2)C)n1 65301,N1(C(c2cncs2)=O)CCCCC2(C1)CN(C(C1(c3ccccc3)CC1)=O)C2 65302,c1(C(C)(C)NC(N(CCNC(=O)OC(C)(C)C)CCO)=O)cc(Cl)ccc1O 65303,C1(NC(c2cccc(CC)n2)=O)CC(O)CN(C(=O)COC(F)(F)F)C1 65304,n1(CC(N2C3CC(C(=O)Nc4cccc(C)c4O)C2CC3)=O)cnc2ccccc12 65305,N1(C(CNC(C(CC)C)=O)=O)CCOCCC1C(=O)NCc1cnc(F)cc1C 65306,C12(NC(C3CCS(=O)(=O)N3)=O)CCCN(C(=O)CSCc3ccccn3)CC1C2 65307,c1(C(=O)NC2CCN(C(c3c(OC)nsc3OC)=O)C2)ccc2nnc(O)n2c1 65308,N1(C(CN(C2CC2)CC)=O)CCC2CN(C(c3scc(OC)c3OC)=O)CC12 65309,c1(C(=O)NCC(CC=C)NC(=O)C2=CC(C)(CC)C2)ccc(OC)c2ccsc12 65310,CC(CF)CC(=O)NCC1(O)CCN(C(c2cc(Cl)sc2Cl)=O)C1 65311,C=CCC(C(=O)NCC1C=CCN1C(c1csc(CS(C)(=O)=O)n1)=O)C(C)C 65312,C(=O)(C(C(=O)NC1(CF)CN(C(C2CCCN2C2CC2)=O)C1)C(C)(C)C)OCC 65313,C(C(CC(C)C)C(=O)NCC1C=CC(NC(=O)CCCN(C)C2CC2)C1)OC 65314,C(=O)(C(F)(F)CC(C)C)NCCN(C(CCC1C(C)C1)=O)C.c12ccc(o1)c(=O)[nH]2 65315,CC1CC(CNC(C2(C)CNC(=O)C2)=O)CN(C(C2(C(F)F)CCCCC2)=O)C1 65316,N1(C(C(CC=C)CNC(=O)C=C(C)C2CC2)=O)CCc2cncnc2C1 65317,CC1(C)CCCN(C(=O)C(C2CCOCC2)=O)C1C(N1CC2(C=CCO2)C1)=O 65318,C1(O)(CN(C(c2cc(C)sc2)=O)C)CCN(C(c2nocc2Cl)=O)C1 65319,C1(C)(CC(=O)N(C(c2ccccc2)CNC(c2ccnn2C)=O)C)CCS(=O)(=O)N1 65320,C(CC(C)N=c1cc(C)nc(NC(c2cc(C)ccc2F)C)[nH]1)OC 65321,C12(C(=O)NCCNC(C34CC(CC(F)F)(C3)C4)=O)CC3CC1C2C3O 65322,c1(OCC)cnc(C(c2nnnn2C2CCOC2)NCCc2cn(C)cn2)nc1 65323,C(CC(C(C)(C)C)NC(C1CCC1COC)=O)N(C(CC(COC)C)=O)C 65324,C1(CN(C(C2CCN(C(C)=O)C2)=O)C)C(=O)NCCN1C1CCCC1 65325,C1(NC(C2CC2F)=O)CN(c2ccnc(CO)n2)C2CCCCC12 65326,N1(C(c2c(CC)oc(C)c2)=O)CCC2(CC1)CN(C(C13CCCCC1C3)=O)C2 65327,C=CCC(CNC(C1COC(=O)C1)=O)NC(=O)CCC1CCCCC1 65328,c1(NC(C2N(C(c3c(Br)cnc(C)n3)=O)CCOC2)=O)cccc2ccoc12 65329,c1(C(=O)NCC2C(C(F)(F)F)CN(C(CCSCC)=O)C2)ccc(Cl)c(F)c1F 65330,C=CCCC(C(=O)NCc1cc(F)ccc1F)NC(C1CCC1c1nc[nH]n1)=O 65331,O=C(CCCCC(F)F)N1CC2CCN(C(=O)C=CC3CCOC3)C2C1 65332,N1(C(C(C)C)=O)CC2CCCC(C1)N2C(C1(C)CC2CCC(C1)S2)=O 65333,c1(C(=O)NCC2OCC(C(=O)NCCOC(C)=O)C2)cccc(O)c1C 65334,c1(OC)cc(C)ccc1C(N1CCN(C(=O)C(=O)NCCC(N)=O)CC1CF)=O 65335,C1(C(=O)NCC(CSC)OC)CCC(C)(C)N(C(=O)C2=C(C)OCCS2)C1 65336,N1(C(CC2CC(=C)C2)=O)CCCC2(CCCN2C(c2cnn(C)c2OC)=O)C1 65337,CC(C)CC(C)C(=O)NC1C2CCN(C(c3ncnc(O)c3Br)=O)C12 65338,c1(CC(=O)NCC=CCNC(C2C(=C)CC2)=O)c(C)cccc1Cl 65339,C1(C(N(C)CC2CCN(C(=O)CN3CCNC3=O)C2)=O)CCOC2(CCC2)C1 65340,C1(C2CCN(C(C3(Br)CC3)=O)CC2)(NC(COc2cccc(C)c2C)=O)CC1 65341,S(=O)(=O)(c1c(F)cccc1F)N(c1ncnc2[nH]ccc12)c1ccc(=N)[nH]c1 65342,C1(C)(COC)CN(C(c2cc(CNC(c3cnc(Cl)s3)=O)[nH]n2)=O)C1 65343,C#CC(C)(C)C(=O)N1CC(C=C)(CC(=O)NCCc2ccc(F)cc2)C1 65344,c1(C(=O)NC2CCN(C(=O)CCc3nnc(O)nc3O)C2)ccc2ccnn2c1 65345,CCCC(C)(C)CC(=O)NCC1(OC)CN(C(c2nc[nH]c2C(F)(F)F)=O)C1 65346,C=CCCC(C)(C)C(=O)N1CC(C(=O)NCC2CCOC2)C2(CC2)C1 65347,c1(C(=O)NCC2N(C(C(C)SC(F)(F)F)=O)CCC2)ccnc(C(F)(F)F)c1N 65348,c1(C(C)(F)F)ccc(CNc2csc(-c3cccc(Br)c3)n2)nc1 65349,c1(C(=O)NC(C)CNC(=O)CSC2CCOC2=O)cncc2c(O)nccc12 65350,C1(C(=O)NCC(CNC(C2(C=C)CCCC2)=O)(C)O)CCC2(CC1)OCCO2 65351,Cc1cccc([N+](=O)[O-])c1C(=O)Nc1nc(C(=O)NC(C)(C)C)cs1 65352,N1(C(c2c(CCC)[nH]cc2)=O)CCCOC(CNC(C2(C3CCCO3)CC2)=O)C1 65353,C1(C)(NC(CC2(NC(C)=O)CC2)=O)CCN(C(c2c[nH]nc2C(F)(F)F)=O)C1 65354,c1(OC)cccc(C(=O)NC2CC(O)(CNC(=O)CCc3cnco3)C2)c1OC 65355,n1(CCOCC)nnnc1C(c1cccn1C1CC1)NC1(CC(C)C)CC1 65356,c1(C(=O)NCC2CCC(NC(c3n(C)c(S)nn3)=O)C2)cc2ccoc2cc1F 65357,CCCC(CC1CCCC1)C(=O)NC1CN(c2ncc(O)cn2)C1 65358,c1(CNC(=NCCOC)NCc2nnc3n2CCC3)nc2ncccn2n1 65359,c1(CN(C)C)ccc(C(=O)N(CCCNC(=O)CC2CC3CCC2O3)C)cc1 65360,C1(C#N)(C(=O)NC(CC)CN(C(=O)CNC(=O)C(F)(F)F)CC)CCOC1 65361,c1(C(=O)NC(CC(C)N(C)C)=O)cccc(C#N)c1.C1CC(C)N1C 65362,c1(C2(CC)CC2)ccc(C(=O)NCC(CC=C)NC(c2n[nH]c(C)c2F)=O)cc1 65363,c1(C(=O)NC2CC2C(=O)Nc2cnn(C3CC3)c2)cccc(O)c1F 65364,c1(C(=O)NC(C(=O)NC(CN(CC)CC)C)CC2CCC2)cc(C)cc(F)c1 65365,CC1CCOCCN1C(C1CCC2(CC2)N1C(=O)C(C)(C)N=[N+]=[N-])=O 65366,C1(C(N2CCCC(CCNC(=O)CC3CCCCCO3)C2)=O)CC2CCC1CC2 65367,c1(OC)cncc(C=CC(=O)NCC23CCC(CC2)N3C(C2CCSCC2)=O)c1 65368,C(=O)(C#CC1(C)CCCO1)NC1CC(C)(CNC(C2(C)CCC(=O)N2)=O)C1 65369,C12(CCC(=O)NCC=CCNC(C3CSCC(=O)N3)=O)CCC(CC1)C2 65370,c1(C(N2C3C(NC(CSCC)=O)(CCC3)CCC2)=O)cc(O)c2ccccc2c1 65371,C(=O)(C(CC(=O)OC(C)(C)C)C(=O)OC)N1CCN(C(C2(CC#C)CCC2)=O)CC1 65372,Cc1c(C(=O)NC2CN(C(C3CC3F)=O)CCC2O)oc(=O)c2ccccc12 65373,c1(N(C)C)cccc(NC(C2CN(C(=O)CNCc3cccs3)CCO2)=O)c1 65374,C1(CC(=O)N(CCCCCC)CCNC(=O)CCC)CC(OC(C)=O)C1(C)C 65375,c1(C(=O)NCCC(CCNC(C(COC)C)=O)C)cc2c(cc1F)OCC(=O)N2 65376,C1(n2cc(C(CC)CC)nn2)CCCCC1NC(C1(C)CCCN1C)=O 65377,c1(Nc2cccc(C)c2)nc2ccccc2nc1N(CCC(C)C)C 65378,C(=O)(C1=CCC(C)(C)CC1)NCCC(C(=O)N(C1CCOCC1C)C)OC 65379,C12(C(N(C(C)CNC(C3COC(C)(C)C3)=O)C)=O)CCC(C(F)(F)F)(CC1)CC2 65380,C=CC(C)(CC)C(=O)NCc1cc(C)c(C(=O)N(CC(O)CO)C(C)C)o1 65381,CCC(CNC(=O)CC1CCCC1O)(CC)C(=O)N1CC(N2CC(O)C2)C1 65382,CCC(CC(=O)NC1(CO)CCCN(C(C)=O)C1)CC(F)(F)F 65383,N1(C(CSCC(N)=O)=O)CC2CC2(CNC(c2csnc2Br)=O)C1 65384,c1(N(c2cc(CNCC3CCC(N)C3)ncn2)CC)ccc(Br)c2ncccc12 65385,N(C(=NCCC(C)=O)NCC1CCCC1CCC)Cc1n(CC)ncn1 65386,C(=O)(C1=C(C#N)CCC1)N1C(CNC(CC(C=C)CC)=O)CCC1 65387,C(C(C)(C)CCNC(=O)CC1COCCO1)NC(C(C1CC1)OCC)=O 65388,C1(C(=O)OC)CCCC(NC2CCCC(c3ccccc3)C2)CC1 65389,c1(C(N2CC(CNC(c3oc(C)c(CO)c3)=O)C2)=O)cc(O)ccc1Br 65390,CCCCCC(CC)C(=O)N1CC2(CCC2)CC1C(=O)NC(CCOC)C(C)C 65391,C12(C(=O)NCc3nc(C)c(C(=O)NCC4CC(F)C4)o3)CCCC1C2(F)F 65392,C1(NC(c2cn(CCC)nc2)=O)CCN(C(=O)CCCCC(N)=O)CCC1(F)F 65393,CC(C)CC(C)CNC(=O)C(O)CNC(=O)CSC(F)(F)F 65394,N1(C(C)=O)CC(CCNC(c2cnc(OC(=O)C(C)(C)C)c(Cl)c2)=O)OC(C)C1 65395,N1(C(c2ccc(C3CC3)[nH]2)=O)CCC2(C1)CN(C(C1(F)CCCOC1)=O)CCO2 65396,c1(CC)cccc(CC)c1C(N1CC(F)(F)CC1C(=O)Nc1cnc[nH]1)=O 65397,C1(NC(CCC=C(C)C)=O)CC(C)N(C(=O)CSc2nncs2)C1 65398,CS(=O)c1ccccc1C(N1CC2(C1)CN(C(c1cnc(F)c(F)c1)=O)C2)=O 65399,C1(C(=O)NCCC2CCCN(c3ccnc(C)n3)C2)CCCC(C)(C)C1 65400,Cn1cnc(C(O)CNC(c2occc2CNC(=O)Cn2cnnn2)=O)c1 65401,c1(C(=O)NC(C)CN(C)C(C2CCCN2c2cnccn2)=O)ccc(Cl)cc1O 65402,CCCS(=O)(=O)C(C)C(=O)NC1CCCC1NC(c1cnc2n1CCCC2)=O 65403,C1(C(=O)NC(CNC(=O)Cc2sccc2Cl)C2CC2)CC=CC(O)C1 65404,C1(NCCCC(=O)Nc2cccc(CCC(=O)O)c2)CCC2(CCCC2)C1 65405,C(C1=CCN(C(=O)C(C)S(C)(=O)=O)CC1)NC(CCCc1scc(C)n1)=O 65406,N1(C(Cc2n(C)ncc2)=O)CC(=O)NCC1C(=O)NCCC(=O)NC1CC1 65407,C1(N2CC(N(C(CCn3c(C)ncc3)=O)C(C)C)C2)CCCN(C)C1=O 65408,C1(CNC(C(C)c2ccsc2)=O)C2CC1N(C(c1ccccn1)=O)C2 65409,C1(CC)C(C)CCN1C(=O)CN(C(c1ccnn1COC)=O)CC 65410,C1(CNC(C2CC(OC)C2)=O)N(C(c2ccc(Cl)cc2Cl)=O)CCCC1(C)C 65411,c1(NCCN2C(C)CCC2)cc(NCCN2CCOCC2)ncn1 65412,C1(NC(C(C)NC(COC)=O)=O)CN(C(C2CC(C)(C)C2)=O)CCC1C(F)(F)F 65413,CC(C)CC(C(=O)NCC12CC1CN(C(c1cc[nH]c1)=O)C2)c1ccccc1 65414,C#CCC(C)(CC)C(=O)NCC(C(=O)N(C)Cc1nc(C)ns1)C(C)C 65415,N1(C(C(C)Oc2cc(C)c(C(C)C)cc2)=O)CC(C)C(O)(C(F)(F)F)C1C 65416,CCC(F)(F)C(=O)NCC(C)(C)CNC(=O)CN1CCNC(=O)C1 65417,C(C)(C(=O)N1CCC1CNC(C1(c2cnc[nH]2)CC1)=O)NC(CC)=O 65418,C1(CC(=O)OCC)CCCC2(CN(c3ccc([N+](=O)[O-])c(Br)c3)C2)O1 65419,c1(C(N2CC(NC(C3CCC3n3cccn3)=O)C(CO)C2)=O)ccc(F)cc1F 65420,C1(NC(C2C(C=C)OCC2)=O)CCN(C(=O)CCC2CC(C)C2)CC1O 65421,C1(C(=O)OC)CN(C(=O)Cc2cnc(Cl)cc2C)CCC1CN 65422,CC(C)(CC(=O)N1CC=CC(NC(c2cccc(-n3cccn3)n2)=O)C1)C1CC1 65423,c1(C(=O)NCC2CCN(C(C(C(C)C)OCC)=O)C2)cccc2nc[nH]c12 65424,C(CNC(=O)CCC(C)OC)(CC(=O)NOCC1(C)CC1)OC 65425,c1(NC(c2cnn(C)c2Br)c2n(C(C)C)nnn2)cc(Br)cc(C#N)c1 65426,N1(C(c2cc(CNC(CCC(C)C)=O)[nH]n2)=O)CCC(O)C12CCC2 65427,c1(CC(C(C)C)NC(=O)NCC2CC(F)CN2)ccccc1C(F)(F)F 65428,C(=O)(C1=COCCO1)NCCOC1(CNC(C(CC)F)=O)CCOCC1 65429,C1(Nc2nccc(N3CC(SC)OCC3)n2)Cc2ccccc2C1OC 65430,c1(OCC)cc(C(=O)NC2CCC2CNC(=O)C(C2CC2)N(C)C)ccn1 65431,C1(C)(CNC(C2C(=C)CC2)=O)CC(F)(F)CN1C(=O)C=Cc1ccc(F)nc1 65432,C1(O)(C(=O)NCCC2CCC(NC(C=CCCC)=O)C2)CCOCC1 65433,Cc1cc(NC(c2cn(C3CC3)cn2)=O)ccc1NC(=O)CN1C(C)CCC1C 65434,C(=O)(CC(O)CNC(C1CSC1)=O)N(C)Cc1scc(C)n1 65435,c1(C(C)(C)NC(C)=O)ccccc1OCCCc1ccc(F)cc1 65436,C=C(Cl)CC(C(=O)NCC(=C)C)NC(C1C=CCS1)=O 65437,C=CC(C)CC(=O)NCC1CC1CNC(=O)C(c1ccn(C)c1)C 65438,N1(C(C(c2ccccc2)SCC)=O)CC2C(CNC(C3CCOC(C)C3)=O)C2C1 65439,c1(C(N(CC(C)NC(=O)C(C)Cc2ccncc2)C)=O)cnc2ccccc2c1 65440,C1(C(=O)NC2C(CNC(c3c(C)nco3)=O)CC2)CN(C)CCO1 65441,C#CC1(C(=O)NCCCc2ccccn2)CCN(C(c2ccc(Cl)cn2)=O)C1 65442,C=CCC(F)(F)C(=O)NCC(C)(C)CC1CN(C(C2C(F)(F)C23CC3)=O)C1 65443,CC(CC(=O)N1CCCCC1c1n[nH]cc1NC(c1ccccc1)=O)C(C)(C)C 65444,C1(C(=O)NCCC2CCC2)CCCCN1C(c1cc(CO)ccn1)=O 65445,C1(C(=O)NC(C=C)C)(CC)CCN(C(=O)Cn2ncnn2)C1 65446,N1(C(c2c(Cl)nn(C)c2Cl)=O)CCC2CN(C(=O)C3=CCCOC3)CCC2C1 65447,C(=O)(C(CC)(CC)CO)N1CC(CC)C(NC(c2snnc2C)=O)C1 65448,CN1CCN(C(C2CN(C(=O)C(C)(C)O)CC(C)(C)C2)=O)CCC1=O 65449,C1(C(N(CCCNC(C(C)OC(C)(C)C)=O)C)=O)CCC(O)C1 65450,N(C1CCSc2ccc(Cl)cc21)S(c1c(C)nn(CC(F)F)c1)(=O)=O 65451,C(CCCCC(=O)NC1CCN(C(=O)COCCCC)C(C2CC2)C1)=CC 65452,c1(C(N2C(CC(N3CC(NC(N)=O)C3)=O)CC(O)C2)=O)ccc2[nH]nc(Cl)c2c1 65453,c1(C(=O)NCC2CC(OC)CN2C(c2ncc(Cl)cc2Cl)=O)cccc(N)c1C 65454,C1(NC(CSCc2ccc(C)cc2)=O)CC(NC(C2(C3CC3)CC2)=O)C12CCC2 65455,c1(C(=O)NCC2C(NC(CC=C)=O)CC2)ccccc1-c1nc(C)no1 65456,c1(C(N2C(CNC(CC(=O)NC)=O)CC(F)(F)C2)=O)c(C)nc2ncnn2c1C 65457,c1(OC)ccc(C(N2CCC3CCC23)C(=O)NCC2CCCO2)c(Cl)c1O 65458,C(C(C)(C)C(=O)N(CC(O)CN(C(=O)CN1CCS(=O)CC1)C)C)OC 65459,N1(C(CC2C(C)=NNC2=O)=O)CC2(C=C(C(=O)NCc3cccnc3F)CO2)C1 65460,c1(N(CC2C(C)N(C(=O)OC(C)(C)C)C2)C2CC2)cnc(-c2ccncn2)nc1O 65461,c1(C(=O)NC(C2(O)CCN(C(=O)C3=C(Cl)CC3)CC2)C)ccc(Cl)c(Cl)c1 65462,c1(CC)cccc(C(N2CCC(O)(CCNC(c3ccc(CO)o3)=O)C2)=O)c1F 65463,C(=O)(C(C#N)C(C)(C)C)N1CC(C(N2CC(SCC)C2)=O)C(F)C1 65464,N1(C(c2c(CC)ocn2)=O)CCCC(N(C(=O)CC2(O)CCCCC2)CCO)C1 65465,Cc1cc(CN2CCC2(C)C(=O)Nc2cc(F)c(F)cc2I)c(O)c(C)c1 65466,CC(C)(C)S(=O)(=O)CC(=O)NC1CN(C(=O)C(O)CC(F)(F)F)C1 65467,C1(NC(C2CC3C=CC2N(C(c2cnc(Cl)s2)=O)C3)=O)CN2CCC1(F)CC2 65468,C(=O)(C(C(C)NC(c1ccc2[nH]ccc2c1)=O)C(C)C)NCC(CC1CC1)OC 65469,Cc1cnc(C(=O)NC2CC3CC2N(C(c2nc(Cl)ccc2N)=O)C3)cc1C 65470,N1(C(C2(Cl)C(C)(C)C2)=O)Cc2[nH]nc(NC(=O)CNc3ccccn3)c2C1 65471,CC(C)(C)C(CNC(=O)C(C)(C)c1ccc(Cl)s1)NC(c1cn(C2CC2)nn1)=O 65472,c1(COC)nc(Cl)cc(=NCC2(O)CN(C(c3c(OC)ncnc3OC)=O)C2)[nH]1 65473,CCCCC(C(=O)NC(C(N1CC2(CCC(=O)NC2)C1)=O)C(C)OC)C(C)C 65474,CCC(CC(=O)NOCC(=O)NCC1CCC(=O)O1)CC(C)C 65475,c1(OC)cc(Br)ccc1C(c1nnnn1C(C)C)NCc1cccc(Br)c1 65476,c1(NC(C(N2CCC(C)(C)C2)=O)=O)ccc(F)c(S(=O)(=O)N(C)C)c1 65477,CCC1=NOC(CNC(C2CCC(NC(C3(c4cc[nH]n4)CC3)=O)CC2)=O)C1 65478,N1(C(COC(C)C)=O)CC2CCN(C(=O)CCCF)CC12 65479,C#CC(CNC(=O)CC1CCN1C(=O)CCc1cscn1)CC 65480,c1(C2(C(=O)NC3CN(C(c4c(C)[nH]cc4)=O)CC3F)CC2)ccc(Cl)c(F)c1 65481,N1(C(c2cc(CCC)[nH]n2)=O)CCC(C2CC2)C1CNC(=O)CSC(C)C 65482,c1(C(N(CC(CC)NC(c2occc2C)=O)C)=O)sccc1Cl 65483,c1(NCCC(CCC)O)ncc(C)cc1S(=O)(=O)NCC#CCCO 65484,c1(C(=O)OC)cccc(-c2nc(N(C(C)C)Cc3nnnn3C)n(C)n2)c1 65485,c1(CC(=O)NCC(CC(C)C)NC(=O)C2CC2)ccc(S(=O)(=O)N2CCCC2)s1 65486,Cc1oc2cc(C(N3CCC(C)N(C(=O)CC4(C)CCCO4)CC3)=O)[nH]c2c1C 65487,N1(C(C2N(CC)CCC2)=O)C2CCC(C(=O)Nc3ccc4occc4c3)C1CC2 65488,N1(C(C(C)SC)=O)CCN(C(c2cc3n(n2)CCN(C)C3)=O)CC(C)(F)C1 65489,c1(-n2cc(C3(O)CN(C(C4N(C(C)C)CCCC4)=O)C3)nn2)cccc2ccnn12 65490,C1(CN(C(c2nnc(-c3ccccc3)s2)C(=O)NCC(F)F)C)CCCSC1 65491,c1(C(N2CCC(F)(C(=O)Nc3c(OC)ccc(Cl)c3)C2)=O)cc(F)c(Br)cc1F 65492,CC(C(C)C(=O)NCC(F)F)NC(C1COC(=O)N1C)=O 65493,c1(C(=O)NCC(C(=O)NC(C)(C)CCO)CC2CC2)n[nH]cc1[N+](=O)[O-] 65494,C1(C(=O)NC23C(CN(C(Cc4ccn(CC)n4)=O)C2)C3)CN2CCN1CC2C 65495,C12(C(=O)NCC(CC)NC(c3cc4sccc4cn3)=O)C3CC(CC13)C2(F)F 65496,c1(CC(C)C)ccnc(NC(=O)CSc2ncccc2F)c1 65497,N1(C(C23CC(CN(C(C(CC(C)C)C)=O)C2)C3)=O)CC(C)C12CCOCC2 65498,Cc1cc(C(=O)NC2CN(C(=O)C#CC3CCCOC3)C2)cc(S(C)(=O)=O)c1F 65499,C(c1ccccc1OC)=CC(=O)NCC(=C)CCNC(c1cnsn1)=O 65500,c1(CC(N2CCC(O)(CNC(CCS(C)=O)=O)C2)=O)ccc2c(c1)OCO2 65501,CCN=c1ccc(C(N2CC3CC2C3CNC(C2OCCN(C)C2=O)=O)=O)c[nH]1 65502,CC1CN2CCN1CC2C(=O)NCC1CCCCN1C(c1cnco1)=O 65503,C(C)(C(=O)NC1CC1NC(=O)Cc1cncs1)OCC(C)C 65504,c1(C2(C(N(CC(C(=O)CCn3cnnn3)=O)CC)=O)CC2)ccsc1.OC 65505,C(=O)(C(C(C)C)C(C)C)N1CCCC(NC(CN(C2CC2)CC)=O)(CO)C1 65506,c1(C(C)=O)cn(C)nc1C(N1CCC(NC(=O)CC23CC(C2)C3)C1)=O 65507,c1(CC(N2CCCC(NC(C(CCC)NC(C)=O)=O)C2)=O)cc(Cl)cc(Cl)c1 65508,C(N=c1[nH]c2cc(F)cc(F)c2o1)C1CC(NC(C2C(S(C)(=O)=O)CCC2)=O)C1 65509,Cc1cnc(C(N2CCC3(CC3C(=O)NCCOCC(F)F)C2)=O)c(C)c1 65510,c1(CCC(=O)NCC2(CN(C(C3C(CC)CC3)=O)C)CC2)ncccn1 65511,c1(NCC(C)N(C)C(c2cc(F)c(CO)c(F)c2)=O)ncccc1S(C)(=O)=O 65512,C(C)(CS(C)(=O)=O)N(C(C1CCC=CO1)C(=O)NC1(C)CC1)CC 65513,C1(CC(=O)NC(C(=O)N(CCCOC)C)Cc2cn[nH]c2)CC(=O)NC1=O 65514,n1(CCC(=O)NCCC(C)NC(CC(=C)C)=O)c(=O)n(CC)c2ccccc12 65515,c1(OC)c(C(=O)NC(C)(CNC(c2cnc(CC3CC3)s2)=O)CO)csc1Cl 65516,CC1C(NC(C2CCCCC2O)=O)CCCN1C(C1CC(=O)N1)=O 65517,CNS(=O)(=O)N1CCN(Cc2ccc(OCC(F)(F)F)nc2)CC1 65518,N1(C(C(CC)OC)=O)Cc2occ(C(=O)NC3CC4C=CC3CC4)c2C1 65519,c1(CC)cccc2c(C(=O)NCC(C)NC(=O)C(C)(C)C3CCOCC3)c[nH]c12 65520,c1(C(=O)NC2(OC)CC3(CCCC3)C2)c(N(C)C)c(O)nc2ccccc12 65521,CC(C)C(CO)C(=O)NC1CCC1NC(=O)CN1CCC(CO)CC1 65522,C1(C(=O)NC(C(=O)OC)(C)C)COCCN(C(C2CCC(C#N)CC2)=O)C1 65523,N1(C(C2C(C#N)CC2)=O)CCCC(CCC(=O)NC2(C(F)(F)F)CC2)C1 65524,CN1CC=C(CC(=O)N2C3CCCC2CC(NC(=O)CC2(C)CCCO2)C3)CC1 65525,CCC(C)(C)C(O)C(=O)N1CCC(C(C)(C)NC(C2CC3(CCCO3)C2)=O)C1 65526,C1(C(C)C)(C(=O)NCCN2CCC(CO)C2)CCCN1C(=O)CN1CC(C)(C)C1 65527,c1(C(=O)NCC2CCN2C(c2cccc(F)n2)=O)ccc2cc[nH]c2c1 65528,C1(C(=O)NC(CNC(c2cc(CC)on2)=O)C2CC2)(COC)CCCNS1(=O)=O 65529,c1(C(N(CCNC(C(CC#C)C)=O)CC)=O)n[nH]c2ccc(F)cc12 65530,N1(C(c2cn(C)nc2)=O)C(C(=O)NC2CC(=O)NC2=O)CCC12CC2 65531,N1(C(=O)C=Cc2ccoc2)CCC2C(CCN2CC(O)CCc2ccccc2)C1 65532,C1(CC(N2CCCC(CCNC(=O)CC3OCCCO3)C2)=O)CN2CCN1CC2 65533,C1(C(N2CCCC(NC(C3C(c4n(C)ncc4)C3)=O)C2)=O)CCS(=O)(=O)CC1 65534,Cc1cc(C(=O)NC(C2CCOC2)CNC(c2cc(CO)n(C)n2)=O)ccn1 65535,C(C)(C)(CC(=O)NOC1CCOC1)N(C(=O)CC1CCCO1)C 65536,Cc1cc(C)c(NC(=O)C(C)C(C)NC(=O)CCC2CCCCC2)cc1C 65537,CCC(C(=O)N(C(C)CN(C)C(c1cnn(CC)c1)=O)C)N(C)C 65538,Cc1sncc1C(=O)NCCCNC(C1CC1(C)C)=O 65539,c1(-c2c(F)ccc(C)c2F)cccc2c1CCN(C(c1c(C)cccc1C)=O)C2 65540,C1(C(N(CC(C)OC)C)=O)(OC)CCN(C(c2ccc(Br)cc2F)=O)CC1 65541,c1(C(C)C(=O)NC2(C(=O)O)CC3(CNC3)C2)cnc2n1CCCC2 65542,CC1C(NC(c2nn(C(F)F)cc2Cl)=O)CCCN1C(=O)C(C)CC1CC1 65543,S(=O)(=O)(CC(=O)N1CCC(C)C1CNC(c1cccc(NS(N)(=O)=O)n1)=O)NC 65544,c1(C(=O)NCC(CC(C)C)NC(=O)C2=C(Cl)CCC2)ccc2c(c1)CCCC2=O 65545,c1(C(=O)NC2CC(C)(CNC(C3CCN(CC)C3)=O)C2)cc2cncn2c(O)n1 65546,N1(C(C(N2CCOCC2)C)=O)CCCC(O)(CNC(=O)C2=CSCCO2)C1 65547,CC1CC(C(=O)OC(C)(C)C)CN(C(=O)C(=O)NC(C)(C)C)C1.C1(=O)CCO1 65548,CC(C)C(CCN(C(=O)CC1COC(=O)C1)C)N=c1nc(-c2ccccc2)[nH]s1 65549,N1(C(CCC(C)OC(F)F)=O)CC2(CCCN2C(c2sccc2N(C)C)=O)C1 65550,c1(CSC)nsc(N(C)C(C2CCC(F)C2)=O)n1 65551,c1(CC)nc(C)c(C(N2CCCCC2CNC(c2cnn(C)c2Cl)=O)=O)c(C)n1 65552,N1(C(c2csc(Br)n2)C(=O)NC2(C)CC2)CCCCC1CCn1ccnn1 65553,C(N=c1ccc(C(N2CCCC(Br)C2)=O)c[nH]1)c1ccc(N(C)C)cc1F 65554,N1(CC(=O)NC(C2CCOC2)CNC(C(C)(C)C2CC2)=O)Cc2ccccc2C1 65555,N1(C(C(c2ccnn2C)NC(C(C(C)C)NC(C)=O)=O)=O)CCN(C)CC1C 65556,n1(CC)cc(NC(C2(CNC(C3C4CC5C(C4)C35)=O)CC3(CC3)C2)=O)c(C)n1 65557,N1(CC)CC(C(=O)NC(CCC2CC2)C(=O)NCC2(CC3CC3)CCC2)CC1=O 65558,N1(C(c2c(C)nn(CC)c2C)=O)CC(NC(c2n[nH]c(C)c2F)=O)C2(CCC2)C1 65559,Cn1cc(-c2cn(CC(C3CN(C(=O)CNC(=O)ON)C3)F)nn2)cn1 65560,N1(C(c2cc(C)sc2C)=O)CCC(CNC(=O)CCOCCN(C)C)C12CC2 65561,C1(CCC)CN(C(=O)Cn2cc(Cl)cn2)CCN1C(=O)CN1CCC(C)(C)C1 65562,CCC(CC)C(CNC(=O)C1CC1)N1CCC(c2cccc(F)c2F)C1 65563,N1(C(C=C(C)c2ccccc2F)=O)CCCCC2(CCN(C(C3CCO3)=O)C2)C1 65564,c1(C(N2CC3CC(NC(C4(C)CCN(C)CC4)=O)C3C2)=O)n[nH]c2c1COCC2 65565,CC1=NOC2(CCN(C(C3CSCCN3C(=O)OC(C)(C)C)=O)CC2)C1 65566,C1(Nc2ccc(C(=O)OC)cn2)(CNC(=O)Cn2ccnc2)CCCCC1C 65567,c1(C(C(=O)OC)NCC(=O)NCC(=O)Nc2ccccc2)cc(Cl)ccc1Cl 65568,c1(NC(c2c(C)nc(C(=O)Nc3c(C)nsc3)s2)=O)ncc2[nH]ncc2n1 65569,C(C(=O)N1CCOC(CC)C1)(C(C)(C)O)NC(C(C=C)C)=O 65570,C=CCCN=C(NCC1(F)CCC(CO)CC1)NCC1CCC(C(=O)OC)O1 65571,C1(NC(c2cnc(C3CC3)nc2)=O)CCCCC12CCN(C(=O)C=CI)C2 65572,c1(CC(=O)N(CCCNC(C2C(CC)OCC2)=O)C)ccc(O)cn1 65573,C=CCC(CC)C(=O)N1CCCC(NC(=O)CCOC(C)C)C1C 65574,C(=O)(CCCCC1CC1)NC1(CC)CN(C(C(C)OCC#C)=O)C1 65575,C1(CNC(C2N(CC)CCC2)=O)CN(C(C2CC(N(C)C)C2)=O)CCN1C 65576,c1(N(C(=O)Cn2cc(C(C3CCCNC3)C)nn2)C2CC2)ccnc(OC)c1.CO 65577,N1(C(C(CCC)OC)=O)C2CCC1CN(Cc1nc(C(C)OC)no1)CC2 65578,N1(C(c2cc(C)sc2)=O)C2CCC(C(=O)NCc3cncc(Cl)c3)C1CC2 65579,c1(C(N2CCCC(NC(C(CC)(C)O)=O)C2)=O)ccc(OC(C)C)c(Cl)c1 65580,CC1CC(NC(=O)CCP(C)(C)=O)CN(C(=O)COc2ccc(Cl)nc2)C1 65581,N1(C(C=CCC)=O)CCN2CCOCC2(CNC(C2COCCO2)=O)C1 65582,c1(C(=O)NCC(C)NC(c2nnc(CN(C)C)s2)=O)ccccc1C1CC1(F)F 65583,N1(C(C(CSC)O)=O)CC2(CCCC2NC(=O)Cc2ccnc(F)c2F)C1 65584,CC(C)C(C)(C)C(=O)NC1CC(CNC(C2(C)CC3CCC2C3)=O)C1 65585,Cc1ncccc1CCC(=O)NCC1(O)CCN(C(C2CCCC2)=O)C1 65586,CON1CC(NC(=O)N(CCC(=O)OC(C)(C)C)C)CC1=O 65587,CON(CCC(=O)N1CCC2CC2C1)C(=O)Cc1ncoc1C 65588,C1(NC(CN(C2CC2)CC)=O)CC2CN(C(c3nc(OC)c(C)s3)=O)CC2C1 65589,C1(NC(C(F)=C(C)C)=O)CCCC1CNC(=O)CC(=O)NC1CC1 65590,O=C1NCc2cc(CNc3onc4ccccc34)ccc21 65591,c1(OC)cccc(C(C(=O)NC2CC(NC(c3sc(C)cc3Cl)=O)C2)OC)c1 65592,N1(C(C(C)NC(C(C)NC(=O)NC)=O)=O)CC(S(C)(=N)=O)C1 65593,c1(C(=O)NCC2(O)CCN(C(C3CC(C)(F)C3)=O)C2)cc2cccnc2cc1F 65594,c1(-c2ccc(F)c(F)c2)ccc(NCc2cnco2)c(F)c1F 65595,C(=O)(C1=NN2CCCN=C2N1)N1CCC(C2CC2)(C(=O)O)C1 65596,c1(OC)ccc(C=CC(=O)NC2(CO)CN(C(=O)Cc3ccno3)C2)c(OC)c1 65597,C1CC(=O)NCC2CC(C2)C(=O)N1CC=C.C1(SC)CC1(C)C 65598,c1(C(=O)NC2(C)CCN(C(C(C)C#N)=O)C2)cncc(S(C)(=O)=O)c1 65599,CC(C)C(C(C)NC(=O)CCC(F)F)NC(=O)C=C1CCCCC1 65600,Cc1cc(O)ncc1C(N1CC(C2CC2)(C(=O)NCC2CC(C#N)C2)C1)=O 65601,Cc1ccc(C(=O)NC2CC(O)CN(C(c3ccc[n+]([O-])c3)=O)C2)c(N)c1 65602,C1(NC(CC2(OC)CCOCC2)=O)CCC2(CC1)CN(C(=O)C(C(C)C)SC)C2 65603,c1(C(F)(F)F)nc(NC2C3CCCCCC23)cc(=NC2CC(n3cncn3)C2)[nH]1 65604,N#Cc1ccc(C(O)C(=O)NC2CC(NC(=O)C(F)=CCCF)C2)cc1 65605,N1(C(=O)Cc2nccs2)CC2CC2(CNC(C2(N3CCCC3)CCC2)=O)C1 65606,C1(C(=O)Nc2cccc(NC(C(CC)(C)CC)=O)c2)CC2CCCCN2C1 65607,C1(CNC(c2cc(C)n(C(F)F)n2)=O)CN(C(=O)Cc2ccon2)C2CCN1C2 65608,C1(NC(c2c(C)coc2)=O)CCCC1(C)CNC(c1ccoc1Cl)=O 65609,c1(CC(=O)NC2CC(N(C(c3c[nH]c(=NC)o3)=O)C)C2)c(OC)cccc1Cl 65610,C1(NC(C(C)c2ccsc2)=O)CC2CCC1N2C(=O)COc1ccc(F)cn1 65611,C1(C(=O)NCCOCC(=O)NCC(COC(C)C)O)CNC(=O)N1 65612,N1(C(Cc2nn(C)c(Cl)c2)=O)CCC(NC(=O)COCCN(C)C)C12CCC2 65613,C#CC1(O)CCCN(C(=O)COCCNC(c2ccsc2)=O)C1 65614,C(=O)(C#CC1CCCCO1)NCCCC1OCCN(C(c2c(C)nc(O)[nH]2)=O)C1 65615,CC1(C)C(CNC(=O)C(=O)NCC2(C)COC(=O)N2)CCS1(=O)=O 65616,[N-]=[N+]=NCCC(=O)NC(C(=O)NCC(F)Br)C1CC1 65617,Cc1cnn(CC(N2CCC(C)(CCNC(=O)COCC3CCC3)C2)=O)c(=O)c1 65618,Cc1ccc(C(N2CC(N(C)C(c3ncn4c3CCCC4)=O)C2)=O)c2c1CCC2 65619,c1(C(N2CCCC(NC(c3n(C)c(S)nn3)=O)C2)=O)cccc(F)c1O 65620,C(CC(=O)NOCC1CC1)(c1ccccc1)NC(C1(CC)CCCO1)=O 65621,N1(C(c2cncc(C)n2)=O)CCCC2C(CCCN2C(=O)COCC(C)(C)C)C1 65622,C1(CNC(C=CC=CCC)=O)CCN(C(=O)C(=O)C2CCCC2)C12CCC2 65623,N1(C(C2(C)CC2)=O)CC2(CC2)CC1CNC(C1CC2(CCC2O)C1)=O 65624,Cc1cc(C(=O)NC(CO)C(C)NC(=O)C(O)Cc2ccccn2)c(Cl)cn1 65625,c1(CNC(c2ccn(CCC(F)(F)F)n2)=O)csc(CNC(C2CCOC2)=O)n1 65626,C=CCC(CC=C)C(=O)NCC1CCCN(C(C2(OC)CS(=O)(=O)C2)=O)CC1 65627,C(=O)(C1CCCc2nncn21)NC1CC(NC(C2(C)CCSCC2)=O)C1 65628,N1(C(C(COC)(F)F)=O)CCN2C(=O)C(NC(c3cnn(C(C)C)n3)=O)CC2C1 65629,O=C1CC(CC(=O)Nc2ncc(C3COC3)s2)c2ccccc2N1 65630,c1(C(C(=O)NCC(CNC(CNS(CC)(=O)=O)=O)C)=O)ccccc1 65631,C(=O)(CC1=CCOCC1)NC1CN(C(CCOCCCOC)=O)C1 65632,c1(C(N(CCNC(=O)C=CC=C(Cl)Cl)CC2CC2)=O)cccc2nccn12 65633,C(c1cnc2ccccc2n1)=CC(=O)NC(C)(CNC(c1ccnnc1)=O)CO 65634,c1(CN2CCC(C(=O)NCCC(=O)OCC)CC2)cc(C(F)(F)F)cc(Cl)c1F 65635,CCC(=O)CCC(=O)N1CCOCC1CCNC(=O)CCc1cccc(C)c1 65636,C1(C(N2CCC(C(C)(C)O)C2)=O)(SC)CN(C(=O)Cc2ccccc2)C1 65637,Cc1ccc(C(N2CCC3CCCC23CNC(c2csnn2)=O)=O)c(=O)n1C 65638,CC1CN(C)CC(C(=O)NCC(C2CC2)N(C)C(c2nccnc2N)=O)O1 65639,c1(CCC)n[nH]c(=NCC(C)(C)NC(c2cnc(O)nc2O)=O)s1 65640,Cc1ncsc1C=CC(N1CCC(N(C(=O)C(C)CF)C)C1)=O 65641,N1(CC(Cn2cnc(C(=O)OCC)n2)O)CCc2ccccc2C1 65642,Fc1ccc(CCCNCc2csc(-c3ccccc3)c2)cc1 65643,N1(C(CC(C)OC)=O)CC(C2(NC(=O)Cc3ccc(Cl)cc3C(F)(F)F)CC2)C1 65644,S(=O)(=O)(c1cc(F)cc(Br)c1)NC1CC(C(=O)NCC2CCCCC2)C1 65645,Cc1ccc2nc(C(=O)NCC3CCCC3NC(=O)COCCO)ccc2c1 65646,N1(S(C(C)C)(=O)=O)CCN(CCCNC23CC(C(F)(F)F)(C2)C3)CC1 65647,N1(C(CSc2c(C)cccc2)=O)CC2(CCN(C(=O)C=CC(C)C)CC2C(=O)O)C1 65648,C1(C(=O)NCCN(C(=O)COC)CCC)C2CCC1(c1ccco1)C2 65649,C(=O)(C(C)(F)C(=O)NCC1(NC(=O)Cc2nc[nH]n2)CC1)OC 65650,CS(=O)(=O)C1(C(=O)NCC2(CCNC(C3CC(N=[N+]=[N-])C3)=O)CC2)CC1 65651,c1(C(CO)NC(C2OCCC(C)C2)=O)cccc(Cl)c1F 65652,C(=O)(C(C)(C)C)NCC(=O)NC(C)CN(C)C(C1CC(=C2CC2)C1)=O 65653,N1(C(c2cc(F)ccc2F)C(=O)NCCSC)CCN(C)C2(CC2)C1 65654,N1(C(=O)C=CC2CCCC2)CCOCC(NC(=O)C(F)(F)Cl)C1 65655,C(C1=CCCN(C(c2cnncc2OC)=O)C1)NC(C(C=C)OC)=O 65656,C1(NC(c2c(C)n[nH]c2)=O)CCCCCN(C(=O)C(O)C(C)(C)C)C1 65657,c1(C(N2C(CNC(=O)Cc3cncnc3)CC2)=O)ccc2c(c1)NCCC2 65658,C1(C(=O)NCCn2c(CC)ncc2)CC(C)CN1C(C1CCCC(C)C1)=O 65659,Cc1n[nH]c(C)c1CC(N1CCC(c2ccccc2)(NC(C2CC23CC3)=O)C1)=O 65660,N1(C(c2c(C)n(C3CC3)cc2)=O)CCCN(C(C23CCCC2(C(N)=O)C3)=O)CC1 65661,CCCC(C(O)C(=O)N1CCC1C(C)O)NC(c1c(F)cncc1F)=O 65662,N1(C(CCCC#C)=O)CCCCCC1CNC(c1cc(C)nnc1CC)=O 65663,N1(C(C2NCCN(C(c3scc(C)c3C)=O)C2)=O)CCCC(C)(O)C1 65664,N1(C(C(=O)NCc2ccc(-c3ccc(Cl)cc3)cc2F)=O)CCC2CCC(C1)O2 65665,C(=O)(C1=CC2(CCOCC2)C1)NCCC1(O)CCN(C(C(CC)(C)F)=O)C1 65666,c1(C(N2CC(NCc3ccc(C#N)cc3)C3(C2)CC3)=O)c(Cl)ccc(Cl)c1F 65667,c1(C(c2nnnn2CCCSC)NCC(=O)NCCC)cccc(OC)c1F 65668,N1(CCC)CC(C(=O)N(C(C)CN(C(=O)CCc2cccnc2Cl)C)C)CC1=O 65669,Cn1ccnc1CCCNC(=O)C(N)Cc1ccoc1 65670,C(=O)(C(C)CC(F)(F)F)NC(CC(C)C)CNC(=O)C1=CCSC1 65671,N#Cc1c(F)cc(NC(N2CCN(CC3CC3)CC2)=O)cc1Br 65672,CC1C(NC(=O)CN(C)S(=O)(=O)N(C)C)CCCN1C(=O)CN1CCCCC1 65673,CC1CC(NC(=O)Nc2ccccc2SCC(N)=O)CCN1CC(N)=O 65674,C1(C(N(CC#C)CCF)=O)(CC2CC2)CN(C(=O)CC2CCC(C)C2)C1 65675,CON1CC(C(=O)NC(C(N2CCC(C)(CCO)C2)=O)c2ccco2)CC1=O 65676,C(=O)(C(CC#CC)NC(=O)COc1ccn(C)n1)N1CC(CC#C)OCC1 65677,c1(CCC(=O)NC2CN(C(C3(COC)CC3)=O)C2)ccccc1Br 65678,N1(C(C2(COCC)CC2)=O)CCCCC(N(C)C(C2CCCC2(F)F)=O)C1 65679,c1(C(N(C2CCN(C(C3(C)ON=C(C)C3)=O)CC2)C)=O)c(Cl)ccc(F)c1N 65680,CC(CCCCNC(=O)CC1CC(=O)C1)NC(=O)C(C)CCOc1ccccc1 65681,C#Cc1ccc(CC(=O)N(C2CN(C(=O)CC(C)OC)CCC2O)C)cc1 65682,n1(Cc2nc(C)on2)nnc(NC)c1C.C1(N=[N+]=[N-])(C=O)CC1 65683,Cc1ccc(C=CC(=O)NCC23CCCC2CCN3C(=O)COC(C)C)cc1C 65684,C1(CNC(c2c(C#C)c[nH]n2)=O)CC2CN(C(=O)CC(F)(F)F)CC12 65685,c1(C(N(C(C)CNC(c2cc(O)nc(O)c2)=O)C)=O)ccc(F)c2ccncc12 65686,Cc1cc(Cl)c(Br)cc1S(=O)(=O)NC1Cc2ccccc2N(C)C1=O 65687,c1(C(=O)NCC(CNC(=O)C(F)(F)c2nccs2)OC)cccc(F)c1N 65688,c1(C(=O)NC(CNC(CC2N(C)CCCC2)=O)C2CC2)cccc2c1COCC2 65689,CC1CCCC1CC(=O)NCC(C)(F)CNC(=O)Cc1cccs1 65690,C(CS(=O)(=O)CC(=O)NCC(C)(CNC(c1c(C)ncn1O)=O)OC)OC 65691,C(=O)(CCCCSC)NC(C(=O)OC)C1CN(C(C2(C(=O)N(C)C3CC3)CC2)=O)C1 65692,c1(NC(C(=O)NCCC(OCC)OCC)=O)cc(C)n(-c2ccc(Cl)cc2)c1C 65693,c1(OC)ccc(C(C)C(=O)N(CCCCCNC(=O)CC2CSC2)C)c(C)c1 65694,c1(C(N2CCN(CC3CN(C(=O)CCC4CC4)C3)CC2)=O)ccc2nc[nH]c2n1 65695,C(=O)(C(C)(C)CCC#N)N1CC(C(N(c2ccc(F)cc2)C)=O)C2(C1)CC2 65696,c1(C(N(C(C)CNC(=O)C=Cc2ccnn2C)CC)=O)ccc(C(C)C)cn1 65697,C1(C(C)NC(C(C)(C)NC(=O)NCC)=O)CCCN(C(=O)Cc2[nH]cnc2C)C1 65698,CCC(CC(=O)NC1CC2CCC1CC2NC(c1cn(C)[nH]c1=N)=O)C(C)C 65699,FCCCCCCNC(c1nnnn1C1CCCC1)c1ccon1 65700,c1(-c2cccc(NC(C3N(CC)CCCC3)=O)c2)cnn2c1NCCC2 65701,CN1CCC(F)(CNC(=O)C(C)(CO)NC(=O)CC2CNC(=O)O2)C1 65702,CC1OC2(C(=O)NC3CC(NC(C4(C)COC(=O)C4)=O)C3)CC1C2 65703,C1(O)(C(CNC(C(C=C)C)=O)C)CCN(C(C2CCS(=O)CC2)=O)C1 65704,Nc1ccc(-c2nc(C(N3CCCC3)=O)n(-c3ccnc(Br)c3)n2)nc1 65705,CCCC(CNC(=O)CC(C)n1cccn1)C(=O)NC1(C2(OC)CCC2)CC1 65706,c1(CC(=O)NC2CC(CNC(C(CCC)NC(C)=O)=O)C2)ccc(CO)c(C)c1 65707,C=CCCCCCCCC(=O)NC(C1CCN(C(=O)CCC(=C)C)C1)(C)C 65708,c1(C(N2CCC(C(=O)NCCNC(CCC#C)=O)CC2)=O)cccc2nncn12 65709,C1(C(N2CCOCC2)=O)(NC(C=C(C)C)=O)CCCCC1.c12cccc(c1)C2 65710,N1(CCc2cccc(C(=O)NC)c2)CCC(=O)N(Cc2ccc(F)cc2C)C1=O 65711,C1(NNC(C(=O)CCN(CC(F)F)CC2CC2C2CCCO2)=O)CCS1(=O)=O 65712,CN1CCc2[nH]nc(C(=O)NCC3CC3CNC(=O)C3=C(Cl)CCC3)c2C1 65713,c1(N2CCC(CNC(C3C(C(C)C)(C(=O)O)C3)=O)C2)ccc(Br)cc1 65714,N1(C(=O)CC2CC3(CCC3)CO2)CC2CN(C(C34CCC(CC3)CO4)=O)CC2C1 65715,N1(C(C(C(C)C)C#N)=O)CCc2nc(CNC(=O)CCn3ccnn3)sc2C1 65716,c1(C(=O)NC(CO)C2CC2)cnn(-c2cccc(F)c2)c1C(F)F 65717,Cn1cnc2c1CCCC2C(=O)N1CCC(CCNC(c2ccon2)=O)C1 65718,C1(N(C(=O)CC=C(C)C)CCC)CCN(C(=O)CC2COCC2O)C1 65719,c1(N(C)Cc2nc(CC)sc2)cc(C)c(S(=O)(=O)N2CCCC(C)CC2)cn1 65720,C1(C(=O)NCCC2CCOC2)CC2(CC2)CN1C(=O)C=CC(F)F 65721,C=CCC(C)(C)CC(c1nnnn1CCSC)NC1CC(C)C1 65722,Cc1nnc(CCCN(C)C)n1C.c12ccc(cc1)CCC(=O)NC2C 65723,N1(C(CS(CCC)(=O)=O)=O)CCC2CCN(C(C3CCCSC3)=O)C2C1 65724,c1(C(N(CCCOCCN(C(C=CC(CC)C)=O)C)C)=O)cn(C)nc1Cl 65725,C1(Cc2cn(CCC=C)nn2)CCCCN1C(c1scnc1C(C)(C)C)=O 65726,c1(C(=O)NCC2CCCC(NC(CCN(C)CC)=O)C2)ccc2ncccn12 65727,N1(C(C(C2CCOC2)NC(CCCCC)=O)=O)CC2(CCC(=O)NC2)C1 65728,c1(C(N2C3CN(C(C(C)C4CCC4)=O)CC2CC3)=O)c(Cl)c([N+](=O)[O-])nn1C 65729,CC1=NOC(C(=O)NC(CNC(C2CC(NS(C)(=O)=O)C2)=O)CC(C)C)C1C 65730,N1(C(c2c(C)nc(COC)s2)=O)CCC(C2CC2)C1CNC(C1CC1C(C)O)=O 65731,c1(CCC(=O)NCC(CN(C(c2nc(CCC)sc2)=O)C)O)nnc(S)nc1O 65732,n1(CC(=O)NC2(CCNC(C(C(COC)C)C)=O)CC2)nnc2ccccc12 65733,N1(C(c2cnc(OC)s2)=O)CCCCC1CNC(=O)CCc1cc(Cl)cs1 65734,c1(C(=O)NC2CC3(CN(C(C(C(C)C)C)=O)C3)C2)ccc2c(c1F)CCC2 65735,CCC(C)(C#N)C(=O)N1CCC(NC(c2cc(Cl)ccc2OC(C)C)=O)CC1 65736,c1(-c2ccc(C)c(F)c2)ccccc1S(=O)(=O)NCC(O)CN(C)C 65737,N1(C(C(CC)N(C)C)=O)CC(NC(C23CCC(CC2)CO3)=O)CCC1C 65738,N1(C(=O)CC(C2CC2)C2CC2)C(C(=O)NCc2nccs2)CCC1C1CC1 65739,C1(C(=O)NCC2(OC)CN(C(c3coc(C4CCC4)n3)=O)C2)CC(C)OC1C 65740,c1(COC)cc(C(=O)NCC(c2cccc(C)c2)NC(C2CC2(F)F)=O)c(C)o1 65741,C1(C(=O)NCC(C(CC)C)(C)O)CC(C)(C)CCN1C(=O)Cn1nccn1 65742,c1(C(N2CCOCC(C)C2)C(=O)NCCC2(C)CC2)ccc(F)c(Br)c1F 65743,C1(C)(C(N2CC(N(C(=O)CCCF)C)C(O)C2)=O)CCC2(CC1)OCCO2 65744,c1(OC)nn(C)cc1C(=O)NCC1(C)CCCN1C(C1CC1c1ccccc1)=O 65745,C(CC(=O)N1CC2(CSC2)C1)(C(F)(F)F)NC(=O)C=CC1CCOC1 65746,Nc1cc(F)cnc1C(=O)NC(CCOCCO)C(=O)NCC(O)C(F)F 65747,c1(C(N(CCCN(C(=O)Cc2ccc(F)c(Cl)c2)C)C)=O)nc2cnccc2s1 65748,CN=c1[nH]c(C(=O)NCC2CCCCN2C(c2cn(C)cn2)=O)cs1 65749,N1(C(CC2N(CC)CCC2)=O)CC2(CC(NC(=O)CC34COCC(C3)C4)CO2)C1 65750,Cc1cc(Br)c(F)cc1C(=O)NC1CC(NC(=O)CCOC(C)C)C1 65751,C1(OCC)CC2(C1)CC2C(N1CC(OCCNC(=O)CN2CC(OC)C2)C1)=O 65752,C#CC1(C(N2CCOCCC2C)=O)CCN(C(=O)CCC(=O)CC)CC1 65753,CC1CCCC(CC(=O)NC(C2CCN(C(c3ccn(CCF)n3)=O)CC2)C)O1 65754,c1(C(=O)NCC(c2ccccc2)CNC(CSC)=O)cc(C2(O)COC2)on1 65755,C(C(CNC(c1cc2n(n1)CCC2)=O)C(F)(F)F)NC(CSCCOC)=O 65756,C1(C(=O)NCC(C)NC(C2C(=C)C2)=O)CC1(C)C 65757,C1(C(=O)NC(CC(C)C)CO)CC12CCN(C1CCC(=O)N(C3CC3)C1=O)CC2 65758,CN=c1cc(C(=O)NC2CC(C)N(C(c3cncc(OC)n3)=O)C2)cc[nH]1 65759,N1(C(=O)CCc2cccnc2)CC2(C1)CN(C(C1(CCO)CC1)=O)CCO2 65760,c1(C(c2nnnn2C2CC2)NC(C=C)C2CCC2)cn(C)nc1C(F)F 65761,CCC(C(=O)Nc1cccc(C(C)(C)C)n1)C(C)C 65762,C1(CNC(=O)C(N2CCN(c3ccc(F)cc3F)CC2)=O)CCc2cncn2C1 65763,Cc1ccc(C(c2ccncc2)NC(=O)NCC2CC2c2nn[nH]n2)cc1 65764,C1(NC(C=CC(C)(C)SC)=O)COCCC1NC(=O)C(C)(O)C1CC1 65765,c1(C(=O)NC2(CCOC)CCN(C(=O)C3=CCCO3)C2)cc(Cl)ccc1C 65766,C1(CN(C(C2C(C)C2C)=O)C)CCN(C(C2(c3ccccc3)CCCO2)=O)CC1 65767,C1(CNC(c2ccc(Br)o2)=O)CCC2(CN(C(c3c(O)cccc3F)=O)C2)O1 65768,CC1CCCC1C(N1CC(C)(CNCc2ccc(Cl)s2)C1)=O 65769,C1(CC23CN(C2)C3=O)CCCS(=O)(=O)C1.C1(C(=O)OCC)CCCC(C(N)=O)C1 65770,Cc1ncncc1C(=O)NC(C1CC=CCC1)C(=O)N(C1CCN(C2CC2)C1)C 65771,C1(N(C(=O)CC2CCC2)CCC)CCN(C(=O)CCc2ccn(C)n2)CC1 65772,C(=O)(C(C)=NOCC#N)NC(COC)C(=O)NCC(O)(COC)CO 65773,N1(CC2CCN(c3n(C)ccn3)C2)CC(=O)N(Cc2cn(CCCF)nn2)C1=O 65774,N1(C(CC(=O)NCC)=O)CCCC1(C)C(=O)NC(C1(OC)CCC1)C 65775,Cc1cc(=O)oc(C)c1C(=O)NCC1CC1NC(=O)Cc1ccccc1Br 65776,C1(F)(C(N2CCC(C)(CCNC(C3(C#C)CCC3)=O)C2)=O)CCCN(C)C1 65777,c1(C(=O)NCCCN(C(=O)C(C)(O)C2CCOC2)CC)scnc1Cl 65778,c1(C(=O)NCc2cccc(CNC(C3(CC)CC3)=O)c2)cnc(Cl)cc1Cl 65779,CCCC(CCC)C(=O)N1CCC(C(=O)NC(C)CC(C)C(F)F)O1 65780,C1(CCNC(C2CC(=O)NC2)=O)CCCCN1C(=O)CCNc1ccccc1 65781,c1(OCCC(=O)NCC(C)CN(C)C(C2CC(F)C(=O)N2)=O)cccc(Cl)c1 65782,c1(NC(C)CCCNC(=O)OC(C)(C)C)ccc(F)c(C=O)c1 65783,N1(C(C(N2CCN(C)CC2)C)=O)CCC(C2CCCN(C(C3(CF)CC3)=O)C2)C1 65784,C(CC(F)F)(C(=O)NCCN1CCCCC1C)NC(CC=C)=O 65785,c1(C(=O)NCC(CNC(c2oc(C)nc2C)=O)OC)ccc(C(C)C)nc1O 65786,N1(C(c2nnc(C)o2)C)CCC(NC(c2cccc(F)c2Cl)=O)C(C)C1 65787,C(CNC(c1cncnc1)=O)(CC(F)(F)F)NC(c1cnc(SC)s1)=O 65788,C=CC(C)(CC)C(=O)NCCOCCCNC(c1ccc(CCCCC)o1)=O 65789,n1(C(C)C)cc(Br)c(C(=O)Nc2ccccc2CC2NC(=O)NC2=O)n1 65790,c1(C(=O)OC)cccc2c1CN(C(C1C3CCC1N(Cc1ccccc1)C3)=O)CC2 65791,c1(C(=O)NCC2(NC(C3CC(C)OC3)=O)CCCCC2)cc2n(c1)CCOC2 65792,C1(NC(c2cccc(C)c2)=O)CC2(C1)CN(Cc1cc(O)ncc1Br)C2 65793,C(=O)(CC(CC)CC)NC(CCC)CNC(=O)CC(C)OC 65794,C1(CC)CN(C(=O)Cc2occc2C)CC1NC(c1ccc(SC)cc1)=O 65795,C12CCN(C1)C(=O)CO2.c1(SCCNC(C2CC(=C3CCC3)C2)=O)cccnc1 65796,Cc1c(C(=O)NCCC2(C(=O)NC3COCCN(C)C3)CCC2)cncc1F 65797,CCC(C)CC(C)C(=O)NCC(C(C)C)NC(c1n[nH]c(C)c1Cl)=O 65798,c1(C(=O)NC2CCC(NC(C(CC)n3ccnc3)=O)C2)ccc(F)c(C)c1O 65799,Cc1cnc2n1CC(C(=O)NCC(F)CNC(c1csc(Br)c1)=O)CC2 65800,C(=O)(CCP(C)(C)=O)NC(C(=O)NCC#CCOC)CCOC 65801,c1(NC2C(C)C2)ccc(Cl)c(C(=O)OCC2CCCO2)c1.N12CC(C1)CC2=O 65802,c1(N(C(c2ccc(Br)cn2)C(=O)NC2COC2)C)cccc(Br)c1F 65803,C(=O)(CCC(O)C(C)(C)C)NCC(C)CNC(c1csc(=N)[nH]1)=O 65804,Cc1cc(C)c(C(N2CCCC2C(=O)NC2CC2)C(=O)NC2CCCC2)cc1C 65805,N1(C(c2c(C)con2)=O)CCC2(CCCN2C(=O)C=CBr)C1 65806,N1(C(c2cc(CC)nnc2C)=O)CCCC12CCN(C(c1cc(Cl)ccn1)=O)C2 65807,Cc1nnnn1C(=O)NC1CCN(C(c2ccc(NC(=O)OC(C)(C)C)o2)=O)C1 65808,c1(C(=O)NC2COCC2CNC(C2CCC(=O)N2C2CC2)=O)nnc(O)nc1O 65809,CC1CCCC1NC(=O)C#CCNC(=O)COCc1nc[nH]n1 65810,Cc1cc(C(N2CCC(C)C(CNC(=O)CC3(C)CCOC3)C2)=O)cc(C#N)c1 65811,c1(C(N(C(CNC(C2(C(=O)OC)CC2C)=O)C2CC2)C)=O)ccc(F)cn1 65812,C(c1ccc(C)c(Cl)c1)=CC(=O)NCC1CN(C(CC(=O)NCC)=O)CC1(F)F 65813,Cc1cccc(CC(=O)NCCCNC(=O)CN2CCNC2=O)c1Cl 65814,C(=O)(C(CCC)CC(C)C)N1C(CC(=O)NC2(C#C)CC2)CC(F)C1 65815,C(=O)(C1CCCc2n[nH]cc21)N1CCC(COC)(NC(c2c(C)ncn2O)=O)C1 65816,C1(C(=O)NC(C(C)(C)NC(CC=CC=C)=O)C)C(C=C(C)C)C1(C)C 65817,c1(C(=O)NC(c2ccccc2)C(C)NC(C(C)=C2CC2)=O)ccc(Cl)c(C)c1Cl 65818,CC(N=c1[nH]c(=NC2CN(CC3CC3)C2)[nH]c2c1CCCC2)c1cn(C)nn1 65819,N1(C(C(C)N(C(C)=O)C)=O)CCC(NC(=O)C2=C(Cl)CC2)C2(CCC2)C1 65820,CCC(CC(F)(F)F)C(=O)N(C)CC1CCCN1C(=O)C(F)(F)c1cnnn1C 65821,c1(OCC)cc(C(N2CCCC2CNC(c2ccc(C#N)o2)=O)=O)ccc1OC 65822,N1(C(C(C(C)C)(C)O)=O)CCC2(CCCN(C(=O)CCn3cc(Cl)cn3)C2)CC1 65823,C1(F)(CNC(c2ncn(CC)c2)=O)CCC(CNC(c2ccnn2C2CC2)=O)C1 65824,CC1(C)C2CCC1(COC(=O)C(c1ccccc1F)(C)F)C2 65825,c1(CNC(c2cccc(F)c2)C(C)C)ccc2cccnc2c1Br 65826,Cc1cc(N)ccc1C(N1CCCC(N(C)C(C2CN(C3CCC3)C2)=O)CC1)=O 65827,C(C1=NOC2OCCCC12)OC(C1CS(=O)(=O)CC12CC2)=O 65828,n1(CC(=O)NCC2(OC)CN(C(=O)CC3NC(=O)NC3=O)C2)c(C)c(C)sc1=O 65829,c1(C(N2CCC(NC(c3c(CC)ocn3)=O)C(C)C2)=O)nccn2cc(C)nc12 65830,c1(C(=O)NCC2CCCN(C(C(C=C)(C)O)=O)C2)cnc(OC)cc1C(F)F 65831,c1(OC)ncc(C(N2CCC(C(N3CCN(CCF)CC3)=O)C(O)C2)=O)cc1Br 65832,N1(C(C2C(C(C)O)C2)=O)CCCC1CNC(=O)CCn1cc(Cl)cn1 65833,c1(C([N+]2([O-])C(C)CN(C(C3CC3C#N)=O)CCC2)=O)ccc2nnn(O)c2c1 65834,c1(C(N2C(C(N(CCCC)CCO)=O)CC3CC32)=O)ccc([N+](=O)[O-])cc1O 65835,c1(C(=O)OCC)cc(N2CCC(NC(c3cnn(C)c3Cl)=O)C(C)C2)nc(C)n1 65836,N1(C(C2N(C(C)=O)CSC2)=O)CCCCC1CNC(c1cc(OCC)n(C)n1)=O 65837,C(C)(CC(=O)N1CC=CC1C(=O)NCCCc1nc(C)no1)SC 65838,C1(CNC(C(c2cccs2)NC(C(C)NC(=O)NC)=O)=O)CNC(=O)C1 65839,Cc1cc(C(N2CCOCC2CC2CCCN(C(=O)C(C)C)C2)=O)cn(C)c1=O 65840,c1(C(N2CCC(C)(NC(CCC=C)=O)C2)=O)[nH]c2ccc(F)cc2c1C 65841,CCCC(C(=O)NCC(C)(C1CC1)NC(c1sc(C(C)C)nc1C)=O)N(C)C 65842,N1(C(CCN(C(=O)CCC2CCCO2)CC2CC2)=O)C2C=CCC1CC2 65843,c1(CN(C2CCCC(O)C2)C)cc(Cl)cnc1O 65844,C1(CCCNC(C2(F)CCCCC2)c2n(CC3(C)CC3)nnn2)CCC(C)CC1 65845,N1(C(C(C)(C)O)=O)CCCC2CN(C(c3cnc4sccn4c3=O)=O)CCC12 65846,C12(N(C)C)CCC(C(=O)NCCC(C)(C)NC(=O)Cc3cnnn3C)(CC1)CC2 65847,C1(NC(c2c(C(C)C)cco2)=O)CCCC(CNC(=O)CCCc2cnn[nH]2)C1 65848,c1(C(=O)NCC2N(C(c3nn(CC)c(O)c3)=O)CC2)cc[nH]c2nccc1-2 65849,C1(F)(CNC(c2cc(Cl)c[nH]2)=O)CN(C(C2CCCSC2)=O)C1 65850,c1(CC(=O)NC2C(C(N(CCC(C)C)C)=O)OCC2)ccnc(O)c1 65851,CCC(CC(=O)NCC1CN(C(=O)C(c2cnn(C)c2)=O)C(C)(C)C1)C(C)(C)C 65852,c1(C(=O)OCC)cnc(NC(C2CC3(CCO2)CC3)=O)c([N+](=O)[O-])c1 65853,C1(CC)CC(CC(N2CCC(O)(CC3CC3)C2)=O)CCO1 65854,c1(C(=O)OCC)nc(Br)c[nH]c1=NC(=O)c1ncc(-c2ccc(SC)s2)cn1 65855,C(C(C)CC(=O)N(C1CCN(C(=O)C=Cc2ccc(C3CC3)o2)C1)CCO)OC 65856,C(=O)(CS(=O)(=O)C1CC1)N(C(CNC(c1cc(N(C)C)ccn1)=O)C1CC1)C 65857,C1(C(=O)NC2(C)CCOC2)C2CN(C(=O)CCc3nc[nH]n3)CC12 65858,c1(C(=O)NCC(C)(CNC(C2(Cl)CCCCC2)=O)OC)cc[n+]([O-])cc1 65859,C1(CNC(CC(C)SC)=O)CC(F)(F)CN1C(=O)C=C(C)C1CC1 65860,CC(c1ccc(F)cc1)=CC(=O)NC1CCC(CNC(=O)C(C)(C)CO)C1 65861,C1(NC(C2(C)C(C)C2)=O)CCC12CCN(C(c1ccc3nn(C)cc3c1)=O)CC2 65862,N1(C(c2nc(C)nc(O)c2)=O)CCC2(CCCN(C(=O)CC3(O)CCOC3)C2)C1 65863,N1(C(c2cc(OC)n(C)n2)=O)CC(NC(c2sccc2Cl)=O)C2CCCC2C1 65864,c1(OC)cc(=O)n(C)cc1C(N1CC(N(C(=O)C#CC2CCCC2)C)C(O)C1)=O 65865,N1(C(C2(C)CC(C)C2)=O)CCCCC12CC(NC(c1cccc(CF)c1)=O)C2 65866,CCC(C)CCCCC(=O)NCC1(CNC(=O)C(C)CC(F)F)CCCCC1 65867,C1(C(=O)Nc2cnc(N(C)C)c(Br)c2)CCC2(CC1)CS(=O)(=O)C2 65868,c1(C(N2CC(Cn3cc(-c4ccc(Cl)c(F)c4)nn3)C2)=O)cc2n(n1)CCCC2 65869,c1(OC)c(C(=O)NCC2(NC(C3(C)CCOC3)=O)CCC2)ccc(Cl)c1Cl 65870,C1(CNC(CN(CC)CC)=O)CC2CCC1N2C(c1cc(F)ccc1OC)=O 65871,C1(CNC(c2c(CC)cccn2)=O)CCN(c2ncnc(Cl)c2F)CCC1(F)F 65872,N1(C(c2scc(C)c2)=O)CC2(CC2)CC1C(=O)NCc1c(Cl)cccc1Cl 65873,C12(NC(C=Cc3c(C)cccn3)=O)CCCN(C(=O)C=CC3CCOC3)CC1C2 65874,C(=O)(CCCCC(C)=O)NC1CCC(N(C(CC(CC)(C)C)=O)C)CC1 65875,CC(C)(C(=O)N1CCCC(Nc2nnc(C(F)(F)F)s2)C1)C(N)=O 65876,C12CCOC1CNC2=O.C(=O)(C(C)CO)OC 65877,c1(C(=O)NCC2(O)CN(C(C(C=CCCC)O)=O)C2)cc2nc(C)cc(C)n2n1 65878,Cc1ocnc1C(N1CCCC1CC(=O)N(C1CC(O)C1)C)=O 65879,N1(C(c2n(CCCC)ncc2)=O)CCC(NC(=O)C=CC(C)C)C(O)C1 65880,C(F)(F)(C(F)(F)F)OCC(=O)N(C)CC1(NC(Cc2ccc(C)o2)=O)CC1 65881,C1(CC=C)(NC(c2ccnc(OC)c2)=O)CCCN(c2nc(Cl)ns2)C1 65882,Cc1cscc1C(=O)N(C)CCOCCN(C(=O)CCc1nnc(C2CC2)o1)C 65883,c1(-c2nc(C(c3c(OC)cccc3)(C)C)on2)cc(C)cc(O)c1 65884,C1(CC)(NC(=O)COCc2nccs2)CCCN(C(=O)C=Cc2ccccc2)C1 65885,N1(C(c2ccn(CCCC)n2)=O)CCC(C2CC(NC(C3CC3(F)Cl)=O)C2)CC1 65886,CC1CC(C)CN(C(=O)CC2CCN(C(=O)CCc3nc[nH]n3)CC2)C1 65887,c1(C(N2CCC(NC(CCCC=C)=O)C2C2CC2)=O)ncc(P(C)(C)=O)cn1 65888,CCC(C)C(=O)N(C(C)CCNC(c1ccn(C2CCC2)n1)=O)C 65889,c1(CCC)ccccc1C(N1CCCC1c1cn(Cc2ccco2)nn1)=O 65890,CCCC(CCNC(=O)CN(CC(C)C)C(c1cncc(OC)n1)=O)C1CC1 65891,C1(NC(C(=O)NCC)=O)CC2CCC1N(C(C1(N(C)C)CCCC1)=O)C2 65892,N1(CC)CCCC(C(=O)NCc2cc(C(=O)NC3(C(F)F)CCCC3)n[nH]2)C1 65893,C1(NC(c2cc(C)n(C)n2)=O)C2CC(CN(C(C3CCNC(=O)C3)=O)C2)C1CO 65894,C1(C(=O)NCC(C(=O)NC2(CC)CCCCC2)O)CC(=O)CC12CCC2 65895,N1(C(c2c(COC)nn[nH]2)=O)CCN(C(=O)Cc2n[nH]c(C)n2)CC1C(C)C 65896,c1(C(=O)NCC2(C)CCN(C(CC(C)n3cccc3)=O)C2)n[nH]c2c1CSCC2 65897,CN1CCN(C(c2ccccc2CC#N)=O)CC1CNC(=O)C(C)(C)C(N)=O 65898,c1(C(=O)NC(CN(C(c2ccc(C)s2)=O)C)C)ccc(C)c(Br)c1C 65899,C(=O)(C(O)CC(C)C)NCCCN(CCC)C(c1ccccc1C(=O)OCC)=O 65900,N1(C(C(CC)F)=O)CC2(CC(CC3(CC(=O)NCC)CCCC3)C2)C1 65901,C(CCC(C)C)(C(=O)NCCN1CCCCC1=O)NC(CC(CCC)C)=O 65902,N1(C(c2cn(CCC)nn2)=O)CCC2(CNC(=O)C=CC3CCC3)CCCCC12 65903,C1(NC(CC2CC(=C)C2)=O)CN(C(C2(CCCC)CCC2)=O)CC2(CCC2)C1 65904,C12(C(N3C(CC(=O)NC(C(C(=O)OC)C)C)COCC3)=O)CCC(C1)OC2C 65905,C1(NC(COCC(c2ccccc2)C)=O)CCC2CC1CN2C(n1cncn1)=O 65906,C1(C(=O)NCCNC(c2ncnc(C)c2C)=O)CC12CCc1ccccc12 65907,C1(C(F)F)(CNC(c2scc(OC)c2)=O)CCN(C(C2CN(C(C)C)C2)=O)C1 65908,C(=O)(CCC(C)(C)[N+](=O)[O-])NCC1(C)CC(NC(c2c(C)onc2C2CC2)=O)C1 65909,CC(C(=O)NC1CCN(C(c2[nH]cc3c2CCC3)=O)CC1)C(F)(F)C(F)F 65910,CC1CC2=C(C(=O)N1)C(c1sc(Br)cc1Br)NC(=S)N2c1ccc(F)cc1 65911,N1(C(CCn2ccc(C)n2)=O)CC2CC2(CNC(C2CCC(=O)N2)=O)C1 65912,C=CCC(C)(C)CC(=O)NCCN(C(=O)CC1CCC(=O)NC1)C1CC1 65913,C1(NC(=O)C=CC2CCCCC2)CCCCN(C(=O)Cc2ccc(Cl)cc2Cl)C1 65914,C1(CC(=O)NC2(C(=O)O)C(c3ccc(Br)cc3)(C)C2)CCC2(CC2)CO1 65915,c1(C(=O)Nc2scc(C(c3c[nH]c4ncccc34)=O)n2)cc2c(Cl)ccnc2s1 65916,C1(C(=O)NC2(CC=C)CN(C(=O)COCC(F)(F)F)C2)CCc2nncn2C1 65917,c1(C(=O)NC2(CCCNC(Cn3ncc(CC)c3)=O)CC2)ccc(N)cn1 65918,C12(NC(c3cn(C)nn3)=O)CCCC1N(C(c1cc(C(C)(C)C)on1)=O)CC2 65919,C1(NC(=O)CCCc2ccccc2)CC12CCN(C(=O)CCC1OCCO1)CC2 65920,CCCS(=O)(=O)C(C)C(=O)NCCCN(CCO)C(c1ccc([N+](=O)[O-])cc1)=O 65921,c1(C(=O)NC(CNC(C(C)SCCCC)=O)C2CCC2)c(C)cnnc1O 65922,c1ccc(C2CCCC2NC(c2ccncn2)c2nnnn2C2CC2)cc1 65923,CCC(CN(C(=O)C=CC(C)(C)C)C)NC(=O)COC1CC=CC1 65924,CC1(C)CCC(CCNC(=O)Nc2c(NC(c3ccccc3Cl)=O)cnn2C)C1 65925,C1(NC(C(C)OCc2ccncc2)=O)CCCCC1CNC(C1CCC(=O)N1)=O 65926,O=C1COC2(CCN(C(C3CC(c4cccc(Br)c4)(O)C3)=O)CC2)CN1 65927,C(=O)(C(C)(C)CC(C)(C)C)NC1CN(C(CC(CC)CC)=O)CC(C)C1 65928,N1(CCC(=O)N(C)CCNC(C2(C)CC2Br)=O)CCOCC1 65929,C12(NC(=O)CSc3ccncc3)CC(C1)N(C(c1cccnc1O)=O)C2 65930,N1(C(c2ccc(CSC)cc2)=O)CC2CC(NC(=O)CCC3CCCO3)CC1C2 65931,C1(C(N2CC(C)(OC)C2)=O)COCCC1Nc1coc(C)n1 65932,C1(COC)(CNC(C2CC(C(C)C)C2)=O)CCN(C(=O)C(c2ccc(Cl)s2)=O)C1 65933,C(=O)(CCC(C)NC(=O)Cc1cnoc1)NCC1(CC)CCOC1 65934,c1(C(=O)NCC2N(C(CSC)=O)CCCC2)cc(C)cc(O)c1 65935,c1(N2CCC(N(C(C=C(CC)CC)=O)C)CC2)cc(C)nc2nc(C)nn12 65936,N1(C(C(C)O)=O)CC(CNC(=O)CNc2ccc(Br)cc2)C2(CCC2)C1 65937,Cc1cc(C(=O)NCC(O)CNC(C2NC(=O)OC2C)=O)ccc1C1CC1 65938,N1(CC(=O)N(CC(C)CNC(=O)CN2CCC(C)(O)C2)C)CCc2sccc2C1 65939,N1(C(C(COC)(F)F)=O)CCC(NC(c2ccc(F)cc2F)=O)C2(CCC2)C1 65940,C1(CC=C)(NC(=O)Cc2cnn(C(F)F)c2)CCN(C(=O)CN2CSCC2=O)C1 65941,C(=O)(CCC(C)(C)C)NC(C1(O)CCN(C(Cn2c(C)csc2=O)=O)C1)C 65942,N1(C(c2n(CC)ncc2Cl)=O)CC2CCC2(NC(=O)CCc2cnn(C)n2)C1 65943,c1(C(=O)NC(CCOC)CNC(C23CC4CC2C3C4)=O)nn(C)c(C)c1Br 65944,c1(C(=O)NCCC2(NC(C(C)Sc3ccccc3Cl)=O)CC2)cnc2n1CCC2 65945,c1(CN2CCC(NC(c3c(C)nc(OC)s3)=O)C(F)C2)ccc([N+](=O)[O-])cn1 65946,Cc1ccc(C)n1CC(=O)NCC1CC(C)N(C(=O)CCc2ccccc2O)C1 65947,CCC(C)(COC)C(=O)NC(C)CCCNC(c1ccn(COC)n1)=O 65948,C1(C(=O)NC(C2CCCN2C(c2cnc(O)s2)=O)C)CS(=O)(=O)C1 65949,C1(C)(OC)CCN(C(=NCCF)NCC(C)(O)C(F)(F)F)C1 65950,Cc1cc2c(CCNC(c3cc(CNC(=O)OC(C)(C)C)sn3)=O)csc2s1 65951,C=CCC(CC(=O)N(CCCF)C)NC(c1coc(N(C)C)n1)=O 65952,C12(NC(C(C)c3cccs3)=O)CCCC1N(C(c1ccc3n[nH]cc3n1)=O)CC2 65953,C1(NC2(C=C)CN(C(=O)OCC(C)(C)C)C2)CCC(=O)NC1c1ccnn1C 65954,N1(C(c2ccc(C#C)o2)=O)CCC(F)CC1C(=O)NCCc1ccncn1 65955,C1(C(=O)NCCCN(C)C(C2(F)CCCC2)=O)Cc2cccc(OC(F)F)c2O1 65956,c1(C(N(C)CC2COCCN2C(C2CC23CCC3)=O)=O)cc2c(nn1)CCCO2 65957,c1(C(N(CCN(C(=O)CC2C=CCCC2)C)C)=O)nn(C(C)(C)C)cc1Br 65958,c1(C(N2CC(OC)(CNC(=O)CNS(=O)(=O)CC)C2)=O)cc(NC)ccc1C 65959,CC1=C(C(=O)NCC2CC3COCC3N2C(=O)Cc2csc(Cl)c2)CCS1(=O)=O 65960,c1(C(=O)NC2CC(CCNC(=O)CC(=O)Nc3nccs3)C2)cc([N+](=O)[O-])c[nH]1 65961,C(=O)(C1COc2ccccc21)N1CC(CNC(CC(C)NS(C)(=O)=O)=O)C(C)C1 65962,C12(NC(c3cc(Cl)cc(Cl)n3)=O)CCCN(C(C3CCC=CCCC3)=O)CC1C2 65963,c1(OC)ccc(Cl)cc1CC(=O)NC1CCN(C(c2cccnc2Cl)=O)CC1C 65964,C1(C(=O)NC2CC(F)(CNC(=O)C=Cc3ccco3)C2)CCN2CCOCC12 65965,N1(C(C(C)NC=O)=O)CCC2(C1)CN(C(c1cnc3[nH]cnc3c1)=O)C2 65966,c1(C(=O)NC2CC(CNC(c3cc(F)ccc3Cl)=O)C2)cc2n(n1)CCCO2 65967,N1(C(C=C(C)c2ccco2)=O)CC2CCC1CN2C(=O)C=Cc1ccncc1C 65968,Cn1c(C(=O)NC(C(N2CCOC(C3CC3)C2)=O)C2CCC2)cccc1=O 65969,N1(C(CC2CCCN(C)C2)C(=O)NC2CCCCCC2)CCCCC2(CCC2)C1 65970,C1(C(=O)OC(C)CF)CC2CC1N(C(=O)OC(C)(C)C)C2 65971,N1(C(C(=C(C)C2CC2)F)=O)CCC(NC(c2cnn(-c3nccs3)c2)=O)C(F)C1 65972,Cc1cccc(C(C(=O)O)NC(=O)NCC(c2cccc(O)c2)O)c1C 65973,[N-]=[N+]=NC1CN(C(C2CCCCC23CC3)=O)CC1NC(=O)Cc1cccnc1Cl 65974,C(CC(C)(O)CNC(=O)C(C)(CNC(=O)Cc1csnn1)OC)OC 65975,N1(C(C(CC)OCC)=O)CCC(C)(CCNC(c2cnc(C)[nH]2)=O)C1 65976,Cc1cocc1C(N1CC(C(C)NC(C2CCCC2)CC2(CO)CCCC2)C1)=O 65977,C(C)(CCC(=O)NC(CO)C(C)NC(c1cnc(C(N)=O)cn1)=O)OC 65978,c1(C2CCN(c3n(C)c(C4CCC(F)(F)C4)nn3)CC2)ccc(Cl)c(F)c1F 65979,N1(C(c2c(CC)ncs2)=O)CCC(C2CC2)(CNC(=O)C(C)CO)C1 65980,C(C)(C(C)C(=O)N1CCOC(C)C1)NC(C1(C(C)C)CCC1)=O 65981,c1(C(N(C2CCN(C(=O)CC3CCNC3=O)C2)CCC)=O)ccc(CC2CC2)s1 65982,c1(C(N2CCC(C(C)NC(c3ncccn3)=O)C2)=O)sc2sccc2c1Cl 65983,C(=O)(CCCCCCCCC1CC1)N1CCCC(NC(C(C)CC(N)=O)=O)CC1 65984,C#CCCCCC(=O)NCC(CC1CC1)C(=O)N(CCCCC=C)C 65985,N1(C(C23C(CN(C(c4c(CC)noc4)=O)C2)C3)=O)CCC(C#N)CC12CC2 65986,C1(C2(O)CN(C(c3cc(C)n(C4CC4)n3)=O)C2)(CNC(CC(C)OC)=O)CC1 65987,N1(C(c2c(C(C)C)onc2)=O)CC(C)CN(C(=O)C(O)CN(C)C)C(C)C1 65988,C(=O)(C1CCCc2ncccc21)N1CCC(N(C(CC)=O)CCO)CC1 65989,c1(C(=O)NCC(C2CCC2)NC(C(CC)n2cncn2)=O)cncc(Br)c1 65990,N1(C(C2CC(CNC(C(C(C)C)=O)=O)C2)=O)CCN(C)C(CO)C1 65991,c1(NC(c2c(SCc3nc(CC)c(C)s3)cccc2)=O)cnn2c1C(=O)NCC2 65992,N1(C(C2(CSC)CC2)=O)C2CCC1CN(C(=O)CN1CCCCC1)C2 65993,C(=O)(CCCCCC(C)C)NCC(CNC(=O)C#CC1CCOC1)OC 65994,C(CS(C)(=O)=O)N(C)C(C1CCC1NC(=O)CCC1CC1(C)C)=O 65995,c1(C(=O)NC(C)CCCNC(=O)C=Cc2ccco2)cccc(Br)c1 65996,CCC1=NOC(C(N2CCCC(N(CCF)C(c3cn(C)cn3)=O)C2)=O)C1 65997,N1(C(c2c(C)nn(C3CCC3)c2)=O)CCN(C(=O)CC2CCC(C)C2)C(C)C1 65998,c1(OC)cc(C(=O)N(C)CCN(C)C(c2cc(N)ccn2)=O)cc2cnn(C)c12 65999,c1(NC(=O)NC2CCN(Cc3cc(O)cc(Br)c3)C2)ccc2c(c1)C(=O)CC2 66000,CONC(=O)CNC(C1(F)CN(C(=O)C(=C2CCCCC2)F)C1)=O 66001,C1(C(=O)NC2CN(C(CCC(=C)C)=O)CC2(C)C)CC2CCCC(C1)C2 66002,CC(C)CC(=O)C(=O)NC1CCCC(C(=O)NCCC2(O)CCOC2)C1 66003,c1(C(N(CC(=O)N(CC2CC(=C)C2)C(C)C)C)=O)n[nH]c2c1COC2 66004,C1(C(=O)NC(CC)COCC2CC2)CN(C(=O)C(C#N)C(C)C)CCN1C 66005,CC1CC(NC(c2nccnc2Cl)=O)CN(Cc2ncccc2C(F)(F)F)C1 66006,CCC(CC)C(C)C(=O)NCC1CCCN1C(=O)CNC(c1cccc(C)c1)=O 66007,CC(C)C(C(=O)NC(C)(CO)C1CCC1)N(C)C 66008,c1(SC)cc(C(=O)NC(C)C(C)NC(c2conc2-c2ccccc2)=O)c(C)o1 66009,Cc1ccc2nc(C(=O)NCc3ccc(C(F)F)cn3)[nH]c2c1 66010,CC(C)(CNC(c1cc(O)ccc1F)=O)CC(=O)NC(C(N)=O)C1CC1 66011,C(C(C)(O)C(=O)NCC1(CNC(=O)CC(F)F)CC1)OC 66012,c1(C(N2CCC(CNC(c3cc(C)on3)=O)C2)=O)cc2ccccc2c(O)n1 66013,C1(OC)CN(C(=O)CN2CSCC2=O)CC1NC(=O)CCC1CCN(C)CC1 66014,c1(CN2CCC(C(=O)NCCSCC)C2)cccc(Br)c1Br 66015,CN1CCn2cc(C(=O)NCC3CCCN(C(C4CCSC4)=O)CC3)nc2C1=O 66016,C1(C)(CNC(C2(CC=C)CC2)=O)CN(C(=O)Cc2cc(Cl)n(C)n2)CC1C 66017,c1(C(C(=O)NC2CC(C(=O)OC)C2)N(C(C#C)C)C)csc(C(C)C)n1 66018,C(C(C(C)(C)C)NC(=O)Cc1cc(C)on1)NC(Cc1ccc(C)o1)=O 66019,CCC(C)C(O)C(=O)N1CCC(CF)(NC(C2CCCN2C(C)C)=O)C1 66020,c1(C(=O)NCCCC2N(C(C3C(C)=C3)=O)CCC2)cc2n(n1)C(C)CCC2 66021,N1(C(C2CCC(OC)CC2)=O)CC(NC(C2CCOC(C)(C)C2)=O)C(C)(C)C1 66022,N1(C(c2cc(OCC)n[nH]2)=O)CC2(CCN2C(C2CCC(=O)C(C)C2)=O)C1 66023,Cc1[nH]cc(C(N2CC(O)(CN(C)C(C3(O)CC4CCC3C4)=O)C2)=O)c(=O)c1Cl 66024,CC1=NS(=O)(=O)NC=C1C(=O)N1CC2CC1C2CNC(=O)CC(O)C(C)C 66025,C(=O)(CC(C)(C)CCOC)N(CCCNC(C(C)=C(CC)C)=O)CC 66026,N1(C(COCC=C)=O)CCN(C(=O)C(C)NS(C)(=O)=O)C(C(C)C)C1 66027,CC(CC(=O)N1CC2CCC1CC2NC(C1(C)CCCCO1)=O)P(C)(C)=O 66028,c1(NC(C2C(C(=O)OC)C2)=O)ccc(I)c(C(c2cc(F)ccc2Br)OC)c1 66029,C(=O)(C(C)(O)C(F)(F)F)N1CC(NC(c2c(OCCOC)cccc2)=O)C(C)C1 66030,C1(CNC(C2(CC)CCC2)=O)CCCC1NC(=O)C=CCO 66031,CC1CC(CNC(c2cccnc2O)=O)CN1C(=O)C(c1cnn(C(C)C)c1)=O 66032,n1(CCCC)ncc(C(=O)N(CCC)CCNC(=O)CC(C)N(C)C)c1C 66033,CCC(O)C(C)C(=O)NCCN(C(=O)C(c1ccc(F)c(F)c1)(F)F)C 66034,N1(C(c2c(SC)c(F)ccc2)=O)CCCC1C1CCCN1C(=O)C(F)F 66035,N1(C(c2cccc(NCc3cc(C)[nH]n3)c2)=O)CCC2(CC1)OCCO2 66036,c1(C(c2ccccc2)OC)cn(C2CCN(C(c3cnoc3C3CC3)=O)C2)nn1 66037,c1(OC)cnc(F)c(C(=O)N(C(=O)C(c2cc(F)cc(F)c2)OC)CCC#N)c1 66038,N1(C(CC(C(=O)OC)C)=O)CCC(C)(C)CC1C(=O)NCC1NC(=O)OC1(C)C 66039,c1(C(N2CCC(NC(=O)Nc3cccc(C)c3)C2)=O)c(Cl)ccc(O)c1Cl 66040,C1(NC(C2ON=C(C)C2)=O)(CNC(c2cncc(F)c2Cl)=O)CC2CCC1CC2 66041,c1(NC(C2N(C(C(CSC)O)=O)CC(F)C2)=O)ccc(O)cc1C 66042,Cc1cc(CCC(N2CC(NC(c3c(Cl)n[nH]c3C)=O)CC(C)C2)=O)cc(C)c1 66043,C(=O)(CC(O)C(C)C)NCCN(C(=O)Cn1ccc(O)nc1=O)CC 66044,N1(C(C2CC(=C)C2)=O)CCC(C)C1CNC(c1cnc(C2CC2)nc1)=O 66045,Cc1ccc(CCCC(=O)NCC(CC(C)C)NC(C23CCC2C3)=O)cc1C 66046,c1(C(=O)NC2CC3CC2CN3C(=O)C(O)O)ccc2nnc(Br)n2c1 66047,N1(C(CSCCC)=O)CCN(C(c2cn(CCC)nc2C)=O)CC(O)C1 66048,C1(CNC(CSCC=C)=O)COCC1NC(=O)CSCCC#N 66049,C(=O)(C#CC1CCCC1)NC1(COC)CCCN(C(=O)C(=C2CCCCC2)F)C1 66050,CC(C)C1=CCC(NC(C2(NC(=O)C=CC3CC3)CCN(C)C2)=O)CC1 66051,C(=O)(CC(C)(C)n1cc(CN2CCOCC2)nn1)N(CC(C)C)CCC 66052,C1(CNC(CCCC(C)O)=O)CC2(CO1)CN(C(=O)C(F)(F)CO)C2 66053,C(=O)(CCC(C)(C)F)N(CCC(C)(C)NC(=O)CC1CCCC1(F)F)C 66054,n1(CCC)ncc(CNC(=O)CCN2CCN(C(=O)C(C)NC(C)=O)CC2)c1C 66055,N1(Cc2c(C)cc(OC)nc2)CCC2C1CCCN2c1nc(OC)cc(C)n1 66056,N1(C(C2C(OC)CC2)=O)CC(NC(c2ccc(Cl)c(F)c2N)=O)C2(CCC2)C1 66057,N1(C(C(N2CCOCC2)C)=O)CCCCC(N(C(=O)C=C(C2CC2)C2CC2)C)C1 66058,CC1CC(C(=O)NCC2C3CN(C(c4ccc(Cl)o4)=O)CC23)CCC1C 66059,N1(C(C(C)OCCCC)=O)CCN(C(c2ccc(C(F)(F)F)s2)=O)CC1CCC 66060,C1(C#N)(C(=O)NC(CC)CNC(c2nnsc2C)=O)CCSCC1 66061,c1(OCC)ccc(CCCNC(c2nc(CC)no2)=O)cc1 66062,C(=O)(C(c1ccoc1)NC(=O)C(C)N(CCSC)CC)NCC(=C)C 66063,NS(=O)(=O)N1CCCC(C(=O)NCC(O)CNC(c2c[nH]c(C(N)=O)c2)=O)C1 66064,c1(NCC)scnc1C(=O)NCCCC(C)NC(=O)Cc1csc(C(C)C)n1 66065,CCCCCCCCCCC(CC)NCCCOc1cc(C)ccc1C 66066,Cc1ccccc1C=CC(=O)NC(C)CCN(C)C(C1CC2CC2C1)=O 66067,c1(C(N2CCC(NC(CN(CC)CC)=O)C(O)C2)=O)cccc2c1OCCO2 66068,c1(SC)cc(C)c(C(N2CC(CNC(C3(C)CCOC3C)=O)C(O)C2)=O)o1 66069,CC1N(C(=O)C(Cc2ccoc2)NC(c2cccnn2)=O)CCOC1(C)C 66070,CCCCC(C(=O)NCC(CC(N1CC(CO)CC(C)(C)C1)=O)OC)C(C)C 66071,C(C)(CC(=O)NCC1CCC1NC(c1cc(N)c(F)cc1F)=O)(C(F)F)N(C)C 66072,C1(CNC(CCOC)=O)CC2(CCOCC2)CN1C(=O)CC1CC2CCC1C2 66073,C1(NC(C2=NOC(C)C2)=O)CCC(O)CN(C(=O)Cc2c[nH]c3ccccc23)C1 66074,n1(C2CCN(C(Cc3cc(C)cc(F)c3)=O)C2)ncc2c1CCCC2 66075,C1(CNC(=O)Nc2ccc(Br)cn2)CCCC(CF)C1 66076,CC1(C)CN(C(=O)NCc2cc3cccnc3s2)C2CCCC12 66077,N1(C(c2c(C)ncs2)=O)CCC2(CC1)CCN(C(c1csc(C)c1C)=O)C2 66078,c1(CC(=O)NCC#CCNC(C)=O)ccc(Cl)s1 66079,Cn1cnc(S(N)(=O)=O)c1C(=O)NC1CC(CNC(c2cncn2C)=O)C1 66080,C=CCC(CC(F)F)C(=O)N1CC(CNC(=O)CSCc2cccs2)CC1(C)C 66081,C12(C(N3CCCC(c4cn(CCCC)nn4)C3)=O)CC3CC(C(=O)N1)C2C3 66082,c1(C(CC(=O)OC)=O)ccc(F)cc1[N+](=O)[O-].C1CCC(=O)O1 66083,C1(=O)NNc2nccnc2N1.C1(CNC(=O)OC(C)(C)C)CC2CCC1O2 66084,c1(OC)ncccc1C(N1CC(CNC(C2(n3cc(Cl)cn3)CC2)=O)CC1C)=O 66085,Cc1cccc(C)c1C(=O)NCCC1COCCN1C(C1CC1C)=O 66086,C1(C(=O)NCC2(COC)CN(C(c3occc3C)=O)C2)CCc2nnn(C)c2C1 66087,c1(C(=O)NC2C(C)(C)CCN(C(C(C=C=C)C)=O)C2)cc(C)cc2c1OCC2 66088,C#CCC(C)(CC)C(=O)NC1COCCC1C(N1CCOC(C)C1)=O 66089,CCC(CC(=O)N1CCC(CCNC(=O)C(C)(C)CF)C1)c1ccc(OC)cc1 66090,c1(CNC(C(C=C=C)C)=O)nc2c(s1)CN(C(C1CC(C(=O)OC)C1)=O)CC2 66091,c1(CC(N2CC(CNC(C3(F)C4CCCC34)=O)C2)=O)ccc2ncccc2c1 66092,CC1(C)CCOC(C(N2CCC(C3CC(NC(=O)CC#N)CCO3)CC2)=O)C1 66093,O=C(CCC1CC1C(F)(F)F)NCC1CC1NC(=O)CC1CCC1 66094,c1(C(=O)NCC2(F)CCN(C(C3CC(OCC)C3)=O)C2)ccc(C)c(C)c1 66095,C12(C(=O)NCC3CCC(NC(C(C)(C)C(N)=O)=O)CC3)CCCCC1OCC2 66096,C1(C(=O)NC(COCC)C)(NC(c2nccn2C)=O)CCC(C)CC1 66097,C(CC(C)(C)CC(=O)NCC1(O)CCN(C(C2(O)CC(CF)C2)=O)C1)OC 66098,C1(NC(=O)CCCCN2CCCC2)CC(F)(F)CC1C(=O)O 66099,C1(CNC(Cn2cnc(CC)n2)=O)CN(C(=O)COC2CC=CC2)CC1C 66100,C1(NC(C(C)(C)CF)=O)CCN(C(C2(O)CC(F)(F)C2)=O)CC1c1ccccc1 66101,c1(C(N(C)CC2CCCCN2C(=O)CC2(CO)CC2)=O)cnc2ccccc2n1 66102,C1(CC)CN(C(=O)Cc2nc(Cl)cs2)CCN1C(c1cscc1C)=O 66103,C(CCOCC)(C(=O)N(C)CCN1CCCC1)NC(C(CC)n1ccnc1)=O 66104,c1(OC)cc(CO)ccc1C(N1CCCC(C)C1CNC(=O)CSC)=O 66105,Cc1cc(=O)oc(C)c1C(=O)NC1CS(=O)(=O)CC1NC(C1CCCC(=O)C1)=O 66106,C1(O)(CNC(C2CC(=C)C2)=O)CCCN(C(c2ccc(Br)c(C)c2)=O)C1 66107,c1(OCC)cc(C(=O)NC(CCN(C)C(C2(O)COC2)=O)C(C)(C)C)oc(=O)c1 66108,N1(C(c2c(C)n(CCO)cc2)=O)CCCC(NC(C2CC(C)(F)C2)=O)C1C 66109,c1(C(=O)NC2C(NC(c3cc(C)sn3)=O)CCC2)ccc2c(c1)CN(C)C2 66110,c1(C(N2CCC(NC(c3cncc(C(C)(F)F)c3)=O)CC2)=O)nnn2c1CCC2 66111,c1(CC(C(=O)N(C(CC#C)C)C)NC(=O)C(C)CC=C)cnn(C)c1O 66112,Cn1cc(C(=O)NC2C3CC(NC(=O)CCC4CCC4)CC23)ncc1=O 66113,c1(OCC)ncccc1CC(=O)NCC1CCN(C(C2(n3nccn3)CC2)=O)C1 66114,C(=O)(C1=CCCCC1C)NCC(C)(C1CC1)NC(c1occ(C)c1)=O 66115,Cc1nc(Cl)ccc1S(=O)(=O)N1CC2CN(C(c3ccc(C#N)s3)=O)CC12 66116,c1(-c2c(C(N)=O)csc2)ccc2c(c1)CN(Cc1ccc(F)cc1)CC2 66117,Cc1cc(F)c(Cl)cc1C(=O)NCC(C)CN(C)C(c1ccc(C#N)nc1O)=O 66118,c1(NC(CC2(CNC(C3(COC)CCC3)=O)CC2)=O)cc(C#N)ccc1C 66119,N1(C(C=CCC)=O)CCN(C(c2cnn(CC)c2CC)=O)C(C(C)C)C1 66120,c1(NC(C2(OC)CCC(C)CC2)c2nnnn2C)ccc2nn(C)c(C)c2c1 66121,C1(C(=O)NC(C2CCOCC2)C(=O)NC2(CC)CCOCC2)CCC2CC1CO2 66122,CN1CC(CC(N2CC(NC(C3CC(N4CCCC4)C3)=O)C2)=O)C1 66123,C1(CC)(NC(C2CC3(CC3)C2)=O)CCCN(C(C2(C)CCC2)=O)C1 66124,c1(OC)cc(C#N)ccc1CNC1CC1C(=O)NCC1CCO1 66125,C(=O)(C1CCc2snnc21)NC(C(C)NC(c1cnn(CCN(C)C)c1)=O)C 66126,c1(CSCCC)nc(-c2cccc(N(C)C)n2)nn1CC1COCCO1 66127,C1(CNC(CCc2nc(C)sc2)=O)CCCCN1C(C1(C)CCCC1)=O 66128,C1(O)(C(C)NC(C2(F)CCOC2)=O)CCN(C(=O)COCC2CCCO2)CC1 66129,Cn1cc(C(=O)NCC2CN(C(=O)Cc3ccsn3)CC(C)(C)C2)c(O)nc1=O 66130,C1(C(=O)NC(c2nn[nH]n2)CC)(C(C)C)CCN(C(C2CCS(=O)CC2)=O)C1 66131,N1(C(c2ncn(CC)c2)=O)CC2(C(=O)N(C)Cc3cnc(C)s3)CCC1CC2 66132,C=CC(C(=O)NC(Cc1ccco1)C(=O)N1CC(C)(CCO)C1)OC 66133,C1(CNC(C(C)OCC)=O)CCC(F)(CNC(c2cnc(C(F)F)s2)=O)CC1 66134,N(C(=NCCC(=O)NC(C)C)NCC(C)(C)C#N)Cc1c(SC)cccc1 66135,C12(NC(CC3(OC)CC3)=O)CCC(CC1n1cc(-c3ccc(Cl)cn3)nn1)C2 66136,N1(C(c2cc(CC)oc2C)=O)CCN2CCN(C(c3cc(F)c[nH]3)=O)CC2C1 66137,CC(=O)CCC(=O)N(C(C)CN(C(=O)CCNC(c1ccsc1)=O)C)C 66138,c1(CC(=O)N(CCOC(C)(C)C)C2CC2)ccc(F)cc1I 66139,Cc1ccsc1C=CC(N1CCC(OCCNC(c2ccnc(O)c2)=O)C1)=O 66140,C(=O)(C(=O)N=S(C)(C)=O)NC1C(CNC(c2c(C)n(CC3CC3)cc2)=O)C1 66141,N1(C(c2n(C)ccc(=O)c2)=O)CCOC2(CCCCC2NC(C2CCOC2)=O)C1 66142,N1(C(CCCC#C)=O)CCC(NC(c2cccc(N)c2F)=O)C(F)(F)CC1 66143,N1(C(CN(C)S(N)(=O)=O)=O)CC(NC(C2CCC(=O)NC2)=O)CC2(CCOCC2)C1 66144,N1(CC(C2CCOC2)F)CCC(NCC(F)F)CC1 66145,N1(C(CCNC(C(C)NC(C)=O)=O)=O)CCCC1CC1(C)CC1C 66146,CC1CN(C(C2(O)CCSC2)=O)CC1CNC(c1cc(-c2cnn(C)c2)on1)=O 66147,c1(-n2cc(-c3ccn(C)n3)nn2)ccccc1NC1CN(c2ccc(F)cc2)C1 66148,N1(CC)CC(C(N2CCC(CN=c3[nH]nc(C4CC4)s3)C(C)C2)=O)CCC1=O 66149,C1(C(=O)NCc2cn(CC(=O)NCC(O)C(F)(F)F)nn2)CC2C(C1)C2(F)F 66150,C1(C(N2CC(OCCO)C2)=O)CCN(C(=O)C(F)(F)c2ncccn2)CC1 66151,c1(CC(C(=O)N(C(C)CNC(C2CC2F)=O)C)C)ccc([N+](=O)[O-])cc1 66152,Cc1cccc2[nH]cc(C(=O)NC34CCOCC3CN(C(C3CCC3)=O)C4)c12 66153,C(=O)(C1=NOC(C)C1C)NC1(CC=CC(=O)NCC(CC)(C)OC)CCCCC1 66154,C1(NC(CSCC(C)C)=O)CCN(C(=O)CC(=O)NC2CC2)CC1O 66155,C1(C(=O)NC2(C)CCN(C(=O)Cc3n[nH]c(=N)s3)CC2)CSc2ccccc2O1 66156,c1(CC(=O)NCC(CNC(CC2(C)CC2)=O)O)ccc(C(N)=O)cc1 66157,N1(C(c2c(CC)noc2)=O)CCN(C(=O)Cn2c(C)csc2=O)C(CC(F)F)C1 66158,c1(SC)nccc(=NC(CNC(c2n[nH]cc2C(F)(F)F)=O)C(C)C(C)C)[nH]1 66159,CC(=O)CCN=C(NCCc1cc2ccccc2o1)NCC1COCCN1C 66160,c1(NC(COC)C2CC2)nc(N2CCOC(c3ccccn3)C2)nc2sccc12 66161,C#CCC(CC#C)C(=O)NCC1=CCN(C(=O)C2=CCCCC2)CC1 66162,O=C(C1c2c[nH]nc2CN1C(c1cnc(O)o1)=O)NC1C2COCC12 66163,c1(CNc2cc(C(F)(F)F)cc(C(C)C)c2C)ccc2c(c1)C(CC)C(=O)N2C 66164,C(=O)(C1=CCCSC1)NC1C(NC(CCc2ccc(OC(C)C)cc2)=O)CCC1 66165,C1(NC(c2ccnc(OCC3CC3)c2)=O)CCOCC1F 66166,CCC(C)CC(=O)NCC1CCC(NC(=O)C(C)(Cl)Cl)C1 66167,N1(C(CCCc2c(C)ccs2)=O)C(CNC(C2(N(C)C)CCC2)=O)CC2CC12 66168,C#Cc1ccc(CN2CC(C)(CNC(=O)Cc3ccc(OC)c(Br)c3)C2)cc1 66169,C12(NC(=O)CN3CCCCC3)CCC(CC1)N(C(C1CC3C=CC1C31CC1)=O)C2 66170,C1(CNC(c2ncn(C)n2)=O)CN(C(=O)C(C)(F)F)CCO1 66171,C1(C=O)CCC(C#N)C1.C1(NC)CC(O)(CC2(C)COC2)C1.n12cc(nn1)C2 66172,CCCCC(C)CCC(=O)NC1(CC(=O)N(C(C(N)=O)C2CC2)C)CCC1 66173,C(=O)(C(F)CCC(C)(C)C)N(C1(C(N2CCC(C(=O)NC)C2C)=O)CC1)C 66174,C1(C(=O)NCCC2(C(NOCCOC)=O)CCC2)CCCC1C 66175,Cc1nnc(O)c(C(=O)NC2CN(Cc3cccs3)C2)c1C 66176,C1(C(=O)NCCC(C)NC(c2ncoc2Br)=O)CCCCCC1(F)F 66177,c1(C(=O)NC2(C(NOCCOCCOC)=O)CCCC2C)ncc(F)cc1N 66178,C1(CC#C)(C(N2CCCC(NC(=O)CCN3CCOCC3)C2)=O)CCOCC1 66179,N1(C(C(C=C)(C)CCOC)=O)CCOC2(CCN(C(c3cncnc3C)=O)C2)C1 66180,N1(C(c2c(C)onc2C(F)(F)F)=O)CC2CC1CN2C(=O)C=CC(F)(F)F 66181,N1(C(CNC(N)=O)=O)CCC(F)(C(=O)NC(CC2CC2)CC2CC2)CC1 66182,N1(C(C2N(C)CCC2)=O)CCN(C(=O)C(F)=CC2CC2)CC1c1ccccc1Cl 66183,C1(C)(NC(C(N2CCOCC2)C)=O)CCN(C(C2CCOCC2)=O)C1 66184,C1(C2(O)CCN(C(c3cscc3Cl)=O)CC2)(NC(=O)COCC2CCOC2)CC1 66185,C1(NC(c2cnc(Cl)s2)=O)CCCN(C(c2cnc3c(c2)COC3)=O)CC1F 66186,N1(C(C(C)=CC)=O)C2CCC1CN(C(=O)Cc1ccc(O)c(O)c1)C2 66187,c1(CC)ccnc(N(C)C(=S)NCC(c2ccc(F)cc2)O)c1 66188,N1(C(CC2C=NN(C)C2=O)=O)CC(NC(c2ccn(C(C)(C)C)n2)=O)CC(F)C1 66189,c1(N(C)C)c(F)cc(C(=O)NC2CC2C(=O)NCc2nc(Br)cs2)cc1F 66190,CCCCC(O)CC(=O)N1CCCC1C(C)(C)NC(=O)CSCCN(C)C 66191,N1(CC=CCNC(C=CCN(C)CC)=O)CCC(NC(c2sccc2Cl)=O)CC1 66192,c1(C(N2C(CNC(C(CC)=O)=O)CCC2)=O)cc(C(C)(C)C)cc(C(C)(C)C)c1 66193,C(CCC(O)C(=O)NCC1CC(=C2CCC2)C1)NC(=O)C(F)F 66194,S(=O)(=O)(c1cccnc1NCc1nnc(O)o1)NC(C(C)(C)C)CCO 66195,C1(NC(C2(C=C)CCC2)=O)CCCN(C(c2ocnc2-c2ccccc2)=O)C1 66196,C(C(CO)C(C)CC)NC(c1cc(CNC(C(C=C=C)C)=O)nn1C)=O 66197,c1(C(N2CCC(C(C)NC(C(C)NC(=O)NC)=O)C2)=O)cccc2c1CCCC2 66198,C(=O)(C(F)C1=CCCCC1)NCCN(C(C(Cc1c(C)cccc1)C)=O)C(C)C 66199,N1(C(c2c(CCC)[nH]cc2)=O)CC2CC1CN2C(C1CC1C(C)C)=O 66200,N1(C(c2c(C)oc(C(C)C)c2)=O)CC(NC(=O)CC2OCCC2(C)C)C2(CC2)C1 66201,c1(SC)cc(C)ccc1C(N1CCN(C(C2CSC2)=O)CC1CS(C)(=O)=O)=O 66202,c1(C(N2C(C(=O)NCCSC)CCC2)=O)cccc(-c2cccs2)n1 66203,N1(C(c2ccc(NC)cn2)=O)CC=C(C(=O)NC2CC2C2CC2C)C1 66204,c1(NC(=O)NCc2cc(=N)[nH]cc2)nc2ncccc2o1 66205,c1(C(=O)NCc2c(C3CN(C(C(C=C)O)=O)C3)ocn2)ccc(C2CC2)cc1C 66206,Cc1n[nH]cc1C(=O)N(C1CCC(NC(=O)CC2(CN(C)C)CCCC2)C1)C 66207,CC(C)C(CC(=O)NCC(C)(C)NC12CC=CC(C1)OC2)NC(=O)OC(C)(C)C 66208,c1(CC)nc(C#N)cc(=NCC2CN(C3CCN(C4CCN(C)CC4)CC3)C2)[nH]1 66209,Cc1nc(C)c(C(=O)NC2CCCC(NC(c3cnc[nH]c3=N)=O)C2)o1 66210,Cc1n[nH]c2nc(O)c(C(=O)NC3(CNC(=O)C=CC(F)(F)F)CCOC3)cc12 66211,N1(C(C2CCC(OCC)CC2)=O)CC(F)(F)CCC1C 66212,N1(C(C2N(C)CCC2)=O)CC(O)C(O)C1CNC(C1CC(=C(F)F)C1)=O 66213,N1(C(C2(CN)CC2)=O)CCCC1CNC(N)=O 66214,CC1(C)CN(C(=O)COc2ccc(F)c(F)c2)CC1NC(=O)CC1CC12CC2 66215,C1(NC(C2N(CCC)CCCC2)=O)CC2CCC(C1)N2C(c1c[nH]c(=NC)s1)=O 66216,c1(OC)cncc(C(=O)NC(C2CCN(C(=O)CC3CCC(=O)N3)C2)(C)C)n1 66217,c1(OC)ccc(CC(=O)N(C2CCCN(C(C3CCSC3)=O)C2)CCO)c(Cl)c1 66218,c1(C(=O)NC2CC(N(C(C(C3CC3)OC)=O)C)C2)sc2ccccc2c1CSC 66219,CC1C(NC(=O)CC(C)(C)C(F)F)C(C)CCN1C(=O)CCOCC(F)F 66220,CC1CC(N=c2[nH]c(=NCC3(c4ccccn4)CCC3)c3ncccc3[nH]2)CS1 66221,c1(C(N(C2CCCN(C(=O)C(O)C(F)F)CC2)CC)=O)nc(C)c(C)nc1C 66222,N1(C(c2ccc(NC(=O)NC)cc2)=O)CC(C)OC(C)C1C 66223,N1(CC(=O)NC2CN(C(CCOCC#C)=O)C2)CCCC1C 66224,C1(NC(c2cccc(COC)c2)=O)CCN(C(c2cccc(CO)n2)=O)CC1O 66225,C1(C(C)C)CN(C(C2CCC(C)(F)CC2)=O)CCC1NC(c1ncccc1N)=O 66226,c1(NC(C2(C)CCCN(CC(c3n(C)ccc3)=O)C2)=O)cc(Cl)cnc1Br 66227,C1(CN=[N+]=[N-])CCCN(C(c2cncc(CNC(=O)C=CC3CCC3)c2)=O)C1 66228,C(N=c1[nH]cnc2c1SCCC2)C1C(C)(C)CN(C(c2cnc(C3CC3)[nH]2)=O)C1 66229,C(C(O)CCNC(c1csc(CC(F)(F)F)n1)=O)NC(C(=O)N(C)C)=O 66230,c1(C(N2C(C(N3CCC(=C)C3)=O)CCC2C)=O)ccc(C#N)n1C 66231,C1(CCNC(c2cnc(C(F)F)s2)=O)CN(C(=O)Cc2nnc(O)s2)CCO1 66232,c1(C(=O)NC2C(NC(CCN(CC)CC)=O)CC2)cnc(O)cc1O 66233,c1(CC(=O)NC2CCC(CNC(Cc3ccn(C)n3)=O)C2)c(F)cccc1C#N 66234,Cc1ccnc(C(N2CCSC(C(=O)NCc3cnc(Cl)s3)C2)=O)c1 66235,C12(CNC(C3CC(C)N3C(=O)C=Cc3ccnn3C)=O)CCC(CO1)C2 66236,N1(C(C(CCSC)(C)C)=O)CCC=C(C(=O)N(C)CC2C(C)(C)C2(C)C)C1 66237,c1(NC(C2CN(C(c3n(C)c(S)nn3)=O)CC2F)=O)cccc2c1CCO2 66238,C1(C(C)NC(C(C2CC2)OCC)=O)CCN(C(c2csc(CC(C)C)n2)=O)CC1 66239,C12(C(=O)NC(C3CN(c4snc(CCOC)n4)C3)C)CCC(CO)(CC1)CC2 66240,c1(C(=O)NCC(CC(=O)N2CCCC2CCC(C)C)OC)ccc(C#N)cn1 66241,c1(C(=O)NC2(CNC(C3CCNC(=O)C3)=O)CC(OC)C2)n[nH]c2c1CSCC2 66242,c1(CN(C(=O)CC2(C)CCC2)C)cccc(Br)c1 66243,c1(C(=O)NC2CCCN(C(=O)CSCC(F)(F)F)C2)ccc2c(c1)B(O)OC2 66244,N1(C(C(C)Cc2ccccc2)=O)CCC(CN(C)C(c2cnc(O)n2C)=O)CC1 66245,CC1CN(C(c2cc(CNC(c3ccon3)=O)[nH]n2)=O)CCC1O 66246,C1(C(N2C(CN(C(=O)C(CC(C)C)OC)CC)CCCC2)=O)CCCCCCC1 66247,C1(C(=O)NCC2(CCNC(c3cc(OC)n[nH]3)=O)CC2)CCCC1S(C)(=O)=O 66248,N1(C(C(C)OC)=O)CC(NC(c2ccc(F)c(C(F)(F)F)c2)=O)CC2(CC2)C1 66249,C(C(F)C(=O)NCC(O)CCNC(C1(C#N)CCC1)=O)N(CC)CC 66250,C1(NC(c2cc(CC)nnc2C)=O)CC2CCC1C(NC(=O)CN1CC=CC1)C2 66251,C(=O)(C(C)(C)CC1CC1)NCC1(N(C(=O)C=CCF)C)CC1 66252,C1(C(=O)NC(C)CNC(c2cncc(Cl)c2)=O)CCC2(CC1)CC2(F)F 66253,N1(C(C(c2cccc(C)c2)O)=O)CC2CC(C1)C2NC(C1CC1C)=O 66254,c1(C(=O)NC2CC(O)(CNC(=O)CC3CCC=CCC3)C2)ncnc2ccsc12 66255,C1(C(=O)NC(CNC(=O)C=Cc2ccncc2)C2CCC2)CCC2(CCC2)O1 66256,c1(NC(c2ncccc2NC(c2ccnc(Cl)c2F)=O)=O)cc(Cl)cc(Cl)c1Cl 66257,C1(NC(=O)C=Cc2ccsc2)(CF)CCN(C(C2CCC(=O)N2)=O)C1 66258,N1(C(CC(C)CF)=O)C2CCC1CN(C(=O)Cc1cc3ccccc3o1)CC2 66259,C1(C(=O)NC2C=CC(CNC(=O)CSC(F)F)C2)C2CC3C(C2)C13 66260,N1(C(C2CCN(C)C2=O)=O)C2CCC1C(F)C(NC(c1coc(C(F)F)n1)=O)C2 66261,CCC(CC(=O)N1CCCC(N2CC(C)(C)C2)C1)c1ccccc1 66262,N1(C(CCOC(C)C)=O)CC(CNC(=O)CNC(=O)C(F)(F)F)CC1C 66263,c1(C(=O)NC2C(NC(Cc3nc(C)sc3)=O)C2)ccccc1OC1CCC1 66264,C1(CN(C(=O)NC(CC=C)(C)C)Cc2ccccc2)OCCCC1(C)C 66265,C1(CC(=O)NCCCN(C(c2coc(C3CCCCC3)n2)=O)CC)COC(=O)N1 66266,C1(C(C)C)CN(C(C2CCC3(CCC3)C2)=O)CCN1C(c1cncs1)=O 66267,Cc1noc(N)c1C(N1CCC1CNC(=O)Cc1ccc(F)nc1)=O 66268,C(CC(C)C(=O)N1CCC(NC(=O)CC2CC(SC)C2)C1CC)=CC 66269,N1(C(=O)CCc2cc[nH]n2)CCCC2CN(C(C34CCCCC3C4)=O)CC12 66270,Cn1nc(C(=O)NCC2CCC2C(=O)NC(CC(N)=O)C2CC2)cc1F 66271,N1(Cc2ccc(C(=O)NCC(=O)O)cc2)C(=O)NC2(CCOC2)C1=O 66272,N1(C(CCC(=C)C)=O)CCCC12CCN(C(=O)Cn1cc3ccccc3n1)CC2 66273,CC(C)(C)C(C#N)C(=O)NC1COCCC1NC(c1cnc(S)n1C1CC1)=O 66274,C1(CCC(=O)OC)CC(OC)N(C(=O)C(c2ccc(C(N)=O)cc2)O)C1 66275,C(=O)(C1=NOC(C)C1)NCCC1(C(N(C)Cc2nc(C)sc2)=O)CCC1 66276,n1(CC(N2CCC(O)(C(C)NC(c3cocn3)=O)C2)=O)cnc2sccc2c1=O 66277,N1(C(CCc2scc(C)n2)=O)CC(NC(=O)C(c2ccccc2Cl)O)C(C)(C)C1 66278,N1(C(CNC(C2CCC2)=O)=O)CC2CCC(C1)N2C(c1ccc(O)nc1)=O 66279,N1(C(Cc2c(C)ocn2)=O)CC2(CCN(C(=O)C(c3ccc(O)cc3)(C)C)C2)C1 66280,N1(C(c2ccc(F)c(Cl)c2F)=O)CCCC2(CCN(c3ncc(CO)cn3)CC2)C1 66281,CC1COc2c(C(=O)N(CCCCN(C)C(C3C=CCCC3)=O)C)cccc21 66282,C1(C(=O)NCC(CO)NC(c2c(COC)nn[nH]2)=O)CC2C(C1)C2(F)F 66283,c1(C(N(C)CC2(O)CN(C(C(F)=C(C)C)=O)C2)=O)ccccc1Br 66284,C(N=c1[nH]c(=NC)[nH]c(=NC2CCCc3occc32)[nH]1)C1(CCC)CCC1 66285,CC#CCCCC(=O)NC(COC(C)C)C(=O)NC(c1scnc1C)C 66286,N1(C(CNS(C)(=O)=O)=O)CC(NC(=O)C(c2cccc(F)n2)(F)F)C(CO)C1 66287,C1(OCC)CC2(C1)CC2C(=O)NCC(C)CN(C)C(c1sc(C2CC2)nc1C)=O 66288,c1(OC)ccc(CNCC2CCC3(C2)CC3(F)F)c([N+](=O)[O-])c1OC 66289,c1(NC(=O)NC2CCCC(Cc3cn(CC)nc3)C2)cncc(C#N)c1 66290,c1(N(C(=O)CNC(=O)CNC(=O)C2CC2)CC)cnn(CC2CCC2C)c1 66291,c1(NC(C2C3CN(C(Cc4c(C)noc4C)=O)C2C3)=O)cnc(C#N)nc1 66292,c1(C(CC)C)nc(C)cc(=NC2CC(NC(=O)CC3CC4CCC3C4)C2)[nH]1 66293,C1(NC(=O)CC2CCCC(OC(F)F)C2)CCCN(C(c2cnn3cc[nH]c23)=O)CC1 66294,N1(Cc2c(C(=O)OCC)n[nH]c2)c2cccc(O)c2CCC1C 66295,N1(C(C2(CC#C)CCOC2)=O)CC2CC(NC(c3c[nH]cc3C3CC3)=O)CC1C2 66296,Cc1[nH]nc2c1CC(C(N1CCC(CO)(NC(=O)Cn3cccn3)CC1)=O)CC2 66297,n1(CC(=O)OC)nnnc1CN(c1ccccc1)C(=O)CCC1CCOC1 66298,C12(CNC(c3cccc(CS(C)=O)c3)=O)CCC(C1)N(C(=O)C=C1CCCC1)C2 66299,c1(C(=O)NC(C(=O)N(CCNC(c2cccs2)=O)CC)C)ccccc1Cl 66300,c1(CC)ncc(Cl)c(C(N2CCCC(NC(=O)COC3CCCCCC3)C2)=O)n1 66301,C1(CN(CCO)CC2(OCC)CCCC(C)(C)C2)Cc2ccccc2C1C 66302,CCCC(CC)CCC(=O)N1CCC(N(C)C(c2cc(N)ccc2O)=O)C1 66303,c1(C(=O)NC2CC(CNC(c3cncc(F)c3Cl)=O)C2)ccc([N+](=O)[O-])s1 66304,CC1CC2CCC(C(=O)NCCC(C)NC(c3ncc(Cl)n3C)=O)CN2C1 66305,c1(OC)cc(C(=O)NC2CCC(NC(c3ccncc3C3CC3)=O)C2)ccc1F 66306,c1(C(=O)NC2CCNCC2F)cnc2c(cnn2Cc2ccccn2)c1 66307,c1(C(N2C3(CNC(C=CC(C)C)=O)CCC2CC3)=O)cnc2c(c1)N(C)CCO2 66308,c1(CC(=O)NCC2C(NC(c3cncc(C)c3Cl)=O)C2)cccc2nsnc12 66309,N1(C(C(C2CCOC2)OCC)=O)C2CCC1CC(CNC(C1CC(F)(F)C1)=O)C2 66310,CC1CN(C(C2(C#N)CCCO2)=O)CC1CC(=O)NCC(C)S(N)(=O)=O 66311,CC1CCCC(OCC(=O)NC(Cn2cc(-c3ccccc3Cl)nn2)C2CC2)C1 66312,N1(C(C(F)=C(C)C)=O)CCC(C(F)(F)F)C(NC(=O)C=C2CCN(C)C2)C1 66313,Cc1cnccc1C=CC(=O)NCC1(CN(C)C(c2cc(O)n(C)n2)=O)CC1 66314,Cc1cc(C(=O)NC2(C)CC(C(=O)NCc3ccc(C)o3)C2)nc(O)n1 66315,C(=O)(C1=C(C)CCC1)N(C(C(N1CC(CCC#C)C1)=O)C1CC1)C 66316,C1(NC(CCCOC)=O)CCC(NC(C23CC(CN2C2CC2)C3)=O)CC1 66317,C12(CNC(c3ncccn3)=O)CCCN(C(=O)C=Cc3cccc(F)c3)C1C2 66318,C1(NC(CSCCOC)=O)CCN(C(=O)CN(C)C(c2ccc(N)cc2)=O)C1C 66319,C1(C#N)(C(=O)NCC(CC)(CC)NC(=O)Cc2cc[nH]n2)CC2C=CC1C2 66320,C1(C(N(CCCCNC(C23CCC(C)(CC2)C3)=O)C)=O)CC12CCCOC2 66321,C1(C)(C(=O)NC(CN(C(c2ccccc2SC)=O)CC)C)CC(OC)CN1C 66322,C1(NC(=O)OC(C)(C)C)CN(Cc2cc(Br)cc(Br)c2O)CC2(CCOCC2)C1 66323,CN1CC(C(=O)NC2(CNC(C3CCOC3)=O)CC2)CC1=O 66324,C1(CCCNC(C(C)c2ccco2)=O)CCCCN1C(=O)CSc1nncs1 66325,N1(C(c2nc(CC)sc2)=O)CCC2CCN(C(C3(C)CC3C)=O)CC12 66326,C#Cc1cccc(NC(C2CN(C(C3(CC(=O)OC)CC3)=O)CC2C)=O)c1 66327,c1(CN(CCOC)CC2CC=CCC2)ccc(Cl)s1 66328,c1(C(=O)NC2CC(F)(CNC(C)=O)C2)cnc(C(F)(F)F)c(F)c1 66329,C1(N(C(C(Br)=C(C)C)=O)C)CN(C(c2cncc(N)n2)=O)CC1(C)C 66330,c1(CN(c2nnnn2CCCF)CC)cc(F)c(F)c(O)c1F.C1(C)(C)CCOC1 66331,CC#CCCC(=O)NC(C)(CNC(=O)CSCC1CCCO1)C(C)C 66332,C(=O)(CC(O)CC(C)(C)C)N(CC(N1CC(C#C)C(O)C1)=O)C 66333,CCC(O)C(F)(F)C(=O)NCC(CCNC(=O)CC1(n2cncn2)CC1)OC 66334,C1(NC(CNC(CN(C)C)=O)=O)CCCC(NC(c2cc(-c3cccs3)on2)=O)C1 66335,N(C(=NCCCNc1sccc1C)N1CCN(c2ccccc2)CC1)C(C=C)C 66336,CCCC(C)CCCC(=O)N(CC(C)NC(C1(c2cccs2)CCCC1)=O)CC 66337,CN=C1NC2=NCCC3=CC=CC=CC4C(N=C(N2)N1)C4C3.c1ccc(C)cc1 66338,C1(CNC(CC(CC)NC(c2cnc(=N)[nH]c2)=O)=O)OC(=O)CC1(C)C 66339,C1(NC(=O)NCC(C(C)C)c2ccccc2)CC2(C1)CC21CCC1 66340,C=C=CCN=c1[nH]c(=NCC2CC(C)CC(C)C2)[nH]c2c1SCC2 66341,c1(C(=O)NC2CCN(C(c3c(C)[nH]cc3)=O)C2(C)C)ccc(Br)c(F)c1F 66342,c1(C(=O)NCCN(C2CCCC2)C(C2C(C(C)(F)F)C2)=O)cc2c(Cl)cncc2o1 66343,c1(C(=O)NCC=CCNC(C(C=C)O)=O)ccccc1C1CC1(F)F 66344,n1(C(C(=O)NC(CCC)C(=O)OCC)CSC)ccc2sccc2c1=O.C(C)(C)C 66345,CC1CC(C)(C(=O)NC(C)CN(C(=O)CCCn2ccccc2=O)C)CC(C)O1 66346,c1(C(N(C2CCN(C(C(CCC)C)=O)CC2)C)=O)ccc2nc(C)n(C)c2c1 66347,C(=O)(CCCCC(=O)NC1CN(C(c2ccc(C(C)=O)c(F)c2)=O)CC1O)NC 66348,N1(C(C(C)OC)=O)CCC(F)(CNC(=O)Cc2cncc(C#N)c2)CC1 66349,CCC(C)C(O)C(=O)N(CCC(C(C)C)NC(C1(C)CC(F)C1)=O)C 66350,C(=O)(C1=CCCOC1)NC(C(C)NC(=O)Cc1ccc(Cl)cc1)CO 66351,C1(NC(CC2(C=C)CN(C(=O)CC(=O)N(C)C)C2)=O)COC2(CCC2)C1 66352,n1(CC)ccc(CC(=O)N(CC(C)CNC(=O)CC(C)C2CCCCC2)C)n1 66353,c1(C(N2CC(CCNC(CCCC)=O)OCC2)=O)cc([N+](=O)[O-])oc1C 66354,c1(OC)c(C(=O)NC2CC(C)N(C(=O)Cc3cccc(Br)c3)C2)ccnc1F 66355,N1(C(c2cccc(C(C)=O)c2)=O)CCN(C(=O)C(c2ccccc2)C)C(CO)C1 66356,N1(C(C2(Oc3cn(C)nc3)CC2)=O)CCCCC1NC(=O)CC(O)C1CCCC1 66357,C1(CNC(c2cc(CNC(CC3(N(C)C)CCC3)=O)on2)=O)CCCC12CCC2 66358,N1(C(CC(C)C)=O)CC(C(=O)NCC(c2ccncc2)C)OC(C)C1 66359,c1(OCC(=O)NC2CC(C)CN(C(=O)CSCCN(C)C)C2)cc(F)ccc1F 66360,C1(CNC(C(C)OC)=O)CCCCCN1C(c1nc(C)ncc1Br)=O 66361,CCC(C)C(O)C(C)C(=O)N(C(C)C(=O)N(CC1CC1)OC)C1CC1 66362,C(=O)(C(F)(F)C(O)C(C)C)NCC1C(NC(C2CN(C(C)=O)C2)=O)CCC1 66363,C1(CCOC)(NC(C2CCCCC2O)=O)CCN(C(=O)CNc2nccs2)CC1 66364,c1(NC(CC)CNC(C2CCCSC2)=O)ncc(C#N)cc1Cl 66365,C(=O)(C1=CCOCC1)NC(C)CN(C)C(c1cc(Br)c(C2CC2)s1)=O 66366,C1(NC(=O)CCCC2CCCCC2)CCCN(C(C2CC23CCCC3)=O)CC1 66367,C1(c2n(CC=C)nnn2)(NCC2(C3CC3)CC2)CCOC(C)C1 66368,CCC(CCC(=O)NCC(CNC(=O)Cc1cnn(C)c1C)OC)OC 66369,CN1CC2CCN(C(C3(CNC(=O)CCN4CCOCC4)CCC3)=O)C2C1 66370,C(=O)(C(CC(N)=O)NC(=O)CC(C)COC)NCC(CC)(C)O 66371,C(=O)(N=c1cc(N(CCOC)C(=O)OC(C)(C)C)n(C)[nH]1)C1(COC)CCC1 66372,C1(C(=O)NCC(CCCC)NC(=O)C2=CCCCC2)CCc2nc(C)sc2C1 66373,c1(OCC)ccc2c(c1)CC(NCCC=C1CN(C(=O)OC(C)(C)C)C1)O2 66374,Cc1ccc(C(O)CNC(=O)N(CCC#N)C2CC2)cc1 66375,CCCCCC(=O)N1CCC(C(=O)N(Cc2ccccc2)OC)C1 66376,CCCCCCC(F)C(=O)NCC(C)(C(C)C)NC(c1cc2ncccn2n1)=O 66377,C1(C(=O)NC(CC)CC(=O)OC)CNC(=O)CN1C(=O)C(C)NC(=O)NC 66378,Cc1ccc(CC(N2CCCC(N(C(=O)C(C)CO)C)CC2)=O)c(C)c1 66379,Cc1cccc2[nH]cc(C(N3CCCC(CC(=O)NCc4ccccc4)C3)=O)c12 66380,CCCC(CCC)CC(=O)NCCN1CCN(C(C2CN(C)CC(C)O2)=O)CC1 66381,C(C(C)(C)C(=O)N1CCC(C)(CNC(C2(c3cnn(C)c3)CCCO2)=O)C1)OC 66382,c1(C(N2CCC(CNC(C3(C)CCCC3)=O)C2)=O)cnc(Cl)c(Cl)c1 66383,CC1(C)CC(=O)CCC1C(N1CCCC(C)(NC(=O)CCCCC2CC2)C1)=O 66384,N1(C(Cc2ccn(C(C)C)n2)=O)CC(NC(c2cc(C(N)=O)no2)=O)CCC1C 66385,c1(-c2nc(CC(C)C)nn2CCCN(C)C)cn(C)ccc1=O 66386,C(=O)(C(CC)C(F)(F)F)CNC(CC=CC(=O)NCC(=O)NCC)(C)C 66387,Cc1ccc(C)c(OCC(=O)N(CC(C)NC(=O)C(C(C)(C)C)C2CCC2)C)c1 66388,c1(C(=O)NC2CCN(C(c3nc(OC)c(C)s3)=O)CC2O)ccc2c(c1)COC2 66389,C1(NC(C(C)OCCOCC)=O)CC(OC)CN(C(=O)Cc2ccsn2)C1 66390,CCCCC(F)C(=O)NC1CCC(C)(CNC(c2cnoc2C)=O)C1 66391,c1(CC)nn(C)c(Cl)c1C(=O)NCCCC1(NC(c2cnc(O)c(F)c2)=O)CC1 66392,N1(C(C2C(C)(C)COC2)=O)CCOC2(CCN(C(=O)CCc3cnoc3)C2)C1 66393,C1(N(C(CCC(=O)OC)=O)CCC(=O)N2CC(F)C2)C2CCC1CNC2 66394,c1(SC)cc(Br)ccc1C(=O)NC1CC(C)(NC(=O)C2=CCCCC2)C1 66395,c1(N(C)C)cccc(CCC(=O)NCC2CCCN2C(=O)C(F)C2CCOC2)c1 66396,N1(C(C(COC)O)=O)CC2C3CCC(C2C1)N(c1ccc(OC)c(NC(C)=O)n1)C3 66397,N1(C(c2ncc(F)cn2)=O)CC2(CCCN(C(c3ccnc4c3CCC4)=O)C2)C1 66398,C1(NC(NCCC(C)=O)=NCCCCC2CC2)Cc2n[nH]cc2C(C(F)(F)F)C1 66399,c1(C(N(C(c2c(C)cccc2)CO)C)=O)cc2ccc(Br)cc2[nH]1 66400,c1(C(=O)NCc2c(O)ncc(C)c2)coc2c1CN(C(=O)C(C)c1cc[nH]n1)C2 66401,CCC(C)(C#N)C(=O)N(C)CCNC(=O)C(C)O 66402,n1(C(C)C)cc([N+](=O)[O-])c(=NCC2CCCCC2NC(=O)CC(C)C(C)C)[nH]1 66403,N1(C(Cc2c(C)occ2)=O)CC(CNC(c2ccsc2C#N)=O)CC1C 66404,C1(CNC(c2c(C(C)C)nn(C)c2)=O)CCN(C(c2cc(O)n(C)n2)=O)C1(C)C 66405,Cc1cn(C)nc1C(=O)NCC1CN(C(c2ccc(CO)o2)=O)CC1C(F)(F)F 66406,C1(NC(C(C2CCCCC2)C)=O)COC2(C1)CN(C(C1(C)CCCO1)=O)C2 66407,Cc1cc(F)c2ncc(C(N3CCC(NC(=O)CC(C)O)C34CC4)=O)cc2c1 66408,C1(F)(CNC(CCCOCCC)=O)CCCN(C(C2CC2CN(C)C)=O)CC1 66409,C1(n2cc(C3CCN(C)C3)nn2)CON(C(=O)C2C3CCC(C3)C2c2cn[nH]c2)C1 66410,C1(C(N2CC3CC(C)(C)C3C2)=O)CC12CCc1ccccc12 66411,c1(OC)ccc(CC(N2CCC(NC(C3(C)CS(=O)(=O)C3)=O)C(F)C2)=O)cc1F 66412,c1(CN2CCCC(C)(CNC(=O)CC3CCOCC3)C2)ccc2c(c1)CNC2=O 66413,C1(CNC(Cc2c(C)nc(Cl)cc2)=O)CN(C(C2CC2CF)=O)CC12CCC2 66414,c1(-c2nc(CCCOCCOC)nn2-c2ccc(C)c(F)c2)cc(C)cc(Cl)c1 66415,C1(NC(c2cn(C)nc2Br)=O)CN(C(=O)CCc2ncc[nH]2)CC(C)(C)C1 66416,c1(C(=O)NCCCCNC(CCCC(CCC)C)=O)sc2nccc(C)c2c1C 66417,N1(C(c2ccn(CCOC)n2)=O)CCC2(CCN(C(=O)Cn3ccc(C)n3)C2)C1 66418,c1(COC(c2ccc(OCCCc3ccccc3)cc2)=O)cccnc1Cl 66419,C12(NC(Cn3c(C)nnn3)=O)CCCC(NC(=O)C3=COCC3)(C1)C2 66420,c1(NC(C(C)N(C)C2CC2)=O)ccoc1C(=O)NCCCc1cnn[nH]1 66421,N1(C(CC2CC(CC)C2)=O)CC2C(C(N3CCCC(CCCO)C3)=O)C2C1 66422,c1(C(=O)NC2CC3CCC2N3C(=O)CCN2CCCC2=O)cnc2ccccn12 66423,c1(CNC(C)=O)ccc(C(=O)NC(C)CCNC(c2c(Cl)cnn2CC)=O)cc1 66424,S(=O)(=O)(c1ccc(Cl)nc1)N(C1C2CCC1CNC2)c1cc(C)on1 66425,N1(C(C2(C#N)C(C)C2)=O)CC=C(C(=O)NCc2cocn2)C1 66426,N#Cc1ccc(C=CCOC(C23CC(CC4CC4)(CO2)C3)=O)cc1 66427,c1(NC(C2C(CNC(c3ccc(CC)cc3)=O)OCC2)=O)cccc2occc12 66428,C1(CNC(c2n(CCOC)ncc2)=O)C(C)CCCN1C(=O)C=Cc1ccsc1 66429,N1(C(Cc2cnc(C)s2)=O)CCCC(O)(CNC(C2CC2C(F)(F)F)=O)C1 66430,CCC(C(=O)N1CCC1C(=O)N(CC(C1CCCC1)O)C)SC 66431,N1(C(CCNC(=O)CO)=O)CC(O)(C(F)C(=O)N(C2CC2)Cc2ncccn2)C1 66432,CCC(CC(F)F)C(=O)NC1(C(C)(C)C)CCN(c2ccc(C#N)c(C)n2)C1 66433,c1(NCc2cc(OC)cc(F)c2)nc2ccccc2nc1NCC1CC1C 66434,c1(C(=O)NCC(C(=O)NCCc2nc[nH]n2)N(C)C)ccc(CO)nc1 66435,C(c1ccsc1)=CC(=O)NCCN(CCOC)C(c1nscc1C)=O 66436,C(N=c1[nH]c(=NC)[nH]c(=NCC(CC2CC2)CO)[nH]1)C1C(CCC)C1 66437,C(=O)(C(F)C(C)(F)F)N(CCCOCCNC(=O)CCc1nc(O)n[nH]1)C 66438,CC1COc2c(NC(N3CCc4cc(Br)ccc43)=O)cnn2C1 66439,N1(C(CCC=C)=O)CC2CCN(C(C3CC(=O)N(CC(C)C)C3)=O)CC(C2)C1 66440,CC(C(=O)NCC1(NC(c2cc(N)c(Cl)cn2)=O)CCCCC1)C(C)C(C)(C)C 66441,c1(Cn2c(C(=O)NC(c3ccccc3Cl)(C)CO)ccn2)ccc(F)cc1 66442,n1(CC)nccc1C=CC(=O)NCC(C)(C)CNC(c1cc(=O)cc[nH]1)=O 66443,C(CCSC=O)(C(=O)N1CC(N(C)C(c2cc(C3CC3)[nH]n2)=O)C1)OC.C(C)C 66444,n1(C(C(=O)NCCN(C(CC)C)C)C)cc(CC(O)C(C)C)nn1 66445,c1(CCC(=O)N(CC(C)N(C(C(C)O)=O)C)C)ccc(Cl)cc1Cl 66446,CCC(C)(C)C(O)C(=O)N1CC(OCC(=O)NC2CCN(C(=O)NC)C2)C1 66447,C1(CC(=O)NCCN(C(=O)CCC2CC2(F)F)CC)CCCOCC1 66448,c1(C(=O)OC)cc2c([nH]1)CCN(C(=O)C(N1CCCC(C(O)C(F)F)C1)=O)C2 66449,C1(NC(=O)CCC2CCCO2)CCSC12CN(C(=O)C=Cc1cncnc1O)C2 66450,C12(C(=O)NC(c3n(CC)ccn3)C)CC(CN1C(c1cc(O)cs1)=O)C2 66451,C1(CCNC(C(C)CN2CCOCC2)=O)CCCCN1C(c1cn(C)c(O)n1)=O 66452,N1(C(C)C)CC(C(=O)NCC(C)NC(=O)C(C)(C)C2CCCO2)CC1=O 66453,C=C(C)CCCC(=O)NC(CNC(C1CCCN(C(C)C)C1)=O)CC 66454,C1(C(=O)NCCCOCCNC(CC2CC(SC)C2)=O)CC2(CCC2)C1 66455,C(=O)(C(C(C)C)NC(=O)COc1cccnc1)OC 66456,c1(C(=O)NCC(CNC(C2(N(C)C)CCCOC2)=O)O)ccc2c(n1)NCC2 66457,CC1CC(C)(C(=O)NCc2cccc(NS(C)(=O)=O)c2)CC(C)O1 66458,N1(C(CCCC)=O)CCC(NC(=O)CCc2ccccn2)C1C(C)(C)C 66459,Cc1ccc(CO)c(NC2(c3nnnn3C3CCCCC3)CCOC2C)c1 66460,c1(CNC(C(N2CC(F)(C(=O)OC)C2)=O)=O)cc2ccccc2nc1Cl 66461,C1(CC=C)CCCCN1C(=O)Cc1cn(C(C)C)cn1 66462,c1(SCC(=O)N(CCCCN(C(=O)CCF)C)C)nccc2ccccc12 66463,C1(C)(CC)CCN(C(c2cc(CNC(C3CN(C(=O)NC)C3)=O)cs2)=O)C1 66464,CC1C(NC(=O)C=Cc2cocn2)C(C)CCN1C(=O)C=Cc1ccnn1C 66465,N1(C(CCC#CC)=O)CCCCC1C1CCCN1C(=O)C=C1CCCCC1 66466,C#CCC(CC#C)C(=O)N1CCCCC(CNC(c2scnc2COC)=O)C1 66467,C1(CC(=O)NCCC2CN(C(=O)C3CC3)C2)SC2=NCCN2C1=O 66468,C1(C(N2CCC(Nc3ncnc4sccc34)CC2)=O)CCCC(F)(F)CC1 66469,N(C1CCCc2nc(O)ccc21)C(=O)COC1CN(C(C2CCOCC2)=O)C1 66470,C1(C(=O)NCc2n(CCC)ncn2)CC(N=[N+]=[N-])CN1C(=O)C(C)C1CCCC1 66471,C12(NC(COc3cccc(C)c3)=O)CCN(C(=O)Cc3cncnc3)CCC1C2 66472,CC1CCC(C)(C(=O)NCC2(C)CCN(C(=O)Cn3cncn3)C2)C1 66473,c1(-c2scc(C)n2)cccc(C(N2CCSCC2CCNC(C2CC2C)=O)=O)c1 66474,C(C)(C(CC(=O)NCC1(C)CC(C)(C)C1)NC(=O)C(C)C(F)(F)F)OC 66475,CC1CN(C(c2ccc(Br)o2)=O)CC1NC(c1cn(C(C)(C)C)nn1)=O 66476,C1(NC(c2c(C)nc(C)[nH]2)=O)CC2CCC(C1)N2C(=O)CC1OC(C)(C)OC1=O 66477,N1(C(COC)=O)CC(NC(=O)CCCOC(C)C)CC12CCCOC2 66478,N1(C(c2n(CC=C)ccc2)=O)CC(O)CC1CNC(=O)CNC(=O)NC1CC1 66479,c1(CNC(c2n(CC)nnn2)(C)CC2CN(C(=O)OC(C)(C)C)C2)ccccc1Br 66480,C12(CNC(CCC(CC)C)=O)COCCN1CCN(C(C1(C)CCOCC1)=O)C2 66481,N1(C(C(=O)NC2CC2)=O)CCC(C(N2CCC(CC(F)F)C2)=O)(CO)C1 66482,c1(OCC)cc2ccccc2cc1C(N1CCC(N(C)C(C2C=C2C)=O)CC1)=O 66483,Cc1n[nH]c2cnc(C(=O)NC3CC(CNC(=O)C=C4CCN(C)CC4)C3)cc12 66484,N1(CCS)CCC(c2cnn[nH]2)C1.C1(N2C(=O)CN(C)CC2)CC(C#N)C1.CO 66485,c1(C(N(CC(C)NC(C2(CC#C)CC2)=O)C)=O)cnc2c(cnn2C)c1N 66486,c1(C(=O)NC2C(NC(c3cnc(C(N)=O)s3)=O)COC2)cnc2n1CCS2 66487,C1(NC(C(CC)Oc2cccc(F)c2)=O)CCN(C(C2(C)C=CCC2)=O)CC1C 66488,C1(CC)C(NC(=O)CCN(S(C)(=O)=O)C)CCCN1C(=O)C(C)CC(N)=O 66489,N1(Cc2ccc(OC)nc2C)CCC(=O)N(CC2(n3cncn3)CC2)C1=O 66490,N1(C(c2cn(C)nc2)=O)CCC(CNC(=O)CN2CCCS2(=O)=O)C12CC2 66491,c1(C(C)C)ncccc1NC(=O)C(C1CCN(C(C2CCCC(C)C2)=O)CC1)C 66492,C1(C)(C(N(CCCCNC(=O)CCc2ccncc2)C)=O)COC(=O)OC1 66493,CCC1=C(C(=O)NC23CCC2CN(C(=O)CC2=CCOCC2)C3)CCCO1 66494,C1(NC(c2cnc(Cl)cc2Cl)=O)CCC2CCN(C(c3cc(Cl)no3)=O)C1C2 66495,CCCCCCN(C)CC1C(NC(CNC(C2(C)CC(C(=O)OCC)C2)=O)=O)C1 66496,c1(C(N(CCCN(C(C2CC(SC)C2)=O)C)C)=O)c[nH]c2cccc(F)c12 66497,C1(NC(=O)C=CC2CCCC2)CCCCC1NC(=O)CSc1ccccc1Cl 66498,CCC(=O)CCC(=O)N1C(CC(=O)NC(C2CCOCC2)CC)C2CCCC12 66499,N1(C(C(C(C)C)SC)=O)CC2CCCC(C1)N2c1nccc(-n2ccnc2)n1 66500,c1(C(C(C)NC(c2cscn2)=O)N)ccccc1 66501,N1(C(C(c2cnn(C)c2)OC)=O)CCCC(n2cc(-c3cccc(F)c3)nn2)C1 66502,N1(C(CC2(C)CC2(Cl)Cl)=O)CC(NC(c2ccnc(OC(F)F)c2)=O)CC1CO 66503,C1(NC(CCOCC)=O)CN(C(c2ccc(C3CC3)c(C)c2)=O)CC12CC2 66504,c1(C(=O)NCC(CC)NC(c2cc3ccncc3[nH]2)=O)ccc2oc(O)nc2c1 66505,C(=O)(C(O)C(F)(F)F)N1C(C2(NC(CCOCCOC)=O)CC2)CCC1 66506,C12(C(=O)NC(C)Cc3nc[nH]n3)CC(CN(C(=O)C(O)CN3CCCC3)C1)C2 66507,N(C(=N)N1CCC(Cc2ccccc2)C1)C(C)CC#N 66508,c1(C(=O)NC(CC)CNC(=O)CCc2cnn(C)n2)cnc(C(F)(F)F)cn1 66509,Cc1cccc(C)c1SCC(N1CCCC(N2CC(F)(F)C2)C1)=O 66510,C(CC(C)C(=O)N(C1CCCCC1NC(=O)Cc1ccsc1Br)C)=CC 66511,N1(C(c2cn(CCNC(c3c(CC)nccc3)=O)nn2)=O)CCCC(CC)CC1 66512,C1(CC(=O)NC(CC)CN(C)C(C2(c3cc[nH]n3)CCC2)=O)CC(C)(C)CO1 66513,CC1CN(C(=O)C=CCF)CCC1NC(c1nn(C)nc1Br)=O 66514,c1(SC)cc(C)ccc1C(=O)NCCN(C(c1ccn(C2CC2)n1)=O)CC1CC1 66515,Cc1cc(C(=O)NC2CSC(C)C2)nc(N(C)C)n1 66516,N1(C(C2C(C)C2)=O)Cc2nccn2CC(NC(=O)Cc2ccnc(Br)c2)C1 66517,c1(C(N(CCCNC(=O)C2=COCC2)CCO)=O)ccc2nn[nH]c2c1 66518,N1(C(CC=CCCCCC)=O)CCCC1C=CC(=O)NC(c1nnc(C)o1)C 66519,C1(CC(=O)NC2(CNC(=O)Cc3cccc(Cl)c3)CCOC2)CCCC1(F)F 66520,C1(COC)(NC(=O)CSS(C)(=O)=O)CCCN(C(=O)C(C)(O)C2CC2)C1 66521,c1(C(=O)NCC2CCN(C(CCOCC#C)=O)C2)scc(C)c1OC 66522,C1(NC(C(c2ccncc2)C)=O)CCC2CC1CN2C(C1CCCNS1(=O)=O)=O 66523,n1(CC(N2CC(SC)C(NC(C3(C)CCCO3)=O)C2)=O)cnc([N+](=O)[O-])c1 66524,CC1(C)CCCCC1C(=O)NCC1CC(NC(C2CCC23CCC3)=O)C1 66525,N1(C(C2CC(C)N2C(=O)COC2CC2)=O)CC=CC12CCCC2 66526,Cc1[nH]nc(CO)c1C(=O)NOCC(C(C)C)NC(=O)CCNC(C1CCC1)=O 66527,C1(F)(CNC(C(C)SC)=O)CCN(C(=O)C(C)(C)C2CC2)CC1 66528,C(=O)(C(C)(C)CCC#N)NC(C1CCCN(C(c2[nH]ccc2C2CC2)=O)C1)C 66529,N(C1CCc2ccccc21)C(c1cncc(NC(c2nccc(OC)c2)=O)c1)=O 66530,c1(C(N2CC(OCCNC(=O)CCOCC(F)F)C2)=O)nc2cc(F)ccc2s1 66531,N1(C(C(C(C)C)SC)=O)CC2(C1)CN(C(C1CCC(=O)N1C)=O)CC2CO 66532,C1(C(N(C)CCN(C)C(C2COCCC2(F)F)=O)=O)CCn2cncc2C1 66533,Cc1cccc(C(F)C(=O)NCC(C)N(C(=O)CN2CC3CC3C2)C)c1 66534,Cn1cnc2c(NCC3C4CN(C(c5ncoc5C5CCC5)=O)CC34)ncnc12 66535,c1(CC(N2CCC(N(C(CSCCOC)=O)C)C2)=O)cccnc1OC(C)C 66536,Cc1ccc(SCCC(=O)NC2CC2NC(C2CCS2(=O)=O)=O)cc1 66537,N1(C(COCc2c(C)cccc2)=O)C2CCC1CC(NC(=O)CC13CC(C1)C3)C2 66538,C(=O)(CCN=c1cc[nH]c2ccccc12)N(C)C 66539,N1(CC)N=C(C(=O)NCC(C)NC(c2cc(C)nc(N(C)C)n2)=O)CCC1=O 66540,c1(C(=O)NCC2(NC(C3C(OCC)C3)=O)CCC2)cc2ccc(Cl)cc2c(O)n1 66541,C(=O)(C(CC(C)C)NC(=O)CC(COC)SC)NC.C12CN(C1)C2=O 66542,c1(C(=O)NCCCN(CC)CC2CC2C)cc(-c2ccns2)on1 66543,CCCCC(C)(F)C(=O)NC(C)CCCCNC(=O)Cc1cnc(C(F)(F)F)s1 66544,c1(C(=O)NC(CC(F)F)C(=O)NCC(Cl)=CCl)ccc2n[nH]cc2c1 66545,c1(CC(=O)NCC(C)CN(C(=O)C(C)CC2CCCC2)C)ccn(C(F)F)n1 66546,N1(C(c2c(COC)scc2)=O)CC(O)C(O)C1CNC(C1(c2cc[nH]n2)CC1)=O 66547,N1(C(C(CC)(C)O)=O)CCCCC(CNC(=O)CCc2csc(=N)[nH]2)C1 66548,N1(C(C(=O)NCC)=O)CCN(C(C2CCN(C(=O)NC)CC2)=O)CC(O)C1 66549,Cn1cccc(C(=O)NC2CC(C(N3CCC(F)(CF)C3)=O)C2)c1=O 66550,C#Cc1cccc(CC(=O)NC(CCC=C)C(=O)N(CC2=CCCOC2)C)c1 66551,Cc1ccccc1-n1nc(CC2CC2)nc1-c1cnc(C(F)F)s1 66552,c1(NC(C2CCCC(Nc3ccnc(C)n3)C2)=O)ccc2c(c1)C(=O)NCC2 66553,C(=O)(C1=NOC2COCC12)N1CCC(C)(C(=O)NCc2c(C)oc(C)c2C)C1 66554,N1(C(C(CC=C)OC)=O)C(CNC(=O)C(CC2CC2)OC)CC2CCCC12 66555,c1(N(CC(=O)NCCNC(C2(C(C)(F)F)CCC2)=O)C)ccc(Cl)nn1 66556,C(=O)(CCC(C)(C)N(C)C)NCC1(C(=O)NC2C(C)N(C)CC2)CCCO1 66557,c1(C(N(C(CCNC(c2cc(C(C)C)[nH]n2)=O)C)C)=O)cc2cccn2c(O)n1 66558,C1(CNC(Cc2ccn(CC(C)C)n2)=O)CCN(C(=O)COCCCF)C1(C)C 66559,CCC(C)C(C)(O)CNC(=O)C(C)(CNC(=O)Cc1cc[nH]c1)CC 66560,N1(C(C(CC(C)C)C)=O)CCCC2CN(C(C3(F)C(C)(C)C3(C)C)=O)CC12 66561,C(=O)(C1=C(C(F)Cl)N(c2ccc(C)cc2)C(=O)NC1c1ccc(F)cn1)OCC 66562,c1(C(C)C)nccc(C(=O)NC2CC(NC(=O)Cc3ccc(Br)cc3)C(O)C2)n1 66563,c1(C(=O)NC(C2CN(C(C3(C)CCCCO3)=O)C2)C)ccc(F)c(F)c1F 66564,S(=O)(=O)(c1cccnc1N1CCc2oc(C)nc2C1)NC(CCC)CC 66565,c1(NCc2cccc(C(N)=O)c2)ncccc1S(=O)(=O)N1CCC2(CCCC2)C1 66566,CC(F)(F)CN=c1[nH]c(=NCC2(CCO)CCOC2)[nH]c2c1COCC2 66567,c1(SC)cccc(C(N2CCC(NC(=O)CN3CCC(O)CC3)C2)=O)n1 66568,c1(CC(N2C(CNC(C3CCCOC3)=O)C=CC2)=O)c[nH]c2ccc(Cl)cc12 66569,N1(C(C(=O)NCC)=O)CCCC2CCN(C(=O)C=COCC)CC12 66570,c1(C(N(CC(CNC(c2cn(C(C)C)nc2)=O)O)C)=O)cc2cccnc2s1 66571,c1(C(C)C)ccc(C(=O)N(CC(C)NC(c2c(Br)nnn2C)=O)C)c(O)n1 66572,N1(C(COCC#C)=O)CCCCC12CN(C(=O)C(O)C(C)C)C2 66573,C1(C(N2CC(n3cc(COCC(=O)OC)nn3)C2)=O)CCC(N=[N+]=[N-])C1 66574,N1(c2ccc(SC)s2)CCN(C(=NCC(=O)NC(C)C)NCCCC(F)F)CC1 66575,c1(C(=O)NC(CCNC(C(c2cccs2)SC)=O)C)cn(C)c(=O)n(C)c1=O 66576,C(=O)(C(CCOCCO)NC(=O)Cc1cccc(O)c1)NC(CC(=O)NC)C 66577,c1(C(=O)N(C(C)(C(=O)O)C2CCC2)CCO)ccc(C(N)=O)cc1.n12cc(nn1)C21CC1 66578,CC1=CCSC1C(=O)NC1(CCNC(=O)CCC2CCCCO2)CCC1 66579,c1(C(N2C3C(NC(C4(C#C)CCC4)=O)CC(C3)C2)=O)cc(F)c(OC)c(F)c1N 66580,C1(C(=O)NCC(CCNC(C(CC)COC)=O)OC)OC(C)(C)OC1(C)C 66581,N1(C(CC(C)N(C)C)=O)CCC(C)(C(=O)NCCCC(N)=O)CC1 66582,N1(C(c2nc(OCC)sn2)=O)CCC(CCNC(=O)C(CCO)N(C)C)CC1 66583,N1(C(C2(CC#C)CCOC2)=O)C2CCC1CC(NC(=O)Cc1csc(=N)[nH]1)C2 66584,c1(C(=O)NCC2(F)CCCN(Cc3n(C)ccc3)C2)cc2ccccc2o1 66585,C1(C2CCCO2)(C(=O)NC2C(C)CCN(C(CN(C)CC)=O)C2)CCCO1 66586,Cc1ccc(F)cc1CC(N1CC2(C)CC1C2NC(C1CCC1)=O)=O 66587,N1(C(c2c(C(=O)OC)c(C)[nH]n2)=O)CCC(NC(c2cnc[nH]2)=O)C(F)C1 66588,c1(C(=O)NCCC2(CNC(C3(C#N)CCCO3)=O)CC2)coc2c1C(=O)NCC2 66589,c1(C(N2CCC(C(C)NC(CCC(=C)Cl)=O)C2)=O)cncc(Cl)c1C 66590,c1(N2CCC(COC)(CO)CC2)nc(NCC(C2CC2)OC)nc2c1ncn2C 66591,CC(CCC(=O)NC(c1ccccc1)(C)C)NC(C1CNC(=O)O1)=O 66592,C(c1cccnc1)=CCN(C(C(C)N(C(c1c(C)c[nH]n1)=O)C1CC1)=O)C(C)C 66593,c1(N)cncc(C(c2cn(CC(C(=O)N3CCCC3C(=O)O)F)nn2)=O)c1 66594,C=C1CC2CCCC(C1)N2C(=O)CCCCCCNC(c1cncnc1)=O 66595,N1(C(CCCc2onc(C)n2)=O)CC(NC(c2c(Cl)c(C)nn2C)=O)CC(C)C1 66596,c1(C(N2CC(C(=O)Nc3ccc(OC)nc3)C(O)CC2)=O)ccc(C#N)c(F)c1 66597,C1(NC(C(C(C)C)O)=O)CN(C(c2cnc(=N)[nH]c2)=O)C(C)(C)C1 66598,C12(NC(COCCC)=O)CCOC(CNC(c3cn(C)nn3)=O)(C1)C2 66599,Cc1ccc(OCC(=O)NCC2CC(CNC(c3cncc(Cl)c3)=O)CO2)cc1 66600,C(=O)(CCCCc1ccc(F)cc1)NCC(C)(CO)NC(=O)CCc1ccco1 66601,c1(CC)cc(C(=O)NCc2cn(CCNC(=O)CCc3cn[nH]c3)nn2)ncn1 66602,C=CC1OCCC1C(N1CCC(C(C)(C)NC(c2ocnc2C)=O)C1)=O 66603,CC1(C)CCCCC1=CC(=O)NC1(C)CCN(C(C2OCCOC2(C)C)=O)C1 66604,C1(C(=O)NC(CC)CNC(C2(CC(C)C)CCNC2=O)=O)CC2C=CCC(C1)C2 66605,c1(C(C)NC(C(COCC)NC(=O)C(C)C2CCCC2)=O)cccc(C)n1 66606,C(=O)(C(C(C)(C)C)n1cc(C2CCCCCC2)nn1)NCC(C)CC1CCC1 66607,C1(CNC(=O)C2=CCCCO2)CC12CCN(C(C1C3(CCC3)C13CCC3)=O)CC2 66608,CC(C)C1=NOC(C)(C(=O)NCC(C)(F)CNC(=O)C2=NOC(C)C2)C1 66609,N1(C(CC(C)SC)=O)CCC(O)C(NC(C2SC3C=CC2CC3)=O)C1 66610,N1(C(C(CCOC)(C)C)=O)CCS(=N)(=O)C(C)C1 66611,C1(O)(C(C)NC(=O)C=Cc2cc[nH]n2)CCN(C(c2nncs2)=O)C1 66612,C1(NC(C2OCCC(C)C2)=O)COCCN(C(C2CCCSC2)=O)C1 66613,Cc1cc(CC(=O)N(C2CCN(C(C3CC(C)(C)C3)=O)CC2C)C)cc(F)c1 66614,C1(CNC(COCC(=C)C)=O)CCN(C(=O)Cn2nc(O)ccc2=O)CC1C 66615,C(=O)(C(C(C)(C)C)NC(C1CC12CCN(C(c1noc(C)c1C)=O)C2)=O)NC 66616,c1(C(N2CCC(=CC(CC)C)CC2)C(=O)NCCCSC)ccc(F)nc1C 66617,C#CCCCC(=O)NCC1(CNC(c2ccc(C(C)=O)o2)=O)CC12CCC2 66618,C(=O)(C(C(C)(C)C)NC(C)=O)NCCN(C(CCOCC#C)=O)CCOC 66619,C1(CCC=C)(C(=O)NCc2sccc2C)CN(C(=O)CCn2ccnn2)C1 66620,CCC(CC(=O)NCC1CCCN(C(=O)CCC(F)F)C1)SC 66621,C1(C(=O)OCC)C2CC(NC(c3ccccc3OC)COC(F)(F)F)CC12 66622,C1(NC(c2cc(C)ns2)c2nnnn2C2(C)CC2)CCc2ccccc2C1 66623,CC(C)C(C(=O)NCC1CN(C(=O)CN2CCCCC2=O)CC1O)N1CCCC1 66624,N1(C(C(C(C)C)n2cnnc2)=O)CCC2(C1)CN(C(c1cc(C#N)on1)=O)C2 66625,c1(CC(=O)NC(C)(C)CNC(c2cccc(CF)c2)=O)ccc2c(c1)COCC2 66626,c1(C2(C(=O)NCCCNC(=O)C(O)CN3CCCC3)CCC2)c(F)cccc1F 66627,C1(CC)CCC(C(=O)NCC2(C(=O)NCc3nc(C)cs3)CCCC2)O1 66628,c1(OC)cc(Cl)ccc1C(N1CCCCC1CN(C)C(C1(CO)CC1)=O)=O 66629,N1(C(C2C=C(C)CS2)=O)CCCCC(N(C(=O)CSc2nccn2C)C)C1 66630,c1(C(=O)NCC(CNC(C(N2CCOCC2=O)C)=O)(C)O)cccc(F)c1O 66631,Cc1sc2ncc(C(=O)NCC(=C3CN(C(=O)C(C)(C)C)C3)F)n2c1C 66632,C=C(F)C1(CC(=O)NC2CC(CCNC(=O)NCCCl)C2)CCOCC1 66633,c1(C(N2CC(=C(CNC(Cn3c(C)ccn3)=O)F)C2)=O)ccc(F)c(O)c1F 66634,CCC1=C(C(=O)NC(CNC(c2cn(CC)c(C)n2)=O)CC(F)(F)F)SCCO1.CC 66635,c1(CC(N2C(CNC(C(CC)(C)CC)=O)CC2)=O)cn2cc(F)ccc2n1 66636,C12(CNC(c3ncc(CC)nc3)=O)CCCCC1N(C(=O)CC1(CO)CC1)CC2 66637,c1(-n2c(C3COC(=O)N3C)nc(C(C3CC3)OC)n2)ccc(Br)c(F)c1 66638,Cc1cc(C(N2CC(CNC(C3CCCC(=O)N3C)=O)C3(CC3)C2)=O)nnc1O 66639,Nc1cc(C(N2CCC(=CCNC(c3cccc[n+]3[O-])=O)CC2)=O)cnc1N 66640,N1(C(C(C)Cc2ccccc2)=O)CC2(CCC2NC(c2cc(Cl)no2)=O)C1 66641,C1(C(=O)NCC(CC)n2cccn2)(NC(c2cc(CO)on2)=O)CCC(C)(C)C1 66642,C1(NC(C(CC)C)=O)CN(C(c2ccc3n[nH]cc3c2)=O)CC(C)(C)C1 66643,c1(OC)cc(C(N2CCC3(NC(c4nccnc4C)=O)CC3C2)=O)cc(Br)c1 66644,c1(CC)scnc1C(=O)NC1CCC1NC(=O)CNC(c1ccoc1)=O 66645,c1(C(c2cn(CCO)nn2)OC(C(CCC)(F)F)=O)ccc(OC)c(OC)c1C 66646,N1(C(C=CCCC)=O)CCC(C)C(CNC(C2(COC)CCCO2)=O)C1 66647,CCCCCCC(C)(C)C(=O)NC(CNC(c1cc(C)no1)=O)CCC 66648,N1(C(C(CSC)C)=O)CCC2C(C(=O)NC(c3cc(C)on3)C)C2C1 66649,N1(C(C(CC)CC)=O)CCC(C2CCN(C(=O)COC)CC2)CC1 66650,N1(C(C2C(CCC)CCC2)=O)CC2CC(C(=O)NCC(F)CO)(C2)C1 66651,n1(CC(=O)N(CCC2N(C(C3C(CC)C3)=O)CCCC2)C)cccc(N)c1=O 66652,N1(C(C2(CC#C)CCOC2)=O)CC2CCC2(CNC(=O)Cc2cnn(C)c2)C1 66653,C(=O)(C1=CCCOC1)N(C1CCCC(N(C(=O)Cn2cc(Cl)cn2)C)C1)C 66654,C1(NC(CC(=O)NC)=O)CN(C(=O)C(C(C)C)C(C)C)CC12CCCC2 66655,c1(C(N(CCNC(C(C(=O)OC)F)=O)CC2CC2)=O)coc2ccc(OC)cc12 66656,c1(CC(=O)NCC2CC(NC(=O)CC3(O)CCOCC3)C2)cncnc1O 66657,CC1CN(C(C2CCCC2F)=O)CC(C)N(C(=O)Cc2cc(Cl)cs2)C1 66658,c1(C(C(=O)NCC)N(CC(=O)Nc2cccc(C)c2)C)cn2cc(Cl)ccc2n1 66659,C(=O)(CCCC(N)=O)NC1CN(C(C=CCOC)=O)C(C)C1 66660,C1(C(=O)NC2C(OC)CN(C(C3CCN(C)C3)=O)C2)CSC(c2ccccc2)=N1 66661,C1(NC(c2c(C(C)C)occ2)=O)CN(C(c2sccc2Br)=O)CC1F 66662,C1(O)(CCNC(CC#N)=O)CCCN(C(c2cccc(C(F)(F)F)n2)=O)C1 66663,C(=O)(C(CCC(C)C)NC(C1CC2CCC(C1)O2)=O)NCC(C(=O)OC)OC 66664,N1(C(C(CC)n2cccn2)=O)CCC(O)(CN(C)C(C2CCC=CCC2)=O)C1 66665,N1(C(Cc2nc(C)sc2)=O)CC(NC(=O)CCC(=O)c2ccc(O)cc2)C(C)C1 66666,c1(C(N2CCOC(C3CCCOC3)C2)C(=O)NCCOC)cnc(C(=O)OC)nc1 66667,Cc1cnn(CCCNC(=O)C(CN(C)C)NC(C2CC2C(N)=O)=O)c1 66668,c1(C(N2CCC(NC(C=C(CCC)C)=O)(CO)CC2)=O)cccc2c1C(=O)NC2 66669,C12(C(=O)NCC(C(C)C)(C)NC(c3cocn3)=O)CCCC1CC(=O)C2 66670,CC1CC(C(=O)OC(C)(C)C)CN1C(=O)Oc1c(NC(N)=O)cccc1 66671,C#CCC(CC(=O)OC)NC(=O)C(CNC(=O)C1=C(Cl)CCC1)CCC 66672,c1(-c2n(CC=C)c(N(CCCO)CC)nn2)c(OCCC)ccc2ccccc12 66673,c1(C(N(C)CC2(NC(Cc3c(C)nc(C)s3)=O)CC2)=O)ccc2oc(O)nc2n1 66674,c1(NC(c2ccc(OC)s2)=O)cn(C)c(C(=O)NCC2CC(=O)N2)n1 66675,c1(C(=O)NC2CC(NC(C3(CC)CCOC3)=O)C2)cnc2cccnn12 66676,CC1CCC(NC(=O)CNc2ccccn2)CN1C(C1C2CCCOC12)=O 66677,C(=O)(C(C)(CSC)NC(c1cc(Cl)cs1)=O)NCC(COC)C 66678,CC(C(=O)N1CC(c2ocnc2CNC(=O)Cn2cncn2)C1)P(C)(C)=O 66679,CCC(CC(=O)N1CC(CNC(=O)CN2CC3C=CC2C3)CC1C)C1CC1 66680,c1(NC(C2C(C)C2c2ccccc2)=O)ccccc1C1CCCC1 66681,c1(C(=O)NCC(C2CC2)NC(C(CC)N(C)C)=O)cnn(C)c1S(C)(=O)=O 66682,C1(NC(C2C(OCC)C2)=O)CN(C(c2cccnc2C(F)(F)F)=O)CC1(C)C 66683,CCC(C)CC(=O)N1CC(C(=O)NCc2cc(C3CC3)on2)C(C(C)C)C1 66684,Cc1ccc(C(=O)NC(C)CCNC(c2nc[nH]c2C(F)(F)F)=O)c([N+](=O)[O-])c1 66685,c1(C(N2CCCC(N(C(=O)C(O)P(C)(C)=O)CC)C2)=O)ccc2oc(=N)[nH]c2c1 66686,c1(C(N(C2CN(C(C3(CF)CC3(F)F)=O)CC23CC3)C)=O)ccc(CO)c(Cl)c1 66687,C(CCC(=O)N1CC(CNC(=O)C(C)CN2CCCCC2)C1)OC 66688,C1(N(C(C(C)OCCOC)=O)C)CCCC2CN(C(=O)CCc3cccs3)CC12 66689,C1(C(C)(C)C)C(NC(=O)CC2CCC2(C)C)CCN1C(=O)CCCn1cccn1 66690,N1(C(CC23CC(C)(OC2)C3)=O)CCCCCC(NC(c2scnc2C2CC2)=O)C1 66691,C1(OC)CCCN(C(=O)CCC2CCN(C(=O)C(O)Cn3cncn3)C2)CC1 66692,C(CC(CC)C(=O)NC12CCC(C1)N(C(=O)CSc1nnc(S)s1)C2)=CC 66693,N1(C(C2(C)C(C(=O)OC)CC2)=O)CCN(C(c2cnns2)=O)C(CCO)C1 66694,Cc1cccc(OC2CCN(C(=O)C(=O)NC3(C#N)CCOC3)CC2)n1 66695,N1(C(C23C(CN(c4c(C)cncn4)C2)C3)=O)CCC(O)(CF)CC1 66696,C1(CNC(C(C)NC(N)=O)=O)CN(C(=O)CC2(C#N)CC2)CCC12CCOCC2 66697,C12(CNC(CCOCCOC)=O)CSC(C1)C2 66698,c1(C(=O)NC(CCNC(COCCC#C)=O)C)cc(Cl)cc2ccccc12 66699,C(C)(C(=O)NC1(CN(C)CC(=O)CC2CCC2NC)CSC1)OCCOC 66700,Cc1nc[nH]c1CC(O)C(=O)N(CC(C)N(C)C(c1cn(C(C)C)nn1)=O)C 66701,C1(NC(C(CCSC)O)=O)CC2CCC(C1C)N2c1ncnc2onc(C)c12 66702,c1(NC(C2(C)CCN(C(=O)C(=O)Cc3ccc(O)cc3)C2)=O)ccc(Br)nc1Br 66703,N1(CCN2CCCC(C(=O)OC)C2)CC(=O)CCC1=O 66704,c1(COC)ccoc1C(=O)NCC(CNC(=O)Cn1[nH]cnc1=N)CO 66705,C1(C)(CC)CCN(C(C2CCCCC2(C)NC(=O)CN=[N+]=[N-])=O)CC1 66706,C1(CC(=O)NC2(CC)CN(C(=O)COCCOC)C2)CC(c2ccccc2)=NO1 66707,C1(CNC(CC2CCCC(C)C2)=O)CC(C)(C)CN1C(=O)CC1C=CCC1 66708,N1(C(CC(C=C)C)=O)CCN(C)CC1C(=O)NCCC12CC(CO1)C2 66709,c1(OCC(N2Cc3nnsc3C2)=O)cc(Br)cc(F)c1F 66710,C(=O)(CC(C(F)(F)F)c1ccon1)NCCCNC(C1=NOC(C)C1)=O 66711,c1(CC)[nH]nc(C(N2CC(OC)C(NC(c3ccc(CC)[nH]3)=O)C2)=O)c1[N+](=O)[O-] 66712,c1(CC(=O)NC2C(C)CN(C(c3cc(CO)on3)=O)C2)ccc2c(c1)CC2 66713,CC1CCOC(C(=O)N(C(C(=O)N2CC(n3ccnn3)C2)C2CC2)C)C1 66714,C1(C(=O)OCC)CCC(F)(CNC(=O)NCC2CCOCC2(F)F)CC1 66715,C1(C(N2CCC(C)(O)C2)=O)CC2(CCN(Cc3cc(F)c(F)cc3Cl)CC2)CO1 66716,c1(C(=O)NC(c2ccccc2)C(C)NC(CCSC)=O)cc2scc(C)c2[nH]1 66717,c1(OCC)ncc(C(=O)NC2CCCC2CNC(c2ccsc2OC)=O)s1 66718,C(=O)(C(C)CCCC(C)C)N(CC(CC)NC(=O)CC1CC(=O)NC(=O)C1)C 66719,CC(C)CS(=O)(=O)N1CCSC(C(N2C(C)CCC2C)=O)C1 66720,N1(C(c2cccc(C(=O)NC)c2)=O)C2CCC1CN(C(=O)C1=CC(C)(C)C1)CC2 66721,O=C(C1=CCCC1)NCC1(CNC(c2cnc(-c3cccs3)o2)=O)CC1 66722,C12(CNC(C(F)=C(C)C)=O)CCC(CC1)N2C(=O)C=C1CCC(C(C)(C)C)CC1 66723,C1(NC(C(CCC)O)=O)CCCCCN(C(=O)C(=Cc2ccccc2)OC)C1 66724,Cc1ccc(C)c(C(=O)NCC2(C(=O)NC(CO)C3(O)CC3)CC2)c1 66725,C1(CNC(CC(C(C)C)C)=O)COC(C)(C)CN1C(c1cc(O)cc(O)n1)=O 66726,C1(C(=O)NCC(=O)OCCCC)CCC(C)(C)N(C(=O)CCOC)C1 66727,Cc1ccn(CC(C)(O)C(=O)N(CC(C)NC(c2ccco2)=O)C)c(=O)c1 66728,c1(C(=O)OC)cc(CN(c2ncc(F)c(C)n2)C2CCNCC2)cc(F)c1 66729,S(=O)(=O)(c1cc(C)c(Br)cc1C)NCC1CC2(CC(OC)(OC)C2)C1 66730,C#Cc1cnn(C)c1C(N1CCCC(C(=O)NCCC(C)CCO)CC1)=O 66731,C1(C)(CC)CC(NC(C23CC2CN(C(C2CC=CC2)=O)C3)=O)CCO1 66732,c1(C(=O)NC2(CO)CC2)sccc1CO.C1(C(=O)OC)(N(C)C=O)CC1 66733,N1(C(=O)CSC(F)(F)F)CCN(C(C2(CCF)CC2)=O)CC(O)C1 66734,C1(NC(c2c(OC)csc2)=O)CN(C(c2cnc(C)[nH]2)=O)CC1O 66735,C1(C(N2CC(O)(CCNC(C3C(C)C3)=O)C2)=O)CCc2cc(Br)ccc2O1 66736,C1(NC(C2(C)CC2)=O)CC(C(F)C(=O)NCCn2cnnc2)C1 66737,N1(C(C(CC)O)=O)CCCC(CNC(=O)Cc2ccc(OCC(F)(F)F)cc2)C1 66738,C1(NC(C2CN(C)C(=O)CC2)=O)CCN(C(=O)CCC2CCCO2)CC12CCC2 66739,C1(NC(c2ccnc(Cl)c2)=O)CN(Cc2cccnc2O)CC1(F)F 66740,c1(OC)ccc(CN)cc1-c1ccc(CNC(C2(CC#N)CC2)=O)o1 66741,CCCCC(CNC(c1ccccc1)=O)NC(C1CC(=O)N(C(CC)CC)C1)=O 66742,c1(C(=O)NC2CCN(Cc3cncc(Cl)c3)CC2F)ccc2ncsc2c1 66743,N1(C(C=C(C=CC)CC)=O)CCC(F)(CNC(=O)C(C)Sc2ccc(F)cc2)C1 66744,Cc1cc(Cl)ccc1-n1cc(CC2COCCN2C(c2sc(Cl)cc2Cl)=O)nn1 66745,C1(NC(CN(C(=O)Cn2c(O)nnc2O)CCOC)=O)CN(C)NC1=O 66746,Cc1c(C(=O)NC2CCC(c3cn(CC(=O)O)nn3)CC2)cccc1C1CC1 66747,Cn1cc(C(N2CCC(C)(CNC(c3nsnc3O)=O)C2)=O)ncc1=O 66748,N1(C(CN2CCC(C)(C)C2)=O)CC2(NC(=O)COC3(C)CCCC3)CCC1CC2 66749,C(=O)(C(=O)N=S(C)(C)=O)NCC1CCC(NC(C(C)Cc2ccccc2)=O)C1 66750,CC1(C)CCCCC(NCc2cnoc2-c2ccc(Cl)s2)C1 66751,C1(CC(N2CCCC2c2cc(C3CC3)on2)=O)CCCC2CC12 66752,Cc1cc(C(N2CCOC(CNC(C3CCN(C)C3C)=O)C2)=O)c(C)n1C(C)C 66753,c1(NC(C)=O)cccc(CC(=O)NCC(C2CC2)N(C(=O)C(C)N2CCC2)C)c1 66754,N1(C(C2(F)CCC(C)CC2)=O)CC(C(=O)NCC(C)(C)CO)C2(CCC2)C1 66755,C1(S(C)(=O)=O)(C(=O)NC(C2CCN(C(C=CCC)=O)C2)C)CCOCC1 66756,Cc1cnc(O)c(CNC(C2COCCN(C(C3(C#N)CC(F)(F)C3)=O)C2)=O)c1 66757,c1(NC2CCCN(C(C3CC4(C3)CC4(F)F)=O)C2)ncc([N+](=O)[O-])cc1Br 66758,C1(C(=O)NCC2(CC)CC2)C=CCN(C(c2cccc(O)n2)=O)C1 66759,N1(CCC)CC(C(=O)N(CCCCNC(c2ccc(C(=O)OC)[nH]2)=O)C)CC1=O 66760,c1(OC)ccc(C(=O)NC(c2ccc(F)cc2)c2ccsc2)cc1 66761,N1(C(C(CC)OCC)=O)CC2CCC1C(CNC(c1cc(C3CC3)[nH]n1)=O)C2 66762,CCC(CC)CC(=O)N1CCN(C(c2csc(-c3ccccc3)n2)=O)C2CC12 66763,c1(C(N2CCN(C)C(CNC(=O)COCC3CCC3)C2)=O)cc2ccncc2s1 66764,N1(C(c2ccc(CC)o2)=O)CC(OC)C(NC(=O)C(C)NC(=O)CC(C)(C)C)C1 66765,C1(S(N)(=O)=O)(C(=O)NCC(CNC(CC(C)c2ccncc2)=O)O)CC1 66766,N1(c2cc(N(C)CCN3CCCCC3)nc(C)n2)CCCc2sccc2C1 66767,C1(NC(CN2C(C)CC2)=O)CCC(NC(c2ccnc(OC(F)F)c2)=O)CC1 66768,c1(N2CC3CN(CC)CC3C2)nc2c(c(=NC3C=C(C)CCC3)[nH]1)COC2 66769,c1(OC)ccc(Cl)c(CN2CCN(C(C3CCC(=O)NC3)=O)C3CC23)c1F 66770,n1(CC(=O)NCC(CCNC(C2(CC)CC(C)(C)C2)=O)O)nnc2c1CCCC2 66771,N1(C(c2c(C)ccc(C(C)C)c2)C(=O)NCCC#N)CCCNC(=O)C(F)(F)C1 66772,c1(C(=O)NCC(CNC(C(CC(CC)C)C)=O)(C)C)cnc2ncnc(O)c2c1 66773,c1(C(N2CCC(CNC(c3nn(C)c(Cl)c3)=O)C2(C)C)=O)ccc2ncsc2c1 66774,Cc1cc(N)cnc1C(=O)NCCNC(=O)CCC1CC(C)(C)CO1 66775,CC1SCCCC1C(=O)NCCC1(NC(c2cnc(C(C)(C)C)[nH]2)=O)CCC1 66776,C=CCC(C)(C)C(=O)NC1CCC1c1cn(CCNCC2CCC3CC3C2)nn1 66777,c1(CC)c[nH]cc1C(N1CCC(Cc2cn(C3CCC3O)nn2)C1)=O 66778,C1(C(N2CC(N(CCC)CC)C2)=O)CN(C(=O)C(CC)OCC)CC(C)(C)C1 66779,c1(OCC)cc(-c2cccc(NC(c3cnn(C(C)(C)C)c3)=O)n2)ccn1 66780,CCCC(C(=O)OC)C(=O)NC(C)CN(C)C(c1sc(C)c(C)c1C)=O 66781,N1(C(C(CNC(C(COC)OC)=O)C(C)C)=O)CCC(N(C)OC)CC1 66782,N1(C(C(COCC)(C)C)=O)CC(CNC(C23CC(C)(CO2)C3)=O)CC(C)(C)C1 66783,C1(O)(C(C)C)CCCN(C(C2CCCCN2C(C2(F)CCCCC2)=O)=O)C1 66784,CC1(C)C(NC(=O)Cn2cnnc2)CC1C(=O)NCC(Cl)C(C)(F)F 66785,Cc1cc(C(=O)NC(C)CCCNC(=O)CC2CC3CC3C2)c(C)s1 66786,C(C(C)C)(C(O)C(=O)NC1CCCC(C(N2CCC(O)C2(C)C)=O)C1)OC 66787,c1(OCC)ccc(Cl)nc1C(=O)NCCC(C)NC(=O)C1=NOC(C(C)(C)C)C1 66788,C1(NC(C(C)NC(=O)NC)=O)CN(C(=O)C(F)OC(F)(F)F)CC2(CCC2)C1 66789,N1(CC(=O)NC(C=CC(=O)NC(c2ccnc(O)c2)C)(C)C)C(=O)CNC1=O 66790,C1(NC(CCCc2n(C)cnn2)=O)CCN(C(C2CC3(CCC3)C2)=O)CC1F 66791,c1(C(N2CC(CNC(CCCCCOC)=O)C(F)(F)C2)=O)c[nH]c2ccncc12 66792,C1(NC(c2ccc(C=C)cc2)=O)CCN(c2ncc(C(F)(F)F)cc2Cl)C12CCC2 66793,N1(C(c2n(C)c(C#N)cc2)=O)CCC2(CC(NC(=O)C(C)(C)c3cnsc3)C2)C1 66794,N1(C(C(C)(C)C2CCCN2C(=O)C(Cl)Cl)=O)CCCC(CCO)CC1 66795,c1(C(N2CC(CCNC(CC3(OCC)CCC3)=O)(OC)C2)=O)ccc(C)cc1 66796,c1(-n2cc(C(C)(C)NC(C3CCCC3O)=O)nn2)ccc(I)c(Cl)c1 66797,C(C(C)(C)C(=O)NCC1CN(C(C2CCC(C)CC2)C)CCO1)OC(C)C 66798,N1(C(C(C=CC)O)=O)CCN(C(C2(CC(C)=O)CCCC2)=O)CC1CCOC 66799,c1(N2C(CCNC(=O)CC34CNC(=O)C(C3)C4)CCCC2)nc2ccccc2o1 66800,CCC(CC(=O)NC(c1ccc(CNC(C2CSCCS2)=O)cc1)C)C(C)(C)C 66801,c1(C(=O)NC2(CC)CN(C(c3ncn(CC)c3)=O)C2)ccc2cccnc2n1 66802,c1(CCC(c2n(C(CC)C)nnn2)NC23CC(F)(C2)C3)ccc(OC)c(C)c1 66803,CON=Cc1ccc(C(N2CCC3CN(C(c4cc[nH]c4)=O)C3C2)=O)cc1 66804,C(=O)(N=c1[nH]c(Cl)ncc1O)c1c(CNc2c(C)cc(F)c(C#N)c2)cccc1 66805,N#Cc1ccc(CCC(=O)NC2(C(F)(F)F)CCCNC2)cc1 66806,c1(CC(=O)N(C(=O)C(C)(C)CF)C)ccccc1CNC(=O)C(C1CC1)C1CC1 66807,Cc1cc(C)c(C(N2CC(C(C)NC(=O)C(C)S(C)(=O)=O)C2)=O)c(=O)o1 66808,c1(C(=O)NCC(CO)NC(c2[nH]cc(OC)c(=O)c2)=O)ccc(C)c(Cl)c1F 66809,c1(CC(=O)NC(C)CCNC(C23CCC(F)(CC2)C3)=O)cnc2ccccc2c1 66810,CC(C)CC(C(=O)N(C)C)N(CC(F)(F)F)C.C1(=O)C(C)NC(=O)N1 66811,N1(C(C(C)Cn2cccn2)=O)CCCOC(CNC(c2cnn[nH]2)=O)C1 66812,N1(C(c2cc(OC)cc(C)n2)=O)CCC(C)N(C(=O)CC2CCCCN2C)CC1 66813,C12(CNC(C3C(=C)C3)=O)CCC(C1)N(C(=O)CCC(=O)c1ccccc1)C2 66814,C(C(C(=O)N(CCC(N1CC=C(C)C1)=O)C1CC1)OC)OC 66815,C(=O)(C1=CCCN(C(c2ccc(F)c(F)c2F)=O)C1)Nc1c(OC)cc(F)cn1 66816,c1(NCCNC(c2ccsc2CO)=O)nccc(SNCn2cc(Cl)cn2)n1 66817,Cc1nc(C2CCC2)oc1C(=O)NC(C)(C)CNC(C1(C#N)CC1C)=O 66818,CC1(C)C(NC(=O)C(C)(C2CCC2)NC(=O)COC2CCCOC2)C1(C)C 66819,N1(C(C2=NOC(CNC(Cc3ccn(C)n3)=O)C2)=O)CCCC(C2(C)CC2)C1 66820,C1(O)(C(N2CCCC(CNC(=O)CCc3ccsc3)C2)=O)CN2CCC1CC2 66821,CCC(C)CC(=O)C(=O)N(CC(C)NC(=O)Cc1cccnc1O)C 66822,Cc1nnc(=NCC2CC(C)N(C(=O)C(C)CS(C)(=O)=O)C2)[nH]c1C 66823,c1(COC)cc(CSc2ccccc2OCC2CCOC2)ccc1F 66824,N1(C(C(C)=C(C)C)=O)CCC(F)(F)C(CNC(c2cnoc2-c2ccco2)=O)C1 66825,CCC(CS(=O)(=O)c1ccccc1)OC(c1ccc(C2CCOC2)cc1)=O 66826,C1(C(N2CC(F)(CC)C2)=O)CN(C(=O)CN(C2CCC2)C)CC1C1CC1 66827,n1(CC)nc(C(=O)NCc2nc(C(N3CCN(C(C)CO)CC3)=O)co2)cc1C 66828,N1(C(c2c(C)ncnc2C)=O)CC2(CC(NC(=O)CC3CC3)c3nccn32)C1 66829,N(C(=NCCF)N1CCC2(O)CCOCC2C1)CC1(C)CCCCC1 66830,CC1CCCCN1C(=O)C(c1cn(C)nn1)NC(C1CN(C(N)=O)C1)=O 66831,c1(N(CCC)C)ccc(C(=O)NCC2CC2CNC(c2cnn(C)n2)=O)cc1 66832,c1(C(=O)NC2CCCN(C(C(=C(C)C3CC3)F)=O)C2C)c(Cl)cccc1[N+](=O)[O-] 66833,C1(NC(c2nc(CC)oc2)=O)CCC2CCN(C(c3cnoc3C(C)C)=O)C1C2 66834,CC1CCC(NC(c2cnn(C)c2)=O)CN1C(=O)C=Cc1ccc(C(N)=O)cc1 66835,c1(C(N2C(C)CC(NC(c3cnc(O)o3)=O)C2)=O)cc(Br)c(C#N)s1 66836,C1(CNC(c2cc(C(F)(F)F)no2)=O)CC2C(O)CC2O1 66837,CC12CCCC1N(C(=O)CCc1cncs1)CCN(C(c1cnc[nH]c1=N)=O)C2 66838,Cc1cc(C(=O)NC2CCN(C(C3CS(=O)(=O)C3)=O)CC2C)nc2[nH]nc(O)c12 66839,C1(C)(C(=O)NCC2C(C(=O)NCC(C3CCCCC3)C)CC2)CC(F)C1 66840,C#Cc1cccc(C(=O)NC2(C(=O)OC)CC(c3cn(CC(=O)OC)nn3)C2)c1 66841,C1(NC(C2C(C(C)=O)C2(C)C)=O)COC2(CCN(C(C3(C)COCCO3)=O)C2)C1 66842,c1(C(=O)NCCCNC(C(C)CN(C)C)=O)ccc(C2CCC2)cc1 66843,Cc1c(CSc2cn(C3CN(C(=O)OC(C)(C)C)C3)nn2)oc2ccc(Br)cc12 66844,N1(C(c2c(C)[nH]cc2-c2ccccc2)=O)CCCC(NC(c2csnn2)=O)C1C 66845,c1(C(N2CC(CNC(C(CCC)=CCC)=O)C3(C2)CC3)=O)cc2cccn2cn1 66846,N1(Cc2nc(-c3ccc(OC)cc3)on2)CC(CO)OC2(CCC2)C1 66847,c1(C(=O)NCC2C(C)CN(C(C3CCOC3)=O)C2)nc2ccccc2cc1Cl 66848,C1(C(CN(C(CCC)=O)CC)F)CCN(C(=O)C#CC2CC2)CC1 66849,c1(-n2cc(C3(O)CN(C(C4(C)CC(C(F)(F)F)C4)=O)C3)nn2)cccc(F)c1Br 66850,c1(CC(C(=O)NCC(CO)NC(C2(C)CC=CCC2)=O)N(C)C)ccccc1F 66851,c1(CC)nc(=N)[nH]cc1C(=O)NC1CCN(C(=O)C(F)C(C)(F)F)C1 66852,CC(CC(F)F)C(=O)NC1CC2C1CCN2C(c1ncccc1Br)=O 66853,Cc1cc(C(N2Cc3ccccc3C2)=O)c2c(c1)CCCN2 66854,C1(NC(C2C(C)(CC)C2)=O)(COC)CCN(C(=O)C=Cc2ccc(C)nc2)CC1 66855,C(=O)(CCCC(C)NC(=O)CC1CCC(=O)C1)Nc1cc(C)sc1C 66856,C1(C(=O)NCCCCNC(C2SCCS2)=O)C2(CCC2)C12CCC2 66857,N1(C(CCC(C)SC)=O)CC2(C(=O)Nc3ccc4c(c3)OCC4)CCC1CC2 66858,c1(C(=O)NCC2CC(OC)CN2C(C2CC(SC)C2)=O)ccc2nc(C)nn2c1 66859,CC(O)CCCCCC(=O)NCC1(O)CN(C(=O)C=CC2CCCO2)C1 66860,c1(C(N2CC(N(C(Cc3cnc(C)o3)=O)C)C2)=O)cc2nn[nH]c2cc1F 66861,N1(C(C=CC)=O)CCC(CN2CCN(C(c3ccc(OC)nn3)=O)CC2)CC1 66862,C1(NC(c2cc(C(F)(F)F)on2)=O)CC2CCC(C1)N2C(c1cccc[n+]1[O-])=O 66863,Cc1cc(C(N2CCC2C(=O)NCc2cc(Cl)ccc2O)=O)cc(O)n1 66864,C1(OC)CC(C(N2CCC(NC(c3c(C4CC4)cnn3C)=O)CC2)=O)C12CCC2 66865,C1(NC(C=Cc2n(CC)ncc2)=O)C(C)CCN(C(c2n[nH]c(=N)[nH]2)=O)C1C 66866,C1(OC)(CNC(c2cc(C(C)(F)F)ccn2)=O)CCN(C(C2(C)C=CCC2)=O)C1 66867,N1(C(c2c(-n3cc(CC(=O)O)nn3)cccc2)=O)CC2CC3CCCN3C2C1 66868,C(=O)(C1=CN=C2N=CNN2C1)NC1CCCN(C(CSC(C)C)=O)C1C 66869,N1(C(CCCC(C)NC(C2N(CC)CCCC2)=O)=O)CCC2CN(C)CC2C1 66870,c1(OC)cccc(C)c1C(=O)NCC1CN(C(=O)C(O)C(C)(C)C)CCS1 66871,Cc1ncc(C=CC(N2CC=CC2CNC(c2c(C)ccnc2O)=O)=O)c(O)n1 66872,CC1(C)C(C(N2CCC(OC3CC3)CC2)=O)CC1COc1nc[nH]n1.C1(=O)CN1 66873,n1(CC(C)C)cnc(S(=O)(=O)NC2CCCCCC2)c1 66874,N1(C(=O)NCC(CCSC)OC)CCCCC(OC(C)C)C1 66875,c1(C(=O)NC2C(F)CCN(C(C3C(=C)CC3)=O)C2)ccc2c(c1)N(C)C(=O)CC2 66876,C(=O)(CC(C(F)(F)F)OC)NC(CCNC(C1CN(CC)C(=O)CC1)=O)(C)C 66877,Cc1cc(NC2CC(NC(c3ccc(O)nc3)=O)C23CCC3)c([N+](=O)[O-])c(C)n1 66878,C(=O)(CC(O)CC1CC1)NC(CNC(C=CCC)=O)(C)Cn1cccn1 66879,C12(C(N3CCCC(CNC(Cc4ccc(CC)cc4)=O)C3)=O)CCCC1CCC2 66880,Cc1noc(C)c1CC(N1CSCC1C(=O)NC1CC(C(C)(C)O)C1)=O 66881,CC1(C)CCC(C(=O)NCC2(O)CCN(C(c3cccc(F)c3)=O)C2)CO1 66882,c1(CNC(CC(C)C)c2cccs2)cc([N+](=O)[O-])ccc1Br 66883,CC(C)(C)C(=O)C(=O)N1CCC(C)(NC(=O)C(CCc2ccccc2)C2CC2)C1 66884,C1(NC(C(C)(C)C)=O)CN(N2CCC(ON3CCCCC3)C2)C1 66885,c1(C(=O)NC2CC(CNC(c3cc(C)c(N)cc3)=O)C2)ccc2cccnc2n1 66886,Cc1nc2cccc(C(N3C(CNC(C4(O)COC4)=O)CC4COCC34)=O)c2[nH]1 66887,C1(C(=O)NC(CC2CC2)C(=O)NC2C3COCC23)CC2(CCC2)CO1 66888,N1(C(C(C=C)(C)O)=O)CC2(C1)OC1(C)CC2(NC(C2CCN3CCCC3C2)=O)C1 66889,N1(C(c2cnc(C)s2)=O)CC2CC(NC(C3CCCC(F)C3)=O)CC1C2 66890,CC1(C)CC(C(=O)NC2(CNC(C34CCCC3C4)=O)CCCCCC2)=NO1 66891,N1(C(=O)NCc2nn(C)c(=O)o2)CCCC(C)(C(=O)NC2(CO)CCCCC2)C1 66892,C(=O)(CC(C(C)(C)C)NC(c1cnnn1C)=O)NC(c1ccco1)C 66893,C1(C(=O)NC(C)C(C)NC(=O)C=C(C)CN2CCOCC2)(OCC)CCCC1 66894,C1(C(=O)NC(C)CCNC(=O)C(O)C2CCC2)C(c2ccncc2)C1(C)C 66895,c1(NC(C2CCN2C(=O)C2=CS(=O)CCC2)=O)ccc2scnc2c1 66896,c1(NC(C2CCN2C(c2cc(Cl)cc(Cl)c2)=O)=O)ncc(F)cc1Br 66897,C12(C(=O)NC3CN(C(COc4ccn(C)n4)=O)CC3O)CCCCN1CCC2 66898,C1(NC(c2c(CC)scc2)=O)CCN(C(c2ccccn2)=O)C(C)C1 66899,c1(C(NNC(NN(C(C)(CC(=O)O)C(C)C)CC)=S)=O)cc(Cl)c(Br)cc1F 66900,c1(C(=O)NC2CCN(C(C3=NNC(=O)C3)=O)CC2F)ccc(F)c2ccsc12 66901,S(=O)(=O)(c1ccc(C2OCCO2)cc1)NCC1(NC(=O)OC(C)(C)C)CC1 66902,C12(C(N3CCN(C(COC(CC)(C)C)=O)C(CF)C3)=O)CCCC(=O)N1CCC2 66903,C(=O)(C(C(C)Cc1ccc(CC#N)cc1)N1CCCC(C(F)F)C1)NCCOC 66904,CCCCC(CNC(=O)C(C(C)C)NS(C)(=O)=O)NC(=O)Cc1ccc(O)nc1 66905,c1(C(N(CCOC)CCNC(=O)CC2COCC2O)=O)cc(F)ccc1C(F)F 66906,N1(C(C2CC(OC)(OC)C2)=O)CC2CC(NC(c3cncc(C4CC4)c3)=O)C1C2 66907,C(=O)(CC(F)(F)C(F)F)NCC1C(NC(C(c2cccc(C#N)c2)C)=O)CC1 66908,C=C(C)C(C)(C)C(=O)N1CCN(C(c2c[nH]cc(Br)c2=O)=O)CC1 66909,CC1(C(N2CCC(COC)(CNc3ccccc3)C2)=O)CC2CCC(C1)S2(=O)=O 66910,c1(NC(c2noc(C)n2)CC)ccnc2c(Cl)cnn12 66911,CC(C)(CNC(c1cc([N+](=O)[O-])c[nH]1)=O)CC(=O)NCCCOCC1CCC1 66912,C1(CC(=O)NCC(C)N(C(C)=O)C)CC2(CCC2)CN1C(=O)C=Cc1cocn1 66913,c1(OC(=O)Nc2ccc(NCc3c(C)cccc3)cn2)cc(F)cc(C)c1O 66914,C12(NC(C(C)OCC#C)=O)CCC(C1)N(C(=O)CCCC(=O)NC)C2 66915,Cc1ccc2c(C(=O)NCC3CCN(C(=O)C#CC4(C)COC4)C3)cnn2c1C 66916,C1(OC)CCC(C(=O)NCC(=O)NC2(C(C3CC3C)NC3CC3)CC2)CC1 66917,CC1CC(C(=O)N2CCC(CNC(c3ccn(C)c3)=O)C2)c2ccccc2N1 66918,c1(CCC(=O)NCCC2CCCN(C(C(CC)F)=O)C2)nc2cnccc2[nH]1 66919,c1(OC)ccc(CN2CCOC(CC(=O)Nc3nccnc3Br)C2)cc1[N+](=O)[O-] 66920,C1(NC(C2(C(=O)OCC)CC2)=O)CCN(C(c2ccc(N(C)C)nc2)=O)C1C 66921,N1(C(c2ccc(CCC)cc2)=O)CC(NC(c2nc(C)no2)=O)C(C)(C)C1 66922,c1(CC(=O)NC(C)CNC(=O)CC2CCS(=O)(=O)C2)cc2ccccc2c(O)n1 66923,c1(OC)cc(NC(=O)C(=O)NC2C(C)CCCC2C)ccc1Cl 66924,c1(C(=O)NC2C(CC)N(C(c3ccc(C4CC4)s3)=O)CC2)ccc(N=[N+]=[N-])cc1 66925,c1(C(=O)NCC2CC(NC(CCN)=O)C2)ccc(Br)c(F)c1.O=CC1CC1 66926,Cn1ncc(Cl)c1CC(=O)NC12CC1CN(C(C1CC1CF)=O)C2 66927,C(C)(CC(C)(C)O)NC(C(C)N(C(=O)C(c1ccnn1C)C)CCC)=O 66928,N1(C(CSCCC)=O)CCCC(CCC(=O)N)C1.N1(CCO)CCC(C)CC1 66929,N1(C(CNC(C(CC)CC)=O)=O)CC2CCCCN2CC1CNC(=O)C=CCO 66930,C(C(O)CC(=O)N(C1CC1C)C)NC(c1c(C)ocn1)=O 66931,c1(C(N2CCC(OCCNC(C(C)SC)=O)C2)=O)ccc(-c2ccco2)nc1C 66932,CC(C)C(C(=O)N(CCCCNC(=O)CC1(C(F)F)CC1)C)N(C)C 66933,C(CC(C)C(=O)NCCCC1CCCN1C(=O)C(=O)NCC(F)F)=CC 66934,N1(C(C2C=CCS2)=O)CCC2CN(C(=O)CSC3CC3)C2C1 66935,C1(CNC(Cc2nnc(C)o2)=O)CCCC2CN(C(=O)CN(C)C(C)C)CC12 66936,Cn1cc(C2CC2NC(c2c[nH]nc2CNC(c2cnn[nH]2)=O)=O)cn1 66937,c1(OC(F)F)ccccc1-c1noc(CSC2CCCC(c3ccc(Cl)cc3)C2)n1 66938,C1(C)(C(N2CC3C(CNC(c4c(OC)noc4C)=O)C3C2)=O)CCC(C)CC1 66939,c1(OC)cc(C(N2CCC(NC(c3ccc(N)cc3Cl)=O)C2)=O)cc([N+](=O)[O-])c1 66940,Cc1cccc(O)c1C(N1CCCC(CN(S(=O)(=O)CCCl)C)C1)=O 66941,CC1CN(C(C2(c3ccno3)CC2)=O)CC(C)N(C(c2cc(O)nc(O)n2)=O)C1 66942,C1(C(=O)NCC2(CCOC)CC2)CCOCC1NC(=O)C=C=C(C)C 66943,c1(C(N2C(C(=O)NCCCOC)C3C(C2)C3(C)C)=O)cccc([N+](=O)[O-])c1C 66944,CC1CN(C(C2CC=CCC2NC(C23CCCN2CCC3)=O)=O)CCCO1 66945,N1(C(CCSC)C(=O)NCC2CCOC2)CCCC(F)(CO)C1 66946,C(=O)(C1=CCCCC1C)N1CC2C(NC(c3c(C)nc(C4CCC4)o3)=O)C2C1 66947,c1(CNS(C)(=O)=O)ccccc1NC(=O)C(=O)NCCC1CCOC1 66948,N1(C(c2c(C)nc(COC)s2)=O)CC2(CCCC2NC(C2CCCN2C=O)=O)C1 66949,Cc1cc(C(=O)NC23CCC2CN(C(c2c(C(C)C)cnn2C)=O)C3)cc(F)c1 66950,C(=O)(CC(C(C)C)NC(=O)Cn1c(C)ccc1C)NC(C(=O)OCC)C1CC1 66951,C1(CNC(=O)Cc2csnn2)CC2CCC1N(C(c1csc(CO)n1)=O)C2 66952,Cc1nc(C(=O)NCC2CC(CNC(c3c(C)cnn3C)=O)CO2)n(C)n1 66953,CCCC(CC(C)C)C(=O)NC(COC(C)C)C(N1CC(CO)C1(C)C)=O 66954,Cc1cc(=NCCC2CCCOC2C(C)C)[nH]c(=NCCCCCF)[nH]1 66955,c1(C(C(=O)NC)N(CC(F)F)CC2CCCO2)ncc(OC)cn1.C(C(C)C)S 66956,CC(C)CC(O)CC(=O)NC1(Cc2ncc(F)cn2)CC1 66957,C12(OC)CCC1CN(C(C1CCN(C(=O)CCCC3CCC3)C1(C)C)=O)C2 66958,Cc1c(C(N2CCSCC2CCNC(C2CN(C)C2)=O)=O)sc2nccn12 66959,N1(C(CC2N(C(CCC(C)OC)=O)CCC2)=O)CCc2nc(C)[nH]c2C1 66960,c1(C(N(C2CCN(C(c3cnco3)=O)C2)CC#C)=O)nocc1C 66961,c1(C(=O)NCC2C3N(C(C=CCOC)=O)C(CC3)C2)cc(Br)cc(C)c1F 66962,O=C(CCCCCO)NC1CC(F)CN(C(c2ccc(OC(F)(F)F)nc2)=O)C1 66963,N1(C(CCCC#C)=O)CCC(C2CCCN(C(=O)CCC(=O)C(C)(C)C)C2)CC1 66964,N1(C(CC2CCC(=O)NC2)=O)CCN(C(c2cccc(Cl)c2F)=O)CC(CO)C1 66965,Cc1cccn(CC(=O)NCC2C=CCN2C(c2cc[n+]([O-])cc2)=O)c1=O 66966,CN=c1ccc(C(N2CC(O)CC2CC(=O)NCC(=O)N2CCCO2)=O)c[nH]1 66967,O=C(CS(=O)(=O)C12CC(C1)C2)NCCCNC(c1sccc1-n1cnnn1)=O 66968,c1(NC(C2CC23CCN(Cc2c(F)ccc(Cl)c2Cl)C3)=O)nccc2[nH]ccc12 66969,CCCCCC(O)C(=O)NC(C1(O)CN(C(C2CN(C(C)=O)CCO2)=O)C1)C 66970,c1(CC)ccc(C(=O)NCC2CC(CCNC(=O)C(CC)SC)C2)cc1Cl 66971,C1(C(=O)NCC(CN(C(CC(C)NC(N)=O)=O)C)O)CCC(=O)N1C 66972,C1(C(CO)NC(C(C)CF)=O)CCN(C(C2(F)CC2(Cl)Cl)=O)CC1 66973,S(=O)(=O)(c1cccnc1)N1CC(C(=O)NCCOCCN2CCOCC2)C(O)CC1 66974,N1(C(c2scnc2C)C(=O)NCCCCCC)CCC2(O)CCOCC2C1 66975,c1(NCC2(CCCC)CCC2)cc(NCC2(CC3CCC3)CC2)ncn1 66976,CC(CCBr)(c1nnnn1CC1CCCO1)Sc1nnc(CN2CCCCC2)s1 66977,c1(NC(C2OCCN(C(C(C)(C)C)=O)C2)=O)ccc2c(c1)OCC2 66978,N1(C(CCCCOCC)=O)C2CCC1CN(C(c1cc(C)n(C(F)F)n1)=O)CC2 66979,N1(C(c2ccc(SC)s2)=O)CC2CCN(C(=O)C(c3cccc(F)c3)O)CC2C1 66980,N1(C(CCc2nnc(C)o2)=O)CCc2cc(Br)c(Cl)cc2C1 66981,C1(CNC(c2nncc(OC)c2)=O)CC2(CO1)CN(C(=O)CCc1cnco1)C2 66982,N1(C(CSCCC(C)C)=O)CCCN(C(c2cnc(Cl)c(N)c2)=O)C(C)C1 66983,Cc1nc(C=CC(=O)NC2COCCN(C(C3SC4C=CC3CC4)=O)C2)[nH]c1C 66984,CN1CCCCC1CC(N1CCC1(C)CC(=O)NC1(CN(C)C)CCC1)=O 66985,c1(OCC)ccc(C(=O)NC(C2(CNC(c3cc(C#N)c[nH]3)=O)CC2)C)cc1 66986,C1(CNC(CC(=O)NCC#C)=O)CCCCN(c2nnc(C(=O)OC)s2)C1 66987,C1(C(=O)NC(CNC(C2(NC(N)=O)CC2)=O)C2CCC2)CC12CCOCC2 66988,C(=O)(C1CCc2c[nH]nc21)NCC(CO)NC(c1ccn(CCF)n1)=O 66989,c1(C(C)=O)ccc(CC(=O)NCC2CC2NC(=O)C(n2cnc(C#N)n2)C)cc1 66990,C1(NC(C2C(OC)CCCC2)=O)CCC2(CC1)CN(C(=O)CS(=O)(=O)C1CC1)C2 66991,Cc1cc2occ(C(=O)OCc3nonc3C)c2cc1C 66992,Cc1cc(C(=O)OC2CN(C(c3nnc(C)n3C)=O)C2)c(Cl)cc1N 66993,n1(CCCC)cc(C(N2CCC(CNC(C3CC(n4cnnc4)C3)=O)C2)=O)nn1 66994,N1(C(c2c(C(C)C)occ2)=O)CCC(C)(C(=O)NCCC(N)=O)C1 66995,C(=O)(N=c1cc(-c2ccc(F)cc2)[nH][nH]1)NC(c1cccc(Cl)c1F)C 66996,c1(COC(C2CS(=O)(=O)CC(=O)N2)=O)ccc2ncccc2n1 66997,C(CC(=O)NCCCC(C)(F)F)(C(F)F)NC(CC(C)c1ccco1)=O 66998,C1(C)(C(N(CC(C)CNC(c2ccncc2C2CC2)=O)C)=O)CCCCC1(F)F 66999,C1(C(N(C)Cc2cc(C)no2)=O)CCCN(C(c2nc(C)oc2C)=O)C1 67000,Cc1nccc(C(=O)NCCC2CC(F)(F)CN2C(=O)CC2CCOC2)c1C 67001,C(CC(=O)NC1(C)CC(NC(C2(O)CC2(C)C)=O)C1)(C(N)=O)NC(C)=O 67002,CC(CC(F)F)C(=O)N(CC(O)CNC(c1ccnc(CO)c1)=O)C 67003,N1(C(c2c(C)noc2-c2ccccc2)=O)CCC2CC(C)CCC12 67004,N1(CC(=O)NCC2(O)CN(C(C3CCC(=O)O3)=O)C2)CCCCCC1 67005,N1(C(CC(C)SC)=O)CCC2(CC1)CC(NC(c1sc(F)cc1Cl)=O)CO2 67006,C1(O)(C(C)NC(C(N2C(=O)CCC2=O)C)=O)CCN(C(=O)C2=CCC2)C1 67007,CC1CCN(C(c2conc2C(C)(C)C)=O)CCN1C(=O)CCc1ccccc1 67008,n1(CC)ncc(C(=O)NC(C)(C)C(=O)NC2CCCC2CF)c1C 67009,N1(C(c2c(CC)cc(N)cc2)=O)CC(NC(c2coc(Br)n2)=O)CC2(CCC2)C1 67010,n1(CC)nnnc1C(c1cccnn1)NC1(NC2CC(c3ccccc3)C2)CC1 67011,CC(C)C(O)CNC(=O)C(C)(C)NC(=O)CCc1ncnn1C 67012,C1(C(=O)NC(CN(C)C)CCO)(CC)CCCN1C(C1CC(N=[N+]=[N-])C1)=O 67013,Cc1cnc2c(C(=O)NCC(CO)NC(=O)C(c3ccc(C)o3)C)c(C)nn2c1 67014,N1(C(c2cnc(OC)nc2C)=O)CCCC12CCN(C(=O)C(C)CF)C2 67015,c1(C(N2CC(C#C)C2)=O)cncc(CNC(=O)COCc2nc[nH]n2)c1 67016,c1(N2C(C(=O)NCc3c(OCC)cccc3)C(O)CC2)ncnc2c1CCC2 67017,C1(N(C(CCC)=O)C)CCCN(C(c2cnn(CCCOC)c2)=O)CC1 67018,CC(CC(F)F)C(=O)N1CC(N(C)C(C2CC2c2ccc(F)c(F)c2)=O)C1 67019,c1(C(=O)NCCNC(c2c(C)cccc2Br)=O)ccc2nc(N(C)C)[nH]c2c1 67020,c1(OCC)c(F)cc(C(N2CCC(CN3CCN(C)CC3)C2)=O)cc1F 67021,CCCCCCOCC(=O)NCC1(NC(c2ccc[nH]2)=O)CCC1 67022,CN1CC2CC2(NC(=O)C(=O)NCCOC2CCCCC2)S1(=O)=O 67023,N1(C(c2cc(C(N)=O)[nH]c2)=O)CCC2(CC1)CN(c1ccc(C#N)nc1)CCO2 67024,c1(NC(C2C(C(=O)OC)C2)=O)ccc(C(=O)Nc2cc(Cl)ncc2F)cc1C 67025,Cc1ccc(CN2CC(F)CC2C(=O)Nc2ccnc(-c3cccs3)c2)cc1 67026,Cc1cnc(NCC2CC3C=CC2O3)c(S(=O)(=O)NC(c2ccco2)CO)c1 67027,C1(C)(CC(=O)NCC(=CC(=O)NC2(CCOC)CC2)C)CCOC1 67028,n1(CC)ccc(C(=O)NCC2(NC(=O)C=CC(=O)NC3CC3)CCOC2)c1C 67029,C1(NC(C(CC2CCC2)NC(C(C)SCCCC)=O)=O)CCOCC1F 67030,c1(CC(=O)NC2CC2)ccc(OCCNC(C(COC(C)(C)C)N(C)C)=O)c(Cl)c1 67031,C1(NC(C(C)Cc2ccco2)=O)CC(NC(=O)Cc2cnoc2)CC1O 67032,N1(C(C2CCCN(C)C2)=O)CCC2(CC(NC(C3(C)CS(=O)(=O)C3)=O)C2)C1 67033,C1(NC(c2cc(OC)ncn2)=O)CCCN(C(C2CCSC2)=O)C1C 67034,c1(C(=O)NCCCCNC(Cc2c(C)cco2)=O)sc(N2CCCC2)nc1Cl 67035,CCCCCCC(C)CC(=O)NC1CCN(C(c2cnc3n2CCC3)=O)C12CC2 67036,N1(C(c2c(CC)nccn2)=O)CCCC2(CCN(C(=O)C(C)NC(C)=O)CC2)C1 67037,C1(C(N2CC(C(C)C)N(C(=O)Cc3cncs3)CC2)=O)CC12CCC1(CC1)CC2 67038,c1(OC)c(CNCC2CCCN2C(=O)CCC(N)=O)cc(F)cc1F 67039,CC1CC=C(C(=O)N2CCN(C3CN(C(C4C(C5CC5)C4(F)F)=O)C3)CC2)CC1 67040,C(=O)(C(C(C)(C)C)OC(C)(C)C)N(CC(C)NC(C12CC(C(C)(C)C)(C1)C2)=O)C 67041,N1(C(CN2CC(=O)NCC2)=O)CC2CC(F)(F)CC2C1 67042,C#Cc1cccc(C(=O)NCC2(F)CCN(C(=O)C(C)(C)CCOC)CC2)c1 67043,c1(C(=O)NCCCN(C)C(c2ccc([N+](=O)[O-])o2)=O)cnc(N)c(N)c1 67044,C1(c2nc(-c3ccc(OCC)cc3)nn2CC2CCOC2)CC2C(C1)C2(F)F 67045,Cc1cc(C)n(CC(c2nc(C3CC34CC4)nn2-c2ccc(Cl)cc2)=O)c(=O)n1 67046,Cc1nc(C#N)ccc1C(=O)N(CC(C)NC(c1ccnn1CC(C)C)=O)C 67047,c1(C(=O)NCC(COC)NC(=O)C(C)n2cccn2)conc1C1CCCC1 67048,N1(C(C2CCCS2(=O)=O)=O)CCC2C(C1)CN2C(=O)Cc1cccc(Cl)c1 67049,C1(NC(c2ccc(CO)o2)=O)CCC(CNC(c2cccn2C2CC2)=O)C1 67050,C1(O)(C(=O)NCC2(CCNC(C3(C)COCCO3)=O)CC2)CN2CCC1CC2 67051,C1(CC(=O)NCC(CC)NC(c2cc(C(N)=O)c[nH]2)=O)COc2ccccc2O1 67052,C1(C(=O)NC(Cc2ncn(C)c2)C(=O)O)CC12CCSCC2 67053,C1(NC(c2cc(C)c(Cl)s2)=O)C2CC1N(C(=O)C(O)Cc1ccccc1)C2C 67054,c1(OC)c(C(=O)NCCC(C)N(C)C(c2cnn(C(C)(C)C)c2)=O)csc1C 67055,c1(C(=O)NCC(CNC(CSCC=C)=O)S(C)(=O)=O)cc2n(n1)CCCC2 67056,Cc1csc(C(N2CCOC(CN(C(=O)CN(CC(C)(C)C)C)C)C2)=O)c1Cl 67057,c1(CNC(Cc2ccc(S(=O)(=O)N(C)C)s2)=O)cc2ccc(Cl)cc2[nH]1 67058,CCCCCCN(CCNC(=O)CN(C(C)CCC)C)Cc1ccoc1 67059,N1(C(c2cc(C)n(C)c2)=O)CCOC(C)(CNC(=O)CSc2ccc(F)cc2)C1 67060,C1(C)(C(=O)NCC(C(C)C)C)CCN(C(=O)C(=O)NCCC(N)=O)CC1 67061,CCC(C#N)C(=O)N1CC(CNC(=O)C=C(C)C)(COC)C1 67062,CCCC(CC)C(=O)NCC1CC2CC2N1C(c1cnn(CCOC)c1)=O 67063,O=C1CN(C(C23CCCCC2C3(F)F)=O)C(c2ccccc2)c2ccccc2N1 67064,c1(C(=O)NC2C(C)CN(C(=O)CC3CCNC3=O)C2)ccc2c(c1)C(C)CN2 67065,N1(CC)CCOCC1CC(=O)Nc1ccccc1.C12CC(C1)CC(=O)OC2=O 67066,N1(C(C=CCCC=C(C)C)=O)CCC12CN(C(c1cc(C)c(Cl)cn1)=O)C2 67067,C1(CC)CC(C(=O)NCCCC(C)NC(c2ccc(F)s2)=O)CCC1=O 67068,C(=O)(CCCCC(F)(F)F)NC1CN(C(C2(C#C)CCCC2)=O)CC12CC2 67069,c1(C(C)=O)ccc(C(N2CCC(C(=O)NC(c3nccn3C)C3CC3)C2)=O)o1 67070,N1(C(C(CC)n2cccn2)=O)CC(C2CCN(C(=O)C3=NOC(C)C3)CC2)C1 67071,C1(NC(c2ccn(CCC)n2)=O)CCCCN(C(c2ccc(O)nc2)=O)C1 67072,Cc1cnc(CCC(=O)N(CCN(C(=O)CCC2CC2CC2CC2)C)C)[nH]1 67073,CCC(CC(=O)NC1CC2CC1N(C(c1c(F)cncc1Cl)=O)C2)C(F)F 67074,c1(CC)nc(CC)cc(=NC2CCC(C(=O)N(CC)Cc3cncn3C)CC2)[nH]1 67075,c1(C(=O)NCC(=C)CCNC(C2(CC)CCNC2=O)=O)cc([N+](=O)[O-])ccc1Cl 67076,c1(C(N(C(C)CNC(c2onc(C)c2C)=O)CC)=O)cc(C(N)=O)ccn1 67077,C1(CNC(C(COCC)C)=O)CN(C(=O)CCCF)CCC1(C)C 67078,C(=O)(C1=CCCCC1C)NC(C)CCN(C(=O)Cn1nnc(C2CC2)n1)C 67079,c1(C(=O)O)n[nH]c2c1CN(C(=O)CCCn1cc(C3CCC(O)CC3)nn1)CC2 67080,c1(NC(C(CCNC(CN(C(C)C)C)=O)O)=O)cc(O)cc(F)c1 67081,N1(C(C2C(C)OC(C)C2)=O)CCC2(CNC(=O)CC3CSC3)CCCC12 67082,N1(C(CNC(=O)NC)=O)CCC(C(=O)NCC2CN(C3COC3)C2)C1 67083,N1(C(C(c2ccoc2)NC(C2C(OC)(OC)CC2)=O)=O)CC2CC(O)CC1C2 67084,c1(C(=O)NCC(C(C)O)O)ccc(-c2ccccc2Br)n1C 67085,N1(C(C(c2cncc(F)c2)C)=O)CC2CC(NC(C3(n4cncn4)CC3)=O)C(C2)C1 67086,C1(C(=O)NCCC(=O)NC(CSC)(C)C)CCS(=O)CC1 67087,N1(C(CCCCC#C)=O)CC2CN(C(=O)C=CC(F)(F)F)CCC2(CO)C1 67088,C(C(N=c1[nH]c(=N)[nH]c(=NCC2(OC)CCOCC2)[nH]1)c1ccco1)OC 67089,N1(C(C2C(OC)CN(C(C3(SC)CC3)=O)C2)=O)Cc2cnn(C)c2C1 67090,C1(C(=O)OC)(NC(C2CC2C(=O)NCCC2CCC(C)CC2)=O)CCCCC1 67091,N1(C(c2c(CCC)n(CC)nn2)=O)CC2CC1CN2C(=O)CCc1ccncc1 67092,C12(NC(=O)CSC(F)F)CC1CN(C(c1sc(N3CCCC3)nc1Cl)=O)C2 67093,C1(N(C(=O)CNc2ccccc2Cl)C)CCCCN(C(C2CC3(CC3)CO2)=O)C1 67094,c1(C(=O)NC(C(C(=O)NCCOCCC)C)C)cccc(F)c1C 67095,NC(=O)CCC(C(=O)NC1CC=CC1)n1cc(Cn2cc(Br)cn2)nn1 67096,N1(C(C(CCOC)OC)=O)CC2(CCN(C(=O)CC3CCOC(C)(C)C3)C2)C1 67097,C1(CC(=O)NC2CCCC(N(C(C3(CC)CC3)=O)C)C2)CN2CCN1CC2 67098,N1(C(C(c2ccc(CC)s2)=O)=O)CCC(NC(c2n[nH]cc2Cl)=O)C(O)C1 67099,N=c1[nH]c2ccccc2cc1C(N1CCCC1C(c1ccccc1)O)=O 67100,C1(NC(CCc2ccc(C)s2)=O)CC1C1CCCN(C(=O)Cn2ccsc2=N)C1 67101,CC1(C(=O)NC2CC(CNC(=O)CSc3cccc(Cl)c3)C2)CCCCC1(F)F 67102,N1(c2nnc(CCC)s2)CC2CC(NC(c3ccn(C(CC)CC)n3)=O)CC1C2 67103,c1(C(C)CNC(C2CC2c2cccnc2)=O)ccncc1Cl 67104,C(C(F)(F)C(F)F)OCCC(=O)OCC(c1ccccc1F)(C)C 67105,C12(NC(=O)CC(O)C3CC3)CCCC1(F)CN(C(=O)C(F)(F)C1CCCC1)C2 67106,N1(C(C2(F)CCC(C)CC2)=O)CCOC2(C1)CN(C(=O)CC1(C)CCOCC1)C2 67107,C(=O)(C1=NOC(C)C1)NCC1CC(NC(c2cccc(SCC#C)c2)=O)C1 67108,N1(C(CN(c2ccccc2)CC(=O)OCC)=O)CCCC(C)(C)C1CNC 67109,C1(CC)CC(C(=O)N(CC(CC)NC(=O)C=C(C)c2ccco2)C)CC(=O)N1 67110,N1(C(c2cc(SC)c(N)cc2)=O)CC2CCN(C(c3snnc3C(C)C)=O)C2C1 67111,c1(C(C)F)cccc(NC(C2CN(C(C3OC4CCC3C4)=O)CC2C)=O)c1 67112,c1(C(=O)OC)cc(C(=O)NC2CCCCC2NC(=O)CCS(C)=O)n(C)n1 67113,N1(C(C23C(NC(C4=CC(C)(C)C4)=O)C4CC2C3C4)=O)CCCC(C2(C)CC2)C1 67114,C(C)(C(=O)N1CC(CNC(c2cocc2C)=O)CC(C)C1)(C(C)C)OC 67115,N1(C(c2c(C)nsc2)=O)CCN(C(c2nocc2Br)=O)C2CC12 67116,C(=O)(C(CC1CC1)N1CCCC1)N(C1CCC1NC(C1CCOC1)=O)C 67117,CCC(C)CC(C)C(=O)N1CC(N(C(=O)CCOc2ccccc2Cl)C)C1 67118,C1(C(=O)Nc2ccc(C)cc2F)CN(C(c2cc(C#N)oc2C)=O)CC12CCC2 67119,c1(NC(C2(F)CCN(Cc3sc(Cl)nc3Cl)CC2)=O)cc(F)c(F)c(F)c1F 67120,N1(C(CCc2cccc(C)c2)=O)CCCCC(NC(c2nn(C)cc2Br)=O)C1 67121,C1(C(N(CC(=O)N(CC(=O)NC)C)C(C)C)=O)COCCN1C 67122,NS(=O)(=O)CCC(=O)NC1(CO)CN(C(C2(F)CCCOC2)=O)C1 67123,C(CC(=O)NOCCC1CC1)(C(C)(C)C)NC(C1CC(CC)C1)=O 67124,c1(NC(=O)CC2CC3CC(=O)C2C3)ccc2nccnc2c1I 67125,c1(C(=O)NCC2C=CC(NC(c3c(CCC)nns3)=O)C2)n[nH]c2c1CCC2 67126,C1(C(=O)NCC(C)(CO)NC(CCS(=O)(=O)NC)=O)CCc2ccnn2C1 67127,CC1(C)CCCC(CC(=O)NC2(C)CCN(C(C3(O)CC3)=O)CC2)O1 67128,C1(C#N)(C(=O)NC(C(C)NC(c2ccc(NC(C)C)nc2)=O)C)CCCOC1 67129,C1(NC(CCN(C(C(C=C)O)=O)C(C)C)=O)CCNC(=O)CC1 67130,N1(C(=O)CCc2cc[nH]n2)CCN(C(C23CCCC(C2)OC3)=O)CC1CCO 67131,c1(NC(C(CCNC(=O)CCCn2cncn2)O)=O)ccc(O)c(F)c1 67132,Nc1cc(Cl)cc(F)c1C(=O)NCC(CO)NC(=O)CCC(=O)N1CCOCC1 67133,c1(C(=O)NCCN(C(C2CCCN2N=O)=O)CC)cc(Cl)cc(F)c1Br 67134,S(=O)(=O)(c1cncn1C)NC(C)Cc1nccn1C 67135,C1(NC(C2C(=O)NCCCC2)=O)CCC(O)CN(C(C2(C(F)(F)F)CC2)=O)C1 67136,C1(NC(CC(=O)NCC#C)=O)CS(=O)(=O)CC1NC(c1nccc(N)c1Cl)=O 67137,c1(C(=O)NCC2C(NC(CCCN(C(C)=O)C)=O)C2)c(Cl)nsc1Cl 67138,C(=O)(C(O)CCC(C)C)N1CC2C(NC(c3ccc(OC)c(C4CC4)c3)=O)(C2)C1 67139,c1(NCCN(C(=O)CC2CCCCC2(F)F)CC)ncn(C)c(=O)c1Br 67140,c1(CC)ncc2c(n1)CCC(C(=O)N(C1CN(C(C3CCCCC3)=O)C1)C)C2 67141,C=C(CC)CN=C(NCc1cccs1)NCc1ccc(OC)c(OC)c1C 67142,C1(NC(C2(C)CCC(=O)N2)=O)CCC(O)CN(C(=O)Cn2ccc([N+](=O)[O-])n2)C1 67143,C(C(CC(=O)Nc1cnn(C(F)F)c1)NC(C1C=CCCC1)=O)OC 67144,O=C1CN(CC(N2CCN(C(c3nc(C4CCC4)no3)C3CC3)CC2)=O)CCCN1 67145,c1(C(=O)NCC(CC(C)C)NC(=O)C(O)c2ccsc2)csc2ccc(F)cc12 67146,C(=O)(C#CC(C)(C)C(F)F)N(C(C)CNC(C1CCCN1c1ncccn1)=O)C 67147,C1(CNC(=O)CCF)CN(C(=O)Cc2sccc2Cl)CCO1 67148,Cc1ncc(Cl)c(C(=O)NCC2CCN2C(=O)Cc2nnn(C(C)(C)C)n2)n1 67149,N1(CC(=O)NCCC2CCN(C(c3cnn[nH]3)=O)C2)CCC(n2cccc2)CC1 67150,C1(CC)CCN(C(=O)Cc2ccsc2C)C(C(=O)N(CC(O)C2CC2)C)C1 67151,C(C1C(C(=O)NCCC(C)N(C)C(C2CCC=CO2)=O)C1(C)C)=C(C)C 67152,C(=O)(C(CCC1CC1)NC(c1cscc1C)=O)N1C(CCC)CCC1 67153,C=C(C)c1cncc(C(=O)NCCSCC)c1.C(C)(=O)O 67154,N1(C(C(C)c2ccco2)=O)CCCC(NC(c2ncc(Cl)nc2Cl)=O)C1C 67155,Cc1ncnc(C)c1C(N1CCCC(C(=O)NCC(C)(O)C2(C)CC2)C1)=O 67156,c1(-n2cc(C3OCCN(C(CCC4CCC(C)O4)=O)C3)nn2)cc(F)cnc1Br 67157,N1(C(C(CN(C)C)NC(C(N2CCOC2=O)C)=O)=O)CCCC2OCCC12 67158,c1(CC)noc(C)c1NC(=O)COC1CC(NC(C2(C#N)CC2C)=O)C1 67159,c1(CCNC(C(C)SC)=O)ccc(CNC(=O)C(N2CCSCC2)C)cc1 67160,Cc1cccc(Cl)c1CC(N1CC2C(N(C(=O)COC3CCCC3)C)C2C1)=O 67161,C1(CC)CNC(=O)CN1C(=O)C(C1CCCC1)NC(=O)CC1(N(C)C)CCCC1 67162,CCC(CC(=O)NCC1(OC)CCN(C(c2nn(C)nc2Br)=O)C1)SC 67163,C1(NC(C(C)OCC(C)C)=O)CCCC(CNC(c2cnc[nH]c2=N)=O)C1 67164,c1(C(N2CC(C)C(NC(C3CCCC(CF)C3)=O)C2)=O)nn(C)c(Cl)c1Cl 67165,N#Cc1ccc(CC(C#N)C(=O)Nc2cccc(F)c2)cc1 67166,Cn1c(NC(=O)CC(O)c2ccccc2)nc2cc(Br)c(Cl)cc12 67167,C(C(=O)NCCC1CCN(C(=O)C(C)N(C)C)C1)(C(C)C)NC(C)=O 67168,CCC(CCOC)C(=O)NC(C)CCCC(=O)N1CC(F)(C2CC2)C1 67169,N1(C(CCCNC(=O)OC)=O)CCN(C(=O)CCc2ccc(C)cc2)C2CCC12 67170,c1(CC(=O)N(CC(C)(C)CNC(=O)C=C2CCC2)C)ccccc1O 67171,C#Cc1ccc(C(=O)NCC2CC2CNC(C2CC(C)(F)C2)=O)c(F)c1 67172,C(c1ccc(=N)[nH]c1C)=CC(N1CC(COC)(NC(=O)CC(C)C)C1)=O 67173,CC1(C(=O)NCc2cc(C(=O)NCCCC3(O)CCC3)on2)CCOC1 67174,C1(C(=O)NCC(CC)NC(c2scnc2C)=O)CCCNS1(=O)=O 67175,N1(C(C(C=C)(C)CC)=O)CC2CC(NC(c3ccc(Cl)c(O)c3)=O)C(C2)C1 67176,N1(C(COC(C)C)=O)CC2CCCC1(CNC(c1coc3ccccc13)=O)C2 67177,C(=O)(C#CC1(C)CCCO1)NCC1C(NC(CN(CCC)C)=O)CCC1 67178,C1(NC(C2CCC(CC)O2)=O)CC2CCC1(C(N1CCC1c1ccccc1)=O)C2 67179,C1(CNC(c2c(C)oc(CO)c2)=O)CC2(CCN(C(C3(C)CC3(F)F)=O)C2)CO1 67180,c1(C(=O)NCC2N(C(C3C(C)C3C)=O)CC(C)(C)OC2)c(F)cc(F)c(F)c1F 67181,Cc1ncc(C(C)NC(=O)NCCCN(C(=O)OC(C)(C)C)C2CC2)cn1 67182,c1(CN2CC(C#N)C(NC(c3cc(Br)c[nH]3)=O)C2)cc2cc(F)ccc2s1 67183,C1(NC(c2cc(Br)n3c2CCC3)=O)CN(C(=O)CCC2CCC2)CC2(CC2)C1 67184,c1(C(=O)NCC23CCCC2CN(C(c2cnns2)=O)C3)cnn2c1C(=O)NCC2 67185,N1(C(Cc2cc(OC)c(F)cc2)=O)CC2CCC1CC2NC(=O)CC(C)(C)C 67186,O(N1CCC(NC(=O)CC2CCCC2NC(=O)C2=C(C)CCC2)CC1)CC 67187,CC1CCC(NC(=O)CC2COCCOC2)CN1C(c1cc(C(N)=O)ccn1)=O 67188,c1(CCC(=O)NC2CN(C(=O)C)C2)ccc(F)cc1.C1(CC#C)CCCC1 67189,N1(C(c2cc(C(C)=O)[nH]n2)=O)CCOC2CN(Cc3c(C)cc(Br)cc3C)CC12 67190,CC1(C)C(=O)NC2CCC(C(=O)Nc3ccc(SCc4nc[nH]n4)cc3)CC12 67191,C1(CC2(C(=O)NC3CC3)CC2)CCN(C(c2cn(C)cc2C(F)(F)F)=O)C12CC2 67192,c1(CS(C)(=O)=O)ccc(CN(C)C(C2CCN(C(CC(C)O)=O)C2)=O)cc1 67193,C1(OC)(OC)CC(C)(C(=O)N(C)CC2(O)CN(C(c3n[nH]c(C)c3Cl)=O)C2)C1 67194,CCS(=O)(=O)c1ccc(Cl)c(C(N2CCC(NC(=O)C(C)CO)C2)=O)c1Cl 67195,c1(C(CNC(C2CC(OC)C2)=O)NC(=O)C(C)=C2CC2)ccc(C)cc1 67196,N1(C(c2nn(C)c(=O)cc2)=O)CC2(CCC2)CC1CNC(=O)C(F)C1CCOC1 67197,S(=O)(=O)(c1ccc(C#N)c(N(C)CCF)c1)N(C1C(C)CCC1)C 67198,C1(CNC(CC(C)OC)=O)CN(C(=O)CC2CCCOCC2)CCC12CCOC2 67199,C1(NC(CCC(C)OC)=O)CN(C(=O)CCn2nc(C)cc2C)CC2CC12 67200,C1(NC(Cc2c(C)n(C)nc2)=O)CCCN(C(c2cc[n+]([O-])cc2)=O)C1C 67201,c1(C(N2C(C)CCC(NC(=O)CC3NC(=O)NC3=O)C2)=O)cc(N)cc(O)c1F 67202,N1(C(C(c2ccoc2)SCC)=O)CCCC(C(=O)NCc2nnc(O)o2)C1 67203,N1(C(c2c(CC)csc2)=O)CC(NC(c2cnc(C)s2)=O)C2CC12 67204,c1(C(=O)NCC2(F)CN(C(=O)CCC3CC(F)(F)C3)C2)cncc([N+](=O)[O-])c1 67205,CN1C(=O)CN(C(=O)CC2C3CN(C(C4CC(C)(C)CN4C)=O)CC23)CC1=O 67206,c1(C(N2CC(O)(C(C)NC(=O)CN3CCC(C)(O)C3)C2)=O)ccc(N(C)C)cn1 67207,C1(=O)CC(C)C(=O)N1.c1(C(N2CCC(O)CC2)CCC)cc(F)ccc1F 67208,C1(O)(CNC(C2(CC=C)CCC2)=O)CN(C(=O)C(C)OCC2CCCO2)C1 67209,C(=O)(C(C(C)(C)NC)C1CCCC1)NC1C(CC)CN(C(=O)OC(C)(C)C)C1 67210,c1(CC)[nH]c(=N)sc1C(=O)NCC(O)CN(C)C(c1ccns1)=O 67211,c1(C(C)C(=O)NC2CCCN(C(=O)C=CCO)C2)ccc(S(=O)(=O)N(C)C)cc1 67212,N1(C(Cc2ccc(C)o2)=O)CC(C(N2CCC(C(F)F)CC2)=O)CC(C)C1 67213,c1(C2C(C(=O)NC(CC)CNC(=O)CCn3cncn3)C2)ccc(C)cc1 67214,Cc1c(Br)ccc(N2CCN(C(=O)CCC34CCC(CC3)C4)CC2C)c1[N+](=O)[O-] 67215,Cc1cc2cc(C(=O)N(C)CCNC(C3(C(F)F)CC3)=O)c(Cl)cc2[nH]1 67216,C1(C(=O)NC2CCC(C(=O)NCC(C)CC3CCC3)C2)(OC)CCOC1 67217,C(=O)(CC1CC(C)(OC)C(=O)N1)N1C(CCC#C)CCC1.C1CC1.OC 67218,N1(C(COCCCCC)=O)CC2(C1)C(NC(c1cc(C)oc1C)=O)CCS2(=O)=O 67219,C1(C)(CNC(C23OCC(CC)(C2)C3)=O)CCN(C(=O)COCC2CCCC2)CC1 67220,Cc1nc2sc1C(=O)NC2.C1(C(=O)Nc2nccs2)CCOC(C)C1 67221,N1(C(C2Cc3cc(F)ccc3O2)=O)CCCCC2(C1)CN(C(c1cc[nH]c1)=O)C2 67222,C1(C(C(=O)N(CC=C)CCOC)NC(c2cnco2)=O)CC=CCC1 67223,c1(C(CNC(C)=O)NC(c2c[nH]nc2[N+](=O)[O-])=O)ccc2ccccc2c1 67224,N1(C(C(C)SC)=O)CC(NC(=O)C=CCCC(C)C)CCC1C 67225,c1(NC2(C(=O)OC)CCOC2)ccccc1C.C1(CC2CCC2)C(=O)N1C1CC1 67226,Cc1nc2cccc(C(=O)NC3COCC3CNC(C34CCC(C3)C4)=O)c2[nH]1 67227,c1(CC2CCN(C(C(=O)NCC3(F)CCNC3)=O)C2)ccc(F)cc1 67228,c1(NCCCC(=O)OCc2nc(SC)nc(O)c2)ccc2c(c1)CCO2 67229,C1(COCC)(CO)CC(N2CCC(Oc3ccc(OC)cc3)CC2)C(O)C1 67230,C1(CC(=O)NCC2N(C(C(F)=CCC)=O)CCC2)COC2CC1C2 67231,c1(OC)c(N(C)CC2CCCN(C(c3ccc(F)o3)=O)C2)ncnc1Cl 67232,N1(C(C=NOC)=O)CCC2(CC1)CC(NC(=O)C(CO)NC(N)=O)C2 67233,S(=O)(=O)(CCCCCl)C1C(C(=O)NC(C2CCCCC2)CO)C1 67234,C12(C(=O)NCC3C(C)CCN(C(C4(O)CCSC4)=O)C3)CCC(CC1)C2(C)C 67235,C=C1Cn2c(C(=O)NCC3CC4CN(C(=O)C=CSC)CC34)nnc2S1 67236,C1(NC(c2cc(OC)c(Cl)cc2Cl)=O)COC2(CCN(C(=O)C3CC3)CC2)C1 67237,N1(C(Cn2c(C)c(Cl)cn2)=O)CC(C)N(C(=O)CC(F)(F)C(C)C)CC1C 67238,CC1C(NC(=O)CN(CC(C)(C)C)C)CCCN1c1ccc(C(F)(F)F)cn1 67239,N1(C(CC(=O)OCC)=O)CC2(CC(CC(=O)NCC3(C#N)CC3)C2)C1 67240,N(C(=NCCCCC(F)(F)F)NCCC1(O)CCCC1)C(CC)CC 67241,C1(C(=O)NC(c2cccc(F)c2)c2n(C)ccn2)CC(C2CC2)=NO1 67242,Cc1cc(NC(C2CC(O)CN2C(c2cccc(I)c2Cl)=O)=O)ccc1O 67243,c1(OCC)ccc(Cl)c(NC(C2CCN2CC2CCCC2)=O)n1 67244,N(C1CN(C(=O)C2=CCCOC2)Cc2ccccc21)C(Cn1c(C)nnn1)=O 67245,CC1CCCC(CC(=O)NCC(C2CCCCC2)NC(C2CC(F)C2)=O)C1 67246,CC(C(=O)N1CC2CC1C2NC(c1ccc(F)c(C(F)(F)F)c1)=O)C(F)(F)F 67247,c1(N2CCC(CNC(C(COC)(C)C)=O)C2(C)C)cc(C#N)nc(C2CC2)n1 67248,c1(C(N2CCN(C(C(CC)OC)=O)C(C3CC3)C2)=O)cc2ccc(F)c(F)c2o1 67249,C1(c2cn(CC)nc2)CN(C(c2cnn(C3CCOCC3)c2Cl)=O)CCO1 67250,C1(NC(CCC(C)NC(c2c(C)ncs2)=O)=O)CN(C)CC1(F)F 67251,C(=O)(CCN(CCO)C(C1(C)CC1)=O)NCC1C(C(=O)OC)C1 67252,C1(CC)CN(C(c2cnc(=N)[nH]c2)=O)CC1C(=O)NC1CC=CC1 67253,C1(COC)(NC(c2coc(C3CCC3)n2)=O)CCN(C(C2COC2)=O)C1 67254,Cc1cccnc1C(C(C)(C)C)NC(=O)C(=O)NC12CC(c3ccccc3)(C1)C2 67255,C(C)(CCCC(=O)NCCCCn1ccnc1)NC(Cc1c(C)scc1)=O 67256,C1(NC(C2(C)CCCCCC2)c2n(CCOCC)nnn2)CCCC(C)(C)C1 67257,N1(C(CNC(CCC(C)C)=O)=O)CCC(NC(=O)CC2CNC(=O)C2)C12CCC2 67258,c1(CC2N(C(CN(c3cccs3)C)=O)CCC2)c(N)cccc1Cl.C1(=O)CO1 67259,N1(C(C(=O)NC(COCC)C)=O)CC2CC2C2CC12 67260,c1(C(=O)NC2CC(CNC(C3CCCC3(F)F)=O)C2)ccc2nc(S)oc2c1 67261,C1(C(N(CC(CCC)O)C)=O)CCN(C(=O)C#CC2(C)COC2)C12CCC2 67262,C1(=CC(=O)NCC(CN(C(C(CC)O)=O)C)O)CC2CCC(C1)N2C 67263,N(C(=NCCCN(S(C)(=O)=O)C)NCC1CCCCO1)C(CC)C 67264,CC1=C(C(=O)NC2CC3CC(NC(C4CC(C(C)C)=NO4)=O)CC3C2)CCCC1 67265,CC1CCCN(C(=O)Nc2ccccc2NC2(C)CCCO2)C1 67266,c1(C(N2CC(CNC(c3n(CC)nnc3C)=O)OCC2)=O)c[nH]c(C)cc1=O 67267,Cc1c(C(N2CC3(CC3)CC2CNC(=O)CNC(N)=O)=O)sc2ccccc12 67268,C(CC(C(=O)N1CC(O)C(O)C1)NC(C1SCC=C1C)=O)SC 67269,c1(CNC(C(C)NCCC)=O)nc(C(C)N)n[nH]1 67270,C1(C)(CNC(CC2C=NN(C)C2=O)=O)CN(c2cc(C(F)(F)F)ncn2)CCO1 67271,CC1CCN(C(=O)CCc2c(Cl)cncc2Cl)CC1NC(c1ccoc1Cl)=O 67272,c1(CC(=O)NCC(C)NC(=O)Cc2cncs2)ccnc(O)c1 67273,C1(CNC(C(C)OC)=O)CCCC1NC(C1CCC2CC12)=O 67274,c1(C(=O)NCC23CCC(CC2)N(C(C2CC2(Cl)Cl)=O)C3)ccc(F)cc1[N+](=O)[O-] 67275,c1(-c2cccc3nc(C(=O)OC)[nH]c32)cc2ccccc2cc1O 67276,C1(CNC(CC=CC)=O)CC(NC(c2cn(C)cn2)=O)C12CCC2 67277,N1(C(C2CCOCC2)=O)CCC(N(C2(C3CCCO3)CC2)C(C2CC2)=O)C(F)C1 67278,C(=O)(CC1C(=O)Nc2ccc(Cl)cc21)NC1CC(NC(C(CC(=O)OC)C)=O)C1 67279,N1(C(CC2(CNC(c3cc(C)c(O)nn3)=O)CC2)=O)CCCC2(C)CCC12 67280,C1(NC(c2ccc(I)c(Br)c2)=O)CN(C(=O)Cn2cc(Cl)cn2)CC1(F)F 67281,c1(CN(CCC)C(=O)Nc2nc(C(C)C)ns2)cc(Cl)ccc1Br 67282,C(=O)(C(F)C(CC)CC)N1CCN(CC(C)NC(c2nc(CC)oc2)=O)CC1 67283,C(=O)(C1=CS(=O)(=O)CCC1)NC(C)CCCCNC(=O)CC1C=CCCC1 67284,n1(CC)cnc2nc(N3CCN(C)C4(CCC4)C3)nc(N(CC(F)(F)Br)C)c12 67285,CCC(CC(C)CO)NC(=O)N(C1CCSC1)C 67286,CCS(=O)(=O)CC(=O)N(C(C)CCNC(=O)CCCC(C)c1ccccc1)C 67287,CCC(CNC(=O)CC1CCCC1NC(=O)CCC(=O)NC)C(C)C 67288,C1(CNC(C(C)(O)CCc2ccccc2)=O)CC2CCC1N(C(=O)CCF)C2 67289,C1(NC(CSCC(=O)OC(C)(C)C)=O)CCCN(Cc2ccc(O)c(O)c2)CC1 67290,C1(CNC(CNC(C(c2ccccc2)N(CC)CC)=O)=O)(CO)CCN(C)C1 67291,c1(C(N2C(C)C(NC(=O)CCSC(F)(F)F)CCC2)=O)ccnc2c1ncn2C 67292,C(=O)(CN=c1[nH]c(C)cs1)NCC1CN(C(c2cnc(OC)c(C)c2)=O)CC1C 67293,N1(C2CN(C(COC(C3CC3c3ccco3)=O)=O)C2)CCCS1(=O)=O 67294,c1(C(=O)NC(C2CCOC2C)C)ccc(-c2cnco2)cc1Cl 67295,C1(CCC)CN(C(=O)CC(C)C)CC1C(=O)NCC(C)(O)C1CCC1 67296,C1(C(C)C)CN(C(=O)CC(C)c2cnn(C)c2)CCN1C(c1ccoc1Cl)=O 67297,C1(CN(C(C(C)OCc2ccccc2)=O)C)CCCN1C(=O)CC1CCCO1 67298,C(=O)(C(F)C(F)(F)F)NCC(C)N(C)C(c1ccc(C(F)F)cc1F)=O 67299,CN1CCC(C(=O)NC2(CNC(C3CCC(F)C3)=O)CCC2)CC1=O 67300,N1(C(c2n(CCC)ncc2Br)=O)CC(C#N)CC1C 67301,C(c1ccc(F)nc1)=CC(=O)NCC(CNC(c1c(C)nc(N(C)C)s1)=O)C 67302,C1(N(C(c2ccc(CNC(C)=O)s2)=O)C)CCCN(C(C2COC(=O)O2)=O)CC1 67303,C(=O)(CC(C)(C)CNC(c1cc(Cl)n[nH]1)=O)NCC(C)Cc1cn[nH]c1 67304,C(=O)(C(C)(O)C(F)(F)F)NCCC1CN(C(C2CC(OC)C(OC)C2)=O)C1 67305,C(CCC(CCC)NC(c1n[nH]c(C)c1C)=O)NC(c1cn(CCCC)nn1)=O 67306,C1(CNC(C(C)SCC)=O)(CO)CCCN(C(C2CCCN2C(C)=O)=O)C1 67307,C(=O)(CC1=CCOCC1)N1CC(C(=O)Nc2cc(C)c(O)cc2)C(C)(C)C1 67308,Cn1ccc(=O)c(C(=O)NCCCN2CCN(C(C3CCS(=O)(=O)C3)=O)CC2)c1 67309,Cc1cc2ccccc2nc1C(N1CC2CCN(C(c3csnn3)=O)CC2C1)=O 67310,C(CCCCC(=O)N1CC(NC(=O)CSC)CC(C)C1)OCC 67311,c1(OC(=O)CCc2cccc(OC(F)F)c2)cc2n(n1)CC(O)CO2 67312,CC1(C)CC(CC(=O)NCCCNC(C2(C(F)F)CCCO2)=O)CO1 67313,N1(C(CCS(=O)(=O)NC)=O)CCC2(CC1)CC2NC(=O)C(c1cccc(C)c1)C 67314,c1(C(=O)OC)cc(NC(c2sc(NC(C3CCCS3)=O)nc2C)=O)c(C)cc1Br 67315,c1(C(N2CC(C)OC(CCNC(=O)C3=CCCC3)C2)=O)cc(C#N)ccc1F 67316,c1(C(=O)NC2(CO)CCN(C(CC3ON=C(CC)C3)=O)C2)cc(C)nc2ccnn12 67317,N1(C(c2c(C)nco2)=O)CCCC(O)(CN(C(=O)C(C)CN2CCCCC2)C)C1 67318,C1(NC(C(C2CCC2)NC(=O)C(F)OC(F)(F)F)=O)CN2CCCC1C2 67319,CC(CN1CCOCC1)N=c1[nH]c(=NC(C)c2nc[nH]n2)[nH]c2c1CCCCC2 67320,Cn1ccc(-n2cc(C(CC(N)=O)NC(C3CCCS3)=O)nn2)cc1=O 67321,C1(CNC(c2n(C(C(=O)OC)C)nnn2)c2ccoc2)CCOC1(C)C 67322,c1(C(=O)Nc2cc(Br)cc(I)c2)cccn2c(-c3ccc(O)c(CO)c3)cnc12 67323,n1(CCCOC(C(C=C)C)=O)nc(O)c2ccccc2c1=O 67324,c1(CN2CC3CN(C(=O)CCc4ccccn4)CC32)ccc(I)c(F)c1F 67325,C(=O)(C#CC1CCCOC1)NCCOCCN(C(CC(C(=O)OC)C)=O)C 67326,CCC(C)C(C)(O)CNC(=O)C(CC(C)C)ONC(C1CC12CC(NC)C2)=O 67327,N1(CCN(C(CN(C(=O)C(C)SCC)CCC)=O)CCC)CCCCC1 67328,CC1CCCC(O)(CNC(C2(NC(=O)Cn3ncccc3=O)CCCC2)=O)C1 67329,N1(C(c2c(CNC(CCCCC)=O)n[nH]c2)=O)CCCC(C)(N(C)C)C1 67330,c1(CNC(C(CO)OC)=O)ncccc1C(=O)N(CCCCSC)N(C)C 67331,N1(C(c2c(CC)ocn2)=O)CC(NC(c2cc(O)ncn2)=O)C2CCCCC12 67332,Cc1ccc(Cl)c(C(=O)NCC2(O)CCN(C(C3CC34CCCC4)=O)CC2)c1N 67333,C1(OC)CC(CN(C(=O)CC(C)(C)C)CC)N(C(=O)CC(C)c2cccnc2)C1 67334,CCCC(O)C(CO)NC(C12CC1CCN2C(C1CCCC(=O)CC1)=O)=O 67335,C(=O)(C(F)C(C)(C)O)N(CC(C)(C)C)CC(C1CCN(C(=O)CCNC)CC1)C 67336,N1(CCC)CCCCC1C(=O)N(C)CCC1CCCCN1C(c1cnc(C)s1)=O 67337,N(C(=NCc1cccs1)NC1CC12CCCC2)CC(F)F 67338,CCCC(CCO)NC(=O)CC1(N(C(=O)C(CC)OC)C)CC1 67339,c1(OC)cc(C(=O)NCCc2ccccc2O)cc(C)c1 67340,c1(CNC(C(=O)NC2CCC(OC(C)(C)C)CC2)=O)ccc(Cl)cc1Cl 67341,C12(CNC(C(C(C)O)C)=O)CC(NC(=O)C3=CCCC3)(C1)C1(CCOCC1)O2 67342,N#Cc1cc(C(N2CCC(F)(C(=O)N(C3CCOCC3)C3CC3)C2)=O)cs1 67343,C1(NC(=O)C=C2CCCCC2)(CF)CCN(C(=O)C(c2cccc(F)c2)O)C1 67344,N1(C(C2(CCCC)CC2)=O)CCCC(C2CCCN(C(C3C4COCC34)=O)C2)C1 67345,N1(C(CP(C)(C)=O)=O)CCOCC(NC(c2ccccc2Cl)=O)C1 67346,N(C(=NCCN1CCOC1=O)NCC1CCCCO1)C1CC(C)OC1 67347,CS(=O)(=O)c1cnn(CC(=O)NC2CCCC(NC(=O)CSC(F)(F)F)CC2)c1 67348,c1(OCC(=O)NCCC2CCN(C(c3nc(OC)oc3)=O)C2)cncc(Cl)n1 67349,C1(C(N2C(CCNC(c3cnco3)=O)CCC2)=O)CC(F)(F)C12CCC2 67350,Cc1cc(CN2CCC2Cn2cc(C3CCCC3O)nn2)cc(C(F)(F)F)c1 67351,CCCC(CC)CC(=O)N1CC2CCC(C1)N2C(c1nc(Br)c[nH]1)=O 67352,C1(CNC(C2(OCC)CC2)=O)CN(C(=O)C(C)C(F)F)CC1(F)F 67353,N1(C(=O)NCC(c2cccs2)=O)CCC2CC2C1 67354,C1(NC(c2nccc(OC)c2)=O)CN(C(=O)C(C)(C)N(C)C)CCC1C(F)(F)F 67355,C1(COC)CC(CNC(C2CC2C(C)(C)C)=O)N(C(=O)COCC(C)C)C1 67356,c1(CN(C)C(C23COCC(C2)C3)=O)ccccc1CNC(C1(F)CC=CCC1)=O 67357,c1(C(=O)NC2CC(CNC(C3(CC)CCNC3=O)=O)C2)nnn2c1C(=O)NCC2 67358,C(=O)(C(C)(C)C(C)(C)C)NC1CN(C(CC2C(C(=O)OCC)C2)=O)C1 67359,Nc1ncc(C(N2CC(CNC(c3ccco3)=O)C2)=O)cc1Br 67360,c1(C(=O)NC2CCC(N(C(=O)CCc3cccc(F)c3)C)C2)nccc(N)c1Cl 67361,c1(C(N2CCN(C(=O)OC(C)(C)C)CC2C(F)F)=O)cc(F)cc2nccnc12 67362,Cc1ccc(F)c(CN2CCN(Cc3cnc(Cl)c(Cl)c3)CC2)c1Br 67363,C1(C(=O)NCC2CC(OC)C2)(NC(=O)CCC2(C#N)CCC2)CCSC1 67364,C(=O)(C(C)(C)C(=O)NC(C1CCCCN1C(c1cc(Cl)n(C)n1)=O)C)OCC 67365,C1(CNC(c2ccc(OC)o2)=O)CCC(CNC(=O)C(O)C2CC2)CC1 67366,Cc1cc(Cl)c(Cl)cc1C(N1CCCCC1C1(NC(=O)CSC2CC2)CC1)=O 67367,C1(C(N2CCC(N(C(=O)CC(C)(C)C3CC3)CCC)CC2)=O)CC(C2CCC2)C1 67368,c1(CC)ccoc1C(=O)NC(C)(CNC(=O)CCOCCOCCCO)CC 67369,Cc1[nH]c2ccccc2c1C(N1CCC2(C1)CN(C(C1C(F)(F)C13CC3)=O)C2)=O 67370,C=CCC(C(=O)N1CC(CNC(c2cc(Br)cnc2C)=O)(OC)C1)C(C)C 67371,c1(CNC2CN(C(CCc3c(C)noc3C)=O)CC2C)cc(F)cc(C#N)c1 67372,c1(N(CCNC(C2CC2C(=O)OC)=O)CC)cc(C(C)C)nc(C)n1 67373,N1(C(C(C)N2CCCC2)=O)CCCCC(CNC(=O)CN(c2ncccn2)C)C1 67374,N1(C(CC=C)=O)CC(CN(C)C(c2cc(Br)ccc2C)=O)C2(CC2)C1 67375,C1(N(C(c2cc(OC)ns2)=O)C)CCN(C(c2cccc(C)c2O)=O)CC12CC2 67376,C1(CNC(C2(OCC)CCOC2)=O)(CNC(=O)CC(F)F)CC12CCC2 67377,C(CCC(C)(C)C(=O)NC(C1(O)CCC1)C)NC(c1c(=O)cc(C)[nH]c1)=O 67378,N1(C(CC2CC(C(=O)OC)C2)=O)CCCC(N(C(=O)C=CSC)C)C1 67379,c1(NC(=O)Nc2ccccc2)ccccc1OC1CC(c2nccc(CO)n2)C1 67380,CC(C)CCC(C(=O)NCc1ccnc(F)c1F)NC(c1cnn[nH]1)=O 67381,CC1CN(C(C2(Cl)CC2(F)F)=O)CC1NC(c1cc(CC(F)(F)F)nn1C)=O 67382,c1(C(=O)NC2CCN(C(C3CC(C#N)C3)=O)CC2O)cccc2c1OCCO2 67383,N1(C(CCOC(C)C)=O)CCC2CCN(C(c3cc(C(F)(F)F)n(C)n3)=O)C2C1 67384,c1(CNC(=O)Cc2cccc(C3CC3)c2)ncc([N+](=O)[O-])cn1 67385,c1(OC)cccc(CN2CCC(CNC(c3csc(C)n3)=O)C2)n1 67386,c1(C(=O)NCC(C)(C2CC2)NC(c2nncs2)=O)ccc(-n2ccnn2)cc1 67387,n1(CC(N2CCC(C(C)NC(C3CC(N=[N+]=[N-])C3)=O)CC2)=O)ncc(O)nc1=O 67388,C(CCN(C)C(c1ccc(OC)o1)=O)(C(C)C)NC(c1cc(SCC)on1)=O 67389,Cc1csc2ccc(C(=O)NC(C)CCCNC(C3CCC(O)C3)=O)cc12 67390,C(N=c1cc[nH]cc1S(=O)(=O)NCC1CN(c2ccccc2Br)C1)C1N(C)CCC1 67391,C1(C(=O)NC23C(CN(C(C4(CC=C)CCC4)=O)C2)C3)COc2ccc(F)cc2C1 67392,C1(C(=O)NCCCN(C(=O)CN(C)CCOC)CC)CC=CCC1 67393,C(CC(C(C)(C)C)NC(c1ccnc(C(F)F)c1)=O)N(C)C(C1CC=CCC1)=O 67394,N1(C(C2C=C(C)CS2)=O)CC2(C)CC1(C(=O)N(C1CCN(C(C)C)C1)C)C2 67395,Cc1ccc(C(N)=O)cc1C(=O)NCC1CC(NC(=O)C(C)CC(N)=O)C1 67396,Cc1nc(CCC(N2CCC(CO)(NC(=O)CC3CC34CC4)C2)=O)oc1C 67397,C#Cc1ccc(C(=O)NCCC(CNC(=O)CN2CCC(=O)CC2)OC)cc1 67398,C1(OC)CCC(C(=O)NCCn2cc(C(N3CC(C(C)(C)C#N)C3)=O)nn2)CC1 67399,Cc1cc(F)c(F)cc1C(N1CC2CC2(C(=O)Nc2ncc(Br)nc2Cl)C1)=O 67400,c1(CN2CC(C(=O)NCc3c(C)cccc3)SCC2)cc([N+](=O)[O-])cc(O)c1O 67401,C1(CC)CN(C(=O)Cc2cccnc2)CCC1NC(c1sncc1C)=O 67402,N1(C(CCS(=O)(=O)N(C)C)=O)CCOC2(C1)CN(C(C1CC13CCOC3)=O)C2 67403,c1(C(N(CC(O)CN(C)C(C2CCCN2N=O)=O)C)=O)ccn(C)c(=O)c1O 67404,C1(CC(=O)NCC(CO)NC(C2CC2Cc2ccccc2)=O)CCCCCC1 67405,Cc1cccc(CNCC2COCCN2C(c2ncc(Br)cc2Cl)=O)c1F 67406,C1(CNC(C(C)NC(C)(C)C)=O)CC2(CC2)CN1C(=O)CC1(C)CCCCC1 67407,N1(C(CCN(C)CC)=O)CCC2(CCCCN(C(C3(Cl)CC3(C)C)=O)C2)C1 67408,N1(C(N=c2nc(C)s[nH]2)=O)CC(C)(C)OC2(CCOC2)C1 67409,c1(C(N2CC3CN(C(C(C)(C)C(F)F)=O)CC3C2)=O)nc2ccc(Cl)nn2n1 67410,N1(C(c2c(CC)csc2)=O)CC2CS(=O)(=O)CC2(NC(c2ccc(=N)[nH]c2)=O)C1 67411,N1(C(C2C(C)OCC2)=O)C2CCC1CN(C(=O)Cc1ccnn1C)C2 67412,c1(OC)c(C(=O)NC2(C)CN(C(C3(C)CC3(F)F)=O)C2)ccnc1Cl 67413,C1(NC(Cn2c(C)nnn2)=O)CC2CC(C1)N(C(=O)CC1CC(F)(F)C1)C2 67414,Cc1cc(C(F)(F)C(=O)N(CC(O)CNC(C2CCC(C)O2)=O)C)cc(C)c1 67415,C1(C(=O)NCc2cc(C(N(CC(C(C)C)OC)C)=O)n(C)n2)CCC(N=[N+]=[N-])C1 67416,c1(C(=O)NCCC2(O)CCN(C(=O)CN3CCOCC3)C2)nccc2nn[nH]c12 67417,c1(NC(c2sc(Br)cc2C)c2n(CC)nnn2)ccc2c(c1)C(O)CCC2 67418,c1(C(=O)NC2(CCNC(CCc3cn(C)nc3)=O)CC2)cnc2[nH]ccc2n1 67419,C(CN=C(NCC1CC1)NC1CN(Cc2cnccn2)C1)n1cncn1 67420,C1(CCC)CN(C(C2(C3CCCN3C(=O)CCC(C)SC)CC2)=O)CCO1 67421,CC(C)C(C)C(C)CC(=O)NC1(CF)CCN(C(=O)CC2(CO)CCOCC2)C1 67422,c1(NC)cccc(C(=O)NCCCCOC)n1.N12CC(O)(C1)C(F)C2=O 67423,C(C(N=c1[nH]ccn2nnnc12)c1cnn(C)c1)OC 67424,c1(C(=O)NC2CCN(C(c3n(CC)nnc3C)=O)C2)cc(C)cc(Br)c1O 67425,c1(C(N2CC(CN(C(C(CCC)C)=O)C)OCC2)=O)cnc(O)c2ccccc12 67426,N1(C(c2c(S(=O)(=O)NC(C)=O)cc(Cl)s2)=O)CCC2(CC1)CC(=O)CCO2 67427,c1(C(CCC)C)c(C(N2CCC2CNC2=NCCS2)=O)cnn1-c1ccccc1 67428,c1(C2(C(=O)NCC(CC=C)NC(c3c(C#C)c[nH]n3)=O)CC2)cccc(Cl)c1F 67429,C1(C)(C(N(C)CC)=O)CC(SCC(C)(C)NC(=O)CCOC(C)=O)C1 67430,c1(CC(N2CC(C)C(NC(c3nc(=O)n(C)[nH]3)=O)C2)=O)ccc2sccc2c1 67431,N1(C(CSCC=C)=O)CC2=C(C1)CN(C(c1cc(C)sc1Br)=O)C2 67432,CC(CCO)C(=O)N1CCCCC1Cc1cn(-c2cccc(F)n2)nn1 67433,C1(C2(N(CC(COCC)(F)F)C)CCC2)CCCCO1 67434,N1(C(C2N(C(CN(C(=O)OC)C)=O)CCC2C)=O)CC2CCCCC12C 67435,C1(C(=O)NC2(CC(=O)NC3CCCC(C(C)C)C3)CC2)(OC)CCCCC1 67436,c1(CN2CC2=O)ccc(O)cc1.c1(C(N2C(NCC)CCC2)=O)cc(C)c(Br)s1 67437,N1(C(CSCCOC)=O)CC2CCN(C(c3ccc4nonc4c3)=O)C(C2)C1 67438,O=C(C1=NOC2(CCC2)C1)N1CC(C2CC2C(=O)NCC23CCC(CC2)CC3)C1 67439,N1(C2CN(C(C3(C(C)C)CC3)=O)C2)CCN(C(C2CCC2C(F)F)=O)CC1 67440,C(c1cncnc1O)=CC(N1C(CCNC(C(CC)SC)=O)COCC1)=O 67441,C1(CNC(=O)C2=C(Cl)CCOC2)CC(N=c2[nH]c3cccnc3s2)C1 67442,C12(C(=O)NC(C(=O)NCC(C)(C)O)CC3CCOCC3)CCC(CC1)C2 67443,CCS(=O)c1ccccc1C(=O)NCC1CC1NC(c1nccc2ccsc12)=O 67444,c1(C(N2CCC(CNC(C(c3cccc(Cl)c3)CC)=O)C2)=O)ccc(F)c(N)c1 67445,c1(CC(N2CCCC(NC(C(C)OCC)=O)C2)=O)ccc2nsnc2c1 67446,Cc1ccc(CC(=O)NCC2CCN(C(=O)CN3CCCCC3)CC2)c(F)c1F 67447,C=CCC(C)C(=O)N(CCCCN(C)C(C1(COC)CCCOC1)=O)C 67448,CCC(CC(=O)N1CCC(CCN(C(=O)CC2(O)CCCCC2)C)CC1)OC 67449,C(=O)(CC(C)(C)C(F)F)NCC1N(C(c2c(Cl)cn(CCC)n2)=O)CCN(C)C1 67450,Cc1c(C(=O)NCC2CN(C(=O)C=CC3CC3)CC2O)noc1-c1ccccc1 67451,C1(CNC(c2c(C)cco2)=O)CC2CCC(C1)N2C(=O)C(C)Oc1ccccc1 67452,c1(C(=O)NCC23CC(NC(C(C)OCC4CC4)=O)(C2)C3)ccc2nccn2c1 67453,C1(C(=O)NCC(c2ncn(C)c2)O)CCCN1NC(=O)c1cnc(Cl)s1 67454,c1(CC(=O)N(CCCCNC(C2(C)C(C)CCC2)=O)C)c[nH]c2cnc(Cl)cc12 67455,N1(C(c2c(NC)cccc2)=O)CCC2C(CCCN2C(C2(C)CCCCC2)=O)C1 67456,CC1(F)CCC(C(=O)NC2C3CN(C(=O)CC4CC=CCC4)CC23)CC1 67457,C1(C(=O)NCCN(CCC)C(c2cc(C)ccc2OC)=O)CCC2C1C2(F)F 67458,CC1CN(C(C2OCCCC2(C)C)=O)C(C)CN1C(C1CN2CCCN1CC2)=O 67459,N1(C(C(=O)NC(=O)NCC(C)C)C)CCC(C)(NC(c2sccc2Cl)=O)C1 67460,c1(NC(C(=O)N(C)CC2CCC(C(F)F)CC2)=O)ccc(F)c(Cl)c1 67461,C1(NC(C(CN(C)C)O)=O)CN(C(c2cc(F)c[nH]2)=O)CCC1CO 67462,C(=O)(C1CCCc2cc(O)ccc21)NCCCNC(C1CCN(CC(C)C)C1)=O 67463,N1(CC2C(c3n(C)nnc3)C2)CCN(C(=O)Cc2ccsc2)CC1 67464,C1(CC)CN(C(=O)CSc2nncn2C)CCC1NC(=O)Cc1cc(Cl)cs1 67465,c1(CNc2nc(-c3ccc(OCCC)nc3)sc2)ccc2[nH]c(C)cc2c1 67466,N1(C(CNC(CC)=O)=O)CCC(C(C)C)CC1CNC(=O)C=CBr 67467,C(=O)(CCCCC(C)(C)C)NC(C(=O)N(C)Cc1c(C)ccs1)Cc1ccco1 67468,C=CCC(CC)C(=O)NCC(c1ccccc1)CNC(C1(O)CC(C)(C)C1)=O 67469,C1(CC(C)NC(C23CSC(C2)C3)=O)CCN(C(=O)CN2CC(=O)NC2=O)CC1 67470,CN1CCC2CCN(C(=O)C(O)CCCNC(c3ccc(F)c(F)c3)=O)C2C1 67471,N1(C(Cn2cc(CCCC=C)nn2)=O)CCC(O)C1C(C)(C)C 67472,C(C)(C)(CC(C)(C)O)NC1C(n2cc(CS(CC)(=O)=O)nn2)CCC1 67473,C=CCCCCC(=O)NC(CC(=C)C)C(=O)NCc1cn(C)nc1C 67474,C(C(=O)N1CC(F)(F)C1C1CC1)(C(C)(C)C)n1cc(-c2c(C)nccc2)nn1 67475,Cc1c(Br)ccc(F)c1C(=O)NC(C)CCNC(=O)C(O)c1ccco1 67476,N1(C(C2=NNC(=O)C2)=O)CC(NC(=O)CC2CCC(=O)NC2)CC(F)(F)C1 67477,O=C1CNC(=O)C(CC(=O)NCCN2CCN(C(=O)CNC=O)CC2)N1 67478,C1(C)(NC(CSC)=O)CCCCC1C(=O)NCc1ccncc1C 67479,C(CC(C)C)(C(=O)NC1(CF)CCN(C(c2cscc2C(F)(F)F)=O)C1)OC 67480,C1(OC)CN2CC1N2C.C1(C(=O)NC=O)CCN(C2COC2)CC1 67481,N1(C(C2CC(F)CN2C(=O)Cc2ccc(Cl)c(F)c2)=O)CCCC2CCCCC12 67482,c1(C(N2CCC(C(=O)Nc3c(C(N)=O)ncs3)C2)=O)ccc2nc(Br)sc2c1 67483,C(=O)(C(F)C(C)(F)F)NCc1ccc(C(N(CC)CC2CCOC2)=O)s1 67484,C1(NC(=O)OC(C)(C)C)C2CC3C1C3C2NC1C(F)(F)C12CCC2 67485,C1(N(C(c2cc(CCC)[nH]n2)=O)C)CCCC(NC(=O)CN2CCCCCC2)C1 67486,C12(CC(N3CCC4(CCC4)C3)=O)CCC1CN(C(c1cccc(CO)n1)=O)C2 67487,C1(C)(C(=O)NCC2(O)CC(C)(C)C2)CCCN(C(=O)Cn2cnc(C#N)n2)C1 67488,c1(C(=O)NCC2N(C(C(c3ccncc3)C)=O)CC2)c(F)cccc1Cl 67489,C(=O)(C(F)(F)Cn1cc(CNc2ccc(-c3ccncc3)nc2)nn1)OC 67490,C(=O)(CN=c1ccc(Cl)n[nH]1)N1CC(CNC(c2ccc(C)o2)=O)CC12CCC2 67491,CCC(C)C(C(=O)NCCc1cnc(C)o1)N(C(=O)CCCC1CCC1)C 67492,C#CCC(C)(C(=O)NCCC1CC(=O)N(C)C1)NC(c1cc(C)sn1)=O 67493,c1(-c2c(C)ccc(CN3CC4CC4C3)c2)cc(C(=O)N(C)C)cc2c[nH]nc12 67494,C1(C2CCN(C(C3CCCO3)=O)C2)(NC(c2cccc(C(C)C)n2)=O)CC1 67495,C1(CNC(CCCC=C)=O)CN(C(=O)CN2CCC(=O)NC2=O)CC1(C)C 67496,c1(C(C(=O)NC(CC)(C)C)N(C2(CCO)CC2)C)cnc(C2CCCO2)s1 67497,C1(C(=O)NC2CCC(N(C)C(C3CC34CCCC4)=O)CC2)CC2CSCC(C1)C2 67498,N(C(=NCCC1CCOC1)NCc1nc(C)c(C)s1)Cc1cc(C)on1 67499,C#CC1(C(N2CC(C(C)(C)C)C2)=O)CCN(C(c2nn(C)cc2Cl)=O)C1 67500,Cc1c(Br)noc1C(N1CCC(C)C1CNC(=O)CN1CC2CC2C1)=O 67501,C(=O)(C1=CC2CCC(C1)C2)N1CC(C(=O)NC2C3CCCC23)C(F)(F)C1 67502,c1(C(=O)NCC(CNC(c2cc(CCC)nn2C)=O)(C)C)cc2occc2[nH]1 67503,N1(C(C(C)CC(N)=O)=O)CCCCCC(Nc2ncnc(C(C)(C)C)n2)C1 67504,N1(C(CCC#C)=O)CCCC(CCCCNC(C2(Cl)CC2(F)F)=O)C1 67505,c1(C(=O)OC)c(NC(=O)CC2CCCN2S(=O)(=O)CCCl)cccc1F 67506,c1(NC(C(N2CCN(C(c3cc(C)c(C)o3)=O)CC2)C)=O)ccn2nccc2n1 67507,CC(=O)C(C)(C)CC(=O)NCc1cc[nH]c1C(=O)NCC1COCCN1C 67508,c1(CN2CCC(NC(C(C)OCCC=C)=O)C2)ncc(Cl)n1C 67509,c1(N2CCCC(CNC(C)=O)C2)ccc(S(=O)(=O)N(CCCCO)C)c(Cl)c1 67510,CC(C)(C)C#CC(=O)NCC1CCCCN1C(=O)CC1CCC(=O)O1 67511,N1(C(C(CCC)N(C)C)=O)CC2CCCC1(CNC(C1CC13CC3)=O)C2 67512,N1(C(c2ccnc(Cl)c2O)=O)CC2(C1)CN(C(C13CC(O)C1C3)=O)CC2CO 67513,Nc1c(C(=O)NC2(CNC(C3CC34CCC4)=O)CCCC2)nnc2ccccc12 67514,c1(CC(=O)N(CC(CNC(C2CCN(CC)CC2)=O)C)C)c(C)nn(CC)c1C 67515,C=C(C)C(O)CC(=O)NCCC1CN(C(=O)CCCc2nc(CC)no2)CCO1 67516,c1(C(=O)NCC2CC2NC(c2cc(F)c(F)cc2Cl)=O)cc2n(n1)CCNC2=O 67517,c1(C(N2CCN(C(CCC(C)OC)=O)C(CCO)C2)=O)nc2ncccn2n1 67518,c1(NC(C2(CNc3c(C)cncn3)CC2)=O)cc(C(F)(F)F)ccc1I 67519,C(=O)(CC(CC)C(F)F)NC(CCC#C)C(=O)NC(C)Cc1ncn(C)n1 67520,C(=O)(C(F)Cc1ccccc1)N(CCNC(C1CC(CF)C1)=O)C1CC1 67521,C#CCC(CC(F)F)C(=O)NC(C(=O)NCC1=C(C)CCOC1)C(C)CC 67522,N1(C(CC2(OC)CCC2)=O)C(C(=O)Nc2sncc2C#N)CC2CC12 67523,CN(C(=NCC1C=CCCCC1)NC1CCC1)Cc1ncnn1C 67524,c1(CC(=O)NC2CC(NC(c3ccsc3)=O)CC2O)n[nH]c2ccccc12 67525,c1(C(=O)NC2CCC23CN(C(=O)CCC2CCCO2)C3)[nH]nc2ncccc12 67526,c1(CC(=O)NCCC(C)NC(c2c(F)ccc(CC)c2)=O)cnn2c1CCCC2 67527,C12(CNC(c3ccc(OC)s3)=O)CC(C1)C(NC(c1cccn(C)c1=O)=O)CO2 67528,CC1=C(C(=O)NCC(C)NC(C2(C)CNC(=O)N2)=O)SCCO1 67529,c1(N)nc(C)c(C)s1.n1(CCC)nnnc1C(C1CC1)NC1CC(CCOC)C1 67530,N(C(=NCCOCc1ccc(N(C)C)cc1)Nc1ccc(Cl)cc1)C(CSC)C 67531,Cc1cccc(C)c1C(=O)NC(C)CC1CCN(C(C2CCC2(F)F)=O)CC1 67532,Cc1ccccc1-n1cc(C(=O)NCC2CC2NC(C2CC(C)(C)CO2)=O)nn1 67533,c1(C(=O)NC(CN(C(C(CC)n2nccc2C)=O)C)C)cnc2c(C)nsc2c1 67534,Cc1cccc(N2CCC(OC(=O)Cn3cc(-c4ccc(C)cn4)nn3)C2=O)c1 67535,C(F)(c1ccccc1)=CC(=O)NCCC(C)(C)NC(C1CCC(F)(F)C1)=O 67536,c1(C(C(N2C(CN(C(c3c(CC)ocn3)=O)C)CCC2)=O)C)ccncc1C 67537,N1(C(CC(CC)O)=O)CC2CC(NC(=O)C3=CCCCCC3)CC1C2 67538,CC(C)C(F)C(=O)NCCN(C(C1CC(=C(F)F)C1)=O)C(C)C 67539,C(CN=c1cc[nH]c(C(=O)OC)n1)N1CCN(C(C2(C#C)CCCC2)=O)CC1 67540,c1(C(=O)NC(C)CCNC(=O)C(C(C)O)NC(=O)C2CC2)cnc(N)c(Cl)c1 67541,N1(c2ncnc(CC)c2F)CCC2CN(C(=O)COC3CCCC3)CC2C1 67542,C(=O)(C1=NOCC1)N(CC(=O)NC(c1nc[nH]n1)CC)CCOC 67543,c1(CCC(=O)OC(C2(CCC(=O)OC)CC2)=O)cccc(C#N)c1 67544,CCC(C#N)C(=O)NCC1CN(C(c2cccc(C(N)=O)c2)=O)C1 67545,C12(C(=O)OCC)CCCC(CN3CCC(O)(CCN4CCOCC4)CC3)(C1)OC2 67546,C(CCS(C)(=O)=O)(C(=O)NCCCN(C(c1ncccc1O)=O)C1CC1)OC 67547,C12(NC(CNC(=O)OC)=O)CCCC1CN(C(=O)C(C)CN1CCOCC1)C2 67548,Cc1ccccc1COC(C)C(=O)NC1CCCN(C(=O)Cc2cncnc2)C1 67549,C1(OC)(CNC(c2cc(C3CC3)on2)=O)CCN(C(C2CCCCS2)=O)CC1 67550,Cc1ccc(C)c(C(=O)NCC2(C)CCCN(C(C3CCC(=O)N(C)C3)=O)C2)n1 67551,C1(CNC(C(CC=C)OC)=O)COC(C)(C)CN1C(c1ncc(F)cc1F)=O 67552,Cc1cc(C(=O)NCC(CC2CC2)C(=O)NC(C)(CO)C(C)C)cc(O)n1 67553,c1(C(N(CCN(C(C2CCC(C)NC2=O)=O)C)C)=O)cccc2c1CCN2 67554,n1(CC(N2CCC(CC(N3CCC(C(=O)NC)C3)=O)C2)=O)nc(C)oc1=O 67555,c1(C(=O)NCC(CC)NC(C2(C3CCC3)CC2)=O)cc(C)c(OC(C)=O)c(Cl)c1 67556,C(=O)(CCS(=O)(=O)Cc1ccccn1)N(CCCCNC(=O)C#CC1CCC1)C 67557,Cc1cc(CCC(=O)NC(C)CCCNC(=O)CSc2nnnn2C2CC2)on1 67558,N1(C(C(F)=CC)=O)CCC(COC)(NC(C2CCCC2)=O)C1 67559,C1(CNC(c2c[nH]nc2C(F)F)=O)COC(CNC(c2ccnn2CCF)=O)C1 67560,CCCCS(=O)(=O)CC(=O)N(C1CCN(C(=O)C(CO)N(C)C)CC1)C 67561,C1(C(N(CC(C)N(C(Cc2scc(C)c2)=O)C)C)=O)C(C)(C)C1(F)F 67562,c1(COCCNC(C(CCC=C)NC(=O)OC(C)(C)C)=O)nc2ccccc2s1 67563,C(=O)(CC(C(C)OC)NC(C1CC(=O)CS1)=O)N1CCC(C#C)C1 67564,c1(N2C(CNC(c3ccc(F)cc3)=O)CC(F)C2)nc2cc(F)cc(F)c2o1 67565,N1(C(C(COC)NC(C)=O)=O)CC2CCC1CN2C(C1(C)CCC(F)(F)CC1)=O 67566,CCCC(O)C(=O)NC(C1CCN(C(=O)COCCc2ccc(Cl)s2)C1)(C)C 67567,n1(CC#C)c(C)cc(C(=O)NC2CC2CNC(c2cc(CC)no2)=O)c1C 67568,C1(NC(CS(N)(=O)=O)=O)CN(C(c2ccc(C3CCC3)cc2)=O)C2CCCCC12 67569,c1(CS(N2C(C)(C(N(C)CCc3ccccc3)=O)CC2)(=O)=O)ccc(Br)cc1F 67570,C(c1ccc(C(C(=O)NCC2CC2)N(C)Cc2nc[nH]n2)cc1)=CC(=O)OC 67571,c1(CCC(=O)NC2C(NC(C3CC(C)(C)C3)=O)C2)ccncc1Br 67572,CCC(CC)C(C)C(=O)N(CCC(=O)NCc1csc(C)c1)CCCO 67573,N1(C(C(C)SC)=O)CCCC(CCNC(c2c[nH]nc2-c2ccccn2)=O)C1 67574,C(CS(=O)(=O)CC(=O)N1CC(NC(c2cc(C)sn2)=O)CC12CCC2)OC 67575,C1(NC(C(C2CC2)SC)=O)(CO)CN(C(c2ccc(C(C)=O)o2)=O)C1 67576,c1(C(C(=O)NCC(C)C)N(C2CCSCC2)C)nnc2n1CCC2 67577,CC1CCCC(C)N1C(=O)C(N1CCC(CN(C)C(c2cc(Br)n[nH]2)=O)CC1)=O 67578,N1(C(N(c2c(OC)ccc(OC)c2)C)=O)CCCC12CCOCC2 67579,c1(CCC(N2CC(O)(C(C)NC(C(C)OCCCC)=O)C2)=O)ccnc(C)n1 67580,c1(OC(C)(C)C)cccc(Cl)c1NC(=O)C(CC(C)C)OC(=O)Nc1ccccc1 67581,C1(CNC(c2csc(C)c2C2CC2)=O)C(C)CCCN1C(c1cnns1)=O 67582,c1(CC(=O)NC2C(NC(CCCC#C)=O)CCCC2)csc2nc(C)cn12 67583,c1(N2CCCC(CCCC)C2)ccncc1S(=O)(=O)NCc1nccn1CCC 67584,CC(C(C)(C)NC(=O)CCCn1cncn1)NC(=O)COCCc1ccccc1 67585,c12nnc(n1CC1(C)CC1)CN2C.c1(CC2CCCC2)ncn(C)n1 67586,C(=O)(C1=CCC(C)(C)CC1)N1CC(C)C(CNc2ccn3ccnc3n2)C1 67587,c1(C(=O)NC2C(NC(C3(CC)COC3)=O)C2)ccc2ccn(C)c2c1 67588,N1(C(CC(=O)OCC)=O)CC(NC(=O)Cc2ccc(OC)c(F)c2)C(C2CC2)C1 67589,C1(NC(c2nc(C)oc2)=O)C2CC1N(C(c1c[nH]nc1OCC(F)(F)F)=O)C2 67590,Cn1nnc2c1CCN(C(=O)CCCCCNC(=O)C(C)(F)C(C)(C)F)C2 67591,Cc1c(C(=O)NC2CCN(c3ccnc(C4CC4)n3)CC2)ccc(F)c1F 67592,C1(C(=O)OC)C(C)CCN1C(C1CC(NC(=O)C(C)(C)N(C)C)CCO1)=O 67593,C1(C(N2CC(O)(CNC(CC3(COC)CC3)=O)C2)=O)CCc2cnn(C)c2C1 67594,c1(OCC(=O)NCC(C(C)C)NC(=O)C(O)c2cnc[nH]2)cccc(Br)c1 67595,N1(C(C)=O)CCC(C(=O)N(CC(C)NC(=O)C(c2ncc(Cl)n2C)(F)F)C)CC1 67596,N1(C(CC23C(CN(C(Cc4c(CC)con4)=O)C2)CC3)=O)CC(=O)NCC12CC2 67597,c1(C(N)=O)ccc([N+](=O)[O-])c(N(CCNc2ccc([N+](=O)[O-])o2)C2CC2)c1 67598,N1(C(C(c2cccc(Cl)c2)(C)C)=O)CC2CCN(C(C3CCCS3)=O)CCC2C1 67599,C1(NC(c2c(OC)n[nH]c2)=O)CCN(C(=O)CN2CCCC2=O)CC1O 67600,C1(C(=O)NCCc2onc(C)n2)CC(C)CN1C(=O)C(N1CCOCC1)C 67601,C1(C(=O)NCc2scc(CNC(C(C)SCC)=O)n2)CC2CCCC(C1)C2 67602,c1(-n2ccc(C(=O)NC3C(NC(=O)C=Cc4cscn4)C3)n2)ccccc1Cl 67603,c1(SCCC)cccc(C(=O)NC(C)CNC(c2oc(SC)cc2C)=O)c1 67604,C(CCCCCCC(=O)N1CC2CC(NC(=O)CCc3ccccn3)C1C2)SC 67605,c1(C(=O)NC2C3CC(NC(C(C)SCCCC)=O)CC32)cc(C)cc(C)c1N 67606,C#CCC(CC(=O)NC1CCC(NC(=O)C=CC(C)(C)C)C1)c1ccccc1 67607,C(=O)(CCCC(C)(C)C)N1C(CNC(c2cnn(CCC)c2C)=O)COCC1 67608,c1(C(N(CCNC(c2c(O)cc(C)nn2)=O)C2CC2)=O)c(C)nc2ccccn12 67609,CCCCC(O)CNC(=O)CC1CN(C(c2cccc(C3CC3)c2)=O)CC1C 67610,CC1CCCCCC1NC(c1coc(CNC(C2CC2[N+](=O)[O-])=O)n1)=O 67611,c1(NC(=O)C(N2CCCCC(CO)C2)=O)cc(N2CCCC2)cc(F)c1 67612,N1(C(CCCCCSC)=O)CC(C)N(C(C2(C)CC3(CC(O)C3)C2)=O)C(C)C1 67613,C1(C)(CNC(c2cc(-c3cn(C)nc3)no2)=O)CCC(NC(C2CC23CC3)=O)C1 67614,c1(C(=O)OCC)ccc(Cl)c(NC(c2oc(C(=O)OC)nc2C)=O)c1 67615,c1(OC)cc(OC)cc(CCNCc2cnc(C3CCCCC3)s2)c1 67616,C1(NC(C(c2cccc(Cl)c2)C)=O)CN(C(c2cc(F)n[nH]2)=O)CCC1O 67617,CC1(C(=O)O)C=CCN1C(C1COCCC1NC(C12CCC(C1)C2)=O)=O 67618,c1(C(=O)NCC(=O)NC(C2(O)CN(C(C3CC=CCC3)=O)C2)C)cnc(O)nc1O 67619,C1(C)(C(N(CC(CC)NC(=O)CCOCCN(C)C)C)=O)CC2CC2C1 67620,c1(C(=O)NCCCN(C(=O)Cc2csc(Cl)n2)C)nccc2c1NCCC2 67621,CCC(CC)(CCNC(c1cnc(COC)s1)=O)NC(=O)CC1CCCOCC1 67622,CCC(C)CCCCC(=O)N1CCC(NC(C2CCCC(C)(C)C2)=O)C(C)(C)C1 67623,N1(C(C(C(C)C)c2cccnc2)=O)CCOCC(NC(c2cccnc2)=O)C1 67624,C1(C(N2CC(c3ccccc3)(NC(CC(C)OC)=O)C2)=O)CCCCC1(C)C 67625,c1(N2CCC(CC)OCC2)nc(N2CCSC(c3cccs3)C2)c2c(n1)CCS2 67626,Cc1nc(N(C)CP(C)(C)=O)cc(N(C)Cc2cn(C)cn2)n1 67627,c1(C(N2C(C(C)(C)NC(=O)CCC3CCC3)CCC2)=O)ccc2nc[nH]c2c1F 67628,C1(N(C(CSCCCC)=O)C)CCN(C(=O)CCCc2cccs2)C1 67629,C(C(F)(F)C(C)(C)O)NC(C1(CNC(C(CN(C)C)O)=O)CC(C)(C)C1)=O 67630,CC(O)(C(=O)NCC12CC(NC(=O)CN3CCCNS3(=O)=O)(CO1)C2)C(F)(F)F 67631,CCCCCCCC(=O)NCCCC(C)NC(C1CCCC1CF)=O 67632,CCCCCC(F)C(=O)NC(C)(C)CCNC(c1cnn(CC)c1C)=O 67633,CN1CCCc2cc(CN(c3nccc(F)n3)C)ccc21 67634,N1(C(CC)=O)C2CCCC1CN(C(c1c([N+](=O)[O-])c(C(F)(F)F)nn1C)=O)CC2 67635,CC1(C)CC(C(N2CC3(CCC3O)C2)=O)CN1C(c1ccco1)=O 67636,CCC(O)C(C)(C)C(=O)NCC(CC(=O)N(CC(C)(CC)OC)C)OC 67637,n1(CC2C(C)CCCC2)ncc2cc([N+](=O)[O-])ccc2c1=O 67638,c1(C(N(C)CC2CN(C(C(C(C)O)C)=O)C2)=O)cn2cc(Cl)cnc2n1 67639,C1(CCOC)(NC(=O)CNC(C)=O)CCN(C(c2[nH]ccc(=O)c2C)=O)CC1 67640,C1(C(=O)NCCCC(C)NC(=O)CCC#N)(CO)CCCCO1 67641,Cc1ccccc1-n1cc(CN2CCC(O)CC2)cn1.N12CCC(CC1)NC2=O 67642,CC#CCC(C(=O)Nc1cnccc1OC)NC(=O)C(CC1CCC1)OC 67643,O=C(CC=C(Cl)Cl)NC1CCCC1CNC(=O)C=Cc1cc[nH]c1 67644,c1(C(N(C2CN(C(=O)CCCC#N)CC23CC3)C)=O)cc2ccsc2n1C 67645,N1(C(C(c2cncnc2)C)=O)CCC(NC(=O)C=Cc2ccco2)C12CC2 67646,N1(C(CC)=O)CCC(C)C1C(=O)N(C)Cc1ncc(Br)cn1 67647,C1(C)(C(=O)NC2(CC(N3CCC(C(C)O)C3)=O)CCC2)CCCC1O 67648,S(=O)(=O)(c1ccc(NCC(c2ccccc2F)OC)cc1Br)NCC=C 67649,c1(C(N2CCN(C(c3c(C(C)C)nns3)=O)CC2)=O)cccc(Cl)c1O 67650,C(CNC(c1c(C)noc1CC)=O)(C(C)C(C)C)NC(CCCC=C)=O 67651,C#CC1(C(=O)NC(C)Cc2ccnn2C)CCN(C(c2cscn2)=O)C1 67652,C1(CNC(C(CCOC)NC(c2cnncc2O)=O)=O)CC2CCCC2C1 67653,Cc1ccc(C#CC(=O)NCC2CCOCO2)cc1 67654,C1(NC(c2cncc(OC)c2)=O)CN(C(C2CCSC2)=O)C2CCCC12 67655,C12(NC(c3ccnc(OCC(F)F)c3)=O)CCCN(C(c3csnn3)=O)CC1C2 67656,O=C(C1=NOC2(CCOC2)C1)NC12CCC1CN(C(=O)C=CC1CCC1)C2 67657,c1(OCC(=O)NC2CN(C(C(=O)NCC)=O)C(C)C2)ccc(Br)c(F)c1F 67658,c1(CNC(CSCCC)=O)cnn2c1CN(C(c1[nH]nnc1C)=O)CC2 67659,N1(C(CCCOCCOC)=O)CC(NC(=O)C(F)(F)CO)CCC(O)C1 67660,c1(SC)nc(=NC2CC(NC(c3cncnc3)=O)C2)s[nH]1 67661,Cc1c(Cl)sc(Cl)c1C(=O)NCCCC1C=CCC1 67662,C1(CC(=O)N(C2CCN(C(c3cc(C(C)=O)c[nH]3)=O)C2)CC)CC2CCC1CC2 67663,N1(C(c2cc(OC)n[nH]2)=O)CCCC(CNC(=O)C(O)Cc2cnc[nH]2)C1 67664,C12(CC=C)CCN(C1)C(=O)CC1(CCC1)NC2=O.N1(OC)CCNC(=O)C1 67665,c1(NCC=CCNC(Cc2c(C)ncnc2C)=O)cc(=O)n(C(C)C)c(O)n1 67666,N1(C(CN(CC)CC)=O)CC(CNC(=O)CCc2ccc(SC)cc2)C2(CC2)C1 67667,N1(C(CC(C)CN(C)C)=O)C2CC1CN(C(=O)CN(C)C(C)C)C2 67668,N1(C(CCN(CC)CC)=O)CCC(CO)C(NC(=O)CC23COCC(C2)C3)C1 67669,C1(NC(C2CC(CC)C2)=O)COCCN(C(c2c(N)cccc2Cl)=O)C1 67670,CC1CCOC(C(=O)NC2CC3C(NC(=O)C(N4CCOCC4=O)C)C3C2)C1 67671,C1(NC(c2ccnc(N3CCCC3)n2)=O)CCCN(Cc2cc[nH]c2)C1 67672,C1(C(=O)NCC2CCC(C)C2)(OC)CCN(C(=O)C=NOC)C1 67673,N1(C(CC=CC)=O)CC(CNC(c2cc(CO)[nH]n2)=O)CC1(C)C 67674,C(=O)(CCCCC1CC1)NC(c1ccccc1)CNC(c1ncc(CC)s1)=O 67675,N1(C(c2c(CC)snn2)=O)CCN(C(=O)C(C)C(F)(F)F)C(CCOC)C1 67676,N1(C(CSCCC)=O)CC2(C=C(C(=O)NCP(C)(=O)OCC)CO2)C1 67677,N1(c2cc(C(=O)OCC)ncn2)CCCN(C(=O)CC(C)c2ccccc2)CC1 67678,c1(OCC(=O)N(CCCCN(C(C(CCC)O)=O)C)C)c(C)cccc1Cl 67679,c1(CCN(CC(O)CN(C(=O)C(F)C(F)(F)F)C)C)ccc(C#N)cc1 67680,C1(NC(C2N(C)CCC2)=O)CC2(CCCCN2C(=O)CCC(N)=O)C1 67681,N1(C(=O)CSCc2ncc[nH]2)CCC2(CCCN(C(=O)CC3CCOC3=O)C2)C1 67682,CCC(C)C(=O)N(CC(CNC(=O)C(C)(C)N(C)C(=O)OC(C)(C)C)OC)C 67683,C(=O)(C(C(C)(C)O)NC(=O)CC1COCC(C)O1)N(CCC)C 67684,N1(C(C2CN(C(C3CC(F)(F)C3)=O)C2)=O)CCOCC1C.c1(C)ccccc1 67685,N1(CC)C(=O)CCC1CC(=O)N(CC(O)CNC(=O)C(Cl)=CCl)C 67686,c1ccc2c(c1)nc(N1CCC(CCN3CCCC3)CC1)c1cncn21 67687,C1(CNC(C(CC=CC)C)=O)CN(C(=O)COC2(C)CCCC2)CC1(C)C 67688,N1(C(CSCCCC)=O)CCCCC(CCC(N2CCC(F)(C#N)C2)=O)C1 67689,c1(C(=O)NC2CN(C(c3c(C)snc3)=O)CC2O)cn(CCO)c(=O)nc1O 67690,c1(C(=O)NC)cccc(C(N2CCOC(C(C)(C)C(=O)OC)C2)=O)n1 67691,S(=O)(=O)(c1cc(F)c(F)c(F)c1)N1CCC(C)(C(=O)Nc2ccc(O)cc2O)C1 67692,C1(NC(Cc2n(C(C)C)cnn2)=O)CCC(C)N(C(=O)Cn2ccnn2)C1 67693,N1(C(c2cc(CC)[nH]n2)=O)CCC(NC(c2ccc(C(C)C)s2)=O)C(C(C)C)C1 67694,CC1=C(C(=O)N2C(C)CCC2(C)C)C(C)n2nnnc2N1C 67695,CCCCCCC(C)NC(=O)C(C)=CCNC(c1coc(C2CC2)n1)=O 67696,N1(C(CCOCC(C)C)=O)CCCC(CC(=O)NCc2n[nH]c3c2CCC3)CC1 67697,c1(C(N2CC3(CCCN(C(C4C(CC)C4)=O)C3)C2)=O)ccc2c(Cl)nccc2c1 67698,C(=O)(CCC(F)(F)C(F)F)NC1CN(C(c2ccn(CCC)n2)=O)CC(O)C1 67699,c1(CC(=O)NC2CCC(NC(C(CC=CC)C)=O)C2)ccc(C)c(F)c1F 67700,c1(OC)ccc(C(N2CC(O)(C3CCCN3C(=O)CC(C)OC)C2)=O)cn1 67701,C12(C(=O)NCC(C)CNC(=O)Cc3ccsn3)CCCCC(F)(C1)C2 67702,c1(C(=O)NCC2CN(C(CCCC(C)O)=O)CC2C)ccc2ccncc2n1 67703,c1(C(=O)NC2C(C)CN(c3nccc(Br)n3)C2)cc2ccccc2cc1O 67704,C12(C(N(CC(C)NC(C3C(OCC)CC3)=O)C)=O)CC3CC(C(=O)N1)C2C3 67705,C(=O)(C1CC(=O)c2ccccc21)NC(C)CNC(=O)COC1(C)CCCC1 67706,C1(NC(=O)Cn2ccnn2)C=CC(CNC(c2cc(Br)c[nH]2)=O)C1 67707,c1(OC)ccc(C(N2CC(NC(c3ccc[nH]3)=O)CC(C)C2)=O)c(F)c1 67708,C1(NC(C=CCOC)=O)CCC2CN(c3cc4nnc(C)n4cn3)CCC2C1 67709,c1(OC)cc(C(=O)NC2CCC2CNc2ncccc2C(=O)NC)ccn1 67710,C(CC(=O)Nc1cccc(Cl)c1O)(C(C)(C)C)NC(c1cnc(C)o1)=O 67711,CC(C)CC(C(=O)NC1C2CN(C(C3CCCC(C)(C)CC3)=O)CC12)C(N)=O 67712,CCC(O)(C(=O)NCCN(C(=O)CC(C)(O)c1ccccc1)C)c1ccccc1 67713,C(CC(=O)N(CC(O)C1CC1)C)N(CC(C)C)C(C)=O 67714,Cc1c(C(N2CCCC(SC)C2)C(=O)NC2CCCCC2)cccc1Cl 67715,CN(S(N)(=O)=O)CC(=O)NC(CNC(=O)Cc1ccsn1)CO 67716,c1(C(=O)NC2(CC)CN(C(c3ncccc3O)=O)C2)cccc2nc(COC)cn12 67717,N1(C(CCCCC=CC)=O)CCC(NC(=O)COc2cccnc2)C(CO)CC1 67718,N1(C(c2ccc(C(C)C)cn2)=O)CC(CNC(=O)CP(C)(C)=O)C2(CCC2)C1 67719,c1(CC(=O)NCC2C(NC(c3c(CC)csc3)=O)CCC2)ccc(OC)c(Cl)c1 67720,C1(C(=O)NC(c2nc[nH]n2)CC)CCCN1C(=O)CC1CCSC1 67721,N1(C(C2(C)CCC(=O)N2)=O)CCC2CC(NC(c3ccc(F)cc3)=O)CCC2C1 67722,C1(NC(C2CCC(F)(F)CC2)=O)CN(C(C2CC2(Cl)Cl)=O)C2(CCOCC2)C1 67723,c1(C(N2CC(N(C(=O)Cc3cccc(O)c3)C)C2)=O)ccnn(C)c1=O 67724,C1(N(C(C=CC(=O)OCC)=O)C)CCCCC1N(C)C(C1CC1F)=O 67725,c1(SC(C)C(=O)NCC(C)(O)CNC(c2ccn(C)c2)=O)ccccn1 67726,n1(CC(=O)NC(N2CCN(C(C3CCC3)=O)CC2)C)ncc2ccccc12 67727,N1(C(C2CN(C(c3cc(C(C)C)[nH]n3)=O)CC(F)C2)=O)Cc2ccccc2C1 67728,C1(C(=O)NC2CCCN(C(c3c(CC)oc(C)c3)=O)CC2)CC2(CCCC2)CO1 67729,Nc1cc(Cl)cc(F)c1C(N1CCCN(C(C2CCSC2)=O)CC1)=O 67730,CC1CN(C(c2c(Cl)ccnc2O)=O)c2cnccc2NC1=O 67731,C1(CN(C)C(C2(C)CC2(F)F)=O)COCCN1C(=O)CN1CC(=O)NC1=O 67732,C(=O)(C(C)S(N)(=O)=O)NCCCCCNC(c1c(C)nc(Br)s1)=O 67733,N1(C(Cn2ccc(C)n2)=O)CCC12CCCN(C(c1n[nH]c(C)c1C)=O)C2 67734,c1(CNN2CCC(C)(C(N(CCCCO)CC)=O)C2)ccc(C)cc1[N+](=O)[O-] 67735,c1(C(=O)OCC)cc(-c2ccccc2)n(CC(=O)NCC2CC=CCN2C)c1C 67736,CCC(C)(CNC(c1cc2n(n1)CCC2)=O)C(=O)NCc1nnn(C)n1 67737,c1(SCC)nc(C)c(C(CC)C(=O)Nc2csc(CC)n2)s1 67738,C(=O)(C(CS(=O)(=O)c1ccccc1)C(=O)NC(C(C)=O)(C)C(C)C)OC(C)(C)C 67739,C(C)(CC(=O)NC1CC(F)CN(C(=O)CSC(F)(F)F)C1)(C(F)F)N(C)C 67740,N1(C(C=C(C)C)=O)CCN(CCN2CCN(C(=O)Cc3ncoc3C)CC2)CC1 67741,N#CC1(C(N2CCC(NC(C3CCCC(C(N)=O)C3)=O)C2)=O)CCCO1 67742,N1(C(COC(C)=O)=O)CCC(O)(C2(NC(c3cnc4scnc4c3)=O)CC2)CC1 67743,CN1CCCCCC1C(=O)Nc1ccc(Oc2cccc(C#N)c2)cc1 67744,c1(NC(=O)CNC(CC2CCCC2)Cc2ccc(F)cc2)ccnc(C(=O)O)c1 67745,C#CC1(C(=O)NCC(C)S(N)(=O)=O)CCN(C(C2CC2(F)Cl)=O)C1 67746,C1(NC(C(C)(O)C2CC2)=O)CCOCC1C(N1CC(F)(F)C1C1CC1)=O 67747,C1(NC(C(C=C)O)=O)CCCC12CCN(C(=O)COCC(=O)OC(C)(C)C)CC2 67748,CC1CN(C(=O)C2=COCC2)CC1CNC(C1OCCC1c1cnn(C)c1)=O 67749,c1(C(N(CCCCNC(C2COCC(C)O2)=O)C)=O)ccnc(C(F)(F)F)c1F 67750,c1(C(=O)NCC(C)N(C)C(c2ccnc(Cn3cnnc3)c2)=O)nnn(C)c1N 67751,N1(CC(=O)NCCC(C)N(C(=O)C=Cc2cscn2)C)CCC(CO)CC1 67752,C12(NC(C(COC)N(C)C)=O)CC3CCC(C1C2)N3C(C12CCOC(C)(C1)C2)=O 67753,c1(OCC)cc(C(N2CCC(C)(NC(c3cnc(C)s3)=O)C2)=O)ccc1OC 67754,Cc1nccnc1C(=O)NC(C1CCCCC1)C(=O)NC(C)CC(F)(F)F 67755,c1(C(N2CCC(C)C(CNC(=O)CC3CCC3)C2)=O)ccc(C#N)nc1O 67756,C#Cc1cccc(C(N2CC3CC(N(C)C(c4cc(C)no4)=O)C2C3)=O)c1 67757,C1(NC(C(C2CC2)OCC)=O)CCN(C(c2ncc(C)cc2OC)=O)CC1CC 67758,c1(C(c2nnnn2CC(F)F)NCC(=C)CC)c(N(C)C)ccnc1Br 67759,N1(C(C2CC(CNC(c3ncc(C)cc3C)=O)OC2)=O)CCC(O)CC(C)C1 67760,C(CCN=C(NC1CCC1)N1CCSC(C(C)C)C1)NC(COC)=O 67761,C12(CNC(CCC(=C)Cl)=O)CCCCC1CN(C(C1CCC(CCC)CC1)=O)C2 67762,N1(C(C2CC(=C)C2)=O)CC2(CC(CNC(C3(CCOC)CC3)=O)C2)C1 67763,N1(C(Cc2cc(C)sc2)=O)CC(C)CN(C(c2ccc(N(C)C)nc2)=O)CC1C 67764,C1(N(C)Cc2ccc(Nc3ccccn3)nc2)CCC(F)(F)CC1 67765,c1(CCc2n(CCC=C)nc(-c3ccnc(Cl)c3)n2)ccc(C)c(C)c1 67766,c1(N2CCN(C(C)C)CC2)nc(N2CCC3(CCCN3C)C2)nc2c1CSC2 67767,c1(C(N2C(CC(N3CC(c4nc(C)[nH]n4)C3)=O)CC2)=O)cc(C)c(C)o1 67768,C1(CNC(Cn2ncc(CC)c2)=O)CN(C(=O)CSC(F)F)CCC1C 67769,CC1(C)C(CN2CCCC2c2ncc[nH]2)CC1O.c12ccnc(n1)N2 67770,C(=O)(CC(C)CCC=C(C)C)N1CCCCC(CNC(CNC(C)=O)=O)C1 67771,CCC(C)C(=O)C(=O)N1CC(C(=O)NC2CCN(C3CC3)C2=O)C(F)(F)C1 67772,C1(NC(C(CN(C)C)O)=O)(CO)CCCN(C(=O)CCCC2CCCC2)C1 67773,c1(N(C(CC)=O)CC)ccc(O)c(C(N2CCN(C(=O)Cc3ccco3)CC2)=O)c1 67774,C1(C(=O)NCC2N(C(c3c[nH]c(=N)s3)=O)CCC2)CCN(CCF)CC1 67775,C#CCCC(C(=O)NCCCc1ccncc1)NC(c1cnc(OC)s1)=O 67776,c1(CCC(=O)NCC2(F)CCN(C(C(C)(F)F)=O)C2)ccc(Br)c(F)c1 67777,C=CCC(CC(=O)N1CCN(C)C(CC)C1)NC(c1c[nH]nc1Cl)=O 67778,N1(C(C2CCN(C(C3(COCC)CCCC3)=O)C2)=O)CCC(CC(C)O)CC1 67779,C1(C(=O)NC2CCCCN(C(c3ccc(F)cc3Cl)=O)C2)CCN2CCOCC12 67780,C1(NC(c2ccc(=O)oc2)=O)COC2(C1)CN(C(c1c[nH]nc1[N+](=O)[O-])=O)C2 67781,N1(C(CNC=O)=O)CCN(C(CNC(=O)CC2CCC(=O)N2)C(F)F)CC1 67782,C1(N(C)C)CCCN(C(=O)C(O)C2CN(C(C3(O)CCCCC3)=O)C2)CC1 67783,CC1CCCCC1OCC(=O)N(CCCCCCN(C(=O)CC(=O)NC1CC1)C)C 67784,Cc1nnc2n1CC(C(=O)NCCCOCCNC(c1ccncn1)=O)C2 67785,C1(C(=O)Nc2ccc(OC)c(N3CCOC3=O)c2)Cc2ccc(F)cc2C1 67786,C1(NC(CCc2n(C)ccn2)=O)CCCCC1NC(=O)CCN1C(=O)CCC1=O 67787,c1(CC)nn(C)cc1C(=O)NCCN1CCC(NC(=O)CCOC2CCC2)CC1 67788,c1(C(=O)NCC(C(=O)NCC(COC)O)C)cnn2ccccc12 67789,N1(C(CC2ON=C(CC)C2)=O)CC(CNC(c2ccc(Cl)cc2)=O)C2(CCC2)C1 67790,C1(COC)(CNC(=O)C=CC(C)C)CCCN1C(=O)CCc1nnc(C(F)F)o1 67791,C1(CN(C(=O)CN2CC3C=CC2C3)C)C(C2CC2)CCN1C(=O)CC1CC(F)C1 67792,c1(C(N2C(C)CC(CNC(=O)CCc3cnn(C)n3)C2)=O)cc2ncccc2o1 67793,N1(C(CNC(C(CC)CC)=O)=O)CCC(NC(c2coc(O)n2)=O)C(C)C1 67794,c1(C(=O)NCCCN(C(CCSCC)=O)C(C)C)ccn2cc(C3CC3)nc2c1 67795,N1(C(C(CCOC)OC)=O)CCN(C)CC1C(=O)NCc1ccnc(O)c1 67796,c1(C(N2CC(OC)C(NC(C3CC(N(C)C)C3)=O)C2)=O)c(F)ccc(F)c1F 67797,C=CC(C)(CCOC)C(=O)N1CC(O)(CCNC(=O)CC(O)CCCC)C1 67798,N1(C(C(COC)CC(C)C)=O)CCCC(C)(C)C1C(N1CC2(CC(O)C2)C1)=O 67799,CCS(=O)CCNC(=O)CC1(N(C)C(c2cccn2C2CC2)=O)CC1 67800,c1(N(C2CN(C(c3cn(CC)nc3)=O)C2)C)c(F)cc([N+](=O)[O-])cc1F 67801,Cc1coc(C(=O)N(C2(C(=O)NC3CC(OC(C)C)C3)CC2)C)c1 67802,N1(C(C2N(C(C)(C)C)CC2)=O)CCC(NC(=O)CC2CCCCC2O)CC1 67803,C1(NC(C2(CS(N)(=O)=O)COC2)=O)CCC2CN(c3ccnc(CO)n3)CC2C1 67804,Cc1[nH]c(=NCCC2CC(C(=O)NC3CCC(C(C)C)NC3=O)C2)ccc1C#N 67805,N1(C(C2N(CC)CC2)=O)CCC(=CCNC(=O)CCCCN2CCOCC2)CC1 67806,N1(C(c2ncc(C)c(C)c2)=O)CC2CCC1CC2NC(c1cnsn1)=O 67807,C1(C(=O)NCC(C(=O)NC2CC(O)C2)O)Cc2nccn2C1 67808,Cn1nnc2c1CCN(c1nnnn1CC1CC13CCC3)C2 67809,C1(NC(C(F)=CC)=O)CCN(C(c2ccc(C)cc2C(C)=O)=O)CCC1CO 67810,c1(CCN(C(=O)N)CCO)ccc(F)c(Br)c1.c1(N2CCOCC2)ncc(Br)s1 67811,N1(C(COCC(C)C)=O)CCC(CN(C)C(C2CC23CCOC3)=O)CC1 67812,c1(C(=O)NC(C(C)NC(c2ccc(C(C)C)cc2)=O)CO)cc2occc2n1C 67813,C1(C(=O)NC(c2ccncn2)C)CN(C(=O)CCC2CCCOC2)C2(CCC2)C1 67814,C(C(=O)N1CC(NC(=O)C(C)(C)CNC(C)=O)C(C)C1)(C(C)C)SCC 67815,CC1(C)OCc2c1n[nH]c2C(=O)NC1CC1NC(=O)Cc1cccnc1Br 67816,CC(CCC(=O)NC1CC1)NC(C1CCCN1C=O)=O 67817,N1(C(Cn2cc[n+](C)c2)=O)CC2CC2(NC(=O)CC2CC=CCC2)C1 67818,C(=O)(C=CS(F)(F)(F)(F)F)NCCN(C(CC(CC)(C)C)=O)CC 67819,C1(NC(C2C(C)C2C)=O)CN(C(C2CCC(C(N)=O)C2)=O)C2CCCC12 67820,N(C(=NCCc1cnccn1)N)C1C(C)C1.c1(C2CCCC2)ccc(=N)[nH]c1 67821,C1(CC(N2C(CN(c3ccncn3)C)CCC2)=O)CCC2CC12 67822,N1(CC)C(C)CN(C(C2CC(O)CN2C(=O)C(c2cnn(C)c2)C)=O)CC1C 67823,C(C)(CCC(F)(F)F)NC(CC1(NC(c2n(CC)c(O)nc2)=O)CCC1)=O 67824,c1(NC(C2N(C(CCCC#C)=O)C3C(C2)C3)=O)c(C(=O)OCC)ccc(Cl)c1Cl 67825,CCN(OC)C(=O)C(C1CCCC1)NC(c1sccc1OC)=O 67826,c1(OC(C)C)ccc(C(=O)NCC2C=CCN2C(=O)C(F)C(C)C)nc1 67827,c1(NCC2N(C(N3CCC(C(N(C)CC)=O)CC3)=O)CCC2)cc(O)cc(O)c1 67828,C(=O)(C(C)(C)C(C)(F)F)N1CCCC(C)(C(=O)NCC2C(C)C2)C1 67829,Cc1[nH]nc(SC(C(N)=O)C2CCCC2)c1C(=O)O.N12CCC(CC1)NC(=O)C2 67830,c1(CS(N2CC(C)N(c3ncccn3)CC2)(=O)=O)ccc2c(c1)OCO2 67831,CCCC(CC(=O)NC1CCC(=O)N(CC)C1)NC(=O)Cc1ccco1 67832,CC1CN(C(C2CCN2C(C)(C)C)=O)CC1CNC(=O)C(c1ccccc1)O 67833,N1(C(c2ccc(N3CCCC3)cc2)=O)CCN(Cc2ccc(I)c(O)c2)C2CC12 67834,c1(C(N2CCC(N(C(=O)CCn3ccnc3C)CC)C2)=O)cc(Cl)cc(F)c1N 67835,c1(C(=O)OCC)cnc(C(=O)OC2CC(C(=O)NC3CC3)C2)n1C 67836,C(=O)(CCCCC(N)=O)NCC1CCCCN(C(Cc2c(C#N)cccc2)=O)C1 67837,C1(CNC(Cn2cc(COCC(=O)OC)nn2)=O)OCCNC(=O)C1 67838,C1(OC)CC(CNC(=O)Cc2cc(C3CC3)no2)N(C(C2CCC(F)(F)C2)=O)C1 67839,c1nnc(C)n1C.C(C(F)C(=O)NCC1CCN1C(=O)CN(C)C)N(CC)CC 67840,c1(C(N2C(CNC(COCC#C)=O)C=CC2)=O)nn(CC)cc1[N+](=O)[O-] 67841,CC1C(NC(=O)C2=COCCC2)CCCN1C(c1ncc(F)cc1N)=O 67842,N1(C(CC2(C)CC2(F)F)=O)CCCC(c2n[nH]c(CNC(=O)CSCC#N)n2)C1 67843,n1(CC(=O)NC2(COC)CCN(C(=O)CNC(C)=O)C2)ncc2cc(C)cnc12 67844,C(CC(=O)NCCCCNC(c1cc(C)ccn1)=O)(C(C)C)OCC 67845,C1(C)(NC(C(C)SCCCC)=O)CCCN(C(=O)Cn2ccc(C)cc2=O)C1 67846,N1(C(c2cnccc2Cl)=O)CCCC12CN(Cc1ccc(Cl)nc1Cl)C2 67847,C1(C(C)C)CN(C(=O)CCCn2cccc2)CCCN1C(=O)CS(C)(=O)=O 67848,c1(N(CCN(C(C)C)CC)C)ccc(S(=O)(=O)N(C(C)CC#N)CCO)c(Cl)c1 67849,c1(C(=O)NCCCN(C(c2cnc(C)n2C)=O)CC)cc(C)c2nc(C)cn2n1 67850,C1(CNC(CCCOCCOCC)=O)CN(C(C2CC2COC)=O)CCO1 67851,c1(C(=O)NCC2C(NC(CCCCOC)=O)CC2)cccc(O)c1C 67852,N1(CC(N2C(CN(C(c3cnc(C)s3)=O)CC)CCC2)=O)CCC(F)CC1 67853,C1(NC(C(CC)F)=O)CCOC12CCN(C(c1nc(C)c(C)nc1C)=O)CC2 67854,O=C(CCCC(F)(F)CO)NC1CC2CCC(C1F)N2C(C1CC2CCC2C1)=O 67855,CC(O)C(C)(C)CNC(c1cc(CNC(=O)C(O)CCN(C)C)no1)=O 67856,c1(C(N2CC(CCCCNC(=O)CCCOC3CCOCC3)C2)=O)ccnnc1Cl 67857,C1(C)(CNC(c2c(CC)noc2)=O)CCN(C(=O)CC2CC2(Cl)Cl)C1 67858,CC(C)(C)C(=O)N1CCCC1NC(=O)NC(CC(=O)O)C1CCCC1 67859,CCCCCCC(=O)N1CCCC(N(C)C(c2nccc(C(F)(F)F)n2)=O)C1 67860,c1(C(N2C(CNC(CC=C(C)C)=O)C=CC2)=O)ccc(C)c(S(C)(=O)=O)c1 67861,C1(F)(CNC(CCS(=O)(=O)NC)=O)COCCN(C(=O)CS(=O)(=O)NC)C1 67862,Cc1cc(Br)cc(Cl)c1NC(=O)NCc1nccn1C 67863,N1(C(C2C(C(=O)OCC)CC2)=O)CCC(C(=O)N(C)Cc2cccs2)C(C)(C)C1 67864,c1(C(C(=O)NC)N(C(C)CCO)C)ccc(Cl)c(C)c1 67865,c1(C(C)NCC23OCC(C(=O)OCC)(C2)C3)cc(Cl)ccc1Cl 67866,N1(C(C(C)C(F)(F)F)=O)CCCCCC(NC(c2cncc(C3CC3)c2)=O)C1 67867,N1(C(C2N(C(c3cn(C(C)C)nc3)=O)CC(O)C2)=O)CCCCC(CO)C1 67868,C(=O)(CC(C)(C)CNC(c1cccs1)=O)N1C(CO)CC(OC)C1 67869,CC1(CNC(C2CCNC2=O)=O)CCN(C(C2SCCCS2)=O)C1 67870,CCC(C)CCCCC(=O)NCCCCCN(C)C(C1(OC)CCC(C)(C)C1)=O 67871,C(=O)(C1=CCCOC1)NC1C(CC)N(C(c2cnc(CC(C)C)[nH]2)=O)CC1 67872,N1(C(c2c(CC)scc2)=O)Cc2[nH]nc(C(N3C(CC)CCC3C)=O)c2C1 67873,C1(NC(CCS(=O)(=O)NC)=O)(CNC(c2ncccc2C)=O)CC2CCC1CC2 67874,c1(OC)ccc(OC)c(CCC(=O)N2CCC2CNC(C2Cc3nccn3C2)=O)c1 67875,C12(C(=O)NCc3ccc(COC)c(F)c3)CC3CC(C1)C(=O)C(C3)C2 67876,C1(OC)CN(Cc2ccc(N3CCCC3)cc2)CCC1NC(c1ncon1)=O 67877,N1(C(c2cccc(NC(C)=O)c2C)=O)CCCC12CN(Cc1ncsc1C)C2 67878,C1(C)(OCC(=O)NCC(C)CNC(C2CCCSC2)=O)CCOCC1 67879,N1(C(CNC(CNC(C)=O)=O)=O)CC2CC1CCN2C(c1ncc[nH]c1=O)=O 67880,c1(C(=O)O)cnc(-c2cn(CCC(N3CC4(CC4)C3)=O)nn2)cn1 67881,C1(CCNC(CCCC)=O)CCCCN1C(=O)COCc1scnc1C 67882,CCC(CC)C(C(=O)N1CCC(C(=O)N(CCCSC)C)(CC)CC1)OC 67883,CC1CCN(C(C2CC(C)(C)C2)=O)CC1NC(c1ccncc1C(F)(F)F)=O 67884,c1(NC(N2CC3(CN(C)C(=O)CC3)C2)=O)cc(Cl)c2cc(Br)ccc2n1 67885,c1(C(=O)NCc2c(C)cco2)ccnc(CNC(=O)COc2ccsn2)c1 67886,c1(C(c2n(C3(C)CC3)nnn2)NCC2CCC3(CC3)C2)cccc2sccc12 67887,c1(C(N(CC(CNC(COC(c2nccn2C)C)=O)O)C)=O)ncc(Cl)s1 67888,c1(C(CNC(=O)C(N2CC(O)(C(F)(F)CO)C2)=O)=O)cc(F)ccc1F 67889,c1(C(N(C)CC2CCCCN2C(C23CCC2CC3)=O)=O)cnn(C)c1S(N)(=O)=O 67890,C1(C(=O)NC2(C)CN(C(=O)CO)C2)C2Cc3ccccc3C12 67891,c1(C(=O)NC(CC(C)NC(C2CC(=C)C2)=O)C)noc(-c2ccccc2)c1C 67892,CC(CC(=O)NC1COCC1C(=O)N(C)CC1CCCS1)N(C)C 67893,CCCC(CCC)C(=O)N(C1CCN(C(C2(CCOC)CCCC2)=O)C1)C 67894,c1(OC)ccc(CCC(N2CCC(CNC(=O)CSC)C2(C)C)=O)cc1O 67895,c1(C(N2CC3(CN(C(C(C(C)C)OC)=O)C3)C2)=O)cc2c(cc1N)CCCC2 67896,C1(NC(c2n(CC#C)ccc2)=O)CN(C(=O)CNc2cnn(C)c2)C(C)(C)C1 67897,CC(C)C(C)(O)CNC(=O)CCN(C(=O)C=Cc1cccnc1)CCO 67898,Cc1nc2c(s1)CCN(C(c1cnccc1C)C(=O)NC1CCC1)C2 67899,C1(C(=O)NC2(CCCNC(CSCC)=O)CC2)CC(C)CC(C)C1 67900,C#Cc1cn(C)nc1C(=O)NCCC1CCCN1C(c1cccc(O)c1C)=O 67901,c1(C(=O)NCCCOCCC(=O)N(CCCC)CCCO)cc(C(C)(C)C)n[nH]1 67902,n1(CC(N2CC(C)(NC(CC=C)=O)C2)=O)cc(C)c(O)nc1=O 67903,C(=O)(CCC(C)(C)[N+](=O)[O-])NC(C(=O)NCC(CC(C)O)(C)C)CCN(C)C 67904,C(=O)(CCCCC(C)C)NCC1(COC)CN(C(C2CC(CC)OCC2)=O)C1 67905,N1(C(CCCOC)=O)CCN(C(=O)CCc2nnc(S)nc2O)CC12CC2 67906,c1(C(=O)NC2CC3CN(C(CSC(C)C)=O)C2C3)cc2n(n1)CC(C)NC2=O 67907,C=CC1CCCN(C(c2ccc(CN(C(=O)CN(C)C(=O)C3CC3)CC)nc2)=O)C1 67908,CCCCC(C)(F)C(=O)NCC1CC(C(=O)NCC#Cc2cccnc2)C1 67909,N1(C(c2ccc(SC)o2)=O)CC(C(=O)NCC(c2ccccn2)N(C)C)C2(CC2)C1 67910,Cc1cc(N(C(=O)CC2(NC(c3cnc(S)nc3)=O)CC2)C)cc(C)c1 67911,c1(C(N2CC(CNC(C3(Cl)CC3)=O)C(O)C2)=O)cc(F)c(C(F)(F)F)c(F)c1 67912,C=CCC(CC)C(=O)NCCC(CCC)NC(C1CC(=O)CC(=O)N1)=O 67913,C1(N(C(=O)C(C)(N)C(=O)O)C)CC2CCCC1N2C 67914,CCCC(C)CC(=O)NCC(C)(CC)C(=O)NC1CC(O)CC1O 67915,n1(CC(=O)NCCCCNC(C2CC2F)=O)nnc(-c2ccccc2)n1 67916,CC(Cc1cnc[nH]1)C(=O)N(C1CCN(C(=O)C(F)(F)c2cscn2)C1)C 67917,c1(OC)ccc(C2CCCN(C(=O)CC(C)(C)CS(=O)(C)(C)CSC)C2)cc1F 67918,c1(CC(=O)NC2(CO)CCN(C(=O)CC3CC4CC4C3)C2)ccc2occc2c1 67919,CC1(C)OCCC1C(N1CC(OC2CCN(C(=O)COCC3CC3)CC2)C1)=O 67920,c1(C(N(CC(C)NC(C(CCC)C)=O)C)=O)cnc(CC2CC2)nc1O 67921,N1(C(c2c(CC)cccc2)=O)CCCC(C)C1CNC(=O)CC1CCS(=O)(=O)C1 67922,C1(CNC(=O)CNC(=O)C2CC2)CN(C(=O)Cc2nc[nH]n2)CCC12CCC2 67923,C1(C(=O)NCC=CCNC(COC(C)C)=O)CCCC(C2CC2)O1 67924,N1(C(C=C(C)CN2CCOCC2)=O)CCOC(C(F)F)CC1 67925,c1(COC)ccc(CN2CCCC(NC(=O)Cn3cncn3)C2)cc1 67926,C(CC(=O)NC1CCCC2(C1)N=N2)(C(F)(F)F)NC(C(CC)=CCCC)=O 67927,C(C1CCCN1C(=O)CC1CC2CC2C1)=CC(N1CC(C)(C(=O)OC)C1)=O 67928,c1(C(=O)NC2C3(CCN(C(CCC)=O)C3)CCC2)ccc2ccc(Br)cc2n1 67929,N1(C(C2(C)C(C)OCC2)=O)CCC(CNC(C2(c3ccno3)CC2)=O)C(O)C1 67930,C(CCCC(=O)N1CCOC(CCO)C1)NC(C(C=C)O)=O 67931,c1(CC(=O)NC2C(CNC(c3[nH]cc(CC)c3)=O)C2)ccnc(F)c1F 67932,C1(C(N2C(C(=O)OC)CC2)=O)CCC(NC(c2cc(C(C)=O)on2)=O)C1 67933,c1(-c2cn(CCN(C(C3C(=C)C3)=O)C)nn2)cccc(Cl)c1Cl 67934,S(=O)(=O)(c1cccs1)NCC(=O)N(C1CCCN(C(C(CC)F)=O)C1)C 67935,C1(CNC(Cc2scc(C)n2)=O)CN(C(=O)C(F)(F)C(F)F)CCC1(C)C 67936,C1(OC)COCCC1CC(=O)NCC(C)(C)CNC(c1scc(C)c1Cl)=O 67937,C1(CC(=O)N(C2(CC)CC2)C)CN(C(=O)C(CO)NC(N)=O)CC1C 67938,CC(CN(C)C)CC(=O)OC(C)(C)C(=O)NC1CC(=O)N(C(C)(C)C)C1 67939,C1(NC(c2ccc(Cl)o2)=O)C2CN(C(=O)Cc3ccccn3)CC12 67940,C(c1ccc(OC(=O)NNC(C2CC3(CC3)C(=O)O2)=O)c(OC)c1)=CC.C1CN1 67941,N1(C(CN(CCCCCC)C)=O)CC2CC1C2CNC(=O)CC(C)(C)O 67942,c1(OCC)nc(C(=O)NC2(C(=O)NC3CC(C(N)=O)C3)CC2(C)C)co1 67943,CC(C)C(CNC(c1cc(C(c2ccccc2)=O)c[nH]1)=O)NC(=O)CCC#N 67944,N1(C(C2=CC(C)(CC)C2)=O)Cc2ccccc2C(NC(C2(F)CCCC2)=O)C1 67945,CC1CN(C2CCCN(N3CC(C)CCC3C=O)C2)S(=O)(=O)C1.C(=O)O 67946,N(C)(C1CCc2c(Cl)cccc21)C(c1ccc(OC)c(F)c1)C(=O)NC(C)C 67947,C1(C(N2C(C)(CCC)CC2)=O)CCCN(C(=O)C(C)(F)c2ccon2)C1 67948,c1(C(N(CC(C)N(C)C(C2CC2CF)=O)C)=O)ccc2c(c1)C(=O)CCS2 67949,C1(C2CC2)(CNC(CC2C(C)(C)CC2)=O)CCN(C(c2ccc(Cl)cc2O)=O)C1 67950,C1(NC(c2ccn(CCCC)n2)=O)CN(C(=O)CCn2cccnc2=O)CC1O 67951,c1(C(N2CC(O)CC2C2CCCCC2)C(=O)NCCCSC)ccccc1Br 67952,N1(C(C23CC(C)(OCC2)C3)=O)CC2(CC(NC(=O)CC3=CCCCC3)CO2)C1 67953,C12(CNC(C3C(C=C)CC3)=O)CCC(CC1)N(C(C1CC3CC3C1)=O)C2 67954,C(=O)(CC1CCc2ccccc21)NC(C1(CNC(c2cc(C)c(C)o2)=O)CC1)C 67955,C1(C(=O)NCC2CCC(O)C2)CC2CC2N1C(=O)CO 67956,c1(CC(=O)NC2C(NC(C3(C(N)=O)CC3)=O)C2)ccc(Br)cc1Cl 67957,C(=O)(CC(C(F)F)C(C)(C)C)NC(CNC(c1c(N(C)C)cccn1)=O)C1CC1 67958,c1(OCC)ncccc1C(N1CCC(C)C1C(=O)NOCc1ccncc1F)=O 67959,N1(C(C=CCC)=O)CCN(C(=O)CNC(N)=O)CC1CC 67960,c1(NC2C(NC(C(C)SCC)=O)CCCC2)ncnc2cnccc12 67961,c1(NC(=O)NCC(c2ccc(C)o2)C)ccc(-c2ccccc2)nc1 67962,C1(CC=C)(NC(=O)Cc2cccc(Cl)c2)CCCN(C(c2cocc2C)=O)C1 67963,C1(CNC(C2CC(C)(C)OC2)=O)CC2CCC(C1)N2c1cnc(C(=O)ON)cn1 67964,c1(N(C)CC2CCCN2C(=O)CC2CCOCC2)ncccc1S(C)(=O)=O 67965,C1(c2n(C)nnn2)(NCCOCC2CC2)CC2COC1C2 67966,C(=O)(CC1=NNC(=O)C1)NC1CCN(CCNC(C2(C=C)CCC2)=O)CC1 67967,c1(C(=O)NCC(C(C)C)NC(C2(O)CCSC2)=O)cscc1S(C)(=O)=O 67968,C(C)(C(C)(C)C(=O)NC1C(C)(C)C1(C)C)NC(c1ccc(CC)[nH]1)=O 67969,N1(C(c2c(C)snc2)=O)CCC2CCN(C(c3cc4n(c3)CCCC4)=O)C2C1 67970,CC1Cc2cccc(C(=O)NC3(CNC(c4ccc(F)cc4)=O)CCC3)c2O1 67971,N1(C(Cc2cccc(C)n2)C)CCC(O)C(C(=O)N(C)Cc2cccc(F)c2)C1 67972,C1(NC(=O)Cc2c[nH]nc2O)C=CCN(C(C2(F)CC2c2ccccc2)=O)C1 67973,C(CN=c1[nH]c2c(c(=NC(C)CC(N)=O)[nH]1)CCC2)c1cc(OC)c(N)cc1 67974,CCC(O)CC(=O)N1CC(CF)(NC(c2cccc(C(F)F)c2)=O)C1 67975,N1(C(c2n[nH]c(C)c2C)=O)CCCC12CCCN(C(C1CCCCC1(F)F)=O)C2 67976,C1(NC(c2c(C)nc(N(C)C)s2)=O)CN(C(=O)C=CC(=O)N(C)C)CC1C1CC1 67977,C(=O)(CCC(C)(C)c1ccccc1)N(C1CCCC(O)C1)CC 67978,c1(C(=O)NC2CN(C(c3c(CC)noc3)=O)C(C)CC2)cnc(O)c([N+](=O)[O-])c1 67979,C(=O)(C1=CC(O)C(NC(C2(O)CCSC2)=O)C1)NC1CN(CC)C(=O)C1 67980,c1(C(=O)NC(CCNC(CCSC)=O)(C)C)cn(C)c(-c2ccccn2)n1 67981,CN1CC2(CN(C(=O)C(C3(O)CCC3)NC(=O)CCc3ccc[nH]3)C2)C1 67982,N=c1ccc(C(=O)NC(CNC(c2cccc(OCCF)c2)=O)C2CCC2)c[nH]1 67983,N1(C(=O)CC2CN(C(=O)CC3CC4CC4C3)CCO2)CCc2nn[nH]c2C1 67984,CCS(=O)C1CCCCC1NC(=O)C(=O)N(C1CCC1C)C 67985,N1(C(CCC#CC)=O)CCN(C(=O)C=C(C)C(C)C)CC2CCCCC12 67986,N1(C(c2cn(CC=C)nc2)=O)CCC2(CCN(C(=O)C(F)=C3CCCC3)C2)C1 67987,C1(CN(C(CC2(C=C)CC2)=O)C)CN(C(=O)CC2CCC(=O)N2CC)CCO1 67988,C(=O)(C(O)C1CN(C(c2ccoc2)=O)C1)NCC(=C)Cl 67989,c1(-n2cc(CNCc3cccc(F)c3)nn2)ccc(Br)c(Cl)c1F 67990,c1(C(C(=O)NCC(=C)CCNC(C2CC(C)(F)C2)=O)(C)C)cccc(C)c1 67991,c1(C2(NC(=O)Nc3cc(C)ncc3)CC2)cc(F)ccc1F 67992,C1(C(=O)NC2CN(C(c3ccc(-n4ccnc4)cc3)=O)C2)CC2(CCC2O)C1 67993,C(=O)(CC1=CCOCC1)NCC1C(C(=O)NCc2cccc(OC)n2)CC1 67994,N#Cc1ccc(Br)cc1CNCC12CC1CN(C(c1c(F)cc(F)cc1Cl)=O)C2 67995,c1(C(N2C3C(CNC(c4cnn[nH]4)=O)C(C3)C2)=O)cc(Cl)cc(Cl)c1OC(F)F 67996,C1(CNC(=O)CCF)CC2(C1)CN(C(c1csc(C3CCCCC3)c1)=O)C2 67997,c1(C(N2CCC(F)(C(=O)OC)CC2)=O)cnc2ncc(-c3ccc(O)cc3)cn12 67998,C(C(C(=O)NCC1(F)CC(CO)C1)NC(C1C=CCC1)=O)OC 67999,c1(-c2cn(CC3(C)CCC3)nn2)nc2ccccc2s1 68000,CC1CCC(NC(c2nc(Cl)ccc2F)=O)CN1c1ncc(F)cn1 68001,CCCCCCC(CC)(CC)C(=O)N1CCC(N(C(=O)C(F)C(F)(F)F)C)C1 68002,N1(C(C2C(NC(c3ncn(C(C)C)c3)=O)C2(C)C)=O)CC(S(N)(=O)=O)C1 68003,CC(=O)N1C(=O)C(C)(C(CC(C)C)C(=O)OCC(C)(C)C)Oc2ccccc21 68004,c1(C(N(CC(CNC(c2nc(C)sc2C)=O)C)C)=O)cc(N)cc(O)c1C 68005,C(=O)(C1=Cc2ccc(Cl)cc2OC1)N(C1CCN(C(C2CC(=O)NCC2)=O)C1)CCO 68006,c1(OC)ccc2c(c1)CC1(CCN(C(c3ccc(N)cc3Cl)=O)CC1)C2=O 68007,C(=O)(CC(O)CC(C)C)N(C)CC1(O)CCN(C(C(C=C)(C)C)=O)CC1 68008,C(=O)(Nn1cnnc1C)C1N(C(CNC(CC)=O)=O)CCCC1 68009,CCC(C)CCCCC(=O)NC1CCCC1CN(C(=O)CC1CC2CCC1C2)C 68010,C1(C(=O)NCC(C)Cn2cccn2)CC(=O)CN1C(C1OCCC1(C)C)=O 68011,N1(C(CCCOCCC)=O)CCC(CNC(=O)CCCN=[N+]=[N-])C(C)C1 68012,c1(C(=O)OCC)cn(C)nc1NC(=O)CCN(CC(C)C(C)C)C 68013,N1(C(CN(CC#C)C(C2CN3CCN2CC3)=O)=O)CC2CC(N(C)C)C(C2)C1 68014,c1(CC)cc(C(=O)NCC(C)N(C)Cc2cccc(Cl)c2F)cc(O)n1 68015,C1(C)(C(=O)NC(CC=CC(N2CCCC(CCOC)C2)=O)(C)C)CCC(=O)CC1 68016,C(=O)(CC(C(F)F)NC(=O)Cc1ccns1)NCC(C)SC 68017,Cc1ccc(-c2cc(C(=O)NCCCCC(C)NC(=O)CC(C)(C)F)on2)cc1 68018,c1(OCCC=C)cccc(CC(=O)NCC2CC2CNC(=O)CCOC)c1 68019,Cn1cncc1CC(N1CC(O)(C(C)(C)CNC(C2CC2F)=O)C1)=O 68020,c1(C(=O)NC2CN(C(C(CCC)N(C)C)=O)CC2C)cncn(C)c1=O 68021,c1(OC)cccc(CCC(N2CC=CC(NC(=O)Cc3cc(Cl)cs3)C2)=O)n1 68022,c1(C(=O)NCC(CNC(C(F)=C(C)C)=O)(C)O)c[nH]nc1[N+](=O)[O-] 68023,CCCC(C)(C)C(=O)NC1CCCC(CN(C(=O)C=Cc2ccnn2CC)C)C1 68024,c1(C(CNC(c2c(C)snc2)=O)NC(=O)CC2CC(C)(C)C2)ccc(F)cc1F 68025,Cc1cc(C(N2CCCC2c2nc(-c3ccccn3)cs2)=O)c(C)n1C(C)C 68026,CC(C)C(F)C(=O)NC12CC1CN(C(c1cnn(C)c1C(N1CCCC1)=O)=O)C2 68027,N1(C(C2C(C(=O)OC)C=C2)=O)CCN(C(=O)Cc2ccccc2F)C(COC)C1 68028,c1(CNCC2CCC(C(N)=O)O2)ccc(-c2ccccc2)nc1 68029,C1(NC(C(C(C)C)n2cnnc2)=O)CCN(C(c2n[nH]cc2Cl)=O)CC(O)C1 68030,C1(CCCNC(=O)C2CC2)(CC2C(CNC(=O)C(O)c3ccco3)C2)CCCC1 68031,C(=O)(C#Cc1ccc(Cl)cc1)N1C(C(=O)Nc2c(C)c(Cl)ccc2)CCC1 68032,c1(OC)cc(C)c(CN2CC(O)(CNC(c3cnn(C(C)C)c3)=O)C2)cc1OC 68033,C1(NC(c2coc(Br)c2)=O)CCC2CCN(C(=O)CCC3CCCC3)C12 68034,CC1=C(CNC(C2CN(CC(F)F)C2)=O)SCCO1 68035,c1(C(=O)NCC2(C)CCN(C(C3C(C#C)C3)=O)CC2)cc(C)c(F)cc1F 68036,c1(C(N2C(CNC(C(C)OCC3CC3)=O)CC2)=O)ccc(O)cc1[N+](=O)[O-] 68037,N1(C(c2cnn(CCO)c2)=O)CCN(C(c2ccc(O)nc2Cl)=O)C(CF)C1 68038,C1(C(=O)NCC(=O)OCCCC)CC(O)CN1C(c1ccn(C(F)F)n1)=O 68039,C(=O)(C(C)(C1CCC1)NC(C1CCN(C)C1)=O)NCC(C1CCC1)OCC 68040,N1(CC=C)C(=S)NC(c2csc(C3CCCCC3)n2)C(C(=O)NC2CC2)=C1C 68041,CC1CN(C(=O)CCC(F)(F)F)CC1(C)CNC(=O)CC1(C)CCC1 68042,C12(OCC)CCC(C(N3CCC(CF)(NC(=O)CSCC(N)=O)C3)=O)(CC1)C2 68043,N1(C(C=CC=CCC)=O)CC(=O)NCC1C(N1CC(O)(CCC)C1)=O 68044,N1(CC=C(C)C)CC(NC(C2CCCCC2N2CCCC2=O)=O)CCC1C 68045,c1(C(N2CCC(C(C)(C)NC(CC(C)SC)=O)CC2)=O)n[nH]c2c1CCCCC2 68046,c1(OCCOC)ccc(NC(=O)C(c2cnn(CC(C)C)c2)C)cc1 68047,C1(CN(C2(c3nnnn3CC(F)F)CCCC(C)C2)CC)C2CC3CC(C2)CC1C3 68048,c1(C(N2CCC(N(C(=O)CN3CCC3C)CC#C)CC2)=O)ccc(O)c(F)c1 68049,C12(NC(C#CCNC(Cc3c(C(=O)OC)cccc3)=O)=O)CC1COC2(C)C 68050,Cc1nn2cc(C(=O)NC3CC(C(=O)NCCC4CCC(C)O4)C3)nc2s1 68051,C1(O)(CC)CCN(C(C2C(NC(=O)Cc3cc[nH]c3)C2(C)C)=O)CC1 68052,C1(CC=C)CCN(c2cc(C)ncn2)CC1C.N12CCC(C1=O)N1CC2C1 68053,C1(C(N(CCN2CCCC2)CC)=O)CCCN(CCSc2cc(C)oc2C)C1 68054,C(CC(=O)NCCS(C)(=N)=O)(CC(C)C)NC(c1c(C)cc(C)nc1)=O 68055,C(=O)(CC(C)C(C)(C)C)N1CCC(F)(CNC(c2c(C)n(C)cn2)=O)CC1 68056,C=CCC(CC)C(=O)NCC1(NC(=O)CC2(O)CCOC2)CCOCC1 68057,c1(C(=O)NCC2(C)CCC(NC(C=C(C)C(C)C)=O)C2)ccc2cc[nH]c2n1 68058,CCC(C(=O)N(CCCN(C)C(c1cc(O)cs1)=O)C)OC1CCCC1 68059,C(=O)(C(C)(C)N(C)C)N1C(C(=O)NC(C=C)C2CCC2)CC1 68060,N1(C(C2C(C)CC2)=O)CCC(CO)(CNC(C2CC(n3ccnn3)C2)=O)CC1 68061,N1(C(COC2(C)CCC2)=O)CC(NC(=O)Cn2cc([N+](=O)[O-])cn2)C2(CC2)C1 68062,C1(CNC(C=CC(C)NC(C=CC(C)(C)SC)=O)=O)CCOC(C)C1 68063,C(=O)(C1=CC2(CCOC2)C1)N1CC2C(CNC(c3c(C)nncc3)=O)C2C1 68064,N1(Cc2c(OC(C)C)ccc(Br)c2)CC2CCN(C(c3cc[nH]c3)=O)C2C1 68065,c1(C(N2C(C)CCC(NC(c3csc(C#N)c3)=O)C2)=O)ccn2nccc2c1 68066,c1(OC)cc(OC)c(N)c(C(N2CCC(C(C)NC(c3ncccn3)=O)C2)=O)c1 68067,C1(CNC(C(c2cccc(F)c2)C)=O)CN(C(C2CC(=O)C2(C)C)=O)CCCO1 68068,Cc1cnc(C)c(C(=O)NC(CNC(C2COC2)=O)CC(C)C)c1 68069,N1(C(c2ccc(-c3csc(C)n3)s2)C(=O)NC)CCCN(C2CCC2)CC1 68070,Cc1ccncc1C(N1CCC(N(CC(N2CCC(C(=O)N(C)C)CC2)=O)C)C1)=O 68071,c1(OC)ccc2c(c1)OCC(C(=O)NC(CNC(c1ccc(C)s1)=O)CO)C2 68072,CC(C)CN=C(NCC(C)(C)C(C)(C)C)N1CCC(C)(F)C1 68073,n1(CCC(=O)N(C(C)CNC(=O)Cc2cnsc2)C)cnccc1=O 68074,c1(C(N2CCC(NC(C(C3CCC3)OCC)=O)C2CC)=O)cc(N)ccc1O 68075,CCC(C(=O)NCC1(NC(=O)CCc2cccnc2)CCC1)C(C)C 68076,C1(CNC(Cc2cc(C)sc2C)=O)N(C(=O)C(C)CC(C)C)CCC1(C)C 68077,C(=O)(CCC(C)(C)C#N)NCC=CCNC(c1nc(C)sc1)=O 68078,c1(CC)ccc(C(=O)NC(CNC(C2CC2(F)F)=O)CC)cc1[N+](=O)[O-] 68079,c1(NCc2c(NC(c3cc[nH]n3)=O)cccn2)cccc2c1oc1ccccc21 68080,C12(OC)CCN(CC1)C2=O.C1(C(C(C(C)(C)OCc2ccccc2)=O)=O)C2CC3C(C2)C13 68081,CC(C(=O)NC1CC(CNC(=O)C=Cc2cnc(C(C)(C)C)s2)C1)S(N)(=O)=O 68082,C(=O)(CCCCCOC)NC1CN(C(CC(CC)OC)=O)CC1O 68083,CC1(C(=O)NC(C2CCCCC2)CNC(C2CCCCS2)=O)CC2(CCC2)C1 68084,O=C1CCC(O)CN1Cc1cn(CC2CCN2C(C2(c3cccnc3)CC2)=O)nn1 68085,CCC(C)CC(C(=O)NCCCn1cc(C)cn1)NC(c1cnc2n1CCC2)=O 68086,C(N=c1[nH]cnc(Cl)c1Br)C1(CNC(CCCC(C)C)=O)CC12CCC2 68087,C12(NC(c3cc(Br)co3)=O)CCCN(C(c3cc4cccnc4[nH]3)=O)CC1C2 68088,N1(C(C(C)Cc2ccc(Cl)cc2Cl)=O)CCC12CN(C(c1ncccc1O)=O)C2 68089,CC(C)CC(O)CC(=O)NCC1(O)CC(CNC(c2ncn(C(C)C)n2)=O)C1 68090,C1(C(=O)NC(CNC(COC(C)(C)C)=O)C2CCC2)CC2(C1)CC21CCC1 68091,N1(C(C(C(C)C)O)=O)CC2(C1)SCCC2NC(c1ccc(-n2cncn2)nc1)=O 68092,C1(C(N(C(C)Cc2sccc2Cl)CCN(C)C)=O)(CC)CCCCC1C 68093,CCC(C(=O)N(C)CCOCCCN(C(=O)C(C1CCCCC1)OC)C)OC 68094,C1(CNC(=O)CCN2CCC2)CC(O)CN1C(=O)CCc1csnn1 68095,C1(C(=O)NC2(CNC(CC(CCCC)O)=O)CCCC2)CCCCC12OCCO2 68096,CCC(O)C(=O)N(C)CC1CCN(C(=O)CCNC(c2ccoc2)=O)C1 68097,C(=O)(C(C)C(O)CCCC)NC(C(=O)N1C(CC#C)CCCC1)CCCC=C 68098,c1(CNC(c2c(CC)n[nH]c2)=O)ccnc(C(=O)N(C(C)CN(C)C)C)c1 68099,N1(C(CCc2cnn(C)n2)=O)CCC2CCCN(C(=O)C=Cc3ccsc3)C2C1 68100,N1(C(C23CCC(NC(C)=O)(CC2)CC3)=O)CCC(C2(C(=O)O)CC2)CC1 68101,C=C(C)C1OCCC1CNC(=O)C(CCN(C)C)NC(c1cc(C)c(N)cn1)=O 68102,c1(CC(=O)NCC(c2ccccc2F)NC(CC=C=C)=O)cn(C)nc1C(F)F 68103,c1(OC)ccc(C(=O)NC(CO)C(C)NC(c2sccc2C#N)=O)nc1OC 68104,C=CCCCCCC(=O)N1CCC(c2ccccc2)C(NC(=O)C(F)=C(C)C)C1 68105,C#CCC(C)C(=O)NCC(C)(C)NC(c1cn(C2CCC2)nn1)=O 68106,c1(C(N2CC3C(C2)N3C(c2cnnc(Cl)c2)=O)=O)cc(Cl)c2cn[nH]c2c1 68107,c1(C(=O)OCC)cc([N+](=O)[O-])c(N(C)CC2CCC2OC)cc1OC 68108,C#CCC(O)C(=O)N1CC(C(=O)NCCc2ccn(C)n2)C(CC)C1 68109,c1(OC)nc(C(N2CC(CC(C)NC(=O)C=Cc3cn(C)nn3)C2)=O)cc(O)n1 68110,C1(O)(CNC(=O)CCCn2ccnc2)CCCN(C(c2cc(O)nc(O)n2)=O)C1 68111,N1(C(c2cc(C)sc2)=O)CCCC(O)(CNC(c2c[nH]cc(F)c2=O)=O)C1 68112,c1(C(N2CC(N(C(CC=C=C)=O)C)C(O)C2)=O)ccc(F)cc1CC 68113,c1(C(=O)NC2CCCC(NC(C(C)CC(N)=O)=O)C2)cc(Cl)c(F)cc1O 68114,c1(C(N2CCCC(NC(c3c(OC)oc(C)n3)=O)C2)=O)c(C)cc(C)cc1C 68115,CC1(CNC(c2cc(C#N)c[nH]2)=O)COCCN(C(=O)CN2CCCC2CO)C1 68116,c1(C(=O)NCCC2OCCN(C(C3(F)C(C)C3)=O)C2)cnc2ccnn2c1N 68117,c1(C(=O)NC(C(C)C)CNC(=O)Cc2ccccc2F)ccc2[nH]ccc2n1 68118,CC1(C)CCCCC1=CC(N1CCC(CCNC(=O)C2=COCCC2)C1)=O 68119,C1(C(N2CCCC(NC(c3c(C)nn(C)c3)=O)C2C)=O)CCC(C2CCCO2)O1 68120,C1(NC(COc2c(C(C)C)cccc2)=O)CCN(C(=O)CC2CCCO2)CC1C 68121,C1(c2nnnn2Cc2ccco2)(NCc2n(C(C)(C)C)ccn2)COCCOC1 68122,c1(C(N2C(C)(CNC(COCC)=O)CCC2)=O)ccc(=O)n(C)n1 68123,C=CCCN=C(NCC1CN(C(C)=O)C1)N1CCC(c2nncs2)C1 68124,C1(NC(Cc2scc(C)n2)=O)CC(NC(=O)Cc2ccn(C)n2)C12CCOCC2 68125,c1(C(N(C(c2ccccc2F)CNC(=O)CCC2CC2)C)=O)ccc([N+](=O)[O-])o1 68126,N1(C(CCC2(C)CC2(F)F)=O)CCC12CCNC2=O 68127,c1(CC(=O)NCC(C)(C)NC(c2ccnn2-c2ccncc2)=O)ccccc1F 68128,C1(C2CCN(C(=O)Cc3cccnc3N)C2)(NC(C(C)SC)=O)CC1 68129,C1(C)(C(=O)NC2CC(N(C)CC)C2)CCCN(C(c2cc(C3(C)CC3)on2)=O)C1 68130,Cc1ccc(CC(=O)NC(C)(CNC(C2CCC(C)O2)=O)C2CC2)c(Br)c1 68131,C1(CNC(c2cc(C(C)C)on2)=O)CC2(CC2)CN1C(=O)CC1CCC=CCC1 68132,C1(NC(Cn2c(C)nc(C)n2)=O)COC2(CCN(C(c3nnn(C)c3C)=O)C2)C1 68133,C(N=c1[nH]c(N2CCC3CC3C2)nc(=N)[nH]1)C1(SC)CC1 68134,C(=O)(C1=Cc2ccccc2C1)NC1C2(CCN(C(CCSCC)=O)C2)C1 68135,C(c1ccc(-c2ccccc2)cc1)=CC(=O)NC1CC(NC(C=CS(C)=O)=O)C1 68136,C(=O)(C1CCCc2ncccc21)N1CC=C(CNC(C2C(C)CCCC2)=O)CC1 68137,C1(NC(c2cnc(Cl)s2)=O)CCN(C(c2ocnc2C2CC2)=O)CCC1(F)F 68138,N1(C(C(CC)(C)O)=O)CC(N(C)C(c2cc(C)c(Cl)cn2)=O)C2(CC2)C1 68139,C=CCCN=C(NCc1ccc(CS(C)=O)cc1)NCC1CCCCC1 68140,N1(C(c2c[nH]c(=NC)o2)=O)CCC2(CC2C(N2CCC(C)CC2)=O)C1 68141,CC1(CNC(=O)CCCc2nc(C3CC3)no2)CCN(CCC2CCOC2)CC1 68142,c1(CC)c(C(=O)NCCC(O)CNC(=O)CCCN2C(=O)CNC2=O)cnn1C 68143,N1(C(COCCC)=O)C2CCC(C(N3CC(OC)C(OC)C3)=O)C1CC2 68144,C1(C(N2C(C(=O)OCC)CCC2)=O)CCCN(C(=O)C(C)(C)c2cccnc2)C1 68145,C(CC)(C(=O)N(CC(=O)O)CSc1cccnc1)OCC 68146,N1(C(=O)CC2CN(C(c3nc[nH]n3)=O)CCO2)CCn2nccc2C1 68147,N#Cc1ccccc1C=CC(N1CC(NC(=O)CCc2ncc[nH]2)C(O)C1)=O 68148,Cn1nc2c(c1C(N1CC(F)C(F)C1)=O)CN(Cc1c(F)cccc1Cl)CC2 68149,N1(C(C(C2CC2)OC)=O)CC(O)(C2(CNC(C3(Cl)CCC3)=O)CC2)C1 68150,C(=O)(C1=CC(C)(CC)C1)NCC(CN(C(=O)Cn1cc(C)cn1)CC)(C)C 68151,C(CCCCC(=O)N1CC(NC(=O)C=Cc2ccccn2)C(C)C1)=CC 68152,C1(O)(CN(C(C2(OC)CC2)=O)C)CCN(C(C2CCCOC2C)=O)CC1 68153,C1(CNC(CC(C=C)C)=O)CC2CCC1N(C(=O)CCc1cn(C)cn1)C2 68154,C(=O)(CCCC(F)F)N1CC2C(N(C(=O)CCN3C(=O)CCC3=O)C)C2C1 68155,C1(NC(CC2C(C)(C)N(C(c3cc(Cl)ns3)=O)CC2)=O)CCCOC12CCC2 68156,C(C)(c1cccnc1)=CC(=O)NCCN(C(=O)C(F)C(F)(F)F)CCC 68157,S(=O)(=O)(c1[nH]c(=NCc2c(C)cccc2Cl)ccc1Br)NCCOC 68158,C(=O)(CC(=O)N1CCC(N(C(=O)C(C2CCCC2)OC)CC)C1)NCC#C 68159,C(=O)(CN=c1ccc(C#N)c[nH]1)N1CCCC(N(C(C(CCC)C)=O)C)C1 68160,C(=O)(CC(F)(F)C(F)(F)F)N1C(C(C)NC(c2cncs2)=O)CCC1 68161,CCC(CC(=O)NC1CC(CNC(c2cnns2)=O)C12CCC2)CC(C)C 68162,CC(CCNC(c1cc(Br)n[nH]1)=O)CCNC(C1CCS(=O)CC1)=O 68163,CCCCC(C)CCC(=O)NCC1CCC(C(=O)NC(C2CCCC2)C)O1 68164,O=C1COC2CCN(C(c3cccc(C(F)(F)F)n3)C(=O)NC3COC3)CC2N1 68165,C1(F)(CNC(C2(C)C(C)C2)=O)CCC(NC(=O)CCc2ncc(F)cn2)C1 68166,N1(C(C(C)N(C(C)=O)C)=O)CC=CC(C(N2CCC2(C(=O)O)C(=O)O)=O)C1 68167,Cc1c(C(=O)NC(CNC(=O)C(CC(C)C)C(N)=O)C(C)C)sc2nnc(S)n12 68168,C(CC(C)C)(C(=O)NC1CCN(C(=O)CCc2c[nH]c(=N)[nH]2)C1(C)C)OC 68169,C1(CCC)(NC(c2ccc(C(F)F)o2)=O)CCCN(C(c2cccc(C)n2)=O)C1 68170,C1(NC(C2N(CC)CC2)=O)CCN(C(c2ccoc2CC(=O)NC)=O)C1CCOC 68171,c1(C(N2C3CCC2CC(N2CC4CC2CC4(F)F)C3)=O)ccc2ncccc2c1 68172,C(C(CNC(C1(CC(C)C)CCC1)=O)OC)NC(C1C(CCC)C1)=O 68173,N1(C(C(CC2CCC2)NC(c2ccco2)=O)=O)CCC(C(F)F)CC1 68174,C1(C)(C(=O)NCC(c2ccccc2F)OC)CCN(Cc2ccc[nH]2)CC1 68175,CC(C)C(CCNC(=O)C(N)=O)NC(=O)C(C(C)O)c1ccccc1 68176,CC1CN(C(C2(F)CCOCC2)=O)CCC1N=c1[nH]c(Cl)ncc1Br 68177,c1(C(N(C2CC(NC(c3cnc(=N)[nH]c3)=O)C2)C)=O)cccc(F)c1C(F)(F)F 68178,C1(NC(CCN(CC#C)C(C2CC(C)(F)C2)=O)=O)CC2(CC2)C1 68179,C1(F)(C(N2CC(CNC(C3(CC)CCC3)=O)OCC2)=O)CCC(C)CC1 68180,c1(CC(=O)N(CC(C)O)CCNC(C2CCN(C(CC)=O)C2)=O)ccccc1F 68181,CC1=C(C(=O)N(CCNC(c2cc(F)ccc2Br)=O)C2CC2)SCCO1 68182,Cc1nc2c(N3CCN(C(c4c(F)cncc4F)=O)C4CC34)ncnc2[nH]1 68183,N(C1CCc2ccccc21)C(CCCCNC(CC=C)=O)=O 68184,c1(C(N2CCC(OCC(N3C(C)CC3CO)=O)C2)=O)cc(C#N)n(C)n1 68185,c1(C(N2C(CC(C)C)CCC2)=O)cccc(S(=O)(=O)NCc2cc(O)no2)c1 68186,c1(C(=O)OCC)nc(C(N2CCC(C(C)NC(=O)CC3CCC3)C2)=O)cs1 68187,c1(CNC(=NC)NC2CCCN(c3ccccn3)C2)nn(C)nc1C 68188,c1(OC)ccc2ncnc(N3CCNC(C(N4CC5C(C4)C5(C)C)=O)C3)c2n1 68189,N1(C(C)=O)CCN(C(=O)C(O)C2CN(C(c3c(C)csc3C)=O)C2)CC1 68190,Cc1ccc(C#N)c(NC(C2CC(NCc3cncs3)C2)=O)c1 68191,N1(C(C(=O)Nc2ccc(F)cc2)c2csnn2)CCc2ccc(Cl)nc2C1 68192,c1(OC)c(C)csc1C(N1CC(F)CC1CN(C)C(c1cnc(C)[nH]1)=O)=O 68193,c1(C(=O)NC(CC2CN(c3snc(CCOC)n3)C2)C)ncc(F)cc1F 68194,c1(N(C(=O)CC2(C(=O)O)CC2)CCOC)ccc(C#N)c([N+](=O)[O-])c1 68195,C1(NC(C(C=C)(C)O)=O)CCC2(CC1)CN(C(c1cccc(C(=O)OC)c1)=O)C2 68196,C1(CNC(CSCC(C)C)=O)CCC(C)N(C(c2ccc(C(F)F)nc2)=O)C1 68197,CCC(C(=O)OC)C(=O)NC(C)(C)CN(C(=O)C(COC)OC)C 68198,c1(C(N2C(CNC(CCOC(C)=O)=O)CCCC2)=O)ccc(C(F)(F)F)c(F)c1C 68199,C(=O)(CC(C(F)(F)F)c1ccccc1)NCC(C)NC(=O)Cc1cnc[nH]1 68200,C12(C(=O)NCCNC(CCc3nc(=N)[nH][nH]3)=O)CC3CC1(CO)CC3C2 68201,c1(C(=O)NC2CCC2CNC(c2cc(SC(F)(F)F)c[nH]2)=O)ncc(F)cn1 68202,N1(C(C(C=C)c2ccccc2)=O)CCC2CCN(C(C3(C)CC(C)C3)=O)CC12 68203,C12(C(N(CCNC(=O)CCSCC(C)C)CC)=O)CC(C)C1C2 68204,c12cnc(F)cc1C(=O)NC1CCN(CC1O)C(=O)N2.c1(OC)ccccn1 68205,C1(C(=O)NC(CC=C)C2CC2)CN(C(C2CCC(N(C)C)C2)=O)CC1F 68206,C1(O)(C(C(=O)NC2C(O)CC2O)NC(CC)=O)CCCCC1 68207,C(=O)(CCCCCC(C)(C)C)N1CC(N(C)C(c2nccc3occc23)=O)C1 68208,CC(CCCNC(c1csc(O)n1)=O)NC(c1csc(O)n1)=O 68209,c1(C(=O)NCCC(=C)CNC(=O)CC2CCCOC2)ccccc1SC 68210,C1(C(=O)NCC2CC(C)N(C(c3coc(CO)c3)=O)C2)(OC)CCC(F)(F)CC1 68211,C(CCC(C)CC(=O)NC1CN(C(=O)Cc2cnn(C)c2C)C1)=C(C)C 68212,N1(C(C=CCCC)=O)CCC2(CCCC2NC(c2cnc(N(C)C)o2)=O)C1 68213,c1(C(=O)NCC2C(C)CN(C(=O)CCSCC(N)=O)C2)nn(C)c2ccccc12 68214,C1(C(=O)NC2C(CNC(=O)CC3(O)CCC3)CC2)(NC(N)=O)CCCCC1 68215,C(=O)(C1c2c[nH]nc2CCC1C)NC1C(S(CC)=O)CCC1 68216,CN1CC(NCc2cccc([Si](C)(C)C)c2)Cc2ccccc21 68217,C(=O)(C(O)CNC(C1CC1(C)C(F)F)=O)N(C(C)CO)C1CC1 68218,n1(C(CC)C)nc(C(=O)NC(C)CNC(=O)C=Cc2csc(C)n2)cc1C 68219,C(=O)(C(F)C(C)CNC(=O)C(C)(C)C(F)F)NCCc1c(C)ncs1 68220,c1(CNC(C(=O)NCc2cncc(OC)c2)=O)csc2ccc(Br)cc12 68221,c1(NCc2cccc(C(=O)Nc3ccccc3CCO)c2)nc(Cl)c(Br)cc1O 68222,c1(N(C2CCCN(C(CCC(C)SC)=O)C2)C)snc(C)c1C#N 68223,C1(N(C)C)CN(C(c2cocc2Br)C(=O)NC2CCOCC2)CC12CC2 68224,c1(C(=O)NC2C(F)CCN(C(C=Cc3c(C)ncs3)=O)C2)ccc2c(c1)CCC2 68225,c1(NC(C2(O)CCN(C(=O)CCc3cc(F)ccn3)C2)=O)cccc2[nH]ccc12 68226,Cc1c(C(=O)NCC(C(=O)Nc2ccccc2CO)N(C)C)cccc1O 68227,C(N=c1[nH]c(=NC2CCCCCCC2)c2ncccc2[nH]1)c1c(C)ccc(C)c1 68228,c1(C(N(C(C)C(=O)NCC(C)C2CCC2)CCC)=O)ncc2ccccn12 68229,C1(NC(c2c(C)onc2)=O)(CNC(C2(C)CCCO2)=O)CC2CCC1CC2 68230,C1(CC(=O)NC)CN(C(=O)Cn2cncn2)CCN1C(=O)C(C)c1ccon1 68231,C1(C(=O)NCC(n2cccn2)C)CCOCCN1C(c1ccc(C#N)o1)=O 68232,c1(C(=O)NCC2C(NC(C3(C)C=CCCC3)=O)CCC2)cc(F)c(F)c(O)c1F 68233,c1(C(=O)NCCN(C(C2CCC(=O)NC2)=O)CC)coc2ccccc12 68234,C=Cc1cc(C(=O)NCC2(C)CCN(C(c3ccnc(OC)c3)=O)C2)cc(F)c1 68235,c1(COC)nn(C)c(Cl)c1C(N1CCCC1CNC(C1CC(C)(C)C1)=O)=O 68236,Cc1ccc(C=CC(=O)NCC(C2CC2)NC(=O)C(n2nccc2C)C)cc1Cl 68237,C1(CC(=O)NCC(CC)C(C)C)CCN(C(=O)CCC2CCC(=O)C2)C1(C)C 68238,c1(OC)cc(C(N2CCCCC2C2CCCC2O)=O)cc2cccnc12 68239,N1(C(CSC)=O)Cc2ccccc2C(CNC(c2cnc(NC(C)=O)o2)=O)C1 68240,C1(CNC(C=C(C)C(C)(C)C)=O)CC2CN(C(C3(C#N)CC4CC4C3)=O)CC12 68241,CCC(CC(=O)NCCC(=O)NC(C)(C)CC(C)C)CC(C)C 68242,N1(C(=O)Cn2cnc(Br)c2)CCC2CCCC(C1)N2C(C1C2COCC12)=O 68243,C1(C(=O)NC(C)C(C)(C)NC(=O)C=CCN2CCCC2)CS(=O)(=O)CCO1 68244,C1(NC(c2cn(C)c(=O)nc2O)=O)CC(C2CCN(C(=O)CC3CC3)C2)C1 68245,CC(C)(O)C(F)C(=O)N1CCOC(c2cn(Cc3cncc(N)c3)nn2)C1 68246,N12CCC(C3CCN(C3)C1=O)C2.c1(-c2ccn(CCOC)n2)cc(C)ccc1C 68247,CC1(C)CN(C(c2ccon2)=O)CC1NC(c1cc(-c2ccco2)cs1)=O 68248,CCCCS(=O)(=O)NC(N(C)CCCc1cn(-c2ccccc2Cl)nn1)=O 68249,N1(C(C(C)C2CC2)=O)CC2(CCC2NC(=O)Cc2nn(C)cc2Br)C1 68250,C1(NC(C(CSC)(C)C)=O)CCCN(C(c2cc3sccc3s2)=O)CC1 68251,CN1CCC(c2nnnn2CCCOC2CC2)(NCCCC(O)C(F)(F)F)CC1 68252,C1(C2CCN(C)CC2)(C(N(CCC(C(C)(C)C)NC(CCCSC)=O)C)=O)CC1 68253,CC1CCCC(OCCNC(=O)NCc2ccsc2)C1 68254,CC1(NC(C2COC(=O)C2)=O)CCCN(C(c2cc3occc3[nH]2)=O)C1 68255,c1(CC(=O)NCCNC(CCCOCCOC)=O)ccc(OC(F)F)c(F)c1 68256,c1(NC(=O)CC2CCN(C(c3cn(COC)nn3)=O)C2)nc(Cl)sc1Cl 68257,c1(NC(C2N(Cc3ccc(OCC#C)cc3)CC(F)C2)=O)nc(Cl)cnc1Cl 68258,N1(C(c2n[nH]cc2C(F)(F)F)=O)CC(N=c2[nH]nc(CO)s2)C2(CCC2)C1 68259,N1(C(C)=O)CCCC(O)(CC(N2CC(O)(CNC(c3cc(OC)ns3)=O)C2)=O)C1 68260,CCC(CC)CC(=O)NCC1CN(C)CCN1C(=O)CCOc1ccc(Cl)cc1 68261,n1(COC)nccc1C(N1CCC(OCC(=O)NC(C)Cc2ccnn2C)C1)=O 68262,N1(C(CC(C)(C)C)=O)CC2(CCC2)CC1CNC(c1ccnc2c1CCC2)=O 68263,C(=O)(CC(=O)NCC1CC(NC(c2c[nH]nc2C(C)(F)F)=O)C1)N(C)C 68264,N1(C(C)=O)CCN(C(=O)CCCn2cc(CCOC(C)=O)nn2)CC1 68265,Cc1nn(C)c(C)c1C(N1CC(NC(=O)CCN2CCCS2(=O)=O)CC(O)C1)=O 68266,N=c1[nH]cc(C(=O)NCC(O)CNC(c2csc([N+](=O)[O-])c2)=O)c2cc[nH]c12 68267,C1(C(NOCC(O)C(C)C)=O)CCC(O)CN1C(c1c(C(NOCC)=O)cnnc1)=O 68268,N1(CC(N2CCN(C)CC2)C)CC2(CCC1CO)CC2 68269,c1(C(=O)NC2CCCN(C(C(CC)NC(C)=O)=O)CC2)cc(=O)c(OC)cn1C 68270,c1(NCC)snc(C)c1C(=O)NCCCNC(=O)C(CC1CC1)OC 68271,c1(C(N(CCN(C(CCC2CC(OC)C2)=O)C)C)=O)ccc(N)c2ccncc12 68272,C1(C2(O)CCOCC2)(CNC(N2C(CC)C(O)CC2)=O)CC1 68273,c1(OCC)cccc(C=CC(=O)N(CCCNC(=O)Cc2c(C)noc2C)C)c1 68274,c1(C(=O)NC)cccc(CCNC(=O)NC2CCC2C(C)(C)C)c1 68275,Cc1cnc(NC2CCCCC2CNC(c2cc[nH]n2)=O)nc1C 68276,N1(C(CC=C(C)C)=O)CCC(NC(c2cc(C(F)(F)F)ccc2N)=O)CC1C 68277,C(=O)(C(C)(CC)CO)NCC(CC=C)NC(c1ncc(C(F)(F)F)cc1Cl)=O 68278,C(=O)(C(O)C(C)(C)C)N1CC(C)C(NC(=O)Cc2ccncc2Cl)C1 68279,C#CCC(C)(CC)C(=O)N1CCCC(CC(N2CCc3sccc3C2)=O)C1 68280,C(c1ccc2occc2c1)=CC(=O)NCC1C(NC(C(C(C)O)C)=O)CCC1 68281,C(=O)(CC(C)CC(F)(F)F)N1C(CCNC(C(=C(C)C2CC2)F)=O)CCC1 68282,CCC(CC)(CCN)NCc1ccc(C(F)F)c(F)c1 68283,C1(C(=O)OCC)COCC1C(=O)NCCCCNC(=O)CC1(N(C)C)CCC1 68284,c1(NC(C(=O)NCCN(C(CC)C)C)=O)ccc2c(c1)C(=O)OC2(C)C 68285,C(CNC(=O)CCc1cnn(C)n1)(CCOC)NC(C(C)NC(CC)=O)=O 68286,c1(C(N2CCC(C(=O)OCC)CC2)=O)ccc(F)c(-c2c(C)cccc2F)n1 68287,C(=O)(C1=CCCSC1)NC(C(C)C)CNC(=O)COC1CCCOC1 68288,C1(NC(C(CC)C)=O)CN(C(C2(Cc3ccccc3)COC2)=O)CC1(C)C 68289,c1(NCCCCN(C(C2CCOC2)CO)C(C)=O)cc(C)nn1C 68290,N(C(=NCC1CCOc2ccccc21)NC1CCN(C(C)=O)CC1)C(C=C)C 68291,Cc1cc(C)n2nc(C(C)NCCOc3cccc(Br)c3)nc2n1 68292,c1(SCC)ccc(Cl)cc1C(=O)N(CC(CC)NC(=O)C(F)CC1CCC1)C 68293,C12(NC(C(COC)COC)=O)CCC(F)(F)CC1CN(C(=O)C(F)C(C)(C)O)C2 68294,c1(C(=O)NC2CC(NC(c3nc(C)sc3C)=O)C2)ccc2nn[nH]c2c1O 68295,c1(C(=O)NC2C(NC(c3c(C(C)=O)cccc3)=O)CC2)cc(Br)cn2ncnc12 68296,C1(NC(C(C)C)=O)CCN(C(c2csc(C(C)(C)C)c2)=O)CC1CO 68297,C#CCCCCCC(=O)NCC1(F)CN(C(c2c(C)csc2C)=O)C1 68298,C12(CNC(C3N(C)CCC3)=O)CCCC(CN(C(=O)CC3CCC3)C1)C2 68299,O=S(=O)(c1cccc(-n2cnnn2)c1)NCC1=NOC2CCCC12 68300,c1(CNC(CCn2c(=O)sc(C)c2C)=O)c(F)ccc2c1OCO2 68301,C12(CNC(C=CCOC)=O)CC1CN(C(C1CC(C)CCO1)=O)C2 68302,C(=O)(CCCCCOC)NCC1C(C(N2CCC(=C)C2)=O)C1 68303,c1(C(=O)NC(C(C)C)CCN(C)C(c2cn[nH]c2)=O)cc(=O)c2ccccc2[nH]1 68304,C1(NC(C(C2CC2)OC)=O)COCC1NC(c1ccoc1I)=O 68305,CC(Cc1ccccc1)(C(F)F)NC(=O)OCC(F)(F)F 68306,c1(C(=O)NC(C2(O)CN(C(CC(C=C)C)=O)C2)C)n[nH]c2c1CS(=O)(=O)CC2 68307,c1(C(N2CCCC(CNC(CCC3CC(C)C3)=O)C2)=O)cn(C)c(=O)n(C)c1=O 68308,N1(C(C=C2CCC(C)CC2)=O)CCC(O)(C(C)NC(=O)CC(C)(F)F)CC1 68309,c1(CC)cc(C(c2nnnn2C2COC2)NC(C)CCC(C)C)ccc1C#N 68310,C#CC1CCC(C(N2CCN(C(c3cn(C)nc3Br)=O)C(CC)C2)=O)CC1 68311,CC(C)(C)C(CNC(c1ccn(C(F)F)n1)=O)C(=O)NC(C1CCC1)C1CC1 68312,C1(C(N(C)CC2CC2)=O)CN(Cc2cncn2C2CCCC2)CCC1O 68313,c1(C(=O)NCC=CCNC(=O)CC2(O)CCOCC2)cnn2c(=O)cc[nH]c12 68314,C1(CNC(C2(C)CC(C)C2)=O)CC2(CCN(C(c3cc(C(N)=O)no3)=O)C2)CO1 68315,Cc1[nH]c(C)c(C(=O)NCC2=CCN(C(=O)C(C)Cc3cnc[nH]3)CC2)c1C 68316,C1(CNC(CS(=O)(=O)NC)=O)CCC2(CCC2)CN1C(c1cncn(C)c1=O)=O 68317,C1(CCNC(CCOCCCOC)=O)CN(C(=O)CC2CS(=O)(=O)C2)CCO1 68318,c1(OC)cc(C(=O)NC2CC(C)CN(C(=O)OC(C)(C)C)C2)ccc1C 68319,N1(C(C(CCOC)OC)=O)Cc2ccccc2CC1CNC(=O)CC1CCOC1 68320,c1(CCC(=O)NCCC(Cn2cc(C=CC(C)C)nn2)F)ccc(C#N)cc1F 68321,Cc1nocc1CCC(=O)NC1CC(CNC(c2csnc2Br)=O)C1 68322,C1(C(=O)NCCc2ccc(O)cn2)CCc2nnc(-c3ccccc3)n2C1 68323,c1(CC)oc(C(=O)NCC2CN(C(=O)C(CC3CC3)CC3CC3)CC2C)cc1C 68324,C1(COC)(CNC(=O)CCc2cc(C)no2)CCCN1C(C1CCCC1)=O 68325,c1(CCC(=O)NCC(CNC(c2cc(CC)on2)=O)(C)O)c(C)n[nH]c1C 68326,C1(CC(=O)NC(CC2CCCO2)CO)CC2(C1)CN(C(=O)CCc1cccs1)C2 68327,N1(C(c2c(C)nncc2)=O)CCN(C(c2ocnc2C)=O)CC(O)C1 68328,c1(N(C)C)nccc2c1CCN(Cc1ncsc1Br)C2 68329,C(C)(C)(CCCNC(=O)CCC1CCC(C)O1)NC(c1c(CC)ncs1)=O 68330,C1(CCNC(C(C=CCCC)O)=O)CCCN(C(=O)CNC(=O)CCC(C)C)C1 68331,N1(C(C(C=C)(C)O)=O)CC(NC(C2CC3(CCOCC3)C2)=O)CC2(CCC2)C1 68332,C1(NC(C=C(C)C(C)C)=O)CCN(C(C23CC(C)(CCO2)C3)=O)CC1CO 68333,Cc1cc(C(c2ccco2)NCc2cn(C3CCOC3)nn2)on1 68334,c1(N2C(CC(=O)Nc3cc(CCC)no3)COCC2)ncc2cccc(Br)c2n1 68335,C1(C)(C(=O)OC)CC12CCN(C(c1ccc(Nc3cn[nH]c3)cc1Cl)=O)CC2 68336,c1(C(N(C(CNC(C(C)CC2CCC2)=O)C)C)=O)c[nH]c2nccc-2c1 68337,C1(CNC(c2ccn(CC)n2)=O)CC(NC(=O)C(O)Cc2cnn(C)c2)C(O)C1 68338,N1(C(CCOCC)=O)CCN(C(C23CC(C2)S(=O)(=O)C3)=O)CC1C 68339,c1(C(=O)NC(C2CN(C(=O)C3=NNC(=O)CC3)C2)C)cc(F)c2cn[nH]c2c1 68340,Cc1nc(CC(=O)NC2(C(=O)N(C)C(C)C3CC3)CSC2)cs1 68341,N1(C(C2(CC(C)C)CCNC2)=O)CCC(C#N)(NC(N)=O)C1 68342,c1(C(N2C(CNC(CC3N(C(C)C)CCC3)=O)CCCC2)=O)cc(N)nc(Cl)c1 68343,N1(C(CNC(CCC(C)C)=O)=O)CCC(C(=O)N(C)Cc2ccsc2)C(C)(C)C1 68344,CC1(CNC(=O)CC2CCCNC(=O)C2)CCCN(C(c2nccs2)=O)C1 68345,c1(CC)cnc(OC)c(C(=O)NCC(CNC(=O)COC2CCCOC2)OC)c1 68346,C(=O)(C1=C(Cl)CCCC1)NCC1(O)CCN(C(C(C)c2ccon2)=O)CC1 68347,CCC(CC)C(C)C(=O)NCC(C)(CC)NC(=O)CSc1nncn1C(C)(C)C 68348,c1(CNC(C(COCC)n2cc(C3CC3)nn2)=O)ccc(-c2cn(CC)nn2)cc1 68349,N1(C(c2scc(C)c2Cl)=O)CCC(CCNC(C2C(C)C2C)=O)C(F)(F)C1 68350,c1(C(N2CC(c3cn(C4(C(=O)OC)CC4)nn3)(C)C2)=O)ccnnc1C 68351,C(=O)(C1CCc2ccccc21)NCc1c(C(=O)NC2(C(C)(F)F)CCC2)con1 68352,N1(C(c2cnc(CC(C)C)s2)=O)CC2CC(NC(=O)CC3=NNC(=O)C3)CC1C2 68353,CCCC(C)(CC)C(=O)N1CCCCCC(NC(C2(O)CCC2)=O)C1 68354,O=C(C1=COCC1)NCC1CN(C(=O)Cc2cccc(OC3CC3)c2)CCO1 68355,C1(CC(=O)N(CC(C)NC(=O)C(c2ccccc2)C)C)(CC)CCOCC1 68356,C1(OC)CCC(C(=O)NC2(CNC(=O)CCc3ccc(C)cc3)CCOC2)CC1 68357,C12(C(=O)NCC3C4CN(C(C(C)(C)N(C)C)=O)CC43)CCC(C)(C(=O)O1)C2(C)C 68358,Cc1nc(N2CCC3(CC3C(=O)NC(C)(CO)CO)C2)c2sccc2n1 68359,c1(C(=O)OC)cccnc1C(=O)N(C)CCOCCN(C(=O)C(F)C1CCC1)C 68360,CC1CC(NC(=O)CC2CCC(=O)N2C)CCN1Cc1cncs1 68361,C1(C(N2CCC(C)(NC(c3nc(C(C)C)oc3)=O)C2)=O)CC12CC(F)(F)C2 68362,N1(NCc2cc(C)n(-c3cccc(C(N)=O)c3)c2C)C(C(=O)O)CC2OCCC12 68363,C1(NC(c2ccc(N(C)C)nc2)=O)CN(C(C2CC2C(F)(F)F)=O)CC1C1CC1 68364,C(=O)(C(O)CCC(F)(F)F)NC(C1CCCC1)CNC(CC(COC)(C)C)=O 68365,c1(C(N2CC(NC(Cc3c(C)cccn3)=O)C(C)C2)=O)c(C)nc2cccnn12 68366,C1(CNC(CC=CC)=O)C2CN(C(=O)Cc3cncc(F)c3)CC12 68367,N1(C(=O)COc2ccsc2Cl)CCC(O)C(O)c2ccccc21 68368,c1(C(=O)Nc2ccc(C(N3CC(CN(C(C)=O)C)C3)=O)s2)c(F)cccc1Br 68369,Cc1ccc(C=CC(N2CCCN(C(=O)C(C)C3CC3)C(C)C2)=O)cc1Cl 68370,C1(NC(C)=O)CCCN(C(C2(O)CN(C(c3cnncc3N(C)C)=O)C2)=O)C1 68371,CCCCC(CC)CC(=O)N1CC(F)CC1CN(C(=O)CC(C)(C)C(F)F)C 68372,C1(NC(C2C(C)CN(C(c3cnc(O)o3)=O)C2)=O)CCN(C)CC1C#N 68373,C(CC(C(=O)NCCCOCCNC(=O)C=Cc1ccoc1)NC=O)SC 68374,C(=O)(CC1=NNC(=O)C1)N1CC(NC(c2n(C)nnc2)=O)C(C(F)F)C1 68375,O=C(C#CC1CCOC1)NCC1CCN(C(=O)CCOC2CCCC2)CC1O 68376,C=CC1(CC(=O)N(CC(=O)NC)C(C)C)CN(C(=O)CC(CC)SC)C1 68377,C(CC(=O)NCC(C)(C)N1CCCC1)(C(F)F)NC(C(COC(C)C)(C)C)=O 68378,C1(c2n(CC(=C)C)nnn2)(NCc2ccccc2-n2cncn2)CC(C)N(C)C1 68379,c1(C(=O)NCC(C(=O)NCC(COCC)C)O)ccc2[nH]ccc2c1 68380,Cc1cscc1C(=O)NC(C(=O)NCCc1cn(C)nn1)C1CCCO1 68381,c1(NC(C(C2CCC2)NC(c2c(CC)cco2)=O)=O)ccc(O)c(OC)c1 68382,C1(C(=O)NCCN2CCC(C)CC2)CN(C(c2cn(C)nn2)=O)C(C)(C)C1 68383,c1(NC(=O)NCC2(NC(C3CN(S(C)(=O)=O)C3)=O)CCOC2)c(C)ncn1O 68384,C(=O)(C(C(=O)NCC12CC1CN(C(C1CCC1COC)=O)C2)C(C)C)OCC 68385,c1(C(=O)NCC2(C)CCN(C(C(C(C)C)NS(N)(=O)=O)=O)C2)cccc(=O)n1O 68386,C1(CC)COCCN(C(C2CCCN(C(c3cnn(CC)c3C)=O)C2)=O)C1 68387,c1(C(=O)NC2CCCCN(C(C(C(C)C)(C)C)=O)C2)cc2c(nc1N)CCC2 68388,c1(C(=O)NCC(C)NC(c2cccc(C(F)(F)F)n2)=O)cnccc1C(C)(C)C 68389,N1(C(C)C)CC(C(N2CC=CC(NC(=O)C(=O)NCC(F)(F)F)C2)=O)CC1=O 68390,C1(C(=O)NCc2c(C(=O)NCC(C3CC3)SC)con2)CCC(C)=C(C)C1 68391,C1(C(COC(n2cccc2N(C)C)=O)=O)CCCN(C(=O)C(C)(C)C)C1 68392,C(C(O)C(=O)NC1CC(F)(CNC(c2csnn2)=O)C1)SC 68393,C1(NC(C2(COC)CN(C(=O)CC(O)C3CCCC3)C2)=O)CC12CCCCC2 68394,C(=O)(C(C)(C)CS(N)(=O)=O)NCC1(F)CC(NC(CC(=O)NCC#C)=O)C1 68395,C(=O)(CC1=CCN(C(C2OCCC2(C)C)=O)CC1)N(C(CSC)C)C 68396,Cc1cccc2nc(C(=O)NCC(O)CNC(C34CCCCC3C4)=O)cn12 68397,C1(F)(CNC(C2C(OCC)C2)=O)CC(CNC(C2(O)CC2)=O)C1 68398,c1(OCC(=O)N(C2CCN(C(CC(=C=C)C)=O)CC2)CCO)cc(F)cc(F)c1 68399,c1(CC)ncc(C(N2CCC(CC(N3CCNC(=O)C3CC)=O)C2)=O)c(C)n1 68400,CC1CCN(CCNC(=O)Nc2cc(-c3cccc(C(F)(F)F)c3)nn2C)CC1C 68401,c1(CC)nn(C)c(C(=O)NC2CCN(C(=O)C(C)(C)C)C2)c1Cl 68402,N1(C(=O)OC)CCN(C(C2CCCN2C(=O)C=Cc2ccsc2)=O)CC1 68403,CCC(C)C(CC(=O)N1CCn2nncc2C1)NC(=O)CSCC(F)F 68404,c1(NC(=O)NC2C(C(=O)OC)COCC2)ccc(F)c(F)c1 68405,C(=O)(CCCCNC(N)=O)NCC(C)(C)CNC(C1(C)CCNC1=O)=O 68406,C1(NC(CCC=C=C)=O)CCN(C(=O)CCC2CCOC2)C12CC2 68407,C=CC(C)CC(=O)NC(CNC(=O)CC1CNC(=O)O1)C(C)C 68408,C1(CC(=O)NC2CCC(CNC(CCC)=O)C2)CC(=O)NC(=O)C1 68409,N1(N(C(=O)C(F)(F)F)C(C2CC(F)C(=O)N2)=O)CCCCC1.Cn1ccnc1C=O 68410,Cc1ccc(CS(N2CC(CNC(=O)CC3(S(N)(=O)=O)CC3)CC2C)(=O)=O)cc1 68411,c1(N2CCC(F)(CNC(c3ccc4nccn4c3)=O)C2)ncnc2[nH]cnc12 68412,c1(C(=O)NC(CNC(C(CC)c2cccnc2)=O)CO)ccc(Cl)nc1O 68413,c1(CNCCS(=O)(=O)NCC)ccc(-c2nc(C3CC3)no2)cc1C 68414,C1(C(=O)NC2(C)CN(C(C(=Cc3cnc[nH]3)C)=O)C2)CCS(=O)(=O)N1 68415,c1(CNC(=O)CN(C2CCSC2)C(c2cn(C3CC3)nn2)=O)ccc(F)cn1 68416,CCC(F)(C(=O)OC)C(=O)NCCNC(c1ccc(CCF)cc1)=O 68417,N1(C(C(C)CCN(C)C)=O)CCC(C2CC2)C1CNC(=O)C=CC(N)=O 68418,Cc1noc(C)c1C(C)C(=O)NCCN(C1CC1)Cc1ccc(C(F)(F)F)nc1 68419,C12(CC)CCC(C(=O)NCCCN(C(C3CCCC(=O)O3)=O)C3CC3)(CC1)CO2 68420,CN1CC(C)(C(N2CC=CC(C(=O)Nc3cccc(NC=O)c3)C2)=O)CC1=O 68421,C1(CN2CC(c3nc(C(C)C)[nH]n3)OCC2)CCCCCCC1O 68422,c1(CCOC(CC(C)CC2CCC2)=O)ccccc1[N+](=O)[O-] 68423,C1(C(N2CCC(CC(F)(F)F)CC2)=O)COC2(CNC2)C1 68424,C12(NC(Cc3c(CC)cccc3)=O)CC3CCC(C1C2)N3C(c1cnsc1C)=O 68425,N1(C(C2CC=C(C)CC2)=O)CCC(C)(C(=O)Nc2ncc(C)c(Cl)n2)CC1 68426,CN1CCCC1(C)C(=O)NCC1CCN1C(=O)Cn1[nH]cnc1=N 68427,C(N=c1[nH]cnc(Cl)c1C(=O)OC)C1(NC(CCOCCOC)=O)CCOC1 68428,n1(CC(=O)NCC(CC)NC(=O)C(C)n2cccn2)nc(C)cc1C 68429,N1(C(CCCC#C)=O)CCCC2C(NC(c3cc(O)cc(C#N)c3)=O)C(C)(C)C12 68430,C=CCCC(=O)N(CCCCCNC(=O)C=CC(=O)NC1CC1)C 68431,c1(SCC(=O)NCC(C)NC(C(C)NS(CCC)(=O)=O)=O)nc2ccccc2s1 68432,c1(C(N(CCC)CCNC(C2(CCC)CCC2)=O)=O)cc(Cl)cc(Cl)n1 68433,c1(CC(=O)NC2CN(C(c3c(OC)nsc3)=O)C3C2C3)cc2ccccc2o1 68434,c1(C(=O)NC2COCCN(C(C3CC(C(C)C)C3)=O)C2)cn2ccccc2n1 68435,N1(C(C)=O)CC2C(CNC(=O)C(N)=O)C2C1.CC1(C)CC1(C(=O)OC)C=O 68436,C(=O)(C(C(C)(C)C)NC(N)=O)N(CC(C)NC(=O)C(=O)Cc1cccs1)C 68437,c1(C(N2CC(O)CC(NC(C3SCCS3)=O)C2)=O)cnn2c(Cl)cccc12 68438,C(=O)(C#CC1CCCC1)NC(C1(O)CCN(C(CCCOC(C(C)C)=O)=O)C1)C 68439,CCC(C)C(CC(=O)N(CC(F)F)CC)NC(C1CCC2(CCC2)C1)=O 68440,c1(C(=O)NCCC2CN(C(C3C(C(=O)OC)CCC3)=O)C2)c(C)cccc1O 68441,C1(C(NC=O)=O)CCCN1NCC1(F)CC1.C1C(=O)N1 68442,C(C(=O)NC)(C1=Cc2cc(Br)ccc2OC1)N(CC(CC)C)C1CC1 68443,Cc1c(C)n(C)c2ccc(C(=O)NCC3CN(C(=O)CO)CCC3C)cc12 68444,N1(C(c2c(CC)n[nH]c2)=O)CC2(CCN(C(=O)Cc3c(F)cccc3C#N)C2)C1 68445,N1(C(CCOCC)=O)C2CCCC1CN(C(=O)C(c1ccccc1)=O)C2 68446,Cc1cncc(C(=O)NC2CC(C)N(C(=O)COCCC(C)C)C2)c1 68447,C(=O)(CCC(CC)NC(=O)CCCCOC)N1C(C=C)CCC1 68448,C1(C(N2CCC(C(C(=O)OC)(C)C)C2)=O)CC(=O)N(CC(C)C)C1 68449,C1(N(C(Cn2nc(C)oc2=O)=O)C)CN(C(c2cc[nH]c2C)=O)CC1(C)C 68450,CCC(C(=O)NCC(C)(C)NC(C1CC1c1cncn1C)=O)SC 68451,C1(NC(C2CC3(CCC3O)C2)=O)CCC(O)CN(C(c2cc(CO)on2)=O)C1 68452,Cc1ccc(F)cc1C(=O)NCC1(F)CC(NC(c2cnc(C)n2C)=O)C1 68453,c1(C(N2C(CN(C(COC(CC)C)=O)C)CCCC2)=O)ccnc2ncsc12 68454,C(=O)(CN=c1cc[nH]cc1)NC(CC#C)(C)C(=O)NC1C2COCC12 68455,C1(NC(CCCC)=O)CCC2(CC1)CC2NC(=O)CC1CCC(=O)N1C 68456,C(=O)(CC(C)(C)NC(=O)Cc1ccccn1)NC(C(=O)OCC)C 68457,C#CC1CN(C(=O)CC2CC(F)CN2C(=O)CC2CNC(=O)O2)CCN1C 68458,C1(NC(c2c(C(C)C)noc2)=O)CN(C(C2COC(=O)N2C)=O)CC1O 68459,CCCCC(=O)C(=O)NC1CCC1C(N1CC(C2CC2)OC(C)C1)=O 68460,N1(C(c2ccc(F)cc2)CC)CCC2(CCCN(C(c3cncc(F)c3)=O)C2)C1 68461,C(=O)(CS(=O)(=O)CCC)N1CCCC(c2cn(C(C3CC4(CCC4)C3)CC)nn2)C1 68462,C1(O)(CCNC(Cc2ccc(C)nc2)=O)CCN(C(=O)C(C)(C)CC#N)CC1 68463,N1(C(c2cc(Cl)c(Br)c(Cl)c2)=O)CCC2C(CCN2Cc2cc(I)ccc2Br)C1 68464,C1(C(=O)NC2C3CN(C(CC(CC)CC)=O)C2C3)CCc2nnnn2C1 68465,Cc1nn(CC(=O)NC(C)(CNC(=O)C=CS(C)=O)C(C)C)c(=O)o1 68466,n1(CC)nnc(-c2nc(CC(C)CC)nn2-c2ccc(OC(C)(C)C)cc2)c1C 68467,C=C(F)C1(CC(N2CCC(C(=O)OC(=O)Cn3nc(C)cc3C)C2)=O)CCOCC1 68468,c1(C(N(C)CC2(NC(C(F)=CCC)=O)CC2)=O)cn2c(n1)CCC2 68469,C1(C(N(CCNC(C=COCC)=O)C(C)C)=O)C2CC1(c1ccccc1C)CO2 68470,C1(C(N(CCC(C)NC(c2cc(C3CC3)ccc2F)=O)C)=O)CCC(C)(C)CO1 68471,C1(C(N2CCN(C(CC(C)(C)C)=O)C(CC(F)F)C2)=O)CC2CC(O)C(C1)C2 68472,Cc1cnc(C(=O)NC2CCC(C(=O)N(C(C)C)Cc3ccccc3F)C2)cn1 68473,Cc1cncc(C(N2CCCC2CCCNC(=O)C(C)OCC2CC2)=O)c1C 68474,Cc1ccc(Cl)cc1NC(=O)C(C)(C)C1CCCN1C(=O)CC(C)N(C)C 68475,c1(CCCC(=O)N(CCNC(C=CC=CC)=O)CC)cccc(Cl)n1 68476,c1(CC(=O)NCC=CCNC(C2C(COC)C2)=O)ccc(F)c(Cl)c1 68477,N1(C(C(CCC)NC(c2nn(C)cc2C)=O)=O)CCC2(CCCOC2)C1 68478,Cc1nc(N(CC(F)(F)Br)C)cc(N2CCCC(C(N)=O)C2)n1 68479,c1(NC(C2N(Cc3c(OC)cccc3)CCCC2)=O)ccc(C)c(NC(C)=O)c1 68480,c1(C(N2CCC(NC(COCC#C)=O)CC2C)=O)cc2nc[nH]c2cc1F 68481,C(=O)(C(C)S(C)(=O)=O)NC1CCCC(NC(CSC(C)C)=O)C1 68482,C1(OC)CC(C)(C)C(=O)N1CN1CCC1CCF 68483,N1(C(=O)NCc2cc(C(=O)OCC)n[nH]2)CC(=O)N2CCCCC2C1 68484,C1(NC(C2(Cl)CC2(F)F)=O)COC2(C1)CN(C(=O)CCOC1CCCC1)C2 68485,c1(C(=O)NC2(C(=O)OC)CC(OC)C2)csc(N=S(C)(C)=O)n1 68486,C#Cc1ccc(C(N2CCC3(CC(NC(=O)CCCCSC)C3)C2)=O)cc1C 68487,CCCCCCCCC(=O)NC1CCC(NC(c2csc3ccccc23)=O)CC1 68488,N1(C(CN(C)C(N)=O)=O)CCCC(O)(CN(C)C(c2cnn(CCO)c2)=O)C1 68489,c1(N(C)C)ncc2c(n1)CN(c1cc(NC(=O)NCCCl)ncn1)C2 68490,c1(C(=O)NC(C2CCN(C(C3=C(C)OCC3)=O)C2)C)cc(C)cc(Cl)c1N 68491,C1(C(C)C)CC(NC(C2CC(C)(C)O2)=O)CO1 68492,Cc1cccnc1CC(=O)NC(CN(C)C(C1CCC(CO)CC1)=O)(CO)CO 68493,c1(-c2c(OC)ccc(-c3nccn3CC(O)CO)c2)cc2cccc(OC)c2o1 68494,C(CC(C(=O)N1CC(CC(=O)NCC2(F)CCCCC2)(OC)C1)OC)OC 68495,c1(SC)ccccc1CC(=O)NCC1CCN1C(c1cccc(NC(C)C)n1)=O 68496,N1(C(c2c(OC)nccc2)=O)CCN(C(=O)CNC=O)CC1CC1CC1 68497,C(CCCCCCC(=O)N(CCNC(=O)CC1CC2CCC1O2)CC1CC1)SC 68498,C1(NC(c2c(OC)c(C)cc(C)c2)=O)CC2(CN(C(=O)CCN=[N+]=[N-])C1)CC2(F)F 68499,C1(NC(=O)CCc2cncs2)C=CCC(C(=O)NCCCCn2ccnc2)C1 68500,Cc1ccc2cc(NC3CCC(C(=O)NOCNC)C3)ncn12.N1CCC1C1CC1 68501,n1(CCNCC(C)(C(C)C)N(CC)Cc2cccnc2)nc(C)c(C)c1C 68502,C1(CC)CN(C(C2CNC(=O)O2)=O)CC1C(=O)Nc1c(C)nsc1C 68503,N1(C(CCCCCOC)=O)CC2CCOC2(CNC(=O)Cc2nc(C)sc2C)C1 68504,c1(OCC)ccc(NC(CN(c2ccccc2N=[N+]=[N-])C(=O)CC)=O)cc1OC 68505,c1(C(N2C(C)CC(CNC(C3(C=C)CCC3)=O)C2)=O)sc2ncccc2c1N 68506,N1(C(CC=C)=O)CCCC(C)(C)C1CNC(c1c(C)cc(Cl)cc1N)=O 68507,c1(COC(N(C)C)=O)ccc(NC(=O)CC(c2ccccn2)N(C)C)cc1 68508,CC(CC(C)(F)F)C(=O)NC(c1cn(CCN2CCNC2=O)nn1)(C)C 68509,C1(C(N(C2CCN(C(=O)Cc3sccc3C)C2)CC)=O)Cc2nccnc2C1 68510,c1(C(N2CCCC(C)(OC)CC2)C(=O)NC(CC)C)cc(Cl)c(OC)cc1F 68511,c1(OCC(=C)C)cc(CN(C)C)ccc1OC.O1NC(=O)NCCC1 68512,c1(C(C(=O)NCC(CCOC)NC(c2sccc2C)=O)(F)F)ccc(C)cc1 68513,N1(C(C2=C(C)OCCC2)=O)CCOC2(C1)CN(C(=O)CC13COC(CF)(C1)C3)C2 68514,c1(NC(C2CC(c3ccccc3)CN2C(c2ccsc2)=O)=O)ncc(Br)cc1Cl 68515,c1(OC)cc(OC)c(F)c(C(=O)NC2CC(C)CN(C(C3CCCS3)=O)C2)c1 68516,c1(C(N(CC(CNC(CC2(C=C)CCC2)=O)C)C)=O)cnnc(C2CC2)c1 68517,Cc1nc2ncnn2cc1C(=O)NC1CCCCC1NC(=O)Cc1cccnc1 68518,C1(NC(CN2CC(=O)NCC2)=O)CCCC12CCN(C(=O)Cc1cccs1)CC2 68519,c1(C(=O)NC(C)CNC(=O)Cc2ccncc2Cl)ccc(S(N)(=O)=O)cc1Cl 68520,C1(CC)(NC(=O)C(C)C(C)(F)F)CCN(C(=O)C(C)Cc2ccncc2)CC1 68521,C1(CNC(c2ccc3[nH]ccc3n2)=O)CCCC2CN(C(c3nncs3)=O)CC12 68522,C1(COC(c2ccccn2)=O)CN(Cc2ccccc2Br)CCO1 68523,C(C(O)C(=O)NC1(C)CC(NC(c2cc(C3CCC3)[nH]n2)=O)C1)=CC 68524,c1(N(C)C)cncc(C(=O)NC2CC(CO)N(C(=O)C(N3CCOCC3)C)C2)c1 68525,CC1CCc2nc(N3CC4CSCC(C4)C3)[nH]c(=NCC(Cl)(Cl)Cl)c2C1 68526,c1(C(=O)NC2C(C(N(CCCC(O)CO)C)=O)COCC2)ccc([N+](=O)[O-])[nH]1 68527,c1(C(=O)NC(C(=O)NC(CC)C(=O)NC)CC2CCC2)ccn(C)c(=O)c1 68528,CC(C)C(CC(=O)NCC1CC2CCC1CC2)NC(C1CC2(CCO1)CC2)=O 68529,c1(C(N2CCC(c3sc(C(=O)OCC)c(C)n3)C2)=O)c(F)ccc(O)c1F 68530,C1(CC)CN(C(c2cc(-c3cccnc3)no2)=O)CCN1C(=O)C1=CCC1 68531,C(=O)(C1CCCc2nncn21)NC(C1CCCCC1)=O.c12nnc(s1)CC1CN2C1 68532,C(=O)(C(CN(C)C)CC)N(CCCOCCN(C(C(C)OCCCC)=O)C)C 68533,c1(C(CCNC(=O)NCC=CC)C)ccc(C(F)(F)F)cc1 68534,C(CC(C)CC)(C(=O)NCCC(=O)NCC)NC(CCCC)=O 68535,c1(CC2(NN(CCC3(CC)CC3)C=O)CCC2)nc(C(C)C)nc2[nH]ccc12 68536,N1(C(C2(NC(C(C)OCC#C)=O)CCOCC2)=O)CC2CC(C)C2C1 68537,C(=O)(CCCC(=O)NC1CCOC(c2cnn(C)c2)C1)c1ccc(OC)cc1 68538,c1(OC)ccccc1CC(=O)NC1(CCCNC(c2nocc2C)=O)CC1 68539,C(C1=NOC2CN(C(=O)CCN3CCOCC3)CC12)NC(c1cc(OC)no1)=O 68540,C1(CC(N)=O)(NC(c2n(C)ncc2)=O)CCN(C(C2CC23CC(F)(F)C3)=O)CC1 68541,C(C(C)(C)C(=O)OC)(c1n(CCC)nnn1)NCC1(c2ccccc2)CC1Br 68542,c1(C(N2CCC(C)(CC(=O)NC(CCO)C3CC3)C2)=O)cc2ncccc2[nH]1 68543,C1(C(=O)OCCN(C)C(=O)NC(C)(C)C)C2CCC(C2)C1C(F)(F)F 68544,c1(C(=O)NC2CC(CCNC(C3(Cl)C(C)(C)C3)=O)C2)cc2cn[nH]c2cn1 68545,c1(N2CCC(CC(=O)NCC(C(=O)N(CCC)CCC)C)C2)cc(CC)ncn1 68546,c1(CNC(C(C2CN(C(c3oc(CC)c(C)c3)=O)C2)OC)=O)ccc(C)nc1O 68547,C1(C)(NC(C(C2CCCCC2)NC(c2c(C)snc2)=O)=O)CCC2(CC1)CC2 68548,C1(C(N2CC(CC(=O)NC(CCC)C3CC3)(OC)C2)=O)COCCN1CC 68549,C1(C(=O)O)CN(C(c2nccs2)=O)CC12CN(C(c1cc(Br)cc(Cl)c1F)=O)C2 68550,C=C1CC2CC1CN2C(=O)C(C1(O)CN(C(=O)CC2CCC2)C1)F 68551,c1(C2C(C(=O)NCC(CNC(c3cccc(N)c3)=O)OC)C2)cccc(F)c1 68552,C(CC(=O)N1CCCC1)NC(CNC(COCC(=O)NC)=O)=O 68553,C(c1cnc[nH]1)=CC(=O)NCC(CN(C(=O)Cc1ccno1)C)O 68554,N1(C(c2cc3sccc3s2)=O)CC2(CCN(C3CCc4ccc(Cl)cc43)C2)C1 68555,c1(C(=O)NCC(CC)NC(C2CCCCC2C(N)=O)=O)ccnc(OC)n1 68556,N1(C(C2(CCNC(=O)CC3CCCOC3)CC2)=O)CC2CCCC1C2CO 68557,N(C1CCc2cccnc21)C(CC1(C)CCN1C(=O)C1CC1)=O 68558,N1(C(C2(CC)CCCO2)=O)CC(CNC(c2cc(C)ncn2)=O)C(O)C1 68559,Cc1nc2n(c1CNC(c1c(C)sc3ccccc13)=O)CCCC2 68560,c1(C(=O)NC2CCCN(C(CCCCCSC)=O)C2)cccc2c1NCC2 68561,Cc1nnc(C2CN(C(=O)NCC3CCC(O)C3)C2)o1 68562,N1(C(C2C(Cl)(C(=O)OC)C2)=O)CC2CCC(CNC(C3CC(C(C)C)C3)=O)(C2)C1 68563,C(=O)(C(CC(F)F)N(C)C(c1ccc(F)cc1F)=O)N(CCCSC)C 68564,C1(NC(c2ccc(-c3ccccc3)s2)=O)CCCN(C(c2ccncc2)=O)C1 68565,C1(C(N2CC(C)(CNC(=O)Cc3ccon3)OCC2)=O)COc2ccccc2C1 68566,N1(C(C(CC2CCOCC2)NC(c2cnsc2)=O)=O)CC2COCC2C1 68567,N#CC1(C(N2CC3(CCC3NC(=O)CCCc3ccncc3)C2)=O)CCOCC1 68568,C=C(C)CCC(=O)N1CCC(N(C(=O)C(=Cc2cnc[nH]2)C)C)CC1 68569,C#Cc1cccc(C(N2CC(NC(c3ccc(CSC)o3)=O)CC(C)C2)=O)c1 68570,C1(F)(CNC(C(C)NC(C)(C)C)=O)CCN(C(=O)CC2OCCCC2(C)C)CC1 68571,N1(CC(=O)OCC(C)CC(F)F)C(=O)Cc2ccccc2C1=O 68572,N1(CCNC(C2CC(NC(c3scc(C(C)=O)c3)=O)C2)=O)CCN(C)CC1 68573,C1(C(C)NC(=O)N(CCO)CCO)CCCC(C(F)(F)F)C1 68574,c1(N2C(C)CCC(NC(CCc3c(C)nn(C)c3)=O)C2)ncc2ncnc-2[nH]1 68575,c1(C(=O)NC2C(CNC(COC(C)=O)=O)COC2)cccc2c1CC(C)(C)C2 68576,Cc1ccc(Cl)c(OC(C)C(=O)NC2CN(C(=O)C3=NOC(C)C3)C2)c1 68577,C1(CNC(C(CC)(C)O)=O)CN(C(c2cc(Cl)cc(Cl)c2O)=O)CC(C)(C)C1 68578,C1(C(=O)NCC2(C)CCCN2C(C2(F)CCC2)=O)Cc2ccccc2S1(=O)=O 68579,N1(C(C(=O)NC2CCN(c3ccc(F)cc3F)C2)=O)CC2CCCCCC2C1 68580,C1(NC(C(C)CC2CCC2)=O)CCCC12CN(C(c1sc(F)cc1Cl)=O)C2 68581,C(=O)(CC(C(=O)N1CC(N(C(=O)C=Cc2ccsc2)C)C1)NC(C)=O)OC 68582,c1(OC)cncc(NC(C2CCC2NC(c2ccccc2C)=O)=O)c1 68583,Cc1cc2[nH]c(C(N3CC4=C(C3)CN(C(C3(C)CCCCO3)=O)C4)=O)cc2s1 68584,c1(C(=O)NCC(C)CN(C(=O)CC2COC(=O)N2)C)ncc(Cl)nc1Cl 68585,Cc1cccc2c1CC(C(N1CC3CN(C(=O)C(C)C(F)F)CC3C1)=O)O2 68586,CCCC(O)CN=c1[nH]c2cc(Cl)c(S(=O)(=O)NC3C4CCCCC34)cc2s1 68587,C(=O)(C1=NNC(=O)CC1)N(C(C)CNC(c1cnc2n1CCS2)=O)C 68588,C=CCC(CN(C)C(=O)NC1CC1)NC(=O)C(OCC)OC(C)(C)C 68589,N1(C(=O)CCC2CCOC2)CCCCC(C(=O)NC2(C3CC3)CCCC2)C1 68590,N1(C(C2(CC)CC2)=O)C2CCC1C(C(=O)NCc1ncn(C3CC3)n1)C2 68591,c1(C(=O)NC23CCC(CN(C(c4ccnnc4)=O)C2)C3)cnc(O)c2cncn12 68592,Cc1csc(=NCC(=O)N(C2CCCN(C(C3CS(=O)(=O)CC(=O)N3)=O)C2)C)[nH]1 68593,N1(C(c2cscn2)=O)CCN(C(C2CC3(CCC3)CO2)=O)C(CF)C1 68594,N1(c2snc(CC)n2)CCC2C(CCCN2C(=O)CC2(C)CC2)C1 68595,c1(N(C)CC2(OC)CCOC2)[nH]c(=NC(C)c2cnn(C)c2)nc2sccc12 68596,Cc1cc(C(N2CC3(CC(NC(c4cnsn4)=O)CO3)C2)=O)c(Cl)cc1Cl 68597,C1(NC(=O)NC)CCC12CCCO2.c1(CNC(=O)OC(C)(C)C)c[nH]nc1C 68598,c1(N2C(C)(C)C(NC(=O)Cn3cncn3)CC2)cc(C#N)ccc1[N+](=O)[O-] 68599,N1(C(c2ccn(CCC)n2)=O)CCN(C(c2cc(CN(C)C)on2)=O)CC1CF 68600,C(C)(CC(C)NC(c1ccnn1C1CC1(F)F)=O)NC(COCCOCC)=O 68601,c1(C(N2CCCC(C(C)NC(C3(SC)CCC3)=O)C2)=O)cc(C)nc(O)c1 68602,N1(C(C2C(CCOC)C2)=O)CCN(C)C(C(=O)NCC2(CO)CC3CC3C2)C1 68603,Cc1ccc(F)c(C(N2CC(O)CC2CNC(=O)Cn2nc(O)ccc2=O)=O)c1 68604,Cc1[nH]c(C#N)cc1C(=O)NC(c1nocc1C(=O)NCCOCC(F)F)C 68605,C1(C(N2C(C(C)NC(Cn3c(C)c(Cl)cn3)=O)CCC2)=O)CCn2cnnc2C1 68606,N1(C(CC(c2ccc(Br)cc2)NC(C)=O)=O)CCCC(NC(C)C)C1 68607,N1(C(C(CC)O)=O)CC2(CCC2)CC1CNC(c1ccnc(-c2ncc[nH]2)c1)=O 68608,Cc1cc(C)n(CC(=O)NCC(C2(O)CCN(C(c3[nH]c(O)nc3C)=O)C2)C)n1 68609,C1(NC(C2C(C(=O)NCC#C)C2)=O)C=CCN(C(=O)CC23CCC(CC2)C3)C1 68610,N1(C(CC(C)=C(C)C)=O)CCCC(C)(C(=O)Nc2cccc(Cl)c2)C1 68611,C(CC)(CC)(CCNC(c1c[nH]cc1-c1cc(C)no1)=O)NC(C=COCC)=O 68612,C12CN(CC1F)C2=O.c1(CNC(C(=O)OCC)=O)ccc(N2CCNCC2)cc1 68613,Cc1cccc2c(NC(=O)Nc3ccc(NCC45CC=CC(C4)OC5)cc3)coc12 68614,CCC(F)(C(=O)OC)C(=O)NCCC12CCC(CC1)N(C(c1cn[nH]c1)=O)C2 68615,Cc1cncc(C(N2CCC(CNC(c3nncs3)=O)C2)=O)c1 68616,C1(NC(c2c(CC)[nH]cc2)=O)CCN(C(=O)C=Cc2cncc(O)c2)CC1C 68617,c1(C(N2CCC(N(C(COCC(C)C)=O)C)C2)=O)cc(N)cc(F)c1 68618,CCCCC(O)CC(=O)N1CC2C(CNC(=O)C=C(Cl)Cl)C2C1 68619,Cc1ccc(F)c(CNC(C2(CNC(C3CCSC(C)C3)=O)CCOCC2)=O)c1 68620,C1(NC(=O)COCCc2ccccc2)CCN(C(c2cnco2)=O)CCC1CO 68621,c1(C(=O)NC2(C(=O)OC)CCC2)ccc(NC(C2(C(F)(F)F)CC2)=O)cc1F 68622,N1(C(C2C(C)(C)C2)=O)CCCC2CCN(C(=O)C=Cc3nccs3)CC12 68623,C1(NC(COc2c(C)cccc2)=O)CCCN(C(c2cccc(F)c2F)=O)C1C 68624,C1(NC(=O)NC2(c3ccc(Br)cc3)CC(O)C2)CCSC2(C1)CC(C(=O)O)C2 68625,C(CCCCNC1CCCO1)N(C(C(c1ccccc1)NC(=O)OC)=O)C 68626,Cn1cc(C(=O)NCC2(NC(=O)CC3=CCOCC3)CC2)c2ccccc12 68627,CC(c1ccccc1F)=CC(N1CC(N(C)C(C2COCCN2C)=O)C1)=O 68628,C1(CNC(C2(C(C)C)CCOCC2)=O)CNCC(C)(C)C1 68629,N1(C(CCCNC(N)=O)=O)CC2CCC1CC2NC(=O)CC1CCCSC1 68630,C1(CCNC(C2(NC(=O)COCC3CCC3)CC2)=O)CCCCC1 68631,c1(NC)ccc(C(=O)NC2CCC2NC(=O)CCc2ccncc2)cc1[N+](=O)[O-] 68632,C1(C(=O)NCCN(CCC)C(C2COCCN2C=O)=O)CC2CCC(C1)S2 68633,c1(C2CCN(CC(=O)NC(C(=O)OCC)CC)C2)c(C)noc1C 68634,C1(NC(=O)CC2(O)CCC2)CC2CCC1CN2C(C1CNC(=O)N1)=O 68635,C#CCCC(C(=O)Nc1cccc(C#N)c1)NC(c1[nH]nnc1C)=O 68636,C(=O)(CC(C)CC(C)(C)C)NCCC(=O)NCc1ncc(C)cn1 68637,Cc1ccc(C(=O)NC2CCOCC2NC(C23CC(F)(C2)C3)=O)c(F)c1F 68638,N1(C(C(C(C)NC(=O)C(N2CCNC2=O)C)(C)C)=O)CCC2CCCC2CC1 68639,C1(C(=O)NCC23C(CN(C(CNC(=O)OC)=O)C2)C3)CCc2nc(C)[nH]c2C1 68640,Cc1nc(CNC(=O)CC2C3CN(C(=O)CCc4ccccc4F)CC23)oc1C 68641,c1(C(N(C(C(=O)NC(CCC)c2nn[nH]n2)C)C2CC2)=O)snc(C)c1N 68642,CN1CCC(NC(c2ccn(CCNC(=O)Cc3ccsn3)c2)=O)C(C#N)C1 68643,C(=O)(C(C(C)O)NC(C)=O)NCCN(C(c1cc(C2CC2)ns1)=O)CC 68644,c1(C(=O)NC2C(NC(c3ccoc3)=O)CC2)c(F)cc([N+](=O)[O-])cc1Br 68645,c1(C(N2CCCC(CCNC(C(C)=CC)=O)C2)=O)cccc2c1OC(C)C2 68646,CCC(C)(C(=O)N1CC(CO)(NC(=O)CCc2nc(O)n[nH]2)C1)OC 68647,N1(C(CCC=CC)=O)CC(NC(=O)C=Cc2ccccn2)CC1(C)COC 68648,CC(C(C)(C)NC(c1cnc(C(F)(F)F)s1)=O)NC(c1csnn1)=O 68649,c1(C(=O)NC(CC2CN(C(c3cc(C)[nH]n3)=O)C2)C)cc2sccc2s1 68650,O=C(C#CC1CCOC1)N1CCCOC(CN=c2cc[nH]c(-c3nccs3)n2)C1 68651,N1(C(C(CC)N(C)C(c2ncnc(C)c2C)=O)=O)CCCC(C)(C)C1C 68652,N1(CC(C2CC2)OC)CC2CCC1CN2C(C1CC(NC(=O)OC)CCO1)=O 68653,N1(C(C2(CC=C)CCN(C(=O)C(C)OCCC(C)C)C2)=O)CCC(O)CC(C)C1 68654,N1(CC)CCN(C(C2(CF)CCN(C(=O)C=CC(C)C)C2)=O)C(C)C1 68655,c1(CCCCC(=O)NC2CCCC(CNC(CSCC)=O)C2)ccc(C#N)cc1 68656,N1(C(COCCC)=O)CC(NC(=O)C(C)(C)Cc2cnn[nH]2)CC1(C)C 68657,CCCCCCOCC(=O)NCC1(NC(c2cnc(O)o2)=O)CCOC1 68658,CN1CCC(C(N2CCC(N3CCCC3)C2)C(=O)NCc2ccco2)CC1 68659,c1(OC)cc(C(CO)NCc2cc(Cl)ncc2NC(=O)OC(C)(C)C)cc(F)c1 68660,C1(NC(c2cncc(F)c2)=O)CN(C(=O)C#CC2CCCO2)C2(CCC2)C1 68661,C1(COCC)CCCN1C(=O)C(C1CC1)N(C(=O)C=CC(F)(F)F)C 68662,C1(C2CC2)(CNC(CN(C2CC2)CC)=O)CCN(c2nc3ccccc3o2)C1 68663,c1(C(N(CCOC)CCNC(=O)CC2(OC)CC2)=O)cc2ccc(Cl)c(F)c2[nH]1 68664,N1(C(CC(=C)C)=O)CCCC2CN(C(C3CCc4c(nnn4CC)C3)=O)CCC12 68665,C1(C#CC(=O)N2CCCC(NC(C34CC(c5ccccc5)(C3)C4)=O)C2)(CC)COC1 68666,N1(C(C2C(C)(C)CCN2C(C2CCCOC2)=O)=O)CCCC2C(=O)NCC12 68667,Cc1cccc(C)c1N1CCC(NC(=O)CN(C(=O)CC(C)(C)C#N)C)C1 68668,c1(CC(N2CCC(C(C)CNC(=O)CC(F)F)CC2)=O)c[nH]c2ncccc12 68669,Cn1c(O)nc2cc(C(=O)NC3CN(c4cnc(F)cn4)CC3(C)C)ccc12 68670,Cc1noc2ncc(C(=O)NC3CC4CC3N(C(c3ncccn3)=O)C4)cc12 68671,CC1(C)CC(O)(CC(N2CC(CCCCNC(c3nn[nH]c3Cl)=O)C2)=O)CO1 68672,c1(NC(c2c(C)cccc2)CO)cc(Br)ccc1S(=O)(=O)NCCC1CCCC1 68673,Cc1ccc(CN(C)Cc2cn(-c3cc(Cl)cc(Cl)c3Cl)nn2)c2cccnc12 68674,C(=O)(CC(C)CC(F)(F)F)NC1(CNC(C2ON=C(C(C)C)C2)=O)CCCCC1 68675,Cc1cc(C(=O)NC2CN(C(C3CCOC(=O)N3)=O)CC2F)oc1C 68676,C(=O)(C1=CC2C=CC1C2)N(CCC(=O)Nc1cccc2c1OCC2)C1CC1 68677,C1(NC(CN(C(C)=O)C)=O)CCC(C)(CNC(=O)Cc2csnc2C)C1 68678,C1(=CC(=O)NC(CCC)CCCNC(=O)C(C)CF)CC2CCC(C1)N2C 68679,C#CCCCCCCC(=O)NC1CC(NC(c2ocnc2CC)=O)CC1O 68680,N1(C(CNC(=O)CC(F)(F)F)=O)CCN(C(=O)C=CC2CCOC2)C2CCCC12 68681,C(=O)(C1=CS(=O)CCC1)NC12CCC(CNC(c3cnc(C)[nH]3)=O)(OC1)C2 68682,c1(C(N2C(CCNC(CC3ON=C(C)C3)=O)COCC2)=O)ccc(Cl)cc1O 68683,c1(C(N(C)CC2(NC(=O)CCC3CC3(C)C)CC2)=O)ccnc(Cl)c1Cl 68684,c1(SC)cccc(NCCNC(=O)C(c2ccccc2)NC(C)=O)c1 68685,N1(C(C(C(C)C)n2ccc(C)c2)=O)CC(O)C(O)C(O)C1C=O.CCO 68686,C1(C(N(C)Cc2nc(CC)on2)=O)COCCN(C(C)CC2(O)CCOCC2)C1 68687,c12ccc(F)c(c1)NC(=O)N2CC.C1(C(N2CCCC2)=O)CN(S(N)(=O)=O)C1 68688,c1(CC(=O)NC(CNC(Cc2c(C)ncs2)=O)C)ccc(F)c(Br)c1 68689,c1(CC(N2CC(F)(CNC(C3(COC)CCCC3)=O)C2)=O)cc(F)ccc1C 68690,C1(NC(=O)NC(CSC)(C)CO)C(=O)NCCC1C 68691,C1(C2CC2)(C(N2C(C)CC2(C)C)=O)CN(C(=O)CC2CC3C=CC2C3)C1 68692,c1(CC(=O)NC2CN(Cc3n(C)cnc3)CC2O)ccc2c(c1)OCO2 68693,CC(C)(C)CC(O)CC(=O)NC1CCCCC1NC(c1cc2cccnn2c1)=O 68694,C(C)(N=c1ccnc(NCC2CC2(C)C)[nH]1)c1ccc(SC)cc1 68695,CCC(C)CCC(=O)NCC(C)(CNC(c1ccc(F)cn1)=O)OC 68696,CCC(CC(=O)N(CC(C)C(=O)NC(c1ccncn1)C)C)C(F)F 68697,C(=O)(C#CC(C)(C)CNC(=O)CN(C)CC)N(C(C#C)C)C 68698,C(=O)(C1=C(Cl)CCC1)N1C(C(C)NC(=O)CCOCC(F)F)CCC1 68699,C1(n2cc(C(C3CC(=O)NC3=O)C)nn2)CCN(C(=O)CC2CCCOC2)CC1 68700,CCCCC(C(=O)NCC1(CC(C)C)CCC1)NC(c1cn(C)nn1)=O 68701,CC(C)CCCC(C)C(=O)N1CCC(C)(C(=O)NCC23CCCC2OCC3)C1 68702,N1(C(CN(C2CCC2)C)=O)CCN(C(C2CC23CCOC3)=O)CC(O)C1 68703,Cc1c(C(N2CC3CC3(NC(=O)CC3CC4(CCC4)CO3)C2)=O)cncc1N 68704,C=CCCCCCC(=O)NC1(C2CC2)CCN(C(c2ccc[n+]([O-])c2)=O)C1 68705,N1(C(c2c(C)ccc(=N)[nH]2)=O)CC2CCCC2(NC(=O)CCC2CCOC2)C1 68706,C1(CNC(C(C2CCN(C(=O)CCC(C)N(C)C)C2)C)=O)C(C)(C)C1(C)C 68707,N1(CC(=O)NC2CN(C(C3(C(F)F)CCCO3)=O)CC23CC3)CCS(=O)(=O)CC1 68708,C1(CCC)COCCN1C(C1CCCCC1NC(c1ccncc1OC)=O)=O 68709,Cc1cc(=N)[nH]cc1C(=O)NCC1CC1CNC(=O)C(C)(C)C(C)C 68710,c1(CC)nc(C(=O)NCCC2CCN(C(C3(CC)COC3)=O)C2)c(C)o1 68711,N1(C(c2c(CC)nco2)=O)CCC(NC(c2ncccc2OC(C)C)=O)C(C)C1 68712,C(C1NC(=O)c2ccccc21)CNC(C1NCCC1C(F)(F)C(F)(F)F)=O 68713,N1(C(CC2C(=O)OCC2)=O)CC(O)(C2CCN(C(=O)CCC3CC3)CC2)C1 68714,N1(C(C2CN(C(c3c(C)nc(O)s3)=O)C(C)(C)C2)=O)C2CCC1CC(=O)NC2 68715,C1(C(C)NC(C2CCCC2)=O)CN(C(=O)CCCNC(C2CCC2)=O)CC12CC2 68716,N1(C(c2c(OC)nsc2)=O)CC2=C(C1)CN(C(=O)CC1C=NN(C)C1=O)C2 68717,c1(NC(=O)Nc2cc(C)sn2)cccc(CC2CC2)c1 68718,C1(NC(C(C)(C)NC(C=COC)=O)=O)CN(C(c2cnc(C(C)C)s2)=O)CC1F 68719,C1(C)(CNC(CC(C)CF)=O)CCCN(C(c2cc(NC(N)=O)ccc2O)=O)C1 68720,c1(OC)cc(NC(C2(F)CCN(C(c3c(Cl)ccnc3Br)=O)C2)=O)nc(Br)c1 68721,C12(C(=O)NC3C(C)(C(=O)NCc4ccc(OC)cn4)CCC3)CC(C)(CCO1)C2 68722,c1(C(N2CC(CNC(COC(C)(C)C)=O)OCC2)=O)ccnc2[nH]ncc12 68723,C(=O)(C#CC1CCCC1)NC(CNC(C(CCC)(F)F)=O)C 68724,C(C(C)(C)CC(=O)NCCOc1ccccc1)NC(C(C1CCC1)OC)=O 68725,C#CC(C)(C)C(=O)N1CCC(NC(c2cc(SC)c(C)o2)=O)CC1 68726,C1(NC(c2ccc(CCCC)cc2)=O)CN(C(=O)CN(C)CC)C2CCCCC12 68727,N1(C(c2cnc(CC)s2)=O)CC2CC(NC(=O)CNS(=O)(=O)NC)C2C1 68728,c1(C(=O)NCC(C(C)C(C)C)NC(CCC(=C)C)=O)ccc(P(C)(C)=O)cn1 68729,Cc1nn(C)c(C)c1NC(C1CCN(C(c2ccc(C(F)(F)F)cc2I)=O)C1)=O 68730,C1(NC(C(C2CC2)NC(CCOC(C)=O)=O)=O)CN2CCC1(C)CC2 68731,N1(C(COCCCCC)=O)CCc2sccc2C1CNC(C12CC(CCO1)C2)=O 68732,CC1CN(C(=O)C#CC(C)(C)C)CCC1NC(c1cccc(NS(N)(=O)=O)n1)=O 68733,c1(C(=O)NCC(C(C)C)NC(c2ccccc2CN(C)C)=O)cc2n(n1)CCCC2 68734,N1(C(C2(NC(CSCCC(C)C)=O)CCC2)=O)CCOC(C(N)=O)CC1 68735,c1(C(N2CC(OC)C(NC(c3cnc(Cl)s3)=O)C2)=O)cc(C)n(C2CC2)c1C 68736,C(=O)(C1=NOC(C(C)(C)C)C1)NC(C)CNC(=O)CC(C)(C)c1ccc(F)cc1 68737,C1(CNc2ccc(N3C(=O)OCC3)cc2)CC2OC1C1CC21 68738,Cc1cccc(C(N2CCN(Cc3ccc(F)c(F)c3)C(C)C2)=O)c1C 68739,c1(OC)cc(CCNC(C2CC(C)(C)C23CCC3)=O)cc(OC)c1C 68740,C(C(C(=O)N1CCC2(C1)CN(C(c1cc(C)c(C)s1)=O)C2)C(F)(F)F)OC 68741,C1(NC(c2cccc(C3CC3)c2)=O)CC1C1CCCN(C(c2cccnn2)=O)C1 68742,c1(OC(C(=O)N(CCN(C(c2cc(CCC)on2)=O)C)C)C)ccc(Cl)cc1C 68743,C1(OC)CC(CNC(=O)CN2CCN(C)CC2)N(C(C2CCC2C(C)(C)C)=O)C1 68744,N1(C(C=CCN(C)CC)=O)CC2CCCC2(CNC(=O)CCCCN(C)C)C1 68745,c1(C(N(C2CCCN(C(C3CCCC4CC34)=O)CC2)C)=O)nc2ncccn2n1 68746,N1(CC)CCC(N(C)Cc2cscc2-c2cncc(CO)c2)CC1C 68747,c1(OC)ccc2oc(C(N3CC4CC3C4C(=O)Nc3ccc(O)nc3)=O)cc2c1 68748,c1(OCC(=O)NC(C(C)(C)C)C(=O)NCC2CSC2)ccccc1[N+](=O)[O-] 68749,N1(C(C(C)Cn2ccnc2)=O)CCn2ncc(NS(C)(=O)=O)c2C1 68750,CC1CC(CNC(c2cnc[nH]c2=N)=O)CN1C(=O)CCc1cnccn1 68751,O=Cc1cccc(CN2CCC3(CC3C(=O)Nc3ccc4c(c3)OCO4)C2)c1Br 68752,C1(C(=O)NC(C(=O)NCCC2CC=CC2)c2cccs2)(C2CC2)CCCO1 68753,c1(CS(=O)(=O)N(C)CC2C(C)C2)cccc(F)c1 68754,N1(C(C2CC(C)(C)NCC2)=O)CC(C)(C)C(O)C1(C)C 68755,C12(NC(c3n(C)ccn3)=O)CCC(CC1NC(C1CC1c1ccc(F)cc1)=O)C2 68756,C1(N(C(=O)C(F)CC)CCCC)CCN(C(=O)C(C2CCOCC2)F)CC1 68757,C1(CC(=O)OC)(NCC(c2ccc(C)cc2)O)CS(=O)(=O)C1 68758,c1(CN2CCC(NC(c3cnc(O)nc3O)=O)CC2)c(Cl)cc(Cl)cc1Cl 68759,C(=O)(C1=NOC2COCC12)N1C2C(NC(CCNC(=O)CO)=O)CC(C2)C1 68760,c1(CNC(COCC(C)C)=O)nc(CNC(=O)C(C)(C)c2cncs2)cs1 68761,CC1CCN(C(C2CCCC2(C)C)=O)CCN1C(c1cnco1)=O 68762,CCCCC(C(=O)NCCC1CCCCN1C(=O)CN(C)C)C(C)C 68763,n1(CC(=O)N(C(c2ccccc2)CNC(c2cnnn2C)=O)C)nnc(C2CC2)n1 68764,C(CCCCCNC(c1c(Br)noc1C)=O)NC(CC1CC(CC)C1)=O 68765,C(CCCC(=O)OC)(C(=O)NCc1cccc(Br)c1)N1CCCC(COC)C1 68766,C(=O)(C(C)CC(C)C)NCc1c(C(=O)NC(CCCC)(C)C)occ1 68767,Cc1cc(C(=O)NCC(=O)N(CCCN(C(=O)C(F)CC2CC2)C)C)c(C)o1 68768,C(=O)(C1CCc2c(Cl)cccc21)OCC(=O)NC(Cc1ccc(C)cc1)C(=O)O 68769,N1(C(c2cc3ncccc3o2)=O)CCC2(CCCN2C(c2c[nH]nc2Br)=O)C1 68770,CC1=CCCN(C(=O)C(Cn2cncn2)NC(C2CCN(C)CC2)=O)C1 68771,S(=O)(=O)(c1cn(-c2ccccc2)nn1)NCC1(CO)C(C)(C)C1 68772,C(=O)(C(O)CC(C)(C)C)NC(C1CCN(C(C2OCCCO2)=O)CC1)C 68773,C1(C(=O)NCCC(=O)NC(CC)C)CCOCC1NC(C1OC2CCC1C2)=O 68774,c1(C(=O)NC2C(CNC(C3(Br)C(C)(C)C3)=O)C2)ccn2c(O)nnc2c1 68775,C(C(COC)C(=O)NC(CO)C(C)NC(C1(N(C)C)CCC1)=O)OC 68776,c1(CCC(=O)NCCN(C(=O)Cc2nc(C)cs2)CC)ccc(Cl)cc1F 68777,C12(COC)CC(CNC(c3ccc(Cl)o3)=O)(CN1C(C1(C(F)F)CCCO1)=O)C2 68778,C1(NC(C2(CCNC(C(CC)(C)C)=O)CC2)=O)CC2CC1C(O)C2O 68779,C1(C(=O)NC2(CSC)CCC2)CN(C(C2CCO2)=O)CCC1C 68780,N1(C(c2ccc(C3CC3)nc2O)=O)CC2CCCN(C(=O)Cc3cccs3)C2C1 68781,Cc1cc(C(=O)N(CC(C)CNC(c2c(C(F)F)cnn2C)=O)C)sc1C 68782,C(C(=O)NCc1cn(C2CN(C(=O)CC(C)C)C2)nn1)(C(C)(C)C)NC(C)=O 68783,N1(C(C(C(C)CNC(c2coc3c2COC3)=O)F)=O)CCCCN(C)CC1 68784,c1(-c2scc(CC(=O)NCCN(C(c3c(CC)nco3)=O)C)n2)ccc(O)cc1 68785,Cc1cc(C(=O)NCC(C)(C(C)C)NC(=O)CC2CCCC(C)(C)O2)nc(O)c1 68786,C1(N(C(CN(C2CCSC2)C)=O)CC2CC2)CN(c2nncs2)C1 68787,c1(C(=O)NC2C(NC(c3sc(CC)c(C)c3)=O)CC2)ccc(F)c(F)c1C 68788,C1(C(=O)NCCN(C(CN2CCN(CC)CC2)=O)C)CC(C2CCCC2)C1 68789,c1(C(N(CCOC)CCNC(=O)Cn2cnccc2=O)=O)cc(O)cc(N)c1C 68790,C(=O)(C(CCNC(c1ccc[n+]([O-])c1)=O)OC)NC(C(=O)OCC)C 68791,C=CCC(C)C(=O)NCC1(CC(=O)NC(CCOC)C(C)C)CC1 68792,N1(C(CSSC)=O)CCC2(CCCCC2NC(c2nncs2)=O)CC1 68793,N1(C(CCCCCNC(CCCCC=CC)=O)=O)CC2CC(C)(C)C2C1 68794,O(C=CC(O)(CNC(=O)C(C)(COC)Nc1ccccc1)C(F)(F)F)CC 68795,c1(OC)c(C(=O)NC(C2CCCCN2C(=O)CCN(C)CCO)C)cccc1F 68796,Cc1cc(C(N2CC(NC(C3C4COCC34)=O)C(n3cccn3)C2)=O)nc(C)n1 68797,C(C)(CCC(=O)NC1CC1CNC(=O)CC1CC1(C)C)OC 68798,Cc1nc(C(C)C)nc(O)c1C(=O)NC1CCCC1NC(C1(CF)CC1)=O 68799,c1(C(=O)NCC2CN(C(CC=CCC)=O)CC2O)nc(C2CC2)ncc1Cl 68800,CC(=O)CCCC(=O)N1CCC(C(F)(F)F)C(NC(=O)Cn2nc(C)cc2N)C1 68801,C#CC1CCCC(NC(C2CC(F)(F)CN2C(=O)CCOCC(F)F)=O)C1 68802,N1(C(c2csnn2)=O)CC2CCC2(CCNC(C23CC(CC(F)F)(C2)C3)=O)C1 68803,N1(C(C(C)NC(N)=O)=O)CC(CNC(=O)Cn2nccn2)C(c2ccccc2)C1 68804,C(=O)(C1=NOC2COCC12)N1CC=C(C(=O)NCCC(C=C)C)CC1 68805,c1(CC(=O)NC2CC(CNC(COCCC(C)C)=O)C2)ccc2ccoc2c1 68806,C1(CCNC(C(CC)(F)F)=O)C(C)CCCN1C(=O)CCOc1cccc(F)c1 68807,C(CSC1CCCO1)(C(=O)NC1CC1NC(=O)CSC(F)(F)F)OC 68808,S(=O)(=O)(c1cccc(Br)n1)N1C(C)(C(=O)NCc2cncc(Br)c2)CCC1 68809,C1(NC(C(CCC)C)=O)CCC12CCN(C(c1c[nH]c(=NC)s1)=O)CC2 68810,C1(NC(C2(SC)CC2)=O)CCCC2CN(C(c3noc4cc(F)ccc34)=O)CC12 68811,N1(C(COCCOCC#C)=O)CC(C)CCC1CNC(=O)C(=O)NC1CC1 68812,CCCCCCC(=O)NCC(N1CCCC1C(=O)Nc1cccc(Cl)c1C)=O 68813,C1(OC)COc2c(C(N3CCCC3CN(C)C(c3scnc3Cl)=O)=O)cnn2C1 68814,O=c1cc(CN2CCC(c3nccc(N4CCCC4)n3)C2)nc2ncccn12 68815,Fc1cncnc1SCc1nnc(Nc2ccccc2)o1 68816,c1(OC)ccc(C(=O)NCC2CC(C)N(C(=O)CCc3cnccn3)C2)cc1Cl 68817,c1(C(=O)NC2CC(C(N3CCC(C4CCCO4)C3)=O)C2)ccnc(CO)c1 68818,Cc1nc(Cl)nc(N2CCC(NC(C3CCCC(F)(F)CC3)=O)CC2)c1[N+](=O)[O-] 68819,CC(C)(C#N)CCC(=O)NC1(CNC(c2cc3ccccc3o2)=O)CCOC1 68820,C1(CNC(c2cnn(CC)c2C)=O)CN(C(=O)CC(O)C(C)(C)C)CC(C)(C)C1 68821,C1(C(NOCC(CC)C)=O)CCC(C)N1C(c1ccc(C)n1C)=O 68822,c1(C(=O)NCC2C(NC(C3CC=C(C)CC3)=O)C2)cn(C)cc(Br)c1=O 68823,C=CC(C)(C)CC(=O)NC1(CNC(=O)COCc2ccnn2C)CCCCC1C 68824,c1(C(=O)NCC2N(C(Cc3cn(CC)nc3)=O)CCC2C)cc(Cl)c([N+](=O)[O-])[nH]1 68825,CC1=NOC(C)(C(N2CC3C(N(C)C(c4cn(C(C)(C)C)nn4)=O)C3C2)=O)C1 68826,c1(CC(=O)Nc2ccc(CNc3ccccn3)cn2)ccccc1F 68827,CC1CC(NC(C2(F)CC2)=O)CCN1C(c1ccc(-c2ccccc2)cc1F)=O 68828,c1(NCC(=O)NCCC(C)NC(C2C3CCCC23)=O)ccc(Cl)cc1Cl 68829,C(C(O)C(=O)NCCN(C(=O)C(C)N(C)C)CCSC)SC 68830,C1(C(C)C)CN(C(C2CC3CC3CC2C)=O)CCN1C(c1ccccc1CO)=O 68831,C1(CC(C)NC(C=C(C)C(C)C)=O)CCN(C(c2cc(C3CC3)no2)=O)CC1 68832,CCC(CCCC(=O)NC1(C)CCCC1(F)F)NC(c1c(C)ccn1C)=O 68833,C#Cc1ccc(CC(N2CCC(F)(C(N3CCC(F)(CO)C3)=O)CC2)=O)cc1 68834,C1(CN(C(C(C2CCOCC2)OC)=O)C)CC(F)CN1C(=O)CCOC 68835,C=Cc1ccc(C(=O)NC(C)C(C)C(=O)N(CC(C)C#N)C2CC2)cc1 68836,n1(C(CC)(C)C)nnnc1C1(NC2(c3cnn(CC(C)C)c3)CC2)CCCC1 68837,c1(C(=O)O)cc(S(=O)(=O)COC2CC3(CN(C(C4CCCO4)=O)C3)C2)ccc1F 68838,c1(C(=O)NCC(=O)NCCC(C)NC(c2cccc(=O)o2)=O)ccc(N)cc1 68839,C(C)(C)(C(C)CC(=O)N(C1CC2CCC1O2)C)NC(CCC(C)CN(C)C)=O 68840,Cn1c(N2C3CCC2(CNC(C2CCCSC2)=O)CC3)c(C#N)c(=O)n(C)c1=O 68841,CCCC(C)CC(=O)N(CCNC(C1(c2ccccc2C)CCCC1)=O)C(C)C 68842,C1(CCC(=O)NC2(COC)CCC2)CCN(C(=O)CCn2ccnn2)C1 68843,Cc1cc(-n2cc(CCC(C3CCCC(OC(C)(C)C)CC3)=O)nn2)cc(C)c1 68844,C1(NC(c2scc(OC)c2OC)=O)CC2(C1)CN(C(C1CCOC1(C)C)=O)C2 68845,C1(COC)(CNC(=O)C(F)CC2CCC2)CN(C(=O)C(F)C2CCCC2)C1 68846,c1(C(N2C(C(N3CC(C=C)C(O)C3)=O)C(C3CC3)CC2)=O)cccc2ccoc12 68847,c1(COC)csc(C(N2CCC(CNC(C3CC3(Cl)Cl)=O)C2)=O)c1 68848,C(=O)(CS(=O)c1ccc(Cl)cc1)N1C(C(C)C)CN(C(=O)COCCN(C)C)CC1 68849,c1(C(C)(C)C)ccc(C(N2CCCC(N(CCO)C(c3cscc3Cl)=O)C2)=O)cc1 68850,CN1CCN(C(=O)Cc2ccc(C#N)cc2)CC1CNC(C1CNC(=O)N1)=O 68851,C1(CNC(=O)OC(C)(C)C)CC(CNC(=O)NCC2CC23CCN3)CO1 68852,Cc1cc(Cl)n[nH]c1=NC(=O)C1CC(O)CN1C(c1cccc2c[nH]nc12)=O 68853,N1(C(C2(COC)CC=CC2)=O)CC2(CC(NC(=O)CN3CCOCC3=O)CO2)C1 68854,C1(C)(NC(C2CC(=O)N(C)C2c2ccccc2)=O)CCc2ccccc2C1 68855,n1(CCC(=O)NCCOCC(=O)NCC(C)(C2CC2)OC)ccnc1C 68856,N1(C(C(CC)C)=O)CCC(NC(=O)CN(C2CCCC2O)C)C1C 68857,Cc1ccc(C)c(CC(=O)NCC(C2CCN(C(c3occc3C)=O)CC2)C)c1 68858,C1(CN(C(C2CCC(C)S2)=O)C)CCN(C(=O)CCc2cccnc2)CC1 68859,N1(C(CCN(C)CC)=O)CCC(C)(CCNC(C2CCC(F)C2)=O)CC1 68860,C1(CNC(CCOCCC)=O)CN(C(=O)CNC(=O)Cc2ccccc2)CC1O 68861,CON(C)C(=O)CN=c1ccnc(NC(c2nc3ccccc3[nH]2)C(C)C)[nH]1 68862,C1(NC(=O)Cn2ncnn2)COC2(C1)CN(C(c1cc(CCCO)on1)=O)C2 68863,CC1(NC(C2CC2C(F)(F)F)=O)CCCN(C(C23CC4CC2C3C4O)=O)C1 68864,C(C)(C)(CCCCC(=O)NC1CCC(NC(c2cscc2OC)=O)C1)OC 68865,C(CC1CC1)(C(=O)NC(C)C1CC1)NC(CNC(CCSCCCO)=O)=O.C1CC1 68866,c1(C(=O)NCCCOCCNC(CSCC#C)=O)nnn2c1CCCCC2 68867,C1(F)(C(N2CCN(CC(C)NC(c3cc(C)no3)=O)CC2)=O)CCC(C)CC1 68868,c1(C(=O)NCC(CNC(=O)C(O)C(F)F)OC)cc(F)c(F)c(F)c1 68869,N1(C(c2ccc(C#C)cc2)=O)CCC(C(=O)NCCN(CC(F)F)C)CC1(C)C 68870,c1(SCC(=O)NC(CNC(c2nc(C(C)OC)oc2)=O)C)ccccc1O 68871,C(=O)(C#CC1CC1)NCCc1c(C(=O)NCc2c(COC)ocn2)c[nH]n1 68872,C(=O)(C(C(=O)NC(C1CCCCC1)CNC(=O)Cc1cncn1C)OC)OC 68873,C(Cc1cn(-c2ccc(N)cc2)nn1)(CC(=O)O)NC(c1ccn(C(C)C)n1)=O 68874,c1(CC)ccc(OCCCNC(=O)NC2CC(NC)C2(C)C)cc1O 68875,c1(C(=O)NCc2cc(OC(CC)C)ncc2)c(C)cc(Br)cc1F 68876,C1(CNC(C(CC)C)=O)CCCCN(C(=O)CCc2ccc(O)cc2)C1 68877,c1(C(N(CCNC(COc2cn(C)nc2)=O)C2CC2)=O)cccc(C#N)c1Br 68878,c1(NC2(C)CC(NC(c3nc(CC)oc3)=O)C2)ncnc(C)c1F 68879,c1(CNC(C(Cc2ccccc2)OC)=O)cccc(NC(C2CC=CCO2)=O)c1 68880,C1(C(=O)NCCCCCCN(C(C(CC2CCC2)OC)=O)C)CC2CCC1CC2 68881,C12(C(N(CCC(=O)NCC)C)=O)CC1CN(C(=O)CCCOC(C)=O)C2 68882,C(CC(C)C)(C(=O)NCc1ncc(C(=O)NC(CO)CC(F)(F)F)cn1)OC 68883,CN1CCC(C(=O)N(C)CC2CC(F)(F)C2)(NC(=O)Cc2cnn(C)c2)C1 68884,Cc1[nH]nc(Cl)c1C(c1nnnn1C)NC(c1cncs1)C 68885,C1(NC(C2C(CC)CCC2)=O)CC12CCN(C(=O)CCc1ccccn1)C2 68886,N1(C(CC2CC(SC)C2)=O)CC2CCC1CC2NC(c1ncnc(C)c1C)=O 68887,C1(C(N2CCC2(C)C(=O)NC)=O)(CC)CCCN(C(c2ccsc2C)=O)C1 68888,c1(SCC(=O)NC2(CN(C(=O)COC)C)CC2)ccc(OCC2CCCC2)nc1 68889,N1(C(c2c(OC)scc2)=O)CC(C(=O)NCC2(C)CCC2)C(C(C)C)C1 68890,Cc1cnc(CCC(=O)NC(C2CCCN2C(c2nnn(C(C)C)n2)=O)(C)C)[nH]1 68891,c1(C(=O)NCC2(NC(C3N(C(CC)=O)CSC3)=O)CCC2)cnccc1Cl 68892,Cc1cc(-c2nc(C(=O)Nc3cnccc3Cl)cs2)cc2c1NC(=O)CC2 68893,c1(C(=O)NCc2ccc(C(N(C)Cc3nc(=O)o[nH]3)=O)s2)cc(C#N)cn1C 68894,c1(Sc2cc(-c3c(C4(NC(C)=O)CC4)cccc3)ncc2)ccc([N+](=O)[O-])cc1 68895,C(CC(=O)NC1CN(C(c2cncn2C)=O)CC1O)(C(F)(F)F)OC 68896,O=C(C1=C(Cl)CCC1)NC(Cc1ccco1)C(N1CC2(CCC2)C1)=O 68897,CC1CCCN(C(c2c[nH]nc2C(F)F)=O)C1CCNC(c1ccc(C#N)[nH]1)=O 68898,C1(C2CCCCO2)(C(N(C)CCO)=O)CCCO1 68899,C1(CC)CCCC1C(=O)NCc1ccc(C(=O)N(CCCF)CC)o1 68900,C1(C(=O)NCC(=O)NC(C)C)CCN(C(=O)COc2ccn(C)n2)C1C(C)C 68901,C(=O)(CCCC(C)c1ccccc1)N(CCNC(C1(OC)CCSCC1)=O)CC 68902,c1(OC)ccc(N2CCC(CNC(=O)C(c3cccnc3)OC)CC2)cc1 68903,N12CCOCC(C1)N(C(=O)C=Cc1ccccc1)C2=O.C(=O)(C=NOC)O.CCC=O 68904,c1(CC(=O)OCC2CC2c2ccccc2)ccc(N2CCCC2)cc1 68905,C1(CC(N2CCN(C(C(C)OC)=O)C(C)C2)=O)SC2=NCCN2C1=O 68906,c1(C(=O)NCCCN(C(CCc2onc(CC)n2)=O)C)ncnc(O)c1Br 68907,c1(CC(=O)NC2CCN(C(=O)COCc3cccnc3)CC2)ccc(F)cc1F 68908,C(=O)(CC(C)CC(=O)OC)N(C(CC)C(=O)NC1COCC1O)C1CC1 68909,c1(C2(C(N(CCNC(CC3(C(=O)OC)CC3)=O)C3CC3)=O)CC2)cccc(Cl)c1 68910,c1(N2C(C)CC(CNC(c3csc4ccccc34)=O)C2)ncnc2c1ncn2C 68911,C=CCC(CC(C)C)C(=O)N1CC2(C1)CN(C(C1CC(O)CN1C)=O)C2 68912,C12(C(N3C(CN(C)C(c4cnc(Br)s4)=O)CCC3)=O)CCC(C)(C1)OC2 68913,N1(C(C(CCSC)OC)=O)CCCC(C)C1CNC(=O)COC1CCCCC1 68914,c1(CN(CCc2ccccn2)CC2CCC(C)CC2)c(F)cccc1F 68915,N1(C(C2CCc3nnc(O)n3C2)=O)CCC2C(CCCN2C(C2CC(F)C2)=O)C1 68916,C(=O)(C(=O)N=c1ncn(-c2ccccc2)[nH]1)NC1C(C)C2CCC1C2 68917,Cc1ccc(CNC(=O)CC2(CNC(C3CCC3C)=O)CC2)cc1F 68918,C1(N(C(=O)C(C)OCC(F)(F)F)CC)CCCN(C(=O)Cc2nccn2C)CC1 68919,C12(NC(C(C)OC)=O)CCCC1N(C(=O)CCc1cn[nH]c1)CC2 68920,CN1CC(C)(C)CC1C(N1CC(CCO)(NC(=O)Cc2cc(F)cc(Cl)c2)C1)=O 68921,C=C(C)C1OCCC1CNC(=O)CN(C(=O)Cn1ccc(C)n1)C1CCC1 68922,Cc1ccc2c(C(=O)NCC(C)(C)NC(C34CCCC3CS4=O)=O)onc2c1 68923,c1(OC)cc(C(F)(F)F)ccc1-c1cc(CN2CCC(Br)CC2)ccn1 68924,C(=O)(C(F)(F)F)NCC(=O)NCCN(C(=O)Cc1cccn1C)CC 68925,C=CC1CN(C(=O)C(C)(F)C(=O)OC)CC1NC(=O)Cn1ncc(Br)c1C 68926,c1(C(=O)NCC2CCC(C)N(C(=O)CSC3CC3)C2)cccc2c1ncn2C 68927,C1(NC(CCc2onc(C)n2)=O)COCCN(C(=O)CC2COCCO2)C1 68928,N1(C(C2C(COC)CC2)=O)CCCC(O)(CNC(c2cn(C)nc2C(C)C)=O)C1 68929,O=C(NNc1cccc2c1CCCC2)c1cnc2ccccc2n1 68930,c1(C(N(CCCN(C(c2c(C)sc(O)n2)=O)C)C)=O)cnc(Cl)c(N)c1 68931,N1(C(C(C2CCCC2)OC)=O)CCCC2(C1)CN(C(=O)COC1CCCO1)C2 68932,C12(C(=O)NCC3(CCNC(C(C4CC4)OCC)=O)CC3)CC(C)(C1)OC2C 68933,C12(C(=O)NCCCNC(C3(S(N)(=O)=O)CCC3)=O)CCCC(=O)N1CCC2 68934,C1(NC(C2(CC(C)C)CC2)=O)CC2CCC(C1)N2C(C1CCCCC1(C)C)=O 68935,N1(C(C2N(CCC)CCC2)=O)CC(C)(C)CC1CNC(C1(SC)CC1)=O 68936,C1(CNC(CSCCOC)=O)CC2COCC2N1C(=O)CCCCN(C)C 68937,C1(NC(C(CC)NC(N)=O)=O)CC(OC)CN(C(=O)Cc2c(O)ncnc2O)C1 68938,C1(C(C(=O)N(CC(CC)O)CC)F)CCN(C(=O)CC2(CC)CCC2)C1 68939,Cc1cnc(NC(C2CCN(Cc3ccc(Cl)cn3)CC2O)=O)nc1Cl 68940,c1(CN=[N+]=[N-])ccc(CNC(C2(CCN)CCCC2)=O)cc1 68941,c1(CN2C(C)(C(=O)Nc3c(C(=O)OC)c(C)no3)CCC2)c(O)cc(O)cc1O 68942,CC(C)CC(CC(C)C)C(=O)N1CC2(CCCC2NC(c2ncc[nH]c2=O)=O)C1 68943,c1(SC)cc(C(=O)N(C)CC2CCCN(C(=O)CC3COCC3O)C2)nn1C 68944,c1(SCC(=O)NC(C2CCN(C(=O)C(CO)NC(N)=O)C2)C)nncn1C(C)C 68945,N1(CNC(C2C(=C)CC2)=O)CC(NC(C2(CCOC)CCC2)=O)CC1=O 68946,Cc1ccc(C(=O)NCCCOC2CCN(C(=O)C3=CCCO3)CC2)nc1F 68947,N1(C(C(C)(O)c2ccccc2)=O)CCC(CO)(NC(c2ccoc2)=O)C1 68948,C(=O)(CCCC(F)(F)F)N1CC(O)(CNC(C23CCCCC2C3(F)F)=O)C1 68949,N1(C(c2cn(CC)nn2)=O)CC2CCC1CN2C(=O)C(C)NC(C1CCC1)=O 68950,N1(C(c2snc(OC)c2I)=O)C(CO)CCCC1CO 68951,c1(C(=O)NCC(C(C)C)C(=O)N2CCOCC2CO)ncn2ccccc12 68952,c1(CN(C(C=CC(CC)=CC)=O)CC(F)Cl)cccc2c1CCC2 68953,c1(OC)ncc(C(=O)NC2CCC(NC(c3scc(C)c3Cl)=O)C2)cc1Br 68954,N1(C(CC(=O)N(C)C)=O)CC=C(CC(=O)N2CCOCC(C)(C)C2)CC1 68955,N1(C(C=Cc2c(C)noc2C)=O)CC2CC(O)C1C2NC(=O)CC(C)C(F)F 68956,C=CC(F)(F)C(=O)NC(CNC(=O)C(CC)=CCCC)C1CCC1 68957,C1(O)(CC(=O)N(C2(C(=O)NCC3(CC=C)CC3)CC2)C)CCCC1 68958,C1(NC(C2(OC)CC(CF)C2)=O)CC2CC(NC(=O)Cc3cccs3)CC12 68959,C=CCCC(F)(F)C(=O)NCCOCCN(C)C(c1cn2cc(C)nc2s1)=O 68960,CC1c2nncn2CCN1C(=O)C(c1ccccc1)(C)NC(=O)C(F)C1CCC1 68961,C1(NC(c2n(CC)nc(C)c2)=O)CCN(C(C23CC(C)(CO2)C3)=O)C12CCC2 68962,C=CCCCCCCC(=O)NC1(CNC(c2cc(C3CC3)ccn2)=O)CCOC1 68963,N1(C(c2cc(C(F)(F)F)c[nH]2)=O)CC2(C1)CN(C(C1(N3CCCC3)CC1)=O)C2 68964,C(C(C)(C)CCNC(C1CCCCN1C(c1sc(C)nc1C)=O)=O)OC 68965,c1(CC)cccc(N(C)C(C2COCC2NC(=O)CCc2ccn(C)c2)=O)c1 68966,N1(CCC)CCCC(C(=O)NC(C)(C)C(C)NC(=O)CC2CC(C(F)F)C2)C1 68967,S(=O)(=O)(c1c[nH]c(=NCCC#N)cc1C)NC(CC)C(C)O 68968,CN1CC2CCCN(C(=O)CCn3cc(CCCN4CCOCC4)nn3)C2C1 68969,C1(C(=O)NCC(C(C)C)NC(=O)CCCC2CC2)CCC(C(=O)N(C)C)CC1 68970,CC(C)(C)C#CC(=O)NCC(CC(=O)NCC1OC(=O)CC1(C)C)OC 68971,c1(OCc2scc(C(=O)NC34CC(C)C3C4)n2)ccc2c(c1)CN=S2(C)=O 68972,c1(C(N2CCC(O)(CNC(C3CCCN(C(C)=O)C3)=O)C2)=O)c(C)cc(C)nc1O 68973,C1(C(=O)N(C)CCN(C(=O)C(C)(C)C2CCOCC2)C)(OC)CCC(C)C1 68974,C12(CNC(C(N3CCCCCC3)C)=O)CCC(CC1)N2C(=O)CC1CC1(C)C 68975,c1(CC(=O)NC(CN(C(c2csc(C3CC3)n2)=O)CC)C)ccccc1C 68976,C1(CNC(C(C(C)C)O)=O)CCCC2CN(C(=O)Cc3ccnc(F)c3F)CC12 68977,N1(C(C=Cc2nnn(C)n2)=O)CCOCC(NC(C2C3CCCCCC23)=O)C1 68978,c1(CC(C)C)cccc(C(N2CCC(C(C)(C)NC(c3c[nH]c(Br)c3)=O)C2)=O)c1 68979,C(C)(C)(CCCNC(=O)C=CC=C(Cl)Cl)NC(C(CC)n1ccnc1)=O 68980,C1(C)(C(=O)NC(C2(CS(C)(=O)=O)COC2)C)CCCN(C(=O)OC(C)(C)C)C1 68981,C1(NC(c2ccc(C(F)(F)F)cn2)=O)C2CC1N(C(=O)CCC1CC1(Cl)Cl)C2 68982,Cc1cc(CN(C)CC2CCCC(c3ccccc3)C2)ccc1F 68983,c1(C(=O)NCC2CCCN(C(CNC(CC)=O)=O)C2)c(F)c(F)cc(F)c1F 68984,C(CC(C)C)(CC(C)C)NC(CCNC(CN(C(COC)=O)C)=O)=O 68985,C(=O)(C(CC(C)C)C(N)=O)NC1N(C(C(CC#C)C2CC2)=O)CCOC1C 68986,N1(C(CSCC(=O)OC)=O)CCCC(CCNC(c2cccn2C)=O)C1 68987,N1(C(Cc2cc(C)nn2C)=O)CCC2CN(C(=O)CCS(N)(=O)=O)C(C)C12 68988,c1(NCc2n(C)nnc2Br)ccc2c(c1)C(C)(C)CC2(C)C 68989,CCCCCCC(C)CC(=O)NC1(C)CN(C(c2c[nH]nc2CC)=O)C1 68990,C1(C(N(C(C)C(N)=O)C)=O)CC12CCN(C(=O)Cn1cnnn1)CC2 68991,CC(C)(C)CCC(=O)NC1(CO)CCN(C(=O)CC2COCC2O)CC1 68992,c1(C(=O)NCC2CC(NC(C(C)C3CCCO3)=O)C2)cc(Br)cs1 68993,CC(c1ccc(F)cc1F)=CC(=O)N(CCCCNC(C1CC2CC2C1)=O)C 68994,C#CC1(C(N2CCC(C(C)O)CC2)=O)CCN(C(c2cc(Cl)c[nH]2)=O)C1 68995,C(CN=c1cc(Cl)nc(C2CN(C)C(=O)C2)[nH]1)OC12CC(c3ccccc3)(C1)C2 68996,c1(C(CC)=O)cccc(NC(N2CCCC(CN(C)C)C2)=O)c1 68997,c1(C(=O)NC(CC)CNC(=O)C(C(C)(C)C)NC(C)=O)cccc2c1OCC2 68998,CCC(C)C(CC(=O)N(C1CCOCC1C)C)NC(c1conc1C)=O 68999,N1(C(C(C(C)(C)C)NC(CSCCCC)=O)=O)CCC2(CC1)CC2CO 69000,c1(-n2cc(C3N(C(CS(C)(=O)=O)=O)CCCC3)nn2)cccc2c1CCCC2 69001,C1(CNC(=O)C2CC2)CC2(CCN(C(=O)CCOc3ccccc3)C2)CO1 69002,C=CCC(C(=O)NCC(CC)NC(C1(c2ccc(F)cc2Cl)CC1)=O)C(C)C 69003,N1(C(C=CC)=O)CCC(O)(C(C)NC(c2c[nH]c(C)cc2=O)=O)CC1 69004,C(C(O)C(F)(F)F)N(C(C1(NC(c2cc(C)[nH]c2)=O)CCSC1)=O)C 69005,c1(OCC)cc(C(=O)NCC(CNC(=O)CCC(C)OC)CO)ccc1C 69006,CC(CC(=O)NCCCN1CCN(C(=O)CN2CCC(C)(O)C2)CC1)P(C)(C)=O 69007,C(=O)(CCCCCCNC(C(F)(F)F)C1CCCC1)OC(C)(C)C 69008,C1(NC(c2c(CC)nns2)=O)CCCC12CN(C(c1cc(O)c(F)cc1N)=O)C2 69009,C(=O)(C(CNC(C1CC1C(F)(F)F)=O)CC(C)C)NC(c1nc[nH]n1)CC 69010,c1(-c2c(C(=O)NCC#CC)cccc2)ccc(C(=O)NC(C)C)c(F)c1 69011,N1(C(C(C(=O)OCC)SC)=O)CC(n2cc(CC3OCCO3)nn2)C2(CCC2)C1 69012,Cc1nc(O)[nH]c1C(=O)N(C(C)CN(C(=O)Cc1ccsc1C)C)C 69013,CC1CN(C(=O)Cc2ccccc2O)CC1CNC(c1ncc(C(F)(F)F)s1)=O 69014,c1(C(C=O)N(N2CCCC2)CC(C)(C)CC)ccc([Si](C)(C)C)s1.CC 69015,C1(C(=O)NC(C)CCCNC(=O)C(C)OCC2CC2)C(C(F)(F)F)C1[N+](=O)[O-] 69016,N1(C(C2N(C(c3c(CC)nn[nH]3)=O)CCC2)=O)CCC(C)(C2CC2)C1 69017,C=CC(C)(O)CC(=O)NC(CNC(=O)C(C)Sc1ccccn1)CC 69018,N1(C(CNC(=O)OC)=O)CCN(C(c2cn3ccncc3n2)=O)CC(O)C1 69019,CCN=C(NCCC1CC1)N1CCC2C(CCCN2C2CC2)C1 69020,C1(C(=O)Oc2cccc(N(CC)CC)c2)CC2CCCC(C1)C2 69021,C(C)(C)(CCC(=O)N1CCC(C)(C(=O)NCC2(C)CCC2)C1)N(C)C 69022,C=CC1COCC1NC(C1CSCN1C(=O)C(C(=O)OC)OC)=O 69023,C1(NC(C=Cc2scc(C)n2)=O)CCCC12CCN(C(=O)CCc1cnco1)C2 69024,N1(C(=O)OC(C)(C)C)CCC2CC12CC(N1CCN(c2ccsc2C#N)CC1)=O 69025,c1(C(C)=O)ccc(C(=O)NCC2CCCN2C(=O)Cc2cc(C)no2)cc1 69026,C1(C(=O)NCC2CC(NC(C(C)(C(C)C)OC)=O)C2)CCc2ncnc(C)c2C1 69027,C1(CNC(c2n(CC)ccn2)=O)CC(C)N(C(c2scnc2Cl)=O)C1 69028,C1(C(=O)NC2C(C=C)CN(C(=O)CC(=C)C)C2)CCCCCS1(=O)=O 69029,C1(CC)CC(N=c2cc(C)nc(N3CC=CCC(C)(C)C3)[nH]2)C1 69030,N1(C(c2c(C)cn(C)n2)=O)C2CCC(C2)C1CC(=O)NCCOCC(F)F 69031,c12ccc(Cl)cc1NC2=O.Cn1cc(-c2cn(CO)nn2)c(C2CC2)n1.C(C)(C)C 69032,c1(C(=O)NCCC(=C)CNC(C2OCCC2CC)=O)cccc2c(C)[nH]nc12 69033,C1(N(C(=O)CC2(O)CCC2)CC)CCCN(C(c2ccc(Br)nc2C)=O)CC1 69034,C(=O)(C1=CCCCO1)N(C1CN(C(CCC=CC)=O)CC1O)C 69035,C1(OC)CN(C(C23CC(C2)C3)=O)CCC1NC(c1cc(B(O)O)co1)=O 69036,N1(C(C(=O)N(C)CCC2CC2)=O)CCC(CCO)(CO)C1 69037,CCCC(C(O)C(=O)NC1CC(F)C1)NC(=O)C(CC)(CC)CC 69038,N1(CCNC(C2(NC(C3CC=CCC3)=O)CCSC2)=O)CCOC1=O 69039,C12(C(N3CC(C)C(CCNC(=O)Cc4cnc[nH]4)C3)=O)CCC(CF)(C1)OC2 69040,C1(CC(C)NC(c2c(CC)onc2)=O)CCN(C(=O)CC(C)C2CCCC2)CC1 69041,N1(C(C=Cc2c(C)n(C)nc2)=O)CCCC(NC(=O)Cc2cncn2C)C(F)C1 69042,C1(C)(NC(=O)C(C2(O)CN(C(c3cc(COC)[nH]n3)=O)C2)F)CCCCCC1 69043,c1(N(C)C)ncc(C(=O)NCC(C2CCCC2)NC(=O)CC2CC2(Cl)Cl)o1 69044,C1(CC(=O)NCCCOC=C)CCN(Cc2cn(C)nn2)C1 69045,CCCCCCC(=O)NCC(C(C)C)NC(=O)Cn1cc(C2CC2)nn1 69046,c1(C(=O)NCCCC(C)(C)NC(c2cc(CC)[nH]n2)=O)c[nH]c2cccc(Cl)c12 69047,Cc1ncc(CC(=O)NC2CC2NC(c2sccc2SC(F)F)=O)s1 69048,c1(N(C(=O)NC2CC3CNC(C2)C3)CC2CC2)ccc(F)c(C(F)(F)F)c1 69049,C1(CNC(c2c(C)n[nH]c2C)=O)CCN(C(=O)CCSc2nccn2C)CC1C 69050,C1(CC(N2C(C)C(NC(=O)C(F)(F)C3CC3)CC2)=O)CSc2ccccc2O1 69051,N1(C(C(CCC)CC(C)C)=O)CCC(C2(O)CCN(C(=O)CNC(=O)NC)C2)CC1 69052,C1(COC)CCCCCN1C(C(=O)NC1CC1)C1CC1(Br)Br 69053,c1(C(N2C(C(=O)NCc3ccc(C#C)cc3)CC(F)C2)=O)ccc2c(c1)CCO2 69054,N1(C(C(C)NC(=O)NC)=O)CCCCC(NC(=O)CN(c2ccc(Cl)cc2)C)C1 69055,C1(COC)CC(C)(C)CN1OC(=O)C(C)CCOC1CCC1 69056,C(CCC(C)CC(=O)N1CC(NC(C2(C)CCC2)=O)C2CC2C1)=C(C)C 69057,C1(CNC(c2c(C(C)=O)ccs2)=O)CN(C(=O)C(c2ccccc2Cl)O)CC1C 69058,C1(Cc2cn(CC)nn2)CN(C(=O)NC2(c3ccccc3C)CC2)CCO1 69059,N1(C(Cc2c(SC)ccc(F)c2)=O)CC2(CCCC(CNC(=O)OC(C)(C)C)O2)C1 69060,C1(NC(C2(C)CC(C)(C)C2)=O)CCN(C(=O)CC2CC(F)(F)C2)CC1O 69061,CSC1=C(C(=O)NC2CN(C(=O)Cc3nonc3C)CC(C)(C)C2)CCCC1 69062,c1(N2CCC(CC=C)(NC(C3NC(=O)CC3C)=O)C2)nc(Cl)nc(C)c1[N+](=O)[O-] 69063,C1(C(C)O)COCCN1C(C1CCOC1CNC(=O)CC1CCN(C)CC1)=O 69064,C1(c2c(OC)cccc2)C(NC(=O)Cc2cccc(C3CC3)c2)CC(=O)N1C 69065,N1(C(C(CCSC)OC)=O)CC(NC(=O)CNC(c2cscn2)=O)CC1(C)C 69066,c1(CCCC(=O)NCC2(O)CCN(C(=O)C3CC3)CC2)c[nH]c2ccccc12 69067,C1(NC(C(N)=O)=O)CN(C(c2cncnc2)=O)C2(CCCOC2)C1 69068,C(=O)(C=C1SCC(=O)N1C)NC12CCCN(C(CC(C)n3cccn3)=O)CC1C2 69069,C(=O)(C(C)(C)CC(F)F)N(C(CNC(CCCC(=O)NCCC)=O)C1CC1)C 69070,C1(NC(C(C)(C)Cc2cccc(Cl)c2)=O)CC2CC(C1)N(C(=O)CCC1CC1)C2 69071,c1(CC)ccc(C(=O)O)cc1.C12(CCOC1)N(C(COC)=O)C2 69072,c1(C(=O)NC2(CNC(=O)CC3CCC3C)CC(OC)C2)nccc2ccn(C)c12 69073,N1(C(=O)C2CC2)CCOC(C2CC2)CC1.C12(CC(O)C1)NC(=O)C=CC(=O)N2 69074,C1(O)(CNC(CCC2C(C)C2)=O)CCN(C(c2ccc(=N)[nH]c2Cl)=O)CC1 69075,Cc1cc(=NC2CC(C)N(C(=O)CCCN(C)C)C2)[nH]c(C(C)(C)C)n1 69076,CC1(C)CN(C(C23CC2CCN3C(c2n[nH]c(=N)[nH]2)=O)=O)CCC1O 69077,C1(C(N(C2CCN(C(c3cc(CC(C)C)on3)=O)C2)CC)=O)CCCC1COC 69078,CN(C)S(=O)(=O)N1CCC(C(=O)NC2C=CCN(C(=O)C3=CCCC3)C2)CC1 69079,c1(NC(C2C3CN(C(CCc4c(OC)cccn4)=O)CC32)=O)ccc(Cl)c(F)c1 69080,c1(C(N2C(CCC(N3CCC(=O)NCC3)=O)CCC2)=O)ccc2c(c1)CCCO2 69081,C(C(C(C)C(C)C)NC(C1(C(F)(F)F)CC(F)(F)C1)=O)NC(CCOCC#C)=O 69082,CCC(C)CCC(=O)NCC(C)C(=O)NC1(CC)CCOCC1 69083,c1(NC(C2(C#N)CCSCC2)=O)cccc2c1C1CCC2O1 69084,C(=O)(C1CCc2ccccc21)N1CCC(C)(CNC(CCC(C)(C)O)=O)CC1 69085,C12(C(=O)NCC(C)N(CC)CC)CCCC1CN(C(=O)CCC(C)(C)F)C2 69086,Cc1cccnc1C(=O)NC(c1ccccc1F)CNC(=O)C=Cc1cocn1 69087,N1(C(CC2OCCN(C(C3C(C)C3C)=O)C2)=O)CC2CCC1C(CO)C2 69088,c1(CNC(C(=C)COc2ccccc2)=O)ncccc1OC(F)F 69089,C1(C(=O)NC2(CN(C)C(C34CC(CC(F)F)(C3)C4)=O)CC2)CCOCC1(C)C 69090,N1(C(CCC2N(C(C3CCCCCC3)=O)CCC2)=O)CCC2(CCOC2)C1 69091,Cc1nccc(C(=O)N(C2CCN(C(C3CCCC34CCC4)=O)C2)C)c1N 69092,c1(CN2CCC(C(N3CC4(CCC4)C3)=O)C2)c(O)cccc1F 69093,N#CCCCCC(=O)NC1CCN(C(C23CC(c4ccccc4)(C2)C3)=O)C1 69094,C#CCC(CC(F)F)NC(c1cn(CCNC(=O)OC(C)(C)C)nn1)=O 69095,C1(CCNC(C2N(CC)CC2)=O)CCCN(C(=O)C(C)(C)c2ccccc2)CC1 69096,c1(C(=O)NCC2=CCCN(C(C3(NC(C)=O)CCC3)=O)C2)cn2ncccc2n1 69097,c1(C(N2CCC(C(=O)NC3(C)CCCC3(F)F)C2(C)C)=O)cc(C#N)ccc1N 69098,CON=Cc1ccc(C(=O)NC(C2CCOC2)CNC(C2(C(F)F)CC2)=O)cc1 69099,c1(C(N(CC(c2ccccc2)OC)C)=O)ccc(C)c(Br)c1F 69100,c1(C(=O)NC(C(C)C)(C)CNC(c2ccoc2Cl)=O)ccc(=O)n(C2CC2)c1 69101,Cc1[nH]c2ccc(C(=O)NCC(C)(C)NC(c3ccc([N+](=O)[O-])o3)=O)cc2c1C 69102,c1(C(C)C(=O)NC2CCC(NC(=O)CSC(C)(C)C)C2)ccc2c(c1)OCO2 69103,c1(C(N2CCC(O)(CNC(Cc3nn(C)c(Cl)c3)=O)C2)=O)cc(N)cnc1Cl 69104,CC1CCCc2nc(C(=O)NCC3(F)CC(NC(=O)C(C)(C)CC4CC4)C3)cn21 69105,C1(C(=O)NC2COCCN(C(CCC(=C)Cl)=O)C2)CC(C2CCCC2)C1 69106,N1(C(C2CC(C(F)(F)F)(OC)C2)=O)CCC2(NC(c3cccc(=O)o3)=O)CC2C1 69107,C1(C(=O)NC(CC)CN(C(=O)CCC2(C)CC2)C)CCN(c2ncccn2)C1 69108,C1(CC(N2CCC(N(C(=O)CCOC3CC3)CC)C2)=O)CCc2ccccc2C1=O 69109,C(=O)(CCCCCC#N)N1C(C)CC(CCNC(=O)CCC(N)=O)CC1 69110,C(=O)(CCCN=c1nccc[nH]1)N(C)CC1CN(C(C2(N=[N+]=[N-])CC2)=O)CCO1 69111,Cc1ncnc(C(=O)NC2CC(O)(CNC(C3CC3c3cnc[nH]3)=O)C2)c1C 69112,C(C(=O)NCCC(C)C(F)(F)F)(C(C)(C)C)NC(C(OCC)OCC)=O 69113,c1(C(=O)NCC(NOCC)=O)cccnc1CNC(=O)Cc1cccn1C 69114,Cc1cc2ncc(C(N3CCC(C)C(NC(c4nocc4Cl)=O)C3)=O)cn2n1 69115,C(=O)(N1CC(O)CCO1)c1c(CNC(C2(C)COC(=O)N2)=O)n[nH]c1 69116,c1(C(C(=O)NC2C(NC(=O)CCCC3CC3)CCC2)N2CCC2)ccc(Cl)cc1 69117,C(N=c1ccc(C#N)c[nH]1)C1C(NC(COC2C(CC)CCCC2)=O)CCC1 69118,c1(C(N2C(CNC(CC3ON=C(C)C3)=O)COCC2)=O)cc(C)cc2ccoc12 69119,N#Cc1ccc(C(=O)NCCCCCNC(c2cnc(Br)s2)=O)cc1O 69120,c1(OCC(=O)NC(CCCC)CNC(=O)CC2COC(=O)N2)cc(Cl)ccc1C 69121,C(=O)(C(CC1CCCO1)C(F)(F)F)NC1CN(C(C(C)=CC)=O)CC1SC 69122,c1(Cc2nnnn2CCCF)ccc2c(c1)OCC2.N(CP(C)(C)=O)C(CC)CC 69123,CC1CC=C(C(=O)NCC2CCCN2c2nn(C)cc2[N+](=O)[O-])CC1 69124,c1(NCC)ccc(F)c(C(=O)NC(CNC(=O)CCC2CC2(Cl)Cl)CC)c1 69125,c1(C(=O)NC(CC)CNC(=O)CC2CCCC3(CC3)C2)c(F)ccc(CC)c1F 69126,C(C(C(C)C)NC(C1CCC1)=O)OCCSC.C1(=O)CCN1 69127,C1(C(=O)NC(CNC(c2c(OC)cc(C)cn2)=O)C(C)C)CCCC1S(C)(=O)=O 69128,c1(C(=O)NC2CN(C(C3C(C)CCC3)=O)C2)nn(C)cc1N 69129,N1(C(CCSCC)=O)CCN(C(c2cnn(CC)c2)=O)CC1COC 69130,C1(NC(=O)CC=C(Cl)Cl)CCC2CN(c3nc(C4CCCCC4)ns3)CCC2C1 69131,c1(C(C)(C)C)cc(Br)cc(Br)c1OC(c1n[nH]cc1C=O)=O 69132,C=CCCCC(C(=O)NCCc1ocnc1CO)NC(=O)CN1CCN(C)CC1 69133,Cc1ccc(NC(=O)COC2CCN(C(=O)CNc3ncccn3)C2)cc1C 69134,c1(C(=O)OCC)cc2n(n1)CCN(C(c1cnc3ccc(Cl)nn13)=O)C2 69135,C1(C(=O)NCC(CC)(C)COC)CN(C(=O)Cc2cc(C)no2)CC(C)(C)C1 69136,N1(CC)CCOC(C(=O)NCCC2(OCC)CN(C(=O)C(CCSC)OC)C2)C1 69137,S(=O)(=O)(c1cnc(N2CC(CCO)C2)c(Cl)c1)NC1C(C(C)C)C2CCC1C2 69138,c1(C(C)C)c(C(N2CCCC(NC(=O)C=CCF)C2)=O)cnn1CCO 69139,C1(NC(N(CCN(C)C)CC2CCC(Br)C2)=O)CCCCCC1 69140,CC1(C)CCN(C(=O)CC2CCSC2)C1CC(=O)NC1(C)CC2(CC2)C1 69141,Cc1cc(C)c(CC(N2CC(O)(CNC(=O)CCC3CCCN3C)C2)=O)c(C)c1 69142,C1(NC(CCc2ccc(OC)cc2)=O)CC2CC1CN(C(c1ccsc1)=O)C2 69143,N1(C(C(CCOC)C)=O)CCC(CNC(=O)Cc2nc[nH]n2)(OC)CC1 69144,Cc1nc(C)c(C(=O)NC(C2CN(C(c3cocc3C)=O)C2)C)[nH]1 69145,N1(C(C(=O)N(C)Cc2c(Br)ccc(OC)c2)=O)CC2CN(C)CC2(C)C1 69146,c1(C(N2C(C)(CC(N3CC(F)(CO)C3)=O)CC2)=O)ccc(=N)[nH]c1 69147,c1(C(=O)Oc2cncc(-c3ccccc3OC(F)F)c2)cnc(O)nc1O 69148,C(C(CC1CC1)C(=O)NCC1CC=CC1)NC(CC1N(C)CCC1)=O 69149,CC1(CC(F)(F)F)CN(C(=O)C(=O)NCCCn2ccnc2)C1 69150,C1(NC(c2cnnc(C)c2C)=O)CC2CCC1CN2C(C1CCOC(=O)CC1)=O 69151,Cc1ccc(Cl)c(C(=O)NC2(C)CC(NC(=O)COc3ccc(F)cc3O)C2)c1 69152,c1(CC)nc2sc(C)cn2c1C(=O)NCC1(O)CCCCCC1 69153,N1(c2n(CC)c(-c3ccc4c(c3)OCO4)nn2)CC(CCO)Oc2ccccc21 69154,N#Cc1cccc(F)c1CC(N1CC2CC(NC(=O)C#CC3CCC3)C1C2)=O 69155,C1(C(N2CCC(C(C)NC(c3cnc(C(F)(F)F)s3)=O)C2)=O)CCS(=O)(=O)N1 69156,C1(CC)CN(C(=O)CCOCC2CC2)CCC1NC(=O)CC1CCC=CCC1 69157,Cc1ccc(S(=O)(=O)NC(c2cc(C)c3ncccc3c2)=O)c(F)c1F 69158,N1(C(C2CN(CC)C(=O)C2)=O)CC(C(=O)NCC(CSC)OC)CC12CCC2 69159,N1(C(C2(C)CCCO2)=O)CC2(CC(CC(N3CCCC3CCCO)=O)C2)C1 69160,c1(C(=O)NC(CNC(C(n2ncc(C)c2)C)=O)C(C)(C)C)cc(F)c(O)c(F)c1 69161,C1(CCCC)CCC(C(=O)NCC(O)CNC(C2(Cl)CC2(F)F)=O)CC1 69162,C(C)(C)(C(=O)N(C)CC1(CNC(C2CSCCS2)=O)CC1)OCC 69163,C(C)(C(=O)OC(C)(C)C)(C(=O)NC1CC(NC(C2CCC2)=O)C1)OC 69164,c1(C(C)(C)C)nocc1C(=O)NC1COCC1NC(=O)C(F)CC1CCCC1 69165,c1(OC)ccc(Cl)cc1COC(N1CC(OC(c2cc(C3CCC3)on2)=O)C1)=O 69166,Cc1nc2ccccc2nc1NC(c1ccc(CN2CCOC(C)(C)C2)cc1)=O 69167,C(=O)(C(C)CC(F)(F)F)NC1(CNC(c2ccnc(CO)c2)=O)CC(OC)C1 69168,c1(C(C)=O)cnc(NC(=O)CC2CN(C(=O)C3=COCCC3)CCO2)nc1C 69169,N1(C(c2cc(OCC)no2)=O)CC(N=c2ccn3ccnc3[nH]2)CC2(CCC2)C1 69170,C1(c2nnnn2CCNCCCC(C)(C)C)(CCO)CCCC(C(F)(F)F)C1 69171,c1(C(=O)NC2C(CNC(c3ncc(NC)nc3)=O)C2)ccc(F)c(Cl)c1F 69172,C1(C(=O)OC(C)(C)C)CCCC(OCC(N2CCCC(CC#N)C2)=O)C1 69173,C(=O)(CCC(C)(C)C#N)NC(C(=O)NC(COC)C(C)C)Cc1ccc(C)cc1 69174,C(CC1=CCOCC1)NC(C1C(NC(=O)CCOC2CCCC2)CC1)=O 69175,Cc1ccn2cc(C(=O)NC3CN(C(C4CCC(=C(F)F)C4)=O)CC3(C)C)nc2c1 69176,N1(C(CC2(C)CC2)=O)CC2CCCC(C1)N2C(=O)CC1CCCCCC1(F)F 69177,CC1CS(=O)(=O)CC(C)N1C(C1SCCS1)=O 69178,C1(CNC(CCC=C)=O)CCC2(CCC2)C1NC(=O)CCN1CCOC1=O 69179,C(=O)(C1=CCOCC1)NCc1cc(C(N(C2CCCC2(F)F)C)=O)on1 69180,c1(C(N2CCCC(OC3CC3)C2)C(=O)NC2CCC2)ncccc1F 69181,C1(CC)CN(c2nnc(CSCCO)n2CC(=O)NC)CC(C)O1 69182,c1(C(N2CC3N(C(c4ccc(F)c(F)c4Cl)=O)C3C2)=O)cc(Cl)c2cn[nH]c2c1 69183,c1(OCCNc2c(NC(CC)=O)c(=O)c2=O)c(F)cccc1Cl.C1CN1.CCNCC 69184,c1(CCC)ccccc1C(=O)NCC(C(C)C)NC(=O)C(N1CCN(C)CC1)C 69185,c1(CC(=O)NC2CCN(C(=O)Cc3ccccc3)C2)csc2ccc(Cl)cc12 69186,N(C(=NCCn1cccn1)NCc1ncccc1O)CC1N(CC)CCC1 69187,c1(OCCC)c(F)cc(-c2nc(C(=O)N(c3ncccn3)CC)cs2)cc1F 69188,c1(CN(C)C(N2CCCC(C(=O)OC(C)(C)C)(C(F)F)C2)=O)cc(F)cc(F)c1F 69189,N1(C(=O)NCCCc2c(C)cccn2)CCN2CCOCC2C1 69190,C(=O)(C(=O)CC(C)CC)NCC1(CC(=O)N(C2CC(=C)C2)C)CC1 69191,Cn1c(C(N2CCC(O)(CNC(=O)CC3CCCOC3)CC2)=O)cc2sccc12 69192,N1(C(=O)C=Cc2ncc[nH]2)CCC2OCCN(C(C3CCC(F)CC3)=O)C2C1 69193,c1(C(=O)NC(C(C)NC(=O)COCCN(C)C)(C)C)ccnc2ccc(Cl)cc12 69194,C(=O)(C(CC(C)C)C(N)=O)NC1CC2N(Cc3n(CCC)c(C)nn3)C(CC2)C1 69195,N(C1CCCc2n[nH]cc21)C(C1C(n2cc(CCCCCCCN)nn2)CO1)C 69196,c1(C(=O)NCC(CO)NC(c2cnc(Cl)s2)=O)cccc2nccnc12 69197,N1(C(c2ccc(Cl)s2)=O)CC(CNC(C23COCC2C3)=O)C2(CCC2)C1 69198,Cc1nc(-c2cn(CC(C3CN(C(C4(C)CC4F)=O)C3)F)nn2)sc1C 69199,C1(NC(c2n[nH]c(=N)s2)=O)CCCC2CN(C(C3CCCC(F)(F)CC3)=O)CC12 69200,O=C(N1CC(n2cc(C3CCCCO3)nn2)CO1)c1cncc(C2CC2)c1 69201,Cc1nc(O)ccc1C(N1CCC(C(=O)NCCc2c(C)n[nH]c2C)C1)=O 69202,c1(CC=C)ccccc1C(=O)NCCCCCNC(=O)C(COC)N(C)C 69203,C=CCC(CNC(=O)CN(C)C(N)=O)C(=O)NCc1nnn(C)c1C 69204,C1(C(C(=O)NC2(c3ncc[nH]3)CC2)NC(c2ccc(CO)s2)=O)CCCCC1 69205,Cc1cc(C(=O)NC23CC(C2)N(C(c2cccnc2SC(F)F)=O)C3)cc(Cl)c1 69206,C1(NC(c2n(C)c(S)nn2)=O)CCCC(C(N2CC(CC(N)=O)C2)=O)CC1 69207,C1(C(N2CC(NC(=O)C(C)(C)C)CC(C)(C)C2)=O)Cc2cc(Br)ccc2O1 69208,N1(C(CSC)=O)CC(NC(=O)CSc2cccc(Br)c2)CCC1C 69209,c1(CC)ccc(N(C(c2c[nH]nc2CCNC(C2CC(C)(O)C2)=O)=O)CC)cc1 69210,CC(C)(C)C(C(=O)NCc1ncoc1CCNC(c1n[nH]cc1Cl)=O)NC(N)=O 69211,N1(C(c2c(C)ccnc2C)=O)CC2CCC(C1)C(NC(c1ccnnc1C)=O)C2 69212,N1(C(C(c2c(C)cccn2)(F)F)=O)CC2(CCC2NC(C2CNC(=O)C2)=O)C1 69213,CCC(CC)C(=O)NC(C)(CNC(c1cccc(C(=O)N(C)C)c1)=O)C(C)C 69214,C1(CC)CN(C)CCCN1C(C1CC2CC1CN(C(c1cc(C3CC3)on1)=O)C2)=O 69215,C1(N(C(C2CCCOC2)C(=O)NC)C)CCC(OC)CC1 69216,C(C)(C)(CCCC(=O)N(C)CC1CCCC1O)NC(c1c(C)cc(O)nc1)=O 69217,C(=O)(C(O)CC(C)C)NC(CCN(C(c1cc(OC)ns1)=O)C)C(C)C 69218,C1(NC(c2cnn(C(C)C)n2)=O)CC(C(=O)NCc2snnc2C)C12CCC2 69219,N1(Cc2c(C(=O)OCC)n[nH]c2)CC2CN(C(c3cc(B(O)O)co3)=O)CC12 69220,Cc1ccccc1C(C)C(=O)NCC(C)CN(C(=O)C(C1CCC1)C1CCC1)C 69221,Cc1cc(-n2cccn2)nc(=NCC2C(C)CCCN2C(=O)C(C)CN(C)C)[nH]1 69222,c1(C(N(CC(C)NC(=O)CCCC#N)C)=O)ccc(-n2cccn2)cc1 69223,c1(N2CC(C)=C(C)C2)ccc(S(=O)(=O)NCC2Cc3ccccc3CO2)cc1Cl 69224,c1(C(=O)NC(CC(C)NC(=O)CC2CCN(C)C2=O)C)cc(N)c(F)c(F)c1F 69225,c1(OC)cc(OC)c(C(=O)NCC2CCC2NC(c2nncs2)=O)cc1OC 69226,Cc1nc(-c2ccc(CN(c3ccccc3)C)cc2)ccc1C(=O)NC1CNC1 69227,N1(c2n(CC(=C)C)c(-c3nccn3C)nn2)CC(C(N)=O)OC(C)C1 69228,C(=O)(C(C)S(=O)(=O)C(C)C)NCC(C)(C1CCC1)NC(C1CCC(CC)O1)=O 69229,c1(C(C)=O)c(Cl)nc[nH]c1=NCC1(F)CC(NC(c2coc(SC)c2)=O)C1 69230,c1(C(=O)NC2(C)CCN(C(c3ccc(N)cc3Cl)=O)C2)ccn2nnnc2c1 69231,C#CC(C(C)OC)NC(C1(C(C)NC(C2CC(CC)C2)=O)CC1)=O 69232,CC(CCC#N)(c1nnnn1CSc1ccccc1)NCCc1cccnc1 69233,Cc1nn(CC(=O)NC(C)C(C)NC(=O)C(CO)c2ccccc2)cc1Cl 69234,C1(OC)CN(CC2CC3CC2C2CC32)C2(CCOCC2)C1 69235,c1(C(N2CC3CC(C2)N3C(c2cnc(Cl)nc2)=O)=O)ccc2nc(Br)sc2c1 69236,N1(C(C23OCC(C(C)C)(C2)C3)=O)CCC(C)(NC(=O)CCS(N)(=O)=O)CC1 69237,Cc1cc(C)c(C(=O)NCC2C(C)CCN2C(=O)CCc2csc(=N)[nH]2)o1 69238,c1(C(N2CC(CC(C)NC(=O)CC3CCC3)C2)=O)ccn(CCO)c(=O)c1 69239,C1(O)(CN(C)C(C2C(C)(C)C2(F)F)=O)CCN(C(C2(c3cc[nH]n3)CC2)=O)C1 69240,C(C)(C(CC(=O)NC(c1cc(C)no1)(C)C)NC(C1C=CCS1)=O)OC 69241,C(N=c1[nH]c(N2CCC(S(N)(=O)=O)CC2)nc2c1SCC2)C1(SCC)CC1 69242,N1(C(C(CO)N(C(N)=O)C2CC2)=O)CC2OCCCC2(CSc2ccccc2)C1 69243,N1(C(C2C3CC(=O)CC32)=O)CC2C=CC1C(C(=O)NCC1(O)CCOC1)C2 69244,N1(C(C2(SCC)CC2)=O)CCC(C(C)NC(C2(CC)COC2)=O)CC1 69245,C(=O)(C(C(F)(F)F)C(F)(F)F)N1CC(N(C(C2CC2C(C)OC)=O)C)C1 69246,C1(C(N(CCNC(CCC2(C#N)CC2)=O)CCOCC2CC2)=O)CC12CCCC2 69247,C(C)(CCC(=O)NC(CNC(=O)C(C)(C)c1cnc[nH]1)CO)OC 69248,C1(C(=O)NC(C#C)C(C)C)CC2CC2N1C(=O)CSc1nc[nH]n1 69249,N1(C(COCc2cc(C)on2)=O)CCN(C)CC1CNC(C1(C(N)=O)CC1)=O 69250,n1(C(C)C)nc2c(c1NC(N1CCCCC3(CC3)C1)=O)CCC2 69251,N1(C(C=CC)=O)CCC(NC(=O)C=Cc2cc[nH]n2)C(C)C1 69252,CN1CC(F)CC1C(=O)N(C1CCCN(C(C2CCCCN2C)=O)C1)C 69253,C1(CC(=O)NC2CN(C(c3cc(F)c[nH]3)=O)CC2CC2CC2)CCCS1(=O)=O 69254,C1(C)(CNC(CC=C=C)=O)CCN(C(=O)C(O)C(C)c2ccc(C)cc2)CC1 69255,CC(C)C(C(=O)NCC(C)N(C(=O)C(F)C1CCOC1)C)n1ncc(N)n1 69256,C1(NCCCC(=O)NCC(CO)OC)CCN(C(=O)OC(C)(C)C)C1C(C)C 69257,C(=O)(C(C)(O)C(F)(F)F)NCCC(C)N(C(=O)C(O)Cc1c[nH]cn1)C 69258,c1(C(N2CCC(NC(C(COC)C)=O)C23CC3)=O)ccc2cccc(C)c2n1 69259,CCS(=O)CC(=O)NCCC1(C)CN(C(=O)COCCN(C)C)C1 69260,C1(=CCC)CCN(C(C2C=CCN2C(c2cnnn2CC)=O)=O)C1 69261,c1(C(=O)NCC2CC3COCC3N2C(=O)C=C(Cl)Cl)cccc2c1CCOC2 69262,c1(C(N2CC(C=C)OCC2)C(=O)NCC2CCCO2)ccc(F)c(C)c1F 69263,C12(CNC(=O)C(CC3CCCCO3)N3CCCC3)CC3CC(CC(C3)C1)C2 69264,C1(CNC(CC)=O)(OCCNC(=O)CN(C)C)CCOCC1.c12cccnc1N2 69265,C1(CNC(c2c(CC)cns2)=O)CC(C)(C)CN1C(c1ccc(F)cc1N)=O 69266,c1(C(=O)NCC2C(NC(CC(CC)SC)=O)CC2)cccc(F)c1NC 69267,c1(CC)nc2sc(C)cn2c1C(=O)NC1CCC1NC(c1ccoc1CC)=O 69268,C1(NC(CC(C)(O)c2ccccc2)=O)CC2(C1)CC2N=c1[nH]nc(C#N)s1 69269,c1(CNC(CC(COC)(C)C)=O)nc2c(s1)CN(C(c1ccnnc1)=O)CC2 69270,c1(C(=O)NC2CN(C(C3C(OCC)C3C)=O)C2)ncccn1 69271,c1(NC(=O)CC2CCC(NC(c3nc[nH]n3)=O)CC2)cc(Br)nc(Br)c1 69272,N1(C(CCc2ccc(C)nc2)=O)CC2(C1)CN(C(C13CC1COC3(C)C)=O)C2 69273,N#Cc1ccccc1C(=O)NCCc1cc(C(N2CCC(F)(F)C2)=O)no1 69274,C(=O)(C(C)(O)C(F)(F)F)NCCCC(C)NC(c1ccc(C2CC2(F)F)cc1)=O 69275,C(=O)(CCC1CCc2ccccc21)NC1(C)CCCN(C(C2(F)CCOC2)=O)C1 69276,C(=O)(CC(C)C(C)C)NC1C(CNC(C(c2ccc(C)s2)C)=O)CCCC1 69277,N1(C(C2OCCN(C)C2)=O)CC2CC1CN2C(=O)COCCc1ccccc1 69278,c1(C(=O)NC2CC(CNC(C3C(C(=O)OCC)C3)=O)C2)cccnc1S 69279,C(=O)(C(CC)C(C)C)NC(CC=C)CNC(c1cnn(C)c1COC)=O 69280,c1(C(N2CC(COC(C(COC)C)=O)C(C)C2)=O)ccc(OC)c(O)c1 69281,c1(CNC(CC2(C)N(C(c3nnn(C)c3N)=O)CC2)=O)ncc(F)cc1F 69282,C12(C(N3CCC(C)(C)C3)=O)CCC(CN(C(=O)CC3CCCO3)C1)C2 69283,N1(C2CC(NCC(N3CC(C4CC4)C3C3CC3)=O)C2)C(=O)c2ccccc2C1=O 69284,Cc1ccc(CC(=O)NC2CCC(NC(C3CCC4C3C4(F)F)=O)CC2)cc1Cl 69285,N1(C(Cc2nnc(C)o2)=O)CC2CC1CN2C(c1ccnc(O)c1)=O 69286,c1(OC)cnnc(C(=O)NCCCOCCN(C)C(C2(N=[N+]=[N-])CC2)=O)c1 69287,C1(CNC(CC2CN(C)C2)=O)CCC2CN(C(=O)COC3CCCCC3)CC12 69288,c1(C(=O)NC(C)CCNC(C2CCCCS2)=O)cc(Cl)cc2ccncc12 69289,c1(OC)c(C(=O)NCC(C2CCN(C(=O)C(C)CO)CC2)(C)O)cccc1Cl 69290,C(=O)(C1Cc2ccc(Cl)cc21)N1CCC(C)(NC(c2c(C)cncc2)=O)C1 69291,CC1CCC(NC(C2(Oc3ccccc3)CC2)=O)CN1C(C1C(C)(C)C1(C)C)=O 69292,c1(C(N2C3CCC(CNC(c4c(OC)n[nH]c4)=O)(C3)C2)=O)c(O)nnc(C)c1C 69293,C1(NC(C2CN(C)C2)=O)CC2CN(C(c3ccc(C(C)(C)C)s3)=O)CC12 69294,C1(C)(NC(C(C)O)=O)CC(NC(c2[nH]ncc2C2CCC2)=O)C1 69295,c1(C(C)NCCN(CC(F)(F)F)CCO)c[nH]c2ncccc12 69296,C(C(C)C(C)C(=O)NCCOC1CCN(C(C2CC3(CSC3)C2)=O)C1)OC 69297,N1(C(c2n(CC)cc(Cl)c2)=O)CCC(CCNC(c2n[nH]c(C)n2)=O)C(F)(F)C1 69298,c1(C(=O)OCC)nn(-c2cccc(COC(C3CC3[N+](=O)[O-])=O)c2)cc1O 69299,Cc1cc(C(N2C(C(N3CCC(C)(N(C)C)CC3)=O)CCC2C)=O)c(C)cn1 69300,N1(C(C(C)CC2CCCC2)=O)CCC(CC(N)=O)(NC(c2cnn[nH]2)=O)CC1 69301,c1(C(=O)NCC=CCNC(C2CCC2F)=O)ccc(-c2nc(=O)o[nH]2)cc1 69302,c1(C(=O)Nc2csc(Cl)c2)cc(C2=CCSCC2)cc2cc[nH]c12 69303,CC1(C#CC(=O)N2C(C(=O)NCC3CC34CC4(F)F)CCC2CO)COC1 69304,Cc1ncc(C(=O)NCC2(F)CN(C(C3C4CC4C4CC34)=O)C2)c(C2CC2)n1 69305,CCCCCCC(=O)NC(C)CCN(C(=O)C(C)OCC)C 69306,Cc1cncc(C(N2CCC(NC(C34CCCC3C4(F)F)=O)C(O)C2)=O)c1Cl 69307,C1(NC(=NCC=C)NCC(CC)(CC)SC)CCc2cc(OC)ccc2C1 69308,C1(NC(C(CC)O)=O)C2CC1CN(C(c1cccc(-n3nc(C)cc3C)c1)=O)C2 69309,N1(C(C(CC)=Cc2cccnc2)C(=O)NCC(C)C)CC(C)(C)OC2COCC12 69310,N1(C(c2cnc(COC)s2)=O)CCC(NC(=O)CC2CC(F)(F)C2)C2(CCC2)C1 69311,c1(NC(c2n(CCC(=O)OCC)nnn2)C2CCC2)ccc2nc(C)ccc2c1 69312,c1(C(=O)NCC2(O)CC(NC(C=CC(C)(C)SC)=O)C2)cc2n(n1)CCC2 69313,c1(CC(=O)NCC=CCNC(C2N(CC)CC2)=O)cc(Cl)ccc1Cl 69314,C1(CC(=O)NC(CNC(C(C2CC(F)(F)C2)OC)=O)(C)C)CCC2(CCC2)CO1 69315,C1(OCC(=O)NC(C2CN(C(C3C(C)C3C)=O)C2)C)CCCCCC1 69316,c1(OCOCC)ccc(CN2CCC(C(=O)NC(C3CCCCC3)C)CC2)cc1 69317,n1(CC)nc(C2CC2)cc1C(=O)NCC12CC1CN(C(C1(O)CCSCC1)=O)C2 69318,N1(C(C2N(C(=O)OC)CSC2)=O)CC2CCC2(CNCc2cc(F)cc(F)c2)C1 69319,c1(C(N(C2CN(C(=O)CC(F)(F)c3ccccc3)C2)C)=O)nccc2ccsc12 69320,CC1(C)CCC(C(N2CC(NC(c3cnc(O)c(F)c3)=O)CC(F)C2)=O)CO1 69321,C1(C(=O)OC)CC1C(=O)N(C)CC=CC(=O)NCC1CC1Cl 69322,C(C(CC(C)C)C(=O)N1CC(C(C)NC(=O)C(C)(C)C(C)O)C1)OC 69323,C1(NC(C2C(C(C)C)(CC)C2)=O)CCCCC1NC(c1ccc(C(F)F)cc1)=O 69324,Cc1c(C(=O)NC2CCC(N(C)C(C3CC4CC3C4)=O)C2)nn(C)c1N 69325,C1(NC(COC(C)C)=O)CCC(C)(CNC(c2ccnc(C3CC3)c2)=O)C1 69326,C(=O)(C1=CCSC1)NC1C(CC(=O)Nc2ccccc2)C(O)C1 69327,C(CCC)(C(=O)N1CC2C(CN(C)C)C2C1)NC(CC1CC(OCC)C1)=O 69328,C12(C(=O)NC3CN(C(CCOCCOC)=O)CC3O)CCCCC1NC(=O)C2 69329,c1(C(=O)NCCNC(c2cccc(CC)c2O)=O)ccc2cc(C)ccc2c1 69330,CC1CCN(C(=O)CCNC(=O)CO)C1C(=O)NCCN(C)C(=O)C1CC1 69331,N1(C(C(=O)NC2CC2)c2cnc[nH]2)CCC2(CCCCC2)CC1 69332,N1(C(C=CC(=O)OCC)=O)CC2CCC1C(NC(=O)CC1CC(SC)C1)C2 69333,C(=O)(CCC(C)(C)[N+](=O)[O-])N(CCCC(=O)N(C(C)CO)C)C 69334,C1(COC)(CNC(=O)Cc2coc(C)n2)CCN(C(=O)C(C)N=[N+]=[N-])C1 69335,N1(C(CC(C)(C)C)C(=O)NCc2cccs2)CCn2c(Br)cnc2C1 69336,c1(SCC(=O)NCc2csc(C(=O)NCCC3CCC(CO)O3)c2)ccccn1 69337,C(=O)(C1=C(CC)OCCC1)N1CC(C(N2CCC(CCC)C2)=O)NCC1 69338,C1(C(C)NC(=O)CC(F)(F)F)CCCN(C(=O)CCc2ncccn2)CC1 69339,N1(C(Cn2c(C)ccc2C)=O)CCN2CCN(C(=O)C(O)C(C)(C)C)CC2C1 69340,C1(C(=O)NC2CCC(CNC(CCC=C(C)C)=O)CC2)CCC(C)(C)OC1 69341,Cc1nc2cc(NC(=O)CCc3cnc(C4(C)CC4)o3)ccc2o1 69342,C1(NC(Cc2ccc(C)s2)=O)C=CCN(C(c2ccnn2CCF)=O)C1 69343,C1(CNC(CC(C(C)C)C)=O)CC2CCC1N(C(=O)CC1C=CCCC1)C2 69344,c1(C(=O)NCC2CC(NC(c3c(OC)cccc3)=O)C2)cc(F)ccc1C 69345,c1(C(N2CC3(N(C(C4CCC(C)(C)OC4)=O)CC3)C2)=O)cccc2nn[nH]c12 69346,C=C(C)CCCC(=O)NC(C)CC(C)NC(=O)C(CN(C)C)C(C)C 69347,CCC(CC(=O)N(CCCC(=O)NCC1C=CCCC1)C)CC(C)C 69348,C=C(C)CC(C)C(=O)NCC1CCN1C(c1cc(F)cnc1OC)=O 69349,C1(C(=O)NCC(C)(C)NC(c2cnc(Cl)cc2N)=O)CCc2ncncc2C1 69350,C1(C(N2CCC(C(C)C(=O)NCCC3CC(C)(C)C3)C2)=O)CC(=O)OC1(C)C 69351,c1(C(=O)NCC(CC)NC(C23CCCC2C3(F)F)=O)ccc(OC)c2ccsc12 69352,c1(OC(C(=O)OC)C)ccc(NC(=O)NCC2(C)CC(C)=NO2)c(C)c1 69353,CC(CC(C)(F)F)C(=O)NCC(C)(C)Cn1cc(C(O)C(C)(C)C)nn1 69354,C(=O)(CC(C)(F)F)N1CCC(n2cc(CNC(CN(c3ncccn3)C)=O)nn2)C1 69355,CC(=O)CCCC(C)C(=O)N1CC2CCCC2C1C(=O)NCC1CC1 69356,c1(C(N2C(C3CCN(C(c4cc(C)[nH]c4)=O)C3)CCC2)=O)cccc(C(F)F)c1 69357,N1(C(Cc2cc(C)sc2C)=O)CCCC(N(C)C(C2CCCC(C#N)C2)=O)CC1 69358,C(C)(CCN=c1[nH]cc(C(=O)OC)cc1C)NC(CCCC(=O)NC)=O 69359,N1(C(C(C)NC(CC)=O)=O)CC=CCC1C(N1CCN(C(C)C)CC1)=O 69360,c1(NC(C(=O)N(CC(C)C)Cc2ccccn2)=O)ccc(C2CCC(=O)N2)cc1 69361,C(=O)(C(O)C(C)(C)C)N(CCN(C(c1sc(CCC)c(CC)c1)=O)C(C)C)C 69362,c1(CC(N2CC3C(NC(c4ncc(C)nc4)=O)(C3)C2)=O)ccnc(Cl)c1F 69363,C1(C(N)=O)CCN(C(=O)NCCc2nccn2Cc2ccccc2)C1 69364,C1(C(=O)NCC(C2CCC2)OCC)CCN(C(=O)CC(CC)C(F)F)CC1(C)C 69365,N1(C(C2C(C)(CC)C2)=O)CCOC2(C1)CN(C(C1(SC)CC1)=O)C2 69366,N1(CCNC(C2(C)C(C)C2)=O)CCC(NC(C2CCC2(F)F)=O)CC1 69367,C(=O)(C1=NN(C)C(=O)CC1)N1CCC(NC(C2(C(=O)NC)CC2)=O)C(CO)CC1 69368,C1(C(=O)NC(c2ncccn2)(C)C)CCC2(CC2)N1C(=O)CCC1CCC1 69369,C1(NC(c2cc(C)ncc2)=O)CCCC12CN(C(c1nccn1C)=O)C2 69370,CC(C)C(C)C(=O)N1CC2CC2(NC(c2cc(-c3ccccc3F)on2)=O)C1 69371,CCC(C)(C)C(=O)NC1CC(N(C(CC2(COC(C)=O)CC2)=O)C)C1 69372,C(=O)(C#CC1CCC1)NCC(C)CN(C)C(C1C2CCCC12)=O 69373,CC1CC2(CCN(C(=O)C3=CC4CCCC34)CC2)CN1.C(C)C(=O)NC1CCCO1 69374,n1(CC)nncc1CN1CCC(N(C(C(=O)OC(C)(C)C)C2CC2)C)C1 69375,c1(C(N2CCN(CC(N)=O)CC2)C(=O)NCCCSCC)ccc(C)c(F)c1 69376,C1(C(N2CCC(F)(CNC(C(C)(C)SC)=O)C2)=O)CCC2(CCCC2)C1 69377,N1(C(C(=O)NC2CCN(Cc3cn(C=C)nc3)CC2)=O)CCCCC(C)C1 69378,C#CC1(OCC(=O)NCC(C)NC(=O)C(c2cnn(C)c2)O)COC1 69379,C1(NC(=O)Cc2cccc(Cl)c2)CC2CCC(C1)N2C(C12COC(C1)C2)=O 69380,CCCCCC(O)CC(=O)N(C(CC(F)F)C(=O)NCc1cn(CCC)nn1)C 69381,c1(NCC2(C)N=C(C)SC2)ccc(S(=O)(=O)N2CCCSC(C)C2)c(Cl)c1 69382,C1(CC=C)(NC(=O)CCCc2cccs2)CCN(C(=O)CCOCCOC)C1 69383,N1(C(CC(=C)C)=O)CCC2(CC1)CC(NC(C1NC(=O)CC1C(F)(F)F)=O)C2 69384,C(c1cnn(-c2ccccc2)c1)=CC(=O)NCC(CC)NC(=O)COCC(F)F 69385,C1(NC(=O)CN2CCCC2=O)CN(C(=O)C(=Cc2cscn2)F)CC1CO 69386,c1(CNCCCc2cccc(N)c2)cc2c(cc1O)OCO2 69387,N1(C(C(C=C=C)C)=O)CC(C(=O)N)C(C)(C)C1.C(C)COC 69388,Cc1ccc(C(N2CC3CC3(NC(=O)OC(C)(C)C)C2)=O)c(N)c1 69389,CC(C)CC(C(=O)NCC1(CNC(c2occc2C2CC2)=O)CC1)n1ccnc1 69390,CC1CN(C(=O)CCNC(c2ccco2)=O)CCC1NC(=O)C(C)(C)C1CCC1 69391,N1(C(C(C(C)C)O)=O)CC2CCN(C(c3cc(C(F)(F)F)ccc3N)=O)C2C1 69392,N1(CCNC(=O)Cc2ccc(F)cc2)CCCN(C(=O)C=CCO)CC1 69393,C(=O)(C1(O)CCCc2ccccc21)N1CCCC(CCC=C)(C(=O)OCC)C1 69394,C#CCC(C)(CC)C(=O)NC(CC(=O)N(C(C)COC)CC)C(F)(F)F 69395,C1(C(N(c2ccccc2)CC)=O)CCCN1NC(=O)CCc1cccn1C 69396,c1(CC)ccc(S(=O)(=O)NC(c2ccc(F)cc2F)C(C)C)cc1C(=O)O 69397,CC1(CCNC(C2SCCS2)=O)CCN(C(c2ccc(F)c(O)c2)=O)CC1 69398,c1(-n2cc(C(=O)NCC(CNC(CN(C)CC)=O)C)nn2)ccccc1C 69399,c1nccc(=NCc2ccc(-c3cc(C(=O)OC)c(F)nc3)cn2)[nH]1.C1CC1 69400,N1(C(C(C)(C)OCC)=O)CC2CCOCC2(NC(c2nc(C(C)C)oc2C)=O)C1 69401,c1(C(N2C(C(=O)NC(c3ccsc3)C)CC(O)C2)=O)cccc([N+](=O)[O-])c1 69402,C1(CNC(C2C(OCCN(C)C)C2)=O)CN(C(=O)CCSC2CCCC2)CC1O 69403,C1(NC(C2(C)CCNC2=O)=O)CC2(C1)CN(Cc1cc(Br)ccc1N1CCCC1)C2 69404,c1(C(N2C3CC(CNC(CC(C)SC)=O)C2CC3)=O)coc2c(F)cc(Cl)cc12 69405,N1(C(C(C=C)O)=O)CCCC(n2cc(CNCc3ccnnc3C)nn2)C1 69406,CC(C)(CO)C(=O)NCCCN(C(=O)CCc1ccon1)CC1CCCC1 69407,N1(C(COCC)=O)CC=CC(NC(c2ccc(OCc3ccccn3)cc2)=O)C1 69408,O=C(CC(C(F)(F)F)NC(C1CC1(F)Cl)=O)NCCOCC(F)(F)F 69409,C1(C(N2CCC(c3ncco3)C2)C(=O)NCC(C)C)CCC(CCC#N)CC1 69410,C1(C(=O)NC(C(=O)NC2CN(C(CC)=O)C2)CCSC)CCCC(=O)CC1 69411,CCCCC(CNC(=O)CCN(S(C)(=O)=O)C)NC(c1cc(COC)cn1C)=O 69412,C=C(Cl)C(C)(C)C(=O)N1CCN(C(=O)C2=C(C)OCC2)C2CC12 69413,CC(C)S(=O)(=O)CC(=O)NC1CCN(C(c2cc(C#N)n(C)n2)=O)C1C 69414,N1(C(c2[nH]ccc2C2CC2)=O)CCN(C(C2CCCCC2)=O)C(C(F)(F)F)C1 69415,N1(CC)CCC(CNC(=O)C(C)(C)C2CCN(C(=O)CCCN(C)C(C)=O)C2)C1 69416,N1(C(C(C)(O)C2CCC2)=O)CCC(O)(CCNC(c2cc(C(F)(F)F)n[nH]2)=O)C1 69417,c1(CC(=O)NCC2C(CNC(=O)CCCC3CCCC3)C2)cn2c(n1)CCCC2 69418,c1(C(C)(C)C)ncc(C(=O)NCC2CC2NC(=O)CC(C)(C)C2CC2)cn1 69419,c1(CCCC(=O)N(C(C)CCNC(=O)C(F)(F)CO)C)nc2ccccc2s1 69420,CC1CN(C(c2nc(C3CC3)cs2)=O)CCC1CNC(C1(CO)CCOCC1)=O 69421,C1(C)(C(=O)NC2CN(C(Cc3c(C)n(C)nc3)=O)CC2C)CCCN(C)C1 69422,C1(C(=O)NCC2CN(C(C3CC3c3ccnn3C)=O)CC2C)(OCC)CCOCC1 69423,C1(C(=O)NCC(CNC(C=CC=CCC)=O)CO)CC(C(C)C)=NO1 69424,C1(CCC)CN(C(c2cc(F)cc(F)c2)=O)CCN1C(=O)C1=CCCSC1 69425,c1(NCC)cncc(C(=O)NC(C2CN(C(c3cnnn3C)=O)CCO2)C)c1 69426,CC(C)(CCCF)C(=O)N1CC=CC(NC(C2CC23CCCCC3)=O)C1 69427,C=CC1CN(C(=O)CN2CCCCC2C)CC1NC(c1cc(C)c(C)cn1)=O 69428,c1(OCC)cccc(CCC(=O)NC(C)(C)CN(C)C(C2C(C)C2C)=O)c1 69429,c1(N(CCCNC(Cc2c(C)cccc2C)=O)C)nc2cc(F)ccc2o1 69430,CC(C)C(C(=O)NCCC1(NC(c2cccc(C(F)F)n2)=O)CC1)n1cnnc1 69431,CC(CCCNC(=O)CCNC(=O)CO)NC(c1nc(C2CC2)cs1)=O 69432,c1(C(=O)NC2(C(N3CC(CCO)(CC)C3)=O)CCCCC2)cc(C)nc(C)n1 69433,C12(NC(c3cc(F)cc(F)c3)=O)CCCN(c3nccc(C4CC4)n3)CC1C2 69434,c1(-n2c(-c3c(N)snn3)nc(-c3ccccn3)n2)cccc(C#N)c1 69435,C12(NC(c3c(C)ocn3)=O)CCC1CN(C(c1ccc(-n3cccc3)cc1O)=O)C2 69436,N1(C(CCN(C)CC)=O)CC2CCC2(CC(=O)NCC(c2ccccn2)O)C1 69437,CON1CC(C(=O)NC2CCN(C(=O)CCc3cncc(C)c3)C2(C)C)CC1=O 69438,c1(-c2nnc(C(ONC(=O)N(C(C)C)C3CC3)C)s2)ccccc1F 69439,O=S(=O)(C1COC1)C1CN(Cc2cn(-c3nc(Cl)ccc3Br)nn2)C1 69440,c1(C(=O)NCC2CC(NC(CCCC=C)=O)CC2O)cc2occc2s1 69441,C(CCC(C)C(=O)NC1CC(=O)N(C2CN(C(C34CC(F)(C3)C4)=O)C2)C1)OC 69442,C1(C(N(CCC(N2C(C(c3cnn(C)c3)C)CC2)=O)C)=O)CC(=O)NC(=O)N1 69443,C1(OC)CN(C(=O)C=Cc2ncc[nH]2)CCC1NC(=O)Cc1ccsc1C 69444,C1(C(=O)NC(c2ccccc2)C(=O)NCCCC(O)CO)CC12CCCCC2 69445,Cn1c(O)ncc(C(=O)NCCNC(c2cc(OC(F)F)cc(F)c2)=O)c1=O 69446,C12(CCN)CC3CC1C2C3O.N1(C(CCSC)=O)CCN(C=O)CC1 69447,N1(C(CN2CCC(C(=O)NC)CC2)=O)CCN(C(=O)OC)CC1.C12CCC(C1)N2 69448,N1(C(C(COC)C)=O)CC2CCC(C1)N2C(c1cccc(C)c1NC(C)=O)=O 69449,C(=O)(CCCC(C)(C)CC)NCC(C(=O)NCC(=O)OCC#C)(C)C 69450,CCCCCCCNC(=O)C(CCN(C)C)NC(c1cc(C2CC2)on1)=O 69451,C12(NC(c3ncn(C)c3)=O)CN(C(=O)C3=CCS(=O)(=O)C3)CC1CS(=O)(=O)C2 69452,c1(NC(C2CCC(CC(=O)NC(c3nncn3C)C)C2)=O)ccc(CO)cn1 69453,N1(C(C2CCOC3(CCC3)C2)C(=O)NC)CCCC2c3[nH]c(C)nc3CCC12 69454,N1(C(C2OCC(C)C2)=O)CCC(NC(c2ccc([N+](=O)[O-])o2)=O)C12CCC2 69455,C1(C(=O)NC2C(N(C)C)CCCC2)C2CC(F)C(C2)N1C(c1ccc(F)cn1)=O 69456,c1(C(N2CCCC(CNC(c3c(SC)snn3)=O)C2)=O)cnn2c1CCCC2C 69457,c1(C(N2CC(CNC(C(CC)C)=O)C2)=O)cc(F)cc(Br)c1 69458,Cc1nc(NC(c2c(CO)cccc2C)=O)ncc1Br.C12CCC(CC1)C(=O)N2 69459,N1(C(c2cncc(COC)c2)=O)CCN(C(c2ccc(C)nc2)=O)CC1COC 69460,CCCC(C)CC(=O)NCc1ncccc1CNC(C12CCN(CC1)CC2)=O 69461,N(C(=NCCCOCC)NCC1(C)CCCCO1)CC(C=C)(C)C 69462,O=C(CCCCN1CCCC1)NCCC1CN(C(=O)Cn2cccn2)CCO1 69463,N1(C(C=C(COC)C)=O)C2CCC1C(NC(=O)C(O)Cc1cc(Cl)cc(Cl)c1)C2 69464,C=CCCC(O)CN(C)C(C1CSCCN1C(C1SCC=C1C)=O)=O 69465,C=CCC(CC=C)C(=O)NC1CCOCC1NC(C1(CCF)CC1)=O 69466,N1(C(C2(CCC)CCNC2=O)=O)CCCCCC(NC(c2c[nH]ccc2=O)=O)C1 69467,c1(C(=O)NC(CNC(CC(C)NC(N)=O)=O)C)cc(C(C)(C)C)n(C)n1 69468,c1(CC(=O)NC(C(=O)NC2(CC3CC3)CC2)C2(O)CCC2)ccc(O)cc1 69469,C(=O)(C(F)(F)C(F)(F)C(F)F)NC1C(CNC(C2CC23CCC3)=O)CC1 69470,C1(CNC(Cc2c(C)noc2)=O)CCC2(CCC2)C1NC(=O)CC1=NNC(=O)C1 69471,Cc1cc(=NC(C)CN(C(=O)Cc2ncncc2Cl)C)[nH]cn1 69472,O=C(C1=CCCN(Cc2c[nH]c3ccccc23)C1)N(c1ccc(F)cc1)CCO 69473,C1(C(N(CC(=O)OC)CCN2CCCC2)=O)C[Si](C)(C)CCN1C 69474,N1(C(CCSCCC)=O)CC(NC(C2CCCC(=O)C2)=O)C(C)C1 69475,CCCCC(C)CCC(=O)NC(C)C(C)(C)NC(=O)Cc1ccc(O)c(C)c1 69476,C1(OC(C)(C)C)(NCCN2CCOCC2c2nc[nH]n2)CCS(=O)(=O)C1 69477,C(=O)(CC1COc2cc(O)ccc21)NCC(CO)NC(Cc1ccc(C)nc1)=O 69478,C(=O)(C(C(C)CC)NC1CC1)N1CCC(O)(CNC(C=CCC)=O)C1.C(N)=O 69479,N1(C(COCCCOC)=O)CCC(C)C(NC(=O)C(F)=C(C)C)C1 69480,c1(C(N2C(CN(C(C(CC=C)C)=O)CC)CCC2)=O)ccc(NC(C)=O)cc1Cl 69481,CCCC(C(=O)OC)C(=O)N1CC(C)CC1C(=O)NCCCC(C)C 69482,Cc1ccc(-c2nc(C(C)O)nn2C(c2ccc(Br)cc2)C)c([N+](=O)[O-])c1 69483,c1(-c2onc(C34CCCC3C4)n2)cc2cc(Cl)ccc2[nH]1 69484,c1(NCCC=CC=C)cc(=NC(C)c2ccn(C)n2)[nH]c(COCC)n1 69485,Cc1cc(C(=O)NC2CC2NC(=O)C2=C(Cl)CCC2)cc(O)n1 69486,N1(C(Cc2c(C)c[nH]n2)=O)CCCC(Cc2cn(CC3CCOCC3)nn2)C1 69487,CC1CCOC1CS(=O)(=O)NC(C1CC(Cl)(Cl)C1)c1nnnn1CCOCC.C1CC1 69488,c1(C(N2CC(CCC)N(C(c3cnnn3C)=O)CC2)=O)ccn2cccc2c1 69489,Cn1ccnc1C(N1CCC(C(=O)NCCOc2cccnc2)C1)=O 69490,C=CCC(C)(O)C(=O)N1CC(C(O)C(=O)NCc2nc(N(C)C)no2)C1 69491,C1(C(=O)NCC(CNC(=O)C(C2CCOCC2)C)CO)(CC)CCCC1 69492,CCC(C(=O)NC(C)CCNC(C1(F)CC=CC1)=O)OC 69493,C(C(CC(C)C)NC(c1csc(F)c1)=O)NC(c1n(CCC)ccc1)=O 69494,CC(F)(F)CCC(=O)N1C2CCC1C(C(=O)NCCC(=O)NC1CC1)C2 69495,N1(C(CCC2N(C(c3c(CC)cco3)=O)CCC2)=O)CCC(C)C2(CCC2)C1 69496,c1(CN(CCCCOCCO)C)csc(-c2cnn(C)c2)n1 69497,CC1CN(C(=O)CC(O)C2CCCC2)CCC1NC(c1cn(C)ccc1=O)=O 69498,N1(C(CC2CC(=C)C2)=O)CCN(C(=O)Cc2ccc(O)cc2)C2CCCCC12 69499,C1(NC(CN(CC)CC)=O)CC2(C1)CC(C(=O)NC1CCC3CCC13)C2 69500,N1(C(C(C)OC)=O)CCC(F)(F)C(N=c2nc(C)nc3[nH][nH]cc2-3)C1 69501,N1(C(CNC(=O)OC)=O)CC2CCC2(CC(=O)NC2CC(=C3CC3)C2)C1 69502,C1(O)(CCNC(COCc2nnc(C)s2)=O)CCN(C(c2cnc(O)o2)=O)C1 69503,Cc1cc(C(N2C(C(N3CCC(F)(F)C3)=O)CC3CC23)=O)c(C)cc1Br 69504,C(=O)(C1CCCc2scnc21)N1C(C)(C)CC(NC(C2CCC(C)CC2)=O)C1 69505,C1(CNC(C2(COC)CC(=O)C2)=O)CCC(CNC(=O)CCOC(C)C)CC1 69506,CC1CC(C(=O)Nc2c[nH]nc2Br)N(C(c2cncc(Br)c2)=O)C1 69507,c1(SC(C)CC#N)ccccc1NC(=O)C(=O)NC1CN(C(=O)CC(F)(F)F)C1 69508,N1(C(COc2cccc(CC)c2)=O)CCC2(NC(=O)C(C)(F)F)CC2C1 69509,c1(NC(c2cn(CC=C)nn2)=O)cccc(CNC(=O)CC2CC2C2CC2)c1 69510,C#CCC(C)(C(=O)NCCC)NC(=O)CCC(=O)NC.C1CN2CCC1CC2 69511,N1(C(CC2CCC(OCCC)CC2)=O)CC2CC1CCC2NC(c1cnsn1)=O 69512,N1(C(Cc2c(C)ocn2)=O)C2CCCC1CN(C(C1CCCOC1)=O)CC2 69513,N1(C(=O)NCC2CCO2)CCN(CC2CC2)CC1 69514,c1(NCc2cc(C)ncc2)nc(C)nc(Br)c1F 69515,c1(C(=O)NC(CNC(c2c(C)ccnc2O)=O)C(C)(C)C)ccc2c(c1)OCC2 69516,N1(C(C2N(C(=O)CC(Cl)Cl)CC=C2)=O)CCOCC(C2CC2)C1 69517,N1(C(c2c(OC)cc(Br)cn2)C(=O)NC2CC(F)(F)C2)CCCNC(=O)C1(C)C 69518,CC1Cc2cc(CCN=c3ccnc(N4CCC(C)(F)C4)[nH]3)ccc2O1 69519,C1(NC(C=CCN(C)C)=O)CC2CN(C(c3[nH]nnc3C3CC3)=O)CC12 69520,N(C(=NCCCC1C=CCC1)N1CC=C(c2cccs2)CC1)CCOC 69521,CCC(C(=O)N(CC(=O)N(CC)CC1CCCC1)CC)SC 69522,C=CC1CN(C(C2CC(=O)CCO2)=O)CC1NC(C1CCCO1)=O 69523,CCC(CC(=O)NC1CCC12CN(C(=O)COc1ccc(C)c(C)c1)C2)C(F)F 69524,c1(CNC(=O)NCc2[nH]nc(CC)n2)cnc(N(C)C)nc1 69525,S(=O)(=O)(c1ccc(NC(c2ccsc2)C)c(Cl)c1)NC(C1CC(F)(F)C1)COC 69526,N1(C(CC=C=C)=O)CCCC(NC(c2nc(C)n(C3CC3)c2C)=O)C1C 69527,C(CCC(=O)NCCC1(NC(=O)CCF)CCCC1)=CC 69528,S(=O)(=O)(c1cnc(NCC2(CO)CCN(C)C2)c(Cl)c1)NCC(C(CC)CC)O 69529,N1(C(C(COC)OC)=O)CC(CNC(=O)Cc2cccc(OC)c2Cl)C2(CC2)C1 69530,CC1CCCCC1C(=O)COC(=O)CC(c1cccc(Br)c1)C 69531,Cc1ccc(F)c(C(=O)NCc2cccc(CNC(c3cn(C)cn3)=O)c2)c1F 69532,C(=O)(C(CNC(C1(CO)COC1)=O)C(C)(C)C)N(CCC)CC 69533,CC1CCC(NC(=O)Cn2cnc(=N)[nH]2)CN1C(=O)CC1(CO)CC1 69534,N1(C(C2(NC(C)=O)CCC2)=O)CCN(C(c2cnc(C3CC3)o2)=O)C(C)C1 69535,CC1(C(=O)NCC2(O)CCN(C(=O)CCCn3cccc3)C2)CCCNS1(=O)=O 69536,N1(C(c2cn(CCC)nc2)=O)CCOC(CNC(=O)Cn2[nH]cnc2=N)C1 69537,c1(C(=O)NC2(C)CCC(NC(C(C)(C)OC)=O)CC2)cc(C)c(F)cc1N 69538,c1(C(=O)NCC2N(C(C3CCN(C)C3)=O)CCOC2)cncc2c(F)cccc12 69539,c1(C(=O)NC2(C)CN(C(C(CCC)(C)C)=O)C2)n[nH]c2c(C)cccc12 69540,Cc1ccc2c(C(=O)NCC34CC(CN3C(C3CC3C)=O)C4)n[nH]c2c1 69541,C(=O)(CC1=CCCC1)NCC(C)CNC(c1conc1C(F)(F)F)=O 69542,c1(C(=O)NCCCCC(C)NC(=O)CSC(F)F)ccn2nccc2c1 69543,C1(C(N2CCOC(c3n[nH]c(CO)n3)C2)=O)CCOC2(CCCCC2)C1 69544,CCC(F)(F)CC(=O)N1C2CCC1C(CNC(c1ccc(OC)c(C)c1)=O)C2 69545,N1(C(CCNC(=O)OC(C)(C)C)=O)CC2CCC(NC(C3(CSC)CC3)=O)CC2C1 69546,C1(C(N2CC(CNC(=O)C(c3cccc(Cl)c3)O)C2)=O)CC2COCC2C1 69547,C(=O)(C(C)(C)C(O)C(C)C)NCCOCCNC(C(CC(C)(C)C)OC)=O 69548,Cc1nc(=N)[nH]c(C)c1C(=O)N(C)CCNC(c1cc(F)ccc1C(F)F)=O 69549,C(=O)(CC1OCc2ncccc21)NC1C2CN(C(C3(C(=O)NC)CCC3)=O)C1C2 69550,N#Cc1cnn(-c2ccccc2)c1NC(C1CCN(Cc2cccnc2Cl)C1)=O 69551,Cc1nc2ccccn2c1C(=O)NC(CNC(C1CC(F)(CO)C1)=O)C(C)(C)C 69552,C1(N(C(C2N(C)CCC2)=O)C)CCCCC1N(C)C(c1cnc[nH]c1=N)=O 69553,CN1CCN(C(c2ccc(O)nn2)=O)CC1C(N1CC(n2cnnc2)C1)=O 69554,c1(C(=O)NCC2(OC)CN(C(=O)CCC(CC)OC)C2)cc(N)c(OC)cc1F 69555,C1(CC(=O)NCCCN(CCC)C(C2CCOC2(C)C)=O)CCC(=O)CC1 69556,c1(CC)ncsc1C(=O)NCC1(CC(=O)NC(C)CCO)CCC1 69557,C(CCCCC(C(=O)NC(C)(C)C)N1CCN(C(C)(C)CF)CC1)OC 69558,S(=O)(=O)(c1cc(C)cnc1NCC(O)C(N)=O)NCc1scc(CC)n1 69559,c1(OC)cc(C)sc1C(=O)NCCNC(c1cc(-c2ccc(F)cc2)n(C)n1)=O 69560,C1(C(=O)NCC)CCN(C(=O)C(=O)NC2CCCC2(C)NC(C)=O)CC1 69561,c1(N2CCC(C(C)O)C2)cc(NCC2(c3cccnc3)CC2)nc(C(F)(F)F)n1 69562,N1(C(C=NOC)=O)CCCC2(C1)C(NC(=O)CC1CC3CC3C1)CCN2C 69563,c1(OC)cc(C2CCCN(C(C3(C4CCC4)CCC3)=O)C2)cc(F)c1 69564,c1(CC)cc(C(=O)NCC2(C(C)(C)C)CCN(C(c3csc(C)c3)=O)C2)ncn1 69565,c1(OC)nc(OC)nc(N(C2CCNCC2)C(=O)CCn2nc(C)nc2C)n1 69566,C1(NC(CCCN(C)C)=O)CC2CN(C(C3CC(c4cccc(F)c4)C3)=O)CC12 69567,c1(CNC(C(C)CO)=O)cc2n(n1)CCN(C(c1cc3n(n1)CCCO3)=O)C2 69568,C12(C(=O)NC(C3CCCOC3)C)CC(CO)(CN1C(c1ccncn1)=O)C2 69569,Cc1ccc(CC(C)NC(=O)NCc2cccc(-c3ccccc3)n2)c(C)c1 69570,N1(C(C=CC(=O)OCC)=O)CC2CC1CN2C(c1ccc(C(N)=O)cc1)=O 69571,c1(CC(=O)NC(C2(O)CCN(C(=O)C3=CCOC3)C2)C)cc(F)cc(F)c1 69572,C1(NC(=O)OCC)CCN(C(=O)C(C2CCSCC2)F)C1 69573,CC1CC(NC(c2cn(CCO)nn2)=O)CN(C(=O)Cn2ccccc2=O)C1 69574,Cc1cc(CN(C)CCc2cccc(C(F)(F)F)c2)nc(-c2cncc(Br)c2)n1 69575,n1(CC)cccc1CCNC(=O)NCCCC(=O)N(C)C(C)C 69576,C(=O)(CC(O)CNC(=O)C(C)(CO)NC(=O)C(n1ccc(C)n1)C)OC 69577,c1(SC)cccc(CC(=O)NCC(C)(CC)NC(=O)Cc2cnc[nH]2)c1 69578,C1(C(=O)NCCC2(COC)CC2)CN(C(=O)CC(C)C2CC2)C2(CCC2)C1 69579,c1(C(N2CC3(CCN(C(c4cnc(C)s4)=O)C3)C2)=O)cccc2nc(O)oc12 69580,C1(CC#N)CN(Cc2ccc(Br)c(O)c2)CCN1C(c1ccc(Cl)c(O)c1)=O 69581,N1(C(C2C(CCC)C2)=O)CCN(C(=O)C=Cc2cc[nH]n2)C(C2CCCC2)C1 69582,N1(C(C2(COC)CCCC2)=O)CCC(NC(=O)CC2COC(=O)C2)C(C)(C)C1 69583,c1(C(=O)NCC(CC)NC(c2cc(C(C)C)ccc2F)=O)cnc(C)c(C#N)c1 69584,C1(CNC(C(C)Cc2ccco2)=O)CN(C(=O)CCNC(=O)CO)CCCO1 69585,c1(OC)ccc(OCC(=O)NCC#CCNC(=O)CC2COCC(C)O2)cc1C 69586,N1(C(c2cc(C(N)=O)[nH]n2)=O)CCCCCCC1C(=O)NCCc1ccccn1 69587,C12(C(=O)NC(C)CNC(=O)CC3CSC3)CCC(N=[N+]=[N-])(CC1)C2 69588,C(=O)(C(C)CCCOC)NCCCN(CCCCNC(CC(C)C)=O)C 69589,C(=O)(C(C)C(C)S(C)(=O)=O)NC1CC(NC(c2c(OC)ccc(C)c2)=O)C(O)C1 69590,CCCCCC(C)CC(=O)N1CC(C(=O)NC(c2cnc[nH]2)C)CCC1(C)C 69591,c1(OC)ccc(C(C)C(=O)NCC2CCCCC2NC(c2cccs2)=O)cc1F 69592,Cc1ccc(NC(C2CCC(NC(=O)C(C)C#N)C2)=O)c(C)n1 69593,c1(SCC(=O)NC(CC=C)CNC(=O)Cc2ccc(O)nc2)c(C)cccc1C 69594,N1(C(C(=O)N(C)Cc2ccc(Cl)nc2)=O)CCn2c(CC3CCCC3)nnc2C1 69595,C(c1ccc(C(N)=O)cc1)=CC(=O)NCC(C)N(C(C(C)C1CCC1)=O)C 69596,CCC(C)C(O)C(=O)NC1CCN(C(C2CN(CC)CCO2)=O)C1C 69597,C1(O)(Cn2cc(C3(CC)CCC3)nn2)CCCN(C(C2(Br)CC2Br)=O)CC1 69598,c1(NC(CCN(C(CC(COC)C)=O)CCCO)=O)ccc(C)c(F)c1 69599,N1(CCC(C)C)CCC(C2(NC(=O)C(C)Oc3ccccc3F)CC2)CC1 69600,c1(OC)c(C(=O)NC2CC(NC(c3ccc(S(C)=O)cc3)=O)C2)nc(O)nc1O 69601,C(CCCC(=O)NC1CN(C(c2ccc(-c3n[nH]c(C)n3)cc2)=O)CC1C)OC 69602,C12(C(=O)NCC(C(C)(C)C)O)CCC(CC1)N(C(=O)C1=CC3C=CC1C3)C2 69603,c1(OCCC(N2CCC(C)(NC(C(CC)F)=O)C2)=O)c(C)cccc1C 69604,c1(NCCOC)ccc(NC(=O)CSC2CCS(=O)(=O)C2)cc1 69605,N1(C(C(C)c2cc[nH]n2)=O)CC2CN(C(c3ccc(CCO)cc3)=O)CCC12 69606,C1(OC)CC(C(=O)NCC(C)C(F)F)N(C(=O)COCC2CC2)C1 69607,Cc1ncc2c(n1)CCC(CNC(c1csnn1)C)C2 69608,Cc1oc(S(N)(=O)=O)cc1C(=O)NCC(C)N(C(=O)C(C)c1cncs1)C 69609,C=CCC(CNC(=O)C(C)OC)C(=O)NC(c1c[nH]ccc1=O)C 69610,c1(OC)ccc(OC)c(C(N2CC3(CCC3NC(c3ccc(O)nn3)=O)C2)=O)c1 69611,CCCCC(F)C(=O)N1CCCC(C)(NC(c2ccnn2C)=O)C1 69612,C1(C(=O)NC(COC)C(C)C)CCCCCN1C(c1nn(C)cc1C)=O 69613,c1(NC=O)ccc(C(N2CCC(NCc3ccc(-c4ccccc4)o3)C2)=O)cc1 69614,Cn1cccc(C(=O)N(C2CCN(C(C3(C(C)(C)C)CCC3)=O)C2)CCO)c1=O 69615,N1(C(CCNC(CCC)C)=O)CCC(C2CN(C(=O)C=CC(=O)NC3CC3)C2)CC1 69616,C1(C(=O)NCCN(C(=O)CSc2n[nH]c(=N)s2)C(C)C)CCCC(C)(C)C1 69617,N1(C(c2ccc(C(C)=O)o2)=O)CC(CNC(=O)CC2CCCO2)OC2(CCC2)C1 69618,C(CC(C)(C)CC(=O)N(CCCN(C)C(c1cc(C#N)ccc1F)=O)C)OC 69619,N1(C(C(CC(N)=O)O)=O)CCCC2CN(C(c3scc4c3CCCC4)=O)CCC12 69620,C12(NC(C=CCN(CC)CC)=O)CCC(CC1)N(C(=O)C(C)CC1CCCO1)C2 69621,CC1N(C(C2CN(C(C3CCCCC3)=O)CCC2O)=O)CCC1(C)C 69622,c1(CC(=O)N(CCCNC(C(C=C=C)C)=O)CCO)noc2ccc(OC)cc12 69623,c1(C(=O)NCCC2C(C)CN(C(=O)CC3CNC(=O)O3)C2)cnc2n1CCC2 69624,C1(CCC(=O)N(C2CCOC2=O)C)CCCN1C(=O)CC1CC(F)(F)C1 69625,N1(C(CCN(C(=O)C(C)c2cccs2)CC=C)=O)CCCC(NC(C)=O)C1 69626,c1(C(=O)NCCOC2CN(C(C(CO)OC)=O)C2)c(C)cc(C)cc1C 69627,c1(C(N2C(C)CC(CNC(C3(CC#C)CCCO3)=O)C2)=O)cc(C#N)oc1C 69628,N1(C(c2ncc(C)c(Cl)c2)=O)CC2CCN(C(C3CCCC3)=O)CC12 69629,c1(C(=O)NC2C3N(C(c4c(C)cco4)=O)CC(CC3)C2)cccc2[nH]nc(O)c12 69630,C(=O)(C1=NN2CCCN=C2N1)NC1CC(CCNC(C(CC)C(=O)OC)=O)C1 69631,Cc1nc(C(=O)NC(C)CNC(=O)CCN2CCNC(=O)C2)cc(O)n1 69632,c1(CN=c2ccc(NC(c3cc(O)ccc3F)=O)c[nH]2)cccc2ncccc12 69633,CC1CN(C(=O)CC2CC3CC3C2)CC(C(=O)NCc2cc(C(F)F)no2)O1 69634,c1(CNC(=O)NC(c2nc(CC)on2)C)c(Cl)ccnc1Cl 69635,Cc1ccc(S(=O)(=O)n2ccc3c(NCC#CCCO)ncnc23)cc1 69636,C(=O)(C1=NOC(C)(C)C1)N1CCCC(F)(C(N(CC(CCC)C)C)=O)C1 69637,c1(C(=O)NCC(=O)N(CC(C)CNC(C2CC=CC(O)C2)=O)C)cccc(F)c1 69638,C1(NC(CN(C)C(C2(C)CCC(=O)C2)=O)=O)C2C3CCC(C3)C12 69639,C(=O)(N=c1cc2ccccn2[nH]1)C1N(C(c2c(C)ccc(C)c2)=O)CC(F)(F)C1 69640,N1(C(c2cccnc2)C(=O)NCCC)CCC2(CCN(C)CC2)C(CO)C1 69641,c1(C(=O)NC2C=CCN(C(c3cc(C)[nH]n3)=O)C2)cncc2sccc12 69642,S(=O)(=O)(c1cc(Cl)ccc1F)N1CCN(C(c2cc(F)c(Cl)cc2Cl)=O)C2C1C2 69643,CC(O)CC(C)(C)CNC(C1(C)CC(NC(=O)CC2CC2(C)C)C1)=O 69644,C1(OC)CCCC(CC(N2CC(F)CC2CNC(=O)CCSCC(N)=O)=O)C1 69645,c1(C(=O)NCC(CNC(c2cccc(C)c2)=O)C)ccc2nnc(C3CC3)n2c1 69646,c1(C(N(CCCNC(CCN(CC)CC)=O)C2CC2)=O)nccc2ccsc12 69647,C1(C(=O)NC2(C)CN(C(C3(C)CCOC3)=O)C2)CCOC(=O)CC1 69648,C1(N(C(C(CSC)C)=O)CCO)CCN(C(c2cncc(C(C)(C)C)c2)=O)CC1 69649,C1(C(N(CCN(C(C=CC(C)(C)SC)=O)C)C(C)C)=O)C(F)(F)C12CCC2 69650,Cc1cccc(-c2nc(-c3cccc(Cl)n3)nn2-c2ncnn2C)n1 69651,Cc1c(CNC(=O)CC2(F)CN(C(c3cc(C(N)=O)[nH]n3)=O)C2)nnn1C 69652,C1(C)(NC(c2ccnc(C)n2)=O)CCN(C(c2cc(C(C)(C)C)ccn2)=O)CC1 69653,C(=O)(C(C)(C)C1=CCSCC1)NC(CCCC)CNC(c1cccnc1OC)=O 69654,CC(O)(CC(=O)N1CC=CC(NC(c2snc(O)c2Cl)=O)C1)C(F)(F)F 69655,N1(C(=O)NCc2nccnc2Cl)CC2CC(CO)C(C2)C1 69656,N1(C(c2c(C)c(C3CC3)on2)=O)CCC(O)(CNC(C2CC23CC(O)C3)=O)CC1 69657,C1(C(C)NC(=O)CCC2CCCO2)CCCN1C(c1n[nH]c(C2CC2)n1)=O 69658,CC(C)C(O)C(F)(F)C(=O)N1CCN(C(C2(C)CC2(F)Cl)=O)CC(O)C1 69659,C1(C(=O)NCCCC)CCCCC1C(=O)NC.c1(C(N)=O)c[nH]c(C(=O)OC)c1 69660,C12CC3CC(C1)N(C3)CCO2.c1(CC)ccccc1OC 69661,C(=O)(C(=O)N=S(C)(C)=O)N1C(COC)CN(C(c2coc(C(F)F)c2)=O)CC1 69662,N1(C(C2(COC)CCCO2)=O)CC2(CC(NC(c3csc4nccn34)=O)C2)C1 69663,CC1CN(C(=O)CC2CC3(CCC3)C2)CC(C)N(C(=O)CCCCN(C)C)C1 69664,NC1(CC(=O)NCCOCCOCCOC2CCC(C3CCCCC3)O2)CCOC1 69665,C1(C(N(C2CCN(C(C3C=CCC3)=O)CC2)CC)=O)CC(O)CN1C(N)=O 69666,c1(C(=O)NC(CN(C(c2n(CC)ccn2)=O)C)(C)C)cc2ccc(Cl)cc2o1 69667,Cn1cc(Nc2cc(NC(c3cccc4c3OCC4)(C)C)ncn2)c(O)nc1=O 69668,N1(c2snc(C(=O)OC)n2)CCC2CCC(NC(c3ccc(F)c(Cl)n3)=O)C1C2 69669,CCC(C)C1C(=O)NN2C(=O)CC(C2)N1.C1(C(=O)NOCC)CC2CCC1CC2 69670,C12(C(=O)NCC(C)(C)CC3CCS(=O)(=O)C3)CC(C(F)(F)F)(CO1)C2 69671,CN1CC(O)CC1C(=O)NC1CCN(C(=O)C(F)(F)c2ccsc2Cl)C1 69672,C12(C(N3CCCC(OCC)C3)=O)CC(CCO1)N(C(C1CC(OC)C1)=O)C2 69673,c1(C(CNC(C2C(C(C)C)CCO2)=O)O)ccc(Cl)c(Cl)c1 69674,c1(C(N2CC(N(C)C(c3cc(Cl)c[nH]3)=O)C(F)C2)=O)ccnc(C(F)(F)F)c1N 69675,Cc1nc2ccc(C(=O)NC(C)CN(C(=O)CC3CCCNC(=O)C3)C)cn2n1 69676,c1(Oc2cccc(OC)c2)cccc2cncc(C(=O)OCC(C)(C)C)c12 69677,c1(CCC(=O)NC(C2CCN(C(C3CC(CC)(CC)C3)=O)C2)C)ncc(F)cn1 69678,C=CC1OCCC1C(=O)NC1CC(CCNC(C2CN(CC)CCO2)=O)C1 69679,CC1(C)CN(C(C2(F)CC=CC2)=O)CC1NC(C1CCC=CCC1)=O 69680,CCC(C)C(C)C(=O)N(CCCNC(=O)CCc1scnc1C)C 69681,C(c1cn(C)nn1)=CC(=O)NC(COC)C(=O)N(C1CC(F)(F)C1)C 69682,CC1(C)CC(C)(CNC(c2cc3cccnn3c2)=O)CN1C(=O)C(F)C(F)(F)F 69683,CC1(C)CCC(C)(C(N2CCC3(NC(=O)CC4(O)CCC4)CC3C2)=O)CC1 69684,C(CN=c1[nH]c(=N)[nH]c(=NCCN2CCCC(C)C2)[nH]1)c1ccn(N(C)CC)n1 69685,C1(CCNC(c2cn(CC)nc2)=O)CCN(C(c2ccc(C)cc2F)=O)C(C)C1 69686,N1(C(CCc2ncn(C)c2)=O)CCC(CNC(C2CC23CCC3)=O)C(O)C1 69687,C(=O)(N=c1cc(C)[nH][nH]1)C1CC2(CN(Cc3c(OC)ccc(Br)n3)C2)C1 69688,c1(C(CO)N(C)CC2CCCO2)ccccc1C(F)(F)F 69689,c1(C(=O)NC2CCC(CCNC(=O)C(F)F)C2)cc(F)c2ccccc2c1 69690,c1(C(=O)NC(CC)CNC(c2cnc(O)s2)=O)cc(OC(F)F)ccc1C 69691,C1(NC(Cn2c(=N)scc2)=O)(CNC(=O)C=Cc2cccnc2)CCOCC1 69692,C(=O)(C#CC(=O)N1CCCC(NC(=O)C(C)n2cccn2)C1)N(C)C 69693,N12CCC3CN(CCC13)C2=O.C1(CC)CC1C 69694,C1(C(=O)NC(C)(CNC(C2CCC(C(F)(F)F)CC2)=O)CO)COC2(CCC2)C1 69695,c1(C(=O)NCC2CC=CCN2)c(F)cc(Cl)cc1Cl 69696,C1(NC(c2sccc2F)=O)CCN(Cc2cc(Br)ccc2Br)CC1F 69697,c1(N2CCC(C)(CC)C2)ncccc1S(=O)(=O)N1CCC(CN(C)C)CC1 69698,C(=O)(C1=NOC(C(N2CC(NC(C3CCC(C)O3)=O)CC2C)=O)C1)OC 69699,C1(C(=O)NC2(CC)CN(C(C3CCCCC3)=O)C2)CCOCC1C 69700,c1(C(N2CCC(CN(C(=O)CCc3cnn(C)c3)C)C2)=O)ccc(N)c(F)c1F 69701,CC12CN(C(=O)CN3CCOC3=O)CC1CN(C(C1(C(F)F)CC(F)(F)C1)=O)C2 69702,N1(C(c2ccc(COC)cn2)=O)Cc2occc2CC1C(=O)OC 69703,C(CN=c1[nH]cnc2ccsc12)C1CCN(C(c2c(Cl)cn(CCC)n2)=O)C1 69704,N1(c2ncc(C(N(C3CCNCC3F)C)=O)cn2)CCN2CCCC2C1 69705,C(c1cn(C)cn1)=C(C(=O)NCC(C)CNC(=O)CSC(F)F)F 69706,CC(C)(C)CCC(F)C(=O)N1CCOC(Cn2cc(C3C4COCC34)nn2)C1 69707,N1(c2n(CC(=O)NCc3ccc(OC)c(OC)c3)nnn2)CCC2CCC(C2)C1 69708,c1(C(N2C3CC(C(=O)O)C2CC3)=O)cc(Br)cc2nc(O)[nH]c12 69709,C1(NC(CCc2onc(C)n2)=O)CC2CC1N(C(C1CC1(F)F)=O)C2 69710,Cc1nc(C)n(CC(N2CCCCC2C(=O)NCC(O)CN(C)C)=O)n1 69711,N1(C(COCC=C)=O)CC(NC(C2CCOC(C)C2)=O)C(c2nccn2C)C1 69712,C(CCC(O)C(=O)N(CCCC)CCO)NC(C(CC#C)C1CC1)=O 69713,C1(C(=O)NCC2CC(NC(C3(CCCC)CC3)=O)C2)COC2(CCC2)CO1 69714,C(CN=c1[nH]c(N2CCN(C3CCC3)CC2)nc2cc[nH]c12)C1C(O)CCC1 69715,c1(OC)cc(C)sc1C(N1CC(N(C)C(c2ccc(C)nn2)=O)C(O)C1)=O 69716,N(C1CCc2cccnc21)C(C1CN(C(c2c(C)c(I)ccc2)=O)CC(F)C1)=O 69717,N1(C(C2C(C)=C2)=O)CCC2(CC1)CC(n1cc(CC3CCOCC3)nn1)CCO2 69718,C1(C(C(=O)NCCNC(Cc2ccc(C(C)=O)s2)=O)C)CCCCCC1 69719,CC1(CCNC(C2(C)CCCCC2)=O)CCN(C(=O)C=C2CCCCC2)C1 69720,Cc1cc(Br)cc(S(=O)(=O)NCCC2(C)NC(=O)NC2=O)c1 69721,c1(C(c2n(CCCOC)nnn2)NC(CCO)CC(C)C)cc(OC)ccc1Br 69722,c1(NC(=O)NS(CC2(COC)CCOC2)(=O)=O)ccc(C(N)=O)cc1 69723,c1(OCC)cc(C(=O)NCC23CC(NC(c4cccnc4)=O)(CO2)C3)ccn1 69724,C1(CCN(C(C(=O)NCC(COCC)C)=O)C2CC2)CC[Si](C)(C)C1 69725,C1(OCC)(CNC(C2COC(=O)N2)=O)CN(C(=O)CN2CCOCC2)C1 69726,C1(NC(c2cn(CCOC)nc2C)=O)CN(C(C2CC3C=CC2C3)=O)CC2CC12 69727,CCC(C)(CNC(C1CC1(F)Cl)=O)C(=O)N(CC(C)(C)OC)C 69728,N1(CCCC(N2CCC(N(C(C(C)c3ccsn3)=O)CCO)C2)=O)C(=O)CNC1=O 69729,c1(OCC(=O)NC(CC=C)CNC(C2C3CC4C(C3=O)C24)=O)nc(O)nc(O)n1 69730,Cc1cccc2c1CC(C(=O)NCC1(C)CCCN1C(C1C3(CC3)C13CC3)=O)O2 69731,c1(CC)onc(C(=O)N(C2CCN(C(=O)CC3CCSC3)CC2)CC)c1C 69732,C(=O)(C(C(=O)N1CCOC(C(=O)NC23CC(C2)C3)C1)OC)OCC 69733,C(=O)(CC(C)CNCc1snc(C)c1N)OC 69734,C1(O)(CC(=O)N(CC(=O)NCC2(C)CCOC2)CC2CC2)CCCOC1 69735,Cc1cc(C(N2CC(F)CC2CNC(C2(C)SCCCS2)=O)=O)[nH]c1C 69736,C1(OC)CN(C(c2cnn(C)n2)=O)CC1NC(=O)C(C)C 69737,c1(C(=O)NC2CCCN(C(c3nccc(C)c3)=O)C2C)cc2cc(Cl)ccc2[nH]1 69738,Cc1cc(C(=O)NCC=CCNC(C2CC3CC(=O)C2C3)=O)nc(C(F)(F)F)n1 69739,C1(F)(C(=O)NCCCOCCCNC(c2c(C)ncnc2)=O)CCCCCC1 69740,C(=O)(CC(C)P(C)(C)=O)N1C(CNC(c2c(C)noc2)=O)CC(O)C1 69741,c1(C(=O)OCC2CC(=O)NC2)cc(Cl)c(F)cc1[N+](=O)[O-] 69742,CC(C)(C)CC(O)C(=O)NCCN(C(=O)CSCCc1ccccc1)C1CC1 69743,N1(C(C2(OCC)CCOC2)=O)CCC(C2(NC(=O)Cn3ccc(C)n3)CC2)C1 69744,CN1CCCC(CN(C)C(C2(NC(C3CCC3)=O)CCC2)=O)C1 69745,C1(CCNC(C(COC)C)=O)CSCCN1C(=O)CC1(O)CCCC1 69746,C1(F)(C(N(CC(C)N(C(=O)CC2CCN(C)CC2)C)C)=O)CC=CCC1 69747,CC1(CC(=O)NC2(CCCNC(c3cn(C4CC4)nn3)=O)CC2)CCOCC1 69748,n1(CC(N2CCCCC(NC(C3(O)CC(C)(C)C3)=O)C2)=O)cnc2ccccc12 69749,C(=O)(C(CC(C)(C)C)NC(=O)CNC(C1CC1C)=O)N1CC(OC)C(O)C1 69750,c1(C(=O)NC2CC(C)CN(C(c3csc(C#N)c3)=O)C2)cnc2ccccn12 69751,C1(NC(CC(=C)C)=O)CC2CN(C(=O)C#CC(C)(C)C)CC2C1 69752,C1(CNC(COCCC(C)C)=O)CN(C)CCN1C(=O)C(C)Cn1ccnc1 69753,C1(NC(C2(N(C)C)CCC2)=O)CC2CN(C(c3cccc(C#N)c3)=O)CC2C1 69754,N1(C(C(=COCC)C#N)=O)CC2(C1)CN(C(c1cncc(F)c1)=O)CC2CO 69755,O=C(C(Cl)=CCl)NC1(C2CCCN2C(C2CC2c2ccncc2)=O)CC1 69756,C1(C(=O)NCCCc2cccs2)CCCN1C(=O)C(c1ccccc1)O 69757,C1(C(=O)NC2(COC)CCCC2)C2CCC(C2)N1C(C1C=CC=CC=C1)=O 69758,c1(C(N2C(CC(=O)Nc3ccc(N(C)C)nc3)CC2)=O)ncc(F)cc1N 69759,CC1(C)CN2CC(O1)C2.c1(Cc2ncccc2C(=O)O)cc(F)cc(I)c1 69760,N1(C(c2c(C)cc[nH]2)=O)CCC2(CC1)CC2CNC(=O)C=Cc1ccc(Cl)cc1 69761,CCS(=O)(=O)CCN=c1[nH]c(N2CCOCC(CNC(C)=O)C2)nc2c1CSC2 69762,CC1COCC1(c1nnnn1CCC1CC1)Nc1ccc(-c2cnco2)cc1 69763,C(C(O)CC(C)(C)CO)NCc1cnn(C)n1 69764,C(=O)(C(C(C)O)N(C)C)NCC(C)CNC(=O)CCNC(c1ccsc1)=O 69765,C12(NC(CCCC=C)=O)CC(CNC(c3cc(C)n(C)n3)=O)(C1)OC2C 69766,C12(NC(c3ccc(F)c(O)c3)=O)CCC(C(N3CCC3CO)=O)(CC1)C2 69767,C(CC(C)(C)CNC(c1cc(C2CC2C)on1)=O)NC(c1cnc(SC)s1)=O 69768,c1(C(N(CC(CNC(COC(C)=O)=O)C)C)=O)ccc(N2N=CCC2=O)cc1 69769,C1(CC(=O)NCCCOC)C2CN(C(C3CCCOC3)=O)CC12 69770,C1(CC(=O)NCCNC(Cc2cn(C(C)C)nc2)=O)CC2(CCC2)CO1 69771,C(c1ccc(=N)[nH]c1)=CC(=O)NC(C)CN(C(=O)COc1ccc(Cl)cc1)C 69772,Cn1cc(S(=O)(=O)N2CCN(C(=O)CSC3CC3)C3CC23)cn1 69773,C1(N(CCOCCNC(C)=O)C(c2ccc(CO)s2)=O)CCCCCC1 69774,N1(C(CC2(COC)CC2)=O)CC(NC(=O)CCc2cnccn2)C(C(F)F)C1 69775,c1(SCC#C)cccc(C(N2CCC(CNC(c3cncc(F)c3)=O)C2)=O)c1 69776,N1(CC(=O)NCCC2(C(=O)NCCN3CCCCC3)CCC2)CCCC(O)C1 69777,C1(C)(C(=O)NCc2cccc(CNC(C(C)(C3CC3)OC)=O)c2)CCCNC1=O 69778,C1(C(=O)NC(CNC(C=CCCC)=O)(C)C2CC2)CC(=O)N(C2CCCCC2)C1 69779,c1(CNC(C=C(C)C(C)C)=O)cccc(CNC(C2(C)CC3CC3C2)=O)c1 69780,CCCCCCC(O)CCC(=O)NC1CC2CCC1N(C(C1CC(C)(C)C1)=O)C2 69781,c1(C(=O)NC2COCCC2NC(c2c(Cl)cccc2Cl)=O)cnc2ccsc2c1 69782,c1(C(c2n(C(CC)C)nnn2)NCC(CCSC)OC)cc(Br)c(C)nc1OC 69783,c1(NC(C2CC3(CCC3)C2)C)cnc2ccccc2n1 69784,c1(CC(N2CCC(CN(C(c3nnc(C)s3)=O)C)C2)=O)ccc2nn(C)cc2c1 69785,N1(CCC)CCC(N=c2cccc(S(=O)(=O)N(C)CC3CCN(CC)C3)[nH]2)CC1 69786,N1(C(=O)C(Br)Br)CCCC(Cn2cc(CN3CCCC3C(=O)O)nn2)C1 69787,c1(C(C(=O)N(C(CC)C)C)N(CC(=O)NC)CC)ccn2nccc2c1 69788,c1(COC)noc(CNC(C2CC(CNC(=O)CCN3CCCC3=O)CO2)=O)n1 69789,C#CCC(CC#C)C(=O)NC1CC(CNC(c2ccc(C)c(Br)c2F)=O)C1 69790,N1(C(C(C)C2(O)CCC2)=O)CCC(C2CC2)(CNC(C2C=CCC2)=O)C1 69791,N1(CC)CC(C(=O)NCC2CC(F)CN2C(=O)CCn2c(C)ccc2C)NC1=O 69792,C1(C(=O)NCCN(C(C2CS(=O)(=O)C2)=O)CC2CC2)CCCC1C1CC1 69793,c1(CC(N2CC3C(CNC(c4occc4Cl)=O)(C3)C2)=O)ccc(O)c(Cl)c1 69794,N1(C(C(c2scc(C)n2)C)=O)CCC(NC(C23CCC(CC2)OC3)=O)CC1C 69795,Cc1ccc(CC(=O)NCCC23CCC2CN(C(=O)CSC2CC2)C3)c(F)c1F 69796,CCC(C)CC(=O)NCCN(C(=O)CC(C)OC)C(C)C 69797,N1(C(Cc2nc(NC(c3n(C)ccn3)=O)sc2)=O)CCC(F)(C(N)=O)C1 69798,N1(C(CC2N(C)CCC2)=O)CCC(OCCNC(C2CCOC2)=O)CC1 69799,C1(CNC(=O)C(=C2CCCCC2)F)(CO)CCN(C(=O)CC2CC3CC3C2)C1 69800,c1(C(=O)NCC(C)NC(C2(CC=C)CCCCC2)=O)nc2nc(C)cc(C)n2n1 69801,CCC(C)(C)C(C)CC(=O)NC1CC12CCN(C(=O)CC(F)(F)F)CC2 69802,C(C(=O)NOCC1CCC1)(C1(C)CC1)NC(c1ncccc1N(C)C)=O 69803,c1(CN(N2CCCCCC2C(C)(C)C)C)ccc(Cl)c(F)c1.C=O 69804,C1(n2cc(C(C3CC=CCC3)=O)nn2)CCN(C(=O)C(F)(F)C(F)F)CC1O 69805,C(=O)(C1=CSCCO1)N(C1CN(C(c2csc(C(N)=O)n2)=O)CC1(C)C)C 69806,C(=O)(CCS(C)(=O)=O)NC1CC(CNC(C(C)OCC2CCCCO2)=O)C1 69807,C(=O)(CCC(C)NC(=O)C(C)(C)CNC(C)=O)NC(CCC)C 69808,c1(C(=O)NCC2C(C)CN(C(=O)CSc3ncccn3)C2)ccc(S(N)(=O)=O)o1 69809,S(=O)(=O)(c1cc(C(=O)NCC2CC2NC(C2(Cl)CC2)=O)ccc1OC)NC 69810,C(CN=c1cc(NCC2(CN3CCOCC3)CCCCC2)nc[nH]1)(C(C)C)OC 69811,C#CCC(C)(CNC(c1cc(C)ncn1)c1nnnn1CCCCCC)CO 69812,c1(C(=O)NC2(CNC(CC3(OC)CC3)=O)CCCCCC2)ccc2nc(C)oc2c1 69813,c1(C2N(C(c3cc(Cl)ccn3)C(=O)NCCSC)CCC2)cc(F)cc(F)c1F 69814,C#CCC(C)(CC)C(=O)NCC(CNC(c1c(C)[nH]c(C)c1C)=O)OC 69815,Cc1cccn2cc(C(=O)NC3CCN(C(=O)C(C)n4cncn4)C3C)nc12 69816,c1(CC(=O)NC(CN(C(CCSCCC)=O)C)C)c(C)cc(OC)cc1C 69817,C1(NC(Cc2n(C)ccn2)=O)CCC2CN(CCCCc3ccccc3)CC2C1 69818,c1(C(=O)NCCCCNC(c2nccc(C(N)=O)c2)=O)ccc2n[nH]cc2n1 69819,CCC(C(=O)NC1(CF)CN(C(C2CCSC2)=O)C1)C(C)(C)CC 69820,c1(CNCCC(C)OC)ccc2nc(C)n(C)c2c1 69821,c1(OC)ccc(NC(=O)C(=O)NCc2ccsn2)cc1OC 69822,C(C(=O)N(C)CC1CCN(C(C2CCC(C(N)=O)CC2)=O)C1)(C(C)C)SCC 69823,Cc1cnccc1N1CCN(c2nnc(C3CC3)n2CCc2ncn(C)n2)CC1 69824,N1(C(C2ON=C(C)C2)=O)CC(NC(c2cc(C)nc(Cl)c2N)=O)CC12CCCC2 69825,CCC(CC1CCCC1)CC(=O)NC1CC(CNC(=O)CCCc2ncco2)C1 69826,CC1=NOC(C(N2CCCC2CCNC(c2cnc(C(C)(C)C)o2)=O)=O)C1 69827,CCCCC(CNC(C1CCN(CC)C1)=O)NC(=O)C(C)(O)c1ccccc1 69828,C1(NC(c2c(C)nn(C)c2)=O)C2CCC(C2)C1C(=O)NC1C2COCC12 69829,C1(C(=O)NC(C=CC(=O)NC(C)Cc2ccncc2)C)CCC(C)(C)O1 69830,C=CC(C)(C)CC(=O)N1CC(C(F)(F)F)CC1CNC(=O)CCC1CCC1 69831,C1(C(C)NC(=O)C=C2CCCC2)CCCN(C(=O)Cc2ccc(Cl)cn2)C1 69832,C1(OC)CC(C(=O)NC(C)C(CO)NC(C2CC(SC(F)F)C2)=O)N(C(C)=O)C1 69833,CC1CC(NC(C2C(C)OCCN2C(=O)CC2(C)CCCCC2)=O)C(C)CN1C 69834,C1(NC(Cn2c(C)ncc2)=O)CCCN(C(c2cncc(C3CC3)c2)=O)CCC1 69835,C1(C(C(N2CC(CO)(NC(C3(CO)CC3(F)F)=O)C2)=O)O)CCCCCC1 69836,CN1CCN(CCC(N2CC3C(NC(=O)COc4ccc(Cl)cc4)C3C2)=O)CC1 69837,C1(C(N2CCC(N(C(=O)CS(=O)(=O)NC(C)(C)C)C)C2)=O)CC(=O)NC(=O)C1 69838,CC1(C)CCCN(C(=O)C(F)C(C)(F)F)C1C(=O)NCCC1COCC1O 69839,c1(NC(=O)NCC(C2CCCCCC2)C)ccc2c(c1)N(C)CCO2 69840,N1(CCc2c(OC)cccc2)C2CCCC1CC(O)C2.n1(CC(=O)O)cccn1 69841,O=S(=O)(c1cnn2ccc(N3CC45CCC4(COC5)C3)nc12)N1CC2CC1CS2 69842,C(CCCC(=O)NCCn1cc(C(=O)NC2CC3CCC2C3)nn1)OC 69843,O=C1CCC(C(=O)NC2CCCCC2NC(=O)Cc2c[nH]ccc2=O)=NN1 69844,C(=O)(CCC(C)S(C)(=O)=O)NCC(CCOC)NC(=O)CCc1c(C)n[nH]c1C 69845,Cn1cc([N+](=O)[O-])c(-c2nnc(-c3ccn(C)n3)o2)n1 69846,c1(CSCc2n(CC)nnn2)ccc(C)c(F)c1F.c1(O)ccccc1.C12(CC1)NC2 69847,N1(C(=O)Nc2ccccn2)CCC2(CCN(S(=O)(=O)c3cncc(Br)c3)C2)C1 69848,c1(NC(c2n(COC)ncc2)=O)ccc(Br)c(OC(F)(F)F)c1 69849,C(=O)(C(=O)N=c1ccn(C2CCOC2)[nH]1)NCCC1CCC(C)O1 69850,N1(CC(C2C(C)C2C)=O)CC2CCC1CN2C(C)C.C12CN(CC1C)C(=O)C2 69851,Cc1ccc2cc(C(=O)NCc3cc4ncccc4[nH]3)[nH]c2n1 69852,C(=O)(CCCCCF)N1CCC(CNC(=O)C(N2CCCC(OCCO)C2)=O)C1 69853,n1(COC)nccc1CN(C1CNC(=O)C1)C 69854,CC1C=C(C(=O)NCC(c2ccccc2)NC(=O)C=Cc2ccc(F)cc2)CC1 69855,N1(C(CC(C)OC)=O)CCCC12CCN(C(C1CCN(C)CC1)=O)C2 69856,c1(C(N(C2CCCC(NC(=O)C=C3CCC3)C2)C)=O)[nH]ncc1C#N 69857,c1(C(=O)NCC(C)N(C(C2CCC(C)(CC)O2)=O)C)cnn2c1NCC(C)C2 69858,C1(C(=O)OC)CCN(C(=O)CC2(C)CCN2C(=O)C(OC)OC)C1C 69859,n1(CC(=O)N(C)CC2CN(C(=O)OC(C)(C)C)C2)ncc2cc(Br)ccc12 69860,Cc1cc(NC(=O)CC2CCN(C(c3cn[nH]c3)=O)C2)cc(C#N)c1 69861,C(=O)(CCCC(C)(C)C)N(CC(C)(C)CNC(=O)CCCOC(=O)CC(C)C)CC 69862,N1(C(C2N(C(CN(CCOC)C)=O)CCOCC2)=O)CCCN(C)CC1C 69863,c1(C(N(CCC(C(C)C)Nc2nnccc2C#N)C)=O)c(Cl)cccc1Cl 69864,C1(CCC(=O)NC2(CC(C)C)CC2)CCN(C(=O)Cc2cscn2)CC1 69865,Cc1n[nH]c(C)c1CCC(=O)NC(C)CNC(=O)CC1CC1C(F)(F)F 69866,C(CC(C(C)(C)C)NC(C1(O)CC1)=O)N(C)C(c1cnc(Cl)cc1N)=O 69867,c1(CC)ccc(C(=O)NC2CC2c2ccco2)cc1OCCSC(C)=O 69868,N1(C(C2CC(C)CN(C(C3(C#N)CC3)=O)C2)=O)CC2(C1)NC(=O)NC2=O 69869,C1(CNC(C(CC2CN(C(CP(C)(C)=O)=O)C2)F)=O)CCC2(CCC2)O1 69870,Cc1ncc2n1CCC(C(=O)NC1COC3CN(C(C4SCCCS4)=O)CC13)C2 69871,CCC(C(=O)NCC1CC(O)CN1C(=O)C1=CCC1)C(C)(C)CC 69872,c1(C(N(C(C)C(c2cnnn2C)=O)C)=O)ccc2ncc(Br)n2c1 69873,N1(C(COC(CC)C)=O)C2CCC1CC(C(=O)Nc1cc(C)nc(C)n1)C2 69874,C=CCCC(C(=O)NCC(C)CCC)NC(=O)C(C)NC(=O)OC 69875,C1(NC(c2c(CN(C(=O)CSc3cn[nH]c3)C)cco2)=O)CC(O)C1(C)C 69876,C(=O)(CS(F)(F)(F)(F)F)NCCN(C)C(c1ncsc1C1CC1)=O 69877,CC1(C2CC2)CCN(C(=O)C(Cc2cc[nH]n2)NC(=O)COC2CCOCC2)C1 69878,N1(C(C(C)(C)NS(C)(=O)=O)=O)CC(NC(=O)COCCCF)C(O)C1 69879,C1(NC(CCOCC)=O)CC1C1CCN(C(c2cn(C)nc2C)=O)CC1 69880,c1(C(=O)NC(CC)(C)CNC(C2(C)CSC2)=O)cncc(-c2ccccc2)c1 69881,CCCC(C(O)C(=O)NCc1ccc(F)nc1C)NC(c1cc(N)cc(F)c1)=O 69882,N1(C(C(C)=CC)=O)CC(NC(=O)CCOc2cccnc2)C2(CCOCC2)C1 69883,CC(C)CC(C)(CNC(=O)CC1CCC1)NC(c1cc(C(F)(F)F)cc(F)c1)=O 69884,c1(C(C)C)nn(C)cc1NC(=O)C(O)CNC(c1ccc(F)cn1)=O 69885,C1(C(=O)NCC(c2ccccc2)(C)O)CCN(Cc2ccnc(F)c2)CC1O 69886,CCC(CC(=O)NCC1CCCN1C(=O)CC1(C(F)(F)F)CCC1)C(F)F 69887,N1(C(CC2N(C(c3c(OCC)cccc3)=O)CCC2)=O)CC2OCC(CO)C2C1 69888,C12(CNC(C(CO)OC)=O)CCCN(CC1)C2 69889,N1(C2C(O)CCCCCC2)CCC(O)c2cc(Cl)ccc21 69890,N1(C(C(C)(C)SC)=O)CCCCC2(CCN(C(C3(C)CCCNS3(=O)=O)=O)C2)C1 69891,c1(NC(C)=O)cc(C(=O)NC2CC2CNC(=O)CCCn2ccnc2)ccn1 69892,N1(C(C(CO)OC)=O)CCCCC(C(=O)NCc2cnco2)C1 69893,c1(C(=O)OCC)ccc(NNC(=O)CSC2COc3ccccc3O2)cc1 69894,C1(NC(=O)Cc2cccs2)CC(F)CN(C(c2ccc(F)c(O)c2)=O)C1 69895,C1(NC(C2N(C)CCOC2)=O)CN(C(c2csc(-c3cccs3)n2)=O)CC12CC2 69896,c1(C(=O)Nc2c(CC)c(Br)ccc2)cn2c(n1)CN(C(=O)C(O)O)CC2 69897,C(C)(CCC(C)C)(c1nnnn1CCN1CCOCC1)NCc1nc(C)c(C)s1 69898,Cc1nn(CC(=O)NCC(C)(F)CNC(=O)C(C)(C)CC2CC2)c(=O)o1 69899,CC1(C)C(NC(C2CC3CC(=O)C2C3)=O)C2CCCN(C(=O)CCC3CCC3)C12 69900,N1(C(COC)=O)CCC(NC(=O)C(=O)N(CC(C)(C)Oc2nnc(C)o2)C)C1 69901,C1(NC(CSCC#C)=O)CC(CNC(c2cc(C)n(C)c2C)=O)C12CCC2 69902,c1(C(=O)NC2(CCNC(C(C(CC)O)C)=O)CC2)cc2oc(Br)cc2s1 69903,C#CCCN=C(NCc1ccc(Br)c(O)c1)NC1CCS(=O)(=O)C1 69904,N1(C(C2(C)CC(C)C2)=O)CCC(CCCCNC(C2(C(F)(F)F)CCC2)=O)CC1 69905,c1(C(N2CC(NC(CC3(C=C)CCCCC3)=O)C(C)C2)=O)cccc2nccn12 69906,CC1CN(C(C2(c3ccnn3C)CC2)=O)CCCN1C(=O)CC(C)(C)C#N 69907,CC1=NC(C)(CNC(C2(CNC(C3CCNC3=O)=O)CCCO2)=O)CS1 69908,c1(OC)ccc(C(=O)NC(C2CN(C(c3sccc3C(F)F)=O)C2)C)c(OC)n1 69909,C1(N(C(c2cc(C)n(C)n2)=O)C)CN(C(=O)Cc2c(O)ncnc2O)CC1(C)C 69910,C1(N(C(c2c(SC)cn(C)n2)=O)C)CCN(C(=O)C(C)(C)c2cscn2)CC1C 69911,C12(C(=O)NC(C)CCNC(=O)CCN3CCCC3)CCCC(CCC1)C2O 69912,c1(NC2CC(F)(CNC(CC(C(C)C)C)=O)C2)cc(O)nc(=O)n1C 69913,C1(OC)CCC(C(=O)NCCC(O)CNC(c2cc(C(C)(F)F)n[nH]2)=O)CC1 69914,c1(OCC)ccccc1-c1nc(C2COCCO2)n(C2CCOC2)n1 69915,C1(NC(C(COC)C)=O)(CO)CCCN(C(c2ccn(CC(F)F)n2)=O)C1 69916,c1(SCC)cc(Cl)ccc1C(=O)NCC1CC(O)(CNC(C2CCS2(=O)=O)=O)C1 69917,c1(C(N(C2CCN(CCc3ccccn3)CC2)C)=O)cc2ccsc2[nH]1 69918,c1(CN2CC(NC(c3scc(C)c3)=O)C(O)C2)cccc(S(C)(=O)=O)n1 69919,N1(C(C2N(S(C)(=O)=O)CC2)=O)CCCC(C)(NC(c2cc(C3CC3)ccn2)=O)C1 69920,N1(C(c2c(CC)oc(C)c2)=O)CC2CN(C(c3cccc(O)n3)=O)CC(C1)O2 69921,C1(NC(=O)CCc2ncc[nH]2)CCCCN(C(C2CC3(CCC3)CO2)=O)CC1 69922,C1(CC=C)(NC(=O)COC(C)=O)CCN(C(c2cc(O)nn2C)=O)C1 69923,n1(CCN(C(=O)C(CC2CCOC2)OC)CC)cc(C(O)C2CC2)nn1 69924,C#CCC(CC(F)F)C(=O)NCC(F)(C(=O)N(CC(C)O)C(C)C)C(C)C 69925,Cc1cc(C(N2CCCCC2CN(C(=O)C(F)(F)C2CCCC2)C)=O)ncc1N 69926,n1(CC(=O)OC)cc(C(N(C(c2ccc(Br)o2)=O)CC)C2CC2)nn1.C1CCOC1 69927,C(C(C)C)(C(O)C(=O)NC(Cc1cnc[nH]1)C(N1CC(C2(C)CC2)C1)=O)OC 69928,c1(CC(N2CC(CC(C)NC(C3CC(F)CN3C)=O)C2)=O)ccc(Cl)nc1 69929,CC(CC(=O)NCC=CCN(C(=O)NC(C)(C)C)C)OCCOC1CC1C 69930,c1(OC(CC)C)cccc(=NC(=O)Cc2cccc(CN=S(C)(=O)N(C)C)c2)[nH]1 69931,N1(C(c2ccc(NC)cc2)=O)CC(C(=O)Nc2ccsc2CO)CC(C)C1 69932,Cn1nnc2c(N3C4CCC3C(CNC(C3(C)C=CCC3)=O)C4)ncnc12 69933,C(C(CC(C)C)C(=O)NC1CC(O)CC1O)NC(c1c(C)noc1C)=O 69934,Cc1n[nH]c(C)c1CC(N1CCC(OC2CN(C(c3cnc(S)[nH]3)=O)C2)CC1)=O 69935,C1(CC(=O)OC)CN(C(c2ccc(OC)c(F)c2)C(=O)NCC(C)C)C(C)(C)C1 69936,c1(C(C(=O)NC(COC)CNC(=O)CCOCC(F)F)O)ccc(F)c(Cl)c1 69937,N1(C(CCN(CCC)C)=O)CCN(C(C2C=CC=CC=C2)=O)CC1C 69938,C=CCCCC(C1CC1)NC(=O)C=CC(=O)OC.C1(=O)C(C)C(C)N1CC 69939,c1(C(=O)NC2CCN(C(C(CCC)C)=O)CC2)sc2ccccc2c1Cl 69940,C1(NC(C(CC(=C)C)C)=O)CN(C(c2cc(C3CC3)nn2C)=O)CC2CCCC12 69941,c1(CSCC)ccc(C(=O)N(C2CC(SC)C2)C)cc1.c12cncc(c1)C(=O)N2 69942,N1(C(C(N(C(c2c(OC)nn(C)c2)=O)C)C2CC2)=O)CCC(F)(C#N)C1 69943,N1(C(c2c(C)c(Br)cnc2)C(=O)NCC(C)C)CC(C#N)C2(CCC2)C1 69944,c1(C(N2CC(CN(C(c3ccc(OC)c(O)c3)=O)C)C2)=O)c(F)ccc(F)c1Cl 69945,C(=O)(CCS(=O)(=O)C(F)(F)F)NCC(C)CNC(=O)CSC1CCCCO1 69946,c1(OC(C(=O)NCC(CC)NC(C2CC(O)C2)=O)C)ccc(Br)cc1 69947,c1(C(=O)NCC(CC)NC(c2coc(C3CCCC3)n2)=O)ccn2ncnc2c1 69948,c1(C(=O)NCCCCCCNC(CCCC)=O)c(Cl)ccc2ccoc12 69949,c1(C(N2CCC(NC(C3(C#C)CCC3)=O)CC2)=O)ccc2oc(N)nc2c1 69950,c1(C(=O)NC2CCN(C(CN(CCC#C)C)=O)CC2)cncc2ncn(C)c12 69951,c1(NCC2CC(NC(C(C=CCCC)O)=O)C2)ccc([N+](=O)[O-])cc1S(C)(=O)=O 69952,C1(NC(c2c(C)nn(C(C)C)c2)=O)CC2(C1)CN(C(=O)C(C)C(C)C)C2 69953,C12(NC(=O)CNC(C3CC4CC3CC4=O)=O)CCC(C1)C(O)C2O 69954,N1(C(C(C#C)(C)C)=O)CCC(NC(=O)CC2CCC(=O)N2CC)C(C)(C)C1 69955,S(=O)(=O)(c1cccc(=NCCCOCCO)[nH]1)NCCN1CCC(=O)NC1=O 69956,C1(NC(c2c(NCC)scn2)=O)CCCCC1CNC(=O)C(C)(C)C 69957,C1(C(=O)NC2CC(N(C)CC)C2)CN(C(=O)Cc2cc(C)nn2C)CC12CC2 69958,C1(C(CNC(C2(CC3CC3)CC2)=O)NC(CCN(C(CCC)C)C)=O)CCCCC1 69959,c1(C(N2CC(NC(=O)CC3(C#N)CC3)CC(C)C2)=O)c(F)cc(F)cc1Br 69960,CCCC(C)(CC)C(=O)NCC1CCCCC1NC(C1CCCC1S(C)(=O)=O)=O 69961,c1(OC)cc(C(N2CCN(C(=O)COCC3CCCC3)C(CF)C2)=O)cc(F)c1 69962,C1(CC(=O)N(CCCNC(=O)C(C)NC(N)=O)CC)COCCOC1 69963,CC1=C(C(=O)NC2CN(C(c3cccc(CCc4cnc[nH]4)c3)=O)C2)CCO1 69964,C1(CNC(Cc2c(C)cc(C)s2)=O)CCC(C)CN1C(=O)CCCCC1CC1 69965,C12(NC(c3cc(C)n(C)n3)=O)CCC1CN(C(=O)C(O)(C1CC1)C1CC1)C2 69966,CCC(CC)(CC)C(=O)NCCC1CC(NC(c2ccc(C#N)c(Cl)c2)=O)C1 69967,Cc1cc2[nH]c(=O)c(C(=O)NC(C)CN(C)C(C3CCCC(C)CC3)=O)cn2n1 69968,C1(CC(F)(F)F)C(C(=O)OC)CCCN1C(=O)NCCN(C)CCO 69969,CC(C(=O)NC1(C(=O)NC(c2ccc(F)cc2)C)CCN(C)C1)C(F)F 69970,N1(C(c2ccc(CNC(C)=O)o2)=O)CCC2CN(C(=O)Cc3cncn3C)CC12 69971,C12(NC(COCCCC)=O)CCN(C(c3cc(C)c(CC)s3)=O)CC1C2 69972,c1(OCCN(C)C)cccc2c1CCN2c1ncnc(C2C3C4CCC(C4)C23)n1 69973,N1(C(C(C)OCC(C)C)=O)CC(NC(=O)CCNC(c2ccoc2)=O)CC(O)C1 69974,Cc1nc(C(=O)NCC2CC2NC(=O)CCC=CBr)cn1C(F)F 69975,C=C=CCCC(=O)NC1CCC(C)(CNC(=O)CCN(CCCCC)C(C)C)C1 69976,C#CCC(O)C(=O)N(C1C=CCN(C(=O)CC(F)(F)F)C1)Cc1ccccc1 69977,c1(C(=O)NC2C(NC(c3n(CC)ccn3)=O)CCOC2)c[nH]c2ccc(F)cc12 69978,N1(C(CC2CC(C)(C)OCC2)=O)CCC(NC(=O)C(C)(F)F)CC(O)C1 69979,N1(C(CC2C(C)=NNC2=O)=O)CC(=O)NCC1C(=O)NC1CCOC(C)C1 69980,CC(N=c1[nH]nc(C2CC2)s1)C1CCN(C(c2ncn3ccccc23)=O)CC1 69981,C(CC(C)(C)C)(C(=O)NCC1CCC1)NC(C(CCCC)C)=O 69982,c1(CNC(C2CNC(=O)N2)=O)ccc2c(c1)CCC2NC(=O)C=Cc1cn[nH]c1 69983,C(=O)(C1CCCc2cccnc21)NC1CCCN(C(c2ccc(C)o2)=O)CC1 69984,C(=O)(CS(=O)(=O)CCO)NC(C)CCCNC(C1CCCOC1C)=O 69985,c1(NC(=O)NC(c2ccccc2)C(C)NC(c2cnoc2)=O)cccc(Cl)c1F 69986,N1(CCNc2cn(CC(=O)Nc3ccco3)nn2)CCN(C(N(C)C)=O)CC1.C1(CBr)CC1 69987,c1(C(N2CC(CNC(=O)C=Cc3cc[nH]n3)C3(C2)CC3)=O)cc(F)c(Cl)cc1Cl 69988,N#Cc1ccnc(C(=O)NCC2CC(NC(c3ccc(CO)o3)=O)C2)c1 69989,C1(CC(=O)NCCCN(C(C2CC2C(C)(F)F)=O)CC)CC2CCC1O2 69990,C(CC(C)CCNC(c1coc(C(F)F)c1)=O)NC(C1CCC(C(=O)OC)C1)=O 69991,Cc1c(C(=O)NC2CCC23CN(C(C2CCCS2)=O)C3)oc2cc(Cl)ccc12 69992,C1(C)(C(=O)NC2COCCN(C(Cc3c(C)n[nH]c3)=O)C2)CCCCCCC1 69993,C1(C(=O)OC)CCC(CCNC(N2CC(CC(=O)OC(C)(C)C)C(C)C2)=O)CC1 69994,C1(CC(=O)NC2CC(C(C)NC(C3CC(O)C3)=O)C2)CC2(CCC2)CO1 69995,S(=O)(=O)(c1cccc([N+](=O)[O-])c1)NC(C(=O)N(C1CNC1)CC)C 69996,N1(C(C=CC(C)(C)SC)=O)Cc2ccccc2CC1CNC(c1ccc(C)o1)=O 69997,N1(C(C(N2CCC(C)C2)=O)=O)CC(C)N(C(c2cc(F)cc(Cl)c2N)=O)CC1C 69998,c1(CC(=O)NCC(O)CCNC(c2cc(-c3cccs3)[nH]n2)=O)ncc(Cl)s1 69999,c1(C(=O)NC2CC(C)N(C(=O)C(O)CCc3ccccc3)C2)cnc(F)c(Cl)c1 70000,CC(F)(F)CC(=O)NC(C1(O)CCCCC1)C(=O)NCc1ncn(C2CC2)n1 70001,C1(C(=O)OC(C)(C)C)CC2(CCC(COC(c3ccc(I)cc3)=O)O2)C1 70002,c1(CNC(c2cccc(C(C)N)c2)=O)nccc(Cl)c1F 70003,N=c1nc(NCc2noc(CCC(=O)O)n2)cc[nH]1 70004,c1(C(=O)NCC(C)N(C)C(C2CCC3C(C2)C3(F)F)=O)cnc2c(Cl)cccn12 70005,c1(C(=O)NCC(CC)NC(=O)C2=CCOC2)ccnc2c(F)cccc12 70006,CCCC(CC)CCC(=O)NCc1cc(C(N2CCOC(CC)C2)=O)on1 70007,c1(C(N2C(CNC(C3(C#N)CCOC3)=O)CC2)=O)ccc2ccnc(Cl)c2n1 70008,c1(C(=O)NCC(CNC(C2(OC)CCSC2)=O)O)cc2c(ccn2C)[nH]1 70009,Cc1cc(N(CCCNC(c2cnn(C(F)F)c2)=O)C(C)C)nc(Cl)n1 70010,C1(CCNC(CSCC#C)=O)CN(C(=O)C(C2CC(F)(F)C2)OCC)CCCO1 70011,Cn1nc(C(=O)NCC2CC2NC(=O)CC2CCC(C)(O)CC2)c2c1CCSC2 70012,NC1(C(=O)NCCCCN2CCCCC2)CC(C(F)F)C1 70013,Cc1ccc(CC(=O)NC23CCN(C(c4ccc(N)cc4Cl)=O)CC2C3)cc1C 70014,CC1(NC(=O)C(N2CC3CCC2C3)=O)CCC(C(F)(F)F)CC1 70015,C(CCCN(C(C)C(=O)NC(=O)N(C)CC1CCOC1)CC)OC 70016,CC(C)CC(C)(O)CNC(=O)CCOC1CN(C(c2cnc(Br)s2)=O)C1 70017,C1(NC(c2cncc(O)c2)=O)CN(C(=O)CCc2ccc(F)cc2)CC1F 70018,N1(C(c2c(C)cco2)=O)CCc2ccccc2C(N(C)C(=O)CSCC(C)C)C1 70019,C(=O)(C1=CC2C=CC1C2)N1CC2C(NC(c3nccc4ccsc34)=O)(C2)C1 70020,Cc1ccc(CC(N2CC(NC(C3(F)CC=CCC3)=O)C(C(F)F)C2)=O)cc1 70021,c1(C(C(CC)(F)F)(C)C)cn(C2c3cccc(Br)c3C2C)nn1 70022,c1(C(N2CC3(C(C(=O)Nc4ccc(C)c(I)c4)C3)C2)=O)cnn2cccc(F)c12 70023,c1(OC)nc(C)ncc1C(=O)NCCCCN(C(=O)C(C)CC1CCCO1)C 70024,C1(C(=O)OC)CCC(OC)(NC(=O)CC(c2ccc(C(C)C)cc2)C)CC1 70025,Cn1cc2c(C(N3CC4CCCN(C(=O)Cc5cc[nH]n5)C4C3)=O)cccc2n1 70026,C(C(N=c1ccc2nnnn2[nH]1)C(C)C(C)C)NC(Cn1c(C)nc([N+](=O)[O-])c1)=O 70027,C1(NC(C(C2CC2)SC)=O)CCCCCC1NC(=O)CC#N 70028,N1(C(c2c(C)nc(CCC)s2)=O)CCC(NC(C2CCCCN2CC)=O)C(F)C1 70029,O(NC(=O)CNCCCO)CC(=C)Cl.C(=O)CCOCC(C)C 70030,CCCCCCC(F)C(=O)NCCN(CC(C)O)C(c1ccnn1CC)=O 70031,C#CCC(CC(=O)NC(C)C(=O)NC)NC(C1CN(C)C1)=O 70032,O=C(C1=CCSC1)NC1CC(F)(CNC(C2CCC(=C3CCC3)CC2)=O)C1 70033,c1(C(N2CC(N(C(CCCCN(C)C)=O)C)C(F)C2)=O)ccc(F)c(N)c1 70034,Cc1ccc(NC(C2(Sc3ccc(Br)cc3)CC2)=O)c(O)n1 70035,c1(C(N2C(C(=O)Nc3cc(Cl)ccc3CO)C=CC2)=O)cc(Br)cc2[nH]ncc12 70036,CCCC(CC)CCC(=O)NC12CC1CN(C(c1nnc(O)nc1O)=O)C2 70037,c1(C(=O)NC(CC=C)C2CC2)cnn(CCNC(C)=O)c1 70038,C1(NC(CN(C(=O)C(O)C2CC2)CCOC)=O)COC2(CCCC2)C1 70039,Cc1ncccc1C(=O)NCCCCN(c1nnnn1-c1ccccc1)C(C)C 70040,c1(N2CC(C)(C)C(NC(C3CCCCO3)=O)C2)nccc(S(C)(=O)=O)n1 70041,C1(C(=O)NC(C(C)NC(c2ccco2)=O)C)CC(=O)N(CCc2ccccc2)C1 70042,CCC(C(=O)NCC(C)CN(C(=O)C(C)C#N)C)n1ccc(C2CC2)n1 70043,CCCCC(CNC(c1c(Br)ncn1C)=O)NC(c1ccc(C)s1)=O 70044,c1(C2CCCC(NC(N3CCC(Oc4ccncc4)C3)=O)C2)ccc(F)c(F)c1 70045,c1(C(N(C)CC2C(NC(CNC(CC)=O)=O)CCC2)=O)ccccc1SC 70046,c1(CC)cc(N)ccc1C(=O)NC(C)(CNC(c1oncc1C)=O)CC 70047,CCCCCC(=O)NCC(N1CC(N(C(=O)C(C)(O)Cc2ccccc2)C)C1)=O 70048,N1(C(c2c(C)oc(Br)c2)=O)CCC2(CC(NC(C3CC(CCO)C3)=O)C2)C1 70049,C1(NC(c2cc(CC)nc(O)c2)=O)CCC(O)CN(C(=O)CC2CN(C)C2)C1 70050,N1(C(c2c(OC)scc2)=O)CC2CC2(NC(=O)Cn2cc(C3CC3)nn2)C1 70051,C(=O)(C1CCCc2sccc21)NC1C(C)CN(C(c2ncn(C(C)(C)C)n2)=O)C1 70052,C(c1ccc(F)cc1)=CCC(N1CCC(N2CCC(NC(C3CC3F)=O)CC2)C1)=O 70053,C(=O)(C(C)(C)C(N)=O)NCC1(COC(C)(C)C)CCN(C(=O)CC2CC2)C1 70054,NS(=O)(=O)c1ccc(C(N2CC3CC(C2)N3C(=O)CCc2ccco2)=O)o1 70055,c1(C(=O)NCC2C(NC(=O)CCc3ccncc3)CC2)n[nH]c2c1COC2 70056,c1(C(=O)NCC2CCC(NC(=O)C(Cl)=CCl)C2)cn2ncccc2n1 70057,N1(C(CC(COC)C)=O)CCN(C(C2(C#N)CC=CC2)=O)C2(CC2)C1 70058,c1(C(=O)NCC2(OC)CCN(C(=O)C(C)CF)C2)ccc(Cl)c(C)c1 70059,C(c1nc2ccccc2o1)=CC(=O)N(C(C)CNC(c1ncnc(O)c1F)=O)C 70060,C(CC(C(=O)N(C1CCCC1)C)NC(c1csnn1)=O)=CC 70061,C1(CN(C(c2cnc(C(F)(F)F)s2)C(=O)NC2CCC2)CC)CCCOC1 70062,CC(C)C(CC(=O)NCCCc1cc[nH]n1)NC(=O)C(c1ccn(C)n1)C 70063,CCC(C)(C)C(O)C(=O)NC1(C2CCN(C(C3CCC(=O)N3)=O)C2)CC1 70064,Cc1cc(C)c(C(=O)NC2CN(C(=O)CC3(CO)CCCC3)CCC2C)c(C)n1 70065,C1(NC(c2csc(O)n2)=O)CC2CC1N(C(C1CN(CC(F)(F)F)C1)=O)C2 70066,c1(Cn2cc(N(CC(CC)N(C)C(=O)OC3CC3)CC)nn2)cccc(F)c1 70067,C=CCC(CC=C)C(=O)N1C2CCC1CC(NC(c1nocc1C(C)C)=O)C2 70068,C1(CCC(=O)NCC(=O)NCC(=O)NC(C2CCCO2)C)CCOCC1 70069,CC(C(=O)NC(CC1CCC1)C(=O)NCCc1cnco1)C(F)(F)F 70070,c1(CNC(C(C)c2ccco2)=O)ccnc(C(=O)NCCN2CCCCC2C)c1 70071,N1(CC(=O)Nc2c(NC(C)=O)c(Cl)ccc2)CCC2(C=Cc3ccccc3O2)C1 70072,C1(C(N(CC=C)CC)=O)CC(NC)CN1C(=O)OC(C)(C)C 70073,N1(C(C2C=CCN(C(c3c(CC)n(C)nn3)=O)C2)=O)CCC2(CCC(O)C2)C1 70074,N(C1CCOc2ccccc21)(CC(N)=O)CC(C1CC1(F)F)=O 70075,n1(CCNC(C2(c3ccncc3)CC2)=O)cc(CCCCCC2CC2)nn1 70076,N(C(=NCCC(C)(C)C)N(C)Cc1ccc2c(c1)OCCO2)C(C)C 70077,c1(C(=O)NCC2CCCCN2C(=O)CCC2CC2CC2CC2)nnn2c1CCC2 70078,C(=O)(CC(C(F)(F)F)P(C)(C)=O)N1CCC(N(C(=O)C#CC2CC2)C)C1 70079,n1(CC)cc(Cl)c(=NC(=O)N2CCNC(C)(C)C2=O)[nH]1 70080,CCC(CCCC(=O)NCC1Cc2nccn2C1)NC(=O)Cn1cccnc1=O 70081,c1(COC)csc(C(=O)NCCN(C(=O)C(=O)N(C)C)CC2CCCC2)c1 70082,CCCC(CC)C(=O)NC1CCC(NC(=O)COCC=Cc2ccccc2)CC1 70083,c1(C(=O)NCCCN(C(C(n2ccc(C)n2)C)=O)C2CC2)cccc(C)c1C 70084,N1(CC)CCOCC1C(=O)NC(C(=O)N(C)CCC1CN(C)C1)C1(O)CCC1 70085,C(=O)(C(O)CC(N)=O)NC1C(C)CN(C(=O)CCCN(C)C)C1 70086,N1(C(C(CC=C)(C)C)=O)CCC2(CC1)CC(CNC(C1CC(C)CC(C)C1)=O)C2 70087,CCS(=O)(=O)c1cnc(O)c(C(=O)NC2C3CN(C(=O)CC4CC=CC4)CC23)c1 70088,C(=O)(C#CC(=O)OC(C)(C)C)NCCCCN(C(=O)COCC(C)(C)C)C 70089,C(C(=O)NCCCN(C(c1c(C)ncn1C)=O)C1CC1)(C(C)C)N(CC)CC 70090,CC1CCN(C(C2CCS(=O)(=O)N2)=O)C(CNC(C2CC(=O)C2C(C)(C)C)=O)C1 70091,N1(C(C(CCCC)F)=O)CCC2CN(C(C3CC3C(F)(F)F)=O)CC2CC1 70092,Cn1nccc1CCNC(=O)CCC1(NC(C2CC2c2ccoc2)=O)CCCC1 70093,C(C)(C)(CC(F)C(=O)NC1CCCOC1)NC(C(C)SCC)=O 70094,c1(OC)ccccc1C(C)CC(=O)N(C1CC(NC(=O)Cc2c[nH]nc2C)C1)C 70095,c1(C(=O)NC2CC(NC(C3C(C)C3C)=O)C2)cccc2c1nnn2C 70096,CC1CN(C(C23CC(C2)C3)=O)CCC1NC(=O)CCc1nc(O)n[nH]1 70097,c1(C(=O)NC2C(CNC(C(=Cc3cccnc3)C)=O)C2)ccc(S(N)(=O)=O)cn1 70098,Cc1cc(=NC(C)CCNC(=O)C#CC2(C)CCCO2)[nH]c(C)c1C#N 70099,CCCCCC(C)NC(c1ccccc1Cc1ccccn1)=O 70100,N1(C(C(C(CC)O)C)=O)CCCC2(C1)CN(C(=O)CCc1ccccn1)CCO2 70101,c1(C(N2CCC(C)(CNC(CN(C(C)C)C)=O)C2)=O)coc(S(=O)(=O)N(C)C)c1 70102,c1(NC(C(C)NC(c2ccc(C)[nH]2)=O)C(C)C)cc2nn[nH]c2cc1[N+](=O)[O-] 70103,C(=O)(C(C)(O)CC(F)F)N(C)C1CC1.c12ccc(o1)C(=O)NCCCNC2=O 70104,c1(CC(=O)NC(CNC(C2CC(F)C2)=O)CO)coc(-c2ccccc2)n1 70105,O=C1Cc2cccc(C(=O)NC3CCN(C(c4c(F)cccc4Cl)=O)C3)c2N1 70106,C(=O)(N(CCC(=O)OC1CCCCC1C1CN(C)CCN1C)OC)NC 70107,N1(C(C2(OCC)CCC2)=O)C2CCC1C(CNC(=O)Cc1cccnc1Cl)C2 70108,N1(C(C(CNC(C=CCOC)=O)O)=O)CCC(C(C)C)(CO)C1 70109,c1(C(=O)NCC(C2CCCC2)NC(c2csnn2)=O)cccc2c1OCCO2 70110,c1(N2C(c3cccc(C)c3C)CCC2)ncc2cc(C)ccn12 70111,c1(C(N2C(CN(C)C(C3CCCOCC3)=O)COCC2)=O)cnn2ccncc12 70112,CCC(C(=O)NCCOCCN(C(=O)CC1CCC(O)C1)C)C(C)C 70113,c1(C(=O)NCC2(C(N(CC=C)CC3CC3)=O)CCC2)cnn(C=C)c1N 70114,C(=O)(C1=CCN(C(c2coc(C)c2)=O)CC1)N(C1COCC1O)CC 70115,C1(O)(CCNC(c2cc(C(C)=O)sc2)=O)CCN(C(=O)C(C)(C)C(F)F)CC1 70116,N1(C(C2(C(=O)OCC)CC2)=O)CC2CC(C1)N(C(C1(F)CCC(C)(C)CC1)=O)C2 70117,N1(C(C(=O)NCc2ncc(Br)cc2C(F)F)=O)CCc2ccc(F)cc21 70118,C(CC(C)C(=O)N1CCC(C)(CNC(c2nn(C)cc2SC)=O)C1)=CC 70119,N#Cc1cccc(NC(=O)C(CCC2CC2)NC(c2ccsc2Cl)=O)n1 70120,C(=O)(C(C)CC(C)(F)F)NCCCCCN(C(C1CC=C(C)CC1)=O)C 70121,C1(CCC(=O)OC)CNc2ccccc2C1Cn1c(=O)oc2ccccc12 70122,Cc1ccc(C(N2CCC(CCNC(C34CCCC3OCC4)=O)C2)=O)c(F)c1F 70123,c1(CC(=O)N(CCN(C(=O)CCN2CCC(F)C2)C)C)ccccc1F 70124,C(=O)(C=CS(=O)(=O)CC)N1CCC(Cn2cc(C(CC)(C)O)nn2)C1 70125,c1(C(N(CCC(C(=O)NC(CC(=O)OC)(C)C)O)C)=O)cc(C)nc(O)c1 70126,c1(SCC#C)cccc(C(=O)NC(CNC(=O)C(c2cscn2)N(C)C)CO)c1 70127,c1(OC)nc(C2=CCNCC2)ccc1C(N1Cc2cccc(O)c2C1)=O 70128,N1(C(=O)NC2(C(=O)O)C(C)C2)CCN2CCN(C(C3CCC(=O)N3C)=O)CC2C1 70129,C1(CNC(CS(C(C)C)(=O)=O)=O)CCC2CN(C(C3CC4CC4C3)=O)CCC2C1 70130,N1(C(C)C)CC2CN(CC34CCCC3C4)CCC12 70131,C1(NC(c2c(CC)nco2)=O)CCN(C(c2c[nH]nc2-c2cccs2)=O)CC1F 70132,c1(Cc2ccnc(N3CCOCC3)n2)nc(C2Cc3ccccc32)no1 70133,C1(CC(=O)N(C)Cc2ccc(F)cc2)CC(C)(C)CN1C(=O)CC1CC2(CC2)CO1 70134,c1(C(N2CCC(C)C(NC(=O)Cc3ccnnc3O)C2)=O)cc(C#N)ccc1F 70135,Cc1nnc(O)c(C(=O)NCC(C)N(C(=O)C(C)Cn2cccn2)C)c1C 70136,N1(C(C(N2CCCC(C)C2)=O)=O)CCC(NC(=O)C(C)(C)c2nccs2)C1(C)C 70137,c1(CCC(=O)NCC(C(C)(C)C)NC(CSC(C)C)=O)ccc(Cl)cc1F 70138,c1(C(=O)OC)cc(Br)c(F)cc1NC(C1CN(Cc2cc(F)cc(Br)c2F)C1)=O 70139,C12=CC(=NC(=O)C3CC(C3)NC1=O)NN2C.C1(CC)CCCCC1F 70140,C1(C(=O)NCCCN(C(=O)C#CC2(C(F)(F)F)CC2)C(C)C)Cc2nncn2C1 70141,C12(C(=O)NC3(C4N(C(CC5(OC)CC5)=O)CCC4)CC3)CCN(CC1)C2 70142,c1(CN2C(C(N3CCC(C(N)=O)CC3)=O)CC2)c[nH]c2cccc(F)c12 70143,c1(C(N2CCC(NC(C(C)SC)=O)C(C)C2)=O)cccc2c1NCC2 70144,C(=O)(C(C(C)CC1CCOCC1)N(C)CC1CCCN(C)C1)NCC=C 70145,C(=O)(C1=CC2(CCOCC2)C1)N1CC(C)(NC(=O)C2=CS(=O)CCC2)C1 70146,Cc1nnccc1C(N1CCC(C(C)NC(=O)CN2CCOCC2=O)C1)=O 70147,N1(C(c2nc(CC)[nH]n2)=O)CC(NC(=O)CC(C)(F)F)CC1C 70148,C1(C(=O)NC(C)CCNC(=O)C(O)C2CCCC2)CCC(N=[N+]=[N-])CC1 70149,N1(C(C2=C(C)CC2)=O)CC2(C(N3CCOC(CCO)C3)=O)CC1CO2 70150,C1(C(=O)NC2CC(NC(C3N(CC)CCCC3)=O)C2)CC2(C1)CC(F)C2 70151,C12CN(CCN1N(C)C)C(=O)C=CC(=O)NCC2.c1(C=O)cc(C2CC2)ns1 70152,C1(C(=O)NC2(C)CN(C(CC(C(C)C)OCC)=O)C2)Cn2c(C)nnc2CN1C 70153,C1(CNC(c2cc(OC)n[nH]2)=O)CN(C(C2CCN(C(C)C)CC2)=O)CCN1C 70154,CC1CCN(C(=O)C(=O)NC(C)(C)C(C)NC(=O)CCCc2ccncc2)CC1 70155,C1(CC(=O)NCCCOCCNC(C(C(C)C)OCC)=O)CCCC2(CCC2)O1 70156,C1(C(=O)OC)CCC(NC(=O)CC2(C)CN(Cc3ccsc3SC)C2)C1 70157,C1(C(=O)NC(CC)CO)C(CNC(c2ccoc2Cl)=O)C1(C)C 70158,c1(C(=O)NC2CC(C)(NC(CC(C)CF)=O)C2)nc[nH]c2ncnc1-2 70159,c1(CC(C)N(C(c2ccc(C(Cl)Cl)cc2)C(=O)NC)C)c(C)nn(C)c1C 70160,CC(N=c1[nH]c2c(c(=NC3CCN(c4ccccc4F)C3)[nH]1)CCC2)C1CCC1 70161,C1(NC(C=CC=CCCCCC)=O)CN(C(c2csnc2C)=O)CCC1CO 70162,c1(NS(=O)(=O)Cc2ccccc2I)ccccc1N1CCCCC1 70163,C=CC(C)(O)C(=O)NCCCN(C)C(C1(c2cccs2)CC1)=O 70164,C1(NC(c2cccc(C3CCC3)c2)=O)C2CCN(C(C3CC=CCC3)=O)C12 70165,N1(C(=O)C=C2CCC2)CCN(C(C2(c3ccc(Cl)c(F)c3)CC2)=O)C(CO)C1 70166,Cc1cc([N+](=O)[O-])cnc1N1CC2(CCC(NC(c3c(C)noc3C)=O)CC2)C1 70167,Cc1cc(C)c(C(=O)NCCC2(CNC(=O)CCc3nncn3C)CC2)s1 70168,c1(C(=O)NCCC(C)NC(c2c(OC)c(=O)cco2)=O)c(C)ccc(C)c1C 70169,c1(C(=O)NCCCN(C(c2cccnc2)=O)CC)cccc2scnc12 70170,C1(NC(CN(C)CC)=O)CC2CC(NC(=O)CSc3n[nH]c(=N)s3)C2C1 70171,C(=O)(CC(F)(F)F)NC(C(=O)N(CC(C)NC(=O)Cc1ccnn1C)CC)C 70172,C1(C(=O)NCCCCCN(C(=O)C(C)(C)C(N)=O)C)CNc2ccnn2C1 70173,C1(C(=O)NCCN(C(=O)C(=O)Nc2ccccc2)CC)COCCN1C 70174,CCCC(CC(=O)NCCN1CCCCC1)NC(C1CC(CF)C1)=O 70175,C(CC(N)=O)(C(=O)N1CCCC(C(C)C)CC1)NC(CSCCC(C)C)=O 70176,C1(C)(C(=O)NC(C)C2CC2)CC12CCN(Cc1cc(C3CCC3)no1)CC2 70177,C1(C(=O)NCc2nnc(CC)o2)CC2(CCC2)CN1C(C1C=CCS1)=O 70178,N1(C(C(=Cc2cccs2)C)=O)CCC2CN(C(=O)COC3CCCC3)CC2C1 70179,CCCCCCC(C)(CC)C(=O)NC1CCC(NC(=O)CCc2nncs2)C1 70180,c1(C(=O)NC2(CNC(c3c[nH]nc3F)=O)CCOC2)cc(Cl)c(Br)[nH]1 70181,N1(C(C(=O)NC(CC)C)CC2C=CCC2)Cc2ccc(Br)cc2CC1C 70182,C(C(=O)N1OC2CCC1C2)C1CCN(C(C(N=S(C)(C)=O)=O)=O)C1 70183,C1(C2CC2)(CNC(C=CSC)=O)CCN(C(=O)C(C)(C)C(=O)OCC(C)(C)C)C1 70184,c1(SCC(N2CCC(N(C(=O)CN3CC4CC4C3)CC)C2)=O)c(O)nc(=N)[nH]c1C 70185,C1(CCN(C)C(c2ccc(F)cc2)=O)CCCCN1C(c1n[nH]cc1Cl)=O 70186,c1(CNC(c2c(C)ncnc2)=O)nc(CNC(=O)CN2CCOCC2)cc(O)n1 70187,C(=O)(C1=Cc2ccccc2C1)N1CC(F)(CNC(=O)C2=CC3(CCOC3)C2)C1 70188,CCS(=O)(=O)CC(=O)NCC1(C(=O)NCC(C)(CO)CO)CC12CCC2 70189,CCCC(CC(C)C)C(=O)NCC1(NC(=O)COC(C)CC)CCOCC1 70190,C(=O)(C1=CS(=O)CCC1)NC(CC)CNC(=O)C(c1ccc(F)c(F)c1)C 70191,C(CCN(C(=O)CC1CC=CCN1C)C)(C(C)(C)C)NC(C1CC(OCC)C1)=O 70192,C1(O)(CNC(C(C)N(C(C=CC(=O)OC)=O)C2CC2)=O)CCCCCC1 70193,N1(C(C2CCC(CC)O2)=O)CCCN(C(c2cnc(O)cc2C)=O)C(CO)C1 70194,N1(C(c2ccno2)=O)CC(C2CCCN(C(C3(CO)CC3)=O)C2)C1 70195,N1(C(CCOCCN(C(C=C(C)C(F)F)=O)C)=O)CCCC(C)(C#N)C1 70196,CC1C(C(=O)Nc2cccnc2F)CCCN1C(C1CC2(C1)CC2(F)F)=O 70197,C1(C)(NC(C(CSC)O)=O)CCCN(C(c2nc(C(C)C)oc2C)=O)C1 70198,c1(NC(c2c(Nc3ncc(OC)cn3)cccc2)=O)ccc(S(C)(=O)=O)cc1C 70199,C1(NC(CCn2ccc(C)n2)=O)CN(C(c2ccsc2)=O)CCC1F 70200,C1(C2N(C(CSC)=O)CCC2)CCN(C(=O)C=C2CCCC2)CC1 70201,c1(COC)cc(C(N2CCOCC2CNC(C2CC2c2cccs2)=O)=O)n(C)c1 70202,C12(NC(C3=NOC(C)C3)=O)CCCC1(F)CN(C(c1ccncc1Cl)=O)C2 70203,N1(C(C(C=C)C)=O)CCC(C)C(CC(=O)NC(CN(C)C)CC(C)C)C1 70204,C(CC(C(=O)N(C1CCC(CO)CC1)C)NC(C1CC1C(F)(F)F)=O)SC 70205,c1(OC)cc(F)c(C(=O)NC2CN(C(=O)C(F)=CCCF)CC2OC)c(F)c1 70206,N1(C(c2c(CC)ccc(Br)c2)=O)CCC(NC(=O)C(CC)OC)C(C)(C)C1 70207,c1(C(N2C(C)(C(=O)NCC(COCC)O)C=CC2)=O)cc(=O)n(C)cn1 70208,C(=O)(C(=O)N(n1cccc1)C)N(CC(C)O)CC(C)O 70209,N1(C(c2c(C(F)F)ccc(C)c2)=O)CCC2CCC(C1)N2C(=O)CCC#N 70210,N1(C(CCc2ccc(C(=O)OC)cc2)=O)CCN(C(C2CSC2)=O)CC1CCO 70211,N1(C(COCCSC)=O)CCC(C(C)(C)NC(=O)C(O)CSC)CC1 70212,c1(C(N2CCC(C)(NC(=O)CC3CCOC3=O)C2)=O)cc(S(N)(=O)=O)ccn1 70213,S(=O)(=O)(c1c(F)cc(F)cc1F)N1CC2CN(C(c3cc(Cl)c(Cl)s3)=O)C2C1 70214,N1(C(CC2COCC(C)O2)=O)CCC=C(C(=O)NC2CC(C#N)C2)C1 70215,CC1CC(C(=O)NCCn2cnc(CO)c2)CN(C(=O)CC2CC(=O)C2)C1 70216,N1N(Cc2cn(-c3ccc(OC)cc3)nn2)CCOC2(CCOC2)C1 70217,C(CCN=C(NCCc1cccc(O)c1)NC1CCCC1)c1c(C)cccc1 70218,c1(-c2cn(C3CN(C(CCOCC)=O)C3)nn2)sc(OC2CCCOC2)nc1Cl 70219,C12(C(N3CC(NC(c4ccc(CO)o4)=O)C3)=O)COCC1CS(=O)(=O)C2 70220,C1(Cn2cc(-c3n(C)cnc3)nn2)CC2CCC1(NC(c1cc(N)cnc1Cl)=O)C2 70221,C1(CNC(CN(C2CC2)CC)=O)CCCCCN1C(=O)C(C1CC(C)(C)C1)OC 70222,Cc1nccc(C(=O)NC2CC(C(=O)NCCSC(C)C)C23CCC3)c1C 70223,CC(CS(N)(=O)=O)NC(C1(C)CC(NC(C2CC=CC2)=O)C1)=O 70224,C(C(CC1CC1)C(=O)N1CC2CC2(CO)C1)NC(C1CC(=C2CC2)C1)=O 70225,NC(=O)CC(O)C(=O)NC(CNC(c1cc(Br)n[nH]1)=O)C1CCC1 70226,c1(CNC(c2n(C)nc(C)c2Br)c2nnnn2C2CC2)ccc2c(c1)CCCO2 70227,C=CC(C)(O)CC(=O)NCCC1(C(=O)NCC2CCSCC2)CCC1 70228,N1(C(C(CC)NC(C)=O)=O)CC(CNC(=O)C(C)Sc2ncccn2)C(C)C1 70229,c1(C(=O)NCC(C2CCOC2)NC(=O)COC2CCC2)ccc(CO)nc1 70230,CC(CCC(C)(C)C)C(=O)NC1CCN(C(=O)CCc2cnn[nH]2)CC(O)C1 70231,N(C1CCc2cc(CCn3cc(-c4cnc(O)nc4)nn3)ccc21)C(=O)OCC 70232,C=CC(CC)CC(=O)N(CCC(C)NC(=O)CCNC(=O)OCC)C 70233,C1(CC(=O)N(CC#CC)CC#C)CCCC(NC(=O)C(C)c2cc[nH]n2)C1 70234,CC1CCCC(C(N2CC(CNC(=O)C3=CSCS3)C2)=O)C1 70235,C1(CC(C)NC(C2(C3CC3)CCCO2)=O)CCN(C(c2ccco2)=O)CC1 70236,C#Cc1cccc(C(=O)N(C2CCCN(C(c3n[nH]c(C)n3)=O)CC2)C)c1C 70237,C(CC(C(C)C)NC(=O)C(n1nc(C)cc1C)C)NC(c1cn(CC=C)nc1)=O 70238,C1(C(=O)NCC2(C)OCCN(C(CC(=O)NCC)=O)C2)CCn2c(O)nnc2C1 70239,C#Cc1ccc(Br)c(OCC2OC(=O)NC2(C)C)c1 70240,N1(C(C2N(C(c3c(NC)scn3)=O)CCC2)=O)CCC(O)CC12CC2 70241,N1(C(CC2(C)CCCCC2)=O)CCC=C(CNC(c2cccnc2)=O)C1 70242,C(c1cnn(C)c1C)=CC(=O)NC(COCCCNC(C(C=C)O)=O)(C)C 70243,c1(C)cccc(C(F)F)c1.C1(C(F)F)(CC)CN(C(=O)NC2=CCC2)C1 70244,C1(CCOC)CN(C(=O)C(N2CCN(C)CC2)(C)C)CCN1C(c1csnn1)=O 70245,CC(C)CC(CNC(C1(F)CCC1)=O)NC(=O)CC(=O)NC1CC1 70246,C1(CNC(c2ccc(C(C)=O)s2)=O)CC(C)N(C(=O)Cc2cnsc2)C1 70247,Cc1cccc(C=CC(=O)NCC(CC2CC2)C(=O)NC(c2ncc(C)o2)C)c1 70248,C1(C(=O)NCC(C)NC(=O)CC2(O)CC2)CC(=O)N(c2ccc(C3CC3)cc2)C1 70249,c1(C(=O)NCC2C3CN(C(C45COC(CCO4)C5)=O)CC23)ccc2cc[nH]c2n1 70250,CC1CC(CNC(=O)CC(C)(C)O)CN1C(c1cnco1)=O 70251,C#CCC(CC#C)C(=O)NCC(CCCC)NC(C1CC2CC2C1)=O 70252,N1(C(CCC(=O)NCC)=O)CCC2(CCN(C(c3cc(C)n(C(F)F)n3)=O)C2)C1 70253,c1(C(=O)NC(C2(O)CN(C(c3cnc(S)nc3)=O)C2)C)cccc(O)n1 70254,c1(C(N2C(CO)CC(NC(C(C)S(C)(=O)=O)=O)C2)=O)ccc(F)c(Cl)c1F 70255,Cn1ccc(C(=O)NCC2CC(NC(c3cnnn3C3CC3)=O)C2)c1 70256,CC(C)CC(C(=O)NCC1C=CCN1C(=O)Cc1cccs1)N1CCCCCC1 70257,C(=O)(C(CCC=C(C)C)N(c1ccccc1Cl)C)NCCCSC 70258,N1(C(C(N2CCC(C)CC2)=O)=O)CC(C)N(C(=O)C=C2CCC2)C(C)C1 70259,C1(C(N(C2CN(C(c3c(OC)c(Cl)ncc3)=O)C2)C)=O)Cc2c(F)cccc2O1 70260,C1(NC(c2c(CC)noc2C)=O)CN(C(=O)CSCC(N)=O)C2(CCCOC2)C1 70261,C(C1=CCCN(C(C2(C)CCCC2)=O)C1)NC(CCn1ncc(C)c1)=O 70262,Cc1cccc(C)c1NC(=O)C(c1ncc(Cl)s1)N(CC(C)C(C)C)C 70263,c1(C(=O)NC2(c3ccccc3)CCN(C(CC)=O)C2)cc(=O)cc(Cl)[nH]1 70264,c1(C(=O)NC(C2CN(c3nnc(C4CC4)s3)CCO2)C)cc(C2CC2)oc1C1CC1 70265,c1(C(N(CC(O)CN(C)C(C2CCS2(=O)=O)=O)C)=O)cc(F)c(F)cc1Cl 70266,N1(C(c2c(COC)cc[nH]2)=O)CCOCC1CNC(C1CC(F)(F)CS1)=O 70267,c1(COC)cc(=NCC2(O)CCN(C(C3(N(C)C)CC3)=O)CC2)[nH]cn1 70268,c1(C(N2CC(NC(CCCOC)=O)CC(C)(C)C2)=O)ccccc1C#CC1CC1 70269,C1(NC(CNC(=O)Nc2sc(C)c(C3CCOC3)n2)=O)COC2(CCC2)C1 70270,c1(C(C)=O)cncc2n[nH]c(C(C)C)c12.N1CC2=C(C1)CN(C(C1(C)CC1F)=O)C2 70271,CCCCCC(O)CC(=O)NCC1CN(C(c2ccccc2-c2ncc[nH]2)=O)C1 70272,N1(CC(=O)N(CC2N(C(C(C)OCC)=O)CCC2)CC)CCNC(=O)C1 70273,CC(CN1CCCCC1)C(=O)NC(C)CCNC(c1nn[nH]c1Cl)=O 70274,c1(-c2cn(C(C)C(=O)NC3CCCN[SH](C)C3=O)nn2)ccc2cnccc2c1 70275,C#CC1(C(=O)NCc2ccc(C(=O)NCCNC(=O)NCCC)cn2)CCCC1 70276,c1(C(N2CC(C)C(NCc3ccc(F)cc3F)C2)=O)cccc2c1CCC(=O)N2 70277,C1(NC(CNC(=O)NC)=O)CCCC(N(CCC(=O)NCC(C)C)C2CC2)C1 70278,c1(CC(N2CC(CCNC(C3CC(CC4CC4)C3)=O)(OC)C2)=O)ccccc1F 70279,N1(C(C2CCCN(CC)C2)=O)CC2(CC(CC(=O)NC3(CCF)CC3)C2)C1 70280,N1(C(C2N(C)S(=O)(=O)CC2)=O)CCCC2(CCCN2C(C2CC(O)C2)=O)C1 70281,c1(C(N2C3C(NC(c4n(CC#C)ccc4)=O)C(CC3)C2)=O)ccc2nonc2c1 70282,N1(C(C=Cc2ccc(C(N)=O)o2)=O)CCCC(C2CN(C(=O)C3=COCC3)C2)C1 70283,C(=O)(CCC(C)(C)NC(c1nnnn1C)c1ccnn1CC1CCC1)OC 70284,c1(N2C(CCNC(C3(CS(N)(=O)=O)CCC3)=O)CSCC2)ncnc(Cl)c1F 70285,C(=O)(C(F)C(F)(F)F)NCC1N(C(CCN(C2CCCCC2)C)=O)CC=C1 70286,N1(C(C(C)CC(F)(F)F)=O)CC2(C)CN(C(C3CC4(C3)CC(O)C4)=O)CC2(C)C1 70287,N1(C(c2cn(CC(=O)N(C)C)nn2)=O)CC2CC2(CNC(=O)C(F)(F)C2CC2)C1 70288,N1(C(c2c(C)cc(C)c(C)c2)=O)CCC2CCN(C(=O)CSCCC#N)CC12 70289,C1(F)(C(=O)NC(C(C)C)CCN(C(=O)C=Cc2nnn(C)n2)C)CC2(CCC2)C1 70290,c1(CNC(=O)NC2(C3CC3)CCCCC2)cccc2c1OCCC2O 70291,N1(C(c2n(CC)cc(Cl)c2)=O)CCC(O)C(NC(C2CC3(CCCO3)C2)=O)C1 70292,CCCC(O)C(CO)NC(=O)C1=NOC(CNC(C2CC3(CC3)C2)=O)C1 70293,C1(C(=O)NC2CCCCCC2)CC2(CCC2)CN1C(c1ccccc1)=O 70294,c12cccc(c1)C2.n1(C(C(N2C(C(=O)OC)CCC2)=O)C)nc(C)cc1C 70295,C(=O)(C(C(C)C)CNC(C1CC(n2cc(CCSC3CCCC3)nn2)C1)=O)OC 70296,C12(CN(C(=O)C(=O)NC3CCN(C(C)C)C3)C(C)C)CCCC(CO1)C2 70297,N1(C(CC(=O)NCC)=O)CCC(C)C(NC(=O)C(CC)n2cccn2)C1C 70298,C=CC1CN(C(C2CC3CC3C2)=O)CC1NC(=O)CCOCC(F)(F)F 70299,c1(C2N(C(c3c(OC)oc(C)n3)=O)CCS2)cccc(Cl)c1Cl 70300,N(C(=S)N1CCC(Oc2ccc(Cl)c(F)c2)C1)CCCF 70301,c1(N2CCN(C(=O)NOCC(F)(F)F)CC2)ncnc2ccccc12 70302,C(=O)(C=C=C(C)C)N1C(C(=O)NCCC2(COC)CC2)CC1C 70303,CCCC(C(=O)OC)C(=O)N1CCC2(C1)CN(C(C1CCCS(=O)(=O)C1)=O)C2 70304,N1(C(Cn2c(CCC)ncc2)=O)CCC(O)C(N(C(=O)CC2C=CCC2)C)C1 70305,Cc1cc(O)cc(O)c1C(=O)NC1CCCC1C(=O)Nc1ccnnc1 70306,C#CC1CCC(C(N2CCOC(CNC(=O)COc3cn[nH]c3)C2)=O)CC1 70307,c1(CCC(=O)NC(C2(O)CCN(C(C3(O)CCCC3)=O)C2)C)ccc(F)c(F)c1F 70308,C(=O)(C1CC(=O)Nc2cc(F)ccc21)N1CC(NC(c2n(C)ncc2)=O)C2C1C2 70309,C(C(C)(O)C(=O)NCCN(CCOC)C(C1CC(c2cccc(F)c2)C1)=O)OC 70310,CCC(C)(C)C(=O)C(=O)NC1(CO)CCCN(C(=O)C(c2ccc(C)cc2)O)C1 70311,c1(C(N2CC(C)(CNC(c3ccc(=O)oc3)=O)OCC2)=O)cccn2cnnc12 70312,CC(CC(F)(F)F)C(=O)N1CCC(C(C)(C)C(=O)NC23CCC(CC2)C3)C1 70313,c1(C(=O)NC(C(C)NC(c2cnn(C(C)(C)C)c2)=O)C)cc(Cl)n(C)n1 70314,C1(NCCC2CC(F)C2)Cc2nc3ccccc3n2C1 70315,C1(CCC(C)C)CCN(CC(=O)NCCC2CCCCC2)CC1 70316,c1(CNC2CC3(N(C(CCCCC(=O)OC)=O)CC3)C2)cccc2cnccc12 70317,c1(C(=O)NCC2CCN(C(C3(C(F)F)CCC3)=O)C2)cc2c(s1)CCCCCC2 70318,Cc1cc(C=CC(N2CCN(C(=O)C(C(C)C)N(C)C)CC2C)=O)c[nH]c1=N 70319,C1(C(N2C(CCCNC(c3cc(C)no3)=O)CCC2)=O)CCC2C(CC1)C2(F)F 70320,Nc1sc2c(c1C(N1CC(O)(CNC(C3C4CCCC34)=O)C1)=O)CCC2 70321,CCC(CNC(C12CC(C)(C1)C2)=O)(CC)NC(=O)CCn1cccn1 70322,C(=O)(CS(=O)(=O)CC(C)C)NCC1CCN(c2snc(SC)n2)CC1O 70323,C1(CC(=O)NC2(C)CC(C(=O)OC)C2)CN(C(=O)CCC2OCCO2)CC1C 70324,c1(C(N2CCOCC(NC(C)=O)C2)=O)cnc2[nH]ncc2c1 70325,C1(OC)(CNC(=O)CC2(C)CCN2C(=O)C(C)OCC(C)C)CCOC1 70326,N1(C(CSCC)=O)CCC2(CCOCC2)C(Nc2cc(-c3nn[nH]n3)cc(Cl)n2)C1 70327,C1(C(=O)NCC(CNC(c2cc(C(C)=O)c(C)nc2)=O)O)OCC2CCCCC12 70328,C1(C(=O)NC2CCSCC2)CCC(c2nn[nH]n2)C1 70329,Cc1ncsc1C=CC(N1CC2C(CNC(c3ccc[nH]3)=O)C2C1)=O 70330,C1(CNC(CCC2CCC(=O)N2)=O)CC2(CC2)CN1C(c1nc(Cl)c(Cl)s1)=O 70331,C(=O)(C(F)(CNC(=O)C(CCC)N(C)C)C(C)C)NCCCCCC 70332,C1(C)(CC(=O)NCCN(C)C2CC2)CCN1C(=O)CC1CC(F)(F)C1 70333,c1(C(N(CCOCCCNC(C(C=C)O)=O)C)=O)c[nH]cc(C)c1=O 70334,Cc1cc(CC=O)cs1.C(=O)(CSC(C)(C)C)N(C)CCNC 70335,c1(SC)cc(Cl)ccc1CN1CCC(c2ccc(OC(F)F)cc2)C1 70336,N1(C(=O)C2=CCCS2)CCC2CCC(NC(=O)C(F)(F)c3nccs3)C1C2 70337,N1(C(c2cc(C(=O)Nc3ccc(C)cc3OC)no2)=O)CCC(COC)C(O)C1 70338,c1(C(C)=O)ccc(OCCCC(=O)NCC(C)N(C)C(c2cc(F)n[nH]2)=O)cc1 70339,C=CCCCCCC(=O)N1CCN(C(c2ccc(C(F)(F)F)nn2)=O)C(C)C1C 70340,CCS(=O)CC(=O)NCC1(C(C)NC(=O)CNC(c2ccc(OC)cc2)=O)CC1 70341,C1(C2CCN(CC(=O)NC(CC)(C)C)C2)CCCCN1C(=O)CN1CCOCC1 70342,C(=O)(CC(CC(N)=O)c1ccc(F)cc1)N(CCCNC(C1COC(=O)O1)=O)C 70343,c1(C(N2CCC(OCCNC(C3C(C)CCC3)=O)CC2)=O)ccnc2c1CCO2 70344,c1(C(=O)NC(C2OCCN(C(c3ncn(CC)c3)=O)C2)C)ncccc1N=[N+]=[N-] 70345,C1(NC(C2CCc3ncnn3C2)=O)Cc2ccc(Br)cc2C1 70346,c1(CCCC(=O)NCC(C)N(C(C(C)OCC2CC2)=O)C)cccc(Cl)c1 70347,C1(C(N(C2CCCN(C(=O)C(C3CCOCC3)=O)CC2)C)=O)CC2CC2CC1C 70348,C(=O)(C(O)CC(C)(C)C)NCC(CCNC(CSc1ccc(C)cc1C)=O)O 70349,CCC(C)CCCCC(=O)NC1CC(C)N(C(c2ccc3oc(O)nc3n2)=O)C1 70350,C(c1ccc(OC)c(F)c1)=CC(=O)NCC(C(=O)OC)CC1CCCC1 70351,c1(C(=O)NC2CC(N(C(CC(OCC)OCC)=O)C)C2)ccc2ccn(C)c2c1 70352,O=S(=O)(c1cc(F)cc(F)c1)Nc1ccc(Br)c(Cl)c1F 70353,c1(C(N(CC(C)NC(c2ccc(=NC)[nH]c2)=O)CC)=O)ccn2nnnc2c1 70354,C1(NC(C2C(=C)CC2)=O)(CNC(=O)CC2CCC(=O)N2)CC(C(F)(F)F)(OC)C1 70355,C1(NC(c2cccc(OC)c2)=O)C2CCC1CN(C(C1CCC(=O)N1)=O)C2 70356,C=CCCC(C)(C)C(=O)NCCC1CC(NC(c2nscc2Br)=O)C1 70357,c1(CSC)nc(-c2c[nH]ccc2=O)n(CC2CCCOC2)n1 70358,C(C(=O)NCCN1CCN(C(=O)C(=O)NCCC(N)=O)CC1)(C(C)(C)C)OC 70359,Cc1ncc(NC(C2(CCC3CC3)CCC2)=O)c(C)c1C.C12(CC1)C(=O)NC2=O 70360,c1(C(N2CC(OCCNC(CC3C(C)CCO3)=O)C2)=O)c(Cl)csc1Cl 70361,CN1CCCCC1C(=O)NC1(CNC(c2cccc(C3(C#N)CC3)c2)=O)CC1 70362,CC(C)CC(C(=O)N1C2CCCC1CC(NC(=O)Cc1cn(C)cn1)C2)C(C)C 70363,C1(C(=O)NC(C(C2CCCCC2)NC(COC)=O)C(C)C)CN(CP(C)(C)=O)C1 70364,N1(C(c2c(SC)snn2)=O)C2CCC1C(CNC(=O)CCC(=O)N(C)C(C)C)C2 70365,c1(C(C)NC(=O)NC(C(=O)OC)C)cccc(F)c1 70366,C(C(CC(=O)NC(C(C)C)C(C)C)C1CCC1)NC(CC1(CO)C(CC)CC1)=O 70367,C#CCCCCCC(=O)NCc1cc(C(=O)NCC(C)C(C)CC)n[nH]1 70368,CCCCCC(O)CC(=O)NCC1CCCN1C(c1cnn(C)c1C(F)(F)F)=O 70369,C(CC1CC1)(CC(=O)NCC1CC1c1ccoc1)NC(C=C(CCC)C)=O 70370,CCC(CC(=O)NC1COCCOC1)NC(=O)C(C)C1(O)CCC1 70371,C#CCCC(C(=O)N(C(CO)C(C)C)C)NC(=O)C(C)SC(C)C 70372,C1(C(=O)NCCC(=O)NC(CC)C)CCN(C(C2CC2Cl)=O)C12CCC2 70373,C1(C(=O)NCC=CCNC(C2(CC=C)CCCC2)=O)Cc2nnc(C)n2C1 70374,C1(NC(CCOCC(C)C)=O)CCC(C(N2CCC2CC2CC2)=O)C1 70375,c1(C(N2CCC(N(C(=O)CCC(C)C#N)CC)CC2)=O)cc2n(n1)CCCC2O 70376,C1(NC(=O)C2=CCCOC2)CCN(C(=O)CC2CC3CC3C2)CC12CCC2 70377,c1(-c2cncc(OC)c2)ccc(F)c(NC(=O)CCCNC(=O)C2CC2)c1 70378,c1(C(N2CC(NC(c3cn(CCC)nc3C)=O)C2)=O)ccc([N+](=O)[O-])cc1F 70379,C12(C(=O)NCC(=C)CCNC(C3NC(=O)OC3C)=O)CCCCC(=O)N1CCC2 70380,N1(C(C(CC)n2nccc2C)=O)CCC(NC(c2cnc(C)cn2)=O)C(C)(C)C1 70381,c1(NCC2C(NC(c3cc(C)ns3)=O)CCC2)cc(C(F)F)nc2ncnn12 70382,C1(NC(C2CC(OCC)C2)=O)CCC(CNC(=O)CSc2nnnn2C)C1 70383,N1(C(C(C)c2cc[nH]n2)=O)CC(CNC(c2cc(C(N)=O)no2)=O)C2(CC2)C1 70384,C1(C)(C(N2CCC(CCOC)C2)=O)CCN(C(=O)C(C)CC(N)=O)CC1 70385,C12(CC(=O)NCC=CCSC)CCC1CN(C(=O)CCc1cccn1C)C2 70386,c1(C(N(CCNC(C2C(C=C)CC2)=O)C)=O)ccc2c(c1)CCCS2(=O)=O 70387,CC#CCC(C(=O)N(CC(C)(CO)CO)C)NC(=O)CC(=O)OC 70388,c1(CNC(C(n2cc(-c3cc(C)ncc3)nn2)C)=O)c(C)ccnc1O 70389,C1(NC(CC(C(=C)C)OCC)=O)CC2CCC1N(C(=O)CNC(N)=O)C2 70390,c1(C(=O)NC2(COC)CN(C(=O)C(C)SC(C)C)C2)cccc2ccsc12 70391,N1(S(CC)(=O)=O)CCC2(CC(C(=O)Nc3cccc4c(O)cccc34)=NO2)C1 70392,C1(OC)CC2CC(C(N3CC(NC(=O)CCOc4ccc(F)c(F)c4)C3)=O)CC12 70393,N1(C(CC(COC)C)=O)CCC2(CCCN2C(=O)CCc2nc(=N)[nH][nH]2)CC1 70394,c1(C(=O)NC2(CCNC(c3cc(C)c(C)nn3)=O)CC2)cnc2n[nH]c(C)c2c1 70395,C(=O)(C1CCCn2c(C)nnc21)NCC(C(C)C)NC(c1n(C)nc(C)c1Cl)=O 70396,N1(C(C(=O)NCCCCCC)CCC2CCCO2)CCCC(CCO)CC1 70397,Cc1nc(N(C2C3CCOC3C2(C)C)C)c2sccc2n1 70398,Cc1ccc(F)c(C(=O)NC(Cc2ccoc2)C(=O)NCc2ccc[n+]([O-])c2)n1 70399,C12(NC(C(CCC)N(C)C)=O)CN(C(c3nc(C)ncc3Cl)=O)C(COC)(C1)C2 70400,c1(C(=O)NC2CCCC(N(C(CN3CC(CC)C3)=O)C)C2)cn2nc(C)sc2n1 70401,N1(C(C(C)=C2CCC2)=O)CCC(CN(C)C(C2CCCN2CC(F)(F)F)=O)C1 70402,C1(C(N2CC3C(CNC(C4CCCC4)=O)(C3)C2)=O)CCN(CCO)C(=O)C1 70403,CCC(CC(=O)N1CC2C(C(=O)NCC(C)(C)CN=[N+]=[N-])C2C1)C(F)F 70404,CCCCCCCCCC(=O)NCC1CN(C(=O)C2=NNC(=O)CC2)CCO1 70405,c1(C(N(C)Cc2ncc(Cl)cc2Cl)=O)nc(S(N)(=O)=O)c2ccccn12 70406,C(C(COC)CC(=O)NCCCC(=O)NCC1COCC1O)OC 70407,c1(C(=O)NC(CC)CN(C(=O)C(O)C2CCCC2)C)ncn(-c2ccccc2)n1 70408,C1(C(N2CCC(CO)(CNC(=O)C3=CCSC3)C2)=O)(OC)CCCOC1 70409,C(=O)(C(C)(C)C(C)O)N1CCCC(CN(C(c2c(C)oc(Cl)n2)=O)C)C1 70410,c1(C(N2CC(NC(c3ncc(OCC)nc3)=O)C(O)C2)=O)cc(C)nc(Cl)c1N 70411,Cc1nc(C(N2CC(O)CC2CNC(=O)CSC2CCCCO2)=O)sc1C 70412,C1(C2CC2)(C(=O)NC2CC(CCNC(C34C=CC(CC3)C4)=O)C2)CCOCC1 70413,c1(CC(=O)NC(CC)(CNC(c2ccn(C)n2)=O)CC)cccc2c1OCO2 70414,Cc1ccc(F)c(C(=O)NC2CC3CC2CC32CC2)c1Cl 70415,C1(CNC(C(CCSC)O)=O)CCCC2CN(C(=O)CCCCC(C)(C)C)CC12 70416,c1(C(N2C(CNC(CC(CCC)(C)O)=O)CC2)=O)cc(F)cc2nccnc12 70417,C1(NC(c2c(C)cc(C)[nH]2)=O)CS(=O)(=O)CC1NC(=O)CCC1CCCCC1 70418,C#CCC(C(=O)NC)NC(=O)NC1(C)CCN(CC)C1 70419,C1(NC(C(CSC)O)=O)CN(C(c2ccc3ncncc3c2)=O)CC1S(C)(=O)=O 70420,C(=O)(C(O)C(F)(F)F)NCCSCC(=O)NCCc1csnn1 70421,c1(C(N(C(CN(C(C(COCC)C)=O)C)C)C)=O)cc2n(n1)CCCC2 70422,N1(C(CCc2cc(NC(=O)OC)ncc2Br)=O)CCc2cccc(F)c2C1 70423,C(CN=c1[nH]c(Cl)ncc1C)C1CC(NC(C2(CC)CCNC2=O)=O)C1 70424,C=CCC(C(=O)NC1CCCCC1CNC(c1c[nH]nc1Br)=O)C(C)C 70425,c1(C(=O)NCCCN(C)C(C2CC(O)(C(F)(F)F)C2)=O)ncn2c1CCCC2 70426,C1(NC(CCc2cnc(C)nc2O)=O)CN(C(=O)Cn2ncnn2)CC1C1CC1 70427,N1(CC(=O)NCC2CC(C)N(C(=O)CN(S(C)(=O)=O)C)C2)CCC(=O)NC1=O 70428,N1(C(=O)C(C2CCOCC2)F)CCN(C(=O)CCCn2ccnn2)C(CC2CC2)C1 70429,Cc1cc(C(=O)NC2CN(C(c3cc(O)cc(O)n3)=O)CCC2CO)cnc1F 70430,N1(C(=O)CC2(O)CC2)CCC2C(C1)CN2C(C1CCOCC1)=O 70431,c1(CC(=O)NC2CCCC(NC(COCCC#C)=O)C2)noc2ccc(F)cc12 70432,Cc1nc(C(N2CCC(C(C)NC(=O)CCCc3cccnc3)C2)=O)c(C)s1 70433,N1(C(c2c(F)cccc2Cl)=O)CCC2C(CCN2C(=O)CCn2cncn2)C1 70434,C=CCC(C)C(=O)NC1CCC(N(C(=O)CC2C(=O)NN=C2C)CC)CC1 70435,c1(C(N2CC(COC)(NC(C3C4CCCC34)=O)C2)=O)ccc(Cl)cn1 70436,C1(C2CC2)(CNC(c2c(C(C)C)ccs2)=O)CCN(C(=O)C(O)C2CCC2)C1 70437,N1(C(=O)NC(c2ccccc2Br)c2cc[nH]n2)CCC2(CCCCC2)C1 70438,c1(CC(N2CC(C(C(=O)NC(c3nccs3)CC)O)C2)=O)cncnc1 70439,C1(CNC(C2CC23CCCC3)=O)CCCN(C(C2(F)CC2(Cl)Cl)=O)C1 70440,CC1C(=O)NC(=O)CN1C(C1(C)CN(C(c2cc(=N)[nH][nH]2)=O)C(C)(C)C1)=O 70441,C(C(CO)C(F)(F)F)NC(C(CC1CC1)NC(c1nn(C)c(O)c1)=O)=O 70442,CCC(CO)C(=O)NC(C)CC(C)NC(C1(NC(C)=O)CCCC1)=O 70443,C1(CC)CCN(C(C2CC23CCC3)=O)C1C(=O)NCC(=O)NC(C)C 70444,CC(CC=Cc1ccccc1)C(=O)N1CCC(NC(C2OCCO2)=O)C1 70445,C(C)(CCCC(=O)NCC1OCC2CCC1C2)NC(CCCNC(C)=O)=O 70446,C12(NC(CN=S(C)(C)=O)=O)CCOCC1CN(C(c1cc(Br)co1)=O)C2 70447,C(=O)(C1CCCn2ccnc21)N1CCCC(O)(CNC(CCCS(N)(=O)=O)=O)C1 70448,c1(C(=O)NCCOCCN(C)C(C2(C)CCNC2=O)=O)ccc2c(n1)CCO2 70449,C(CN=C(NC(C)CNC(=O)OC(C)(C)C)NCCCF)c1ncc(C)nc1 70450,C(c1ccc(C(N)=O)o1)=CC(=O)NCCN(C(=O)C(F)CC1CCCC1)CC 70451,CC(CNC(C1(C)CC1(C)C)=O)CC(=O)N(C)CC1(C)CC1 70452,C1(NC(CCC(=O)NC)=O)CC(O)CN(C(=O)CCCNC(N)=O)C1 70453,c1(C(=O)NC2C(N(C(=O)CCC3CCOC3)C)CCCC2)cccc2nc[nH]c12 70454,c1(C(=O)Nc2scc(-c3c(C)ccs3)n2)cc(F)c(F)c(Cl)c1 70455,C1(CCC(=O)N(C2CC(C)C2)C)CCCCN(C(C2(O)CCOC2(C)C)=O)C1 70456,C1(NC(CC2(NC(C)=O)CC2)=O)CC2C(NC(=O)C(c3ccccc3)C)C2C1 70457,N1(C(C(CC)NC)=O)CC2CN(C(c3cnc(Cl)c(C)c3)=O)CC12 70458,Cn1nnc2c1CCC(C(=O)NC1CCC13CCN(C(=O)C(C)(C)CF)CC3)C2 70459,N1(C(C(CCC)(C)O)=O)C2CCC1C(C)C(NC(C1CCC(C(C)C)CC1)=O)C2 70460,c1(NC(N2CC(CN3CCOC3=O)C2)=O)cc(Cl)ccc1I 70461,N1(C(CCCNC(CCCOC(C)=O)=O)=O)CCCCC1CF 70462,CC(C)CC(CNC(C1CC2CC2N1C(C12CCC(CC1=O)C2)=O)=O)CO 70463,C1(NC(c2cnn(CC(F)F)c2)=O)CC1C1CCCN(C(=O)C(F)(F)C(F)F)C1 70464,C1(CNC(C(=O)NCC)=O)CN(C(c2cn(C3CCOC3)nn2)=O)C(C)(C)C1 70465,C(=O)(CS(=O)(=O)c1ccccc1F)N1CCC(CC=C)(NC(=O)CC=C(C)C)C1 70466,CCCC(CC)CCC(=O)N1CCCC1(C)CNC(c1cncnc1)=O 70467,Nc1cc(C(=O)NCCOC2CN(C(=O)CCc3ccncn3)C2)cc(Cl)n1 70468,C1(C(N2CCCC(CN3CCCC3)C2)=O)Cc2ccc(O)cc2CN1 70469,C#CCC(CC#C)C(=O)N1CC2CCC1C(CNC(=O)CC=CC)C2 70470,c1(C(=O)NCCN(CC(=O)NC2CC2)C2CC2)ccoc1I 70471,c1(CN2CCN(C3CCN(C(C4CC5(CC5)CO4)=O)C3)CC2)cc(Cl)cc(Cl)c1 70472,C12(CC)CCC(C(=O)NC3CC3CNC(=O)CCc3ccc(F)c(F)c3)(CO1)C2 70473,c1(C(N2C(CCCNC(CN(C(C)=O)C)=O)CCC2)=O)cc(C(F)F)ccn1 70474,C#Cc1ccc(F)cc1C(=O)NC1CN(C(=O)CC(C)F)CC1n1cccn1 70475,C(=O)(C(C)C(CC)CC)N1C(C(=O)NCC(=C)Br)CC(=O)C1 70476,c1(C(=O)NC2(CNC(c3n(C=C)nnc3)=O)CCOC2)cc2sc(Cl)cc2s1 70477,C(CNC(c1cnc(C#N)s1)=O)(C(C)(C)C)NC(C1(COC)CC1)=O 70478,C=C(C)C(C)(C)C(=O)NC1CN(C(=O)C(=O)NCC2CC2)CCC1CO 70479,c1(C(=O)NC2(CCNC(CCC#CC)=O)CCC2)ccc2ccnc(Cl)c2n1 70480,c1(C(N2C(C)(COC(c3c(OC)c(Cl)sc3)=O)CCC2)=O)n[nH]c2c1CCC2 70481,C#CCC(C)(C)C(=O)N1CC(C(=O)Nc2cncc(N(C)C)c2)C(C(C)C)C1 70482,C(=O)(CCCCCN(C)C)NC(C)CC(N1CCC(C#N)C1)=O 70483,C1(C(=O)NC2C(NC(c3c(Cl)cn(CCC)n3)=O)CCC2)CCc2nncn2C1 70484,C1(CC(N2CCC(C(=O)NCCCC3CCC3)C2)=O)CC(C2CC2)C1 70485,c1(C(=O)NC2(C)CC(NC(CC(=C=C)C)=O)C2)cc[nH]c2nccc1-2 70486,CC(C)C1=NOC(C(N2CCC(C(C)NC(C3CC(=O)C3)=O)C2)=O)C1 70487,C=C=CCCC(=O)NCCC1CCC(NC(=O)CCS(C)=O)C1 70488,C1(C(=O)NCCc2cn(C)nc2)CN(CC2CCC(=O)NC2)CC1C#N 70489,C1(NC(C=CC(C)(C)SC)=O)CCCC1NC(=O)C(C)CC1CCC1 70490,N1(C(c2cc(C)ncc2)=O)CCC2CC2(C(N2CCC(OC(C)C)CC2)=O)CC1 70491,c1(C(=O)NC)ncnc2c1ncn2C1CC(c2ccccc2OC)C1 70492,c1(C2C(C(N(C3CCN(C(C4(O)CC4)=O)CC3)CC#C)=O)C2)ccc(OC)cc1 70493,N1(C(C(C)(C)O)=O)CCCC(C2CCN(C(=O)C=CCOCC(F)(F)F)CC2)C1 70494,c1(C(=O)NC2CC(CNC(CCCOCC=C)=O)C2)ccc(NC(C)C)c(F)c1 70495,c1(OC)ccccc1NC(=O)C(C(C)C)N1CCN(S(=O)(=O)C(C)C)CC1 70496,C(=O)(C(O)C(C)(C)C)N1CC(C)C(CNC(C2(C)CC(O)CN2C)=O)C1 70497,C1(NC(c2cc3ncccc3o2)=O)CC2CC1CN(C(c1cc(Cl)sc1Cl)=O)C2 70498,N1(C(C2C(C)=CCS2)=O)CC2(CC(C(=O)NC3CN(CC(F)F)C3)CO2)C1 70499,c1(CCC)ccc(C(N2CCCC2CNC(c2cc(C)[nH]n2)=O)=O)cc1 70500,C(CC(=O)NC1CCC12CCCC2)(C(C)OC)NC(C(COC)(C)C)=O 70501,C(=O)(CCCCC(=O)NOC(C)(C)C)NC1CC(NC(C(CC=CC)CC)=O)C1 70502,c1(OC)cc(C)cnc1C(N1CCC(O)(CCNC(C2C(C)C2C)=O)CC1)=O 70503,CC1(C)C(=O)NCC1NC(C1COCCC1NC(c1cccc(O)c1F)=O)=O 70504,C(=O)(CCC(=O)NC1CCC1NC(c1cccc(F)c1)=O)N(CCC)CCC 70505,C1CCCC(NC(C)=O)C1.C12CCC(C1)NC(=O)C1(CC1)CCNC2=O.CC 70506,C(=O)(CCCCNC(c1snc(C)c1N)=O)NCC(C(=O)NC)C 70507,N1(C(C(CC(C)C)N(C)C)=O)CCC2(CC(C(N3CC(O)CC3(C)CO)=O)C2)C1 70508,N1(C(c2cncc(NC)c2)=O)CC(O)C(O)C1CNC(C1CC1OC)=O 70509,N1(C(C=CC)=O)CCN(C(C2CC3CC23)=O)CC1 70510,C(=O)(C(C(C)(C)C)SC)NCC1CN(C(c2c(COC)ncs2)=O)C1 70511,C(=O)(C(CO)C(C)(C)C)N1C(c2n(C)ncc2)CN(C(=O)CNC=O)CC1 70512,CCCCS(=O)(=O)NC(C(=O)N1CC(CO)(NC(=O)C(C)CF)C1)C(C)C 70513,C1(C(=O)NCCCCCCN(C(CCC(C)OC)=O)C)CCCN2CCCCC12 70514,c1(CCC)ccc(C(N2CC(NC(=O)C(F)F)CCC2C)=O)cc1S(N)(=O)=O 70515,C1(C(=O)NCCOC2CN(C(CCc3cnc(C)s3)=O)C2)CN(C)CCO1 70516,C=CCC(F)(F)CNC(C1(C(C)C)CCN(C(c2ccc(CC)[nH]2)=O)C1)=O 70517,N1(c2n(CCOC)c(CC3(S(C)(=O)=O)CC3)nn2)CC2CN2C=NC=CC1 70518,Cc1cc(C(=O)NC(CO)C(C)NC(C2(C3CCCCO3)CCC2)=O)nn1C 70519,c1(C(N(C(CCNC(c2cccc(CC)c2)=O)C)C)=O)ccc2snnc2c1 70520,CN(C)NC(=O)CCC(=O)Nc1ncc(CC2CCC(F)(F)CC2)s1 70521,CC1(C)CNCC1OCC(=O)NCCC(c1ccccc1)CO 70522,C1(NC(c2c(C)cc(CNC(C(C)=CC3CC3)=O)o2)=O)CCCC1C1CC1 70523,C1(CC)CCCN(C(n2nnnc2C)C(=O)N(c2ccccc2)CCC#N)CC1 70524,c1(C(N2C(CNC(C3(CC(C)C)COC3)=O)CCCC2)=O)cnc(F)c(Cl)c1 70525,c1(NC(C2CCN(Cc3c(CC)cccc3)C2)=O)cc(F)c(F)cc1Cl 70526,c1(CN(C(=O)C(N2CCCCC2c2nnc(C)o2)=O)CCOC)ccc(F)cc1F 70527,C1(NCCCNC(N(CCCC#C)CC)=O)CCN2CCCC2C1 70528,C(=O)(CC(C)C(F)F)NC1CN(C(c2nc(C)oc2C)=O)CC1C 70529,Cc1cc(C(=O)NC2CCCCC2NC(c2cccs2)=O)nn1CC(F)(F)F 70530,c1(NC(CN(C(=O)C(N2CCOCC2)C)CC#C)=O)cnc(C)c(C#N)c1 70531,C1(CC)CCN(C(C2CCC2COC)=O)C(C(=O)NC2C(O)CC2O)C1 70532,n1(CC(N2CC(CNC(COc3cccc(C)c3)=O)C2)=O)cc(P(C)(C)=O)cn1 70533,c1(CC)c(C(N2CCN(C(=O)Cc3cc(C4CC4)no3)C3CC23)=O)cccc1C 70534,N1(C(CC2(C#N)CC2)=O)C2CCC1CN(C(C1Cc3cccnc3C1)=O)C2 70535,CC1(C)OC2CC(C(=O)NC3CC(NC(C4OCC5CCC4C5)=O)C3)CC2O1 70536,Cc1ccc(-c2cnc(NC(=O)C(C)NC=O)c(O)c2)c(C)n1 70537,n1(CC(N2C(C)CC(CNC(=O)CSC3CC3)C2)=O)ccc(O)nc1=O 70538,c1(NC(C)=O)ccc(Cl)c(C(=O)NC2CCCC2NC(c2nccn2C)=O)c1 70539,C1(C(N2CC=C(CNC(c3cc(=O)cc[nH]3)=O)CC2)=O)CC1C1CCCCC1 70540,N1(C(C(C)Oc2ccc(F)nc2)=O)CCC(NC(c2c[nH]nc2F)=O)CC1C 70541,C1(CNC(c2ccc(C(F)(F)F)[nH]2)=O)CN(C(C2CSC2)=O)C2CC12 70542,N1(C(c2c(N)ccc(Cl)c2)=O)CCCN(C(C2(CO)CC2(F)F)=O)CC1CO 70543,c1(OC(C)C)cccc(C(=O)NCC(CO)NC(c2cc(O)cs2)=O)n1 70544,CC(O)C(F)(F)C(=O)NC1CC(F)(CNC(=O)C(c2ccccc2F)(C)C)C1 70545,C1(CC(=O)N(C(C)CNC(C2CCC(N(C)C)CC2)=O)CC)CCS(=O)(=O)C1 70546,c1(C(=O)NCCN(C(=O)CC2CC(F)C2)C)cn(C)cc1C(F)(F)F 70547,c1(CN2CCC(CC(=O)Nc3c(C(N)=O)ccnc3)C2)ccc(F)c(F)c1F 70548,Cc1cc(CC(=O)NC2CCCC(NC(=O)CCOCC(C)C)C2)cc(C)c1 70549,c1(CCC)nc(C)c(C(N2CCC(NC(C3CC3C)=O)C2C)=O)s1 70550,c1(C(=O)OCC2CC3(CCC3)C2)ccc([N+](=O)[O-])c(O)c1 70551,Cc1c(Br)ccc(O)c1C(N1CC(NC(=O)CCC2CCC(C)O2)C1)=O 70552,C1(CC)CC(C(N2CCC(F)(CNC(c3cc(F)n(C)n3)=O)C2)=O)CC(=O)N1 70553,O=C(C(=O)C(F)(F)F)NCCC1CCN(C(C2CCCCC2O)=O)C1 70554,C1(C)(CNC(C2(OC)CC2)=O)CCC(NC(c2cc(CCO)on2)=O)C1 70555,C(=O)(CCS(C)=O)N1CC(C(C)NC(=O)C(C)(C)N2CCOCC2)C1 70556,C1(NC(=O)CC2CCCC2)CCCC12CCN(C(=O)CC1CC3(CC3)CO1)CC2 70557,C1(NC(c2cc(O)nc(C3CC3)n2)=O)CC2CN(c3ncc(F)cn3)CC2C1 70558,N1(C(CNC(=O)NC)=O)CCN(C(=O)CC(C)(C)C2CC2)C(C(F)F)C1 70559,C1(CC#C)(C(=O)N(C)CCN(C(=O)CCOCC2CCC2)C)CCOC1 70560,N1(C(=O)C=Cc2ccc[nH]2)CC23CCCC2(C1)CN(C(c1cc[n+]([O-])cc1)=O)C3 70561,C1(NC(C2(F)C(C)C2)=O)CCC(C)N(C(=O)Cc2ccc(C(F)F)cc2)C1 70562,CC(C)C(C)C(CNC(=O)CCN1CCCC1)NC(c1ccc(CO)cc1F)=O 70563,c1(SC)cc(C)ccc1C(=O)NCC1(O)CCN(C(c2nn(C)cc2C)=O)C1 70564,C1(CNC(C2CN(C(C)=O)C2)=O)CC(NC(c2n[nH]cc2Br)=O)C1(C)C 70565,c1(N2C(CCNC(=O)CN3CCS(=O)(=O)CC3)CSCC2)ncccc1[N+](=O)[O-] 70566,C(C1c2ccccc2CCN1C(c1ccc(C(N)=O)c(Cl)c1)=O)NC(C(C)C)=O 70567,c1(OC)cccnc1CN1CCCC(C(=O)NCCCN2CCCC2)C1 70568,c1(C(=O)NCCCN(C(c2cc(CCC)on2)=O)CCC)ccncc1OC 70569,N1(Cc2cn(CCC(C(=O)OCC)C)nn2)CCC12CCSCC2 70570,C1(NC(c2ccc(S)cc2)=O)CN(S(=O)(=O)c2cccs2)CC1(F)F 70571,c1(CC)ccc(C)c(C(=O)NC2(CF)CCN(C(=O)C(C)C(O)CC)C2)c1 70572,c1(CC(C2CCN(CC(F)(F)F)CC2)NC(=O)Cn2cnnn2)ccccc1Cl 70573,C1(C(=O)NCC2CCN2C(=O)CSC(F)(F)F)CCCC1C(F)(F)F 70574,c1(C(N2CC(C(C)(C)O)(CNC(=O)CNC=O)C2)=O)cc2n(n1)CC(F)C2 70575,CC1CC(c2nnnn2CC2CCOC2)(NCC(C)(C)CO)CC(C)O1 70576,N1(C(c2c(C)n(C)cn2)=O)CC(C(=O)NCc2cnn(C)c2O)CC1(C)C 70577,C(C#Cc1cccnc1)NC(C1C(NC(c2cccn3cncc23)=O)CC1)=O 70578,N1(C(C(=O)NCCN(C(C2CC(OC)C2)=O)CC)C)CCCC(O)C1 70579,c1(CC(=O)N(CC(CNC(CC2CC(OCC)C2)=O)C)C)cc(C)on1 70580,N=c1ncn(CCC(=O)NCC2(C(=O)N(C3CCOC3)CCF)CCCO2)[nH]1 70581,C(C1=CCN(C(=O)CC2CCCS(=O)(=O)C2)CC1)NC(CC1CCC(C)CC1)=O 70582,N1(C(=O)OC(C)(C)C)CCC(C(=O)N(C2CCC2)CC2CC2)C1 70583,C1(C)CCC2CC2C1.C1(N(C(C2C(C(=O)OCC)C2)=O)CC)CCN(C=O)C1 70584,C1(C(N2C(C(=O)OC)C=CCC2)=O)CCN(C(=O)CC(C)(C)SC)C(C)(C)C1 70585,N1(CCN(C)C(C2CCOC(=O)CC2)=O)CCSC(C)(C)C1.C12CN(CCO1)C2 70586,C1(Cn2cc(-c3c(C)nsc3)nn2)CCCCN(C(C2(C)C=CCC2)=O)C1 70587,N(C1CCCn2nccc21)C(C1(C=C)CCN(C(c2n[nH]c(C)c2O)=O)C1)=O 70588,Cc1ccc(C(C)CC(=O)NC(C)C(C)(C)NC(c2ccsn2)=O)cc1 70589,c1(NC(c2c(C)n[nH]c2)=O)ccc(C(=O)Nc2ccc(F)c(C(=O)O)c2)cc1F 70590,c1(OC)ccc(CO)cc1C(=O)NC(CNC(=O)CN1CCCCC1=O)C1CC1 70591,c1(C(=O)NCC(CN(C(=O)C=C2CCSCC2)C)(C)C)ccc2ccsc2c1 70592,CCC(CC(=O)NC(C(=O)N(C1CCSC1)C)C(C)O)C(F)F 70593,C12(C(=O)NCC(C)(C)C#N)CC(CN(C(C3C4CCC(F)C34)=O)C1)C2 70594,C1(C)(C(N2CCC(O)(C(C)NC(C(C)NC(N)=O)=O)CC2)=O)CCCCCCC1 70595,N1(C(c2c(CC)cco2)=O)CCCN(CCNC(=O)Cn2cncn2)CC1 70596,Cc1c(C(=O)NCC2CC(NC(C34CC(C)(C3)C4)=O)C2(C)C)cccc1O 70597,C#CC(C)(C)C(=O)NCc1nc(C(=O)NC(C)CC)c(C)o1 70598,C(=O)(CCCCC#N)N1CC(CNC(C2(C)C=CCC2)=O)OCC1 70599,C#CC1(NC(=O)C(C)(C)CN(C)C(c2ccc(=N)[nH]c2)=O)CCOC1 70600,N1(C(=O)COC2CCOC2)CCCC(C2CCCN(C(c3ccc[n+]([O-])c3)=O)C2)C1 70601,C1(NC(CN(C)S(N)(=O)=O)=O)CCCC12CN(C(=O)Cn1cc[nH]c(=O)c1=O)C2 70602,c1(C(=O)Nc2ccc(-c3c(F)cccc3F)cn2)cc(F)c(Br)c(F)c1 70603,C(=O)(C(C)CC(C)C(C)=O)NCCn1cc(C(N2C(C)(CCC)CC2)=O)nn1 70604,C1(CNC(c2cn(C)nc2)=O)CC2CCC1N(C(c1cc3n(n1)CC(F)C3)=O)C2 70605,c1(C(N(C(CNC(c2ccc(C)c(O)n2)=O)C2CC2)C)=O)ccc2[nH]ccc2n1 70606,N1(C(C(COC)(C)C)=O)CCC2(CC1)OCCCC2NC(c1c[nH]nc1OC)=O 70607,c1(CN(C)C)ccc(C(N2CCC2CNC(c2csc(=N)[nH]2)=O)=O)[nH]1 70608,C#CCC(C)C(=O)N1CCC(C(C)NC(c2ccc(C3(C)CCO3)cc2)=O)CC1 70609,c1(C(C(C)C)NC(CCc2cn(CC)nc2C)=O)ccc2ncccc2c1 70610,N1(C(C2N(CCC)CCCC2)=O)CCC(F)(CNC(=O)CC(C)(C)O)CC1 70611,C12CCC(C1)NC2=O.c1(C(=O)NCCNC(C2(Br)CC2)=O)ccco1 70612,c1(OC)ccc(C(N2CCN(C(C3(c4ccn(C)n4)CC3)=O)C(C)C2)=O)c(Cl)c1 70613,C(C)(C)(C=CC(=O)NC1(CC(=O)NCC(C)SC)CCC1)SC 70614,C(CCC(C)CCC)c1nc(-c2ccc(OCC)cn2)on1 70615,c1(CC)nn(C)c(CC(N2CCCC(NC(=O)C(C)CC3CCC3)C2)=O)c1Cl 70616,C1(C(N2C(CNC(c3n(C)cc(C#N)c3)=O)CC(F)C2)=O)CNC(=O)C(C)(C)C1 70617,C(C(=O)N1CC(NC(=O)Cc2ccc(C(N)=O)nc2)C(C)C1)(C(C)C)OCC 70618,c1(-c2nc(C(C)NC)nn2Cc2cncc(F)c2)cc2c(OC)cccc2[nH]1 70619,C1(NC(c2c(C)ocn2)=O)CN(C(=O)C(C)OCC(C)C)CCC1F 70620,C(CCCCC(=O)NCC(C)(C)OCCNC(C1CCC(N(C)C)C1)=O)SC 70621,Cc1nn(C)c(N)c1C(=O)NCC(C)NC(c1cccc(C(N)=O)c1C)=O 70622,CC(C)C(C(=O)N1CC(CCCCNC(C2CC3C=CC2O3)=O)C1)NC=O 70623,C#CC1(NC(C2(CNC(=O)C(C)OCCN(C)C)CC2)=O)CCOC1 70624,CCCCC(CNC(c1ccc(F)s1)=O)NC(=O)C(O)C1CCC1 70625,N1(C(CC2C(=O)OCC2)=O)CCC12CN(C(C1CCCCCC1)=O)C2 70626,Cc1c(C(=O)NCC2COC(C)(C)CN2C(=O)C=CC2CCC2)nc2sccn12 70627,c1(CCCNC(CN(CCOC)C(C2C=CCS2)=O)=O)nc[nH]n1 70628,n1(CC)nc(C(=O)NCC(C)(CNC(=O)Cn2cc(C3CC3)nn2)OC)cc1C 70629,N1(C(c2cc(C)no2)=O)Cc2ccc(O)cc2CC1C(N1CC(F)CC1C#N)=O 70630,C1(CCC2N(C(C(F)OC)=O)CCC2)CCN(C(=O)COC2CCCC2)CC1 70631,c1(CNC2CCN(C(N3CC(C)CC(C)C3)=O)C2)ccc(S(=O)(=O)C(F)F)cc1 70632,N1(CC)CC(C(N2CCCC(N(C(=O)C(C)Sc3ccncc3)C)C2)=O)CC1=O 70633,CCC(CC(=O)NCC(C1CC1)NC(=O)Cc1cnnn1C)SC 70634,CC(C)CC(C)C(=O)N(C1CN(C(=O)CC2COCC2(C)C)C1)C 70635,C1(NC(C(c2cn(C)nc2)=O)=O)CC(NC(=O)CCN2CCCCC2)C12CCC2 70636,Cc1cc(C)c(C(N2CCN(C(=O)CC3COCCN3C)C(CO)C2)=O)c(C)c1 70637,c1(C(N2CCCC(OC3CC3)C2)C(=O)NCC)nc(Br)ccc1OCC(C)C 70638,C(=O)(CC(P(C)(C)=O)P(C)(C)=O)N(C(CNC(C(CCC)O)=O)C)C 70639,c1(C(N2C(C)CCC(CNC(=O)CCC(C)(C)C)C2)=O)ccc2n[nH]cc2c1 70640,c1(CC)ccc(CNC(c2ccn(C3CC3)n2)c2nnnn2CC)o1 70641,C(CC)(CCCCCC)NC(C(CCCC)NC(c1ccc(C)nn1)=O)=O 70642,C12(NC(c3cc4n(n3)CC(F)C4)=O)CCCC1CN(C(c1cc(O)cs1)=O)C2 70643,C=CCC(F)(F)C(=O)NCC(F)CNC(c1ccc([N+](=O)[O-])o1)=O 70644,c1(C(=O)NC2CCN(C(c3ccc(OC)s3)=O)CC2F)ccc2nc(O)oc2c1 70645,Nc1ccc(C(=O)NCC(CO)NC(C2CCCN2C=O)=O)c(Cl)c1 70646,c1(CNC(C(=O)NCC)=O)cccc(CNC(C2CCC(F)C2)=O)c1 70647,N1(C(C=Cc2cn(C)nc2)=O)CC2COCCC2(NC(=O)C(F)=C2CCCC2)C1 70648,C1(CNC(C2(CC#C)CCC2)=O)CCN(C(=O)CN2CCCCC2C)CC1 70649,c1(C(=O)NCC2CN(C(C(C)=C3CC3)=O)C2)ccc(C(F)F)nc1 70650,CCCC(O)C(=O)N1CCC(OCCNC(c2coc(C#N)c2)=O)C1 70651,c1(C(=O)NCC(CC(=O)NCC(CC=C)(C)C)C)cc(F)cnc1O 70652,c1(CC(=O)NC2CCN(c3ccn(C)n3)C2=O)noc2cc(Br)ccc12 70653,C(C(C)N=c1nc(OC)cc(OC)[nH]1)N(C(CCC(=O)NC)=O)C 70654,CC(C)C(C(=O)N1CC(NC(=O)CSC(F)(F)F)C(C)C1)NS(=O)(=O)C1CC1 70655,CC1CN(C(C2CC(C)(C)CO2)=O)CC1C(=O)NC1C=CCC1 70656,C1(NC(c2ccn(CC)c2C)=O)CN(C(C23CCCC2C3)=O)C2(CCCCC2)C1 70657,C(CC(C(=O)NCC1CCCCO1)NC(=O)CC1CCC(=O)C1C)OC 70658,C(CCCCCNC(=O)CC1CCC1(C)C)NC(c1cc(CCC)[nH]n1)=O 70659,C=C=C(C)CC(=O)NC(C1CCCN1C(=O)CCSc1nccn1C)C 70660,C(=O)(C1=CCCCO1)N(C1CCCN(C(C2(CC=C)CCOC2)=O)C1)CC 70661,N1(C(COCCOCC#C)=O)CCN(C(=O)CN2C(C)CCC2C)C2CCC12 70662,C1(CC=C)(NC(C2CCN2C(C)(C)C)=O)CN(C(=O)Cc2ccsc2)C1 70663,c1(OC)ccc(C(=O)NCCC(C)NC(=O)C(O)Cc2ccc(F)cc2)cc1C 70664,N#CC1CN(C(=O)N(Cc2ccncc2)CC23CC(CO2)C3)CC12CCC2 70665,C1(NC(C2CC(NC(c3ccoc3)=O)C2)=O)CCCC(O)CC1 70666,CC(C)(CCCO)CN=c1[nH]c(=NCC2CCOC(C)(C)C2)c2sccc2[nH]1 70667,c1(C(=O)NCCCNC(CC(COC)(C)O)=O)[nH]c2ccccc2c1Cl 70668,CCCC(C(=O)NC(C)CC1CN(C(c2coc(C#N)c2)=O)C1)S(N)(=O)=O 70669,c1(CN(C(=O)NC2CCC(C)(CC)CC2)CC)cc(Br)ccc1C 70670,c1(OC)cc(C)cnc1C(=O)NC(C(C)NC(c1cn(C2CC2)cn1)=O)C(C)C 70671,N1(C(C=C(C)C)=O)CCC2CN(Cc3c(C)cccc3Br)CC12 70672,Cn1cnc2ccc(C(=O)NCC3CC4CCC3N4C(c3cc(Cl)on3)=O)nc12 70673,Cn1ncc2nc[nH]c(=NC3CCCC(C(=O)NCCc4ccc(O)cc4)C3)c12 70674,CP(C)(=O)c1ccc(C(=O)NCC(C2CCC2)NC(c2ncccc2N)=O)cc1 70675,CC(C)(CNC(C1CC2CC1CC2O)=O)CC(=O)NCCC1(CO)CC1 70676,N1(C(C=CCNC(=O)CCC2OCCO2)=O)CC(O)CC12CCC2 70677,N1(C(CC2CN(C)CC2O)=O)CC(NC(c2ccoc2C2CC2)=O)C(C)(C)C1 70678,C(=O)(CC(C(=O)OCC1CCCCNC1=O)N1CCNCC1)OC 70679,C1(C(N2C3(C(N4CCC(O)(CC)C4)=O)CC3CC2)=O)C2CCC(C2)C1C 70680,c1(C(=O)NC2CC(CCC(=O)NC3(CCCC)CC3)C2)cnc(C)n1C 70681,Cc1c[nH]c(C(=O)NCC2CCCN(C(=O)CCc3nccn3C(F)F)C2)c1C 70682,N1(C(C(=O)NC2C(NC(CCCC)=O)COC2)CC)C(=O)CCC1=O 70683,N1(C(C(C)N(C(C2CC(=O)CC(=O)C2)=O)CC)=O)CC(C)CCCC1C 70684,C=CCC(CNC(=O)C(C)(C)N(S(C)(=O)=O)C)NC(=O)C(C)(C)C1CC1 70685,C(C(C)C(=O)NCCNC(N)=O)N(C(C(C)SCC)=O)C 70686,c1(C(=O)NC2C(CNC(CCC#CC)=O)C2)cc(F)cc(Br)c1F 70687,C1(C(N(CCN(C(c2ccsc2)=O)CC)CC)=O)CC2(C1)CC(F)(F)C2 70688,c1(C2(C(=O)OC)CC2)ccccc1F.C(C1(C)CN1)NC(C1C(C(=O)OC)C1)=O 70689,C(=O)(C(CNC(C1CC=CCC1)=O)C(C)(C)C)N(CCCSC)C 70690,C1(NC(=O)CCC2CCOC2)CC(O)(CNC(c2ccc(CO)s2)=O)C1 70691,N1(C(CC2CC(OC)C2)=O)CCC2CN(C(=O)C=CI)C2C1 70692,N1(CC(=O)NCC(CO)NC(C2(COC(C)C)CC2)=O)CCS(=O)(=O)CC1 70693,N1(C(CC(CC)C)=O)CCC(C2CC2NC(c2cc(C)cc(Cl)c2)=O)CC1 70694,Cc1ccccc1CCC(=O)NC1CCN(C(c2cnccn2)=O)CC1 70695,c1(OC)cc(C)c(NC(CCC(F)F)C(N)=O)cc1Oc1ccnc(CO)n1 70696,N1(C(CN(C2CCC2)C(C)=O)=O)CC2CCC(N(C)C)C2C1 70697,C(=O)(C1=CCCN(C(C2(COC)CCCO2)=O)C1)NC(CCCC)(C)C 70698,CCC(CC(=O)NCCCCn1cc(CC(C)(O)c2cccs2)nn1)CC(F)(F)F 70699,S1(=O)(=O)CC(=O)NN1C(C)C.C1(NC)C2CC1N(C(c1ncccc1SC)=O)C2 70700,N1(C(c2cc(C(=O)OCC)ncc2)=O)CC2CCC1CN2C(C1CC(F)(F)C1)=O 70701,C1(C(N2CC(C(N(C(CO)C3CC3)C)=O)OCC2)=O)CC(=O)NC1(C)C 70702,C(=O)(C(C)S(N)(=O)=O)N1C(CNC(c2c(C)[nH][nH]c2=N)=O)CC1 70703,c1(C(=O)NCCC2CCN(C(C=CSC)=O)C2)cccnc1C 70704,c1(C(=O)NC2CCC(CNC(C(C)c3ccco3)=O)CC2)ccn2cnnc2c1 70705,C1(C(=O)NC2CCN(CC)C2=O)CC(C)(C)CCN1C(C1CC1(C)C(F)F)=O 70706,C1(C(N2C(C(=O)NC)CC2)=O)CN(C(=O)CCc2ccccc2)C2(CCC2)C1 70707,c1(C(=O)NCC2(F)CC(CNC(C(C)(C)N(C)C)=O)C2)cc(Cl)c(F)cc1F 70708,c1(C(=O)NCC2C(NC(C3(C)CC4CC4C3)=O)CCCC2)ccc2c[nH]nc2c1 70709,N1(C(C(C)CC2CC2)=O)CC2(C)CC1(C(=O)NCCC1(C)CCOC1)C2 70710,CCC(CC)C(C)NC(C1(C)CN(C(=O)C(C)NC=O)C1)=O 70711,C=CCC(C)C(=O)NCCCC1(NC(=O)C2=CCOC2)CC1 70712,CC(C)(CCC(=O)N1CC(C(=O)NCC(c2cnc[nH]2)O)C(F)C1)[N+](=O)[O-] 70713,c1(NC(C(CC=C)CNC(C2CC3CCC(C2)O3)=O)=O)cnc(C)c(C)c1C 70714,c1(CC)ccccc1CC(N1CC(C)(NC(C2CC(C)CO2)=O)C1)=O 70715,C=CC(C)C(=O)N(CC(CC)NC(=O)Cc1c[nH]nc1O)C 70716,c1(C(=O)NC2(C)CCN(C(=O)CCc3cnoc3)C2)nccc2ccsc12 70717,C1(C(N2CCN(CC(=O)NC(C3CC(F)(F)C3)C)CC2)=O)CC(=O)C12CCC2 70718,C12(C(N(CC(C)CNC(=O)Cc3cc[nH]c3)C)=O)CCCC1C2(F)F 70719,N1(C(C(=O)NCCOC)=O)CC2CC(NC(=O)Cc3cccc(Cl)c3)C2C1 70720,c1(SCC(=O)N(CCC(C)NC(C(CCSC)O)=O)C)ncnc2[nH]cnc12 70721,CCC(O)C(C)(C)C(=O)N1CCOC(CC(=O)NC2(C)CCCC2)C1 70722,c1(OC)ccc2c(c1F)CCC2NCCc1cncc(Br)c1 70723,c1(C(=O)NCC2CCN(C(CC=C)=O)C23CCC3)ccc2nc(N(C)C)sc2c1 70724,C1(CNC(CC2(C=C)CCC2)=O)CCN(C(c2ccc(N)c(O)c2)=O)C12CCC2 70725,CC1CN(C(=O)CCc2cncc(Br)c2)CC1NC(=O)CCc1cnc[nH]1 70726,C1(C)(C(=O)NC(c2cnc(C)s2)C)C=CCN1C(c1cnn(C)c1Cl)=O 70727,C(=O)(C(F)(F)C1=CCOCC1)N(c1cc(N)c(Cl)c(O)c1)C(=O)OC(C)(C)C 70728,c1(C(N(CC(C)O)CCNC(C(C)OCC)=O)=O)cnc(CC(C)(C)C)o1 70729,C(c1ccc(F)cc1)=CC(=O)NCC1(C(=O)Nc2ccc(F)c(F)c2)CC1 70730,C(C(CO)(CO)NC(=O)C=Cc1cncs1)N(C(=O)CCC1(C)CCC(=O)N1)C 70731,CC(C#N)C(=O)NC(Cn1cccn1)C(=O)N(C)Cc1ccsc1 70732,C(=O)(CC(C)CC(C)C)NC1(CC)CCN(C(C2CN(C)CCN(C)C2)=O)CC1 70733,n1(CC(N2CCCC(C(C)C(=O)O)C2)=O)cc2ncccc2n1 70734,c1(C(N(CC(CC)NC(=O)CC2CNC(=O)C2)CC)=O)ccc(SC)cc1.C(C)=O 70735,C1(C(N2CCN(c3cccc(OC)c3)CC2)C)CCC(F)(F)CC1 70736,C1(C(C)C(=O)NCc2ncoc2CN2CCCC2)Cc2ccccc2O1 70737,CC1C(NC(C2CCCO2)=O)CCN1C(=O)Cn1ccnn1 70738,C(=O)(C1CCCc2nc(C)[nH]c21)Nc1cc(C(=O)OC)c(OC)nc1 70739,c1(NC(=O)Nc2c(C=C)cnn2C)ccc2nc(Cl)cc(C)c2c1 70740,c1(C(=O)NCC2N(C(CC3CCC(=O)C3)=O)CC(F)(F)C2)nc2c(s1)CCCC2 70741,N1(C2C(NC(C3CCOCC3)=O)CCC2)CCN(C(C23CCCC2C3)=O)CC1 70742,CC(C(=O)NCC1(CNC(=O)CCn2cncn2)CC12CCC2)S(C)(=O)=O 70743,c1(C(=O)NC2(C)CC(NC(C(C)Cc3cnc[nH]3)=O)C2)cnc2c[nH]nc2c1 70744,Cn1nc(C(=O)NC2CN(C(=O)CC3CCOCC3)C3CC23)c2ccccc12 70745,c1(C(=O)NCC2N(C(C(CC)NC(C)=O)=O)CCCCC2)cccc2sncc12 70746,O=C(CC1=CCCCC1)NC1CCC(NC(C2(C(F)F)CC2)=O)C1 70747,C1(C(C)C)CN(C(C2CCCCCCC2)=O)CCN1C(C12COC(CF)(C1)C2)=O 70748,C(=O)(CC(C)(C(F)(F)F)N(C)C)N1CCC(N(C(=O)C=CCCC)CC#C)CC1 70749,C1(C)(NC(=O)NCCCC(=O)N(C(CF)CF)C)C=CCCC1 70750,C(=O)(CC(P(C)(C)=O)P(C)(C)=O)NC1CN(C(C2C(C)N(C)CC2)=O)C1 70751,N1(C(c2ccn(C)n2)=O)CCC2OCCN(C(=O)C(O)C(F)F)C2C1 70752,C=C(Cl)C(C)(C)C(=O)NCC12CC1CN(C(=O)C(c1ccccc1OC)=O)C2 70753,Fc1cncc(Cn2c(CN3CCC(CO)CC3)nc(-c3cccc(Cl)c3)n2)c1 70754,c1(CNC(C(=O)NCC(n2cccn2)C)=O)ccc(CN2CCNC(=O)C2)cc1 70755,CC(CC(=O)NCC(CC(=O)N1CC(N2CCNC2=O)C1)C1CCC1)C(F)F 70756,C(=O)(C(C(C)C)C(C)C)NC1C(NC(c2c(Cl)c(C)n(C)n2)=O)CCCC1 70757,Cc1nsc(C(=O)NC2CC(CNC(=O)C(O)C3CCC3)C2)c1N 70758,N1(C(CC2CN(C)C2)=O)CC(NC(=O)COC2CCCC2(C)C)C2(CCC2)C1 70759,C12CC(C(F)(F)F)CN1C2=O.C1(C(C)NC(C23CC(F)(C2)C3)=O)CC(C)(C)CO1 70760,C1(CNC(C2(N(C)C)CCCC2)=O)CCC(NC(=O)Cc2cnccn2)CC1 70761,c1(CC)c(C(=O)NC2(CF)CCN(C(C3CCC(CN(C)C)O3)=O)C2)cnn1C 70762,CC1(C)C2CCC(C(=O)NCC3(O)CCN(C(=O)CNC=O)C3)C1C2 70763,C1(CNC(C2C(CC)CCO2)=O)COC(C)(C)CN1C(c1cc(N)ccc1C)=O 70764,c1(CC)cnc(C(=O)NC2(CN3CCN(C(C4CCC(F)C4)=O)CC3)CC2)cn1 70765,c1(OC)nc(=NC(C)CCNC(C2(C)CC2Br)=O)[nH]c2ccccc12 70766,N1(C(C(C)OCCOC)=O)CC(NC(c2cnc(N(C)C)nc2)=O)C(C)C1 70767,c1(C(N(C2CCN(C(C3C(C)(C(F)F)C3)=O)C2)CCO)=O)cc(C#N)ccc1F 70768,C1(CC(N2C(CO)CC2C)=O)(OC)CN(C(=O)C=Cc2ccoc2)C1 70769,c1(N2CC(CNC(=O)Cn3nnnc3C3CC3)OCC2)ncnc2[nH]cnc12 70770,C1(c2n(CC)nnn2)(OC)CC2(C1)CC(C)(C#N)C2.C12(CCOC1(C)C)NC2 70771,C1(CC)C(NC(=O)CCOC(C)CC(C)C)CCN1C(C1(c2cccs2)CC1)=O 70772,CC1(C(=O)NC(C)(CNC(c2ncccc2C2CC2)=O)C2CC2)CCOCC1 70773,c1(C(N(C2CN(C(CCC=C)=O)C2)C)=O)cccc(OC)n1 70774,C#Cc1ccc(NC(=O)C#CC(C)(C)CNC(c2cncnc2C)=O)c(C)c1 70775,C(=O)(CCCC(=O)NC1CCOC(c2ccccn2)C1)N(CC)CC 70776,CN1CCC(C(=O)NC(C(=O)NCC2(C(N)=O)CC2)C2(C)CC2)C1=O 70777,c1(CN(C(=O)CCN2CCC(F)C2)C)ccccc1CNC(=O)CC(F)(F)F 70778,c1(C(=O)NCC(C)NC(C(COC)C)=O)ccccc1-n1cc(Br)cn1 70779,N1(C(COCCCCC)=O)CCC(C(=O)Nc2cccnc2C)CC1C 70780,C1(C)(CNC(C(CC)CCOC)=O)CN(C(C23CC(C)(C2)C3)=O)C(C)(C)C1 70781,N1(C(c2c(C)csc2)=O)CCC(n2cc(-c3cscn3)nn2)C(O)C1 70782,N1(C(c2cc(CC)n(C)n2)=O)CC(NC(=O)Cc2nccn2C)C(C)(C)C1 70783,N1(C(=O)OC(C)(C)C)CC2(CCN2C(=O)CCC(c2ccc(C(N)=O)cc2)=O)C1 70784,c1(C(N2CCC3CCC(C(=O)OC(C)(C)C)C32)=O)cc(S(C)(=O)=O)cc(F)c1Cl 70785,CC1(C)CC(NC(=O)C(=O)NCC2CC2)CN(C(=O)C(C)(C)S(C)(=O)=O)C1 70786,c1(C(=O)NCCOCCN(C(=O)C(C2CC2)C2CC2)C)ccc(Cl)s1 70787,C(=O)(CC(C)CNC(C1COCC(C)O1)=O)NCCc1cnc(C)[nH]1 70788,C1(C(=O)OCC(=O)NCCOC2CCOCC2)CCC(Nc2ccc(Cl)nc2)CC1 70789,C1(C2CN(C(=O)CNc3ccccn3)C2)CN(C(c2ccc(CO)s2)=O)CCO1 70790,O=C1CCc2nc(NC3CCC(NC(c4cc5n(n4)CCC5)=O)CC3)ccc21 70791,N(C1CCc2cccnc21)C(c1cc(-c2c(OC(F)F)cccc2F)ccn1)=O 70792,c1(C(N2CCC3C(NC(C4(F)CCCCCC4)=O)C3C2)=O)ccn2cncc2c1 70793,S(=O)(=O)(c1ccc(NC(c2ccc(Cl)cc2)CCO)cc1Cl)NC(C)CCCO 70794,C1(C(N2CC(CNC(c3c(C)nc(CO)o3)=O)OCC2)=O)CC2CCC(C1)C2 70795,c1(C(=O)NCC2(F)CN(C(C3C(CC)CCC3)=O)C2)cc(Br)cnc1S 70796,c1(CCC(=O)NCC(C2CCOC2)NC(=O)CC2CSC2)nc(C2CC2)no1 70797,C1(CCN(C(=O)Cc2ccc(CO)cc2)C)CCCCN1C(=O)C=CCF 70798,C(=O)(C(O)C(F)(F)F)NC(C(C)O)C(=O)NCCOCCN(C)C 70799,CCCC(C)CC(=O)NC(CNC(c1cc(C)cnc1Cl)=O)CC(C)C 70800,C1(NC(c2c(C#C)c[nH]n2)=O)CCCCCCC1NC(=O)CCCCOC 70801,N#Cc1ccccc1OCC(N1CCN(C(C2CCCC(O)C2)=O)C(CO)C1)=O 70802,c1(C(N(C2CCN(C(=O)C=NOC)C2)CC)=O)cn(C)nn1 70803,C1(C2CC2)(C(=O)NC(CC(=O)OC)C2CC2)CN(C(C2C=CCC2)=O)C1 70804,C(=O)(CC(C)(O)C(F)(F)F)N1CC(C)(NC(=O)Cc2csc(=N)[nH]2)C1 70805,c1(C(=O)NCC2OCCN(C(c3cc(CO)[nH]n3)=O)C2)ccc(Cl)c([N+](=O)[O-])c1 70806,C1(C(=O)NC2(CCNC(CN3CC(CC)C3)=O)CC2)CCN(C(C)=O)CC1 70807,c1(CNC2CC(CN=[N+]=[N-])C2)cc(O)c2ccccc2c1 70808,C1(C(=O)NCC(CC(C)C)NC(=O)C(C)(O)C(C)C)CCCCNC1=O 70809,c1(C(N2CCC(CNC(CC(C(CC)C)O)=O)CC2)=O)cnc2c(c1)ncn2C 70810,Cc1cccc2cc(C(=O)N(CC(C)(C)NC(c3occc3Br)=O)C)cnc12 70811,C=CC1(C(=O)N(CCCN(C(=O)C(C)Cc2ccncc2)C)C)CCC1 70812,c1(C(=O)OCc2c(C(=O)OC)nns2)ccc2cccnc2c1F 70813,O=C(C1=CCCCO1)NCCCOCCNC(C1COC2(CO)CC1C2)=O 70814,C1(C(=O)NC2CCOCC2C)(CC)CCN(C(c2csnn2)=O)C1 70815,CC1(C)CC(C(=O)NCC2CN(C(=O)C3CC3)CC23CC3)CCO1 70816,O(NC(=O)C(O)C1CC1)CC(=O)N(C)C.C12(CCC1)C(=O)N2 70817,C#CCCC(=O)NCCCOCCN(C(=O)C(O)CF)C 70818,C1(NC(C=C(NC(C)=O)C)=O)CC2CCC(C1)N2C(=O)Cc1ccccc1O 70819,C(=O)(C(CO)C(C)(C)C)N1C(CC(N2CCN(CCOC)CC2)=O)C2CCC1C2 70820,c1(C(N(C(C)C)CCNC(=O)CCCCc2cnn[nH]2)=O)ccnc2[nH]ncc12 70821,C1(OCC=C)CCN(C(=O)C(C2CC2)N(C(=O)Cn2cncn2)C)CC1 70822,c1(C(=O)NC(CCN(C(CCSCCCC)=O)C)C)ccc2nonc2c1 70823,N1(C(C(C)C#N)=O)C2CCC1CC(CNC(c1cc(Cl)ccc1OC(F)F)=O)C2 70824,C1(CCNC(C2CC(OC)C2)=O)CN(C(C2CCN2C2CCCC2)=O)CCO1 70825,c1(OCC)cc(F)ccc1C(N1CC2C(C1)N2C(c1cnco1)=O)=O 70826,C12(NC(c3n(CC)ncc3)=O)CCC(C(N3CCC(C)(O)C3)=O)(CC1)CC2 70827,CCCC(CCCNC(=O)COc1ccc(F)cc1)NC(C1(C)CC1C)=O 70828,c1(C2n3cc(nn3)SC2)ccc(Cl)cc1.CCC(CC)N(CC(=O)O)C(C)=O 70829,c1(C(=O)NCCN(C(C(CC#C)C)=O)CCOC)cc2c(nn1)CCCO2 70830,Cc1cc(C(=O)NC2CCCCC2NC(C2CCC(=O)O2)=O)cc(C)c1Br 70831,Cn1cc(Br)c(C(=O)NCC2(CCNC(=O)Cn3cccn3)CC2)cc1=O 70832,Cc1cc([N+](=O)[O-])c(N2CCC(C(F)(F)F)C2)cc1Br 70833,C#CC1CC2(CC2)CN1C(=O)C(C(C)CC)N(C)C(c1oc(C)cc1C)=O 70834,c1(CNC(c2ccccc2Cl)c2n(CC)nnn2)ccc(Cl)nc1 70835,c1(NC(C(=O)NCC(=C)F)=O)cc(C(F)(F)F)ccc1OC 70836,c1(NC(c2noc(C3CC3)n2)CC)cc(C(=O)C(F)(F)F)ccc1F 70837,C(=O)(C(O)CC(F)(F)F)NC1(CC(N2CCC(C(=O)OC)CC2)=O)CCC1 70838,N1(C(C(CC)O)=O)CCCN(C(=O)Cc2ccc(OC)cc2C)CC1 70839,C12(CCC(O)CC1)C(=O)NC2.C1(C(OCC)OCC)CCC(CC)CC1 70840,C1(C(=O)NCCN(C(C)C)C(C2C(C)C2C)=O)CCC(C)(C)O1 70841,C1(NC(c2cn(CC)nc2)=O)CCC(NC(=O)C(C)Sc2ccc(F)cc2)CC1 70842,N1(C(CCC#CC)=O)CCC(CCNC(=O)C(CCC)N(C)C)C(O)C1 70843,N1(C(C2(C(C)C)CCN(C(c3ccsn3)=O)C2)=O)CCC12CCSCC2 70844,C(CCCCC(=O)N1CCCC(C(C)(O)CNC(c2cc[n+]([O-])cc2)=O)C1)OC 70845,C1(C(=O)NC(C)CCNC(c2occc2F)=O)C2CCCOC12 70846,N1(S(C(C)C)(=O)=O)Cc2ccc(NC(=O)C(C)OCc3ccccc3)cc2C1 70847,C1(N(C(C(=O)OC)C)C)CCSCC1.c12noc(n1)C2SC1CCCCC1 70848,Cc1ccc(CN(c2nnc(C3CCC3)n2C)C(C)C(C)C)cc1Cl 70849,CN1CC(=O)N(CC(=O)NC2CC(NC(=O)Cc3cn(C)cn3)C2)C1=O 70850,C1(C(N2C(CNC(c3cc(CC)on3)=O)CC2)=O)CCOCC12CCC2 70851,Cc1[nH]c(=NC(=O)N2CCc3[nH][nH]c(=N)c3C2)ccc1C#N 70852,N1(C(c2c(C)n(C)nn2)=O)CC2CCC1C(CNC(c1c(O)cccc1Cl)=O)C2 70853,c1(NCCN2CCN(C(C3ON=C(C)C3)=O)C(C)C2)nc(C)nc2sc(C)c(C)c12 70854,c1(C(C(=O)NCC2N(C(c3nccc(COC)c3)=O)CC2)O)cc(Cl)cc(Cl)c1 70855,N1(C(C(=O)Nc2ccccc2)=O)CC2CCNCC12.c12ccc(cc1)[nH]c2=O 70856,C1(CC(=O)NC(CC)(C)CO)CN(C(c2c[nH][nH]c2=N)=O)CCO1 70857,C(=O)(CC1=CCCCC1)NCC(C1CCN(CC(CC)OC)CC1)(C)C 70858,Cc1cc(NC(=O)C(=O)NC2CCC2)n(C)n1.C1(n2ncc(N)c2)CCS(=O)(=O)C1 70859,c1(SCC#C)cccc(NC(C2CCCC2)=O)c1.C12CC(C)N(C1)C(=O)N2 70860,C(=O)(C(C(C)(C)C)NC(C1(Cl)CC1(F)F)=O)NCCC(C)N1CCCC1 70861,c1(-c2cn(C3C(C)CN(C(=O)C(F)C4CCC4)C3)nn2)cc(Cl)cc(Cl)c1Br 70862,C1(NC(c2cc(OC)no2)=O)CN(C(=O)CCC=C(C)C)CC1F 70863,C=Cc1cnn(C)c1CNC(=O)N(C)CC1(O)CCOCC1 70864,c1(OC)cccc(NC(c2nnnn2CCSc2cccs2)C2CC2(C)C)c1 70865,C1(NC(c2ccc(CCC)cc2)=O)CCN(C(c2cnc(N)c(O)c2)=O)CC1F 70866,C(=O)(C(CCC1CCC1)NC(=O)Cc1c[nH]ccc1=O)NCC(C(C)O)C 70867,C1(N(C)C(C2CCN(c3ncccn3)C2)=O)CC1C1CC1 70868,C1(NC(C2(CC)CN(C(C(CCCC)C)=O)C2)=O)CCCCC12CCC2 70869,C1(CNC(c2scnc2Cl)=O)CN(C(c2cn[nH]c2)=O)C2(CCOCC2)C1 70870,N1(C(C(C)(C)NC(=O)OC)=O)CCN(C(=O)C(C)c2cccs2)C(CN(C)C)C1 70871,c1(C(N2C(CNC(C(CC#C)C3CC3)=O)CC2)=O)nc(C)ccc1Br 70872,c1(C(N2CCC(NC(C(CC)CN(C)C)=O)CC2C)=O)cc(C)cc2ccoc12 70873,c1(C(=O)NC2(COC)CCN(C(C3CC3CF)=O)C2)cc(Cl)c2[nH]c(O)nc2c1 70874,c1(C(=O)NCC(CNC(C2CCN(C(CC)=O)C2)=O)OC)cc(C)n(C2CC2)c1 70875,C1(C(=O)NC(C)CCNC(c2ccnc(Cl)c2N)=O)CC(C(C)(C)C)=NO1 70876,C(C(C)(C)C(=O)OCC1CCN(C(CCC(C)(C)C2CC2)=O)CC1)NC(C)=O 70877,C(C(=O)N1CCOC(CC(N2CC(O)CC2CN(C)C)=O)C1)(C(C)C)OCC 70878,c1(CC)cccc(OCC(=O)NCCC(C)(C)NC(C2CCC(C)O2)=O)c1 70879,c1(NC(C(CC)C)=O)ccc(SCCC(N2CCC(C)CC2)=O)cc1C 70880,C(=O)(C(C(C)C)SCC)NCC1CCC(NC(C2(CC#C)CCOC2)=O)C1 70881,c1(C(=O)NCC2N(C(C(=O)NCC)=O)CC3(CC3)C2)cn2c(n1)CC(OC)CC2 70882,C(=O)(C(C)(C)CCCNC(=O)CCc1nccs1)NCCOCCN(C)C 70883,C(=O)(N=c1[nH]nc(CN(C)C)s1)N(CC)CC1CCNC1 70884,C1(C(CNC(C(C)(C)n2ccnn2)=O)(C)O)CCN(C(C2CCCCC2)=O)CC1 70885,C(CC(CNC(c1nncs1)=O)OCC)NC(C(C)OCC=C)=O 70886,CN1CC(NC(c2cc(CNC(C3CNC(=O)N3)=O)nn2C)=O)CC12CCC2 70887,CCCCC(CC)NC(N1CCCC(COc2ccccc2)C1)=O 70888,C#Cc1cc(C(N2CCC(F)C(NC(c3ccccc3)=O)C2)=O)cc(N)c1 70889,N1(C(C2(COC)CC=CC2)=O)CCC(F)(CNC(C2(COC)C=CCC2)=O)CC1 70890,c1(NC(CN(C)Cc2cccc(O)c2)=O)cccc(OCc2cccs2)c1 70891,O=C(CCC[N+](=O)[O-])N1CCOCC(CNC(C2(c3ccccn3)CC2)=O)C1 70892,c1(CC(=O)NC(CC=C)C(N2CC(C(N)=O)C3(CC3)C2)=O)ccc(C#N)cc1 70893,CC1CCC(CCC(N2CC(O)(CNC(=O)CC34CC(C3)C4)C2)=O)O1 70894,N1(C(c2c(CC)con2)=O)CCCC(C)(C(=O)NC2CCCC2O)C1 70895,CCCCC(C(=O)N(CC(C)NC(c1nn(C)nc1C(=O)OC)=O)C)C(C)C 70896,c1(C(N(C)CC2CCN(C(C(CCC)O)=O)C2)=O)cnn2c1N(C)CC2 70897,c1(C(=O)NCCN(CCC)C(c2c[nH]nc2CC)=O)c(C)csc1Cl 70898,C1(CNC(c2cnc(O)o2)=O)CC2(CCC2)CN1C(c1ncoc1C1CC1)=O 70899,C(=O)(CC(C)(C)C(=O)N1CC2CC(NC(c3cc(Br)cn3C)=O)CC2C1)OC 70900,N1(C(Cc2ccn(C)n2)=O)CC(NC(C2(c3cncs3)CC2)=O)CC(F)C1 70901,CC#CCCC(=O)NC1CCC(CCC(N2CCN(CCCO)CC2)=O)C1 70902,c1(C(N(CCN(C(=O)C(F)(F)c2cscn2)C)C)=O)ncc(C(C)(C)C)o1 70903,C1(Cc2cn(C(C)(C)C)nn2)CC(C(=O)NCc2ccc(Cl)cc2)C1(C)C 70904,CCC(CC)C(F)C(=O)NCC1(CNC(=O)C(CC)OC)CCCCC1 70905,C(CC1CC1)(C(=O)NCC=CCNC(c1cc(Br)co1)=O)OC 70906,C=C(C)C(CC(=O)NC(C)(CNC(c1cc(O)ccc1O)=O)C1CC1)OCC 70907,C1(CCC#C)CCCN(C(=O)C(C)(CO)NC(=O)C(C)N(C)C(C)=O)C1 70908,C1(C(=O)NC(C(C)C)(C)CNC(=O)CN2CCC(=O)CC2)CCCCC1(F)F 70909,C1(C(=O)NC(C(=O)NC(C(=O)NCC)CC)CCC2CC2)C2CCC(C2)C1C 70910,c1(-c2cccc(NC(=O)C(=O)NC3CC4OC(=O)CC34)c2)nc([N+](=O)[O-])n[nH]1 70911,N1(CCn2c(C)csc2=O)CCCN(C(c2c(Cl)nn(C)c2Cl)=O)CC1 70912,c1(C(=O)CCC2CCN(c3cn(C)nc3)C2)cc(Br)cnc1S 70913,CC(C)CC(O)CN=c1cc[nH]cc1S(=O)(=O)N1CCc2c(C)cccc2C1 70914,c1(OCC)ccc(NC(c2nnnn2C2CC(F)(F)C2)(CC)C2CC2)c(F)c1 70915,c1(CN(C)C(C2CN(c3ccncc3)C2)=O)ccnn1C 70916,CCC(C)C(O)C(=O)NC1(CO)CN(C(=O)C(C)(O)C2CC2)C1 70917,CN1C(=O)OCC1C(N1CCC(F)(C(=O)NC(C2CC2)C2CC2)C1)=O 70918,N#Cc1cnn(CCO)c1NC(=O)NC1(c2ccc(OC(F)(F)F)cc2)CC(O)C1 70919,Cc1cnn(C(C)C(=O)NC(c2cccnc2)C(=O)NCC2(N(C)C)CC2)c1 70920,N1(C(CC=C(C)C)=O)CCN(C(c2ccc(C(F)F)o2)=O)CC1c1cn[nH]c1 70921,C(CO)(CCCCNC(c1ccc(C2CC2)cc1)=O)NC(C=CC(C)(C)SC)=O 70922,c1(N(c2nccc(C(C)C)n2)C(C2CCCNCC2)=O)ncc2ccccc2n1 70923,Cc1cc(C(N2CCC23CN(C(=O)CCC(C)(F)F)C3)=O)c(O)c(C)c1 70924,N1(CC(=O)N)CCCC(CCC2CCC(NC(CC(=C)C)=O)C2)C1=O.C(=O)OCC 70925,C(C(C(=O)N1CC2CC2N1)NC(=O)OC)c1cccc(-c2c(OC)cccc2)c1 70926,c1(OC)cc(C)cnc1C(=O)NCC1C2CN(C(c3cc(Cl)cn3C)=O)CC12 70927,c1(CCC(=O)NCCN(CC(C)(C)C)C(CC2(CC)CCC2)=O)ccc(=N)[nH]c1 70928,Cc1cc(C)c2nc(N3CC(C(N)=O)(CNC(=O)C(C)N(C)C)C3)sc2c1 70929,Cc1ncc(CC(=O)NCCCN(C(=O)CCCN(C)C)CC2CCCC2)s1 70930,c1(C(N(C2CCC(F)C2)CCOCOC)=O)cnc[nH]c1=N 70931,CCC(C(=O)NC1CC(C)N(C(=O)Cc2cc(C)n(C)n2)C1)C(C)(C)CC 70932,c1(C(=O)O)ccnc(N2CCCC2)n1.C12CCCC1C(=O)N(C(=O)CCCF)C2 70933,c1(N2CCCC(CC)C2)nc2cccc(F)c2c(=NCC2CCN(C)C2)[nH]1 70934,C1(CNC(C(C#C)(C)C)=O)CN(C(=O)Cc2cc(C)on2)CCCO1 70935,C1(C)(C(=O)NCC(CNC(C2CCCC2(C)C)=O)OC)CCCN(C)C1 70936,N=c1nc(O)c(C(N2CCCCC(NC(c3ccc(C(N)=O)nc3)=O)C2)=O)c[nH]1 70937,c1(CN(C(COCCNC(c2ccc(CC)[nH]2)=O)=O)C)ccc(C)cc1 70938,c1(COC)ccccc1NC(C1CC1C(=O)Nc1cc(CS(C)(=O)=O)on1)=O 70939,c1(CN2C(C(=O)NC3CC(C)(C)CCO3)CC(OC)C2)cc2ccccc2o1 70940,O=C(C(F)(F)CO)N1CCC(OC2CN(C(=O)Cn3ccc(C4CC4)n3)C2)CC1 70941,CCCC(C)(C)C(=O)NCC(CNC(C1(c2ccc(OC)cc2)CCC1)=O)OC 70942,c1(OCCOC)cncc(C(=O)NC2CC(CNC(=O)C(Br)=C(C)C)C2)c1 70943,C(CC(=O)N(CC(C)CO)C)(C(C)CC)NC(C(CCC)N(C)C)=O 70944,C1(C(N2CCC(CC=C)C2)=O)COCCN1C(=O)Cc1cc[nH]n1 70945,C(C(=O)NCC1CC12CCCCC2)(C(C)(C)C)NC(C1N(C)C(=O)CC1)=O 70946,c1(C(=O)NC2CN(C(CC(C(C)C)C)=O)CC2(C)C)c2c(nn1C)CCCC2 70947,c1(C(N2CC(NC(C3(C)CC4CC4C3)=O)C(C)(C)C2)=O)ccc2oc(=N)[nH]c2c1 70948,c1(C(N2CCC(C)(CNC(=O)CC3CCC(=O)N3)C2)=O)cc2c(Cl)cccn2n1 70949,N1(C(C(C)OCC(C)C)=O)CC(C2CCCN(C(c3cc(C(C)C)[nH]n3)=O)C2)C1 70950,c1(C(=O)NCc2cc(C(=O)NC(COC)(C)CO)n(C)n2)ncc(F)cc1N 70951,CC1CC(CNC(=O)C=CC2CCCCCC2)CCN1C(c1nn(C)cc1Cl)=O 70952,C1(C(N2CC(F)(C(N(c3ccc(OCC)cc3)C)=O)C2)=O)CC(=O)OC1(C)C 70953,c1(CSCCCC)ccccc1-c1ccc(CNc2nc[nH]n2)s1 70954,CC1CN(C(c2cc(Cl)ccn2)=O)CC(C)C1NC(c1cc(N)nc(Cl)c1)=O 70955,C(=O)(C#Cc1ccc(F)cc1F)N1C(C(=O)OCc2ccccc2)CCCC1 70956,Cc1ccc(CNC(=O)C(CC2CC2)NC(c2cnn(C)c2)=O)s1 70957,C1(C(N2CCSCC2)=O)CCCCCN1C(=O)C=CC1CCCCCC1 70958,C(=O)(C(O)CC(C)(C)C)NC(CNC(c1c(C)cc(OC)nc1)=O)CO 70959,c1(C(=O)NC(CCNC(CC2(OC)CCCCC2)=O)C)ncn2cc(Cl)ccc12 70960,c1(C(=O)Nc2snc(Cl)c2C(F)F)ccc(Br)c(CO)c1 70961,N(C)(C(=NCC1CCCO1)NCC1CC2CC1C2)CCCCN(C)C 70962,C(CCCCCNC(c1sccc1CO)=O)N(C(C(C)=C(C)C)=O)C 70963,c1(C(N2CCN(C(C=CCOC)=O)C(C)CC2)=O)ccc2c(c1)C(C)CO2 70964,c1(C(=O)NC2CC(NC(=O)CC3CC3(Cl)Cl)C2)ccccc1S(=O)(=O)C(F)F 70965,CC1SCCCC1C(=O)NC1CCC(CNC(=O)CSC(C)(C)C)CC1 70966,N1(C(CC(=C)Br)=O)CCC2(CCN(C(c3cccc(C(C)C)n3)=O)C2)C1 70967,c1(C(=O)NC2(CO)CCN(C(COCCN(C)C)=O)C2)cc(N(C)C)nc(Cl)c1 70968,n1(CC(=O)NCC(CC(C)C)NC(CSCCCC)=O)cc(F)ccc1=O 70969,C1(C2CCC2)(NC(C(C2CCN(C(c3csc(F)c3)=O)C2)C)=O)CC1 70970,c1(C(N2CCN(CCN(C3CN(C(C)=O)C3)CC)CC2)=O)cnn2cccc2c1 70971,c1(NC(CCN(CCC)C)=O)cccc(CNC(=O)C(c2cccc(C)c2)O)c1 70972,CCCCC(C(=O)NC(C)Cn1ccnc1)NC(=O)COC(C)C 70973,C1(C(=O)NCC2CCC(NC(c3cc(CC)[nH]n3)=O)C2)COc2ccccc2C1 70974,C1(C#CC(=O)NC(C)(C)CCNC(c2cnc(C(C)(C)C)o2)=O)(CC)COC1 70975,C(=O)(C1CCOc2ccccc21)N1C2CN(C(c3nnc4ccccn34)=O)C(C2)C1 70976,C(=O)(CCC(=O)Nc1ccc(C(C)Nc2cn(-c3ccccn3)nn2)cc1)OC 70977,C1(NC(C2N(C(CC(C(C)C)O)=O)CCC(C)C2)=O)CCC2CCCC1O2 70978,N1(C(CC=C)=O)CCC(NC(=O)CCc2ccc(C)nc2)C(CC)C1 70979,C1(CN(C(=O)CS(=O)(=O)NC)CC)CCN(C(C2OCCOC2C)=O)CC1 70980,N1(C(=O)NC2CN(CCOC)C(=O)C2)Cc2ccc(F)cc2CC1C 70981,N1(C(C(=O)NC(C)C)=O)C2CCC1C(NC(C1(c3ccc(Cl)cc3)CCC1)=O)C2 70982,Cc1ccccc1C=CC(=O)NC1(CCCNC(=O)CC2CC3(CCC3)C2)CC1 70983,c1(OC)cc(CNCC(c2nccs2)C)cc(I)c1O 70984,CCCC(C)(CC)C(=O)NCC(C)(C1CC1)NC(C1CCCC1C)=O 70985,N1(C(CSCCC)=O)CC(NC(=O)CC2CCCC23CC3)CC1(C)C 70986,c1(N(C(c2cc(C)c(O)nn2)=O)CC)ccc([N+](=O)[O-])cc1C#N.C12CCN(CC1)C2 70987,C1(C(=O)NCC2(O)CC(CNC(=O)CC3CCCC3)C2)Cc2nccn2C1 70988,C1(C(N(CCNC(COCCCC#C)=O)CCOC)=O)CCC(C2CC2)C1 70989,C1(CNC(CN(C)CC)=O)CCC12CCN(C(=O)Cn1ccc(=O)cc1C)CC2 70990,N1(C(c2nc(C)oc2C)=O)CCc2sccc2C1CNC(C12CCC1C2)=O 70991,C(C(CCC)C(=O)NCc1nc(N(C)C)no1)NC(C=C(CC)CC)=O 70992,Cn1ncc(Cl)c1C(=O)NC12CC(NC(C3CCCN(C(=O)C4CC4)C3)=O)(C1)C2 70993,c1(CC)ccc([N+](=O)[O-])cc1C(=O)NCC=CCNC(c1cnc(C)s1)=O 70994,C(CC(C)(C)C)(C(=O)NC1CCCCC1N=[N+]=[N-])NC(CCC#C)=O 70995,C1(CC(N2CCC(N(C(C3CC(N(C)C)C3)=O)CCO)C2)=O)CC2(CCC2)C1 70996,Cc1cc(C(N2C(C(=O)N(CC(C)C(C)C)C)CC2C)=O)cn1C 70997,Cc1cc(Cl)ncc1CC(N1CCN(C(=O)CC(C)C2CC2)C(C)C1)=O 70998,C(=O)(C(C(C)(C)C)N(C)C(=O)OC(C)(C)C)N(C)CC1CCN(C(C)=O)C1 70999,c1(OC)cc(CCNC(=O)C(C)Oc2cc(C)cc(C)c2)cc(C)c1 71000,c1(C(N(CCC(=O)OC)CCOC)=O)ccc(C2CCCNC2)cc1 71001,C1(N(C)C)CCC(N(C(=O)CC(O)C2CCCC2)C)CC1 71002,CC(C)C(C(=O)NC1CC(C(N2CC3CC2(C(F)F)C3)=O)C1)C(C)C 71003,C1(N(C(C2CCC(C)CC2)=O)C)CN(C(=O)C(C)N2CCC2)CCC1O 71004,Cc1cc(F)c(C(=O)NCC2CCN(C(c3cnc(O)c(Cl)c3)=O)C2)c(Br)c1 71005,CC(CC(=O)NCC(C(=O)N1CCc2ccsc2C1)C(C)(C)C)CC(C)(C)C 71006,c1(COC)cccc(CC(=O)NC2CCC(CNC(C3CC=CCC3C)=O)C2)c1 71007,C1(CNC(CN(CCC)C)=O)C(C)CCCN1C(=O)C(C)N(CC(F)(F)F)C 71008,C1(CN(C(=O)C=CCOCC(F)(F)F)C)COCCN1C(C1CC2CC2C1)=O 71009,C(=O)(C(C)CC(F)(F)F)N(CCNC(C(C=C)(C)O)=O)CCOCCOC 71010,C1(C(N2CCC(=CCNC(C3CC(Cl)(Cl)C3)=O)CC2)=O)CCC2(CCC2)CO1 71011,c1(CC)coc2c1CN(C(=O)Cc1cccc(O)c1)C2.C12(C)CC(O)CN1C2=O 71012,c1(C(N2CCC(OC)(CO)C2)C(=O)Nc2ccccc2)cc2cccc(Cl)c2o1 71013,CCC(CC)=CC(=O)NCC1CCN1C(=O)CCOCCOCCCO 71014,C(=O)(C1COc2ccccc21)NC1CCC(NC(=O)Cc2cccc(Cl)c2)CC1 71015,N1(C(CC2C(OC)CC2)=O)CCCC1C1(NC(c2sccc2C(C)=O)=O)CC1 71016,c1(C(N2CCC(C(C)NC(C(C)OCC#C)=O)CC2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 71017,CC(C)CC(=O)N1CCC(CN(C(=O)CC2C(CN)C2(F)F)C)C1 71018,c1(C(=O)NCC(C)CC(N2CCC(C)(C#N)C2)=O)cccc2[nH]ccc12 71019,N1(C(C)=O)CCN(C(=NCCc2cccc(F)c2)NCC(C)(C)C)CC1(C)C 71020,CC1(C(N2CCC(OCC(N)=O)C2)=O)CCCN(C(=O)CN2CC3CC3C2)C1 71021,N1(C(c2on(C)c(=O)c2)=O)CC(CNC(=O)C(F)(F)C(F)F)OC(C(F)(F)F)C1 71022,C1(NC(Cc2c(C)nsc2)=O)C=CCN(C(=O)C(c2cccc(F)c2)(C)C)C1 71023,C12(NC(CN(CC(=O)NC(C)C)C)=O)CCOCC1CN(C(=O)CS(C)(=O)=O)C2 71024,C1(NC(c2c(CC)con2)=O)CCC(C)N(C(c2cnn(C)c2Br)=O)C1 71025,N1(C(=O)CCn2cnnn2)CCCC(F)(CNC(C2(CO)CCC2)=O)C1 71026,C#CCC(CC(F)F)C(=O)N1CC(NC(=O)CC2(OC)CCOCC2)CC1C 71027,c1(SC)cc(C)c(C(N2CC(NC(c3cc(CCO)on3)=O)C(C)C2)=O)o1 71028,C1(C(N2C(C)(CC(=O)NC(C#C)(C)C3CCC3)CC2)=O)CCCC(=O)C1 71029,CS(=O)(=O)c1ccc(NC(C2COCCN2Cc2cccc3c2CCC3)=O)cc1 71030,N1(C(c2c(C)scc2)=O)CCCCCC1C(=O)N(C)Cc1nnnn1C 71031,C#CC1(C(N2CCC(O)C2)=O)CCN(C(c2cncc(C#C)c2)=O)C1 71032,N1(C(C2C(c3n(CC)ccn3)OCC2)=O)CCOCC1CCNC(=O)CN(C)C 71033,c1(NCCOC)ncc(S(=O)(=O)N2CCC(NCC3CC(SC)C3)CC2)cc1Cl 71034,C1(NC(C(C)SCc2ccccc2)=O)CC12CCN(C(C1CCC(C)CC1)=O)C2 71035,c1(CCC(=O)NCCCN(C(=O)CC2CSCCO2)CC)nnc(C2CC2)o1 71036,c1(C(=O)Nc2ccc(C(=O)OC)c(Cl)c2)cc2ccoc2cn1.C123CC1CN(C2)C3 71037,CC1(CNC(C2CC(NC(=O)Cn3cccc3)CCO2)=O)NC(=O)NC1=O 71038,c1(C(=O)NCC23N(C(C=CSC)=O)CCC2CCC3)ccc2c(c1)CCCO2 71039,c1(C(=O)NCCCOCCNC(=O)CC2CCCO2)cc(=O)n2ccccc2n1 71040,N1(C(C(C)C2CCOC2)=O)CCOC(CNC(C2(C3CC3)CCC2)=O)C1 71041,c1(CC(=O)NC2CN(C(C3(CC#C)CCCCO3)=O)CC2F)ccc(C)c(F)c1 71042,c1(OC)ccc(Cl)c(C(=O)NC2CC(F)(CNC(=O)C(F)(F)C3CC3)C2)c1N 71043,c1(C(=O)NCC(CN(C)C(C2(F)CCOC2)=O)O)nc2cccnc2s1 71044,Cc1cc(OCC(N2CC3CCOC3(CNC(=O)CO)C2)=O)cc(C)c1Cl 71045,c1(CN2CCC(O)(C(=O)NCC(C)OC)CC2)c[nH]c2ncc(Br)nc12 71046,CCC(C)C(C(=O)N1CCCN(Cc2ccc(C(F)(F)F)cc2)CC1)OC 71047,c1(C(N(CCC(C)NC(C2CC2c2ccsc2)=O)C)=O)ccc2c(c1)OCCO2 71048,CCC(C)(COC)C(=O)NC1CC(NC(=O)C(C)N(C)C)C(O)C1 71049,c1(C(=O)NC(C2(O)CN(C(=O)CCNc3ccccn3)C2)C)ccoc1Br 71050,c1(OC)cc(C(=O)N(CCN(C)C)Cc2ccc(C)cc2)c(Br)cc1O 71051,Cc1nn(C)c2c(NCCN3CCCOCC3)nc(=NCC(C(C)C)N(C)C)[nH]c12 71052,N1(C(N2CCC(c3nc(C)on3)C2)=O)CCC(O)CC1CO.n12nc(C)cc1C2 71053,Cc1c(C=CC(N2CCC(CCNC(C3CC4C=CC3O4)=O)CC2)=O)cnn1C 71054,Cn1cc(C(=O)NCCCC(c2ccccc2)NC(C2(F)CC=CC2)=O)nn1 71055,N1(C(C2(CCC=C)CCCC2)=O)CCN(C(=O)Cc2cnn(C)c2)CC1CCC 71056,c1(C(=O)NC2CC(N(C(Cn3c(C)ccc3C)=O)C)C2)ccc(P(C)(C)=O)nc1 71057,c1(C(=O)NCC(CCNC(C(C)CS(C)=O)=O)(C)C)scc2c1OCCO2 71058,CC(CNC(=O)CNc1cccnc1)C(=O)N1CC(O)(C(F)F)C1 71059,c12ccc(nc1O)C(=O)NCC(CC)NC2=O.C#CCC(O)C(=O)OCC 71060,N(C(=NCc1ccn(C)c1)NCc1cccc(OCC(F)(F)F)n1)C(C)C1CC1 71061,N1(C(C(C)OCC)=O)CCC2(CC1)CCN(C(c1cnncc1O)=O)C2 71062,c1(OC)nc(C(=O)NC2(CNC(c3csc(C(N)=O)n3)=O)CCOC2)cc(O)n1 71063,N1(C(CNC(=O)NC)=O)CCCC(C)(C(=O)NC(c2ccncc2)C)C1 71064,c1(CNC(C(C)OC)=O)ccc(CCNC(=O)CC(C)(C)c2cccs2)cc1 71065,Cc1nc2ccccc2n1CC(N1CC(C(C)NC(c2ccnnc2)=O)C1)=O 71066,CCC(C)(CNC(=O)C(F)C(C)C)C(=O)N1CC(O)(C(C)C)C1 71067,C1(C(=O)NCc2c(COC)ocn2)CN(C(C2(C(N)=O)CCC2)=O)CCO1 71068,CCCCC(CNC(c1cnccc1N)=O)NC(c1cc(C(F)(F)F)c[nH]1)=O 71069,N1(C(C2(F)CCCN(C(c3n(C=C)ncc3)=O)C2)=O)CCc2cc(F)ccc21 71070,CCCCC(C)N=c1cc(NCCCCCOCC2CC2)nc(C)[nH]1 71071,c1(OCC)ccc(C(N2CCC(CNC(c3cncc(C)c3)=O)C2)=O)nn1 71072,C1(CC)CN(C(=O)C(=O)NC2CC2)CCC1NC(=O)C(c1cnn(C)c1)O 71073,CC(C)CC(C)CNC(c1csc(-c2ccccn2)n1)=O 71074,N1(C2(C(N(C(CNC(CC=C(C)C)=O)C3CC3)C)=O)CC2)CCCCC1=O 71075,C1(NC(C(CCOC)NC(C(CC)O)=O)=O)CC2C=CC1CC2 71076,CS(=O)(=O)C(C(=O)N(CCNC(=O)CC1CC1)CC)C1CCOCC1.C(CN(C)C)S 71077,c1(C(=O)NCC(C)(CO)NC(C2C(CCOC)C2)=O)cccc(-c2cnco2)c1 71078,c1(CN(C(C(OC)OC)=O)CCCNC(C2(C)CSC2)=O)ccccc1 71079,C(=O)(CCCC(C)(F)F)NC1(CCOC)CCN(C(=O)C(C)C2(O)CCC2)C1 71080,c1(OCC(N2C3CC(NC(COCC)=O)C2CC3)=O)ccc(C#N)cc1Cl 71081,C1(C(N2CCC(C#CC)C2)=O)CCC2CCC1N2C(=O)C(=Cc1ccccc1)C 71082,C(=O)(C1=CCC2CCC1N2C(c1coc(C(F)F)c1)=O)NCCCOCCCC 71083,C(=O)(C#CC1CCCO1)N(CCC)CCNC(C1(NC(=O)C2CC2)CCCCC1)=O 71084,N1(C(C=C(C)CNC(C2CC(=O)N(C)C2)=O)=O)CCc2cc(F)ccc21 71085,C#CCC(C(=O)Nc1cccc(SC)c1)NC(c1snc(C)c1N)=O 71086,N1(C(C(C(C)C)SC)=O)CCCN(C(C2(c3ccc(Cl)c(Cl)c3)CC2)=O)CC1 71087,C#CC(C)(C)C(=O)N1CCC(C(=O)NCCC(=O)NC(C)C)O1 71088,c1(OC)cc(C(=O)NC2CCC2C2CC2)nn1-c1ccc(Cl)cc1 71089,c1(C(N2CCC(C)(C(=O)NCC(C)NC(c3cnco3)=O)C2)=O)ccc(Cl)cc1 71090,C1(NC(c2c(CC)nc[nH]2)=O)CCC(N(C)C(C2CCN(C3CCC3)C2)=O)CC1 71091,Cc1nn(C)c2sc(C(=O)NCCC(P(C)(C)=O)c3nn[nH]n3)cc12.N12CC(C1)C2 71092,c1(C(=O)NC2CN(C(c3cc(OC)c(F)cc3)=O)C2)cn(C)cc(Br)c1=O 71093,C1(N(C(=O)CC2CCOC2)CCC)CCN(C(=O)Cc2cc[nH]n2)CC1 71094,C1(C(N2CC(C)C(CCNC(c3cnc[nH]c3=N)=O)C2)=O)CCCC(C)(C)O1 71095,C1(C(=O)NCC(CSC)OC)CNC(=O)CN1C(c1cc(=O)n(C)cn1)=O 71096,Cc1sc(O)nc1C(N1CC(F)(C(=O)NC2CCOCC2F)C1)=O 71097,N1(C(c2ccc(-c3ccccc3)s2)C(=O)NCCCCCCl)CCC(O)CC1(C)C.CS 71098,c1(CC(C(=O)OC)OCCC(c2cccc(N(C)C)c2)=O)ccc(F)cc1 71099,CCC(C)C(C(=O)N1CCC(NC(=O)C(Cl)=CCl)C(O)C1)NC(=O)OC 71100,C1(OC)CN(C(=O)C=Cc2ccccc2)C(C)(CNC(c2nncs2)=O)C1 71101,c1(C(=O)NC2CCc3n(C)cnc3C2)ccc2c(=N)[nH]cnc2c1 71102,C1(CC(=O)NC(C)CN2CCN(C(c3c[nH]nc3F)=O)CC2)CCCCC1(C)C 71103,C#Cc1ccnc(C(=O)NC(CC=C)C(=O)N2CCOCC2CCO)c1 71104,C1(NC(c2c(NC)nc(C)cc2)=O)CC2CC(C1)N(C(=O)Cc1scnc1C)C2 71105,C1(C(=O)NCC(=O)OCC=C)CCCC(NC(C2(N(C)C)CC2)=O)CC1 71106,c1(C(=O)NC(CC)(C)CNC(c2cccc(CF)c2)=O)cc2cc(C)[nH]c2cc1Cl 71107,C(CC(C)CCNC(=O)CCC1CCCO1)NC(C1N(C(C(C)C)=O)CCC1)=O 71108,C1(NC(C2(CC=C)CC2)=O)CCC(O)CN(C(C2CC23CCSCC3)=O)C1 71109,CCC(CC)C(C(=O)NCCCNC(C1(c2ccccc2F)CCC1)=O)OC 71110,C(C(C(F)(F)F)N(c1ccnc(NCCN2CCCC(O)C2)n1)C)OC 71111,N1(C(C(COC)C)=O)CCOC2(CCCN(C(c3ccc(CN(C)C)[nH]3)=O)C2)C1 71112,C(=O)(C(C)(C)CC(C)(C)C)N(CC(C)CNC(=O)C1=CCCC1)C 71113,C1(CC)CCC(C(=O)CNC(N2CCC2C(C)C)=O)C1 71114,Cc1cc(C)c(C(N2CCCC(NC(C3(C)CC3(F)F)=O)CC2)=O)c(S)n1 71115,C=CCCC(C(=O)OCCCN=[N+]=[N-])NC(=O)CN(C1CCOC1=O)C(C)=O 71116,C1(C(=O)Nc2ncccc2C2CC2)CC(F)CN(C(=O)CC2CCSC2)C1 71117,C=CCC(C(=O)N1CCC1(C)COC)NC(C1CC(C)C1)=O 71118,c1(OC)ccc2c(=O)c(C(=O)OCC34CNCC3CCO4)c[nH]c2c1 71119,C1(NC(C2(NC(C(CCSC)O)=O)CC(F)(F)C2)=O)CCn2nccc2C1 71120,c1(SC)ncc(C(N2CCC(F)(C(N3CCOC(C(F)(F)F)C3)=O)C2)=O)cn1 71121,C1(NC(c2nc(C)nc(O)c2)=O)C(CNC(=O)C(C)(C)CO)CCC12CCC2 71122,CCCC(C)(C)C(=O)N1CC(NC(C2CC2c2cc(Cl)cc(Cl)c2)=O)CC(F)C1 71123,C12(NC(C3=C(C)CCC3)=O)CCCC1N(C(c1ccc3nncn3c1)=O)CCC2 71124,C12(C(N3CCCC(CCNC(=O)Cn4ccnn4)C3)=O)CCCC1C2(F)F 71125,c1(C(N(CC(CN(C(C(CC)F)=O)C)O)C)=O)cnc(OC2CCOCC2)cn1 71126,c1(CC(=O)NC(CN(C(c2cc(C)n(C)n2)=O)CC)C)coc2cc(C)ccc12 71127,C(=O)(CC(C)CC)NC1(C)CN(C(CN(CCC#C)C)=O)C1 71128,Cc1cc(C2CC2)ncc1C(=O)NCC1CCC(C)CN1C(c1cnccn1)=O 71129,C1(C(=O)OC)(C(N2CC3(C2)CN(C(=O)C(O)CN2CCCC2)C3)=O)CC2(CCC2)C1 71130,CC1CCN(C(C2CC23CC(O)C3)=O)CCN1C(=O)CCC1CC1(F)F 71131,N1(C(C2CCN(C(=O)NC)CC2)=O)CCC2(NC(=O)CN(C)C(=O)OC)CC2C1 71132,N1(C(c2nn(CC)nc2C)=O)CCC(C(N2CC(O)CC2C(N)=O)=O)C(C)(C)C1 71133,CC1C(NC(=O)CSC(C)(C)C)CCCN1C(=O)CN(c1ccc(Cl)nn1)C 71134,N1(C(c2ccc(SC)o2)=O)CCCC(C(C)NC(c2nn[nH]c2Cl)=O)C1 71135,N1(C(C(C)OCOC)=O)CCOC(C)C1C(=O)NCCC(O)C(F)(F)F 71136,c1(C(=O)NC(CNC(c2ccc(NC(=O)OC)cc2)=O)(C)C)nn(C)c(Cl)c1Cl 71137,CCCC(CC)CC(=O)NCC1COCCN1C(=O)CN(C)CC 71138,N1(C(CCc2ccc(C)cc2C)=O)CC2(NC(C3CC3C(F)F)=O)CCC1CC2 71139,N1(C(=O)C=C2CCC2)CCCC2C1CCCCN2C(=O)CCF 71140,C1(C2(O)CN(C(C3COC(C)C3)=O)C2)(CNC(Cn2nnc(C)n2)=O)CC1 71141,N1(C(c2cccc(OC)c2)=O)CCCN(CCCCNC(=O)C(O)C2CC2)CC1 71142,C1(NC(=O)CCN2CCCCC2)C=CCN(C(C2(c3ccc(Cl)o3)CC2)=O)C1 71143,C1(CNC(C(CC)CC)=O)CCC12CCN(C(=O)C(O)(C(F)(F)F)C1CC1)CC2 71144,C(=O)(C#CC(C)(C)CNC(=O)C(N1CCNC1=O)C)Nc1c(C)ncc(Cl)c1 71145,c1(CN2CCCC(C(=O)NCCC3N(C)CCC3)C2)csc2ccc(Cl)cc12 71146,c1(C(=O)NC(CNC(c2c(CC)noc2)=O)(C)CO)ccc(C)c2c1CCC2 71147,N1(C(C2C(C)CC(C)O2)=O)CC2CCN(C(c3ccc(=O)n(C)c3)=O)CCC2C1 71148,Cc1scc(C(N2CC(N(C(=O)CC3(C(F)(F)F)CC3)C)C(F)C2)=O)c1C 71149,Cc1ncc(C(=O)NC(C)(C)CCNC(C2CC(C3CC3)=NO2)=O)cc1N 71150,C1(C(N2C(C(=O)Nc3cccc(OC)c3)(CC)CCC2)=O)OC(C)(C)OC1(C)C 71151,CCC(C(=O)OC)C(=O)NC(C(N1CC(C)(F)C1)=O)C1CCC1 71152,N1(C(C2(Cl)C(C(C)=O)C2)=O)CCOCC(C(N2CCN(C)C(C3CC3)C2)=O)C1 71153,C(=O)(CCCCCNC(c1cc(F)c[nH]1)=O)N1C(C)CC1 71154,C(C(F)(C(=O)NCCC1CCCC1(C)C)C(C)C)NC(C1(OCC)CC1)=O 71155,c1(OC)ccncc1C(=O)NC12CC(NC(=O)C(C)(C)CC3CCOCC3)(C1)C2 71156,CC(C)CCC(O)C(=O)N(CC(C)CNC(=O)C=CC1CCCCC1)C 71157,C1(C)(C(N(CC)CC2CCC2)=O)CNC(C)(C)C1 71158,c1(NC(C)=O)cc(=NCC(c2ccccc2C)NCC(C)(C)C(N)=O)[nH]c(C)n1 71159,c12noc(C)c1C(C)N1CCC1CNC2=O.N1(CC(=O)OC)CCCCC1 71160,c1(C(N2CCN(CC(=O)N(C)C)CC2)=O)cn(C)ccc1=O.CC1C(=O)N1 71161,C1(C(=O)NC(C#C)CC)CCN(C(=O)C(C)COC(C)=O)CCO1 71162,C1(C(N2CC(F)(CNC(=O)C(CO)c3ccccc3)C2)=O)(CC)CCCC1 71163,C(=O)(C1CCOc2ccc(Cl)cc21)NC1CN(C(CC#N)=O)C2(C1)CCC2 71164,c1(C(C(=O)NCC(COC)NC(c2c[nH]nc2C(C)(C)C)=O)C)cccnc1 71165,C#CC1CCCC(CNC(C2(C)CN(C(C3CCC(C)(C)C3)=O)C2)=O)C1 71166,C12(NC(C3C(CC)C3)=O)CC1CN(C(=O)CSC(C)(C)C)C2 71167,C12(CNC(C(CC)O)=O)CCC(CC1)N2C(C1CCC(=C2CCC2)CC1)=O 71168,C=CC1(NC(C2N(C(C3CCC3OC)=O)CCC2(C)C)=O)CCOCC1 71169,CC1(C)CC(C(=O)NCC(F)Br)CCN1C(C1(c2ccsc2)CC1)=O 71170,c1(C(=O)NC(CNC(COCCCC)=O)C(C)C)ccccc1C 71171,c1(OCC(=O)NC2CC(NC(C(C(C)O)C)=O)C2)ccc(Cl)c(F)c1 71172,Cc1ccc(OCC(C)NC(C2CCN(CC3CC3)CC2)=O)c(F)c1 71173,Nc1nc(C(=O)NCC2CC(F)(CNC(=O)C(F)n3cccn3)C2)ccc1O 71174,CCCC(CC(C)C)C(=O)NC1CN(C(c2c(CC)nn(C)c2Cl)=O)CCC1F 71175,c1(N(C)C)ccnc(C(=O)NCc2cn(-c3ccccc3)nn2)c1 71176,c1(C(=O)NC(CNC(c2c(CCC)cccc2)=O)C)ccnc(F)c1N 71177,Cc1csc(C(N2CCC2(C)CC(=O)NC2(CC(C)C)CC2)=O)c1C 71178,C1(CC(=O)NCC2(C(N)=O)CN(C(C3(C#N)CC=CC3)=O)C2)CCCCC1O 71179,c1(C(=O)NCC2N(C(c3ccc(=O)oc3)=O)CCOC2)c(Cl)cc(Cl)cc1Cl 71180,c1(CC)ccc(C(=O)NC(CN(C)C)C(N2CCC(C)(CC)C2)=O)cn1 71181,C(=O)(C1COc2ccccc21)NCCN(CCC)C(C1(C)CC(F)(F)C1)=O 71182,n1(CC(N2CCC(O)(CN(C(C(C)C(F)F)=O)C)C2)=O)cnc2ccccc12 71183,C(=O)(CC1=CCCCC1)N1CC(C#C)(C(=O)Nc2[nH]ccc(=O)c2C)C1 71184,C(C(=O)NCCCN(C)C1CC1)N(CCC)C(C1CC1CC)=O 71185,CCC(C)CC(C(=O)NC1CC1)NC(=O)C=CCN(C)Cc1noc(C)n1 71186,c1(C(=O)NCC2C(OC)CCC2)ccc(CNC(=O)CNc2c[nH]c(C#N)c2)cn1 71187,N1(C(C(C)CC(C)(C)C)=O)CCC2(CCCN2C(=O)C(C2CCOCC2)O)C1 71188,CCCCCCN(CC(=O)NCC(C)(CC)NC(c1coc(SC)c1)=O)C 71189,c1(C(N)=O)ccc(Cl)nc1NC(C1CCCC1NCc1ccnc(O)c1)=O 71190,O(C1CCCc2nc(C)ncc21)C(C=Cc1ccc(C(CC)(C)C)cc1)=O 71191,C(=O)(C(O)C(F)(F)F)NCCN(CCOC)C(C1CCCOC1)=O 71192,c1(C(N2CC(CNC(C(CN(CC)CC)F)=O)(OC)C2)=O)cccc(F)c1C 71193,CC1CCc2[nH]c(C(=O)NCCCN(C(=O)CC(C)(C)O)C3CCCC3)cc2C1 71194,N1(CCNC(CCCCC)=O)CCCN(C(=O)Cn2cc(C(C)O)nn2)CC1 71195,C1(C)(CCNC(c2c(OC)ccs2)=O)CCN(C(C2(O)CCSC2)=O)C1 71196,C1(C#N)(C(N(CC=CC(=O)NC2CN(CCC)C2)C)=O)CC2CC2C1 71197,N1(C(C=NOC)=O)CCc2cc(CN3CCC(C)(N(CCO)CCO)C3)ccc21 71198,c1(C(=O)NC2C(NC(c3ccccn3)=O)CCCC2)ccc(O)nc1Cl 71199,N1(c2n(CC)c(-c3cc4n(c3)CCCC4)nn2)CC2NC(=O)C(=O)NC2C1 71200,C(C1C(C(=O)NCC2CN(C(=O)Cn3cnnc3)CCO2)C1(C)C)=C(C)C 71201,c1(C(=O)NC2CC(NC(=O)CC(F)(F)C(F)(F)F)C2)cc(Cl)cc2ccncc12 71202,c1(C(=O)NCC(CCCC)NC(c2cccc(=O)o2)=O)ccc2cncnc2c1 71203,C1(NC(c2ncc(Br)cc2O)=O)CCN(C(c2ccc[nH]2)=O)C12CC2 71204,c1(C(N(C2(F)CN(C)C2)CC)=O)cc(Br)c(C)cc1O.n1(C=O)cccc1 71205,C(C(C)(C)CC(=O)N1CC(CNC(c2[nH]c(C)nc2C)=O)C2(CC2)C1)OC 71206,c1(CC(=O)N(CCN(C(c2cc(C)n(C3CC3)n2)=O)C)C)c(F)cccc1F 71207,N1(C(C2(SC)CN(C(=O)CC3COCCO3)C2)=O)CCOCCC1C1CC1 71208,S(=O)(=O)(c1ccc(N2CC=CCC2)c(F)c1)NCC1OCC(C)C1 71209,C(=O)(C#CC1CCCOC1)N(C1CCCCN(C(C=C(C)C(F)F)=O)C1)C 71210,C1(CC(=O)N(CC#CC)C)CCCCN1C(c1cn(C)nn1)=O 71211,c1(CNC(C(CC)C)=O)ncccc1CNC(c1cc(Br)nn1C)=O 71212,C1(CCC(=O)N(CCN(C)C)C)CN(C(=O)OC(C)(C)C)CCO1 71213,C12(C(=O)N(CCNC(C3(CO)CCCO3)=O)CC3CC3)CCC(CO)(CC1)CC2 71214,CC(C)(C)C(C(=O)N1CC(C#N)(CCF)C1)NC(=O)CCc1ccccc1 71215,c1(C(=O)NC2(CO)CN(C(C3(F)CCCOC3)=O)C2)ccc2nccn2n1 71216,c1(C(=O)NCCCN(C(C)C)C(C2CCC3CC23)=O)ccc2c(c1)CCOC2 71217,CC(CCCNC(c1cccnn1)=O)NC(C1CCCC1c1nc[nH]n1)=O 71218,n1(CC)cnc(CNC(c2coc(CNC(c3nocc3C(C)C)=O)c2)=O)n1 71219,C(=O)(CC(O)CC1CC1)NC(C)CCCNC(=O)CNC(=O)OC(C)(C)C 71220,N1(CCC)CCC(C(=O)N(CC(C)O)CCNC(=O)CCC2CCCO2)CC1 71221,N1(C(C2C(CNC(CNC(CCC)=O)=O)OCC2)=O)CCOCC(C(C)C)C1 71222,c1(C(N2C3CN(C(C(C#C)(C)C)=O)CC2CC3)=O)ccc2c(n1)CCC(C)C2 71223,N1(C(CCc2n(C)ccn2)=O)CCCCN(C(c2cccc(OCC#N)c2)=O)C1 71224,N1(C(c2cscc2Br)C(=O)NCCCSCC)CCCC2(CCNC2=O)C1 71225,Cc1nnc2n1CCC(NC(=O)NC(C)(C)C(C(=O)O)c1ccccc1)C2 71226,c1(N2CC(NC(c3ccc(CO)nc3)=O)(CO)C2)ncc(O)cn1 71227,C1(OCCNC(=O)Cc2cn[nH]c2)CCN(C(C2COCOC2)=O)C1 71228,N1(C(CCN(C(C)=O)C)=O)CC2(CC(NC(=O)C(C)(C)C(C)O)CO2)C1 71229,C(=O)(C(C)Cc1cnc[nH]1)O.C1(C(C2CCCC2)C)CN(C(=O)CN(C)CC)C1 71230,C12(OCOCC)CCC(n3cc(-c4cnc(OC)s4)nn3)C1C2 71231,C(=O)(C(O)C(F)(F)F)N1C2C(C(N(C(CCO)C(F)F)C)=O)C(C2)C1 71232,CCCCC(CNC(C1CC(N(C(=O)CC2(OC)CCC2)C)C1)=O)CC 71233,N1(Cc2c(OC)cccc2C)CCC2(CCN(C(=O)Cn3cc(Cl)cn3)C2)C1 71234,CCCC(CCC)CC(=O)NCC1CN(C(c2ccsc2CC)=O)CC12CCC2 71235,c1(C(=O)NCCN(C(C=CC)=O)CC)cccc(F)c1Br 71236,CN1N=C(C(=O)NC2COCCC2NC(C2COC(C)(C)CO2)=O)CCC1=O 71237,N1(C(c2[nH]nc(OC)c2Cl)=O)CC2(CCC2NC(c2ccc(CO)cc2)=O)C1 71238,C1(C(=O)NCC(C)NC(c2c(OC)cnc(Cl)c2)=O)CCOCC12CCC2 71239,c1(C(=O)NC2CCCN(C(c3c(Cl)ccc(C)c3)=O)C2C)cc2cccnn2n1 71240,N1(C(C2CC(SC)C2)=O)CC2OCCN(C(=O)CCC(=O)C3CCCC3)C2C1 71241,C1(C(N2CC(C#N)C(NC(c3csc(Br)n3)=O)C2)=O)CCc2ccccc2C1 71242,C1(O)(CNC(c2cc(C)nn2C(C)(C)C)=O)CCCN(C(C2(Br)CCC2)=O)C1 71243,c1(C(N2C3C(NC(C4CS(=O)(=O)C4)=O)CC(CC3)C2)=O)cccc2c1CCCC2 71244,C(=O)(C(C)(C)CCCNC(=O)CCC1CC1C)N1CCCC(CCC)C1 71245,CC1CCCN(C(=O)C(=O)NCCC2CC(NC(=O)C(C)(C)C3CCC3)C2)C1 71246,CCC(C)(C(=O)N1CCC(C)(NC(c2ccc(SC(F)(F)F)nc2)=O)C1)C(N)=O 71247,Cc1cc(C(=O)NC2C3CCC2N(C(C2(C(=O)N(C)C)CC2)=O)C3)ncc1CO 71248,c1(CC(N2CCC(F)(C(=O)NCC(C)(C)N(C)C)C2)=O)cc(Cl)cc(Cl)c1 71249,c1(C(N2CC(CN3CCN(C(C4C(=C)C4)=O)CC3)C2)=O)nccn2c(C)nnc12 71250,CCC(O)C(C)(C)C(=O)N1CCC(CN(C(=O)CCc2cnn(C)c2)CC)CC1 71251,c1(OC)ccc(CC(=O)NC2CCC(N(C(=O)Cn3cc(Cl)cn3)C)C2)cn1 71252,Cn1c(C(N2CCC(C(C)(C)C)(CNC(=O)CC(C)(C)O)C2)=O)cc2occc12 71253,N(C1CCCn2ncnc21)C(C(CNC(c1ccc(CC)[nH]1)=O)OC)=O 71254,Cc1ccc(Br)c(CN(C=O)CC(C)(C)C(O)c2ccccc2)c1 71255,N1(C(C(C)Cn2cccn2)=O)CCN(C(c2ccc(Cl)cc2I)=O)CC12CC2 71256,c1(C(c2n(CCSCC(C)C)nnn2)NCCSC)ccnc2c(Br)cccc12 71257,c1(C(=O)NCC2C(CNC(CN)=O)C2)cc(OC)ccc1OC.C(C)CC.S 71258,c1(C(=O)NCC2(C)N(C(c3cc(OC)nn3C)=O)CCC2)cc(O)nc(O)c1 71259,C1(CC(=O)NCCNC(Cc2[nH]c(=N)sc2)=O)CCCC12NC(=O)NC2=O 71260,C(C)(C)(C(C)CC(=O)N1CCC(CCOC)CC1)NC(C=C(CC)CC)=O 71261,C=CCC(C(=O)N1CCCC1COC)NC(=O)CC=C(C)C 71262,N1(Cc2cncc(C)n2)CCC(O)CC1C(=O)NC1CC1c1ccc(Br)cc1 71263,C1(CC#C)(C(=O)NC(CNC(c2cnn(C(C)C)c2F)=O)CO)CC=CCC1 71264,c1(C(=O)NC2CN(C(c3c(C)nsc3C)=O)CC2C(F)F)cccn2ccnc12 71265,N1(C(c2c(C)nsc2)=O)CCC2CN(C(=O)C(O)CC3CCCCC3)CC12 71266,C1(NC(COc2ccc(C)cc2C)=O)CN(C(C2CC23CCC3)=O)CC2(CC2)C1 71267,Cc1cc(C(N2CCSCC2C(=O)N=c2cc[nH][nH]2)=O)ccc1F 71268,C1(CC=C)(NC(c2ccsn2)=O)CCN(C(=O)COCc2ncc(C)o2)C1 71269,C1(C2CCN(C(C3(CC4CC4)CCC3)=O)C2)(NC(C=C(CC)C)=O)CC1 71270,N1(C(CN(C2CCCC2)C)=O)CC(O)(C(F)C(=O)NCc2cc(C(F)F)n[nH]2)C1 71271,CCCCCC(CC)C(=O)N1CC(C)CC1C(=O)NOCC1CCCCC1 71272,c1(C(C)=O)c[nH]c(C(=O)N(C)CCN(C)C)c1C.N12CCC(C1)OCC2=O 71273,C(=O)(C1CSc2ccccc21)N(C)CCNC(=O)COC(F)F 71274,C1(C(=O)NC(CNC(CN2CC(C)C2)=O)(C)C2CC2)CC(c2ccccn2)=NO1 71275,C#CC1(C(=O)NC2CCS(=O)CC2)CCN(C(=O)C(F)n2ccnc2)C1 71276,N1(c2n(CCC=C)c(-c3cnsn3)nn2)CCC2(CCOCC2)C1 71277,Cc1ccc(C(=O)NC2CCCC2NC(c2scnc2C2CC2)=O)o1 71278,C1(NC(CCCC=C)=O)CCCOC12CCN(C(=O)CC(C)=C=C)CC2 71279,c1(C(N2CC(C3OCCN(C(c4c(C)nns4)=O)C3)C2)=O)cc(Cl)cc(Cl)n1 71280,N1(C(C2(N(C(c3cnn(C(C)C)n3)=O)C)CC2)=O)CC(C)C(C)C1C 71281,c1(-c2c(C)ccc(CO)c2)cnc2[nH]cc(C(=O)Nc3ccnn3CCO)c2c1 71282,CCC(C)C(O)C(=O)N1CCCC1C(C)NC(=O)C=CC=Cc1ccccc1 71283,C1(NC(CC=CC=C)=O)CCN(CCNC(=O)CNC=O)CC1 71284,Cc1ccc(C(=O)NCC2C3CN(C(c4c(C)csc4Cl)=O)CC23)c(O)n1 71285,C12(C(N(C3CN(C(C4(O)CCC4)=O)CC34CC4)C)=O)CCC(C)(CC1)CO2 71286,c1(C(=O)NC2C(CNC(c3cc(SC)c(N)cc3)=O)CC2)cnc2[nH]cncc1-2 71287,C1(CN(C=O)CC(c2cc(C)c(F)cc2)O)CCS(=O)(=O)C1(C)C 71288,Cc1cc2cc(C(=O)NC3CC4(C3)CC4C(=O)NC3CCC3)oc2cc1C 71289,C(=O)(C#CC1(CC)COC1)N1C(CCNC(C(C=C)(C)CC)=O)CSCC1 71290,c1(OC(C)=O)ccc(C=CC(=O)NC2CC2NC(=O)COC2CCCC2)cc1 71291,C1(CC)(NC(=O)CSS(C)(=O)=O)CCCN(C(c2cncc(OC)c2)=O)C1 71292,C(c1ccncc1)=CC(=O)NCC(C(=O)NC(c1nc[nH]n1)CC)N(C)C 71293,N1(CCNC(C2(CCCC)CC2)=O)CCCN(C(=O)CC2CC2C(F)(F)F)CC1 71294,c1(COC)nc(C)ncc1C(=O)NCC1CCC1NC(c1ccc(CF)cc1)=O 71295,CC(C)(C(=O)NCC1CCN(C(C2(c3cccnc3)CCC2)=O)C1)C1CCCC1 71296,c1(N2CCC(CCNC(C3CC(CCC)OCC3)=O)C2)cc(C)nc(Cl)n1 71297,c1(C(c2n(C3CC(F)(F)C3)nnn2)NC2CC2C(F)(F)F)cccc2c[nH]nc12 71298,c1(C(N(C(C)C)CCNC(c2cscn2)=O)=O)nnsc1-c1ccccc1 71299,N1(C(c2occ(S(C)(=O)=O)c2)=O)CC2CCCN(C(c3n[nH]c(=N)s3)=O)C2C1 71300,c1(CCC)cccc(C(=O)NCCC2CCCCN2C(=O)C(C)SC)c1 71301,CCCC(C)(O)C(=O)N1CCC(C)(CC(=O)NCC2(O)CCN(C)C2)C1 71302,N1(C(CNC(=O)OCC)=O)CC=CC1CNC(C1CCN(c2ncccn2)C1)=O 71303,C1(C(=O)NC2C(C)CN(C(=O)CCc3cncc(F)c3)C2)CCC2C(C1)C2(F)F 71304,CC(C)CC(O)C(C)C(=O)N1CC(F)(F)CC1C(=O)NC1C=CCCC1 71305,C1(C(N2CCC(OCCNC(=O)CSC3CC3)C2)=O)C(C(F)(F)F)C1[N+](=O)[O-] 71306,N1(C(c2cc3ncc(-c4c(C)cco4)cc3[nH]2)=O)CCc2c(Br)cccc2C1 71307,c1(CC)c(C(N2CC3C(CNC(c4n[nH]c(CC)c4Cl)=O)C3C2)=O)csc1C 71308,c1(C(=O)NC2CC(CNC(C3N(C)C(=O)CC3)=O)C2)cccc2c1nc(O)n2C 71309,C1(CC(=O)NC2(CN(C(=O)CP(C)(C)=O)C)CC2)CCC12CCC2 71310,CCCCCCCC(C)CN=c1[nH]c(=NCC2CCOC2)[nH]c2cc[nH]c12 71311,C12CC(C)N(C1)Cc1[nH]nc(n1)C(=O)OC(=O)C[SH]2CC(=O)OC.C(C)(C)OC 71312,c1(CC(=O)NC(CC)C(=O)N(CC(C)C(=O)OC)C)ccc(C)nc1 71313,c1(CC)ncnc(N2CCSCC2CCNC(C2CCCN2C(C)C)=O)c1F 71314,Nc1c(O)ccc(Cl)c1C(=O)NCC1CCCN(C(=O)C=CC2CCC2)C1 71315,C1(C)(C(=O)NCCN(CCOC)C(c2ccc[n+]([O-])c2)=O)CNC(=O)C1 71316,C(=O)(C(F)(F)C(F)(F)F)N1CCC(COC)(CNC(c2ccc(C)nn2)=O)C1 71317,Brc1ccc(C2CCN(CCCCc3nccs3)CC2)nc1 71318,O=S(=O)(c1ccc(Br)c(Cl)c1)Nc1cc(-c2ccc(CO)nc2)ccn1 71319,c1(C(N2C(CNC(C(c3ccc(Cl)s3)C)=O)CCCC2)=O)cnc2c(c1)CCC2 71320,c1(C(=O)NC2CN(C(C3(COC)CC3)=O)CC(O)C2)cnc2cc(C)nn2c1C 71321,C1(NC(Cc2c(C)nn(C)c2)=O)CC2CCC1N(C(c1nnc(O)nc1O)=O)C2 71322,Cn1cnc2sc(C(=O)NCC3(O)CCCN(C(=O)Cn4nccn4)CC3)cc12 71323,c1(C(N2CCCC(CNC(C(C)OC)=O)C2)=O)cccc2[nH]ccc12 71324,C1(C(=O)Nc2ccc(-c3cn(CCC(=O)NC)nn3)cc2)CCCCC1(C)C 71325,C(CC(C)C)(C(=O)NCC(C)n1cncn1)ONC(=O)C1(CCCC)CC1 71326,c1(OC)ncccc1S(=O)(=O)NC1(c2cccc(C(F)(F)F)c2)CCOCC1 71327,N1(C(CCCNC(N)=O)=O)CC2CC1CCC2NC(C1C2C3CCC(C3)C12)=O 71328,Cc1cc(O)cc(=O)n1CC(=O)N(C)CC1CCN(C(C2C=CCC2)=O)C1 71329,n1(CC(=O)NCC2CN(C(Cc3cn(CC)nc3)=O)C2)sc(=O)c2ccccc12 71330,C(=O)(C(F)(F)Sc1cnn(C)c1)NCCOCCN(C(=O)Cc1ccn(C)n1)C 71331,C(CCN(C)C(C1(C)CS(=O)(=O)C1)=O)(C(C)C)NC(c1cn(CC=C)nc1)=O 71332,c1(C(=O)NCCN2CCC(NC(C(CC)C)=O)CC2)ccc(Cl)c(Cl)c1F 71333,C(=O)(C(C(C)(C)C)NC(C1CC2C(C1)C2(C)C)=O)NC1CCN(C(C)=O)CC1 71334,C1(NC(c2ccc(-n3cncn3)cc2)=O)CCCC(C(=O)Nc2ncc(F)s2)C1 71335,Cc1csc2nc(CNCCC(C)(C)c3ccccc3)cc(=O)n12 71336,Cn1c(COC(=O)CC2(c3ccccc3)CC2(C)C)cnc1Cl 71337,c1(CNC(C2(CNC(C34CCC3C4)=O)CCC2)=O)ccc(C(C)=O)c(N)c1 71338,c1(C(=O)NCC2(O)CN(C(=O)Cc3cccc(Cl)c3)C2)cccc2oc(O)nc12 71339,N#CCCC(=O)NC(CC(N)=O)c1cn(C2COCC2n2cccn2)nn1 71340,N1(C(C(C(C)C)NC(C)=O)=O)CCCC2CN(Cc3ccc(Cl)nc3)CC12 71341,C(=O)(CS(=O)CCC(F)(F)F)N1CCC(N(C(CCC2CCN(C)CC2)=O)C)C1 71342,C#CCC(C)(C(=O)N(CC(O)CCC)C)NC(=O)C1=CC(C)(C)C1 71343,C1(CNC(CC(C)C)=O)CN(C)CCN1C(=O)CCc1ccc(Br)s1 71344,C1(NC(c2cccc(OC)c2)=O)CN(C(c2cc(C)ccc2N)=O)CC2(CC2)C1 71345,c1(C(=O)NCC2C(NC(COCCC(C)C)=O)CCC2)ccc(Cl)c(Cl)c1 71346,N1(C(C(Cc2cn[nH]c2)NC(c2cncc(OC)c2)=O)=O)CCNC(=O)CC1C 71347,c1(C(N2CC(CN(C(C(C)OCCOC)=O)C)C2)=O)n[nH]c2c1CCCCC2 71348,c1(COCC)nc(C)c(C(=O)NCCC2(O)CCN(C(=O)C(C)C3CC3)C2)s1 71349,N1(C(c2cnc(Br)n2C)C(=O)Nc2c(C)cccc2)CCCN(C)C(=O)C1 71350,CC1CCSCCN1C(c1cccc(-c2nn[nH]n2)c1)=O 71351,CC(C(=O)NCCC1CN(C(=O)CCc2nncn2C)CCO1)C(F)(F)C(F)F 71352,C1(OCC)(CNC(c2sc3nccn3c2C)=O)CCCS(=O)(=O)C1 71353,C1(CNC(C2(CC(C)=O)CC2)=O)(CNc2ccncn2)CC12CCC2 71354,CC(C)CC(C(=O)NC1CC(C)OC1=O)NC(C1CNC(=O)O1)=O 71355,C(=O)(C1=CCOC1)NC(C)CC1CN(C(=O)C(C)c2cccs2)C1 71356,C1(CNC(=NCCC)NCC2CCN(S(C)(=O)=O)CC2)C2CCC(C2)C1(C)C 71357,CC(CNC(=O)CC1(N2CCCC2)CC1)(CO)NC(=O)CCC1CCC(=O)C1 71358,CC(C)(C)C1=NOC(C)(C(=O)NC2CCN(CCNC(c3ccc[nH]3)=O)CC2)C1 71359,CCCC(F)C(=O)N1CCC(CC(=O)NCC(C2CC2)N(C)C)CC1 71360,N1(C(CCc2cc(C)on2)=O)CCC2CCC(NC(=O)CCc3cnc[nH]3)C1C2 71361,N1(C(C(C(C)(C)C)=O)=O)CC2CC1CCN2C(=O)CSCC(N1CCCCC1)=O 71362,N1(C(=O)CCC(F)F)CCN(C(=O)CSc2cccc(F)c2)C(CO)C1 71363,c1(C(=O)NCC2C=CC(NC(C(CC)(C)O)=O)C2)cc(S(N)(=O)=O)ccn1 71364,C1(COC)(NC(=O)Cc2csnc2C)CN(C(C2CC(OC)(OC)C2)=O)C1 71365,C1(CNC(C(CC)F)=O)CC2(CCN(c3ncc(S(C)(=O)=O)cc3Cl)CC2)CO1 71366,C1(NC(C2CCN(C(CC)=O)C2)=O)CN(C(=O)CN2CCCCC2)CC1F 71367,Cc1c(C(=O)NCC2CC(C)N(C(c3ccoc3Cl)=O)C2)cccc1C#N 71368,C1(NC(=O)COCCOCCO)CCCC(CNC(=O)CC2CCSCC2)C1 71369,c1(C(N(C2CCCN(C(CCNC(COC)=O)=O)C2)C)=O)ccc(S(N)(=O)=O)s1 71370,c1(C(=O)NCCC2CC(NC(=O)CCn3ccnn3)C2)ccc(C(F)F)cc1O 71371,c1(NC(C2N(C(c3c(C#N)ccc(F)c3)=O)CC=C2)=O)c(O)cccc1[N+](=O)[O-] 71372,c1(NC(CC2(CNC(c3c(NC)cncc3)=O)CCC2)=O)ccc(Cl)c(O)c1 71373,c1(C(N2C(CN(C(=O)CC3CCC4CC4C3)C)CCC2)=O)cc2sccc2s1 71374,C1(NC(c2c(OCC)ccs2)=O)CC(C)CN(c2nccc(C(=O)OC)n2)C1 71375,O=C1CCCCCN1Cc1cn(CC2C=CCN2C(=O)CC2CCCO2)nn1 71376,N1(C(c2c(CC)occ2)=O)CC(OC)CC1C(N1CCC(O)(CN(C)C)C1)=O 71377,c1(COC(CN2C(Nc3nc(C)nc(O)c3)=NCC2)=O)[nH]c2ccccc2c1Cl 71378,c1(OC)cccc(OCCCC(=O)NCC(C)CC2CC(F)(F)C2)c1 71379,CCCCCC(CC)C(=O)N1CC(F)(F)CC1(C)CNC(c1ccc(CC)s1)=O 71380,N1(c2c(F)cnc(OCC)n2)C2CCC1CC(NC(c1cc(F)ccc1I)=O)C2 71381,Cc1ccc(O)c(CNC(=O)CCN(C(C2CC3CC3C2)=O)C2CC2)c1 71382,N1(C(CSCCOC)=O)CCN(C(C2CCC(C)O2)=O)C(C(C)(C)C)C1 71383,N1(C(C(CCOC)C)=O)CCCCCC(NC(c2ccnn2C)=O)C1 71384,C1(O)(C(N2CC(NC(CCC3C(C)(C)C3)=O)C(O)C2)=O)CN2CCC1CC2 71385,N1(C(C(CC(C)C)NC(C)=O)=O)C2CCC1CC(NC(C1CC3CCC1O3)=O)C2 71386,c1(C(=O)NC2CCN(CC)CC2)cc(Br)ccc1OCC1CONC1=O 71387,C1(NC(CCC(C)(C)OC)=O)CC2CCC(C1)N2C(C)C 71388,C1(OC)(CNC(=O)C(c2cccnc2)C)CCN(C(=O)CC2CCCS2(=O)=O)C1 71389,C#Cc1cn(C)nc1C(=O)NCC(CC)NC(c1ccc(N)cc1Cl)=O 71390,C1(C(=O)NC2CCN(C(C3CC(C)C3)=O)C2)CCC(C(=O)N(C)C)CC1 71391,C1(CNC(c2csnn2)=O)(CO)CCN(C(c2occc2C2CC2)=O)C1 71392,Cc1cccc2c1CCOC2C(=O)NC1CCCN(C(c2nn(C)cc2Cl)=O)C1 71393,c1(C(=O)NCCN(C(C)C)C(c2cccc(F)c2F)=O)ccc2c(c1)COCC2 71394,c1(NC(=O)CC2CCN2C(C2COCCO2)=O)cncc(CO)c1 71395,c1(C(N(C2CC(NC(=O)CP(C)(C)=O)C2)C)=O)ccc(-c2ncc[nH]2)cc1 71396,c1(C(=O)NCC(CC)NC(C2CC2(C)C)=O)cnc(-c2ccncc2)s1 71397,c1(C(=O)NC(C)CN(C)C(c2nocc2C2CC2)=O)ccc(P(C)(C)=O)o1 71398,C(C1CCN(C(=O)C2=CCCCO2)CC1)=CC(=O)NCc1cc2n(n1)CCO2 71399,CCC(O)(CNC(=O)CC(C)(C)NC(=O)C(C)(O)C1CC1)CC 71400,c1(CC)ccc(C(N2CCC(OC3CCC3)C2)=O)cc1C#N 71401,c12cccc(c1)C(=O)N2.c1(C(CC)CC)cc(CSc2ncccn2)on1 71402,N1(C(CCC(=C)Cl)=O)CCN(C(c2cc(CC)c(CCC)s2)=O)C(C)C1C 71403,N1(C(C(C)C2CC2)=O)CC2CCN(C(C34CCC(C(F)F)(CC3)C4)=O)CCC2C1 71404,c1(N(CCCNC(c2c3c(nn2C)CCC3)=O)CC)ncnc2c1c(Br)nn2C 71405,c1(N2CC(CN(C(C3C(C)C3)=O)C)C2)nc(Cl)nc2[nH]ccc12 71406,C(c1ncco1)=CC(=O)N(C1CCC(NC(=O)CSc2ccccc2)C1)C 71407,C1(C)(CNC(CS(=O)(=O)N(C)C)=O)CCCN(C(C2CCCC(C)(C)O2)=O)C1 71408,C1(C(N2CCN(C3CCN(C(c4cn[nH]c4)=O)CC3)CC2)=O)C2CS(=O)(=O)CC12 71409,C12(C(=O)NC3CC(CNC(CNC(=O)NC)=O)C3)CCCN1CC(O)C2 71410,CS(=O)CC(=O)N1CCCC1CNC(c1cc(C(C)(C)O)on1)=O 71411,C1(C(=O)NCCC2(C)CCN(C(CSCC)=O)C2)CCc2nc(C)nn2C1 71412,C(=O)(CC(CC)C(C)(C)C)NC1C(CCC)CN(C(c2cn(C(C)C)cn2)=O)C1 71413,C1(C(C(=O)NCC(C(C)C)NCC(=O)N(C)C)C)CCCC(F)(F)C1 71414,C1(CNC(C2(C(C)(F)F)CC2)=O)CCN(C(c2ccncc2O)=O)CC1 71415,C12(CN(C)C(=O)NCc3cnn(C)c3)CCCC1OCC2 71416,c1(CNC(=O)NC(C2COCCO2)C(=O)O)ccc(Br)cc1[N+](=O)[O-] 71417,n1(CC)nc(C(=O)NCC2(CNC(c3cnccc3Br)=O)CC2)ccc1=O 71418,c1(OCC(N2CCC(C)(CNC(COCCCOC)=O)C2)=O)ccc(F)c(F)c1 71419,C(=O)(CCP(C)(C)=O)NC(C(C)C)C(=O)NCCC1(C)CCCO1 71420,n1(CCCOC)nnnc1C(c1cc(C(F)F)on1)NCC1(F)CCOC1 71421,c1(CC(=O)NC(CNC(Cn2c(C(C)C)ncc2)=O)C(C)C)ccccc1Cl 71422,C1(CNC(COCC(C)C)=O)CCC2(CO1)CC(NC(=O)CSC(F)(F)F)C2 71423,C1(NC(C)=O)CN(C(c2cc(C3CC3)ccn2)=O)CCC1C(F)(F)F 71424,C1(C(=O)Nc2c(C)n(C(C)C)nc2)CCN(C(C2CCC(F)(F)C2)=O)CC1O 71425,c1(C(=O)O)ccc(CCNC2(c3ncccn3)CCOC2)cc1 71426,c1(C(=O)OCCc2ccc(C#N)cc2)ccc(S(=O)(=O)CCS(C)(=O)=O)cc1 71427,c1(OCC)cc(C(=O)NCC(c2cccc(Cl)c2)NC(=O)C2=CCSC2)ccn1 71428,Cc1cc(C(N2CCCC2(C)CNC(=O)CC2CNC(=O)C2)=O)c2[nH]cnc2c1 71429,c1(C(=O)NCC(CNC(c2c(C)ncs2)=O)(C)F)c(C)nn2ccccc12 71430,CC(C)(CS(C)(=O)=O)C(=O)N1CC(F)(CNC(C2(CF)CC2)=O)C1 71431,C=CC1CCCCN1C(C1(C)CCN(C(c2nnn(C)c2C)=O)CC1)=O 71432,Cc1noc2ncc(C(=O)NC3CC(CNC(c4cccc[n+]4[O-])=O)C3)cc12 71433,C(=O)(C(C)(C)C(O)C(C)C)N(CCC(=O)NC(CC)CC(F)(F)F)CC=C 71434,c1(OC)cc(C(N2CCSCC2C(=O)Nc2cccnc2Cl)=O)nn1C 71435,c1(C(N(CCN(C(C(C(C=C)C)C)=O)C)C)=O)ccc2c(=N)[nH]cnc2c1 71436,Cc1cc(C(=O)NCC2(C)CCCN2C(=O)CC(C)C2CCCC2)c(O)nn1 71437,CC1(C)CN(C(=O)CCCS(N)(=O)=O)CC(CNC(C2CC3(CSC3)C2)=O)O1 71438,CC1=CCC=CC1C(N1CCC(C(C)NC(C2CCC(=O)N2)=O)CC1)=O 71439,N1(C(c2nc[nH]n2)CC)CCc2cc(F)c(F)cc2C1 71440,c1(C2(C(=O)OCC)CC(NC(C3CCCC(CC)CC3)=O)C2)cc(F)ccc1F 71441,C=C1CCN(C(=O)CCN=[N+]=[N-])C(C(=O)NCCC(O)CO)C1 71442,C1(NC(=O)CC2CCCCC2)CN(C(=O)C(F)n2cccn2)C2CCCCC12 71443,C1(C(N(C)CC2(CNC(c3c(C)scc3)=O)CC2)=O)CCc2nncn2CC1 71444,c1(C(N2C(C(N3CCN(S(C)(=O)=O)CC3)=O)CC3CC32)=O)ccc(F)c(F)c1Cl 71445,N1(C(C)C)CCCC1C(=O)NC1CCCC1NC(=O)C(C)(C)c1ccnn1C 71446,N1(C(C=C(CC)CC)=O)CCCOC(CNC(=O)CCn2cc(Br)cn2)C1 71447,CC1(C)CC(=O)NCC1C(N1CCC(OCCNC(C2CC(=O)N2)=O)C1)=O 71448,N1(C(C=Cc2n(CC)ccn2)=O)CC2CCC1CN2C(C1CS(=O)(=O)CCO1)=O 71449,N1(C(CC2ON=C(CC)C2)=O)CCCCCC1C(=O)NCCc1cnc(C)[nH]1 71450,C12(NC(c3ncn(CC)c3)=O)CCCC1N(CC1CCCCO1)CC2 71451,C(=O)(CC(C(F)(F)F)NC(C1CC2CC2C1)=O)N(CCCCOC)C 71452,N1(c2ncc(CC)cn2)CCC(NC(c2[nH]nnc2C)=O)C(C)(C)C1 71453,CC1CC(N(C(=O)C(c2ccoc2)NC(=O)COCCCN=[N+]=[N-])C)CCO1 71454,N1(C(c2c(OC)cccc2Cl)=O)CC2(CCCN2C(=O)COC2CCCC2)C1 71455,c1(N(C(COC(c2[nH]c(=NC)sc2)=O)=O)C2CCC2)ccc2c(c1)CCC2 71456,C1(N2CCC(C(N3CC(=O)NCC3C(=O)O)=O)CC2)CCC(O)C(O)CC1 71457,N1(C(CCC(C)(C)C)=O)CCC2(CCC2NC(c2csc(C(F)F)c2)=O)CC1 71458,C(=O)(C1CCCc2nncn21)NC1CCCCN(C(c2c(=N)[nH]cnc2)=O)C1 71459,C12COCCN(C1)C2=O.C1(C)(NC(C=CC(=O)N(C)C)=O)CCC1 71460,n1(CC)cnc2nc(N3CCC(C)(CC)C3)nc(NCC3CC(C(F)(F)F)C3)c12 71461,N1(C(c2cncc(C)c2)=O)CCC(C)C(N(C)C(c2cn(C3CC3)cn2)=O)C1 71462,Cc1cc(=NCCCCC(C)NC(c2csc(-c3cnc[nH]3)n2)=O)[nH]cn1 71463,N1(C(C2(C)CCCC2)=O)CC(NC(C2(Cc3cnn[nH]3)CCC2)=O)C(CO)C1 71464,C1(NC(CC2C(C)(C)C2(C)C)=O)CCCN(C(c2nc(F)ccc2Cl)=O)CC1 71465,N1(C(C(C)OC2CCOC2)=O)CCC(N(C)C(C2CC=CCO2)=O)C1 71466,c1(NC(C2CC(OC)CN2C(C2CC2F)=O)=O)cc(F)cc(Br)c1F 71467,CCN=c1[nH]cc(C(=O)NC(C)(C)CNC(=O)Cc2ccc(OC)cc2F)s1 71468,c1(CNC(CC(C(C)C)O)=O)cnn2c1CN(C(=O)CCc1cccn1C)CC2 71469,C12CCC(CC1)C(c1nnnn1C)NC2CCO.C1(C(F)(F)F)(CC)CCCC1 71470,C1(C)(CC=C)CN(C(=O)CCC2CCC(NC(=O)C(C)SCC)C2)C1 71471,c1(CC)nc(C(=O)NCC2CCN(S(C)(=O)=O)C2)c(Br)s1 71472,C#CCCCCC(=O)N(C1CCN(C(=O)CC(C)n2ccnc2)CC1)CCC 71473,C1(C(N2CCC(NC(c3nc(C(C)C)sc3)=O)(CO)C2)=O)CC(C2CC2)=NO1 71474,Cc1cccc(Cl)c1C(=O)NC1CS(=O)(=O)CC1NC(C1CC2(C1)CC(C)C2)=O 71475,c1(C(=O)NCC2OCCC(NC(C3C(C)C3C)=O)C2)ccnc2c1CCC2 71476,N1(C(C(c2n(C)ccc2)=O)=O)CC2CCC2(C(=O)Nc2ccc(O)cc2Cl)C1 71477,c1(CN2CCC(C(N(CCC(=O)OC)C3CC3)=O)CC2)cc(Br)c(O)c(Br)c1 71478,Cc1ccccc1-n1nnnc1C(c1nncs1)NCCCNS(N)(=O)=O 71479,C1(CNC(C2C(C=C(C)C)C2(C)C)=O)C2CCC1CN(C(c1cc(C)[nH]n1)=O)C2 71480,N1(C(=O)CCc2cccnc2F)CCCN(C(=O)CCC2CCOCC2)CCC1 71481,c1(C(=O)NC)ccc(C(=O)NC2CC2NC(c2cccc(C)c2C)=O)cc1F 71482,[N-]=[N+]=NC1CCN(C(=O)C(CC2CCC2)NC(=O)Cc2cn[nH]c2)CC1O 71483,C(c1ccc(F)cc1F)=CC(=O)NC(C(C)NC(=O)CC(C)(C)O)CO 71484,c1(OC)ccc(C2(C(=O)NCCCN(C(=O)C=Cc3cncs3)C)CC2)cc1 71485,c1(C(N2C(CNC(CCCC=C)=O)C(C)CC2)=O)cc(Br)c2ncccc2c1 71486,C1(CC)(CC)CCN1C(C(=O)NCCOCC1CC1)c1cnn[nH]1 71487,c1(CC)nnc(=NCC2(F)CC(N(C(C3CCCC4CCCN34)=O)C3CC3)C2)[nH]c1CC 71488,c1(C(=O)NCC(C(C)C)NC(=O)C2=NOC(C(C)(C)C)C2)cccc2c1CCO2 71489,N1(C(C2(N(C(CC(COC)C)=O)C)CC2)=O)CC(=O)NCC12CC2 71490,C1(NC(CCC=C(C)C)=O)CCCCN(C(C23COC(CF)(C2)C3)=O)C1 71491,C1(COC)(NC(C2CCSC2)=O)CCN(C(=O)CCCSC)C1 71492,C1(CC(=O)NC2CC(C)(NC(C(CC#C)C3CC3)=O)C2)CCCC2(CC2)C1 71493,C(=O)(CCC(=O)N1CCN(C(=O)CCC2NC(=O)NC2=O)CC1)N(CC)CC 71494,N1(C(CCN(C(=O)CC2(COC)CC2)CC)=O)CC(=O)N(C)C(=O)C1 71495,C(c1sc2ccccc2c1Cl)=CC(=O)N(CC(O)CN=[N+]=[N-])C 71496,N1(C(CC2C(=O)NC(=O)N2)=O)CC2CCN(C(=O)CCc3cncc(F)c3)C2C1 71497,C(=O)(CCC(C)C)NC12CC(CNC(C3(CC)CCCO3)=O)(C1)C2 71498,N1(C(C=NOC)=O)CC(NC(=O)CSC(C)C)CC(C)C1 71499,C1(NC(C2(C)CCC(F)(F)CC2)=O)CN(C(=O)C(N)=O)Cc2nccn2C1 71500,Cc1cnc(N)c(C(=O)NC2CCC(C)N(C(c3coc(Br)c3)=O)C2)c1 71501,C=CC1(CC(=O)NCC2CN(C(=O)C=CCO)CCN2C)CCCCC1 71502,C1(C(N2C(CCNC(C3(C(C)(C)O)CCC3)=O)CCC2)=O)C2CCC3C(C2)CC13 71503,Cc1ccsc1C(=O)NC1CCC(NCc2nccs2)C1 71504,CC1(P(C)(C)=O)CCCN1C(c1ccc(F)c(F)c1)=O.c12cccc(c1)C2=O 71505,CC1CC(NC(c2ccn(C3CC3)n2)=O)CN(C(C23CCC(CC2)CO3)=O)C1 71506,c1(OC)cc(N2CC3CC2CN3Cc2cccc(Br)c2Cl)nc(OC)n1 71507,N#CC1(C(=O)NC(CO)C(O)C2CCCCC2)CC12CCOCC2 71508,N1(C(CSCCC(C)C)=O)CCCC(O)(CNC(=O)CCC2CCCN(C)C2)C1 71509,C1(C(=O)Nc2ccc(OC)nc2)(OC)CCN(C(=O)CC2CCCSC2)CC1 71510,CCC(CN(C)C)CC(=O)NC1CCC(CNC(C2CCN(C3CC3)C2=O)=O)C1 71511,n1(CCC)ccc(C(=O)NC(CO)C(=O)N2CCC(n3cccn3)C2)n1 71512,c1(CNC(C(C)Cn2cccn2)=O)ncc(C(=O)NCC(CO)N(C)C)cn1 71513,Cc1c[nH]c2ncnc(N3CCC(O)C(C(=O)Nc4ccc(S(C)=O)cc4)C3)c12 71514,CC(Cn1ccnc1)C(=O)NCc1cc(C(=O)NCC(O)C(N)=O)cs1 71515,C1(C(c2n(Cc3nnn(C)n3)nnn2)NCCC23CC(CO2)C3)CCOC1(C)C 71516,n1(C2CCN(C(=O)C(O)CN3CCCC3)CC2)cnc2c1CCN(C(=O)CO)C2 71517,C1(CNC(C(C)SC(F)(F)F)=O)CCN(C(C2COCCN2C)=O)CC1 71518,CCC(CC)C(=O)NCc1cccc(C(=O)NCc2ncnn2C(C)C)n1 71519,N1(C(C(CNC(c2ncccn2)=O)CC2CC2)=O)CCCC2COCC12 71520,C1(CC=C)(NC(CC=CC=C)=O)CCN(C(c2cnc(NC)cn2)=O)CC1 71521,Cc1noc(C)c1C=CC(=O)NC1CCCN(C(c2ccn(C(F)F)n2)=O)C1 71522,C1(CC(=O)OC)CCN(C(C2CCCC2CNC(C2CCC2C)=O)=O)C1 71523,c1(C(=O)NC2(CNC(C(c3ccc(N(C)C)cc3)C)=O)CC2)cc([N+](=O)[O-])n[nH]1 71524,N1(C(C(C)OCCN(C)C)=O)CC23CCCCC2(C1)CN(C(=O)C(N)=O)C3 71525,c1(CN(c2c(Br)cnc(C)n2)C2CCNCC2F)ccc(C#N)cc1I 71526,N1(C(C(CCCC)C)=O)CCCN(C(=O)Cc2cccc(C3CC3)c2)CCC1 71527,CCCC(CCC)CC(=O)N1CC2(NC(c3cc(CC)c(C)s3)=O)CCC1CC2 71528,c1(C(=O)OC)ccc(C(N2CC3C(C2)N3C(=O)C(=O)c2ccco2)=O)c(F)c1 71529,c1(C(=O)NCC2C3N(C(CN(CCC)C)=O)C(CC3)C2)c(C)ccc(Cl)c1F 71530,CSC1=C(C(=O)N(C(C)CN(C)C(C2(C#N)CC2(C)C)=O)C)CCCC1 71531,N1(C(C=C(CC)CC)=O)CCC=C(C(=O)N2CC(Cc3ccco3)C2)C1 71532,N1(CC)CCN(CC(N2CCSCC2CCNC(c2nsnc2O)=O)=O)CC1 71533,c1(C(=O)NC2CC3(C(NC(CC4(OC)CC4)=O)C3)C2)csc2nccn12 71534,C1(C(C)NC(c2nscc2N)=O)CN(C(=O)C=C2CC2)CCO1 71535,Cc1nsc2ncc(C(N3CC4CCN(C(=O)CCC5CC5C)CC4C3)=O)cc12 71536,C(C(C)(C)CC(=O)N1CC=CC(O)C1)NC(C(C)OCC1CC1)=O 71537,C(=O)(C1=NN(c2ccccc2)C(=O)CC1)NCC1N(C(C2ON=C(C)C2)=O)CC1 71538,c1(C(=O)NC(CNC(C(=O)NCCC(N)=O)=O)CO)cc(C)on1.C(C)(C)(C)S 71539,N1(C(C(C)OC)=O)CCC(C)(NC(=O)CC(C)CNC(=O)OC(C)(C)C)CC1 71540,N1(C(CCC(C)C)=O)C(CO)CCC12CCC2.C(c1cocn1)=CC=O 71541,C(=O)(C(C)(C)C1=CCN(C(=O)C(C)Oc2cc(-c3ccccc3)on2)CC1)OC 71542,C1(NC(N2CC3C(C)C3C2)=O)CCCN(CC(F)(F)F)C1=O 71543,c1(C(=O)NC2CC2C(=O)NC2(c3ccc(Cl)cc3)CC2)ccc(O)c(Cl)c1 71544,C(CC(=O)NNC(=O)C1(Cl)CCC1)C1N(C(=O)OC(C)(C)C)CCCC1 71545,Cc1nc(S)nc(C)c1CCC(=O)NC(CNC(C1CC(C#N)C1)=O)CC(C)C 71546,C(CCC(=O)NC(c1ccoc1)C)(C(C)C)NC(c1cc(OC)n[nH]1)=O 71547,c1(CC2(C(N3CCC(N(C(C4C(CC)C4)=O)CC)C3)=O)CC2)cccc(F)c1 71548,C12(C(=O)NCC(c3ccccc3)N(C(=O)Cc3ccco3)C)COCC1C2(F)F 71549,C(=O)(C(C)C(O)CC(C)C)N1CC(C(=O)NC23CCN(CC2)C3)(CC)C1 71550,C12(CNC(C3(CC)CC3)=O)CC(C(N)=O)(C1)C1(CN(C(=O)CSCC#N)C1)O2 71551,CCCCN=C(NCC1CCCCC1)N1CC(C)(C)OC2(CCOC2)C1 71552,c1(C(=O)NC(CC)CNC(C2(CO)CCCO2)=O)cc(C)cc2c1NCCC2 71553,O(NC(=O)C#CC(C)(C)CNC(c1cc(F)ccc1O)=O)CCCC=C 71554,C=Cc1cc(C(N2CC3C(NC(c4cnc(S)n4C4CC4)=O)C3C2)=O)cc(F)c1 71555,n1(CC(=O)NCCC(C)N(C(=O)Cc2ccon2)C)cnc2c(cnn2C)c1=O 71556,c1(C(=O)OC)ncc(C(=O)NCCN(C(=O)CCc2cc[nH]n2)CC(C)O)s1 71557,N1(C(c2ncccc2Br)=O)CC2CCC1CN2C(c1cccc2c1CCC2)=O 71558,c1(C(C(=O)OC(C)=O)N(C2CCC2)CC)cc(Cl)cc(Cl)c1 71559,Cc1noc(C)c1CC(=O)NC1CCC1NC(C1COC(=O)O1)=O 71560,C1(C(=O)NC(CC)(CC)CO)CCCC(NC(=O)C2=NOCC2)CC1 71561,N1(CC(C)(C)OC)CC(c2ccccc2Cl)OCC1C 71562,C(=O)(C1Cc2ccccc21)NC1CCCCN(C(Cc2cc(C)cc(F)c2)=O)C1 71563,C1(C(=O)NCC2(C)CCN(C(CCCc3ccc(C)s3)=O)C2)Cc2nccn2C1 71564,N1(c2n(CC(=C)Cl)c(CCCC)nn2)CCCC2(CC=CCO2)C1 71565,N1(C(c2c(C)ccc(F)c2N)=O)C2CCC1C(C)C(NC(=O)C1=CCCC1)C2 71566,C1(C)(NC(C(C)N(C(C2(C(C)(C)O)CCC2)=O)C2CC2)=O)CN2CCC1CC2 71567,c1(OC(C(N2CCCC(COC)C2)=O)C)ccc(CNC)cc1 71568,C(=O)(C1(C)OCCc2ccccc21)NCCN(C(c1cnn(C)c1Cl)=O)C1CC1 71569,c1(C(N2CC(CC(=O)N(CCOC)CC)C3(C2)CC3)=O)cc2cc[nH]c2cn1 71570,N1(C(c2cc(CC(C)C)on2)=O)CC(NC(=O)CC(C)n2cccn2)CC(C)C1 71571,Cc1cn(C)nc1C(=O)NCc1nc(C(=O)Nc2cncc(F)c2)c(C)o1 71572,N1(C(CN(C)C(c2cccs2)=O)=O)CCN(C(c2cc(Cl)cn2C)=O)CC(O)C1 71573,C(=O)(C(C(CC)CC)OC)NCC(CC=C)C(=O)NC1C2CCCCCC12 71574,C1(C)([SH]=CC(=O)N(C)CC2N(C(C3CCC(C)O3)=O)CCCC2)NC(=O)NC1=O 71575,N1(C(CC(CCSC)O)=O)CC2(C1)CN(C(c1nocc1C(C)C)=O)CC2CO 71576,CCCCC(O)C(C)C(=O)NCC1CN(C(c2cc(O)ccc2Cl)=O)CC1O 71577,C(CCCCN=c1[nH]c(-n2cccn2)nc(=N)[nH]1)N(S(C)(=O)=O)C 71578,CC(CO)C(=O)NCC1CC(F)(CNC=O)C1.N1(C2(C3(C)CC3)CC2)CCCC1 71579,c1(N2CCCC(NC(C(C)(C)n3cnnn3)=O)CC2)nc2ccc(F)cc2s1 71580,C1(C(C)NC(c2cnn(-c3nccs3)c2)=O)CCCN(C(=O)C(C)(C)C)C1 71581,C(=O)(C(C(C)NC(c1cncc(C)c1)=O)C(C)C)NCC(COC)OC 71582,C1(C)(C(N2C(C)CC2C(=O)NC23CC(F)(C2)C3)=O)CC(C)(C)C1 71583,C=C(C(=O)Nc1cccc(-c2noc(C)n2)c1)C(C)C 71584,c1(C(N2CC(OCCNC(C3CCC(CC)C3)=O)C2)=O)ccc(C)cc1COC 71585,C1(C2CCN(C(c3ncn(C)n3)=O)C2)(NC(c2ncn(C)c(=O)c2)=O)CC1 71586,C1(C(N2CC(OC)C2)=O)CCC2(CC2)N1C(=O)CN1CCNC1=O 71587,C1(NC(c2c(C)sc(C(C)N)n2)=O)CC1C1CCOCC1 71588,Nc1cc(C(N2CC3CC2CC3CNC(C2CCCCS2)=O)=O)cnc1N 71589,C1(C(=O)NC2CC(C)(NC(CC3CCCC(OC)C3)=O)C2)CN2CCN1CC2C 71590,N1(C(c2cc(=O)cc[nH]2)=O)CCC2(CCCN2C(C2CCCS2)=O)C1 71591,c1(NC(C2C=CC(NC(=O)CCc3ccc(F)cc3)C2)=O)ccc(Cl)cc1F 71592,C1(NC(CC=C)=O)CC(F)CN(C(=O)Cc2n[nH]c(=N)s2)C1 71593,N1(C(C2N(C)CCOC2)=O)CCN(C(=O)CCN2C(=O)CCC2=O)C(C2CC2)C1 71594,Cc1cc(C(N2CCCC2Cc2cn(CC(C)O)nn2)=O)c(Br)s1 71595,c1(C(N2CC(N(C)C(C3CC3OCC(C)(C)C)=O)C2)=O)cc(C2CC2)on1 71596,N1(C(C2N(C(COCCCCC)=O)CC(O)C2)=O)CCC(CO)C1(C)C 71597,C1(CC(=O)NC2(CC=C)CCCC2)COCCN1C(=O)CC1OCCCO1 71598,C1(O)(C(C)NC(C2(n3ccc(C4CC4)n3)CC2)=O)CN(C(=O)C(C)(O)C2CC2)C1 71599,N1(C(C2CCN(C)CC2)=O)CC2CCCC1(CNC(c1cc3cscc3s1)=O)C2 71600,N1(C(C(N2C(c3n(C)ccn3)CCC2)=O)=O)CCC(C2CCOCC2)(C(=O)O)C1 71601,N1(C(CC2(C)CN(C(c3cccc(O)n3)=O)C2)=O)CCCN(CCO)CC1 71602,CC(CC1CC1)C(=O)NCCC(=O)N(C)Cc1ccsc1 71603,C(=O)(CC(F)(F)CC(=O)Nc1cc(C(F)(F)F)cc(C2CC2)c1)OC 71604,N1(C(Cc2c(C)cco2)=O)CCN(C(c2c(C)nn(C)c2C)=O)CC1CO 71605,C1(N(C(CCCC(C)=O)=O)C)CCN(C(C2CCC(C)=C(C)C2)=O)CC12CC2 71606,C(=O)(CC(C)C(=O)N1CC2C(N(C)C(c3cnc4sccn34)=O)C2C1)OC 71607,Cc1ccc(C(N2CCC(C)C(CNC(c3ccncc3)=O)C2)=O)cc1Br 71608,Cc1cnc(CNC(C2(NC(=O)Cc3ccco3)CC2(C)C)=O)cn1 71609,C(=O)(C(C1CC1)NC(=O)Cc1cncs1)NCCOCC(=O)OC.C1CC1 71610,c1(CC(=O)NC(C(C(C)C)NC(=O)CCNC(=O)CO)C)ccc2nn[nH]c2c1 71611,C#CC1CN(C(=O)CSCCOC(C)=O)CCN1C(c1[nH]ccc1C)=O 71612,C(=O)(C(CSC)CC1CC1)N(CCCN(C(C1(O)CCSCC1)=O)CC)C 71613,Cc1ncnc(O)c1C(N1CCC(C)(CCNC(C2CC=CC2)=O)C1)=O 71614,C1(C(=O)NC2(C(=O)NCC#C)CC2)CC(C)(C)CCN1C(C1C=CCCC1)=O 71615,n1(C(C)C)ncc(C(=O)NCC(O)CNC(C2(Cl)CC2(F)F)=O)c1N 71616,c1(C(=O)NCCCNC(C(CC=C)CC)=O)ccc(N)c2ccncc12 71617,CC1CN(C(=O)C=CC2(C)COC2)C1C(=O)NCCC(C)N1CCCC1 71618,CCC1=NOC(C(=O)NC2CCC(N(C)C(c3cnnc(O)c3)=O)CC2)C1 71619,c1(NC(CCCOC)c2cccnc2)cc(Br)ccc1S(=O)(=O)NC1CCC1(C)C 71620,C1(NC(=O)NCCNC(=O)C2CC2)CN(C(=O)CC2CCCC2)C2(CCOC2)C1 71621,CCCC(CC)CCC(=O)N1CC(C)(C)CC1CC(=O)NCC1(OCC)CCC1 71622,CCCC(CCC)CC(=O)N1CCN(C(=O)CNC(=O)CC2CSCCS2)CC1 71623,N1(C(Cc2cc(C)sc2)=O)CC(NC(C2CCCCC2)=O)C(C)C1 71624,c1(C(=O)NC2C(NC(=O)CCC3CCCCO3)CCC2)ccc2c(n1)CCCC2 71625,C1(C(=O)NCC2N(C(COC3C(C)CCCC3)=O)CC=C2)CN2CCN1CC2 71626,N1(C(c2c(CC)ccs2)=O)CC2CC1CCC2NC(c1c[nH]nc1C(C)(C)C)=O 71627,C1(NC(C2C(C)(C)C2)=O)CC2CCC1CN(C(C1(C)CC3CCC1O3)=O)C2 71628,N1(C(=O)CCN(c2ccccc2)CCO)CCC2CC12COC(F)F 71629,c1(C(N2CC3CN(C(C(C)(F)C(F)(F)F)=O)CC3C2)=O)cnc2n1CCCCC2 71630,Cc1n[nH]c(C)c1C(=O)NCC(CO)NC(=O)C(C)OCc1ccncc1 71631,c1(CCCC(=O)N(CCCN(C(c2c(C)c[nH]n2)=O)C)C)ccc(O)cc1 71632,C1(CC)CC(C(=O)N(C2CCN(c3nnc(CO)s3)CC2)CC2CC2)CCO1 71633,C1(NC(=O)C=CCO)CC2CCC(C1F)N2C(=O)CCN1CCC1 71634,O=C(NNC(=O)C1CCS(=O)(=O)C1)c1cncc(OCC(F)F)c1 71635,N1(C(CC=CCC)=O)CCc2ccc(C(N3CCCC4OCCC34)=O)nc2C1 71636,c1(N2CC(CNC(C(CC)SC)=O)OCC2)nc(Cl)nc2[nH]ccc12 71637,c1(C(N2C(C)(CC(=O)N(c3c(OC)cccc3)C)CC2)=O)cc(F)ccc1O 71638,CC(C)C(N=[N+]=[N-])C(=O)NC1C=CC(C(=O)NC2(CO)CC3CCC2C3)C1 71639,CC1C(C(=O)N2CCC(C(N3CCCC(N=[N+]=[N-])C3)=O)(CO)C2)=NOC1C 71640,C1(CN(C(=O)COCC(C)(C)C)C)CCCN(C(C23CCCC2C3)=O)C1 71641,c1(OC)cc(C(=O)NC(c2ccccc2)CNC(c2cc(Cl)c[nH]2)=O)ccc1O 71642,C(=O)(CC(C)C(F)(F)F)NC1(C(N(C(C(=O)OCC)C)C)=O)CCCC1 71643,N1(C(Cc2c(C)con2)=O)CCN(C(c2csc(S)n2)=O)CCC1C 71644,N1(C(C2N(C(C)C)CCC2)=O)CCC(F)(CNC(=O)C(C)c2cccs2)CC1 71645,C1(NC(c2ccc(C(F)(F)F)o2)=O)CCC2(CCN(C(c3ccon3)=O)C2)C1 71646,C(=O)(C1=CS(=O)CCC1)NC(CNC(Cc1nnc(C)s1)=O)CO 71647,C#Cc1ccc(C(=O)N(C(C)CCNC(C23CCC(CC2)O3)=O)C)c(F)c1Cl 71648,C1(NC(c2cc(C(C)=O)on2)=O)CN(C(c2cc3n(n2)CCCO3)=O)CC1C1CC1 71649,N1(C(CC(CNC(c2cn(CC)nn2)=O)OC)=O)CCC2(CCCCC2)C1 71650,n1(CC(N2C(CCNC(CCNC(=O)NC)=O)CCC2)=O)ccc(C)cc1=O 71651,CCN=c1[nH]c(C(=O)NCC2CC(NC(c3ccc(OCCF)cc3)=O)C2)cs1 71652,C1(NC(C2CCN(CC)CC2)=O)CCN(Cc2ccc(COC)cc2)CC1F 71653,c1(CC)ccc(C(N2CCOC(C(C)(C)C)CC2)C(=O)NCCOCCC)cc1F 71654,O([Si](C)(C)C(C)(C)C)Oc1sccc1C(N1CC(C(=O)OC)C(F)C1)=O 71655,C(=O)(C1=Cc2ccccc2C1)NC(C(CC)C)C(=O)N1C2CCC1CC2 71656,Cc1cc(C(=O)NCC2CCN(C(C3C4CCC(=O)C34)=O)CC2)cc2c1CCC2 71657,N1(CCNC(N2CCC(CN)CC2)=O)C(=O)NC2(CCC2)C1=O 71658,c1(C(N2C(C3(NC(CCC(=C)Cl)=O)CC3)CCCC2)=O)cccc2nn[nH]c12 71659,c1(C(=O)NCCC(CNC(c2ccc(C)nc2O)=O)O)cccc(C=C(F)F)c1 71660,c1(C(=O)NC(C)CNC(=O)Cn2ncnn2)nccc2c(Cl)cccc12 71661,C=CCC(CNC(=O)C(CC)N(CC)CC)C(=O)NC1(O)CCC1 71662,c1(C(=O)NCCC)ccccc1NC(=O)Cn1cccc1 71663,Cc1cccc(CC(=O)NC2CN(C(C3(O)CCSC3)=O)CC2C)c1Cl 71664,C(=O)(CC1=Cc2ccccc2C1)N1CCC(NC(c2ccc(F)cn2)=O)C(F)C1 71665,C(=O)(CCC(C)(C)C#N)N1C(C(=O)NCC(C#C)OC)CCCC1 71666,c1(OC)cc(O)ccc1NC(C1CCC(CNc2sccc2Cl)C1)=O 71667,C1(CNC(=O)C(C2CCN(C(=O)C3CC3)C2)F)Cc2ccccc2C1 71668,C1(C)(C(N(CCCN(C(C2CCN(C)C2=O)=O)C)C)=O)CCS(=O)(=O)CC1 71669,N1(c2nnc(C(C)C)n2CC2(C)CCCO2)CCN(C)C(=O)C1(C)C 71670,C(=O)(CS(N)(=O)=O)NC(C)CN(C)C(c1ncnn1C1CCOCC1)=O 71671,N1(C(C2CN(C)C2)=O)CCC2CCC12CNC(c1ccoc1Br)=O 71672,N1(C(C(C)O)=O)CC2COCCC2(NC(C2(c3ccccc3Br)CC2)=O)C1 71673,C(=O)(C1=NN(C2CC2)C(=O)CC1)NCCCN(C(C1CC1C)=O)CC 71674,c1(C(CNC(C2(C(=O)OC)CC2)=O)N(C(=O)C(Cl)=CCl)C)ccccc1 71675,CC1CCC=C1C(=O)N(C(C)C(=O)NC1CCC12CCCC2)C 71676,N1(C(CNC(CC)=O)=O)CCC(C(=O)NCC2(C)CC3CC3C2)C(C)(C)C1 71677,C1(NC(=NCCCC)NCC(=O)NCC2CCCO2)CCc2cnn(C(C)C)c2C1 71678,N1(C(C2CC(NC(C(CCOC)OC)=O)C(O)C2)=O)CCOC2(CC2)C1 71679,c1(C(C(=O)NC2CCCC(NC(C(CC)(C)C)=O)C2)O)ccc(F)c(Cl)c1F 71680,CON(C(=O)CC1CN(C(C2CC2CC(C)C)=O)CCO1)C1CCC1 71681,C(CCC(=O)NCC1(C(C)(C)O)CN(C(=O)C(CN(C)C)N(C)C)C1)SC 71682,c1(C(C)C)cc(NC(=O)C(=O)NCC2NCCC2C)ns1 71683,N1(C(C(CC)CCOC)=O)CCC2(CC1)CCN(C(c1ccc([N+](=O)[O-])[nH]1)=O)C2 71684,C#Cc1ccnc(C(=O)N(CCC)CCNC(=O)CCn2ccnc2)c1 71685,C1(NC(C(CCC)C)=O)CCCC2CN(C(C3(CO)CCC3)=O)CC12 71686,C(C(=O)N=c1cc(C)n(CCO)[nH]1)CC1CCN(C(c2ccc(C)cc2F)=O)C1 71687,C(=O)(C(C)NC(=O)NC(C)COC)NCCOCC#C 71688,Cc1cc(NC(C2CC(F)(CO)C2)=O)n(-c2ccc(F)cc2)n1 71689,N1(C(C(C)Cc2ccccc2)=O)CC(NC(=O)CC(C)C2CCCC2)CC(O)C1 71690,CN1CCC(C(=O)N(C)CC2CCCN(C(=O)CC3CCCSC3)C2)CC1 71691,CC(C)CC(C)CC(=O)NC1CC(F)(CNC(c2ccnc(C(F)(F)F)c2)=O)C1 71692,c1(C(=O)NC(C)C(C)NC(=O)C=C2CCOCC2)ccc(-c2csnn2)cc1 71693,C1(C)(C(N(CCCC(=O)NC)C)=O)CC(O)CN1C(C1CCN(C)CC1)=O 71694,c1(C(=O)NCC23OCC(NC(COCCCC)=O)(C2)C3)cc(N)ccc1[N+](=O)[O-] 71695,c1(C(N(C2CCN(c3nnc(CC)o3)CC2F)CCC)=O)cc(C)c(C)nc1O 71696,c1(C(=O)NCC=C)cc(F)ncc1NC(c1ncccc1C(F)F)=O 71697,CC1CCCn2c(CC(N3CC(CCNC(=O)CCc4ccoc4)C3)=O)cnc21 71698,N1(C(C(CO)NC(C2CCCCC2)=O)=O)CCC2CCC(C1)N2 71699,c1(OC)ccc(F)cc1C(C1=CCCCC1)NCc1ccccc1N1CCCC1 71700,C(C(C)(C)CC(=O)N1CCCC1C1(C(=O)NOC(C)(C)C)CC1)OC 71701,c1(C(=O)NC(CNC(c2ccc(COC)o2)=O)(C)CO)ccncc1OC 71702,Cc1cc(C(=O)NC2CC3CCC2CC3NC(=O)C(O)CC2CC2)cc(C)c1N 71703,c1(C(C(=O)NCCCOCC2CCCN2C(=O)CC2CC2)O)ccc(Cl)nc1 71704,N1(C(C(C=C)(C)CC)=O)CCN(C(c2ccsn2)=O)CC2(CC2)C1 71705,C1(COC)CN(C(=O)Cc2ncoc2C)CCN1C(=O)C1=CCCCC1 71706,c1(-c2n(CC(C)(C)CO)nc(Cc3ccccc3)n2)nc2n(c1Cl)CCCC2 71707,c1(OC(C)C(=O)NCC(C)(C)CN(C)C)cccnc1 71708,c1(NCC)cccc(C(=O)N(CCC(C)NC(c2snnc2C)=O)C)c1 71709,C1(C(=O)NCc2ccn(CC)n2)CC(C)(C)CN1C(=O)Cc1cncs1 71710,c1(C(=O)NC(CNC(c2cc(C)no2)=O)CO)oc2ccccc2c1CS(C)=O 71711,S1(=O)(=O)c2ccc(cc2)OC2CCCN12.c1(C(N)=O)cn(CC(F)(F)F)nn1 71712,C1(NC(c2occ(C)c2)=O)CCC2(CCN(C(=O)Cc3nc(C)sc3C)CC2)C1 71713,c1(C(C)CC(=O)NC2CC(F)(CNC(=O)Cn3ncnn3)C2)cncc(F)c1 71714,C(=O)(C(C)(C)C(F)(F)F)NC1CC(C)N(C(=O)CC2OCCCO2)CC1 71715,C1(C(N2C(C(=O)NCCC3(O)CCC3)(CC)CCC2)=O)CC2C(C1)C2(F)F 71716,C1(CNC(CO)CO)C2(CCC2)C12CCC2 71717,CCCCCC(C)(C)C(=O)N1CCOC(CNC(=O)CC(C)N(C)C)C1 71718,c1(NC(=O)Nc2cccc(C3CCC(=O)N3)c2)cc(Cl)n2nccc2n1 71719,C1(NC(CC(COC)C)=O)C2CC3CN(C(C4CCC(C(=O)OCC)C4)=O)C1C3C2 71720,C1(C(=O)NCC(=C)C(F)(F)F)CN(C(c2ccn(C(F)F)n2)=O)CCC1O 71721,C(C(C)(C)OCC1CC1)SCC(=O)OC(C)(C)C.C1C(=O)NCCO1 71722,Cc1cc(O)c(C(N2CC(F)CC2C(=O)Nc2cnncc2Cl)=O)cc1Br 71723,c1(OCC)ccc(S(=O)(=O)N(C2CCCCCC2O)C)cc1C(=O)OC 71724,c1(C(C(N2CC(NC(COCC=C)=O)C(CC3CC3)C2)=O)O)ccc(Cl)c(F)c1 71725,N(C1CCCc2c[nH]nc21)C(CC(CNC(c1cc(CC)nn1C)=O)O)=O 71726,c1(C(C)=O)cc(=NCC23CC(CNC(=O)C(C)C(C)C)(CO2)C3)[nH]cc1[N+](=O)[O-] 71727,C1(CC(=O)NCC2(OC)CCN(C(c3ccc(F)cn3)=O)C2)CC(O)C12CCC2 71728,N1(C2CCN(C(C(C)(C)N3CCCC3)=O)C2)CCN(C(=O)Cc2cccs2)CC1 71729,c1(C(=O)NCCC2N(C(CSCCOC)=O)CCC2)ccc2nc[nH]c2c1 71730,N1(C(c2cc(C(C)(C)C)n[nH]2)=O)CCC(CNC(=O)Cc2cnccc2Cl)CC1 71731,N1(C(C(CC(C)C)ONC(=O)CC2CC3C=CC2C3)=O)CC2(CCOC(=O)N2)C1 71732,c1(CC(N2CC(C(C)NC(c3cccc(=O)o3)=O)OCC2)=O)ccc(O)c(F)c1 71733,CC1(C)CCCC1(N)C(=O)NCc1cn(C2C=CCCC2)nn1 71734,N1(C(c2n(CCC)ncc2)=O)CCCC2CCN(C(c3cnsn3)=O)CC12 71735,CCCCC(C)C(C(=O)NCCCOCC1CC1)N1CCC(OCC(F)F)C1 71736,c1(C(N(C)CC2N(S(CCC)(=O)=O)CCOC2)=O)cc(C)ccc1C 71737,O=C1CC(CC(N2CCCC(C(N3CCN(c4nccs4)CC3)=O)C2)=O)C(=O)N1 71738,N1(C(C(C=CC)O)=O)CC=C(CC(=O)NC(CCC)c2nn[nH]n2)CC1 71739,CN1CC(NC(c2c[nH][nH]c2=N)=O)C(O)C1.C1(=O)C(CC2CC2)CN1C 71740,C(=O)(CCS(=O)(=O)N1CCC(NC(C2CCS(=O)(=O)CC2)=O)C1)OC 71741,c1(NC(C2N(C(c3ccc(OC)cc3)=O)CC=C2)=O)cccc2cc(C)cnc12 71742,C1(NC(CC(=O)N(C)C)=O)CCCC12CCN(C(=O)C(C)(C)c1nccs1)CC2 71743,c1(C(N2CCN(C(C(C)NC(=O)OC)=O)C(C)C2)=O)n[nH]c2c1CS(=O)(=O)CC2 71744,Cc1cncc(C(=O)NC2CCCC(CN(C)C(c3nc(C)n(C)n3)=O)C2)c1 71745,C1(NC(c2cc(C)cc(F)c2)=O)CN(C(=O)COCC2(F)CC2)CCC1(C)C 71746,c1(C(=O)NC(CN(C(C(CC)(C)F)=O)C)C)ccc2c(c1)nc(C)n2C1CC1 71747,C(=O)(C(C(C)CC)N(C)C)NC1C=CC(C(=O)NC2CC(=C)C2)C1 71748,Cc1cc(C=CC(=O)NCC2CC3(C2)CN(C(=O)C(C)CO)C3)ccc1F 71749,N1(C(C2CN(C)C(=O)C2)=O)CC(CN(C(=O)COCC2CCCC2)C)C2(CC2)C1 71750,N1(C(C(=O)NCC(CCOC)NC(c2cc(F)c[nH]2)=O)C)CCN(C)CC1 71751,c1(C(N2CC(F)(CNC(C3CCC(C)C3)=O)C2)=O)ccnc(N2CCCC2)n1 71752,C1(CNC(CC(C)(F)F)=O)CCCN(C(C2(C)CCCS2)=O)CC1 71753,C1(CCNC(C(c2cccs2)NC(CCC=C(C)C)=O)=O)COC(C)(C)C1 71754,C(=O)(C=CS(F)(F)(F)(F)F)NCC1CN(C(C2C3CCCOC23)=O)CC(C)(C)O1 71755,N1(C(C(C)C)=O)CCN(C(C)C(=O)NC(C)CCN(C)C)CC1 71756,C(=O)(C1=CCC2CCC1N2C(c1occc1CC)=O)N1CC(C#C)C1 71757,C(c1ccc(C(F)(F)F)cc1)=CC(=O)NC1C=CCN(C(C(OC)OC)=O)C1 71758,CCC(CC)(CCNC(C1C2(CC2)C12CC2)=O)NC(=O)C(C)OC1CCOC1 71759,c1(CCC(=O)NCCCC(C)(C)NC(C2C(C)C2C)=O)ccc(C#N)cc1F 71760,C=CCC(C)(C(=O)N(C(C)CCNC(C1(O)CCCC1)=O)C)N(C)C 71761,C1(C(C(C)(C)C)=O)CC12CCCCC2.c12cn(nn1)CCOCN1CC(C1)OC2=O 71762,c1(C(=O)NCC23CC2CN(C(c2cc(Cl)no2)=O)C3)cc2c(O)ccc(F)c2[nH]1 71763,C1(C(=O)NCCNC(C2(c3ccc(Br)nc3)CCC2)=O)CCC([N+](=O)[O-])CC1 71764,O(NC(=O)CCOCCCNC(=O)C(F)CC1CCOC1)CCN(C)C 71765,n1(CCC(N2CC3C(NC(CSCC)=O)CC(C3)C2)=O)cc(C#N)c(O)nc1=O 71766,c1(C2(C(N3CCC(CNC(C4CNC(=O)N4)=O)C3)=O)CCCC2)ccc(Cl)cc1 71767,C(=O)(C(C)(C)C(C)NC(=O)C(C)OCOC)NC1(CCC=C)CC1 71768,C(C(F)(F)C(=O)N(CCNC(C1CCCC(CC(F)(F)F)C1)=O)C1CC1)OC 71769,N1(C(COCCCOC)=O)C(C(=O)NCC(c2ccsc2)O)CC2CCCCC12 71770,Cn1c(C(=O)NCC2CCCCC2NC(C2CSCCS2)=O)cc2ccccc12 71771,N1(C(c2cc(SC)ncc2)=O)CC2CN(S(=O)(=O)Cc3cccc(Cl)c3)CC12 71772,N1(C(C(CC=CCC)C)=O)CCC2CCCC12C(=O)NC(c1nc[nH]n1)C 71773,CCC(C)C(C(=O)NC1CCC(NC(c2ccccc2NCCO)=O)CC1)OC 71774,C=CCCCCCCCCC(=O)NCCCCCCNC(=O)CCCC(=O)NCC 71775,N1(C(C(CC)NC(C)=O)=O)CCC2(CC(NC(=O)C=Cc3cnccn3)CO2)C1 71776,C(=O)(C#CC(C)(C)C)NCC1OCCN(C(c2ccn(C)c2C2CCC2)=O)C1 71777,CC1CCCN(C(=O)C(C)N(C(c2cncn(C)c2=O)=O)C2CC2)CC1 71778,C=CCC(C)(C)CCNC(c1cnn(CCNC(c2cncc(C)c2)=O)c1)=O 71779,c1(OC)nc(Cl)c(C(=O)NCCC(C(C)C)NC(c2cn(C(C)(C)C)nn2)=O)s1 71780,CCCCC(CC)C(=O)NCCN(C(c1nc(Cl)sc1C)=O)C(C)C 71781,C1(CNC(C(CCC=C)(F)F)=O)CCC2(CCN(C(=O)C(C)(C)CO)CC2)CO1 71782,N1(C(C2C(C)C2)=O)CCC(C(C)NC(C23CCN(CC2)C3)=O)CC1 71783,C1(CNC(c2c(C(=O)OC)csc2)=O)CN(C(=O)C(=O)NC2CC2)CCC1C 71784,N1(C(C2C(C=C)CC2)=O)CC(NC(c2cc(OC)ccn2)=O)CC12CCCCC2 71785,c1(NC(N2CCC(C3OCC3(F)F)C2)=O)cccnc1F 71786,C1(CNC(COCCC)=O)CCCN(C(=O)CC2CCCS(=O)(=O)C2)CC1 71787,C(=O)(NOCCC1CCSC1)C1(NC(=O)COCC(F)F)CC1 71788,CCCCCCCOC(=O)C(Cc1ccccc1)C1CC1 71789,C1(CNC(CCCC#CC)=O)CN(C(c2coc(Br)n2)=O)CCC1(F)F 71790,CC(C)CN=C(NCc1nc(CS(C)(=O)=O)n[nH]1)NCC1CCOCC1(C)C 71791,C1(NC(c2c(OC)oc(C)n2)=O)CCC(O)CN(C(=O)C(C)CC(C)C)C1 71792,C(=O)(C1=CC2(CCOC2)C1)N1CCC(NC(C(C(C)C)OC)=O)CC(C)(C)C1 71793,N1(C(C23CC(OC)C2C3)=O)CC2CC(NC(c3ccc(C(F)(F)F)nc3)=O)C1C2 71794,c1(N2CCC(Oc3cccc(NC(C)=O)c3)C2)c(F)cc(F)c(N)c1[N+](=O)[O-] 71795,CC1CCC(CNC(=O)CCc2ccncc2)N(C(c2ccc(Cl)cn2)=O)C1 71796,C(=O)(CC1OCc2cc(Cl)ccc21)NC1CC(C)(NC(c2ccc(C)cc2)=O)C1 71797,c1(NC(CCC=CCC)(C)c2nnnn2C2COC2)cc(F)c(F)cc1OC 71798,c1(C(=O)OCC)cnc(N2CC(C(C)NC(=O)Cc3ccc(O)cn3)C2)cn1 71799,c1(C(=O)NCC(CN(C(C2C(C=C)C2)=O)C)C)cc(S(C)(=O)=O)c(C)o1 71800,C1(C(=O)NCCCN(C2CCCC2)C(C2CC(N(C)C)C2)=O)CC2CCC2C1 71801,C1(C(=O)NC2CC(NC(c3ccc(C(F)(F)F)[nH]3)=O)C2)Cc2ccccc2C1 71802,O(N=C1CCCCCC1)CC(=O)NCC1CCCN(C(Cc2nc(C)sc2)=O)C1 71803,C=CCCC(C)N=c1[nH]c(=NCC(CCC)OCC)[nH]c2c1CCCCC2 71804,CC(C)C(CCN(C)C(C1CC(C)OC1C)=O)NC(=O)CCN1CCOCC1 71805,C(CC(C)C(=O)N1CC2(NC(=O)CC(C)n3cccn3)CC1C2)=CCC 71806,CC(CCCc1ccccc1)C(=O)Nc1cc(CC(=O)O)ccn1 71807,CCC(C)C(C(=O)N1CCC(C(N)=O)C1)N(C)C(C12CC1CNC2=O)=O 71808,Cc1cc(=NCc2cc(Br)cs2)[nH]c(=NCc2cccc([N+](=O)[O-])c2)[nH]1 71809,N1(C(c2ccc(C)cn2)=O)CC(C)(C)C(NC(=O)CN(C)C(=O)C2CC2)C(C)(C)C1 71810,CC(C)C(C)CNC(=O)C(c1cn(C)nn1)NC(c1cn(C(C)C)cn1)=O 71811,OC1CC2CC(N=c3nc(N4CCNC(=O)CC4)c4c([nH]3)CCS4)CC12 71812,Cc1ccc(C=CC(=O)NCCCN(C)C(c2cocc2Br)=O)cn1 71813,c1(C(N2CC(O)(C(C)NC(c3c(C)cc(CC)o3)=O)C2)=O)c(C)ccc(F)c1N 71814,Cc1ccc(CNC(c2[nH]ccc2CNC(c2cc(=N)[nH][nH]2)=O)=O)nc1C 71815,c1(C(=O)NC2CC3CN(C(C(C)OC)=O)CC32)oc2c(c1C)C(=O)CCC2 71816,C(=O)(C(CC(F)F)NC(c1ccncc1O)=O)NCCC1CN(C)C(=O)C1 71817,c1(C(=O)NCC2N(C(CCCCN(C)C)=O)CC(F)C2)cnc(O)c2ccsc12 71818,C(=O)(C(CC1CCCC1)NC(=O)CCc1nccn1C)NC(C=C)CO 71819,c1(C(N2CCN(C(CN(C(=O)OCC)C)=O)CC2)=O)cn2c(n1)CCC2 71820,C1(C(N(CCN(C)C)CC)=O)C2CCCC2CN1C(=O)NC1CCCO1 71821,c1(OC)ccnc(C(=O)NCC2C3CN(C(c4ncc(C(F)F)s4)=O)CC23)c1O 71822,N1(C(CC(CC)(F)F)=O)CCC2CCN(C(c3cnc4sccn34)=O)C2C1 71823,c1(CCNC(c2cc(C)n(C)n2)=O)ccc2c(c1)COCC2 71824,CC(C)C(C#N)C(=O)N1CCC(CCNC(=O)C(C)N2CCC2)CC1 71825,Cc1ncc(C(N2CC3C(NC(C45CC(F)(C4)C5)=O)C3C2)=O)cc1N 71826,C(F)(F)(C(F)(F)F)c1cc(C(=O)NCCN(C(C2(C)CC2(F)Cl)=O)CC)no1 71827,CC1CCC2(CO1)CN(C(C1CCC1CNC(c1cn(C)nn1)=O)=O)C2 71828,C1(CC(=O)N(CC(C)C)CC(=O)NCc2nc[nH]n2)CCC(C)(C)O1 71829,C=CCC(CC)C(=O)N(CC(CC)NC(c1ccccc1SCC(F)(F)F)=O)C 71830,C(=O)(C(O)C(F)(F)F)N1CC(c2cn(CC(CC=C)CO)nn2)(C)C1 71831,c1(C(=O)NCC(C(C)C)NC(c2cc(OC(C)C)ncc2)=O)c(F)cccc1Cl 71832,c1(CC)ccccc1CC(=O)NC1CC12CC(NC(=O)C(c1ccc(C)o1)C)C2 71833,N1(C(c2c(C)cc(CNC(=O)C(C)c3ccsc3)o2)=O)CCC(C)C(F)(F)C1 71834,C1(NC(COCCCC)=O)CN(C(c2cc(CCC)nn2C)=O)C2(CCOC2)C1 71835,CC(C)CC(C)(CNC(C12CCC(C)(C1)OC2)=O)NC(c1cc[nH]n1)=O 71836,c1(C(COC)(C)SCCCNCC2(CC(N)=O)CC2)nnnn1CC(F)F 71837,c1(N2CC(C(C)NC(C3CC(C#C)(O)C3)=O)OCC2)ncc(C)c(SC)n1 71838,c1(C(N(C(CNC(c2cc(COC)sc2)=O)C)C)=O)ccc(C2(C#N)CC2)cc1 71839,c1(C(=O)NCC(CCOC)NC(=O)C(c2ccccc2)F)cc(C(C)=O)c(C)o1 71840,C1(CNC(c2coc3c2CCCC3)=O)CCN(C(=O)CC2OCCO2)C12CCC2 71841,CCC(C)CC(C(=O)NCCc1cc(C)[nH]n1)NC(c1cc(CO)[nH]n1)=O 71842,C1(C)(CN2CCCC(CC=CC)C2)CCC(F)(F)CO1 71843,C12(C(NCP(OCC)(C)=O)=O)CC(C)(CN1C(=O)CCCN(C)C(C)C)C2 71844,C1(CNC(c2ccccc2O)=O)CCN(C(=O)CCCOC2CCOC2)C12CC2 71845,c1(N(CC(CC)C)C)cccc(S(=O)(=O)N2CCCOC(COC)C2)n1 71846,C(C)(C)(CC(F)C(=O)NCC#Cc1cnn(C)c1)NC(CC(=O)OCC)=O 71847,c1(C(=O)NC2CC3CN(C(c4coc(Br)n4)=O)CC23)nccn2ccnc12 71848,C=CC1CN(C(=O)CCCOc2cccc(C)c2)CC1NC(=O)CCC1CCC1 71849,CCCC(C(O)C(=O)NOCC(O)CO)NC(=O)CNC(C)=O 71850,c1(C(C(N2CC3C(NC(C4C(C)(C)CC4)=O)C3C2)=O)=O)cc(F)cc(Cl)c1 71851,C1(CNC(c2c(CC)onc2C)=O)CCN(C(c2cc(Br)no2)=O)CC1C 71852,C(CCO)(C(=O)Nn1cc(CCCC#N)nn1)N(C)C.C12CCCC(O1)C2 71853,c1(C(C)C)ncncc1C(=O)NCC1CCCN1C(c1cccc(C(F)F)c1)=O 71854,C(=O)(C1=CCN(C(c2cnn(C3CC3)c2)=O)CC1)NCCCc1c(C)n[nH]c1 71855,c1(OC)ccc2ncc(C(N3CC(CNC(=O)CCc4cc(Cl)cs4)C3)=O)n2n1 71856,Cc1cnc(NC(C2CN(C(c3cnc(N(C)C)o3)=O)CCS2)=O)cc1I 71857,c1(C(C(=O)OC)N(C)C(c2ccc(O)c(OC)c2)=O)cccc(Cl)c1Cl 71858,c1(N(CC(C)C)C)nc(=NC2CCC(CO)C2)[nH]c2cccc(F)c12 71859,C1(C(=O)NC2CN(C(Cc3cc(COC)on3)=O)CC2F)CCCS(=O)(=O)C1 71860,c1(C(=O)NCC2(NC(C3CCC(F)(F)C3)=O)CC2)cc2cc(O)ccc2[nH]1 71861,C(C)(CNC(=O)CC1CCC(=O)CC1)(C(C)C)NC(C(CC)N(C)C)=O 71862,C1(NC(c2c(COC)cco2)=O)(CF)CCN(C(c2[nH]cc(C)c2C)=O)C1 71863,c1(CC(=O)NC(CNC(C2(C(=O)OC)CC2)=O)C2CC2)nc(C)c(C)o1 71864,CCC(CC)CC(F)C(=O)NC(C)(CNC(C1Cc2ccccc2C1)=O)CC 71865,c1(NC(=O)Nc2cc(SC)c(Cl)cc2)cc(Cl)c(C)cc1O 71866,C1(F)(C(NOCC2(C)CC2)=O)CCN(C(C2CCN2C(C)(C)C)=O)C1 71867,C1(NC(C2(CSC)CCC2)=O)CC2(CCC(NC(=O)C3=CCCCCC3)CC2)C1 71868,Cc1ncc(C(=O)NC2CCC(CCNC(=O)C=CCOC3CCOCC3)C2)s1 71869,c1(C(N(C(=O)C(F)CC2CCCCC2)C)=O)ccc2ncccn12 71870,CCCN(OCc1ccccc1)C(=O)C(O)CCCN=[N+]=[N-] 71871,C(=O)(CC(C(F)F)NC(=O)Cc1ccnn1C)NC(c1cc[nH]n1)C 71872,N1(C(C2(F)C(C)C2)=O)CCOC(CCNC(=O)Cc2nnn(C(C)(C)C)n2)C1 71873,N1(C(CC(C(C)OC)NC(=O)CN2CCN(C)C(=O)C2)=O)CCCC12CC(O)C2 71874,c1(C(N(C)CC2CCCN2C(C2CCCCO2)=O)=O)sc(F)cc1Br 71875,O=C(CC(O)C(Cl)(Cl)Cl)N1CCSc2nccnc21 71876,Cc1cnc2cc(C(=O)NC3CCC34CN(C(C3(C#N)CCCO3)=O)C4)nn2c1 71877,C1(C)(N(C)CC)CCN(C(=O)C=CC2CCCN2C(c2ccns2)=O)C1 71878,c1(C(N(CCN(C(=O)C(c2cnn(C)c2)C)CC)CC)=O)cn(C)c(=O)cn1 71879,Cc1c(F)ccc(C(N2CCCC2CCNC(C2C3CCCCC23)=O)=O)c1C#N 71880,C1(C(=O)NC(C)C(C)(C)NC(c2ccc(-n3cccn3)nc2)=O)CC(=O)NC1=O 71881,C1(C)(OCC(=O)N(CCC(C)O)C2CC2)CN(C(C2CC2C#N)=O)C1 71882,c1(C(=O)NCC2(CCNC(CCOCC#C)=O)CC2)ccc(Br)c(O)n1 71883,N1(C(C(CC(C)C)OC)=O)CC2CC(N=c3nc(C)nc4[nH][nH]cc3-4)CC1C2 71884,C1(C(C)C)(C(N2CCC(CN(C(=O)CNC(=O)NC3CC3)C)C2)=O)CNC(=O)C1 71885,CCC(CC(=O)NCc1nncs1)NC(=O)C=C1CCOCC1 71886,c1(N(CCOC)C)nc(N2CC(NC(=O)C(C)C)C(C)(C)C2)nc2c1CCC2 71887,c1(CCN(C)C(C2(CNC(=O)CCC3CCCO3)CCC2)=O)ccc(F)cc1 71888,C=CCCCCCCC(=O)N1CCCC(NC(=O)Cc2cc(C3CC3)no2)C1 71889,c1(SCC)cc(C(=O)NCC2CCCCN2C(=O)C=Cc2cn(C)nn2)ccn1 71890,N1(C(CC=C=C)=O)CCC(NC(C2(c3cc(F)ccc3C)CC2)=O)C(F)C1 71891,c1(N2CCC(CC)C2)cc(C)nc(N2CCC(Cc3ccc(C)cc3)C2)n1 71892,CC1=C(C)CC(C(=O)NCC2CCN(C(=O)CCc3cc(C)on3)CC2)CC1 71893,N1(C(C2N(Cc3n(C)ncc3Br)C3C(C2)C3)=O)C2CCCC1COC2 71894,C1(NC(C(C)=C(CC)C)=O)CC2CN(C(c3[nH]nc(C(F)(F)F)c3C)=O)CC2C1 71895,c1(C(N(C)CCOCCNC(C2CC(C(F)F)C2)=O)=O)ccn2c(O)nnc2c1 71896,Cc1nc(O)ccc1C(=O)NC1CC(C)N(C(=O)CN2CCCC2=O)C1 71897,N1(C(C(C)n2ccnc2)=O)CCC2(CCN(C(=O)CN3CCCC3=O)C2)C1 71898,N1(C(C2C(=C)CC2)=O)CCC2(CCC2NC(c2ccc(Cl)cc2C)=O)CC1 71899,c1(SCCNC(c2n(CCCOC)nnn2)C2CC2)nc2c(s1)CCCC2 71900,C1(O)(CNC(=O)CCOC2CC2)CCCN(C(=O)CC2(C(=O)O)CC2)CC1 71901,O=C1COCC2(CCCN(C(=O)COC(C3CN(CC(F)(F)F)C3)=O)C2)N1 71902,C1(C(N(CC(C)O)CCNC(c2cccc(O)n2)=O)=O)CC2(CCC2)CO1 71903,c1(-c2cccc(NC(c3c(OC(C)C)cccn3)=O)n2)ccc2scnc2c1 71904,CC1(C)CN(C(C2C3CCC23)=O)CCC1NC(=O)CCC1OCCO1 71905,C1(C)(C(=O)NCC(CNC(C2C(C(C)C)CCC2)=O)O)Cc2ccccc2C1 71906,C1(c2onc(-c3occ(C)c3)n2)COC(C)(C)N1C(=O)NC(C)(C)C 71907,N1(C(CCOC)=O)CC2OCC(NC(=O)C(C)(C)Oc3ccc(F)cc3)C2C1 71908,c1(C(N(C)CC2CCCN2C(=O)CN2CC(C)(C)C2)=O)ccc2c(n1)CCCC2 71909,N1(C(CC)=O)CCCCCCC1C(=O)NC(c1ccccc1)C 71910,Cc1c(Cl)ccnc1C(=O)NC(c1cn(CC(C)(C)O)nn1)C 71911,C1(NC(=O)Cc2ccc(Cl)cc2)(CO)CCCN(C(=O)CCc2cnc[nH]2)C1 71912,N1(C(c2c(OC)cccc2O)=O)CCC2(CCN(C(C3CC(CCO)C3)=O)C2)C1 71913,C1(C(=O)OCC(C)C(=O)Nc2ccc(C(=O)OC(C)(C)C)cc2)CCC(F)CC1 71914,CN1CCN(C(C2COCCN2C)=O)CC1C(=O)NCC(O)C(C)(C)C 71915,c1(CC(CC)N(C(=O)C(C)n2cccn2)C(c2ccccc2)=O)ccc(Cl)cc1 71916,N1(C(c2[nH]cc(C)c2)=O)CCN(C(c2csnn2)=O)C(CC(F)(F)F)C1 71917,c1(CCN(C2CCC2)C(=O)Nc2c(C)cc(O)nc2)csc2sc(C)cc12 71918,C#CCC(CC#C)C(=O)NC(C)CN(C(=O)CCC(C)(C)OC)CC 71919,c1(NC(C2CN(C(C3(C(F)(F)F)CC3)=O)CCS2)=O)ccc(F)c(Cl)c1 71920,Cc1cnc(C(=O)NCC2CC3CC3N2C(=O)C(C)n2cccc2)cc1C 71921,C(=O)(C1=NOC(C)(C)C1)N(CCC(=O)N(C(CO)C1CC1)C)CC1CC1 71922,Cc1cc(C#N)cnc1C(N1CCC(C)(NC(=O)CC(=O)NC2CC2)C1)=O 71923,c1(C(=O)NC2CN(C(C3(C)CCCCC3)=O)CC(F)C2)ccc2c(n1)CCC2 71924,c1(NC(c2c(C)c[nH]c2)=O)ccc(NC(=O)CN2CCC(C)(C)C2)cc1C 71925,S(=O)(=O)(c1ccc(NCc2nccn2CCSC)cc1Cl)NCC1(C)CC1(Cl)Cl 71926,C(=O)(C(=O)C(F)(F)F)NCCCOCCCNC(CS(=O)(=O)NCC)=O 71927,N1(C(C(C)CC2CC2)=O)CCCC(C2CN(C(c3ccc4occc4n3)=O)C2)C1 71928,N1(C(c2cc(OC)c(Cl)cc2)=O)CCC2CCN(C(c3cc(C)nn3C)=O)CC12 71929,C(C(C)C)(C(O)C(=O)N(C1(CC(=O)NC2CCC(=O)N(C)C2=O)CC1)C)OC 71930,C1(C)(C(=O)NC2CC(NC(CC(C=C)(C)O)=O)C2)CC(C(C)C)=NO1 71931,CC1CCCC(NC(=O)C(=O)NC(C)(CNC(=O)C2=CCC2)CO)C1C 71932,O=C1CCC(C(=O)N2CC3CC2CN3Cc2c(F)cc(Cl)cc2Cl)=NN1 71933,c1(C(C)=O)nc(C(=O)NCCC2CCN(C(=O)Cn3nnc(=O)[nH]3)C2)cs1 71934,C1(N(C(c2nc(OC)oc2)=O)C)CCCN(C(=O)COC2CCC2)CC1 71935,C12(C(=O)NCC(COCC)C)CCC(NC(c3c(C)ccnc3C)=O)(CC1)C2 71936,CC1CS(=O)CCN1C(=O)C(CCN(C)C)NC(=O)CCN1CCOC1=O 71937,C1(CCN(CCOCC#C)C)CCN(C(c2cn(C)nc2-c2ccoc2)=O)CC1 71938,Cc1cc(-c2nccn2C(c2ccccc2C)C)cnc1O 71939,Cc1cc(C)c(CC(N2CC3CC2C3NC(=O)CC2CC=CCC2)=O)s1 71940,C1(C(=O)NC(CCC)CC)C2CC3C(C2NC(C2(COC)CCC2)=O)C13 71941,c1(C(C)=O)c(NC(C23CC2CN(C(c2ccc(C#N)s2)=O)C3)=O)cccc1F 71942,C#CC1(C(=O)NC(C(C)C)C2CC2)CN(C(c2ccc(Cl)cn2)=O)C1 71943,N1(C(C2(NC(=O)CC3CC4(CC4)CO3)C(C)CCC2)=O)CCC2(CCOC2)CC1 71944,C(CCCCNC(C1(C(=O)NC2CC2)CC1)=O)N(C(C(C)OCCOC)=O)C 71945,c1(C(N2CCOCC(CNC(C(C3CC3)OCC)=O)C2)=O)cc(C)cc(C#N)c1 71946,c1(C(N2CCC(CNC(Cc3ccc(C)s3)=O)C2)=O)cc(O)nc(O)n1 71947,C(=O)(CCC(F)(F)C(F)F)N(C)CC1CCCN(C(C2CCC(=O)N2)=O)C1 71948,C1(C(=O)OC)CC(OC(C2CCN2Cc2ccccc2)=O)(NC(=O)OC)C1 71949,C1(C(N)=O)CC2CC(CNC(=O)N(CCC3CCCC3)Cc3ccccn3)C2C1 71950,C(=O)(C(=O)CCC(C)(C)C)NC1C(CNC(C(CCC)C)=O)CCC1 71951,C1(CC(=O)NC2C(n3cc(C(C4CC4)OC)nn3)CCCC2)CCCCC1(F)F 71952,CC(C)C(C)CC(=O)NCc1ncccc1C(=O)NC(c1ccn(C)n1)C 71953,Cc1cc(C(=O)NC2C3CN(C(=O)Cc4cnco4)CC23)nn1CC(F)(F)F 71954,CCCCC(CC(=O)NC1CCC(OC)C1)NC(c1ccc2cc[nH]c2c1)=O 71955,c1(CC(=O)NCC(C)NC(c2occ(OC)c(=O)c2)=O)noc2ccc(O)cc12 71956,C(=O)(C(C1=CCCCCC1)N1CCCCCCCCCC1)NC(C)(C)C 71957,C1(C(N(CC(=O)N)C(C)C)=O)CCN(C)C1CC.C1(OCC)(CC)CC1 71958,n1(C(CC)C)nccc1C(=O)NC(C1CCCN1C(=O)CCCNC(=O)OC)C 71959,CC1OC2(C(=O)NC3CCC(NC(c4cnc(-c5ccccc5)[nH]4)=O)CC3)CC1C2 71960,c1(CC(C)C(=O)NC2(C)CN(C(=O)CC(C)N(C)C)C2)ccc(Br)cc1 71961,N#CCCCC(=O)NCC#CCNC(C1(c2ncco2)CCC1)=O 71962,CC12CCCC(C(N3CCC(c4cn(C5CCCC5O)nn4)C3)=O)(CO1)C2 71963,c1(OCC(C)SCCC(C)C)cccc(Br)c1 71964,CCCC(C(=O)N1CCC2(C1)CN(C(=O)C=CC1CCC1)C2)S(N)(=O)=O 71965,CC(CC(=O)NCC1CCN(C(=O)CC=CCc2ccccc2)C1)CC(F)(F)F 71966,N1(C(C(CC)SC)=O)CC2(CCC(CNC(=O)C(O)CC3CCCC3)O2)C1 71967,C1(NC(c2cnc(C)n2C)=O)CC12CCC(NC(C1CN(C)CCO1)=O)CC2 71968,C1(N(C(c2ccc(COC)o2)=O)CC)(CF)CCN(C(C2CC3(CCC3)C2)=O)C1 71969,Cc1ccnc(C)c1C(=O)NCC1C(C(=O)NCc2cccc(O)c2F)C1(C)C 71970,c1(-c2nc(Cc3c(C)occ3)n(CC(F)F)n2)ccc2ccccc2n1 71971,Cc1cc2ccccc2n1CC(=O)NCC(CO)NC(=O)CC1CCNC1=O 71972,N1(C(c2ncc(C)c(Cl)c2)=O)CC(NC(=O)CS(=O)(=O)C2CC2)C(C2CC2)C1 71973,CC(C)CC(C(=O)NC(C)C(C)C1CC1)N(C(=O)CSc1cn[nH]c1)C 71974,C1(C(=O)NC(C)(C(=O)NCCc2cc[nH]n2)C2CCC2)CCCC(F)C1 71975,c1(CC(=O)NC(CC(=O)NCC2CCC(C)(C)O2)CC2CC2)ccc2c(c1)CC2 71976,C(=O)(C(C(C)(C)C)C1CC1)NC1C(C)CN(C(=O)C(c2ccccc2)N(C)C)C1 71977,c1(C(=O)NC2(CNC(C(CC=C)C)=O)CCOC2)ccc(C(C)=O)nc1O 71978,C12C3CN(CC13)NC2=O.c1(C)ccc(OCF)nc1.C1(CCCO)CCCO1 71979,c1(C(N(C)CC2CCN(C(c3cscc3Br)=O)CC2)=O)cc(F)cc(F)c1Cl 71980,C(N=c1[nH]c(=N)[nH]c(=NC(C)Cn2ccnc2C)[nH]1)C1(OC)CCCC(C)(C)C1 71981,C(=O)(CC(C)(C)C(=O)NCC1CCN(C(=O)COCC(C)C)C1)OCC 71982,C1(F)(C(=O)NC(C2SCCS2)C)CN(C(=O)C(F)OC(F)(F)F)C1 71983,C(C1=CCCCCC1)(c1nnnn1C1CC1)NC1(C(N)=O)CC1 71984,C1(C(N2C(C(C)(C)NC(C(C)NC(=O)NC)=O)CCC2)=O)CCC2CC2C1 71985,N1(C(C(CCC)(C)O)=O)CC2(CC(NC(=O)Cc3cccc(C#C)c3)CO2)C1 71986,N1(C(C(CC)Oc2ccccc2)=O)CCC2CC1CN2C(c1csc(CO)n1)=O 71987,N1(C(CCCCCSC)=O)CC2CCC(N=c3[nH]ccnc3F)CC2C1 71988,c1(NC2(c3nnnn3CCCOCC3CC3)CCN(CC)C2)ccc(I)cc1Br 71989,CCCCC(CC(=O)Nc1ccc(C(C)C)nc1)NC(=O)CCn1cncn1 71990,c1(C(=O)NCCC2COCC(C)O2)cccc2c(O)nncc12 71991,CC1CN(C(c2cc(Br)co2)=O)CC1CCNC(C1(O)CCC1)=O 71992,N1(C(C2(F)CCN(C(C3=C(C)CCC3)=O)CC2)=O)C2CCC1CC(O)C2 71993,c1(CCNC(CN(C(C(OC)OC)=O)CC2CC2)=O)cc(O)ncn1 71994,C1(NC(c2cnn(C(C)C)n2)=O)CCCCCC1C(=O)NCC(c1cnc[nH]1)C 71995,N#Cc1ccc(C(N2CCC23CN(C(=O)Cc2ccc(Cl)cc2F)C3)=O)c(Cl)c1 71996,CC1(C(N2CC(N(C)C)C(CNC(=O)CC3CCS(=O)(=O)C3)C2)=O)CCCC1O 71997,C1(OC)CC2(C1)CC(C(=O)NC1CC(NC(c3coc(C4CCC4)n3)=O)C1)C2 71998,C1(NC(Cc2nc(C)sc2)=O)CCOCC1C(=O)NCCc1ccncc1 71999,C1(CNC(C2C(=C)CN2C(=O)OC(C)(C)C)=O)CCCCC1OC(C)(C)C 72000,Cc1nc(O)sc1C(=O)NC(c1cn(C)nn1)C(=O)NCC(c1ccccc1)F 72001,C(CN=C(NCc1ccc(N(C)C)cc1)N(C)Cc1nc2c(s1)CCCC2)OC 72002,N1(C(c2cnc3cc(C)nn3c2)=O)CCC2(C1)CN(C(=O)C=C(Cl)Cl)CCO2 72003,Cc1ccc(OC(C)C(=O)NC(C2CCCC2)CNC(c2coc(Cl)n2)=O)cc1 72004,Cc1cc(N2CCC(C)C(NC(=O)CSCCC(F)(F)F)C2)nc(C(F)(F)F)n1 72005,C1(C(=O)NC(CC)CN(C)C(c2coc(C)c2)=O)COc2cccc(OC)c2C1 72006,C(=O)(C(CCC1CCC1)N1CCC(Cc2nccn2C)C1)NCCSC 72007,c1(C(N(CC(O)CNC(=O)Cc2ccccc2)C)=O)ccc([N+](=O)[O-])n1C 72008,c1(C(C)C)ncsc1C(=O)NC(C)CN(C)C(c1ccnn1C1CC1(F)F)=O 72009,Cc1ccc(O)c(N(C)Cc2csc(Br)c2Br)n1 72010,N1(C(C(c2cccc(OC)c2)C)=O)CC2CCC1C2NC(c1sccc1C)=O 72011,N1(c2n(CC(=C)C)c(-c3ccccc3F)nn2)CCC2CCCC12CN 72012,FC1(F)C2CCC1CN(CC(=C1CCOCC1)Br)C2 72013,c1(C(N(CCC)CCNC(c2ocnc2C2CC2)=O)=O)c(C)cccc1F 72014,C1(CNC(c2ccoc2)=O)CCCCC1NC(C1CC(O)(C(F)(F)F)C1)=O 72015,N1(C(Cc2cccc(OCC)c2)=O)CCCC(NC(C2(CC(C)C)CC2)=O)C1C 72016,CCC(CC(=O)N1CCC1C(N1CCC(C)(O)C1)=O)SC 72017,C(C(C)C(C)C(=O)NC1C2CC1CN(C(C1CSCCS1)=O)C2)OC 72018,C(=O)(C(C)CCCC(C)C)NC1C(NC(c2c(SC)cccc2)=O)CCC1 72019,C#CCC(O)C(=O)N1CCC(COC)(NC(=O)Cc2csc(COC)n2)C1 72020,c1(C(=O)NCCCCCCN(C(CC(C)O)=O)C)ccc(S(N)(=O)=O)c(N)c1 72021,C#Cc1cccc(OCC(=O)NC2(F)CCN(C(=O)CCCNC(N)=O)CC2)c1 72022,c1(OC)cc(NC(c2[nH]c(C)c(C(=O)NCC3(C4CC4)CC3)c2C)=O)cc(C)c1 72023,C1(NC(CCCC#C)=O)C2CC3CN(C(=O)CCN4CCSC(C)(C)C4)C1C3C2 72024,CN1C(=O)Cc2c(C(=O)NCC(C)(C)NC(=O)C(F)C(F)(F)F)cccc21 72025,C12(C(N3C4C(NC(C5C(C)(C)NC(=O)C5)=O)C(C4)C3)=O)CCC(C1)S(=O)(=O)CC2 72026,c1(C(=O)NC(CCOC)CNC(c2cnc(C(C)C)s2)=O)cncc(C)c1C 72027,c1(CC(C(=O)O)NC(C2CC2c2ccccc2)=O)c(I)ccnc1F 72028,Cc1cccnc1CCC(N1CC2CC2(NC(=O)CSCCC#N)C1)=O 72029,C(=O)(C1=CCCSC1)N1C(CCCNC(CNS(CCOCC)(=O)=O)=O)CCC1 72030,C1(CC(=O)NCCC2CC(NC(=O)C=CC3CCCC3)C2)CC(F)(F)C1 72031,CC1(C)CCCC(C(N2CCC(CO)(NC(C3CC(F)(F)C3)=O)C2)=O)C1 72032,c1(C(=O)OC2(CN(CC)CC)CCCC2)cc(N2CCOCC2)ccn1 72033,c1(C(c2n(CC=C)nnn2)(C)NC2COC(C(F)F)C2)ncccc1C 72034,N1(C(c2c(C)c[nH]n2)=O)CC2CC1CCC2NC(c1cc(C)c(F)c(C)c1)=O 72035,N1(C(CCC2CC(NC(C3C(C)CC(=O)NC3)=O)C2)=O)CCCN(C)CC1C 72036,N1(C(c2n(CC=C)ccc2)=O)CCC(C)(C)C(CNC(c2ccsc2C)=O)C1 72037,N1(C(c2cc(OC)nn2C)=O)CCC(CO)(NC(c2snnc2C)=O)CC1 72038,c1(NC(CC)=O)ncccc1C(=O)NC1COCC1n1cc(CCOC)nn1 72039,N1(C(C(C)(C)CC#N)=O)C2CCCC1CN(C(C1CCc3ccnn3C1)=O)C2 72040,c1(C(=O)NCCCCC(C)NC(C2C(=C)CC2)=O)c(O)cc(Cl)cc1Cl 72041,C12(NC(c3cc(C(C)C)n(C)n3)=O)CCC1CN(C(C1CCOC(=O)CC1)=O)C2 72042,c1(NCC)cccnc1C(=O)N(CC(C)CNC(=O)C(c1cccc(Cl)c1)C)C 72043,C(=O)(CN=S(C)(C)=O)NC1(C)CC(NC(C2CCCN2C2CC2)=O)C1 72044,CC1(C)C(CNC(=O)C(O)C2CCC2)CCN1C(=O)CCCn1cccc1 72045,C(=O)(CCCCCNC(N)=O)N1CCCC(NC(c2c(C)nnc(O)n2)=O)CC1 72046,c1(-c2c(OCCC)cccc2)cccc2c1CCN(Cc1n[nH]c3c1CCC3)C2 72047,c1(C(=O)NC2(CC#C)CC2)n[nH]c2c1CN(C(c1cc(F)ccc1O)=O)C2 72048,c1(C(N2CC(CNC(c3c(O)cccc3O)=O)OCC2)=O)ccc(Br)cc1F 72049,CC(C)(C)C(O)C(C(=O)NCC(c1ccco1)O)C1CCCC1 72050,S(=O)(=O)(c1cccc(Cl)c1)NCC(N1CCC(N(C)C(c2cccs2)=O)C1)=O 72051,C12(CNC(CN3CC(C)(OC)C3)=O)CC1CN(C(=O)CCc1n[nH]c(=N)s1)C2 72052,N1(C(C2CC(C(=O)OC)C2)=O)CC2CC1C2NC(c1cnncc1C)=O 72053,N1(C(C2N(C(C)C)C(=O)CC2)=O)CC(NC(C2C(C)(C)OC2(C)C)=O)CCC1C 72054,C1(CNC(C=CC(C)(C)C)=O)CC2COCC2N1C(C1(F)CC2(CCC2)C1)=O 72055,N1(C(C(CC#C)CC#C)=O)CCC2C(C1)NC(=O)CN2C(=O)CCCC(C)CC 72056,c1(NCc2ccc(C#N)s2)cnc(F)cc1C(=O)Nc1cc(Br)cc(I)c1 72057,C1(CNC(=O)C2=CCCC2)CCC12CCN(C(c1cnc3ccsc3c1)=O)CC2 72058,N1(C(C(CC)F)=O)CC2CC1CN2C(c1ncsc1Br)=O 72059,CCC(C)(C(=O)N1CC(CNC(=O)CO)C1)C(N)=O.CCCC(C)N(CCC(=O)ON)C 72060,N1(CCO)CCC(N)CC1C.N1(C(C)C)CCC(NC(=O)C(F)=C2CCCC2)C1=O 72061,C1(C(=O)NCCCOCCCNC(C=C(C)C)=O)CCC2(CCC2)CC1 72062,C1(NC(c2sccc2CO)=O)C=CCC(C(=O)NC2CCCC2F)C1 72063,N1(C(C(CC=CC)C)=O)CC2CC1CC2CNC(=O)CCNC(=O)CO 72064,N1(C(C(CNC(=O)C(C2CCCCC2)F)OC)=O)CCC(F)(C(N)=O)CC1 72065,N1(S(CC2CCC(N(C)C(=O)OC(C)(C)C)C2)(=O)=O)CCOC(C(=O)C2CC2)C1 72066,N1(C(CC(=C=C)C)=O)CC2(CCCN(C(=O)CNC(=O)Oc3ccncc3)C2)C1 72067,C1(C#N)(C(=O)NC(CC)CN(C)C(c2cc(SC)oc2C)=O)CCCCCC1 72068,c1(C(N(CC(CC)NC(C2CSCCS2)=O)C)=O)cc(C)c(C)o1 72069,C1(C(=O)NC2(CC=C)CCCC2)CN(C(C2CC23CCCC3)=O)CC1(F)F 72070,c1(C(=O)NCCc2ccc(CNC(C=CS(C)=O)=O)cc2)nc2cnccc2s1 72071,c1(C(=O)NC(C(=O)NCC(COC)(C)CO)C2CC2)cn2c(n1)CCC2 72072,c1(C(=O)NCCC(C)NC(C2CC(N(C)C)CCO2)=O)ccc(C(F)(F)F)nc1 72073,N1(C(=O)CC2(O)CC2)CCC2CCCC(C1)N2C(C1CCc2ccccc2C1)=O 72074,C1(C(=O)NC2C3(CC(NC(c4ccnnc4)=O)C3)C2)CC12CCSCC2 72075,O=C(C1CCCc2nccn21)NC1CC1C1CCN(C(=O)C=C2CCC2)CC1 72076,c1(OC)nc(F)ccc1-c1cc(CNC(=O)C(N)=O)ccn1 72077,Cc1scc(NC(=O)NCC2CCCC2C(=O)Nc2ccnc(C3CC3)c2)c1C 72078,c1(C(=O)NCC2N(S(CCCC)(=O)=O)CCCC2)cc(Cl)cc(OC)c1O 72079,N1(C(CCC2C(C)=NOC2=O)=O)CC(NC(c2onc(C)c2C)=O)CC1(C)C 72080,Cn1cc([N+](=O)[O-])c(C(=O)NC2CC(NC(c3coc(Cl)c3)=O)C2)n1 72081,Cc1c(NC(c2ccc(OCc3ccccc3C#N)cc2)=O)cc(F)cc1C#N 72082,N1(C(c2cc(C(C)=O)[nH]n2)=O)CC(n2cc(CN3CCCC3)nn2)CCC1(C)C 72083,c1(NC(CCN(C(C2C(OC)(OC)CC2)=O)C)=O)ccncc1C(C)C 72084,N1(C(C(C)CCO)=O)CC(C2CCCN(C(=O)C(C)(O)C3CC3)C2)C1 72085,N1(CC(=O)NC(c2ccc(Cl)cc2)C(=O)OC)CCC(C(=O)N(C)C)CC1 72086,c1(C(=O)NCCN2C(C(=O)NC3CCC3)COCC2)c(Cl)ccc(F)c1F 72087,CC(CNC(=O)CCC(N)=O)C(F)C(=O)NCCCC(C)(C)C 72088,C1(C2(O)CCN(C(=O)CCNC(C)C)CC2)(NC(CCc2ncc(C)[nH]2)=O)CC1 72089,N1(CC)CCC(N2CC3CC2(CO)C3)C1=O 72090,CCS(=O)(=O)CC(=O)NCC1(F)CCCN(C(c2occc2C(C)C)=O)C1 72091,Cc1cc(CNC(=O)CC(O)CNC(C2CCOC2)=O)sc1C 72092,c1(C(=O)NCC2N(C(CN3C(=N)CCC3)=O)CCC2)ccnc(F)c1F 72093,CC(C)C(O)CC(=O)N(C(C)CCNC(=O)Cc1ccc(Cl)cc1F)C 72094,c1(C(=O)NC2C(NC(CSC)=O)CCCC2)cc(Cl)cc(C)c1O 72095,C1(NC(c2sc(CC)c(C)c2)=O)CN(C(C2(C)CC(C)C2)=O)Cc2ccnn2C1 72096,CC1(c2cn(-c3ccccc3)nn2)CCN(C(c2cc(CC3CC3)on2)=O)C1 72097,c1(C(=O)NC(CC)CNC(C2C=CCC2)=O)csc2ccc(Br)cc12 72098,CCC(O)C(F)(F)C(=O)N1CC2(CNC(c3cc(C)on3)=O)CC1CO2 72099,C1(NC(=O)C=Cc2ccccc2)CN(C(=O)C(O)CC2CC2)CCC1C(F)(F)F 72100,c1(NCC(C)NC(=O)OC)nc(N2CCOC(C)(c3ccccc3)C2)cc(C)n1 72101,C1(CN(C(=O)Cn2cc(C3CC3)nn2)C)CCCN(C(c2cccc(O)n2)=O)C1 72102,CN1CCOC(C(=O)NC(CCOCCO)C(=O)NC2CCC(C)CC2)C1 72103,C1(C(c2ccccc2)C(=O)OC2CCS(=O)(=O)C2)CCCOCC1 72104,N1(C(c2c(C)nc(F)cc2)=O)CCC2(CC1)CCN2S(=O)(=O)c1ccc(Cl)cc1 72105,n1(CCCC)nc(COc2ccccc2)nc1-c1ccc(=O)oc1 72106,C(C(CC(C)C)C(=O)N1CCC(O)(CN(C(=O)C=CCF)C)C1)OC 72107,C(C)(CN=C(NCC(=O)NC1(C)CC1)NC1CCC1)OC 72108,C#CC1(C(=O)NOCC(=O)NCCC2CCC(C)C2)CC(=O)C1 72109,c1(NS(CC)(=O)=O)nnc(N2CCOC(c3nccs3)C2)n1CC1CC1 72110,N#CC1CN(C(c2ncc(F)cc2F)=O)CCN1C(c1sccc1Br)=O 72111,CC(C)C(C(=O)NCC(C)(Cn1cccn1)NC(=O)C=CC(F)(F)F)NS(C)(=O)=O 72112,C1(C(=O)NCCC=C=C)(CC)CN(C(=O)C(CC)OC)C1 72113,C(=O)(CCCCC#N)NCc1cccc(C(N(C(C)C(=O)NC)CC)=O)n1 72114,Cc1cc(C(=O)N(C(C)CNC(=O)C(c2cccc(Cl)c2)C)C)oc1C 72115,C#CC1(C(=O)NC2CCOC(C)(C)C2)CCN(C(=O)CNS(=O)(=O)CC)CC1 72116,N1(C(c2c(C(C)C)scn2)=O)CCC2(COC(CNC(=O)C(C)CO)C2)C1 72117,c1(CNC(=NCC23CC(C)(OC2)C3)NCC2CCCCC2)cc(Cl)cnc1F 72118,C1(C(=O)NCC(C(C)O)C)N(C(=O)Cn2cncn2)CCC1(C)C 72119,C1(C(=O)NCC(CNC(C2N(C(=O)NC)CCC2)=O)(C)C)C2CNC(=O)C12 72120,C1(C(N2CCCC(N(C(c3ccc(N)cn3)=O)CC)C2)=O)CCC(F)(F)CO1 72121,C#Cc1ccc(C(N2CCC(C)(C)C2CNC(C2(N(C)C)CCCC2)=O)=O)cn1 72122,c1(C(N2CCC(C)(C(=O)NCc3ccccc3)C2)=O)cc([N+](=O)[O-])c(F)cc1Br 72123,CC(C(=O)NCC1(NC(=O)CCN2CCC2)CCCC1)C1OCCc2sccc21 72124,CC1CC(N=c2[nH]c(=NCc3cc(Cl)ccc3N(C)C)[nH]c3cc[nH]c23)CC(C)N1 72125,CCCCCC(=O)N(C1CCCC(NC(C2(COC)C=CCC2)=O)C1)C 72126,c1(C(=O)NC(C(C)C)CNC(=O)CC2(C)CC2)ccccc1-c1ccccc1 72127,c1(C(=O)NCC(=C)CCNC(C2(S(C)(=O)=O)CC2)=O)cc(Cl)ccc1Cl 72128,c1(C(=O)NCC2C(C)(C)CCCN2C(=O)CS(N)(=O)=O)ccc2nc(O)[nH]c2c1 72129,N1(C(C(COC)O)=O)CCC(C)(NC(=O)COc2cccc(NC(C)=O)c2)C1 72130,c1(OC)ccc(CC(=O)N(C(CNC(c2ccc(Cl)s2)=O)C2CC2)C)cn1 72131,c1(C(=O)NC(C)(C)CC(=O)N2CCC(CCO)CC2)ccc2c(c1)CC2 72132,CC(=O)CCCCC(=O)N1CC(C(=O)NCC(C2CCCC2)C)CC1(C)C 72133,c1(CN2CCCC(C(C)NC(=O)COC3CCOC3)C2)ccc(F)cc1Br 72134,c1(OC)cc(NC2(CNC(c3ccc([N+](=O)[O-])nc3)=O)CC2)cc(OC)c1O 72135,Cc1cn2cccc(NC(C3CN(C(=O)CSc4nc[nH]n4)CCN3C)=O)c2n1 72136,c1(C(N2CCN(C(c3c(SC)nccc3)=O)C3C2C3)=O)cc2cc(F)ccc2[nH]1 72137,C12(C(=O)NCCOCCN(C)C(c3ccc(CO)s3)=O)CCOC1CCOC2 72138,C(C(=O)NCC12CC(CN1C(=O)CC1CSCCS1)C2)(C(C)C)SCC 72139,c1(C(=O)NCC2CCC(NC(C3CCNC3=O)=O)C2)cc2cc(F)ccc2s1 72140,Cc1nsc(NC(C2CC(F)CN2Cc2c(Cl)cccc2Br)=O)c1C#N 72141,C(=O)(C(C)(C)C(C)(F)F)N(C(C)CCNC(C1CCC2CC2CC1)=O)C 72142,C1(OC)CN(C(=NCCCN2CCCCCC2=O)NC2CCC2)CC1O 72143,Cc1ccc(C(=O)NCC2CCCN2C(=O)CC2CC3CC3C2)cc1S(C)(=O)=O 72144,C1(C(=O)NC2C3CN(C(C4ON=C(C)C4C)=O)C2C3)OCCCC1(C)C 72145,C#CCC(C)(C(=O)NCC(F)(F)C(N)=O)NC(=O)CCC1CC1(F)F 72146,C(CCC)(C(=O)NC(c1ccnn1C)C(=O)Nc1cccc(SCC)c1)=CCC 72147,CC12CC(CCO1)N(C(C1CC3(CCN1C(=O)C(N)=O)CC3)=O)C2 72148,C=CCC(CC)C(=O)N1CC2CC(C1)N2C(C1C=CC=CC=C1)=O 72149,C#CC1CN(C(=O)C(N2CCC(C(C)COC)CC2)=O)CCN1 72150,C1(CNC(c2c(C)cn(C)n2)=O)CC(C)CN(C(=O)C(C)NC=O)C1 72151,C12(C(N3CCC(N(C(C=CC(CC)C)=O)C)C3)=O)CCC(CC1)C(C)(C)O2 72152,N1(C(C(CCSC)O)=O)CC2(CCC2NC(=O)Cn2cnnn2)C1 72153,CC1CC(C(=O)NCCOCCNC(=O)CCC=Cc2ccccc2)C1(C)C 72154,c1(C(=O)Nc2cc(F)c(O)c(F)c2)cn2c(n1)CN(Cc1ccc(Cl)cn1)CC2 72155,c1(C(=O)NC(C)CCCCNC(=O)C=Cc2ccccn2)ccc2c(c1)CCC2 72156,N1(CC)CCC(C(=O)NC2(C(=O)NC3COCC3CN(C)C)CSC2)C1 72157,C1(=O)C(CN=[N+]=[N-])N1.C(=O)(C(CC)n1cncn1)NCCN(CCC)C(C)C 72158,C1(NC(C(F)OC)=O)CC2(C1)CC(CNC(C1CNC(=O)C1)=O)C2 72159,C=C(Cl)CCC(=O)N1CC(CCNC(c2cc(C(F)(F)F)ccn2)=O)C1 72160,C1(NC(CCCC#C)=O)CS(=O)(=O)C12CCN(C(=O)C(C)CS(C)(=O)=O)CC2 72161,c1(C(=O)NCCCNC(Cc2ccn(CC)n2)=O)cc(C)oc1C(F)(F)F 72162,C1(C(=O)NCc2cc(C)oc2)CCOCCN1C(c1ccc(C#N)s1)=O 72163,C#Cc1cncc(C(=O)NC2COCCC2C(=O)NCCc2cncs2)c1 72164,n1(C(C)C)c(O)nc(N2CCC(NC(c3cc(Cl)ccc3F)=O)CC2C)cc1=O 72165,c1(C(=O)NC(C2CCN(C(CC=C)=O)C2)C)ccc(F)cn1 72166,C1(C(=O)NCCCC(C)NC(C=C(COC)C)=O)CCC(=O)N(C(C)C)C1 72167,C=C(Cl)C(C)(C)C(=O)NC1CC(CNC(=O)Cc2cnn(C)c2C)C1 72168,CC1CCC(C(=O)NCC(C2CCCC2)NC(c2cc[nH]n2)=O)CC1 72169,S(=O)(=O)(c1cccc(F)c1F)NCC(c1cnn(C)c1)C 72170,N1(C(C(CC#CC)NC(=O)OC(C)(C)C)=O)CCS(=O)(=O)C(CO)C1 72171,C=CCCC(C(=O)NCCC(C)(C)C)NC(=O)CCCSC 72172,C(=O)(C1=C(C)Oc2ccccc2C1)N1CC(NC(CCC#CC)=O)C(OC)C1 72173,C(=O)(CS(=O)(=O)CC(C)C)N1CCC(N(C(C2CC2c2nccn2C)=O)CC)C1 72174,c1(NC(=O)NCCCNC(C2CCCN(C(C(C)C)=O)C2)=O)cc(N)c(F)cn1 72175,c1(-c2scc(C(N(C)CC3CN(C(C4CC4F)=O)C3)=O)n2)ncccc1F 72176,C(=O)(CC(C)(C)N(C(=O)CCNC(=O)OC)C)N(CCOCC=C)C 72177,C(=O)(C1=CCCCC1)NC(CSCC)C(=O)NCc1nc(C)cs1 72178,Cc1nc(C2CCCC2)sc1C(=O)NC1CCCC1NC(=O)CCN(C)C 72179,N1(C(c2c(Br)ccc(C)n2)=O)CCC2(CCN(C(C3CC3C3CC3)=O)CC2)C1 72180,C(=O)(C(C)C(F)(F)F)N1CC(N2CCN(C(c3c(OC)cncc3)=O)CC2)C1 72181,C1(NC(c2cc(CC)nnc2C)=O)CCN(Cc2nnc(C3CC3)s2)CC1(C)C 72182,C(CCN(C(=O)CCSc1nccn1C)C)(C(C)C)NC(c1ccc(CC)[nH]1)=O 72183,c1(CN2C3C(CNC(C)=O)(CCCC3)CC2)cc2cc(C)ccc2[nH]1 72184,c1(CC)c(C(N2CC(CO)(CNC(=O)COCCSC)C2)=O)nnn1C 72185,C12(CC)CCN(C1)C2.c1(CNC(=O)OC(C)(C)C)cccnc1Br 72186,C1(C(N(CCC(=O)NC)C)=O)CC2(CCC2)CN1C(=O)CN(C)C 72187,C12(C(N(CCC=C)CC)=O)COCC1CN(C(c1cc(OC)n[nH]1)=O)C2 72188,c1(C(=O)NCC2(F)CC(NC(COCC(=C)C)=O)C2)cccn(C2CCC2)c1=O 72189,Cc1cc(C(=O)NC2CC(NC(C3CC3C3CC3)=O)C2)cnc1C(F)F 72190,c1(OC)nc(C)c(C(N2CCCCC2C(=O)Nc2cnn(CCO)c2)=O)s1 72191,c1(CC)nsc(CNC(=O)C(C2CCOC2)NC(c2sccc2F)=O)n1 72192,Cc1cnncc1C(=O)N(C1CC1)CC1CCCN1C(=O)CC12CCCC1C2 72193,c1(C(=O)NC2CCCCC2CNC(c2n[nH]cc2F)=O)ccc2c(c1)OCCO2 72194,N1(C(C2(NC(c3ccc(C)o3)=O)CCCC2C)=O)CC2CSCC(C2)C1 72195,C(=O)(CCC(=O)NC1CCCCC1NC(c1nc(C(C)C)oc1C)=O)NCCC 72196,N1(C(C2CC(C)(C(=O)OC)C2)=O)CCN(C(=O)CN2CCCNS2(=O)=O)C(C)C1 72197,C1(OC)(CNC(c2sc(C)c(Br)c2C)=O)CCC(C)CC1 72198,C1(C(=O)NC(C(=O)N(CC)CC)C)CC2CCN(C3CCC3)CC12 72199,CC(C)CC(C(=O)NCC12CC1CN(C(C1(N(C)C)CC1)=O)C2)c1ccccc1 72200,C1(c2n(CCSC)nnn2)(NCc2ccc(Cl)c(Cl)c2)CCOC2(CCOC2)C1 72201,N1(C(C2CC(O)CN2Cc2cccc(Cl)c2Cl)=O)CCC2(CCCO2)C1 72202,N1(C(c2c(C)nns2)=O)CCC2(CC1)CC2C(=O)NCC(C)S(C)(=O)=O 72203,N1(C(COc2ccc(C(C)C)cc2)=O)CCCC(NC(=O)CS(N)(=O)=O)C1C 72204,C1(OC)CC(CC(=O)NC23CC(NC(c4cc(C(C)(C)C)on4)=O)(C2)C3)C1(C)C 72205,N1(C(C(C)NC(C)(C)C)=O)CCN(C(=O)C=Cc2cncc(F)c2)C(CF)C1 72206,c1(OC)c(C(=O)NCCC(C(C)C)NC(C2CC=CCO2)=O)c(C)nn1C 72207,C1(NC(=O)CC2(C(F)(F)F)CC2)CCN(C(c2ncc(Cl)s2)=O)CC1CO 72208,C1(C(C)NC(C2CCC3CC23)=O)CN(C(c2csc(C(C)(C)C)n2)=O)CCO1 72209,CC1CC(=O)NC1C(=O)NCC1CCCN(c2ncc(Br)cn2)C1 72210,Cn1cc(Cl)c(C(=O)NC2CC(NC(c3cccc(OCC(F)(F)F)c3)=O)C2)n1 72211,N1(C(=O)OC)CCCC(C(N2CCC(OCC(c3ccncc3Cl)=O)CC2)=O)C1 72212,CC#CCCCC(=O)NC1(C(=O)NCCOCCCO)CCSC1 72213,c1(C(=O)NC2C(CNC(CNC(=O)NC)=O)C2)coc(C#Cc2ccccc2)c1 72214,Cc1ccn(C)c1C(=O)NCC(C)CNC(C1(c2ccccc2)CC1Br)=O 72215,c1(OC)ccc(C(=O)NC(C)CNC(c2cc(C(O)C(F)(F)F)ccn2)=O)nc1 72216,CC1CC(C(=O)NCC2CCN(C(c3cc(F)ccc3O)=O)C2(C)C)=NO1 72217,N1(C(Cc2n(C)cnn2)=O)CCN(C(CC(C2CC2)C2CC2)=O)CC1 72218,Cc1c(Br)cnc(O)c1C(=O)NC(C)CNC(C1CCCC(F)C1)=O 72219,O=NN1CCCC1C(=O)NC1C=CCN(C(c2ccc(-c3cn[nH]c3)cn2)=O)C1 72220,Cc1noc(C)c1CC(=O)NCC1(O)CCN(C(=O)C(C)NS(C)(=O)=O)C1 72221,n1(CC)cc(C(=O)NCC(O)CN(C(=O)CCn2ccnc2)C)c(C(C)(C)C)n1 72222,N1(C(CCCOCCC)=O)CCOCC(F)(CNC(=O)CC2CCNC(=O)C2)C1 72223,N1(C(C2CC(=O)NC2)=O)CC2CCC1C(CNC(c1n[nH]c3c1CCOC3)=O)C2 72224,C(=O)(CCCCOC)N1C(C2(C(=O)NCCCCC=C)CC2)CCC1 72225,Cc1ccc2sc(N3CCCC3CNC(=O)C(C)CF)nc2c1C 72226,c1(CC)ccc(C(C)C(=O)NCC2C(C)CCN2C(=O)Cc2n[nH]c(C)n2)cc1 72227,CCC(C)(C)CC(=O)NCCC1(NC(C2CCCN2c2cnccn2)=O)CCC1 72228,C(=O)(CC(O)CNC(C1CN(C2CCC2)C1)=O)N(C1CC(F)(F)C1)C 72229,N1(C(C(C)C)=O)CC(CNC(=O)COCc2nnc(S)n2C)C2(CC2)C1 72230,C=Cc1ccc(C(=O)N(C(C)CN(C)C(c2cccn(C3CC3)c2=O)=O)C)cc1 72231,C1(N(C(=O)CC2CCC2)C)CCCN(C(c2ccccc2N2CCOCC2)=O)C1 72232,c1(CN(C(=O)NCC(CC)(C)COC)C)cccc(Br)c1F 72233,CC1CCc2ccccc2N1Cc1cn(C2CCC(C(=O)NCCO)C2)nn1 72234,c1(C(=O)NCC2(F)CCC(CNC(CCSCC)=O)C2)cccc(Cl)c1F 72235,c1(C(=O)NCC(C(C)C)NC(=O)C2=CCCC2C)cc(C(F)(F)F)cc(F)c1 72236,CC(C)CC(C(=O)NC(c1cnn(C)c1)C)NC(c1cccc(Cl)c1)=O 72237,C1(OCC(=O)NCC(CC)NC(c2cc(C(=O)OC)cs2)=O)CCCCC1C 72238,N1(C(C(=O)Nc2cccc(OC)c2)=O)CC2CC2(C(N(CCNC)C)=O)C1 72239,N1(C(COCC(=O)OC)=O)CC2CCC(C1)C(NC(=O)C(C(C)C)C1CCC1)C2 72240,C(C)(CCC(=O)N1CC(OC)CC1CNC(c1occ(C)c1C)=O)OCC 72241,C1(CNC(=O)CCc2ccsc2)CCCC1C(=O)NCCC1CCOCC1 72242,c1(C(=O)NC2(CN(C)C)CC2)ccc2c(c1)C(C)(C)OC2 72243,c1(C(N(C(C)CCNC(c2cnc(S)n2C)=O)C)=O)c(Cl)nc2ccccn12 72244,N1(C(C(C2CC(F)(F)C2)OC)=O)CCCC2(NC(c3cnsc3C)=O)CC2C1 72245,CCC(F)(F)C(=O)NC1C=CC(CC(=O)NCc2ccc(OC)nc2)C1 72246,Cc1ccnc(C(F)(F)C(=O)NCC(C)(C)NC(=O)CC(C)N2CCCC2=O)c1 72247,c1(OC)ccccc1CN(CC(C)C#N)C(c1ncoc1-c1ccccc1F)=O 72248,N1(C(c2ccc(C)cc2)=O)CC(C(=O)N(C2CC2)CC2CC2)CC(C)(C)C1 72249,CN1CCN(C(C2(F)CCCOC2)=O)c2cnccc21 72250,C1(NC(c2c(C)nncc2)=O)CCN(C(=O)CC23CCC(CC2)OC3)CC1F 72251,C1(CNCc2c(I)cn(CC(F)(F)F)n2)CCCC12CCOCC2 72252,Cc1c(Br)csc1C(=O)NCC1CN(C(=O)C(O)CN(C)C)CC1O 72253,c1(CC)cc(C(=O)NCC(C23CCC(CC2)C3)NC(=O)C=C2CCC2)cc(C)c1 72254,c1(OC)c(C)cnc(C(c2nnnn2C)NC(c2cncc(Br)c2)C2CC2)c1C 72255,c1(C(N2C(CNC(C3C(=C)CC3)=O)CC(O)C2)=O)cc2c(CC)cccc2[nH]1 72256,C=CCCCC(C(=O)NCCC(F)(F)Cl)NC(C1CNC(=O)N1)=O 72257,C(=O)(C(CC(C)C)NC(C1CC(O)C1)=O)NC(COC)CCO 72258,CCCCCCC(CC)C(=O)N1CCCCNC(=O)CC1 72259,c1(C(N2CC(NC(=O)COCc3ccccn3)C2)=O)ccnnc1S 72260,CC(=O)CCCC(=O)NC1CS(=O)(=O)CC1NC(=O)C1=CCC1 72261,c1(C(=O)NC2C(NC(C(C)CC3CC3)=O)CCC2)c[nH]nc1S(N)(=O)=O 72262,C(N=c1ccnc(NC2CS(=O)(=O)CC2N2CCCCC2)[nH]1)c1c(C)coc1C 72263,c1(OC(C)C(N2CCCCC2COC(c2ncn(C)n2)=O)=O)ccc(Cl)cc1 72264,C1(C(N(CCNC(CSCC(C)C)=O)C(C)C)=O)CCC(C2CCCC2)O1 72265,C1(C(C)C)CCC(C)CC1CNC(=O)C(=O)Nc1cc(-c2ccccc2)on1 72266,Cc1cc(C(N2CCN(C(=O)CC3(N(C)C)CCC3)C(C3CC3)C2)=O)cc(C)n1 72267,C1(C)(NC(C(c2csnc2C)N(C(C)C(C)(C)C)CC)=O)CC(C(=O)OC)C1 72268,N1(C(c2c(C)c[nH]c2)=O)CC(CC(=O)NC2CC3C=CC2C3)C2(CC2)C1 72269,N1(C(C(C(C)(C)C)O)=O)CCCC2(CCN(C(c3cc(F)c(F)cc3F)=O)C2)C1 72270,c1(C(=O)NCC(C2CCC2)Nc2nccc(C3CC3)n2)ccc2ocnc2c1 72271,C(=O)(CC(F)(F)C(C)(F)F)N1CCCC(C)(CNC(C=CCCC)=O)C1 72272,C1(NC(c2cc(C)n(CC#C)c2C)=O)CCC2(CC1)CC2NC(=O)CC(C)(C)O 72273,N1(C(C(C=C)CC)=O)CC2(CO)CC1(C(=O)NCC1CCCN1C)C2 72274,N1(C(c2cnn(CC)c2C)=O)CC(CNC(=O)CC(F)(F)Cl)CC12CCC2 72275,Cn1nccc1CC1CCN(C(c2cc(C(C)F)on2)C(=O)NC2CCOC2)C1 72276,CCC(C)C(=O)NC1CC(O)C1CC(=O)N(C(CC)CO)C 72277,N1(C(CSCCC#N)=O)CCC2(CC1)CN(C(c1ccccn1)=O)CC2CO 72278,c1(SC)ncc(N)c(C(=O)N(CCNC(=O)CCc2nc[nH]n2)C2CC2)n1 72279,C1(NC(C(CSC)O)=O)CN(C(c2csc(Cl)n2)=O)CC2(CC2)C1 72280,N1(C(c2ccc(OC)c(Br)c2)=O)CC(NC(C)=O)C(C2CC2)C1 72281,N1(C(=O)NC2CCc3ncccc3C2)CCS(=O)(=O)c2ncc(Br)cc21 72282,C1(n2cc(CC(C)(C)C)nn2)CCC(C(N2CCC(n3cncn3)C2)=O)CC1 72283,C(=O)(CCC(C)S(C)(=O)=O)NC1CN(C(c2ncn(CC)n2)=O)CC(O)CC1 72284,C1(C(N2CCC(COCC)C2)=O)CC12CCN(C(C1(O)COC1)=O)CC2 72285,n1(CCC(=O)NC2CN(C(C3(C4CCCO4)CC3)=O)C2)c(=O)oc2cc(Cl)ccc12 72286,N1(C(c2c(C)nn(C)c2)=O)CC2(CC(C(=O)NCC3(CN(C)C)CCC3)CO2)C1 72287,C1(NC(C(C#C)(C)C)=O)CC2CCC(C1C)N2C(c1nc(Cl)sc1Cl)=O 72288,C12(C(=O)NC3CCC(C(=O)OC)C3)CCCC1CCN2C(=O)C(C)=CC(C)(C)C 72289,c1(OC)ccc(C(=O)NC2CCCC2CNC(C)=O)c(NC(=O)C(C)(C)CF)c1 72290,C1(CC)(NC(=O)CCSC(F)(F)F)CCN(C(c2cc(C(F)F)nn2C)=O)CC1 72291,c1(C(=O)NC2(C)CCN(C(c3c(C)cc(Cl)cc3)=O)C2)cnc2c(c1)nnn2C 72292,c1(OC)cncnc1C(=O)NCC(c1ccc(C)cc1)NC(=O)CN(C)C(C)=O 72293,Cc1ccc(OCCC(=O)NC2CN(C(=O)CC3CCC(C)(C)CO3)C2)c(Cl)c1 72294,C1(C2CCN(C(=O)CNC=O)C2)(NC(C(C)OCCN(C)C)=O)CC1 72295,CCC(CCCC(F)(F)F)NC(=O)C(=O)NC1CCS(=O)(=O)CC1 72296,c1(N2CC3C(C)C3C2)nc2c(c(=NC3CCc4nn[nH]c4C3)[nH]1)COC2 72297,C(=O)(C1=CCC(NC(=O)Cc2ccoc2)C1)Nc1cccc(C(C)F)c1 72298,CC(C)(F)C(=O)NC1CCCC1CNC(c1cn(CCF)nn1)=O 72299,c1(-n2cc(CCC3N(C(CC)=O)CCC3)nn2)ccc(F)cc1Br 72300,Cc1ccc(OCC(=O)NCC2CCC=CCC2)c(Br)c1 72301,C(C(=O)NCCC(O)CNC(=O)CCCN(C)C)(C(C)C)(C(C)C)NC(C)=O 72302,C=CCCCCCCCCC(C(=O)NCCC)N1C2CCCC1CC(O)C2 72303,Cc1cc(=NC2CCC(N3CCOCC3)C2)[nH]c(=NCC2COC(C)(C)C2)[nH]1 72304,CC(C)C(CC(=O)NC1(CCNC(=O)CCc2ncc[nH]2)CC1)C(C)C 72305,C(c1cccc(Cl)c1Cl)=CCN1CCCC(C(=O)OCC)C1c1nn[nH]n1 72306,C1(CNC(C(C(C)C)OC)=O)CCN(C(c2ccc(Cl)c(O)c2)=O)C12CC2 72307,CC1CN(C(C)C(=O)Nc2ccccc2C(N)=O)CCC1O 72308,c1(C(=O)NCC2CN(C(CCCC)=O)C(C)(C)C2)cc(C)cc([N+](=O)[O-])c1N 72309,c1(CC(=O)OC)cccc(C(=O)NC(CNC(=O)CCNC(N)=O)CC)c1 72310,c1(C(N2CCN(c3ccnnc3)CC2)C(=O)NC(CC)C)cc(C)oc1C 72311,c1(OC(C)C(=O)NC2CCC(F)(CNC(C34CC(CO3)C4)=O)C2)cccc(F)c1 72312,c1(C(=O)NC(C2CN(C(CCCOCC)=O)C2)C)cncc(C)c1C 72313,C1(OC)CC2(C1)CN(C(=O)Nc1nscc1SC)C2 72314,Cc1cccc(CNC(c2ccc(-n3cncn3)nc2)=O)c1C 72315,C(CCCCCN=c1[nH]c(Cl)nc2cc(C)sc12)NC(CC(CC)O)=O 72316,N1(Cc2ccc(OCC)c(O)c2)CCC2(CC1)CC(C(=O)NC(C)CC)CO2 72317,CCCC(C(O)C(=O)NCCCc1cccnc1)NC(C1CC(O)C1)=O 72318,C1(C(=O)NC2(C(=O)NCCC(C=C)(C)C)CCCC2)CC(=O)NC(=O)C1 72319,C12CCCC(C1)NC2=O.CCC(C(=O)N1CC(N(C)C)C1)N(CC)CC 72320,N1(C(CCc2ncn(C)c2)=O)CC2(C1)CN(C(=O)C(O)CCc1ccc[nH]1)C2 72321,c1(OC)ccc([N+](=O)[O-])c(N2CC(NC(=O)C(C)CO)CC3(CC3)C2)c1F 72322,C(c1ccccc1)(C(F)(F)F)=CC(=O)N(CCNC(C1CC(F)(CO)C1)=O)CC 72323,C(CCCOC)(C(=O)N1CC(c2nn[nH]n2)C1)NC(CCC=C)=O 72324,N1(C(C(C)OCCC(C)C)=O)CCCC1C=CC(N1CC(O)(CCO)C1)=O 72325,N1(C(C(C)Cc2ccccn2)=O)CCN(CCNC(=O)CC2CCCCC2)CC1 72326,n1(CCC(=O)NCCC(C(C)C)NC(C(C)SCCCC)=O)cnc(C)cc1=O 72327,c1(C(=O)NCC2CCN(C(C3(CF)CC3(F)F)=O)C2)ccc(C(F)F)cc1 72328,C12(CNC(C(C3CCC3)OC)=O)CCC(CC1)N2C(=O)CSC(C)C 72329,c1(OCC)ccc(-c2nc(C3CCCN(C4CC4)C3)n(-c3ncnn3C)n2)cc1 72330,c1(CC(=O)N(C2CN(C(c3c(C)[nH]cc3)=O)CC2F)C)cccc2c1OCCO2 72331,C(CCCCC(=O)NCCCC1(C)CC1)NC(C(C)CN(C)C)=O 72332,Cc1ccc(C(=O)NCC(C2CCC2)NC(=O)CN2CCN(C)CC2)cc1 72333,CC1(CNC(=O)C(c2cc(F)ccc2F)=O)CCCN(C(C2CCSC2)=O)C1 72334,N1(C(C(CC2CCC2)NC(CC2CCC(C)O2)=O)=O)CCN(C)C(=O)C1 72335,c1(CNC(c2c(C)con2)=O)ccc2c(c1)CCC2NC(=O)C(O)CCC(C)C 72336,C(=O)(C(C)CC(C)(F)F)N1CCC(N(C(=O)Cn2nc(C)n(C)c2=O)CC)CC1 72337,C1(C(=O)NC2(C)CCN(C(c3cccc(C(=O)NC)n3)=O)C2)CC(O)C12CCC2 72338,c1(C(=O)NC(C)CC(C)NC(c2cnc[nH]2)=O)nn(C)cc1Br 72339,c1(C(N2CCCC(CCC=C)C2)=O)coc2c1CN(C(=O)CC1CCCN1C)C2 72340,c1(CNC(C(=O)NCC(CC)Oc2cccc(C)c2)=O)ncccc1C 72341,Cc1c(C(=O)N(C)CCNC(C2(C(=O)OC(C)(C)C)CCC2)=O)nnn1C 72342,C(=O)(C(C)CCC(C)(C)C)NC(CCCNC(c1ccc(SCC)nc1)=O)(C)C 72343,C1(C)(C(=O)NCC2(F)CCC(CNC(c3c(C)cncc3)=O)C2)CCN(C)C1=O 72344,C1(COC)(CNC(=O)CC2CC2C)CCCN1C(=O)CCSC 72345,c1(C(=O)NC2CC3(C2)CN(C(C24CC(F)C2C4)=O)C3)cccc2nonc12 72346,c1(CC)cccc(OCC(=O)NCC2CN(C(c3nccc(C)n3)=O)CC2O)c1 72347,C=CC(C)(CCOC)C(=O)NCCN(C(=O)C(c1c(C)cccc1C)O)CCC 72348,c1(SCC)cc(C(=O)NC(C)CNC(C2C(C)C2C)=O)ccn1 72349,c1(CNC(c2cn(CCNC(CCC(C)N(C)C)=O)nc2)=O)c(F)cncc1F 72350,N1(C(COC2CC(NC(c3ccc(C)c(O)c3)=O)C2)=O)CCC2(CCCO2)C1 72351,c1(C(=O)NCCCC(C)NC(C2(C)C(CC)CCC2)=O)c(Cl)ccnc1F 72352,c1(CC(=O)NC(c2ccccc2F)CNC(C(C)SC(C)C)=O)ccccc1Cl 72353,O=C1CC(Cc2cccc(NC(c3csc(Cc4ccccc4)n3)=O)c2)C(=O)N1 72354,C(=O)(C(C)C(F)(F)C(F)F)NC12C(CN(C(Cc3nc(C)sc3)=O)C1)C2 72355,CN1C(=O)CSC1=CC(=O)NCC1CC2CCC(C1)N2C(c1ccc(Cl)cn1)=O 72356,C1(NC(c2c(C)cc(CNC(=O)CC3(O)CCOC3)o2)=O)CCn2nnnc2C1 72357,C1(C(=O)NC2(C3CCCN3C(=O)C=Cc3cc[nH]n3)CC2)CCCC2(C1)CC2(F)F 72358,N1(CC)N=C(C(=O)NCCCCNC(C2CCC(c3cc[nH]n3)O2)=O)CCC1=O 72359,c1(C(N(CCC(=O)NC2CCCOC2)CCO)=O)n[nH]c2c1CCC2 72360,C12(C(=O)NC3C(CNC(Cc4nnc(C)o4)=O)CCC3)CC3CC1C2C3 72361,N1(C(C(C2CCCC2)OCC)=O)CC(NC(=O)C=CC=C(Cl)Cl)C2(CC2)C1 72362,C12CC3CCC(C1)N3N2CC#N.c1cnc(N)c(Cl)c1.n1(CC)ccc(Br)cc1=O 72363,N1(C(CC=C=C)=O)CCN(C(c2cn(-c3cccc(Cl)n3)nn2)=O)C(COC)C1 72364,C1(NC(Cn2c(C)nc(C)n2)=O)CN(C(c2n[nH]c(C)c2F)=O)CC1C1CC1 72365,C1(Nc2c(OC)cc(CC3CCCOC3)cc2)CCC2(CCCC2)C(O)C1 72366,c1(C(=O)OC)nc(=NCC(C)CNC(C2(C3CCOCC3)CC2)=O)c(F)c(Cl)[nH]1 72367,C1(NC(=O)CC2CCCO2)CCC12CN(C(=O)CCSc1ccccc1F)C2 72368,c1(C(N(C2CCN(Cc3ccc(Br)cc3Cl)C2)C)=O)ccc2cccc(Br)c2n1 72369,N1(C(c2nccc(N)c2)=O)CCC2(CC1)CC2CNC(=O)CNC(=O)C1CC1 72370,c1(N2CC(C(N(C)CC3CCN(C(C(C)O)=O)C3)=O)C2)ncc(F)cn1 72371,N1(C(CC(C)(C)CNC(C2CC23CCC3)=O)=O)CC2CC(F)CC2C1 72372,C(=O)(C(O)CCC(C)C)N1C(CNC(C2C(OC)CCCC2)=O)CC2CC21 72373,C1(C2(O)CCOCC2)(C(N2C3CC(NC(C4CC(C)(C)C4)=O)CC2CC3)=O)CC1 72374,CCCN=C(NCC1CN(C(C)=O)C1)N1CCC2(C1)CC2(F)F 72375,c1(C(=O)NC2C(NC(CC(C)CF)=O)CCCC2)cc2c(Cl)ccnc2s1 72376,N1(C(CCCCOC)=O)CC2CCN(C(=O)CC3(N(C)C)COC3)C2C1 72377,C=CCC(C(=O)N1CCOC(C(=O)NCC(C)(C)SC)C1)OC 72378,c1(OC(c2ccccc2)C(=O)NCC2CC3CC2C3)cc(F)ccc1F 72379,n1(C(C)(C)C)ncc2c1CCCC2NC(=O)C(N1C2CCC1COC2)=O 72380,c1(CNC(C2CC(SC)C2)=O)cc(C(=O)NCCOC(C)(C)COC)co1 72381,C(C1c2ccsc2CCN1C(=O)C=C1CCC1)NC(C1CC2CCC2C1)=O 72382,N1(C(C2(CC#C)CCCO2)=O)CCC2C(C1)CN2C(=O)CCc1nc(C)c(C)o1 72383,N1(C(C2OCCN(C(C)=O)C2)=O)CCC(O)C(NC(=O)CN2CCOCC2)C1 72384,c1(C(=O)NC(C(C(=O)NCc2cc(OC)no2)(C)C)C)nccc2[nH]ccc12 72385,N1(C2C(CC)CN(C(=O)C(S)C=C)CC2)CC(=O)N2CCc3ccccc3C2C1 72386,N#Cc1c(O)csc1NC(C1CCCCN1CCO)=O.c1(CN)ccccc1O 72387,c1(C(N(CCOC)CCNC(C2(C(F)(F)F)CC2)=O)=O)cc([N+](=O)[O-])c[nH]1 72388,N1(C(C(COCC)F)=O)CCCC(C2CC2NC(=O)OC)C1.C12(CC1)C(=O)N2 72389,c1(NC(N2C(CC(=O)Nc3cccc(Cl)c3Cl)CCC2)=O)cnnc(O)c1Cl 72390,CC1(C(=O)NC2(CCNC(C3CCC(C(F)(F)F)C3)=O)CCCC2)CCCCC1 72391,C(=O)(C1OCCc2ccccc21)NCC1N(C(C(C)c2cccs2)=O)CCC1C 72392,c1(C(N2C(C)CCN(C(=O)C=Cc3cc[nH]n3)CC2)=O)ccc2c(c1)CCCC2 72393,C(C)(C)(CCC(=O)N1CCCC(C)C1CNC(=O)CN1CC2CC2C1)OC 72394,c1(OC)ncnc(C(N2CCC(C)(CCNC(C3CC3(F)F)=O)C2)=O)c1F 72395,C1(NC(c2cnn(CC(F)F)c2)=O)CC(NC(=O)C2CC2)C12CCC2 72396,N1(C(=O)NC(C2(C)CCN2OC(C)(C)C)C(C)C)CCC(C2CCO2)CC1 72397,C(=O)(C(C(C)C)C1CCC1)N(C(c1ccccc1)CNC(C(C)(C)OC)=O)C 72398,c1(C(N2CCC(NC(=O)C(c3ccc(Cl)cc3)(F)F)C2)=O)cnn2ccsc12 72399,C1(C2CCN(C(C3CCC4(CC3)CC4)=O)C2)(NC(C(C)OCOC)=O)CC1 72400,c1(C(=O)NCC(CN(C(C2C(C)C2C)=O)C)C)c[nH]c2nccc(Cl)c12 72401,c1(C(N(C2CN(C(C3ON=C(C)C3)=O)CC23CC3)C)=O)n[nH]c2c1CN(C)CC2 72402,C1(CC(=O)N(c2nccs2)C)OCC2CN(C(c3cnc(O)c(Br)c3)=O)CCC12 72403,N1(C(C2CC(C#C)(O)C2)=O)CC(C)N(C(c2cnn(CC)c2C)=O)CC1C 72404,C(=O)(C(F)(CNC(=O)OC)C(C)C)NC1C(NC(CCN(CCC)C)=O)CCC1 72405,Cc1nc(C(=O)C(=O)NCC(CNC(=O)CC2CCOC2)CO)cs1 72406,C#CCCC(N)C(=O)NCCCN1CCN(c2cccc(C)n2)CC1 72407,C1(CNC(c2c(C)nco2)=O)CN(C(c2cc(C#N)c[nH]2)=O)CCC1C 72408,c1(C(=O)NC2(C)CCCN(C(C(CC)(C)O)=O)C2)cccn2c(C)nnc12 72409,C=CC1(C(=O)NCC(O)CC(F)(F)F)CCN(C(C2CCC(OC)CC2)=O)C1 72410,C(=O)(C1=CC2CCCCCC12)NC1CC(F)(CNC(CCCCC(C)(C)C)=O)C1 72411,C1(OC)(CNC(C2(C(F)(F)F)CC2)=O)CCN(C(C2(C)CC3CC3C2)=O)CC1 72412,CC(C)CC(C(=O)N(C)Cc1ccncc1F)ONC(=O)COC1CCCCC1 72413,C1(=O)CCC(C)(C)N1.c1(OC)cc(CNC(=O)CN(C)C)ncn1 72414,c1(C(C)C(=O)NCCNC(=O)CNS(=O)(=O)N(C)C)ccc2c(c1)OCCO2 72415,C#CC1(NC(C2CCCCN2C(=O)C=CC=CCC)=O)CCC(C)(C)C1 72416,c1(C(=O)NC2C(CC(=O)NCC3OCCN(C)C3)CCCC2)cnc2n1CCC2 72417,CCC(CN(CC(N=[N+]=[N-])C(=O)OC)CCN)(CC)CC 72418,C#Cc1ccccc1CC(=O)NCC(O)CC(N1CCC2(CSC2)C1)=O 72419,C1(C(N2CCCc3n[nH]cc32)=O)CC2(C1)CS(=O)(=O)C2 72420,N1(C(c2c(CC)nn[nH]2)=O)CC(C2CCCN(C(=O)C(C(C)C)C(C)C)C2)C1 72421,C12(CNC(c3c(C)nccn3)=O)CCC(CN(C(=O)Cn3cnnc3O)C1)C2 72422,c1(CN2CCC(CC(=O)Nc3c(C(N)=O)occ3)C2)cc(O)ccc1F 72423,N1(C(C(=O)NCC)=O)C(C(=O)Nc2cc(C)nn2C(C)C)C2CC(O)C1C2 72424,c1(C(=O)NC2C(NC(COCCN(C)C)=O)CCC2)cc2c(nn1)CCC2 72425,Cn1ncc2c1CC(NC(=O)Nc1ccnn1C1CC1(F)F)CC2 72426,C1(NC(c2c(C)nco2)=O)CCCCC1NC(=O)CC1CC=CCC1 72427,CC1CN(C(C23CC(C2)S(=O)(=O)C3)=O)CCC1NC(C1CC1C1CCCC1)=O 72428,c1(C(C)O)ccc(C(=O)NC2CN(C(C3CCN3C3CCCC3)=O)C2)cc1 72429,c1(CSC)ccc(C(=O)NC2CCCC(N(C(=O)C(F)(F)C3CC3)C)C2)cc1 72430,N1(C(C(c2ccccc2)C)=O)CC(O)CC1C(c1ncccn1)=O 72431,C1(NC(C(C)OCC)=O)CCCCN(C(c2nc(Br)sc2Cl)=O)C1 72432,C1(C(N2CC(CNC(=O)CC(C)(C)C3CC3)C2)=O)(CC)CCCC1O 72433,Cc1cc(C(=O)NCCC2CC(NC(c3[nH]cnc3C#N)=O)C2)cc(C)c1Cl 72434,N1(C(C(CC(N)=O)NC(C2C(C)N(C)CC2)=O)=O)CCOC2C(O)CC12 72435,C12(CNC(CCCCC)=O)CCCC1N(c1[nH]cnc3nc(Cl)cc1-3)CCC2 72436,n1(CC(=O)NCC(C2CCCCC2)NC(C(CC)OC)=O)ncc(Cl)c1C 72437,c1(C(=O)NC2(C)CC(NC(c3c(C)cccc3C)=O)C2)cnc2sc(C)c(C)n12 72438,CC1(C)CN(C(=O)COc2ccccc2)CCC1NC(C1CCc2nn[nH]c2C1)=O 72439,N1(C(C(=O)NCC(CC)NC(CCN(CCCCC)CC)=O)C)CCOCC1 72440,N1(C(COCCC(C)C)=O)CCN(C(=O)CCn2cncn2)CC2CCCCC12 72441,CCC(C)CCCCC(=O)NC1(C2CCN(c3ncc(C)c(C)n3)C2)CC1 72442,c1(C(c2nnnn2C2CCCC2)NC2(CC)COC2)cc(F)nc(F)c1F 72443,S(=O)(=O)(c1ccc2nc(Cl)ccc2c1)N1CC2(CC(CC(=O)OC(C)(C)C)C2)C1 72444,c1(C(C(=O)NC2CCOCC2)N(C)Cc2cnc(CC)[nH]2)cnc(C)n1C 72445,c1(C(=O)NCCC(=C)CNC(c2oc(C(F)F)cc2C)=O)cnc(N)c(N)c1 72446,c1(C(=O)NC)ccc(=NC2CCN(C3CCN(Cc4ccccc4)C3=O)C2)[nH]n1 72447,c1(C(N2CC(OCCNC(C3C(C)CN(C)C3)=O)C2)=O)cc(C#N)ccc1F 72448,c1(SC)nc(O)nc(C)c1C(N1CC(C(C)NC(=O)CCCc2ccsc2)C1)=O 72449,N1(C(C(CCOC)C)=O)CC2CCC1C(CNC(c1csc(Br)n1)=O)C2 72450,C1(CNC(=O)Cc2cscn2)C2CN(CC34CC(c5ccccc5)(C3)C4)CC12 72451,c1(OC)ccc(C=CC(N2CC(CN(C(=O)CCC#N)C)C3(CC3)C2)=O)cc1 72452,N1(C(C)=O)CC2(C1)CN(C(c1cnc(N3CC(CC(=O)OC)C3)c(Cl)c1)=O)C2 72453,C(CCC(C)CC(=O)N1CCN(C(c2ocnc2C(F)F)=O)CC1CO)=C(C)C 72454,CC(C)C(Cn1cc(CO)nn1)C(=O)NC1(C(N)=O)CC1.C12CCCN(CC1)C2 72455,CCCCCCC(C)CC(=O)N1CCN(C(=O)C(C2CCCC2)C(=O)NC)C(C)C1 72456,c1(C(=O)NCCCN(C(C)C(C)C(=O)NC)CC)ccn2ccccc12 72457,C(C1CCOCC1)=CC(=O)NC(CNC(c1n(C(C)C)nnc1)=O)(C)C 72458,C1(CCC(C)(C)NC(C(=O)NC(C)C)=O)CN(C(C2(CO)CC2(F)F)=O)CCO1 72459,c12cn(nn1)CC(=O)OC2.NC(=O)COCCCF 72460,c1(CNC(C(C2CN(C(C3C(OCC)C3)=O)C2)OC)=O)cc(C)cnc1O 72461,C1(CS(=O)(=O)N(C)CC2CNCCC2)CCC(C(F)(F)F)O1 72462,c1(OCC)ccc(C(=O)NCC(CO)NC(C2CCC2CF)=O)cc1 72463,S(=O)(=O)(c1ccc(N2CCc3noc(N)c3C2)cc1Br)NCc1c(C)ncn1C 72464,C12(OC)CCCC(C(=O)NC(CNC(=O)C3=C(Cl)CCC3)CC(C)C)(CC1)C2 72465,c1(C(=O)NC(C2CCN(C(C3CS(=O)(=O)C3)=O)CC2)(C)C)cc(N(C)C)ccn1 72466,C1(NCC2CN(C(C3(CCC#N)CCC3)=O)C2)CS(=O)(=O)C1.c1(C)nn[nH]n1 72467,C1(C2CCCN(C(=O)C3=CCCCC3)C2)(NC(C2C3CCCOC23)=O)CC1 72468,c1(C(=O)NCCCC(=O)NCCC(F)(F)CO)cccc2nccn12 72469,C#Cc1ccc(C(=O)NCC(Cc2ccccc2)NC(=O)C(O)C2CCC2)cn1 72470,c1(C(=O)NC2CCC(NC(CC3(CSC)CC3)=O)C2)ccc(C)c(C#N)c1 72471,CC1CN(C(C2CC3C(C2)C3(C)C)=O)CCC1N(C(=O)CCN1CCOCC1)C 72472,C=CCC(C(=O)NCC1CCC(NC(=O)CCc2ccc(C#N)cc2)C1)C(C)C 72473,c1(C(=O)NC2(CN(C)C(C3(C)CC(C)(C)C3)=O)CC2)cccc(CS(N)(=O)=O)c1 72474,c1(C(=O)NCCN(CC(C)O)C(c2c(C)oc(Cl)n2)=O)c[nH]c2ccc(Cl)cc12 72475,c1(C(=O)NCCN(C2CC2)Cc2c(C)occ2)ccc(-c2ccccc2)cc1 72476,c1(C(=O)NC2CCCC2Cn2cc(CCO)nn2)ncccc1C(F)F 72477,C1(CNC(=O)CCC2CCCC2)CN(C(c2ccc(F)o2)=O)C2(CCC2)C1 72478,c1(C(=O)NC(CC(=O)OCC)c2ccncc2)cccc(CCC(=O)NC)c1 72479,CCCCC(O)CC(=O)NC1C2CCC(C2)C1C(=O)N(CC(C)OC)CC 72480,N1(C(c2cc(C)nn2C)=O)Cc2ccccc2C(CNC(c2nccn2C)=O)C1 72481,C1(C(=O)NCCc2ccncc2)CN(C(=O)Nc2cnccc2Br)CC(F)(F)C1 72482,CC1CCN(C(=O)C(O)C2CCCC2)C(C)C1NC(=O)COCCO 72483,c1(N2CCC(OCCSC)C2)cc(N2CCC(c3cncn3C)C2)nc(C)n1 72484,c1(C(C)NCC(c2c(OC)cccc2)N(C)C)cc2cccc(F)c2o1 72485,N1(C(CCOC)=O)CC(NC(=O)Cc2cccc(C(C)(C)C)c2)C(C)(C)C1 72486,C1(c2n(CCOCC)nnn2)(NCCc2cc(C)cc(C)c2)CCC(C)(C#N)C1 72487,c1(C(=O)NC(CNC(C2(OC)CCCOC2)=O)C(C)C)cc(C)ccc1F 72488,CC1CN(C(c2sccc2CN(C)C)=O)CC1CCNC(c1snc(Cl)c1Cl)=O 72489,C1(OC)CCC2(CCN(C(=O)NC3CCCCC3C(=O)Nc3ccccc3)C2)C1 72490,C1(NC(Cc2scc(C)c2)=O)CC=C(C(=O)NC2C(C)CCC2C)C1 72491,CC1(C#CC(=O)NC2CC2CNC(c2c(F)c(F)cc(F)c2F)=O)CCCO1 72492,c1(C(C)(C)C)ncc(C(=O)NCC2(O)CN(C(=O)CCCc3ccccc3)C2)s1 72493,C1(CNC(CC2C(C)=NNC2=O)=O)CCN(C(=O)Cc2cnsc2)C12CC2 72494,S(=O)(=O)(c1c[nH]ccc1=NCC1CCC(CO)CC1)CN1CCC(SC)C1 72495,C(=O)(C(C)(C)C(=O)NC1CCC(C)(CNC(C2CC=CC2)=O)C1)N(C)C 72496,N1(C(CCCOC)=O)CCCC2(C1)C(NC(c1nc(C)ncc1Cl)=O)CCN2C 72497,C(=O)(CC(C)(C)O)NCCCC(C)NC(=O)C(F)(F)c1cncs1 72498,c1(CCNC(CNC(c2c(CCC)n[nH]c2)=O)=O)cccc(C)c1 72499,Cc1cc(C(C)(C)C(=O)N(CC(=O)NC(C)(C)C)CCO)cs1 72500,C1(NC(c2cc(C(C)(C)C)on2)=O)CCCC(NC(=O)CS(N)(=O)=O)C1 72501,c1(C(=O)NCC(CNC(C(CN(C)C)(F)F)=O)CO)cc2nccnc2cc1F 72502,N1(C(C(C)n2cccc2)=O)CCC2CCN(C(=O)C#CC3CC3)CC12 72503,C1(NC(CCC2OCC(C(=O)OC)C2)=O)COCCC1NC(=O)CN1CC2CC2C1 72504,Cc1csc2ncc(C(=O)NCCOCCNC(=O)CCNC(N)=O)c(=O)n12 72505,c1(-n2cc(SCC3OCCN(C(C(C(=O)OC)C)=O)C3)nn2)cc(Cl)c(Cl)c(Cl)c1 72506,C1(NC(C(C2CCCC2)OC)=O)C2CCC1N(C(=O)Cc1cn(C)nc1C)C2 72507,C(=O)(CC(C)(CN(C)C)C(F)(F)F)NC1C2CN(C(C(CC)=CC)=O)C1C2 72508,C(=O)(C1=COc2ccccc2O1)NC1CC(C)(C)CN(C(c2ccoc2)=O)CC1 72509,Cc1sc(C(N2CCCC(CNC(c3cnn(C4CCOC4)n3)=O)C2)=O)nc1O 72510,CCC(O)C(=O)NC1(CNC(=O)Cc2cncn2C)CCC1 72511,Cc1cc(=O)c(C(=O)NCC2CCN2C(=O)Cn2cnc(C(F)(F)F)n2)cn1C 72512,CC1CC(C(=O)COC(N2CC(CN(C)C(=O)C3CC3)C2)=O)CO1 72513,C(=O)(C(CC(F)F)c1ccccc1)Nc1cccc(NC(c2n(C)nnc2)=O)c1 72514,C(=O)(C1=CC(O)CCC1)NC(C)CCNC(c1c(Cl)csc1Cl)=O 72515,c1(CN(C(C(=O)NC)c2ccsc2)CC)ccc(Br)s1 72516,C1(NC(C2(OCC)CCCC2)=O)CC2CCC1N(C(c1cc(C)c(C)nn1)=O)C2 72517,N(C(=NCC1COCCO1)NCc1ccc(C2CC2)cc1)CCSC 72518,CCC(CC(=O)N(C)CC1CC2(CC2)C1)C(C)C 72519,N1(C(C)CNC(c2coc(CO)c2)=O)CCN(C(C2CCCC2(F)F)=O)CC1 72520,CCCC(C(=O)NC(C)Cn1cccn1)NC(=O)CN(C)CC1CCOC1 72521,N1(C(c2c(C)n(CCO)nc2)=O)CC2CC(C1)CN(C(C1CC(C)CO1)=O)C2 72522,N1(C(C=CCCC)=O)C2CCC1CC(NC(=O)Cn1ccc(Br)n1)C2 72523,N1(C(C(SC)SC)=O)CCCC(CNC(C2(C)CCCN2C)=O)C1 72524,C1(C)(C(=O)NC2CN(C(COC3(C)CCC3)=O)C(CO)C2)CC2(CCC2)C1 72525,O=C(CC1=CCCCC1)NCC12CCC1CN(C(C1CC(=O)NC(=O)N1)=O)C2 72526,C(CCCC(C)(C)NC(C1CCC(NC(C)=O)CC1)=O)NC(C(C=C=C)C)=O 72527,C(C(=O)NC(C(=O)NC1CC=CC1)C1CCC1)(C(C)C)OC 72528,c1(-c2nc(CSc3[nH]n(CC(C)C)c(=O)c3)on2)ccc2c(c1)COC2 72529,CC1CN(C(c2ccccc2C2(C)CC2)=O)CCN1C(=O)COc1ccccc1 72530,Cn1nc(CC(N2CC3CC3(NC(C34CC(F)(C3)C4)=O)C2)=O)cc1C(F)(F)F 72531,N1(C(c2cccc(C)c2C)=O)CCC2CN(C(c3ccc(=N)[nH]c3Cl)=O)CC12 72532,N1(C(CCC(CC)C)=O)CCOC2(CCN(C(=O)C(C)C3CCC3)CC2)C1 72533,C(=O)(C(CC)C(=O)OCC)N1CCC(C(C)(C)NC(c2n(CC#C)cnn2)=O)C1 72534,C(CCCCCNC(=O)C1CC1)N(C(C)C)CCN(C)C(c1ccncc1Cl)=O 72535,c1(COC)sccc1C(=O)N(CC=CC=C(C)C)Cc1cn(C2COC2)nn1 72536,Cc1c(CCC(=O)NCCC2CCC(NC(=O)CC3CCOC3)C2)cnn1C 72537,C=C1CCN(C(=O)CC2CCC2)C(C(=O)NC2CCN(C(C)=O)C2)C1 72538,C1(CNC(Cc2cc(C)sc2C)=O)CC(C)(C)CCC1NC(=O)CCF 72539,N1(C(C(CN(C)C)N(C)C)=O)CCCC1(C)C(=O)NCCc1ccc(O)cn1 72540,N1(C(C2(OC)CCOC2)=O)CCN(C(=O)C=C(C2CC2)C2CC2)C(CC(F)F)C1 72541,c1(CN2CC(NC(CCc3c(C)ncs3)=O)(CO)C2)c(I)ccnc1Cl 72542,C1(NC(c2c(CC)ncs2)=O)CCN(C(c2cccc(C)c2)=O)CC(C)(C)C1 72543,S(=O)(=O)(c1cc(C(=O)OC)c(Cl)cc1Cl)N1C(C#C)C2CCC1C2 72544,N1(C(c2c(OCC#C)nccc2)=O)CCN(C(c2csc(C)n2)=O)C(CCO)C1 72545,C1(NC(CCc2ccc(C)s2)=O)CCCN(C(c2cc(C)n(C(F)F)n2)=O)CC1 72546,CCC(c1ccc(OC)cc1)=CC(=O)N(C)CCN(C)C(c1ccc(C)n1C)=O 72547,C=CCCC(C(=O)N1CC(CNC(c2ccc(N)cc2Cl)=O)C1)c1ccccc1 72548,C1(C2CCN(C(C3CCC4CC34)=O)CC2)N(Cc2ccns2)CC12CCC2 72549,N1(C(CCOc2c(C)cccc2)=O)CC(N=c2[nH]nc(C3CC3)s2)CC(C)(C)C1 72550,C(=O)(CCC(CC)CCC)NCC1C2CN(C(C3(C=C)CC3)=O)CC21 72551,c1(C(c2cncc(Br)c2)F)ccc(F)c(F)c1.CC12CCCN1C(=O)N2 72552,c1(C(C)C)nccn1CC(=O)NC1COCC1N1CCOCC1 72553,N1(C(c2c(C)nsc2)=O)CCCCC1C(=O)N.c1(COC(F)(F)F)cn(C2(C)CC2)nn1 72554,CC1(C)C(NC(=O)C(F)OC(F)(F)F)CCN1C(c1ncc(C(F)F)s1)=O 72555,c1(-c2ccc(-c3nnn(C)n3)cc2)n[nH]c2c1CN(C(=O)COC(=O)CC#N)C2 72556,N1(C2C(NC(=O)COCC3CCOC3)CCC2)CCN(C(=O)C=CCO)CC1 72557,c1(C(N(CCN2CCN(C(C(C)OC)=O)CC2)C)=O)cc2cccnc2[nH]1 72558,c1(OC)ccc(C(N2CCC(N(C(=O)C(O)P(C)(C)=O)C)C2)=O)c2ccoc12 72559,C(=O)(C1=CC(C)(CC)C1)N1C(COC)(CNC(=O)C(c2cccnc2)O)CCC1 72560,C(CC1CC1)(CN=c1ccc(Br)c(S(=O)(=O)NC2CC23CCC3)[nH]1)OC 72561,N1(C(c2c(CC)cns2)=O)CCCCC1C(=O)NCC1(O)CCCOC1 72562,C1(C(C)(C)C)C(NC(c2c[nH]nc2F)=O)CCN1C(=O)CCC1CCCCCC1 72563,C1(NC(C2C(=C)C2)=O)(CO)CN(C(c2coc(Br)c2)=O)C1 72564,N1(C(c2cncc3sccc23)=O)CCC2CCCC(C1)N2C(C1CCC1)=O 72565,c1(OC2(C(N3CC(CC(C)NC(C=CC)=O)C3)=O)CC2)ccccc1 72566,c1(C(=O)NCCC2CCN(C(c3cc(N(C)C)ncc3)=O)C2)c(F)cncc1Cl 72567,c1(C(N2CCC(C)C(CO)C2)=O)cc(P(C)(C)=O)cs1 72568,N1(C(C2C(C)C2)=O)CCN(C)C(C(=O)NCc2ccc(C(=O)OC(C)(C)C)cc2)C1 72569,C(=O)(CCCC(F)(F)F)NCCCCCCN(C(C(C)CC(F)F)=O)C 72570,c1(C(=O)NCC2(OC)CCN(C(=O)Cc3ccoc3)C2)cnc(C)nc1C 72571,N1(C(c2cc[nH]c2C2CCC2)=O)CC2CCC1CN2C(c1snnc1C1CC1)=O 72572,c1(C(=O)NC2C(NC(C(=O)NCC)=O)CC2)sc(C2CCOC2)nc1C.CC=O 72573,c1(C(N(CCCNC(c2cc(CC)sn2)=O)C(C)C)=O)ccn2cnnc2c1 72574,c1(C(=O)OC)cnc(=NCCCN(C(=O)CCOc2ccccc2)C)[nH]c1 72575,CC1CC(C(=O)NC2(C(=O)NC(CO)C(F)(F)F)CCOCC2)CCS1 72576,Cc1cc(C(=O)NC2CC(NC(c3ccccc3C3CC3)=O)C2)c(C)n1C 72577,c1(-c2n(C)c(SCc3ccc(Cl)c(N=[N+]=[N-])c3)nn2)cccc2c(Cl)ccnc12 72578,CC(CC(=O)NN1CCCC1C(=O)NCC1(CO)CC(C)(C)C1)C1CC1 72579,c1(NCC2(SC)CCCC2)ccnc(CNC(C2CC(F)(F)C2)CCO)n1 72580,N1(C(c2cc(CC)ncc2)=O)CC2(CCCC2NC(C2CC2F)=O)C1 72581,c1(CNC(CC2CCN(C(CNC(=O)OCC=C)=O)CC2)=O)c(C)cccc1C 72582,C(=O)(CC(C)C(=O)N1CCC(C(C)C(=O)NC2(C(F)(F)F)CCC2)C1)OCC 72583,C1(NC(c2cnnc(O)c2)=O)CN(C(=O)Cn2nnc(=O)[nH]2)CC1C1CC1 72584,n1(CC(=O)NC(C(C)(C)C)CNC(=O)C(C)(C)c2cnco2)cc(F)ccc1=O 72585,C1(C)(C(N2CCC(OCCNC(CCC(=C)C)=O)C2)=O)CCCNC1=O 72586,Cc1oc(C)c(C(=O)NCC2CC(CNC(=O)COCCN(C)C)CO2)c1C 72587,Cc1ncc(Br)c(N(C2CCCNC2)C(c2ccc(S)cc2)=O)n1 72588,C12(NC(=O)COC3CCC3)CC(C(=O)NCCc3ccon3)(C1)C2 72589,c1(-c2cnc(C)nc2)nc2c(s1)CCN(C(=O)C(F)F)C2 72590,C12(CNC(CCNC(COC)=O)=O)CCC1CCN2C(C1CCC1)=O 72591,CC(C(=O)N1CC(O)CC1Cn1cc(-c2ccc(Cl)c(Cl)c2)nn1)S(C)(=O)=O 72592,c1(C(=O)NC2(CN(C)C(c3ccnnc3O)=O)CC2)cccc(CC#N)c1 72593,N1(C(C(CC=CC)CC)=O)CC2CN(C(=O)C(c3ncc(Cl)n3C)(F)F)CC2C1 72594,C(=O)(C1CCc2cccnc21)N1CCN(C(C2C(c3c(C)occ3)C2)=O)CC1 72595,c1(CN2CCC(C)(C(N3C(CCCC)CCC3)=O)C2)ccc(C#CCO)cc1 72596,CCC(CN(C)C)CC(=O)NC1(CCC(=O)Nc2ccc(OC)c(C)c2)CCC1 72597,N1(C(C(C)OC(C)(C)C)=O)CCC(C2CC2)(NC(c2cnc(Br)s2)=O)C1 72598,N1(C(Cc2ccc(OC)c(O)c2)C)CC(CO)Oc2c(Br)cccc21 72599,c1(C(=O)NCC(CC=C)NC(c2ccnn2CC2CC2)=O)ccnc(C2CC2)c1 72600,C1(CC(=O)NCCCN(C(C2CCC(CC)O2)=O)C)NC(=O)CNC1=O 72601,C(CCN=c1[nH]c(=N)[nH]c(=NC(C)c2ccc(Br)c(C)c2)[nH]1)OC=C 72602,CCC(CC(C)C)C(=O)NCC1=CCN(C(C2CC3CCCC(C2)C3)=O)CC1 72603,CCC(C)(COC)C(=O)NC1CCC(CCC(=O)NCC2(F)CC2)C1 72604,C(=O)(C1=NOC2(CCOC2)C1)NCCN(C(c1n(C)ncc1)=O)C1CC1 72605,c1(CC(C)C)ccc(C(C)C(=O)NCC2(F)CN(Cc3ncccc3O)C2)cc1 72606,C1(C)(NC(C(CC2CC2)OC)=O)CCN(C(C2CCC(C)(C)OC2)=O)CC1 72607,c1(N(CC(C)C)CCNC(=O)CC2(C)CCCC2)nc2ccc(F)cc2s1 72608,C1(NC(c2nc(CNC(C(CC)CN(C)C)=O)oc2C)=O)CC(C)(OC)C1(C)C 72609,N1(C(=O)NC(C)CS(=O)(=O)N2CCCC2)CCN(CC(F)(F)F)C(C)C1 72610,N1(C(=O)Cn2cnnc2O)CCN(C(c2cnoc2-c2ccco2)=O)C2CC12 72611,CC(C(=O)NC1CC(NC(=O)Cn2nnc(C(C)(C)C)n2)C1)S(N)(=O)=O 72612,N1(C(C2CCC(NC(=O)CN3CCCC3=O)CO2)=O)CCCC2(CCOC2)C1 72613,c1(OC)ccccc1ON(CC(=O)NC1CC(CNC(c2nccs2)=O)C1)C 72614,CC1CCCCC1C(=O)NCCC1CCCN(C(=O)CSCC2CCCO2)C1 72615,C1(NC(CC(C)OC)=O)CCC(C(=O)NCC2(CCO)CCCC2)CC1 72616,C(CCCCCNC(=O)CSC(C)(C)C)N(C(=O)Cc1nncn1C)C 72617,CC(CN=c1nc2sccc2c(NCC(C)C2CC2)[nH]1)c1nccs1 72618,C1(NC(C2CCC(C)C2)=O)CN(C(=O)CCc2ccc(F)nc2)CC2(CC2)C1 72619,C(=O)(C(C)(CO)NC(=O)CCc1ccncc1)NCC(C)(C)OCCO 72620,C1(NC(CCN(CCC)C)=O)C2CCCN(C(C3CCSC3)=O)C2C1(C)C 72621,C1(NC(c2ccc(Cl)[nH]2)=O)CCC(CNC(c2ccnn2C2CCCC2)=O)C1 72622,c1(C(=O)NCC(C(C)C)NC(c2cn(C)[nH]c2=N)=O)ccc2ncnn2c1 72623,c1(CC(=O)NCC(CNC(CCC2CCN(C)CC2)=O)O)cccc(F)c1Cl 72624,N1(C(C=C(C)Cl)=O)CCC(C2CCOCC2)(CNC(C2CCCCNC2=O)=O)C1 72625,c1(C(N(C2CCN(C(=O)C(COC)COC)C2)CC)=O)nn(C)c(C)c1Cl 72626,c1(C(N(CCC)CCNC(=O)CC2CCCC(O)C2)=O)c(C)[nH]c(C)c1C 72627,S(=O)(=O)(c1ccccc1F)NCC1N(C(c2ccc(Cl)c(Br)c2)=O)CCC1 72628,c1(CC(=O)N(C2C3CCC2CNC3)c2cccc(Cl)c2)cc(F)cc(F)c1F 72629,C12(C(N(CC(=O)NCCCS(C)=O)CC)=O)CCCC1C2(F)F 72630,C1(CC(N2CC(OCCC(=O)NC(C(C)C)C3CC3)C2)=O)NC(=O)NC1=O 72631,C(=O)(CCP(C)(C)=O)N(C1CCCCN(C(=O)C(c2ccc(F)cc2F)=O)C1)C 72632,c1(C(=O)OCc2c(F)ccc(F)c2Br)cc(I)ccc1[N+](=O)[O-] 72633,n1(CCC)nnnc1C1(NCC(C2CC2)C2CC2)CC(C)C1 72634,N1(C(C2(C)CC(=C)C2)=O)CCC2CN(C(=O)CCCOC(C)=O)C2C1 72635,Cc1cccc(CCC(=O)NCC2CC2CNC(C2CCCS2(=O)=O)=O)c1 72636,N1(C(=O)CCc2ncc[nH]2)CC2CC1CN2C(C1CC1c1ccc(Cl)cc1)=O 72637,N1(C(CSSC)=O)CCC(CNC(=O)C=Cc2cccc(CO)c2)C(F)(F)CC1 72638,c1(C(=O)NCC2CCN(C(CCC3C(C)C3)=O)C2(C)C)ccc2c(c1)ncn2C 72639,Fc1cc2c(cc1Br)CN(c1nc(I)cs1)CC2 72640,c1(C(=O)NCCC(CC)(CC)NC(C(CC)OCC)=O)cc(C)nc(Cl)c1N 72641,Cn1cc(Br)cc1C(=O)NCC1(NC(=O)CNC(=O)C2CC2)CC1 72642,C(=O)(C(CNC(=O)C(O)C1CCCC1)CC(C)C)N1CC(N(CCC)CC)C1 72643,c1(N2CCC(C)(CSC)C2)nc(=N)nc(N2CCC(CCO)C2)[nH]1 72644,C(=O)(CC1=NN(C)C(=O)C1)N1CCC(C#C)(C(N2CCOC(CC(N)=O)C2)=O)C1 72645,N(C1CCc2ccc(Cl)cc21)C(C1CCCN(Cc2cn(CC)nc2)CC1)=O 72646,c1(-c2nc(C3CCCN(c4cn(C)nc4)C3)on2)ccc([N+](=O)[O-])s1 72647,c1(NC(=O)NC2(CC(=O)Nc3c(C)cc(F)cc3)CCC2)cc(F)c(F)c(F)c1 72648,C1(C(N(C2CCN(C)C2)CCC)=O)CN(C(=O)C(F)C(C)C)CC1C(C)C 72649,c1(C(N2CC(NC(CCNC(N)=O)=O)C3(C2)CC3)=O)cccc2c[nH]nc12 72650,CC1(C)CN(CCO)CCN1C(c1ccnc(Cl)c1F)C(=O)NC1CC1 72651,C1(CN(C(=O)COC2CCOC2)C)CCN(C(=O)CCN2CCC(F)C2)CC1 72652,c1(C(N2CCCC(NC(c3ccc(Br)cc3Br)=O)CC2)=O)c(Cl)cc(F)cc1Cl 72653,C(CCC(C)C(=O)N1CC(Nc2cc(C(=O)NOCCN(C)C)on2)C1)OC 72654,C1(NC(Cc2c(C)n(C)cn2)=O)CN(C(=O)C(C)C#N)CCC12CCC2 72655,N1(C(C(C(=O)OC)OC)=O)CC(NC(c2ccnnc2O)=O)C2CCCC12 72656,N1(C(C2CCCCO2)=O)CCN(C(C2(CC(F)(F)F)CC2)=O)CC12CCC2 72657,C1(=O)C(C)(C)CCC(=O)C(N(C(C(CC)CCOC)=O)C)CCC(CC)N1.OC 72658,c1(N2CC(CNC(c3nc(C)nc(O)c3)=O)OCCC2)ncc2ccnc-2[nH]1 72659,c1(C(=O)NCCOCCCN(C)C(c2cc(F)n[nH]2)=O)c[nH]nc1S(N)(=O)=O 72660,N1(C(Cc2c(C)cccn2)=O)CC2(C(=O)NC3CCC(C4CC4)C3)CC1CO2 72661,N1(C(C(c2ccc(Cl)cc2)C)=O)CC2CN(C(c3csc(C(F)(F)F)n3)=O)C2C1 72662,c1(C(=O)NC(C(C)C)CCN(C(=O)C(C)O)C)c[nH]c2c(Br)cccc12 72663,CCCCC(=O)NNC(=O)C1CCN(C(=O)OCC(C)(C)C)C1(C)C 72664,CC(CC(=O)N1CCCC1C1(C(=O)NC2CCC(C)(C)CC2)CC1)C(F)(F)F 72665,C1(C(=O)NCC(CC=C)(C)C)CN(C(c2cnc(C)s2)=O)CC1(F)F 72666,CCN=c1[nH]c(C(=O)NCC(C2CC2)N(C(=O)Cc2nncn2C(C)C)C)cs1 72667,c1(CNC(CC=C)=O)ccnc(C(=O)NCC2C=CCCC2)c1 72668,CC1C(NC(c2cc(Cl)no2)=O)CCCN1C(=O)CCC(=O)c1ccccc1N 72669,C1(CNC(c2c(CC)n(C)nn2)=O)CN(C(=O)Cc2cnnn2C)C2(CCC2)C1 72670,CC1CCC(C(=O)NOc2ccccc2)CN1.N12CC(c3cccs3)(C1)C2=O 72671,C1(NC(C(c2cccc(C)c2)C)=O)CC(F)CN(C(c2cnnc(C)c2)=O)C1 72672,CCC1=NOC(C(=O)NCCCCNC(=O)C=CCn2cncn2)C1 72673,c1(COCCO)cc(Cl)cc2cc(C(=O)O)oc12.C12CCN(C1)C2 72674,c1(C(N2CC(CC=C)(NC(=O)CCCC(C)=O)C2)=O)ccc2c(c1)CCS2(=O)=O 72675,CC(CC(F)(F)F)N(C)C(C1C2CC1N(C(=O)C(=O)N(C)C)C2)=O 72676,N1(C(CS(CC)=O)=O)CC2CC1CN(C(C1(c3ccccc3OC)CC1)=O)C2 72677,N1(C(CC(C)C2CC2)=O)CCC2(CC1)CC2NC(c1cnn2c1OCCC2)=O 72678,C1(CNC(c2c(C)cns2)=O)COCCN(C(C2(F)CCS(=O)(=O)C2)=O)C1 72679,c1(C(=O)NC2(CC=CC(=O)N(CCCCCCC)C)CCC2)cn2c(n1)CCC2 72680,C1(C(=O)NC(CC(C)C)C)CCN(C(c2ccc(F)cc2)=O)C1(C)C 72681,c1(C(N2CCCC(N(c3cc(C)ccc3C)C(C)=O)C2)=O)cccn2nccc12 72682,C=CCCCCCC(=O)NC(C)(C)CNC(=O)C(c1ccc(Cl)s1)C 72683,N1(C(CC=C=C)=O)CCC2CCN(C(c3cn(C)nc3-c3ccc(C)o3)=O)C2C1 72684,C(=O)(C(C)(C)S(C)(=O)=O)N(C1CN(C(CCC(CC)OC)=O)CC12CC2)C 72685,c1(C(=O)NCC2C(NC(CCCC(C)(F)F)=O)CCC2)sc2ccccc2c1Cl 72686,CCC(C(=O)NCCCN(C(=O)CC1(C)CC1)C)C(F)(F)F 72687,CC1OC(C)CC1C(N1CC(CC(C)NC(=O)CCC2CCOC2)C1)=O 72688,N1(c2cc(NCCCCOC)ncn2)CCN(C(c2ccco2)=O)CC1(C)C 72689,c1(C(=O)NCCN(C(=O)C(F)C2CC2)CC(C)O)c[nH]c2cccc([N+](=O)[O-])c12 72690,CC(O)C(C(=O)NC12CC1CN(C(c1n[nH]c(C3CC3)n1)=O)C2)NC(N)=O 72691,C(=O)(C1CCCc2cncn21)NC(C)(CNC(C1CCCC1)=O)C1CC1 72692,C(CN=c1[nH]c2c(c(=NC(C)CC(=O)NC3CCCC3)[nH]1)CC(C)CC2)OCC 72693,N1(C(C2C(OC)CCC2)=O)CC(=O)Nc2ccccc21 72694,C1(C(=O)NC2C(NC(c3c(C)cnn3C)=O)COC2)COc2cc(Cl)ccc2C1 72695,N1(C(C(C)=CC)=O)CC2(CCN(C(c3ccc(=O)n(CCF)n3)=O)CC2)C1 72696,c1(CC)cc(F)c(C(=O)NCCC2(NC(c3ccccn3)=O)CCC2)cc1F 72697,N1(C(c2nc(CC)oc2)=O)CCC2(C=C(C(=O)NCC3CC3CC)C2)C1 72698,C1(C(=O)NC2(C3CCCN3C(=O)COC3CCOC3)CC2)CCc2c[nH]nc2C1 72699,N1(C(C=Cc2scc(C)n2)=O)CCN(C(=O)CCn2ccnn2)CC2(CC2)C1 72700,N1(c2ccc(C(=O)OCC)cn2)CC2CCCN(C(c3cc(Cl)n(C)n3)=O)C2C1 72701,C(=O)(C(C(C)(C)C)c1nn[nH]n1)NCc1cn(CCNS(C)(=O)=O)nn1 72702,C1(N(C(C(n2c(C)ccn2)C)=O)C)CCN(C(c2cc(C(F)(F)F)ns2)=O)CC1 72703,c1(C(N2C3C(NC(C4(CN(C)C)CC4)=O)C(C3)C2)=O)cccc2occc12 72704,N(C(=NCC1(C)CCCO1)NC(C)C)C(C#C)CC1CCC1 72705,c1(-n2cc(C(=O)NC3CCC3CNC(C3CC3(F)F)=O)nc2)cccc(Cl)c1 72706,S(=O)(=O)(c1ccc(CNCCC(O)CCO)cc1)NCC=C 72707,N1(C(CCc2nc(C)sc2)=O)CCC(CO)(NC(C2CCOC2C(C)C)=O)C1 72708,C(CC(=O)NC(C1(CO)CC1)C)(C(F)F)NC(Cc1c(C)n[nH]c1C)=O 72709,N1(C(C(C)CN(C)C)=O)CCN(C(C23CCC(CC2)C3)=O)CC1CC1CC1 72710,c1(C(=O)NCC(C)(C)CNC(=O)C(O)c2cnc[nH]2)cncc(P(C)(C)=O)c1 72711,CC1=NOC(C)(C(=O)NC2CCC(CCNC(=O)CCC=CBr)C2)C1 72712,c1(NC2CCN(C(c3cnc(SC)s3)=O)C2)cncc(Cl)n1 72713,C(C#CCNC(C1(CCF)CC1)=O)NC(CNC(N)=O)=O 72714,N1(C(c2n(C)nnc2CNC(=O)C(=O)NCC2CC2)=O)CCC(N=[N+]=[N-])C1 72715,C1(C2CCC2)(C(N(CCCCNC(c2ncn(C(C)C)c2)=O)C)=O)CCC1 72716,C1(c2onc(C)n2)CN(C(c2nnn(C)c2C)C(=O)NCCC2(C)CC2)CCO1 72717,N1(C(C(C2CC2)SC)=O)CC(F)(CNC(=O)C(CN(C)C)c2ccccc2)C1 72718,c1(C(C)(C)C)ccc(C(=O)NCCN2CCN(C(=O)C(N)=O)CC2)cc1 72719,N1(Cc2cccc(CNC(=O)OC(C)(C)C)n2)CC(C(N)=O)CCC1(C)C 72720,C1(NC(Cc2cn(C)nc2)=O)C2CC1N(C(=O)C(C)(C)Cc1ccc(F)cc1)C2 72721,C1(C(N2CCC(N(C(C(CC)COC)=O)CCO)C2)=O)CN2CCC1CC2 72722,c1(C(=O)NCC(CNC(CCSCCCC)=O)(C)F)cc(F)cnc1O 72723,CC1OCCOC1C(N1CCOCC1CCNC(c1cc(C(F)F)ccn1)=O)=O 72724,C(C)(CCC(=O)N1CCCC1CCNC(C12CC(CCO1)C2)=O)OC 72725,N1(C(c2ccn(-c3ccccc3[N+](=O)[O-])n2)=O)CC2ON=C(C(F)F)C2C1 72726,CCC(C)C(C(=O)NCCCCCCNC(N)=O)NC(=O)CN(C)S(N)(=O)=O 72727,CCC(CC)(CO)C(=O)N1CC2CC1C2NC(C1(CO)CCCO1)=O 72728,Cc1nccc(C(N2CC(c3ocnc3CNC(=O)CCCF)C2)=O)c1N 72729,N1(C(C2(C)CC=CCO2)=O)CC2=C(C1)CN(C(=O)CCNC(c1cccs1)=O)C2 72730,C(CC(C(=O)NC1(C)CC1)NC(=O)C(F)C(C)C)OC 72731,C1(CN(C(CCC2CCC(C)O2)=O)C)CCN(C(c2ccc(C(N)=O)s2)=O)CC1 72732,c1(C(=O)NCC(CNC(C=C(C)c2ccsc2)=O)(C)C)cc2scnc2[nH]1 72733,C1(C(=O)NC(C(=O)OCC)CC)C2CCC(C2)N1C(C1(C)CCCO1)=O 72734,C1(N(C(Cc2ncc(C)o2)=O)C)CN(C(=O)CC2CN(C)C2)CC1F 72735,CC1(C)OCC2CC12C(N1CCC(NC(c2cn3c(n2)SCC3)=O)C1)=O 72736,CS(=O)c1ccc(NC(=O)CCc2ccncn2)cc1 72737,c1(CNC(C2(NC(C3CC3C(F)(F)F)=O)C(C)(C)C2)=O)ccccc1O 72738,CCC(CC(=O)N1CCC(NC(C23CC(CO)(C2)C3)=O)C1C)C1CCC1 72739,C1(C2CC2)(C(=O)NCC(CNC(CCC)=O)OC)CCOCC1 72740,C(=O)(CCC1=CCCCC1)N1CCN(C(CCCC#CC)=O)CC1CC 72741,c1(CC(=O)NCC(C)NC(=O)CCc2ccc(Cl)nc2)cccc(F)c1 72742,C1(NC(=O)CC2CCCCC2)CC12CCN(C(c1ncc3[nH]ncc3n1)=O)CC2 72743,c1(N2CCCC(NC(Cc3n(C)ccn3)=O)CC2)c(C#N)cccc1[N+](=O)[O-] 72744,C(c1cn(CC(CNC(=O)C(C(C)C)N2CCC(C)CC2)OC)nn1)=CC 72745,C1(CC)CCC(C)N1C(C1OCCC1NC(c1cncs1)=O)=O 72746,N1(C(COCCCC#C)=O)CCCC(CCNC(=O)C(c2cccc(Cl)c2)O)C1 72747,C1(NC(C2CN(C)C2)=O)CN(C(c2cccc(CC#N)c2)=O)C2CCCCC12 72748,C(C1CCCCCC1)=CC(=O)N(CCCCN(C(C1CCC(OC)C1)=O)C)C 72749,N1(C(CNC(CC)=O)=O)CCC2C1CCCN2C(c1cc(Br)cc2[nH]ncc12)=O 72750,C(=O)(CC(C)C(=O)OC)NCCC1(O)CCN(C(C2(OCC)CCOCC2)=O)C1 72751,C1(C2CN(C(=O)C(C)Cn3ccnc3)C2)(NC(Cc2c(C)n[nH]c2)=O)CC1 72752,C1(CCNC(C(F)=CCC)=O)CCN(C(=O)CNC(=O)CCC(C)C)C(C)C1 72753,c1(C(N(CCCC2(NC(=O)CCC(=O)NC)CC2)CC)=O)cnc(C)cc1Cl 72754,Cc1nn(C)cc1-c1cn(CCCC(=O)NCCC2CC3CCC2C3)nn1 72755,C1(OC)CC2CC1CN(C(=O)CC1CCCCC1NC(C1(C)CC(F)(F)C1)=O)C2 72756,Cc1ncnc(O)c1C(=O)NC1CCN(C(C2CCC3(CCC3)O2)=O)C1 72757,C(CN=S(C)(C)=O)NC(c1n(CC(=C)C)nnn1)(CCC)C1CCCC1 72758,C(C)(C)(C(C)CC(=O)NC1CCN(C(C)=O)C1)NC(C=CC=CCC)=O 72759,c1(C(=O)NCCC2(C(=O)NCC3(OC)CCC3)CC2)nc(C)sc1C 72760,C(=O)(C(O)(C(F)(F)F)c1ccccc1)N1CCC(CCNC(C2(F)CC2)=O)C1 72761,C(=O)(C1CCCc2n[nH]cc21)NCCCC(C)NC(C1CC1(F)F)=O 72762,N1(C(CC(C)O)=O)CCC(F)(F)C(CNC(c2cc(C3CC3)n(C)n2)=O)C1 72763,Cc1nnc(NC2CC(NC(c3sccc3C)=O)C2)nc1C 72764,c1(N2CCN(C(CCC)=O)CC2)cc(C)nc(C)c1[N+](=O)[O-] 72765,C1(C(=O)NC(COC)C)CC2CN(C(c3ncn4ccccc34)=O)CC2C1 72766,C(C1CCCN1C(c1coc(CO)c1)=O)=CC(=O)N(C)Cc1ccco1 72767,N1(C(C#CC2(CC)CC2)=O)CCCC2CN(C(C3(CO)CCC3)=O)CC12 72768,S(=O)(=O)(C1CN(C(c2cc(CO)[nH]n2)=O)C1)N1CCN(C(CC(=O)NCC)=O)CC1 72769,Cc1c(C(=O)NCc2ncc(C(N3CC(C)(O)C3)=O)cn2)c[nH]c1C#N 72770,CCC(C)C(O)CC(=O)N1CCOC(CC(=O)NCC(C)(F)C(C)(C)F)C1 72771,c1(C(N2CCC(CN(C(C(N3CCC(O)CC3)C)=O)C)C2)=O)cccc(Cl)c1Cl 72772,N1(C(CC(C=C)C)=O)CCN(C(=O)CCc2cc(OC)no2)CC2(CC2)C1 72773,N1(C(C=CC=CC)=O)CCC(NC(c2cn(C)nc2CCC(F)(F)F)=O)C1C 72774,c1(C(C)(C)C)nc(Cl)cc(=NC(CNC(=O)C2=CCCOCC2)C2CC2)[nH]1 72775,N1(C(CSCC#C)=O)CCCC(C(C)(C)C(=O)NCc2cnn(CCC)c2)C1 72776,C1(NC(C2CC2(F)F)=O)CCN(C(=O)C=Cc2ccncn2)CC1CO 72777,C(=O)(C(F)(F)C(F)(F)F)N1CC(NC(=O)Cn2ncc(O)nc2=O)C(O)C1 72778,C1(C(=O)NCC(C)CNC(c2ccno2)=O)CNC(=O)CC1C 72779,c1(NCCN=C(NCc2c(C)nn(C)c2)NC2CC2C)ccc([N+](=O)[O-])c(F)c1 72780,n1(CC(=O)NC23CC(CNC(C(C(C)C)F)=O)(OC2)C3)nc(O)c2ccccc12 72781,C1(C(N2C(C)(COC)CCC2)=O)CC2CCCC2N1C(=O)C1=C(C#N)CCC1 72782,N1(C(CCC=C)=O)CCC(C2CCCN2C(c2cncc(C(C)(F)F)c2)=O)CC1 72783,N1(C(Cc2nnc(C)o2)=O)CCN(Cc2cccc(C)c2O)C2CC12 72784,C(=O)(CCCC(=O)NCC1CN(C(=O)CC2CCCCN2C(C)C)CCO1)OC 72785,N1(C(c2nc(C)n(-c3nc[nH]n3)n2)=O)CC2CC1CN(C(C1CCC(C)O1)=O)C2 72786,C(=O)(CS(N)(=O)=O)NC1(C(N2C(C(C)O)CC2)=O)CCC1 72787,N1(C(C(=O)NCCC(C)c2ccco2)=O)CCC(NCC(F)F)CC1 72788,C(C(CC)(CC)C(N)=O)NC(C1(CNC(CCC=C=C)=O)CC=CC1)=O 72789,N1(C(C(C(C)C)SC)=O)CCCn2cc(Br)cc2C1 72790,c1(CC)cc(NNC(=O)NC2COc3cc(Br)ccc3C2)ncn1 72791,CCCC(CNC(=O)C=CC(F)(F)F)C(=O)NCCN(C(C)CC)C 72792,n1(CCOCC)nc(-c2cccc(C(F)(F)F)c2)nc1CCCC1CCCCC1 72793,CCC(C)C(=O)C(=O)NCC1C(C)CCCN1C(c1cnn(C(C)C)c1)=O 72794,C1(NC(C(C)CO)=O)CCC2(CC1)CN(C(c1cc(C3CCOCC3)[nH]n1)=O)C2 72795,Cc1cc(C(N2CCCCCC2CNC(=O)CC(C)C)=O)cc(C)c1 72796,c1(C(=O)NCCN(C(C(CC)C2CCC(=O)N2)=O)C(C)C)ncc2ccccn12 72797,C(=O)(C1=NOC2COCC12)NC1C(CC)N(C(=O)Cc2ccc(Cl)cc2F)CC1 72798,c1(OC(C)C)ccc(COC(c2ccccc2CS(C)=O)=O)c(Cl)c1 72799,C1(C(=O)NCCC2OCCN(C(C=C(C)C)=O)C2)CCCCN(C)C1=O 72800,C1(C(=O)NC(CNC(c2c(SC)csc2)=O)C2CC2)CCCCCCC1 72801,c1(NC(C2N(C(CC(C)(C)O)=O)CCC2)=O)cc(Br)cnc1I 72802,C1(NC(CC=C)=O)CC2(CCN(C(c3cc4sccc4cn3)=O)CC2)C1 72803,N1(C(C(C)=C(C)C)=O)CCCC1CCNC(c1ccco1)=O 72804,N1(C(C2(C)CNC(=O)C2)=O)CC(C2CN(C(c3nccc(Cl)c3F)=O)C2)C1 72805,N1(C(c2cc(C)cc(F)c2)=O)CCC2(CC2)CC1C(=O)NC(C)C(C)(C)O 72806,c1(C(=O)NCC(C)NC(Cc2c(C)cco2)=O)cc2c(n1C)CCOC2 72807,C(=O)(CC(CC(C)C)NC(=O)CCn1cnc(=N)[nH]1)Nc1cn(CC)nc1 72808,N1(C(c2ccc(N(C)C)cc2O)=O)CC(C2CC2)C(F)(C(=O)O)C1 72809,C1(C(N2CC3C(NC(c4c(SC)cccc4)=O)(C3)C2)=O)CCN(C)S1(=O)=O 72810,C12CCCN(CC1)C(=O)C1(CC1)CNC(=O)C2.N1(C(CC)C)CCCC1 72811,c1(C(N2C(CO)CC(NC(c3cc(C)oc3C)=O)C2)=O)ccc2c(c1)NCCC2 72812,C=C(C)C(C)(C)C(=O)NC1CCCC(CNC(c2ccc(C(F)(F)F)o2)=O)C1 72813,C1(C(=O)OCC)CN(C(=O)C=CC(=O)NCC2(F)CCCC2)CC12CCOCC2 72814,C1(N(c2cccc(-n3cnnc3)c2)C(c2c(C)noc2)=O)CCNCC12CC2 72815,c1(C(c2n(CC=C)nnn2)NCC(C2CCCCC2)OCC)nccc(Cl)c1C 72816,Cc1cnc(C(=O)NC2CC(N(C)C(c3cnc(C)[nH]c3=N)=O)C2)c(C)c1 72817,C1(CC(=O)N(CCCCN(C(=O)Cc2cnco2)C)C)OCCC1(C)C 72818,S(=O)(=O)(c1cccc(C(=O)N(C)C(c2ncccn2)C)c1)NC(CC)C(N)=O 72819,c1(C(=O)NC2CC3(CN(C(CC=CC)=O)C3)C2)cc([N+](=O)[O-])ccn1 72820,N1(C(CCCC#C)=O)CCOCC(NC(=O)CC(C)Cc2ccc(F)cc2)C1 72821,C1(C(=O)NCC2(O)CN(C(CNC(C(CC)C)=O)=O)C2)CNC(=O)C(C)(C)C1 72822,CC(C)C(F)(CNC(C1CCCC12CCC2)=O)C(=O)N(C)CC1CCOC1C 72823,C(=O)(C(C)(C)CC(=O)NC(c1ccccc1F)CNC(=O)C(C)CF)OC 72824,c1(CCC)ccc(OC)c(OC(=O)C=Cc2scnc2C)c1 72825,c1(C(=O)NC2C(OC)CN(C(c3cccn3C)=O)C2)ccc2c(N)nccc2c1 72826,N(C1COc2cc(Br)cc(C)c21)C(=O)NCc1ccc(-n2ccc(C)n2)c(F)c1 72827,C=CCCC(C(=O)NC1CCCN(C(C)C)C1)NC(=O)CC1CCCSC1 72828,N1(CC)CCCC(n2cc(C(C)(C)F)nn2)CC1.c12nc(no1)C(=O)N2 72829,c1(C(COC)(C2CCCC2)NCC2CC2)nnnn1Cc1ccccc1 72830,CC1C(C)N(C(=O)CC23CCC(CC2)OC3)CCN1C(=O)C(C)OCCN(C)C 72831,C1(N)(Cc2nc(C(c3ccc(F)cc3)N(C)C)on2)CCCC(C)(C)C1 72832,c1(C(=O)NC2CC2)cnn2cccc(-c3ccc(OCCCO)cc3)c12 72833,c1(C(=O)NCCC2CC(NC(CC#N)=O)C2)ccc2c(c1)S(=O)(=O)NC2 72834,C(=O)(C(C)(C)CCC#N)OC(C)(C)C.C12COCC1ON2C 72835,c1(NCC(C)(C)OC)nc(C)cc(=NC(C)c2ccc(C#N)c(C)c2)[nH]1 72836,C(=O)(C(O)CC[S+](C)C)N(CCCNC(C(C)OCCC=C)=O)C 72837,C1(OC)CC2(C1)CN(C(=O)CC(O)CNC(=O)C(c1cnn(C)c1)O)C2 72838,C(=O)(NN1CCCC1C(=O)N(C1CCCC1)C)C1CC(N(C)C)C1 72839,c1(OC)cc(C2(C(=O)NCC(C)(O)CNC(=O)CC3CC(F)C3)CC2)ccc1C 72840,c1(C(=O)N)ccnc(F)c1N.c1(C(C(=O)N2CCC(OC)C2)SCC)ccccc1 72841,N1(c2cc(C)ncn2)CCCCC(NC(=O)Cc2c(F)cccc2F)CC1 72842,c1(CC(=O)NC2CCC(CNC(C(N(C)C)C3CC3)=O)C2)cc(Cl)ccc1Cl 72843,n1(CCC(=O)NC(C(C)C)c2ncc[nH]2)cc(CNS(N)(=O)=O)nn1 72844,CCC(C)(O)CCNC(C1(NC(C2C3CCCOC23)=O)CCSC1)=O 72845,Cc1ccc2ncc(C(N3CCCC(NC(c4coc(C)n4)=O)C3)=O)n2c1 72846,c1(C(N2CC(O)(C(=O)OCC)C2)=O)cccc2c1oc1ccccc21 72847,C(=O)(CCCCCF)NC1C(C)CN(C(c2cnc(C(C)(C)C)[nH]2)=O)C1 72848,C1(C(N2CC(C)C(CC(=O)Nc3cnsc3)C2)=O)CCCCCN1C 72849,CC12CN(C(=O)Cc3ncc(Cl)s3)CC1CN(C(c1coc(C(F)F)n1)=O)C2 72850,c1(NC(=O)CCSCCNC(c2n[nH]c(O)n2)=O)cccc(C(F)F)c1 72851,C1(NC(c2c(OC)nsc2)=O)CCCC(CNC(=O)CC2CC=CC2)C1 72852,C(CNC(=O)Cc1cncnc1)(C(C)C(C)C)NC(C(=Cc1ccncc1)C)=O 72853,c1(CC)cc(C(N2CC(CNC(=O)C(C)C)(OC)C2)=O)n[nH]1 72854,c1(N2CCCC(NC(C(c3cn(C)nc3)O)=O)CC2)ncnc2c1ncn2C1CC1 72855,N1(C(C(C)=CC2CC2)=O)CCC2(NC(c3conc3C)=O)CC2C1 72856,C1(NC(=O)Cn2cncn2)CCN(C2CN(Cc3cccs3)C2)CC1 72857,c1(C(=O)NCC2(F)CC(CNC(C(CC(=C)C)C)=O)C2)cncc(S(C)(=O)=O)c1 72858,c1(C(=O)NCC2CN(C(CC3CCC(C)(C)CO3)=O)C2)c(Cl)cccc1[N+](=O)[O-] 72859,c1(SC2(C(=O)NC(C)CN(C)C(C3CCC3C(F)(F)F)=O)CCC2)ccccc1 72860,N1(C(CCCOC)=O)CCC(C2(NC(c3ccc(OC(C)C)cc3)=O)CC2)C1 72861,CC(C)CCCCCC(=O)NCC1C2CC1N(C(c1coc(Cl)n1)=O)C2 72862,C(=O)(C(C)(C(F)F)c1ccccc1)NCC1CC(NC(CSC)=O)C1 72863,c1(C2C(C(=O)NC3CC(CC(=O)OC)OCC3)C2)ccc(-c2nn[nH]n2)cc1F 72864,c1(CN2CCC(NC(CC(CC)O)=O)(CO)CC2)c(Cl)nc(SC)nc1Cl 72865,c1(C(CNC(=O)CSc2nc[nH]n2)NC(CC2(CSC)CC2)=O)ccccc1 72866,CC1CN(C(=O)CC(C)CN(C)C)CCCN1C(=O)CCn1cccc1 72867,c1(OC)cccc(Cl)c1C(N1CCC(CO)(Nc2ccncn2)CC1)=O 72868,C(CN=c1[nH]c(N2CCN(CC(F)(F)F)CC2)nc2c1CCC2)C1C(C)C1 72869,c1(C(c2nnnn2CCC2CC2)NC(C(=O)N(CC)CC)C)ncc(C)s1 72870,c1(CN(c2ccc3c(c2)OCO3)C)nc2c(c(=NCCCP(C)(C)=O)[nH]1)COC2 72871,c1(OCC)cccc(C(N2CC(O)CC2C(=O)Nc2nc(C#N)cs2)=O)c1 72872,C1(NC(C(C(C)C)C)=O)CCN(C(=O)COC2CCCOC2)CCC1CO 72873,c1(COC(c2ccc(-c3cccc(Br)c3)cc2)=O)cccnc1F 72874,Cc1cccc(OCC(N2CC(NC(=O)CSCc3cccnc3)C3CC23)=O)c1 72875,c1(C(N2CCCC2CS(N)(=O)=O)C(=O)NCCSC)ncc(C(C)C)s1 72876,c1(C(=O)NCCCCNC(C2(CC)CC2)=O)ccc(C)cc1.C(=O)C1CC1 72877,c1(C(=O)Nc2cc(C)c(C(F)(F)F)cc2)cccc(S(=O)(=O)NCCN(C)C)c1 72878,C(CC)(CCCC(=O)N(C)CP(C)(C)=O)NC(C1C(=C)C1C(=O)OC)=O 72879,CCCCCC(C)CC(=O)N1CCC(NC(=O)CCc2ccc(O)nn2)C(F)C1 72880,C(=O)(CC(C)CC(C)(C)C)N1C(C(=O)NC(C)C(F)(F)F)CSCC1 72881,C(=O)(CC(F)(F)Cl)NC(c1ccc(F)cc1)CNC(C12CC(C)(C1)C2)=O 72882,CC1Cc2cc(C(=O)NC3COCC3NC(=O)Cn3cnnc3)ccc2O1 72883,C#Cc1nccnc1NC(C1CCCN1C(=O)CCNC(c1ccc[nH]1)=O)=O 72884,N1(C(c2n(CC)ncc2Cl)=O)CC(NC(c2cc(C)cc(C)n2)=O)CC(O)C1 72885,N1(C(CC(n2c(CC)ncc2)C)=O)CC2CC1CN(C(c1ccc(Cl)o1)=O)C2 72886,CC(Cl)(Cl)C(=O)N1CC(C(N)=O)(CNC(c2ccc(C(N)=O)o2)=O)C1 72887,C1(CNC(C23N(C(c4cc(C)ncc4)=O)CC(C2)C3)=O)OC(=O)CC1(C)C 72888,c1(NC(c2n(C)cc(NCc3ccc(Br)[nH]3)n2)=O)ccc(Br)cc1C(C)(C)C 72889,c1(OC)ccc(C(=O)NC2CCN(C(c3cc(C)ccn3)=O)C(C)C2)c(F)c1Cl 72890,C1(C(N2CCN(C3CCCC3)CC2)=O)C2CC(O)C(C2)N1C(=O)C(F)Cl 72891,N1(CCNC(C(c2cccc(Cl)c2)(C)C)=O)CCC(NC(C2CC(F)C2)=O)CC1 72892,N1(C(C2(c3c(C)cccc3)CCC2)=O)C2CCCC1CC(NC(=O)C(C)(C)F)C2 72893,c1(C(N2CC(C(=O)NC3CC3)C2)=O)cnc(CNC(=O)CC2CCC(=O)C2)nc1 72894,N1(C(C2CCC(COC)C2)=O)CCN(C2CCN(C(=O)C(=O)N(C)C)CC2)CC1 72895,c1(C(=O)N(CCCn2cc(-c3cncc(Cl)c3)nn2)C2CC2)c[nH]nc1[N+](=O)[O-] 72896,C1(C(=O)NCCNC(C)=O)CC2(CCN(C(=O)CC3C(C)(C)C3(C)C)C2)C1 72897,c1(OC)ccc(C(O)C(N2CC(O)(CNC(=O)CC3(C)CCCC3)C2)=O)cc1 72898,C1(C(=O)NCCCCN(C(COCCN(C)C)=O)C)CCCCN1C1CCCC1 72899,c1(C(=O)NC2CCCC(CC(=O)NCCOCC)C2)c(C)cnnc1O 72900,c1(C(N2CC(NC(c3n(CC)ncc3)=O)CC2(C)CC)=O)ccc2n[nH]cc2c1F 72901,C(=O)(CCCC(C)(C)C)NC(C1C(CNC(c2ccc(CSCCC)o2)=O)C1)=O 72902,c1(CNC(=NCC=C)NCC(C)C#N)ccc(S(=O)(=O)N2CCCCC2C)cc1 72903,C1(CN(C(C2C(C)=C2)=O)C)CCCN1C(C1CCC(=O)N1)=O 72904,C12(CNC(C3CC4(CC4)C3)=O)CCCC1CCN2C(c1cc2c(s1)CCC2)=O 72905,C(=O)(CC(C)(C)C1CC1)NCCCC(C)NC(=O)CC1C=NN(C)C1=O 72906,CC1CCCn2cc(C(=O)NC3CCC(NC(c4cnc[nH]c4=N)=O)CC3)nc21 72907,c1(C(N2CC3C(CNC(c4c(CC)onc4C)=O)(C3)C2)=O)ccc(F)cc1O 72908,C1(N(CC)CC)CCN(C(=NCC2CCCCC2)NCC2CCCOC2(C)C)C1 72909,N1(CCCNC(c2cccn(C)c2=O)=O)CCC2(CCCCC2)CC1 72910,C1(NC(C(C)=CC2CC2)=O)CC(C(=O)N(C)Cc2cnccn2)C1(C)C 72911,C#CCCCC(C)C(=O)N1CCC2(CC2NC(=O)C(c2ccccc2F)C)C1 72912,C=C(C)C(C)(C)C(=O)N1CC(CO)(NC(=O)CN2CCCC2CO)C1 72913,CCC(C)CCCC(=O)N(CCNC(C1CCS(=O)(=O)CO1)=O)CCOCCO 72914,CS(=O)(=O)c1ccc(C=CC(=O)NC2CCN(C(=O)CC(F)F)CCC2CO)o1 72915,Cc1ccc(C(=O)NC2CCC2NC(c2cc(O)ncc2Br)=O)c(F)c1 72916,N1(C(C2CCC(NC(c3cn(C(C)C)nc3)=O)CC2)=O)C2CCC1COC2 72917,C1(C(=O)N(c2c(C)nco2)CCO)C2CN(C(c3coc(C(N)=O)c3)=O)CC12 72918,N1(C(C2CCC23CCC3)=O)CCC2CC(C1)CN(C(=O)CCc1cnccn1)C2 72919,C1(CNC(=O)CN2CCCS2(=O)=O)C(C2CC2)CCN1C(=O)Cc1ccc(Cl)o1 72920,C(=O)(CC(CC1CC1)NC(=O)CC(O)CN(C)C)NCCc1scc(C)n1 72921,N1(C(CSCC)=O)CC(C2CCN(C(c3ccccc3O)=O)C2)C1 72922,N#CC1(C(=O)NCCCCNC(C2CC2F)=O)CCC(=O)CC1 72923,CC1(C)CCCC1CCCNC(=O)NC1(Cc2ccc(Cl)cc2)CC1 72924,N1(C(C(C(C)C)O)=O)CC(NC(C23CC(c4ccccc4)(C2)C3)=O)CCC1C 72925,c1(C(N2C(C(=O)NCC3C(C(=O)OC)C3)CNC(=O)C2)=O)cccc2cncn12 72926,c1(C(N2CCC(CNC(CC(C(F)(F)F)OC)=O)C2)=O)cc(O)c2sccc2c1 72927,O=C1CCC(N=c2[nH]c3c(c(=NCc4nn[nH]c4C4CC4)[nH]2)SCC3)CN1 72928,C1(C(=O)NC(CC(=O)OCC)c2ccccc2)CCCN(C(C)CNC)CCO1 72929,C1(OC)CC(NC(=O)CCn2ccnc2)CN(C(C2(C#N)CCCC2)=O)C1 72930,C1(NC(c2ncc(OCC)nc2)=O)CC2(CCN(C(C3(CC)CCOC3)=O)C2)C1 72931,c1(C(N(CC(CC)NC(=O)CNC(C)=O)C)=O)cc(Br)cc(C)c1F 72932,C1(CNC(C2N(C(CSC)=O)CC=CC2)=O)CCCC2(CC2)C1 72933,C12(NC(CCCN(C(C)=O)C)=O)CCC(CN(C(=O)CC(C)C3CCCC3)C1)C2 72934,C1(C(N(CC(C)NC(c2cccc(C3(C#N)CC3)c2)=O)C)=O)CCCCC1(C)C 72935,C1(NC(COc2cccc(CC)c2)=O)CCN(C(=O)C(C)c2ccco2)CC1O 72936,N1(C(c2cc(OCCC)c(F)cc2)=O)CC(C(=O)NC)CC(F)(F)C1 72937,CCC(O)CCNC(=O)CC1(CNC(=O)Cc2ccsc2C)CC1 72938,C1(C(N2CCC(F)CC2)=O)CC12CCN(Cc1ccc([N+](=O)[O-])o1)C2 72939,N1(C(C2C(=C)CC2)=O)CCCC2(NC(c3coc(COC)n3)=O)CC2C1 72940,c1(C(N2CCC(C)C2)=O)c(CNC(c2cc(Cl)cs2)=O)cnn1C 72941,c1(SCC(=O)NC2CC(CNC(C3CCC(SC)C3)=O)C2)nnc2ccccn12 72942,c1(OCCC(=O)NCC(N(C(C(CC)OCC)=O)C)C2CC2)cccc(F)c1 72943,C(C(CC)CC)(c1n(CCOC)nnn1)NC(c1cccc(OC)c1)C 72944,C1(C(=O)NC2C(C(N(C(C)C(F)F)C)=O)CCC2)CCCC(=O)N1C 72945,C(=O)(C1=CCCOC1)NC(C(C)(C)C)CNC(=O)CC1OCCO1 72946,C(N1CCOC(C2CC2)C1)N1CCC(C)C1=O 72947,c1(C(=O)NCCCCO)cn2c(n1)CN(C(c1c(F)ccc(O)c1F)=O)CC2 72948,c1(C(=O)NC2C3(CN(C(C4C(C)(C)CC4)=O)C3)SCC2)ccc2cccnc2n1 72949,N1(CC(=O)N(C(C)CNC(C2CC23CCOC3)=O)C)CCS(=O)(=O)CC1 72950,N1(C(c2cnc(C)[nH]2)=O)CCN(C(C2CC=CCO2)=O)CC1CS(C)(=O)=O 72951,CCC(CC)C(C)C(=O)NC(CCOCCO)C(=O)Nc1ccc(F)cc1C 72952,CN1CCC(C(=O)NC2CC2NC(=O)C=Cc2cccc(CO)c2)S1(=O)=O 72953,c1(C(N2C(CNC(c3csc(CC(F)(F)F)n3)=O)CCC2)=O)ncncc1Cl 72954,N(C1CC2(CN(C(C3CC(C)N(C)C3)=O)C2)n2ccnc21)C(C(C(=C)C)(C)C)=O 72955,O=C1CCC(NC(=O)CC2CC3(CC3)CN2C(c2ccc(F)cn2)=O)C(=O)N1 72956,N#CC1CCCC1NC(C1CCCN1C(=O)CCC1CCC(=O)C1)=O 72957,C(CCCCC(=O)NCC(C)(C)C(=O)NCCCc1nccs1)N(C)C 72958,C1(NCc2ccc(C)cn2)CCN(C(c2cc(Br)ccc2Cl)=O)CC1F 72959,Cc1nc(C(C)(C)C)sc1C(=O)N(CCC(C)NC(=O)CCC(C)N(C)C)C 72960,CN1C(=O)CN(CC(N2CCN(C3CN(C(=O)C4=C(Cl)CCC4)C3)CC2)=O)C1=O 72961,c1(C(=O)NCC(CNC(CNS(NC)(=O)=O)=O)F)ccc(C(F)(F)F)nc1 72962,S(=O)(=O)(c1ccc(C#N)c(N(CC(C)OC)C)c1)N1CC(CC)C2(C1)OCCO2 72963,Cc1c(C(N2CCC(CNC(=O)CC(=O)NC3CC3)CC2)=O)sc(Cl)c1Cl 72964,C(=O)(CCS(=O)(=O)CC(C)C)NCC1N(C(c2cc(C(C)=O)sc2)=O)CC=C1 72965,N1(C(CC2(COC)CCCC2)=O)CCCC(CO)(NC(C2CCCCO2)=O)C1 72966,C(CC(F)F)(C(=O)N(C)Cc1ccsc1)NC(C1C(C)C1)=O 72967,C1(C(N2CC(C)(CC=C)C2)=O)C(C2CC2)CCN1C(C1COCCC1C)=O 72968,C1(NC(CNC(=O)NC)=O)CCC2(CC1)CN(C(=O)C(C)(CC)CO)CCO2 72969,N1(C(CCC=C)=O)CCC(C(=O)NC2CN(CCC)C2)=C(F)C1 72970,O=C1NCC2(CCN(C(c3cccc4ccoc34)C(=O)NCc3ccco3)C2)O1 72971,C(=O)(C#CC(C)(C)O)NC(C(NC[Si](C)(C)C)=O)C1(O)CCC1 72972,c1(C(=O)NCCCC(C(=O)OC)O)nc2ccccc2nc1O 72973,c1sc(CNC2CCCC2N2CCCC2)nc1-c1cn[nH]c1 72974,c1(C(=O)NC(CC)CN(C(=O)C=C(CC)CC)C)ccnc(N2CCCC2)n1 72975,N1(Cc2c(OC)cc(Br)cn2)CCn2cccc2C12CCNCC2 72976,C1(CNC(C(C)OCC#C)=O)CCN(C(c2cc(C)nn2C2CC2)=O)CC1(F)F 72977,C(C(=O)NCCCCC(C)NC(=O)C(C)Cc1cnc[nH]1)(C(C)C)SC 72978,c1(-c2ccc(C(=O)NCCOCCCNC(C3CCSC3)=O)o2)cccc(F)c1 72979,C=C(CNC(=O)CC1CCN(c2nnc(S)n2C)C1)c1ccccc1F 72980,C(C(C)(O)C(=O)N1CCC1(C)CC(=O)NCc1nnnn1C)OC 72981,C1(CNC(=O)CCc2cocn2)CCCCCN1C(=O)CC1CC2(CCC2)CO1 72982,C1(C(=O)NC2CC23CC(NC(C2CN(C(C)=O)C2)=O)C3)(CC)CC(C)(C)C1 72983,C1(NC(c2ccccc2)=O)CCCCCN(C(C2CN3CCN2CC3)=O)C1 72984,N1(C(c2c(SC)cnn2C)=O)CC2CCN(C(c3cc4n(c3)CCOC4)=O)C2C1 72985,C(CCCCCN(C)C(C1CC=C(C)CC1)=O)NC(C(C1CC1)OCC)=O 72986,Cn1ccc2ccc(C(=O)NCC3CN(C(C4(C)CCOC4)=O)CC3(C)C)cc12 72987,N1(C(C(=O)NCC)=O)CCN(C(=O)CCc2cnc[nH]2)CC1CS(C)(=O)=O 72988,N1(C(C(C=C)CC)=O)CC(C(=O)NCc2cc(C)nc(O)c2)CC12CCC2 72989,C(C(C)(CC(C)C)NC(=O)Cn1cc(CO)nn1)NC(c1[nH]nc(OC)c1Cl)=O 72990,c1(C(=O)NCC2(CNC3(CC)COC3)CC2)ccc(CC#N)c(OC)c1 72991,c1(C(N2CCC(CCNC(c3cnc(OC)nc3)=O)C2)=O)ccsc1S(C)(=O)=O 72992,C1(CC)(NC(=O)CCCc2ccncc2)CCN(C(=O)C(O)C2CCCC2)CC1 72993,c1(C(=O)NCc2cccc(Cn3ccnc3)c2)cc(O)ncc1Br 72994,C1(N(C(=O)CCc2cnco2)CC)CCCN(C(=O)CC2CC3CCC2O3)C1 72995,C1(NC(C2C(=C)C2)=O)CCC(O)CN(C(c2ccc(C)cc2SC)=O)C1 72996,c1(CC)ccc(OC)cc1.C12CC=CC(C1)CN(CC(O)(COC)CO)C(=O)N2 72997,c1(CNC(C2C=CCN2)=O)cc2n(n1)CCNC2 72998,c1(C(=O)NC2C(NC(c3cncc(C)n3)=O)C2)ccc(C)c(F)c1 72999,Cc1cc(Br)ccc1NC(=O)C(C1CCOC1)Nc1ccsc1 73000,c1(C(=O)NCC2C(C)CCCN2C(C2CC(O)C2)=O)cnn2c1CCCC2 73001,c1(CC(=O)NC2(CC=C)CCN(C(C3CC3C)=O)C2)c[nH]c2cc(F)ccc12 73002,C12(NC(c3c(N)c(F)ccc3)=O)CCCC1CN(C(=O)CCCC1CC1)C2 73003,CC1CC(C#N)(C(=O)NCC2(F)CC(CNC(=O)CCC3CCC(=O)NC3)C2)C1 73004,c1(C(=O)NC2(CNC(c3cccc(C)n3)=O)COC2)cc(F)c(Cl)nc1Cl 73005,O=[N+]([O-])c1cc(CN2CCCC(N3CCCCC3)C2)ccc1Br 73006,C(=O)(NNC(=O)CCCn1cc(C2CCCO2)nn1)c1c(O)ccc(OC)c1 73007,CS(=O)CCC(O)C(=O)NCC12CC(NC(=O)CCCC3CC3)(C1)C2 73008,c1(C(=O)NC2CC(CC(=O)NCc3cn(C4CC4)nn3)C2)c[nH]c(=S)cn1 73009,c1(C(N(CCNC(CNC(CNC(=O)NC)=O)=O)C)C)cccc(OC)c1 73010,Cc1cc(C(=O)NCC2CCN(C(=O)C=Cc3ncc[nH]3)C2)nc(C(F)(F)F)n1 73011,C(=O)(C1CC(=O)Nc2cc(F)ccc21)N(C1CN(S(C)(=O)=O)C1)C 73012,CC1(C)C(NC(=O)Cc2ccc(O)nc2)CC1C(=O)NCC1CN2CCC1C2 73013,N1(c2nccc(OCCOC)n2)CCC(NC(=O)Cn2ncn(C)c2=O)CC1C 73014,N1(C(CN(CCOC)C)=O)CC2(CCN(C(=O)C(c3cscn3)N(C)C)C2)C1 73015,N1(C(c2ncc(C(C)C)s2)C(=O)NCCCOC)CCc2c(nnn2C)C1 73016,CCC(CC)C(F)C(=O)N1CCN(C(=O)CC2CC2(Cl)Cl)C(C2CCC2)C1 73017,C(=O)(CS(=O)(=O)C(C)C)NCC(CCCC)NC(=O)C(c1cnn(C)c1)O 73018,N1(C(c2ccc(C(C)(C)C)s2)C(=O)N(C2CCCOC2)CCF)CCC(O)CC1 73019,C(=O)(C(O)C1=CCCCC1)NC(CC=C)CNC(c1cnn(CC(C)C)c1C)=O 73020,C1(N(C(C2C(CC)C2)=O)CC)CCN(C(C2CCC3(CC3)C2)=O)CC1 73021,Cc1[nH]c(C)c(C(=O)NCCC2CCC(NC(=O)CCNS(C)(=O)=O)C2)c1C 73022,N1(C(C(C)OCCOCC)=O)CCN(C)CC1CNC(c1c(C)nsc1NC)=O 73023,c1(OC)ccc(F)c(C(N2C3CN(C(c4ccno4)=O)CC23)=O)c1F 73024,CC1(C)CCN(C(=O)C(CC(=O)NC(=O)CN)CC2CC2)C1c1ccccc1 73025,c1(OCC)cc(CN(C)C(=O)NC(C)CCNC)ccc1O 73026,N1(C(C2C(C)CC(C)O2)=O)CCCC(NC(=O)CCc2cc[nH]n2)CC1 73027,C(CN=C(NCC(C)(COC)COC)NCC(c1ccc(C2CC2)cc1)O)OC 73028,N12CC(C(C)C1)NC(=O)CSCC2=O.C1(C(=O)N)CCCN1c1ccncn1.CO 73029,c1(OC)ccc(C(Cc2cn(CCCCCO)nn2)O)cc1.C1(C)CC1 73030,c1(C(=O)NC(C(C)C)C(N2CCC(N=[N+]=[N-])C2)=O)coc2c1COC2 73031,C1(CN(C(CC2(CCC#C)OCCO2)=O)C)CCC(OC(=O)C(C)C=C)CC1 73032,CCCCC(CC)CC(=O)NCC(CNC(=O)Cc1c[nH]nc1C)OC 73033,C=CCCCCCCC(=O)NC1CCN(C(c2coc(O)n2)=O)C(C2CC2)C1 73034,c1(C(N2CC(C)C(NC(=O)CC3CCC(C)(C)CC3)C2)=O)onc2ccccc12 73035,C1(NC(C2CCC(C)(C)O2)=O)CC2CCC(C1)N2C(=O)C(C)(C)c1cncs1 73036,CC1CCc2[nH]c(=NC(C)c3cnn(C)c3)[nH]c(=NCCCCC(N)=O)c2C1 73037,C(C)(C(=O)NOC(c1ccccc1)C)(N(C(CCC(=O)NC)=O)C)C1CC1 73038,C1(CNC(C2CC(C)(C)C2)=O)CC(O)CN1C(c1ccnc(C2CC2)c1)=O 73039,C1(OCC#C)CCN(C(=O)CCC2CC2C(=O)OC)C1 73040,C(=O)(CS(=O)(=O)N1CCOCC1)NCC(C)N(C)C(c1ccc(C(C)O)cc1)=O 73041,c1(NC(=O)NC2CCN(C)CC2)cnc2ccnn2c1O 73042,N#Cc1cncnc1N1CCC(NC(c2ccc(C3CC3)cc2)=O)C(F)C1 73043,c1(OC)c(C(N(CC=CC(=O)NC2CN3CCC2C3)C)=O)c(C)nn1C 73044,C=CCC(C)(C)C(=O)NCC1(NC(c2cccc(-n3ccc(CC)n3)c2)=O)CC1 73045,C1(NC(C=NOC)=O)CC2CCC(C1C)N2c1cccc(F)c1C#N 73046,c1(C(=O)NC2CCCN(C(C(c3ccc(CC)s3)=O)=O)C2)cc(C)c(C)nc1C 73047,c1(NC(C2(C)CCN(C(C3(C(=O)OC)CC3)=O)C2)=O)ccc2c(c1)C(=O)C(=O)N2 73048,C(=O)(C1=CCC2CCC1N2C(=O)C(CN(C)C)N(C)C)NC(C#C)(CC)CC 73049,N1(C(c2ccc(C)cc2)C)CCN(Cc2cnn(C)c2)CC1C 73050,c1(NCCC(C)OC)[nH]c(=NCc2cc(F)ccc2C(F)(F)F)nc2scnc12 73051,N1(C(C(CC(=C)Cl)NC(=O)C(C)C(=O)OC)=O)CC(C)(C)C2COCC12 73052,C#CCC(CC(=O)N(CC(C)NC(C1CCC(C)(O)CC1)=O)C)c1ccccc1 73053,C1(C(=O)NCC2C(C)(C)COC2)CN(C(C2CCCC2)=O)CC1(F)F 73054,c1(NC(CC2CCC(NC(CC=C=C)=O)C2)=O)cc(O)ccc1OC 73055,CC1CC(NC(C2CC3CCC2O3)=O)CN(C(=O)Cn2cnc([N+](=O)[O-])c2)C1 73056,C12(C(N3CCC(CNC(c4cc(N)c(N)nc4)=O)CC3)=O)OCCCC1C2(F)F 73057,C1(C)(CNC(C2C(=C)CC2)=O)CCCN1C(C1(c2cccc(N(C)C)c2)CC1)=O 73058,Cc1cc(Cl)c(C(=O)NC(CNC(=O)CC(C)c2ccccc2)CO)s1 73059,N1(C(COCC#C)=O)CCC2CN(C(c3cnc(OC)c(C(F)(F)F)c3)=O)CC12 73060,C1(F)(CNC(C(C)(C)c2cscn2)=O)CCC(NC(=O)C(N)=O)C1 73061,c1(CC)ccc(CNC(=O)C(=O)N(C(C)C(C)C)CC)c(O)c1 73062,C(=O)(C(O)CC(C)C)NC(COC)CC(=O)N1CCOC(C(C)(C)C)C1 73063,c1(C(N2CCC(OCCNC(C3CCC(C)S3)=O)CC2)=O)cc2c([nH]1)CCCC2 73064,c1(NC(C)=O)ccc(C(=O)N(C2CCN(C(C3C(C)C3C)=O)C2)C)cc1 73065,C1(NC(C(C)SC)=O)(CNC(C2CCN2C2CCCC2)=O)Cc2ccccc2C1 73066,c1(CC)oc(C(=O)NC(C)(CNC(c2cccc(C)c2)=O)C2CC2)cc1C 73067,c1(C(=O)NCC(=O)N(CCO)Cc2ccc(C)cc2)cccc(C#N)c1 73068,c1(-c2cn(CC(=O)NCC(CNC(CCC)=O)O)nn2)cccc(C(F)F)c1 73069,c1(C(=O)NC2C3CN(C(c4[nH]c(=N)sc4)=O)C(C3)C2)cc2cc(F)c(F)cc2[nH]1 73070,N1(C(CC(C)(C)NC(=O)C(C2CCCCC2)F)=O)CC(CO)C2(CCC2)C1 73071,N1(C(C)=O)CCCCC1CC(=O)NCC1(F)CC(NC(c2[nH]nnc2C)=O)C1 73072,N1(C(c2n(CC)ncc2)=O)CCCC(CO)(NC(=O)CN(c2ccncc2)C)C1 73073,C1(NC(=O)NCC2CC2C(C)(F)F)CCCN(C(=O)Cc2ccccc2O)CC1 73074,N1(C(c2n(C=C)ncc2)=O)CC(NC(=O)Cc2ccc(OC)cn2)CC12CCC2 73075,CC(CF)CC(=O)N1CCN(C(C2(C(=O)Nc3ccccc3)CC2)=O)CC1 73076,C(=O)(C(C)(C)CC#N)NCCN(CC(C)O)C(=O)CN1CCCC1=O 73077,c1(C(=O)NCCC2(C(=O)NCC(C)CN(C)C)CCC2)ncccc1[N+](=O)[O-] 73078,Cc1nccc(Cl)c1C(=O)NC1CC(F)CN(C(c2ccnn2C(C)C)=O)C1 73079,N1(C(C(CCC)CNC(=O)C(C)OCCOC)=O)C(C)CC2CCCC12 73080,CC1CC(CC(N2CC(C)(NC(c3cnn(CC(F)(F)F)c3)=O)C2)=O)C(C)O1 73081,c1(C(=O)NC(C)CC2CN(C(C3CCCO3)=O)C2)ccc(=O)n2c1CCCCC2 73082,N1(C(C(C)C)=O)CC2(C1)CN(C(c1cccnc1-c1ccccc1)=O)C2 73083,CCCCC(C)(F)C(=O)NCCC1CSCCN1C(=O)CN(C(=O)COC)C 73084,c1(C(C(=O)OC)NC2CC(=O)NC2=O)cc(Cl)cc(Br)c1 73085,Cc1c(C(N2CCCC2CNC(C2CC23CCSCC3)=O)=O)nn2c1CCCC2 73086,C1(NC(=O)CCc2cccs2)CCCC1CC(=O)NCCc1ccsc1 73087,C(=O)(C(CNC(C)=O)NC(C1CC1(Br)Br)=O)OC 73088,C1(C(=O)NC2C(NC(C3OCC(C)(C)C3)=O)CCCCC2)CC2C=CC1C21CC1 73089,N1(C(CCNC(=O)Cn2ccccc2=O)=O)CC2C3C=CC(O3)C2C1 73090,C(=O)(CC1=CCOCC1)NC1CC(CNC(CC2(COC)CC2)=O)CC1O 73091,Cc1cnc(N2CC(O)(CCNC(=O)C=CC(C)(C)C)C2)nc1O 73092,c1(OC)c(OC)cc(C(=O)NCC(O)CNC(C2CC3(C2)CC3F)=O)cc1Cl 73093,N1(C(C(C=C)OC)=O)CCC(CNC(c2cnncc2NC)=O)C1(C)C 73094,c1(C(N(CC(CNC(Cc2c(C)cco2)=O)C)C)=O)c(C)nsc1C 73095,C1(NC(C(C)N2CCC2)=O)COCCN(C(c2c(Cl)csc2Cl)=O)C1 73096,N1(C(CN(C)C)=O)CC(NC(C2CC(=O)N(CCN(C)C)C2)=O)CC(F)C1 73097,C(=O)(CC1OCCc2ccsc21)N(C)CCNC(=O)C(C)(C)c1sccc1Cl 73098,Cc1nn(CC(=O)NCC2=CCN(C(c3cc(N)cc(N)c3)=O)CC2)c(C)c1C 73099,C#Cc1ccc(OCC(N2CCOCC2CNC(C2CCCN2N=O)=O)=O)cc1 73100,N1(C(c2cc(C)[nH]n2)=O)CCC2CCN(C(=O)C3=CSCS3)CC12 73101,C(C1CCCN1C)=CC(=O)N(CCCNC(C(C)=C1CC1)=O)C(C)C 73102,Cc1cccc(C2(C(=O)NC(C)CC(C)NC(=O)CCN3CCCC3)CC2)c1 73103,c1(C(N2CC(CNC(C3CC(O)C3)=O)C3(CC3)C2)=O)cc(Cl)ccc1OCCF 73104,c1(C2C(CC(N3CC(C(C)NC(=O)CN4CCCC4=O)C3)=O)C2)ccc(Cl)cc1 73105,C1(CCNC(C2C(C)C2)=O)CCN(C(=O)OC(C)(C)C)CC1(F)F 73106,C1(O)(C(C(=O)NCCN(C2CCCCC2)C(CCOC)=O)(F)F)CCOCC1 73107,Cc1cccc(C(=O)COC(c2cc(-c3ccoc3)[nH]n2)=O)c1 73108,c1(C(N2CC(C3(NC(C4N(C)CCC4)=O)CC3)C2)=O)cc(F)c2cn[nH]c2c1 73109,c1(CC(=O)NC2C(NC(=O)C#CC3CC3)CCCC2)cc(F)cc(Br)c1 73110,O=C(C1=CCCS1)NCCN1CCN(C(=O)C(=O)Nc2ccncc2)CC1 73111,C1(CNC(C(C(C)C)O)=O)CC12CCN(C(=O)CCNC(C1CCC1)=O)CC2 73112,C1(NC(C=C(Cc2c(OC)cccc2)C)=O)CC2CC(NC(=O)C=C(C)Cl)CC12 73113,N1(C(C(CCN(C)C)O)=O)CC2C=CC1C(C(N1CC(NC(N)=O)C1)=O)C2 73114,c1(CN2C(C(N3CCC3CO)=O)CC3CC32)cc(F)c(O)c(F)c1 73115,N1(C(C2(C)CS(=O)(=O)C2)=O)CC2=C(C1)CN(C(c1cnn3c1SCC3)=O)C2 73116,N1(C(=O)CSc2cccs2)CC2OCCN(C(c3cc(CO)on3)=O)C2C1 73117,N1(C2CC3(NC(c4ccc(OC(F)F)nc4)=O)C(C2)C3C)CCSCC1CCO 73118,N1(C(CNC=O)=O)CC(n2cccc2)C1 73119,c12ncc(o1)NC2C1CCC1.C(C(Cl)=CCl)NC(=O)OC(C)(C)C 73120,c1(C(=O)NCC(C(C)C)(C)C(C)C)cccc(N=c2cncc[nH]2)c1 73121,CC(C)(F)CCC(=O)NCC1CCCC1NC(c1cnoc1-c1ccccc1)=O 73122,CCCCCCCCCC(=O)NC(C)C(C)NC(C1CC=C(C)CC1)=O 73123,CCC(CS(=O)(=O)c1ccc(C)c(C)c1)NC(=O)CS(=O)(=O)c1ccccc1F 73124,c1(OC(=O)NCC(C(C)C)NC(C=CC)=O)cnc(O)n(-c2ccccc2)c1=O 73125,N1(C(Cc2c(C)noc2C)=O)CC2CCCC2(NC(c2cc(C(F)F)no2)=O)C1 73126,N1(C(C(C)=C2CCOC2)=O)CC2CCC(CNC(=O)CCC3CCCCC3)C2C1 73127,N1(C(CC2C(C)(C)C2(C)C)=O)CCC(NC(=O)CCNC(C2CCC2)=O)C(O)C1 73128,C1(C(N2CCC(CNC(COC(CC)(C)C)=O)C2)=O)CCN(C2CC2)S1(=O)=O 73129,Cc1cc(Cl)cc(C(N2CCCN(C(C3C4CCC3(C)C4(C)C)=O)CC2)=O)c1O 73130,CCCCC(CNC(=O)Cc1csc(S)n1)NC(c1cc(O)no1)=O 73131,C=CCC(CC(F)F)C(=O)N1CC2CC(C1)N(C(=O)CC1CCCN1C)C2 73132,N1(C(c2c(C)coc2)=O)CCCC(C2CN(C(=O)CCCc3ccncc3)C2)C1 73133,C1(CCOC)CN(C(c2cc(C)cc(O)c2)=O)CCN1C(=O)C(C1CCC1)OC 73134,S(=O)(=O)(c1ccc(-c2ccc(Cl)s2)cc1Cl)NCc1c(C#C)cccc1 73135,C1(CNC(CCCCN(C)C)=O)CC2CCC1N(C(c1nc(Cl)sc1Cl)=O)C2 73136,CC1CN(C(c2cc3n(n2)CCCC3)=O)CCN(C(=O)COC(C)(C)C)C1 73137,CCC(CNC(=O)CNC(=O)C=Cc1ccsc1)(CC)NC(=O)CCC 73138,c1(NC(C)CN2CCCC2=O)nc(N(C)CCn2cnnc2)nc2c1CCC2 73139,CC1CC(CCC(=O)NC2CN(C(=O)CCc3ccn(C)n3)C2)C(C)N1C 73140,C1(C(N2CC(C(C(N3CCC(C(=O)NC)CC3)=O)OC)C2)=O)CCCCCN1C 73141,c1(C(N(CC(CC)NC(c2ccc(CO)s2)=O)C)=O)c[nH]nc1Br 73142,c1(C(=O)NCC2(CN(C)C(C3CCC4CC34)=O)CC2)cc(S(=O)(=O)N(C)C)c[nH]1 73143,C1(C(c2n(CC=C)nnn2)NCc2cncn2CCC)CCC2(CC1)CC2 73144,C(C(CC)(CC)C(=O)N1CCC12CC(O)C2)NC(c1cc(CC)ncn1)=O 73145,C=CCCCC(=O)NCCCN(C(=O)CC1CCC(C)CO1)CCO 73146,C1(CNC(C)CS(C)=O)(NC(=O)OC(C)(C)C)CC12CCC2 73147,N1(C(c2nnc(C)s2)C(=O)NCc2cccs2)CCn2ncc(Cl)c21 73148,c1(CC)ccccc1CC(=O)NCC(C)CN(C)C(C1CC1c1nccn1C)=O 73149,Cc1nc(C(c2nnnn2CCN2CCOCC2)NCC2CCOC2)nn1C 73150,c1(C(C(=O)NCC=C)N(CC=C)C2CC2)ccc2nonc2c1 73151,n1(C(C)C)cc(C(N2CC3CC2C3CNC(=O)C(C)C2CC2)=O)c(O)nc1=O 73152,c1(C(N2CC(NC(=O)C3CC3)C(F)CC2)=O)ccc2oncc2c1 73153,N1(CC(C2C(C)(C)C2(F)F)=O)CCCC2(C1)OCC(O)C2O 73154,C1(CN(C(=O)C=Cc2ccco2)CC)CCCCN1C(=O)CSc1ccccc1 73155,N1(C(C2N(C(CC(COC)(C)C)=O)CC3(CC3)C2)=O)C2CCC1CC(O)C2 73156,N1(C(C(F)=CCC)=O)CC(C(=O)NCC(=O)OC)C2(CCC2)C1.C1CO1 73157,Cn1ncc(C(=O)NCc2csc(CNC(C3C=CC=CC=C3)=O)n2)c1F 73158,C(=O)(CC(O)CNC(C1(O)CC(CF)C1)=O)N1CCC(OCC(N)=O)C1 73159,C(C1CN(C(=O)C=Cc2ccoc2)CC1C(=O)NC1(C(F)(F)F)CC1)=CC 73160,c1(C(c2nnnn2C)NCC#CC)ccnc2[nH]c(C(F)F)nc12 73161,C1(CNC(Cc2cc(C)no2)=O)CCN(C(=O)CCCF)CC1O 73162,N1(C(Cc2nc(CC)sc2)=O)CCOC(C)(CNC(c2cc(C)cs2)=O)C1 73163,c1(COC)cc(C(=O)NCCCCN(C)C(C2CC2c2cncn2C)=O)no1 73164,Cc1ccc(O)c(CN2CCC(C)(C(=O)NCc3cc(F)cc(Br)c3)C2)c1 73165,c1(CC)[nH]c(Cl)nc(=NC(C)CNC(C23CC(C)(CO2)C3)=O)c1C#N 73166,c1(C(=O)NC(C)CCNC(=O)Cc2ccccc2CC#N)ccc(N=[N+]=[N-])cc1 73167,c1(CC)nc(O)c(C(=O)NCC2CN(C(=O)C(C)COC)C2)cc1C 73168,N1(C(C2CC(=C3CC3)C2)=O)CCC2OCCN(C(=O)Cc3ccc(F)cc3F)C2C1 73169,N1(CC)CCCC(CC(N2CCC(C(=O)Nc3ccc(SC)cc3)CC2)=O)C1 73170,N1(S(C2CCC(=O)CC2)(=O)=O)CCC(C2CCCN(C(=O)C(O)C(F)(F)F)C2)C1 73171,Cc1ccc(NC(=O)C(Cc2ccccc2)NCC(F)(F)F)cc1I 73172,c1(OC)ccc(O)cc1CN1CCC(F)(C(N2CCC(C(F)F)CC2)=O)C1 73173,c1(C(N2CC(NC(C(C)=C(CC)C)=O)C(C(F)(F)F)C2)=O)c[nH]c2cccnc12 73174,N1(c2ncc(C#N)cc2F)CCC2CCN(C(=O)CN3CC4CCC3C4)CC2C1 73175,C1(CC)(CC)CC(NC(=O)CN=S(C)(C)=O)CN1C(c1ccc(N(C)C)nc1)=O 73176,N(S(=O)(=O)N1CC(C#N)C1)Cc1c(OC)cc(OC)c(C)c1 73177,CC1(C)CCCN(C(=O)COCC(F)F)C1CNC(=O)COc1ccncc1 73178,c1(OC)ccc(C(=O)NC2CN(C(=O)CC3COC4CC3C4)CC2OC)cc1O 73179,c1(C(=O)NC(CC)CN(C(=O)C(C)(C)C(C)C)C)cccc([N+](=O)[O-])c1 73180,C(=O)(CC(=O)NCCOC(C)(C)CNC(=O)CCN(S(C)(=O)=O)C)N(C)C 73181,C1(C(=O)NC2CC(NC(CS(CC)(=O)=O)=O)C2)CCCC2(CCC2)C1 73182,c1(OCCNC(N2CC(C=C)OCC2)=O)cccc2ccccc12 73183,C1(c2onc(C)n2)CCCN(c2nccnc2N2CCC(C)CC2)C1 73184,c1(C(=O)NC23CCN(C(CCC(=O)NC)=O)CC2C3)cnn2cc[nH]c(=O)c12 73185,C(=O)(C(F)(F)C(C)O)NC(C(=O)NCc1nnn(CC)n1)CC1CC1 73186,c1(C(=O)NC2C(CNC(c3c(CC)noc3)=O)CC2)ccnc2ccncc12 73187,Cc1ccc2c(C(=O)NCCC3CCCN(C(C4(O)CCOC4)=O)C3)csc2c1 73188,C1(C(N(C2CCC(NC(C3CCNC3=O)=O)CC2)C)=O)CCC(C)(C)O1 73189,C(=O)(C(C)(C)C(=O)N1CC(CNC(c2cnc(C)[nH]2)=O)C2(CC2)C1)NC 73190,C(C(C(C)C(C)C)NC(c1cc(C)n(C)c1C)=O)NC(CCN(CC)CC)=O 73191,C1(NC(C(C)OC(C)(C)C)=O)(CNC(C2CCCN2C=O)=O)CCCCCC1 73192,C=C=C(C)CC(=O)N(CC(C)O)CCNC(c1cn(C)nc1C(F)F)=O 73193,c1(CCC)[nH]nc(C(N2CC3C(NC(=O)C(C)C)C3C2)=O)c1[N+](=O)[O-] 73194,C=CCC(C)C(=O)NCC1(O)CC(CNC(=O)C=Cc2cc[nH]c2)C1 73195,C1(NC(c2c(C)cc(C)o2)=O)C2CCN(C(=O)Cn3c(C)csc3=O)C2C1(C)C 73196,N1(C(Cc2ccc(C)cc2)=O)CC2OCC(NC(c3coc(C(F)F)n3)=O)C2C1 73197,CCC(O)C(C)(C)C(=O)NCC(O)CCNC(=O)CCCCN(C)C(C)C 73198,N1(C(C2(C)CN(C(c3sccc3I)=O)C2)=O)CCC(N2CCCC2)CC1 73199,C1(NC2CC(N(CC(COC)C)C)C2)CCCN(C(N)=O)C1 73200,c1(OC)ccc(Cl)cc1S(=O)(=O)NC1CN(Cc2c[nH]c3c(F)cccc23)C1 73201,c1(-n2c(C(=O)NC(C(=O)OCC)CC)ncc2)cccc(Cl)c1 73202,N1(C(C)=O)CCCC1CC(=O)NCC1CCC(NC(=O)C(C)OCCC(C)C)C1 73203,N1(C(CCCC)=O)CC2CCCC2(C(=O)NC(C2CCCC2O)C)C1 73204,N1(C(C2=C(C)OCCS2)=O)CCCC2CN(C(C3(O)CCSCC3)=O)CCC12 73205,c1(C(=O)NCCCN(C(=O)CC(C)C)CC)cc(Cl)n[nH]1 73206,c1(CC(N2CCC(O)(CN(C(C(CC)SC)=O)C)C2)=O)ccc2cnccc2c1 73207,C1(C(=O)NCC(=O)OC23CC(F)C2C3)CC2(CCCC2)CO1 73208,C1(NC(C(C)OCCCC)=O)CCN(C(=O)Cc2cc[nH]c(=N)c2)CC1C 73209,CC(CN=c1[nH]c(=NC2COC(C3CC3)C2)[nH]c2ccc(Cl)cc12)c1cnc[nH]1 73210,Cc1cnc(C(N2CCC(C(C)(C)C(=O)NCc3cncc(F)c3)C2)=O)cn1 73211,C1(CC(=O)NCC2CN(C(C3CC34CCOC4)=O)C2)CCC=CCC1 73212,C1(CC(=O)NC(C)CNC(C2C3(CC3)C23CC3)=O)COC2(CCC2)CO1 73213,CC1CCC(NC(=O)Cc2ccccc2)CN1C(=O)Cc1cccc(Cl)c1 73214,C1(CN(C)C(c2cc(F)n[nH]2)=O)CCCN1C(=O)CCc1nc[nH]n1 73215,c1(C(=O)NC(CN(C(C2CC2CC(C)C)=O)CC)C)c(Br)ccc(F)c1N 73216,c1(OC)ccc(C(=O)NCC(C2CCC2)NC(=O)Cc2cncc(C)c2)c(F)n1 73217,CC(C)CC(C)CC(=O)NCC1(F)CCC(NC(c2ccc(F)cc2)=O)C1 73218,C1(C(=O)Nc2ccc(OC)c(C(F)(F)F)c2)CC12CCN(C(=O)C(F)F)CC2 73219,c1(C(N2CCC(O)(CC#N)C2)C(=O)NCCCF)cc(I)ccc1F 73220,c1(CCC(=O)NCCOCCNC(C2CCN2C2CCCC2)=O)cccc(O)c1 73221,C12(CNC(=O)Cc3csc(Cl)n3)CCC(CC1)N(C(c1cc(F)cnc1O)=O)C2 73222,C1(C(N2CC(n3cc(CNC(CNC(C)=O)=O)nn3)C2)=O)CCCC(C)(C)CC1 73223,c1(CCC(=O)OCC)c[nH]c2c(C)cccc12.N12CCCC1CCC2=O.N(C)(CCC)C 73224,C(=O)(C1=COCCC1)NC1C(C(=O)NCCn2c(C)ncc2)CCOC1 73225,C12(NC(c3cccn4ncnc34)=O)CCCC1N(C(=O)C1=NOCC1)CC2 73226,N1(C(c2ccc(N)cc2F)=O)CC2CCC(C1)N2C(C1CCCCS1)=O 73227,c1(CC(=O)NCCN(C(=O)C(C)(C)C2CCOCC2)C)ccc2nn(C)cc2c1 73228,Cn1cncc1C=CC(=O)NC(C1CCCCC1)CNC(C1COC(=O)O1)=O 73229,N1(C(c2n[nH]c(CC)c2Cl)=O)CC(NC(C23CC(C#N)(C2)C3)=O)CC12CCOC2 73230,N1(Cc2cnn(CC)c2C)CCC2CN(C(c3cc(OC)ccn3)=O)CCC12 73231,c1(CNCCOCC(N(OC)C)=O)cc(F)ccc1N(C)C1CC1 73232,N1(C(c2c(Br)cn(C)n2)C(=O)NC2CC2)CCC(C(N)=O)(C(N)=O)CC1 73233,N1(C(C(C=CC)O)=O)C2CCC1CN(C(=O)CC(C)(C)O)C2 73234,C(=O)(C1=NOC2COCC12)NCC(CC(=O)Nc1ccc(C)nc1C)O 73235,C#CC1(C(=O)NCc2ccccc2CC)CN(C(c2cn(C)cn2)=O)C1 73236,c1(C(N2CCC(CCNC(=O)CSC3CC3)C2)=O)ncn2c1CCCC2 73237,C1(NC(c2[nH]cc(C(C)=O)c2)=O)CCOC(C(=O)NCC=C2CCC2)C1 73238,c1(C(=O)NC(CC(C)NC(c2c(OC)c(Cl)sc2)=O)C)ccc(F)c2[nH]ccc12 73239,CC1CC(N(C(=O)C(=O)NCc2cccc(C(C)(C)C)c2)CCO)CCO1 73240,CCCC(C)(O)C(=O)NC1CCCC(NC(C2CC(F)(F)C2)=O)C1 73241,N12CCCC(C1)OOCC2=O.C(=O)(C(CC)OC)NCC1(CCOCC)CC1 73242,C1(C(N2CC(C3(NC(CCN(CCC)C)=O)CC3)C2)=O)CC2OC(C)(C)OC2C1 73243,c1(C(N2CC(Nc3ncc(C)cn3)CC(C)(C)C2)=O)cnc(O)c2ccsc12 73244,N1(C(C(C)Cn2ccnc2)=O)CC(NC(c2c(Cl)cnn2C(C)C)=O)C(O)C1 73245,c1(COC(C)C)nc(-c2cccc(C(C)C)c2)n(-c2ccccc2)n1 73246,C1(C)(C(=O)NC2C(NC(Cc3ccn(C)n3)=O)CC2)CCC12CCC2 73247,CC1(CNC(C2C(CNC(=O)CCN=[N+]=[N-])C2(C)C)=O)CCCCO1 73248,N1(C(c2cc(C)c(C)o2)=O)CCCCCC(Nc2ncc3ncn(C)c3n2)C1 73249,c1(CCCC)nc(C(C)P(C)(C)=O)n(-c2cc(C)ccn2)n1 73250,C1(O)(CNC(C(CC)NC(C)=O)=O)CCCN(C(C2CC(=C3CCC3)C2)=O)CC1 73251,Cc1cccc(C(C(=O)NCCCF)N(CCC(C)C)C(c2ccccc2)C)c1 73252,c1(CC(N2CCCN(C(C(C)NC(CC)=O)=O)CC2)=O)coc2ccccc12 73253,c1(C(c2n(C(CC)(C)C)nnn2)NC2CC3(CC3)C2)cc(C)ncn1 73254,c1(SCCNC(CC(C)(C)C)c2n(CCCOC)nnn2)cc(C)ccc1F 73255,C(=O)(CCCS(N)(=O)=O)N(CCC(C(C)C)NC(Cn1nc(C)n(C)c1=O)=O)C 73256,c1(C(N2CCOCC(F)(CNC(CSCC=C)=O)C2)=O)cccc2c1CNC2=O 73257,N1(C(CCCCN(C)C)=O)CCCCCC(NC(c2nc3ccccc3[nH]2)=O)C1 73258,C1(C=O)(COC)CCCC1.N1CCC(CNC(c2n[nH]cc2C2CC2)=O)C1 73259,c1(C2(C(=O)NCC(CN(C)C(C3CC3(Cl)Cl)=O)O)CCC2)ccc(Cl)cc1 73260,C1(C(N2CC(CC(C)NC(C3CCCCC3O)=O)C2)=O)C2CC3CC(C2)CC1C3 73261,C1(NC(c2c(CCC)occ2)=O)CC(C)CN(C(c2ccn(CCO)c2C)=O)C1 73262,N1(C(C2C3(CC(OCC)C3)C2)=O)CC2CC(NC(=O)C(=O)C(C)(C)C)C1C2 73263,CC(C)(CC(F)C(=O)NCC1(CF)CC1)NC(=O)CC1CNC(=O)O1 73264,c1(C(N2CCN(C(=O)C(O)C(F)(F)F)C(C(F)F)C2)=O)cc2ccc(Cl)nc2s1 73265,c1(N2C(C(=O)NC(C)Cc3cnn(C)c3)CCC2)ncncc1Br 73266,c1(-c2nc(CCCC=C)n(CC(C)CO)n2)ccc(OCCOC)c(Cl)c1 73267,CCC(CC)(CC)C(=O)NCC(C(C)C)NC(c1ccc(S(N)(=O)=O)s1)=O 73268,c1(OC)ccc(C(=O)Nc2ccc(C(=O)C(F)(F)F)cc2)c(O)c1F 73269,c1(SC)nc(N2CC(F)(C(=O)Nc3cc(I)ccc3F)C2)ncc1Br 73270,c1(C(C)C)sc(Cl)nc1C(=O)NC(C)CCN(C(=O)C(C1CCOCC1)O)C 73271,C(CNC(=O)CC1CC2(CC2)CO1)(CC(=O)NC)OC.C1(C2CCC2)CCCC1 73272,C1(C)(C(=O)NCC(C)(CNC(=O)C(C)=C(C)C)OC)CCC(C)C1 73273,CC(CC(F)(F)F)C(=O)N1CC(CC(=O)NCC(C)C2CCC2)CC1(C)C 73274,c1(C(=O)OCC)c[nH]nc1S(=O)(=O)NC(CCSC)C(=O)OC 73275,N1(C(CN(C(C(CC)OCC)=O)CCOC)=O)CCCC(C(=O)OC)C1 73276,c1(C(=O)NC(C)CCCCNC(c2ccon2)=O)c(Cl)oc2ccccc12 73277,c1(OC)ncnc(C(=O)NCC2CCCCC2NC(=O)Cn2cnnc2O)c1F 73278,C(=O)(C(CO)C(C)(C)C)NCC1(C)OCCN(C(c2cnc(C(C)(C)C)[nH]2)=O)C1 73279,N1(C(c2nc(C(C)OCC)sc2)=O)CCC(C)(NC(=O)CS(=O)CC)CC1 73280,N#CCCCCCC(=O)NCCC1CN(C(=O)Cn2cc(CO)nn2)CCCO1 73281,c1(C(=O)NCC(CNC(c2ccc(C)s2)=O)(C)C)cc(C(F)(F)F)ccc1O 73282,CC1CCCC(C(=O)NC(c2ccc(Br)cc2)(C)C(=O)O)O1 73283,c1(C(N2C(CCNC(C3CC(CC)C3)=O)CCC2)=O)ccc(N)c(F)c1Br 73284,c1(OC(C(N2CC(N(C(C(C=CC)O)=O)C)C2)=O)C)cc(Cl)cc(Cl)c1 73285,Cc1cccc(C(C)C(=O)NC2CCC2NC(c2cnn(-c3nccs3)c2)=O)c1 73286,C(=O)(CCC(C)(C)[N+](=O)[O-])NCc1c(OC)ncnc1OC 73287,c1(NC(C2CC(O)(CNC(c3cscc3C3CC3)=O)C2)=O)ccc(CCO)cc1 73288,N1(C(C#CC(C)C)=O)CCC(CO)(CNC(C23CCC(CO2)C3)=O)CC1 73289,C#CC(CNC(=O)CCCCNC(C1(O)CCOC1)=O)C(C)C 73290,c1(C(=O)NC(CCCNC(COCCOCC#C)=O)C)ncnc2cc[nH]c12 73291,C1(CNC(C=C(C)C(C)C)=O)CCCCN1C(C1CN(C(=O)OC(C)(C)C)C1)=O 73292,C(=O)(C1CCCc2scnc21)NC1C(CNC(c2c[nH]c(=NCC)s2)=O)CCC1 73293,CC1COCCN(C(C2CNC(=O)CN2C(=O)CC(Cl)Cl)=O)C1 73294,CCCC(C)CCCC(=O)NCC1(F)CCC(CNC(=O)C(F)(F)C2CC2)CC1 73295,C(=O)(C(C#N)(CC)CC)NC(CC)CNC(C1CCC(CN2CCOCC2)CC1)=O 73296,N1(S(CC)(=O)=O)CCN(C2CC2)CC1.C12CCCC1NC(=O)C(=O)N2 73297,C1(NC(C(C)=CC2CC2)=O)CCCC(NC(c2c(C)noc2C(C)C)=O)C1 73298,C1(CNC(=O)CCCc2cnccn2)C(F)(F)C12CC2 73299,c1(NC(CC=C)C)[nH]c(=NCc2cnc[nH]2)nc2c1ncn2C 73300,C(=O)(C1CCOc2ccc(Cl)cc21)N1CC(C)CC(NC(C=CC)=O)C1 73301,C1(NC(c2cc(CNC(=O)C(c3cccnc3)O)cs2)=O)CCC2(CC2)C1 73302,C(CC(CNC(c1cc(C)co1)=O)NC(=O)C=CC1CCCO1)OC 73303,CCCCC(C)(F)C(=O)NC1CCCCC1NC(c1ccc(F)cc1)=O 73304,C1(C(=O)Nc2ccc(C(C)C)cc2)CN(C)CCN1C(=O)C(F)C(F)(F)F 73305,C(=O)(C1=CC2(CCOC2)C1)NC(C(=O)N(C(C#C)C1CCC1)C)CC1CC1 73306,c1(C(=O)NCC(CC(N2CCCC(CC)C2)=O)O)n[nH]cc1[N+](=O)[O-] 73307,C(=O)(C1=CS(=O)CCC1)NC12CC(NC(CC(=O)NCC#C)=O)(C1)C2 73308,CCC(C)C(C(=O)NCC(C)(C)CCOC)NC(c1ccccc1NC)=O 73309,c1(C(c2n(CC=C)nnn2)NCc2ccc(NC)cn2)cccc2c1CCC2 73310,N1(C(C(C)N(C(C)=O)C)=O)CCC(C2CCN(C(C3(F)CCCC3)=O)CC2)CC1 73311,N1(C(C(C)(C)SC)=O)CCCN(C(=O)Cc2ncc(Cl)s2)C(C)C1 73312,CCC(C(=O)NCC1(F)CCN(C(c2cc(OC)n[nH]2)=O)CC1)C(C)O 73313,C1(C(=O)NC(c2nc(SCC3CCCO3)on2)(C)C)CCCCN1S(C)(=O)=O 73314,CC(C)(C)CCCN=c1ccc(S(=O)(=O)NCCCCC2CCCC2)c[nH]1 73315,c1(C(=O)NC)c(C)nc2cc(O)nn2c1C.C1(C)C(=O)N1CCCNC(CC)=O 73316,CCC(C(=O)N(CC(C)(C)CNC(=O)C(Cc1ccsc1)NC=O)C)C(C)C 73317,c1(OC)cc(C(=O)NC(C2CCCCN2C(=O)CC(C)(C)C)C)cc(Cl)c1O 73318,C(=O)(C#CC(C)(C)C)NCC1C(C(N2CCC(CCC#C)CC2)=O)C1 73319,c1(C(N2C(C)CC(CNC(c3n[nH]c(C)c3N)=O)C2)=O)cnn2c1CCCC2 73320,C(C)(Cc1ccccc1)(CC(C)C)NC(C(C=C)CC)=O 73321,C(=O)(CC(C)(C)C)NC1(NCc2nc(-c3ccn(C)n3)sc2)CC1 73322,c1(OC)ccc(O)c(CNC2CCN(C(c3ccc(OC(C)C)cn3)=O)C2)c1 73323,N1(C(=O)OCC=C)CCN(C(=O)CCn2cc(C3CCCC3O)nn2)CC1 73324,C(=O)(C(C)CS(C)(=O)=O)NCC1CCCCN(C(CCCc2ccc(C)s2)=O)C1 73325,N1(C(CN(C)CC)=O)CCC(NC(=O)CS(=O)(=O)N2CCOCC2)CC1C1CC1 73326,C1(NCc2c(C)c(C(F)(F)F)n[nH]2)CC2(CCC2)C12CCC2 73327,S(=O)(=O)(c1ccc(N2CCN(SC(F)(F)F)CC2)nc1)NCC(C=C)(C)C 73328,N1(C(CCC2(NC(c3cncc(O)c3)=O)CCC2)=O)CC2C(CO)C2C1 73329,C1(CNC(C2CC(SC)C2)=O)COCCN(C(c2ccccn2)=O)C1 73330,c1(C(N(CC(C)NC(c2cnc(C3CC3)s2)=O)CC)=O)ccc2ncn(C)c2n1 73331,C12(NC(CCSCC)=O)CCN(C(=O)CN3CCCCCC3)CCC1C2 73332,c1(C(=O)NCCC(=O)NCC)n[nH]cc1CNC(=O)COCC1CC1 73333,C=CCC(CC(=O)NCC(O)C1(Cl)CC1)NC(=O)C=CC 73334,c1(OC)ccc(NC(C2CC(F)(F)CN2Cc2scnc2C)=O)c(Cl)n1 73335,C(=O)(C(O)C(C)C)NCCC(C)NC(C(CC)c1ccccc1)=O 73336,N1(CC(N2CC(CN(C(C(C)SC(F)(F)F)=O)C)C2)=O)CCCC(N(C)C)C1 73337,C(C(=O)N(C)CCN(C)C(C1(Cl)CC1(C)C)=O)(C(C)C)n1cc(C)nc1 73338,c1(C(CNC(C23CC(C)C2C3)=O)N(C(=O)Cc2nnc(O)s2)C(C)C)cccc(Cl)c1 73339,CC(CC(C)(C)O)C(=O)OCn1cc(Cc2ccc(C(CCO)N)cc2F)nn1 73340,c1(NC(CC)C)ccc(S(=O)(=O)NCc2nnnn2-c2cn[nH]c2)cc1Br 73341,c1(C(=O)OC)cc(CC(=O)C(F)(F)C(O)c2ccccc2)n2ccccc12 73342,CCC(C(O)C(C)C)NC(c1ccc(NC(=O)N(C2CC2)CC)cc1)=O 73343,CCCCCCCCCCCCN(C(=O)Cc1ccc(OCCC(C)C)cc1)C 73344,C1(NC(C2(CC)CC2)=O)CN(C(c2cccc(OC)n2)=O)CC2CCCC12 73345,N1(C(c2ccc(NC(C)=O)s2)=O)CCC(C)(C)C1CNC(C1CC(=O)N(C)C1)=O 73346,c1(CNC(C(=O)N(C)Cc2cc3ccccc3s2)=O)cc2ccnc(Cl)c2o1 73347,C12(C(N3CCC(NC(CNS(NC)(=O)=O)=O)C3)=O)CCC(=O)N1CCS2 73348,c1(C(=O)NCC2(NC(c3cc(C(F)(F)F)c[nH]3)=O)CC2)c[nH]cc1C1CC1 73349,C(=O)(C(C)CC(F)(F)F)N1CCC(NC(c2c(OCC)noc2C2CC2)=O)C1 73350,CC1(C)CCCC(O)(CNC(=O)Nc2ccc3ccoc3c2)C1 73351,CC1CCN(CC(=O)N(CC(C)NC(C2(C)CC2c2ccccc2)=O)C)CC1 73352,C1(CCC(=O)NC(C)C(C)NC(=O)CN(C)C(=O)OC(C)(C)C)CCCOC1 73353,N1(C(C(C)CC(F)F)=O)CCC2C(CCCN2C(=O)CC2(O)CCCCC2)C1 73354,c1(CNC(NC(COC)C)=NCC2CN(C)CCO2)nc2c(s1)CCC2 73355,N1(C(C2CCC(CC)O2)=O)CC2CCC2(CC(=O)NCCc2ccc(C)cn2)C1 73356,c1(C(CCC)C)cn(CC(=O)OC)nn1 73357,CCS(=O)c1ccccc1C(=O)NCCOC1CCN(C(=O)CC(C)SC)CC1 73358,C1(NC(C(c2cc(C)oc2C)C)=O)CC2CN(C(=O)CCc3cn[nH]c3)CC2C1 73359,C(CCCC(=O)NSC1CCC(C#N)C1)CCOC.C1(=O)ON1 73360,C1(C(N2CC(NC(C3(C)CCCC3)=O)C2)=O)CCC(N=[N+]=[N-])C1 73361,CN1C(=O)Cc2c(C(=O)NCC3C4CN(C(=O)Cn5cnnn5)CC34)cccc21 73362,c1(N2CCOCC(NC(C(C)c3ccsc3)=O)C2)c(F)cccc1[N+](=O)[O-] 73363,C(=O)(C(C)CCC(C)(C)C)NC1CCN(C(C(=O)NC(C)C)=O)CC1 73364,C1(Cn2cc(COC)nn2)CCCCN1C(=O)CC(C)c1cnn(C)c1 73365,C1(CC(N2CC(NC(C(C)(C)n3cccn3)=O)C(CO)C2)=O)CCCNC(=O)C1 73366,C1(N(C(C2CCN(CC(C)C)C2)=O)C)CN(C(=O)CCc2ccco2)CC12CC2 73367,C1(C(=O)NC2CCCC(O)C2)CN(C(c2ccnn2C2CC2)=O)CC1(F)F 73368,N1(C(C2(COC)CC2)=O)CCC(OCCNC(=O)CC2(C)CCC2)C1 73369,c1(OCC)ccc(C2(CNC(c3c[nH]nc3F)=O)CCC2)cc1.C12(CC1)C(=O)N2 73370,N(C1CCCc2c[nH]nc21)C(c1c(C)nc(CNC(C2C(CC)C2)=O)o1)=O 73371,c1(-c2nc(-c3scc(C)n3)nn2C2CCCCCC2)cc(S(N)(=O)=O)c(C)cc1C 73372,N1(C(C(CC)CC)=O)CCC(C2(CNC(=O)C3CC3)CCOCC2)CC1 73373,N1(C(c2cn(C(C)C)nc2)=O)CCCCC1CCN(C)C(C1CCCOC1C)=O 73374,C1(C(N2CCC(C(F)(F)F)(OC)C2)=O)CCN(C)CC1C(F)(F)F 73375,CC(C)CCC(CO)NC(C1CC(CNC(c2coc(C(F)F)c2)=O)C1)=O 73376,N1(C(c2c(C)nsc2C)=O)CCC(C)C(CC(N2CCCCC2CCO)=O)C1 73377,C1(NC(c2c(C)onc2-c2ccc(C(F)(F)F)cc2)C)CCC(F)(F)CC1(C)C 73378,C(=O)(C(C(C)(C)C)c1cc[nH]n1)N(CCN(C(=O)CCOC1CC1)C)C 73379,c1(C(=O)NCCOCCNC(C2CN(S(CC)(=O)=O)C2)=O)ccn(CC(C)C)n1 73380,CC(C(=O)NOCCN(C)C)C1CCCN(C(C2CN(C(N)=O)C2)=O)C1 73381,N1(C(c2c(CC)noc2)=O)CCCC(C2CCN(CCOC3CCCC3)C2)C1 73382,C(C1=NOC2CN(C(C3(C4CC4)CCOCC3)=O)CC12)NC(c1cccnn1)=O 73383,C(C(C)(C)CC(=O)NCC1(CNC(C2(F)C(C)(C)C2(C)C)=O)CCOCC1)OC 73384,C(=O)(C1=CCCCCC1)N(C(C)C(=O)Nc1cc(Cl)cnc1C)CC 73385,C=CC1(NC(C23CC2CN(C(C2CCC(O)C2)=O)C3)=O)CCCC1 73386,N1(C(C=C2CCN(C)C2)=O)CCC(NC(=O)CC2(C)CC(F)(F)C2)C(O)C1 73387,c1(C(N(CCCNC(C2(C=C)CCCCC2)=O)CCO)=O)cn2cccnc2n1 73388,c1(C(=O)NC2CCC(NC(C3(C4CC4)CC3)=O)CC2)cc2ccncc2o1 73389,CC(C(=O)NC1(C)CCCN(C(c2cccc(Cl)c2F)=O)C1)C(C)(F)F 73390,C(CCCCC(=O)NC1(C(=O)NOCC2(C)CC2)CCCCC1)NC(C)=O 73391,Cc1nc(S(C)(=O)=O)sc1C(=O)OCC1CC(C(=O)OC(C)(C)C)C1 73392,C1(NC(C(C)NC(C)=O)=O)CC(F)CN(C(=O)C(C(C)C)c2cccc(Cl)c2)C1 73393,S(=O)(=O)(c1ccc(NCCc2ccnc(Cl)c2)cc1Cl)NC(CC)CO 73394,c1(CC(=O)N(CCCNC(c2cn(C)c(=O)n2C)=O)C2CC2)ccc2ncsc2c1 73395,CN1C(=O)CC(C(N2CCC(CO)C(NC(C3C4(CC4)C34CC4)=O)C2)=O)NC1=O 73396,c1(OCCC)ncc(C)cc1-c1ccc(C(=O)Nc2nccnc2OC)nc1 73397,N#Cc1cc(Br)ccc1CN1CC2(CC2C(N2CCCC2C(N)=O)=O)C1 73398,c1(C(=O)NC2C(CNC(c3c(C)nc(COC)s3)=O)C2)ccc2nnc(C)n2c1 73399,c1(OC)ccccc1NCC(=O)NCC1(O)CN(C(c2nc(Br)c[nH]2)=O)C1 73400,c1(N2CC(c3cc(C)no3)OCC2)ccc(S(=O)(=O)NCc2sccc2C)cn1 73401,C1(CC(=O)NCC(N(C(c2nc(CC)sc2)=O)C)C2CC2)Cc2ccccc2N1 73402,CCC(C(=O)NC1CCCC1NC(=O)C=CCOC)n1ccnc1 73403,CC(C)CC(C(=O)N1CCC(CO)(NC(c2cnns2)=O)C1)C(C)C 73404,C(=O)(C(CC(C)C)N(C)C)NCc1c(CCNC(CC(=O)NCC#C)=O)ocn1 73405,C=C(C)CCCC(=O)NCC1COCC1NC(=O)C(C)NC(C)=O 73406,c1(N2C(C)CC(CNC(=O)CCc3cnn(C)n3)C2)ncnc2c1CCCC2 73407,C12(NC(C3(F)CCS(=O)(=O)C3)=O)CCC(CC1n1cc(CSCCOC)nn1)C2 73408,CCCC(CC(C)C)C(=O)NCc1ncccc1C(=O)N(C1CC(C)(C)C1)C 73409,CCCC(CNC(c1ccn(C)n1)=O)C(=O)NCCC(O)C1CCCC1 73410,C1(C(N(C2C3CN(CC(F)(F)F)CC23)C)=O)CCCN(C(N)=O)C1.C12CN(C1)C2 73411,C1(CCC(=O)NC(C)CCN(C(=O)CSC2CC2)C)NC(=O)NC1=O 73412,C1(NC(c2csc(CO)n2)=O)CCC12CN(C(=O)C(c1ccc(F)cc1)CO)C2 73413,N1(C(CCc2onc(CC)n2)=O)CC2CC(C1)N(C(=O)CCC1CCC(=O)N1)C2 73414,C(CNC(C12CC(NC(=O)NC3CC3)(C1)C2)=O)(C(C)C(C)C)NC(C#CC(C)C)=O 73415,CC(F)(F)CCC(=O)NC(C)(C)CC(=O)NCC1C2COCC12 73416,Cc1cc(Cl)c(C(=O)NCCN(C(=O)CCC2CCC(C)O2)C2CC2)cn1 73417,N1(C(CC(CNC(C(CC=CC)C)=O)OC)=O)CC2(CNC(=O)OC2)C1 73418,C1(N(C)C)CC(N=c2ccnc(N3CCCC(c4nncs4)C3)[nH]2)C1 73419,c1(-n2cc(CC3(O)CN(C(=O)CCOCC(F)F)C3)nn2)cccc(F)c1F 73420,C(C(=O)Nc1ccccc1)(C1=CCC2CC1C2(C)C)N1CCC(S(CC)(=O)=O)C1 73421,C1(CNC(C2C(C)C2(F)F)=O)CC2(CCC2)CN1C(c1cccnn1)=O 73422,Cc1c(F)c(F)c(CNCc2c(F)ccc(F)c2O)c(F)c1F 73423,N1(c2snc(C(C)(C)C)n2)CCC(NC(C2CCCN(C(=O)C3CC3)C2)=O)C(F)C1 73424,CC1N(C(=O)NCCCC(=O)NC2CCCCC2)CCOC1(C)C 73425,C(CCCC)(C(=O)N(C)CCOCC1CC1)NC(CCCC#C)=O 73426,Cc1nc(O)nc(C)c1C(=O)NCCC(C)NC(=O)Cc1cnn(C(C)(C)C)c1 73427,c1(CNCC2C(C)(C)CCNC2)n[nH]c2ccccc12 73428,Cc1c(C(N2CCN(C(C3CC34CCC4)=O)CC2C(C)C)=O)cnc2nncn12 73429,CCCC(C)C(=O)NC1(CCC(=O)NCc2cn(C)nc2CC)CCC1 73430,c1(OC)cc(C#N)ccc1N(C1CC2CNC1C2)C(=O)CCBr 73431,C1(C(=O)NCCC(C)NC(C2(C)CCSCC2)=O)CCOC(=O)N1 73432,N1(C(C2N(C(c3c(C)cc(C)o3)=O)CSC2)=O)CCCC(C)(O)C1 73433,c1(NC(C(C)(CO)NC(CC(C=C)C)=O)=O)ccc(OC)c(F)c1 73434,N1(C(C(C2CCOC2)OCC)=O)CCN(C(C2CC(C)CCO2)=O)CC1CCO 73435,CC1(C)CCCN(C(c2cc(N)cc(O)c2)=O)C1CNC(=O)CNc1nccs1 73436,C(=O)(C1=C(Cl)CCOC1)N(C1CCN(C(C2C(OC(C)(C)C)C2)=O)C1(C)C)CCO 73437,c1(C(C(=O)NC(CCN(C(CC=C(C)C)=O)C)C)O)ccc(Cl)cc1 73438,c1(CN2CCC(C(=O)NCc3ccc(F)c(Cl)c3)C2)ccc2c(c1)CCO2 73439,C1(C(=O)NC2C(NC(=O)Cc3cscn3)CCC2)CCC12CCC2 73440,c1(C(CNCC2C(=O)NOC2)CBr)ccc(F)cc1Br 73441,C1(C#N)(SC)CN(C(=O)C(Cc2ccoc2)NC(C2CCN2C(C)(C)C)=O)C1 73442,C(=O)(CC(O)C(Cl)(Cl)Cl)NC1CC(C)(NC(c2ccnn2C2CCC2)=O)C1 73443,C1(CC)CC(C(=O)NCC(CC)(CC)NC(c2oc(CO)cc2C)=O)CCO1 73444,c1(CC)ccccc1C(CNC(=O)CSC(F)F)NC(c1ccn(CC)c1C)=O 73445,C1(NC(C2CSCC(=O)N2)=O)CCCC12CN(C(c1ccccn1)=O)C2 73446,C1(NC(c2nc(CC)sc2)=O)CC2CCC(C1)N2c1ncc(Br)cn1 73447,n1(C(CC)CC)nc(C)cc1C(N1CCC(COC)(NC(c2cncs2)=O)C1)=O 73448,C1(c2cn(CC3CCN(C(C4(CF)CCCOC4)=O)C3)nn2)CCCCCCC1 73449,n1(CC)ccc(CCNC(c2c[nH]nc2CCNC(C2CC2F)=O)=O)n1 73450,C(C)(C)(CC(=O)N1CC(F)(c2cn(CC34CCC(OC(C)C)C3C4)nn2)C1)OC 73451,C1(NC(c2cc(COC)[nH]n2)=O)CN(C(=O)C(C)CO)CC1c1ccccc1F 73452,C1(NC(C2N(N=O)CCC2)=O)CC2CC(C1)N(C(=O)Cc1ncn3c1CCC3)C2 73453,C(C(C)(C)C(=O)N(C)CC1(C)CCCC1)NC(CCCOCC=C)=O 73454,S(=O)(=O)(c1ccc(C)cc1F)Nc1[nH]c2ccc(NC)cc2c1 73455,N1(C(C(C(C)C)O)=O)CCC2(CCN(C(c3ncnc4sccc34)=O)C2)C1 73456,C1(C(CNC(C(c2ccccc2F)C)=O)C)CCN(C(C2CC(F)(F)C2)=O)CC1 73457,N1(C(CCN(CC)CC)=O)CCN(C(c2ccc(C#N)o2)=O)CC1CC(C)(C)C 73458,Cc1nn(CCC(=O)NCCN(C(=O)C(C)CC(N)=O)C)c(C)c1C 73459,CC1(C)CCCC(CC(=O)NCC2(CCNC(C3(O)CC3)=O)CC2)C1 73460,c1(C(N2CC(CCNC(CC(CC)C)=O)OCCC2)=O)cnc(C)c(C#N)c1 73461,c1(C(=O)NC2CN(C(c3cncc(OC)c3C)=O)C2)[nH]c2ccccc2c1Cl 73462,Cc1cnc(CNC(COCC2(CN(C(=O)C=CCF)C)CC2)=O)o1 73463,N1(C(c2ccc(C(F)F)cc2)=O)Cc2[nH]nc(-c3c(CO)cccc3F)c2C1 73464,C(N=c1ncc(Br)c[nH]1)C1(O)CCCN(C(c2ncoc2-c2ccccc2)=O)C1 73465,c1(C(N(CCCNC(C(C)Cc2cnc[nH]2)=O)C)=O)cc2ccccc2c(=O)o1 73466,N1(C(C(c2n(C)cnc2)O)=O)CC(NC(c2cnn(C3CCC3)c2)=O)C(C)(C)C1 73467,c1(C(=O)NC2CC(O)(Cn3cc(CCNC(C)=O)nn3)C2)ccc(S(C)(=O)=O)s1 73468,CCCCN=C(NCc1nnn(C)n1)NC1CCCCC1C 73469,C1(O)(C(=O)NCC(CN(C)C(c2ccsn2)=O)(C)C)CCCC(C)(C)CC1 73470,c1(C(=O)NCc2ccc(C(=O)Nc3cn(CCC#C)nc3)s2)ncncc1C 73471,N1(C(c2nnc(C(C)C)s2)C(=O)NCC(=C)C)CCCN(CC2CC2)CC1 73472,N1(C(c2ccc(C(C)C)o2)=O)CCC=C(CNC(=O)C(O)C2CC2)C1 73473,C1(CC(=O)NCC(c2ccco2)O)(OC)CN(C(=O)Cc2cc(C)no2)C1 73474,Cc1cc(S(C)(=O)=O)cc(C(=O)NC2CCN(C(=O)CC3CCOC3)C2C)c1C 73475,c1(N(CC)CC)ccc(C(=O)NC2CN(C(c3coc(C(F)(F)F)n3)=O)C2)cn1 73476,C1(C#CC(=O)NC(C)CC2CCCN(C(=O)COCCCF)C2)(CC)CC1 73477,C(=O)(C(C)CS(C)(=O)=O)N(CC(CN(C(c1c(CCC)nco1)=O)C)O)C 73478,c1(C(N(C)CCOCCC(=O)NC(CO)CCO)=O)ccn2cncc2c1 73479,CC(C)(CNC(C1C=CC(NC(=O)COCC2CC2)C1)=O)CCO 73480,c1(C(C)(C)NC(C(C)O)=O)c(F)cccc1Br 73481,CC(C)CC(CNC(c1coc(Cl)c1)=O)NC(c1cc(=O)n(C)o1)=O 73482,c1(C(=O)NC2CN(C(Cc3scc(C)c3)=O)CC2C)cnc2sccn2c1=O 73483,c1(C(N(C2CCN(C(CC(CC)C3CCC3)=O)CC2)C)=O)cc(OC)ccc1O 73484,N1(C(Cc2nc(C)oc2)=O)CCC(NC(c2ccc(F)c(C)c2)=O)C1(C)C 73485,c1(C(=O)NC(CC(F)F)C(=O)NCC2OCC3CCC2C3)ccc2cccnn12 73486,C1(CC)CN(C(C)=O)CCC1NC(=O)CCCNC(c1ccc(C)c(C)n1)=O 73487,C12(NC(c3n[nH]c4c3CCCC4)=O)CCOCC1CN(C(=O)C1=CCCSC1)C2 73488,N1(C(c2nnc(C)s2)=O)CCCC(N(C(C)CC(C)C)C)C1 73489,CP(C)(=O)c1cnn(CC(=O)NCCCC2CCCN2C(=O)Cc2cnc[nH]2)c1 73490,CC1(C)CCCCC(C(N2CC3CCC2CC3NC(c2cccc[n+]2[O-])=O)=O)C1 73491,c1(C(=O)NC2C(C=C)CN(C(=O)C(C(C)C)SCC)C2)n[nH]c2cccnc12 73492,c1(NC)cc(C(=O)NCC2CCC(C)CN2C(=O)CCOCC2CC2)cc(Cl)n1 73493,c1(C(N2CCOC(C(F)(F)F)C2)C(=O)NCCCSC)cccc(CC2CC2)n1 73494,c1(C(=O)NC2CC(C)CN(C(=O)C3=CC(C)(C)C3)C2)ccc2c[nH]nc2c1 73495,Cc1c(N)ccc(C(=O)NCC2CCCC2NC(=O)CCC=CC(C)C)c1C 73496,c1(OC)ccc(NC(=O)NCC2CCN(C(=O)NCC(F)(F)F)CC2)c(F)c1 73497,c1(OC(C(=O)NC(Cn2cc(C(CC)OC)nn2)C)C)cccc(Cl)c1Cl 73498,c1(C(=O)NCC2(NC(CNS(C)(=O)=O)=O)CCC2)ccc2c(c1)OC(F)(F)O2 73499,CC(C)CC(C(=O)NCCC(C)(C)NC(C1CN(C)CCO1)=O)C(C)C 73500,C1(C(N(CC(COCC)O)C)=O)CCCCN1C(c1scc(C)c1C)=O 73501,C=C(C)C(C)(C)C(=O)NCCN(C(=O)COCC1CCOC1)CCC 73502,CC1CN(C(c2n[nH]cc2C2CC2)=O)CCCN1C(c1n[nH]c2ccccc12)=O 73503,CCCCC(CC)C(=O)NCC1COCCN(C(c2nc(Cl)oc2C)=O)C1 73504,c1(N2C3C(NC(Cc4nc(C)c(C)[nH]4)=O)(CCC3)CC2)ccc([N+](=O)[O-])cc1C 73505,c1(C(=O)NCC2CC(NC(c3n(CC)ncn3)=O)C2(C)C)ccc(C#N)n1C 73506,Cc1cccc(C2=CCN(C(=NCCn3cccn3)NC3CC3)CC2)c1 73507,C1(NC(C(CCCCC)F)=O)CCN(C(c2ncccn2)=O)CC(C)(C)C1 73508,C1(C(F)(F)F)(C(N2CCN(C(CSC)=O)C3C2C3)=O)CC2C=CC1CC2 73509,C1(CC=C)(NC(C2CCCC2C(C)C)=O)CCN(C(c2cc(=O)cc[nH]2)=O)C1 73510,C(=O)(CCC(C)(C)C#N)N1CCCC(CNC(c2[nH]cc(C)c2C)=O)C1 73511,CC1(C)C(NC(=O)Cc2cn[nH]c2)CC1CNC(C1(C2CC2)CCC1)=O 73512,N1(C(CC(C(F)F)NC(=O)C2=CCCOC2)=O)CC(F)(F)C(F)(F)C1 73513,N#Cc1ccc(CNC(=O)CC2CCCN2C(c2c(F)cncc2Br)=O)c(F)c1 73514,Cc1cc(C(=O)NCCN2CCN(C(C3(C)CCOC3C)=O)CC2)n(C2CC2)n1 73515,c1(OC)cc(C)cnc1C(N1CCN(C(C)CNC(=O)C=CC(=O)N(C)C)CC1)=O 73516,C12(CCC1)C(=O)NC2.C(C(=O)NCCOCCC1(CO)CC1)OC(C)=O 73517,C1(NC(C2CC(C#N)C2)=O)CCCCC1NC(C1CCCN1Cc1cccs1)=O 73518,C(C1c2ccsc2CCN1C(=O)C(=O)NCC(F)(F)F)NC(=O)CCCF 73519,C12(C(N(CC=C)CCC)=O)CCCC1CN(C(=O)C(C)(C)OC(C)=O)C2 73520,C(=O)(C1=Cc2ccccc2C1)NC(CNC(C1(CC(=O)OC)CC1)=O)(C)C 73521,c1(C(=O)NCCc2cccc(C)c2)coc2c1CN(C(=O)CCN(C)CCO)C2 73522,N1(C(CC=C)=O)CC2(CCCN(C(=O)CCCC(=O)c3ccc(OC)cc3)C2)C1 73523,C1(OC)CC(NC(=O)CN2CC3CC3C2)C12CCN(C(=O)CC1(C#N)CC1)CC2 73524,N1(Cc2cnc(CC)[nH]2)CCOCC(NC(=O)CCCCCNC(C)=O)C1 73525,C1(CNC(C2(C#N)CCC2)=O)CCCCC1NC(=O)C(O)Cc1ccc(Cl)cc1 73526,C1(C(=O)NCC(C2CC2)NC(C(C2CCC2)OC)=O)CC(C)(C(C)(C)C)C1 73527,N1(C(CCCC#C)=O)CC2CCCC(CNC(=O)C(C)n3cncn3)C2C1 73528,C1(CNC(CCCCC=C)=O)CC2(CO1)CN(C(c1cnc(C)s1)=O)C2 73529,n1(CCC)ncc(C(=O)NC2CCN(C(c3ccc(CS(C)(=O)=O)o3)=O)C2)c1C 73530,N1(CC)CC(C(N2CC(CNC(=O)CCC3CC(C)(C)CO3)C(C)C2)=O)CC1=O 73531,c1(C(=O)NC2C3(CC(NC(=O)C4=CCOCC4)C3)C2)ccc2c(n1)NC(=O)CO2 73532,Cc1sc2ncc(C(N3CC4C(NC(=O)CC5CN(C)C5)C4C3)=O)c(=O)n2c1C 73533,C1(NC(CONC(Cc2nc(=N)[nH][nH]2)=O)=O)CCC2CCCC1O2 73534,C(=O)(C(C)=Cn1ccnn1)N1C(CNC(C2(C=C)CCC2)=O)CCC1 73535,c1(C(=O)NC2(C3CN(C(C(C)CO)=O)C3)CC2)nc2cncnc2nc1O 73536,c1(C(N(C(c2cn(CC3CC4CC4C3)nn2)C)C)=O)cnn(C)c1C#N 73537,C1(CNC(c2cc(C)ncn2)=O)CCN(C(c2c[nH]c(=O)cn2)=O)CC1C 73538,N1(C(CNC(C(CC)C)=O)=O)CC2(C=C(C(=O)NC(c3nnc(C)o3)C)CO2)C1 73539,Cc1nn(CC(=O)NC2(C)CN(C(c3scnc3C3CCCC3)=O)C2)c(=O)o1 73540,C1(C(=O)NCC(=O)NCc2cnc(C)[nH]2)CCCC(C)C1 73541,N1(C(C(C)n2cncn2)=O)CC=C(C(=O)NCCC(=O)NC2CC2)CC1 73542,N1(C(C(CC=C)(C)CC)=O)CCC2(CCN(C(c3cncc(C)n3)=O)C2)C1 73543,C(CC(CC)C(=O)NCC(C)N(C)C(c1nnn(C)c1CCC)=O)=CC 73544,c1(SCC(=O)N(C(C)C)CCNC(C2CCS(=O)(=O)C2)=O)ccc2c(c1)CCC2 73545,c1(OCCCN(C2CCN(C(=O)C=CC(F)(F)F)C2)C)cccc(C#N)c1 73546,C(=O)(C(C(C)(C)C)N(C)C)N(CC(C)C(=O)NC(CO)C(F)(F)F)C 73547,C#CCCCCC(=O)N1CCCCC(C(=O)NC(c2nc[nH]n2)CC)C1 73548,c1(OC)ccc(CNC(=O)NC2C3CCC(C3)C2c2ccccc2)cc1F 73549,c1(-c2nc(CC)c(CN3CCCC3c3cc(F)cnc3Cl)s2)cccc(F)c1F 73550,C1(N(C)C(=O)C2CC2)CCCN1c1nnc(C2CCCC2)s1 73551,c1(C(N2CC(NC(c3cncc(C)c3C)=O)(CO)C2)=O)cnc2c(c1)CCOC2 73552,c1(NC(CC2CC(NC(c3ccc(COC)cc3)=O)C2)=O)ncc(I)nc1Cl 73553,C1(C(N2CCC3(C2)CC3(F)F)=O)C2CCCC2CN1C(c1ccccc1F)=O 73554,C1(NC(C2CN(c3n(C)nnn3)C2)=O)CC2CCC1CC2NC(C1CC1F)=O 73555,N1(C(C(CC)SC)=O)CCCOC(CCNC(c2ccsc2OCC)=O)C1 73556,C(C)(C(C(=O)N1CC=CC(O)C1)C(C)C)NC(C1CC(CCC)C1)=O 73557,N1(C(c2c(CC)ocn2)=O)CCC(NC(=O)C=CSc2ccccc2)CC1C 73558,C1(CC)(NC(C2(C(F)F)CCCC2)=O)CCN(C(=O)C2=COCCO2)CC1 73559,C(=O)(CCCC(C)(F)F)N(CCNC(C(C)(C1CC1)NC(C)=O)=O)C(C)C 73560,C#Cc1ccc(OCCC#N)cc1.C12OCCCC1C(=O)NOC2 73561,N1(C(c2cc(F)cc(C)c2O)=O)CCCC2CN(C(=O)C(C)S(N)(=O)=O)CC12 73562,CN1CC2(CCN(C(=O)CONC(=O)CCCN3CCCCC3)C2)C1 73563,c1(C(N2CCC(c3ccccc3)(C(N)=O)C2)=O)cnc2cc(O)ccc2c1 73564,Cc1ccc(C(=O)NCC2CC3(C2)CN(C(=O)C(F)C2CCC2)C3)nc1O 73565,C1(CNC(CC(CCC)O)=O)CC2(CCN(C(c3cc(C)nnc3O)=O)C2)CO1 73566,C1(C(=O)NCC23CC(NC(CNC(C)=O)=O)(C2)C3)CC12CC(O)C2.C(C)(C)(C)OC 73567,c1(CN2CCC(CNC(c3csc(C)c3C)=O)CC2)ccc(C#N)cn1 73568,C1(C(N(C)C)=O)CCCCC1C(=O)NCC1(c2cnn(C)c2)CCCO1 73569,N12CCC(CC1)CNC(=O)C(C)COC2=O.c1(C(CC)=O)cn(CC)nn1 73570,N1(C(C=CSC)=O)CCC(NC(c2cc(=O)c(C)c[nH]2)=O)C(F)C1 73571,C1(C(=O)NC2CCN(C(c3c(C)[nH][nH]c3=N)=O)C2)(OC)CCCC(C)(C)C1 73572,C(=O)(CC(C)(C)COCC)N(CCCN(C(C1CCN(C(=O)NC)CC1)=O)C)C 73573,C1(C(=O)NOC(CC)CC)(CC#C)CCN(C(=O)Cc2cncs2)C1 73574,C1(CC)CN(C(c2ccc(Cl)cc2)=O)CCC1NC(=O)C=CC1CCOC1 73575,c1(OC)cc(C(N2CCC(O)(C(C)NC(c3ocnc3C3CC3)=O)C2)=O)n(C)n1 73576,C#Cc1cccc(N(C2CCC(NC(=O)CCC)CC2)C(=O)C=CC(C)OC)c1 73577,CC1CN(C(c2cccnc2C2CC2)=O)CC1NC(=O)CCC(N)=O 73578,Cc1cc(C(=O)NCCC2CCN(C(=O)C(F)(F)c3ccccc3)C2)nn1C 73579,c1(C(=O)NCCCOc2cccc(OC)c2O)ccc2nc(C)[nH]c2c1 73580,Cc1noc(C)c1C(N1CC(CCNC(=O)CN(C)C(CCC(F)(F)F)=O)C1)=O 73581,c1(OC)ccn2ncc(C(=O)NCC3CN(C(=O)C(O)C(C)C)CCN3C)c2c1 73582,C#CCC(CC#C)C(=O)N1CCC(CCNC(C2CC2OCC)=O)C1 73583,c1(C(N2CCC(N(C(C3CC(C)(CC)C3)=O)C)C2)=O)c(C)nnn1CC 73584,C1(N2CC(C)(c3ccccc3)C2)C(NCC)CC1(C)C.CO 73585,Cc1nc2c([nH]1)C(Nc1cc(C)c3ncc(Br)n3c1)CCC2 73586,c1(OC)cc(NC(c2cc(-c3cc4ccccc4o3)[nH]n2)=O)ccc1[N+](=O)[O-] 73587,N1(C(C2(Oc3ccccc3)CC2)=O)CCCC(NC(C2CCC3(CC3)C2)=O)CC1 73588,C#Cc1cnn(CC(=O)NCC(C)(C(C)C)NC(c2nc(Cl)sc2C)=O)c1 73589,C12(NC(=O)CCn3cnccc3=O)CCCC1CN(C(=O)C(=O)NCC(F)F)C2 73590,c1(NC2(CNC(CCc3ccc(C)s3)=O)COC2)nc2cccc(F)c2s1 73591,N1(C(C(CC=C)OC)=O)CC=C(CC(=O)N2CCCC3(C=CCO3)C2)CC1 73592,C1(NC(CN(C2CC2)CC)=O)(COC)CCN(C(=O)Cc2c[nH]ccc2=O)CC1 73593,C12(C(=O)NC(CC(C)NC(c3coc(-c4ccccc4)n3)=O)C)CC(C)(CO1)C2 73594,C(C(=O)N1CC(O)C(O)CO1)C12C(CN(C(c3ccncn3)=O)C1)CC2 73595,C12(CC(=O)NCC(CC)CN(C)C)COCC(C1)C2.c12ccc(cc1)c(=O)[nH]2 73596,CN1CCCCC(C(=O)NCC2(C)CCCN2C(=O)CNC(=O)C(C)(C)C)C1=O 73597,c1(C(=O)NC2CCN(C(=O)CC3(C(F)(F)F)CC3)C2)nccc2[nH]ccc12 73598,CC1CC(NC(c2cc(Cl)c(Cl)n2C)=O)CN(C(C2CC(=O)N(C)C2)=O)C1 73599,C(=O)(C1=NOCC1)NCCN(C1CCCC1)C(C1C(OCC)C1)=O 73600,C(=O)(C(O)C(F)(F)F)NC1(CO)CCN(C(C(N2CCOCC2)C)=O)C1 73601,C1(C(=O)NC2CCCN(C(=O)CCc3ccc(F)nc3)C2)CCc2nnnn2C1 73602,C1(C(=O)NCCCCCNC(C2(SC)CC2)=O)CNc2ccccc2O1 73603,Cc1nc(NC2CCC(NC(=O)CC(C)n3ccnc3)CC2)cc(C#N)n1 73604,c1(C(N2C(COC)CCCC2)=O)ccc(Cl)nc1NC(c1ccc(O)cc1F)=O 73605,Cc1nc2ncccc2cc1C(=O)NC1CCC(NC(=O)C(C)CC(N)=O)CC1 73606,C#Cc1ccc(F)c(C(=O)NCCOCCCNC(c2[nH]cc3c2CCC3)=O)c1 73607,Cc1cccn2cc(CC(=O)NC3CC(CNC(=O)CSc4cn[nH]c4)C3)nc12 73608,c1(C(N2C(C)(CC)C(=O)NCCC2)=O)cc(C)nc2ccc(C)cc12 73609,c1(C(=O)NCC2(O)CN(C(C3(OC)CCCOC3)=O)C2)c(C)nn(C)c1Br 73610,c1(C(=O)NCC(C2CCCC2)NC(C(C)n2cccn2)=O)cc(Cl)cnn1 73611,c1(OC)cccc(F)c1C(N1CC(O)(C(C)NC(=O)CCCCCF)C1)=O 73612,CC1(NC(=O)CCC2CCCO2)CCC(NC(c2ccnn2CCF)=O)CC1 73613,C=CC(CC)CC(=O)N1CC(CC(F)C(=O)NC(CCOC)C(C)C)C1 73614,N1(C(C(C(C)CNC(c2ccc(Cl)s2)=O)F)=O)CCCC2(CC(O)C2)C1 73615,c1(CC(=O)NCC2C(NC(CCN(CCCCC)C)=O)C2)cncnc1 73616,c1(C(C)(C)C)nccc(=NC2CCC2)[nH]1 73617,CC(C)CCC(O)C(=O)NN1CCCC1C(=O)NC1(C(C)(F)F)CC1 73618,N1(C(C(C=C=C)C)=O)CC(CNC(c2ccnc(OC)c2Br)=O)C2(CCC2)C1 73619,C12C3CC(CC13)NC(=O)C1(CCOCC1)C(=O)N2.c1(OC)cc(N(C)C)[nH]n1 73620,C(=O)(CCC(C)(F)F)NC(C)CCCNC(C1CCN(C(N)=O)C1)=O 73621,c1(C(N2C(CNC(c3c(OC)c(Cl)sc3)=O)CCC2)=O)cc2n(n1)CC(O)CO2 73622,N12CC(C3(CC3)C1)NC(=O)C1CCC1CC2=O.c1(COC)ccc(C(=O)OC)[nH]1 73623,c1(C(=O)NC(C)CCNC(c2cc[nH]c2C2CCCC2)=O)csc2c1CCCC2 73624,N1(C(c2c(CNC(c3c(OC)n(C)nc3)=O)noc2)=O)CCC(N(C)C)C1(C)C 73625,C12(O)CC(C1)C(=O)NC1C(CCC1)NC(=O)CNC2=O.C1(CO)CC1 73626,C1(COC)CC(CNC(c2cn(C3COC3)nn2)=O)N(C(=O)C(C)C(C)O)C1 73627,N1(C(CCCCC=CC)=O)CC(=O)NC2CN(C(=O)CNC(=O)CC)CCC12 73628,C12CCON1C(=O)O2.C1(C(N(C2(C(=O)OC(C)(C)C)CC2)C)=O)CC(C)(F)C1 73629,C1(CNC(C2N=C(C)SC2)=O)CC(C)N(C(=O)CSC2CCS(=O)(=O)C2)C1 73630,c1(-c2cn(C(C(=O)NCC(C3CCOCC3)CC)C)nn2)ccc(CO)nc1 73631,Cc1cc(C(=O)NC2(C(N3CCC(c4ccon4)C3)=O)CC2C)oc1C 73632,c1(OC(C2CCCO2)C)ccc(NC(=O)NC(c2ccco2)CO)cc1 73633,N=c1cc(C(=O)NCC23CCC2CCN3C(=O)C=Cc2cnccn2)nc(Cl)[nH]1 73634,N1(c2ncc(CC)s2)CCN(C(=O)NCC2CCCC(=O)C2)CC1 73635,C1(NC(C(N2CCCC(C)C2)=O)=O)CCC12CN(C(c1ccncc1)=O)C2 73636,N1(c2cc(NCCc3cnc(C)o3)ncn2)CCN2C(=O)N(C)CC2C1 73637,C(=O)(C1=C(C)OCC1)NC(C1CN(C(C2CCN(C(C)=O)CC2)=O)C1)C 73638,c1(N2CCC(C(=O)NC(CCC)Cc3nccn3C)C2)ccc2c(c1)OCO2 73639,C(=O)(CCC(F)(F)F)NC1CCC(CCC(=O)NC(CC(=O)OC)C2CC2)C1 73640,CC1(C)CCC(CC(=O)NCC2CN(C(c3cc(-n4cccn4)ccn3)=O)C2)C1 73641,CCC(C)(CO)C(=O)N1CC(N(C)C(c2cc(O)nc(O)n2)=O)C2(CC2)C1 73642,c1(-n2c(Cn3ccc(C(F)F)n3)nc(COC(C)C)n2)ccc2ncsc2c1 73643,N1(C(C(C)n2ccnc2)=O)CCCC(C)(C)C1CNC(C1CC1C1CC1C)=O 73644,C(=O)(CN=S(C)(=O)c1ccc(Cl)cc1)NC1C(NC(CCOC)=O)CCC1 73645,c1(OC)ccc(OC)c(S(=O)(=O)NCC(=O)Nc2ccc(OC)cc2)c1OC 73646,Cc1cc(CCN2CCN(CC(C)O)CC2)cc(O)n1 73647,C(CCCC(C)NC(C1CCOCC1)=O)NC(c1nc(C(=O)OCC)sc1)=O 73648,c1(C(N2C3CN(C(C4CCN(C(C)=O)CC4)=O)CC32)=O)c(Br)ccc2c1OCO2 73649,N1(C(Cc2c(C(C)C)cccc2)=O)CC2COCC2C1 73650,C1(C(N2CC(CC(C)NC(=O)CCSCC(N)=O)C2)=O)(OC)CCOCC1 73651,c1(C(C)C)ccc(C=CC(=O)NCCN(C(c2ccccc2)=O)C(C)C)cc1 73652,N1(C(C2(F)CCN(C(c3ccc(NC=O)cc3)=O)C2)=O)CCc2n[nH]cc2C1 73653,C(=O)(C1=CS(=O)(=O)CCC1)NC(C1(O)CCN(C(c2ccn(CF)n2)=O)CC1)C 73654,N1(C(c2c(C)coc2)=O)CCN(C(=O)C(F)(F)Oc2ccccc2)C(C)C1 73655,c1(C(=O)NCC2C(NC(CCn3ccc(C)n3)=O)COC2)ccn2nncc2c1 73656,Cc1nc(-c2cn(CCC(=O)N(C(C)C)Cc3sccc3C)nn2)cs1 73657,N1(C(CSC)=O)CCC(C)C1C(=O)NCCCc1n[nH]c(C)n1 73658,C1(N(C(CCSCCNC(CC(C)SC)=O)=O)C)CCC(CO)CC1 73659,CC1CC(NC(=O)Cc2nncn2C)CN1C(=O)COc1ccc(F)cc1 73660,C(c1c(C)coc1C)=CC(N1CC(C2N(C(Cc3cnc(C)o3)=O)CCCC2)C1)=O 73661,C1(C(=O)NC2CC(CC)(CC)C2)CC(F)(F)CN1C(=O)CC1COCC(C)O1 73662,C(=O)(C(C#N)=CCNCC1(C)CC1(Cl)Cl)NC1CCCC1 73663,C=CCCCCCCC(=O)NC1(CNC(c2cncc(C)c2Cl)=O)CCOCC1 73664,N1(C(C2N(C(C3CC4(CC(C)C4)C3)=O)CC2)=O)CC(O)C(O)C12CCC2 73665,N1(C(C(c2ccnn2C)NC(C(C)C#N)=O)=O)CCCCCCCCC1 73666,CC(C)CC(=O)NC1CC(N(C(=O)CC2CC(C(F)F)C2)C)C1 73667,Cn1cncc1CC(N1CC(CCCCNC(=O)CCCn2cccn2)C1)=O 73668,C1(Cn2cc(C(CC)(C)C)nn2)CC(O)CN1C(c1coc(C)n1)=O 73669,O=C(C1=CCCOC1)NC1(CO)CCN(C(c2ccccc2)=O)C1 73670,Cc1cc(C(N2CC3CC(NC(C4CC45CCC5)=O)C2C3)=O)ccc1C(F)(F)F 73671,C(=O)(C(CC(F)F)NC(=O)CCCF)NCc1n(CC)cnn1 73672,Cc1nc(C(=O)NCc2c[nH]nc2C(=O)NC2CCC2O)c(C)s1 73673,c1(-n2c(-c3cccc(C4CCC4)c3)nc(C(C)OC)n2)ccc(Br)cc1C 73674,C=CC(C)C(C)C(=O)NC1(C)CC(NC(c2cncc(Cl)c2Cl)=O)C1 73675,CCCCCCC(C)CC(=O)NC1CC2CCC1N2C(=O)C(C)(C)CS(C)(=O)=O 73676,C1(CC(C)C)CNC(=O)CN1C(=O)CCCCCn1cc(-c2ccccn2)nn1 73677,C(=O)(C(C)(C(=O)OC)C(C)NC(C1CC(=O)N(c2ccc([N+](=O)[O-])cc2)C1)=O)OC 73678,CN1CCC(C(=O)NCc2ncoc2C2CN(C(=O)COC(C)(C)C)C2)C1 73679,Cc1ccc2oc(C(N3CCN(C(=O)Cc4ccsc4Cl)CC(O)C3)=O)cc2n1 73680,CCCC(C(=O)NCCC(O)C(=O)N(CC(F)F)CCC)C(C)C 73681,C1(CC(N2CCC(C(=O)NC)C2)=O)CC(C)(C)CCO1 73682,CC1(NC(C2CCCS2)=O)CC(NC(c2cnoc2C2CCC2)=O)C1 73683,C1(N(C(c2c(C)ocn2)C(=O)NC(C)C)C)CC(O)C1(C)C 73684,C1(C)(C(=O)NCC(C)(C)NC(C2(C)CC3CCC2C3)=O)CC2CCC1C2 73685,CC1(C(=O)NCC2(C)CCN(C(=O)Cc3csc(Cl)n3)C2)COC(=O)OC1 73686,C1(COC)(NC(=O)Cc2ccccc2Cl)CCN(C(=O)C(F)OC(F)(F)F)CC1 73687,c1(COC(=O)CC(c2ccccc2)n2cccc2)ccc(I)c(Cl)c1 73688,C(CCF)(C(=O)N1CC(C(C)O)C1)NC(COCCC#C)=O 73689,c1(CNC(C2CC2Nc2cc(OC(F)F)ccn2)=O)cccc(I)c1 73690,C1(CCNC(=O)CN2CCOCC2)CCN(C(c2csc(CO)n2)=O)CC1(F)F 73691,CC1OCCC1CNC(=O)Nc1csc(C(N2CCCC2)=O)n1 73692,N1(C(C(C)NC(=O)Nc2ccccc2Cl)=O)CCOc2ccccc21 73693,c1(C(=O)NC2C3CN(C(C(CCSC)NC(C)=O)=O)C2C3)n[nH]c2c1CSCC2 73694,CCC(CO)(C(=O)NC(C1CCN(C(=O)CCN2CCCC2)C1)C)OC 73695,C12(C(=O)NC3C(NC(CCc4cc(C)no4)=O)C3)CCC(CC1)C(C)(C)O2 73696,C1(C(=O)Nc2ccc(C)cc2C(N)=O)C2C(CN1Cc1ccc(I)cc1)C2(C)C 73697,Cc1ccc(C)c(C(N2CCCC(CCNC(C34CC5CC3C4C5)=O)CC2)=O)n1 73698,c1(C(=O)NC23CCN(C(CCC(=C)Cl)=O)CC2C3)cc2c(C)c(F)ccc2[nH]1 73699,C1(CC)CN(C(=O)C(C(C)C)SC)CCN1C(=O)CN1CCCCC1 73700,c1(CN2CC3(N(C(c4nc(Br)cs4)=O)CC3)C2)c(F)cc(Cl)cc1Br 73701,C(=O)(CCCNC(=O)CC1C=CCC1)NCCSC(C)(C)C 73702,C1(CNC(C2(CC)CC2)=O)CN(C(=O)CC2CC(O)C2(C)C)CCCO1 73703,C(=O)(C(CC(N)=O)NC(=O)CCn1ccnc1C)NCC(CC)O 73704,Cc1cc(F)ncc1C(=O)NC1CN(C(c2ccc(N)cc2F)=O)CC1(C)C 73705,CN(CC1CN(c2ccccc2)C(=O)O1)N(C)C1CCCOC1C(N)=O 73706,N1(C(C(CC#C)C)=O)CCN(C)C(CNC(C2(CC(C)C)CC2)=O)C1 73707,c1(OCC(=O)NC2C(NC(C3CCC(C(C)(C)C)CC3)=O)C2)ccc(F)cc1Cl 73708,C12(C(=O)OCC)CCC1CN(C(N1CCN(CCCNC(C)(C)C)CC1)=O)C2 73709,C1(CC)(CC)CN(C(=O)C(C)(C)C(C)NC(=O)COCC(=O)OC)CCO1 73710,C(=O)(C(O)(C(F)(F)F)C1CC1)N1CC2C(CN(C(Cc3nc(C)oc3)=O)C)C2C1 73711,N1(c2nnc(-c3[nH]n(C)c(=O)n3)n2CC2CCCCN2C2=CC=C(Cl)CC2)CCC(F)(F)C(F)C1 73712,c1(N(C)C)ccc(C(=O)NC2COCC2NC(C2(C(F)(F)F)CC2)=O)nn1 73713,C1(C(N(C2CCN(C(c3cn(CCO)nn3)=O)C2)C)=O)CC(=O)NC(=O)C1 73714,c1(CC)nnc(O)c(C(=O)NCC2(NC(c3cc(O)cc(O)c3)=O)CC2)c1CC 73715,CC(CCCCNC(=O)CCCCn1ccnn1)NC(=O)Cc1ccc(F)cc1 73716,C1(NC(CN(c2ccc(Cl)cc2)C)=O)CN(C(=O)C=C2CC2)C2(CCOCC2)C1 73717,c1(C(=O)OCC)c(NC(C2CC(F)CN2C(=O)C2=CCCS2)=O)cccc1C 73718,CC1(CO)C=CCN1C(=O)CCOCCNC(c1cccc(O)c1)=O 73719,C(=O)(C(C)C(=O)NCC(C)CNC(C1(c2ccccc2F)CCC1)=O)OC 73720,C(CC(C)(C)C(=O)NCCC1(CO)CCC1)NC(C(CCSC)O)=O 73721,CN1CCN(C(C2(CNC(=O)CCCN3CCCC3)CC=CC2)=O)CC1 73722,C1(CC)(CNC(C2(CCNC(=O)CSc3nnnn3C)CC2)=O)CCCC1 73723,c1(C(N2CCC(NC(CCc3cccc(OC)n3)=O)C2C)=O)cc(C)c(O)nn1 73724,N1(C(CC2OCC(C)(C)C2)=O)CCC2CN(C(C3CS(=O)(=O)C3)=O)CCC12 73725,c1(SC)c(NC(c2nnnn2CCC2CC2)c2ccsc2)cncc1F 73726,c1(SC)ccc(-c2cn(-c3ccccc3NC(=O)CCN(C)C)nn2)cc1 73727,c1(CN(C)C)cccc(C(N2CC=CC2CNC(c2cccc(Cl)c2)=O)=O)c1 73728,N1(c2cc(N3CCN(CC)C(C)(C)C3)nc(C)n2)CCC2OCC(=O)NC2C1 73729,C(=O)(CC(C)(C)NC(C1(OC)CCC1)=O)NCC(=O)NCC#C 73730,c1(C(N2C(C(C)NC(C(n3ccc(C)n3)C)=O)CCC2)=O)oc(CO)cc1C 73731,C1(O)(CNC(C2CC2CF)=O)CCN(C(=O)CCC=CBr)CC1 73732,Cc1cc(C(N2CC3C(CNC(C4(C)CCN(C)C4=O)=O)C3C2)=O)cc(C)c1 73733,C1(OC)CN(c2cc[nH]c(=N)n2)CC1NC(=O)NC(C)C 73734,CC(=O)CCCC(C)C(=O)NC1CCN(C(=O)CCC2CCOCC2)C1 73735,C1(C(N(C2CCN(C(C3(C)CC=CC3)=O)C2)CC)=O)COCC1(C)C 73736,c1(C(=O)NC2C3CCC2N(C(c2occc2F)=O)C3)cc2ccc(F)cc2o1 73737,Cc1cc(C(N2CC(C(C)NC(=O)CC3(C)CC3(F)Cl)C2)=O)on1 73738,N1(C(C(c2ncc(C)s2)C)=O)CC(O)CC1CC1CCNCC1 73739,c1(C(N2C(CCNC(C3CN(C(C)=O)C3)=O)CCC2)=O)cc(Cl)cc(F)c1F 73740,c1(C(=O)NCC2CCN(C(C(CC=C)CC)=O)C23CC3)cc2ccccc2cn1 73741,C1(CNC(=O)Cc2ccns2)CN(C(=O)C=Cc2cc[nH]n2)CC12CC2 73742,C1(C(=O)NCCN(C(=O)CN(C)CCO)CCOC)CCCSC1 73743,c1(C(=O)NCC#CCNC(c2c(CC(C)C)onc2)=O)cnc2[nH]ncc2c1 73744,N1(C(C2C(=C)C2)=O)CCN(C(=O)CCc2ccc(Cl)cc2)CC1C(F)F 73745,c1(CC)cc(N2CC3C(CNC(=O)C(C)Cn4ccnc4)C3C2)ncn1 73746,c1(CC(C(=O)NCC2(O)CN(C(C3(OC)CCC3)=O)C2)O)cc(Cl)sc1Cl 73747,C1(C(=O)NCCCN(C(c2cccc(C)c2O)=O)CC)CC12CCC(F)(F)CC2 73748,O=C1CC(C(=O)NC(C(=O)NCC2CCCC2)CO)C2(CCC2)C1 73749,c1(C(=O)NC2C=CCN(C(C3C(C)CC(=O)NC3)=O)C2)cc2ccc(Cl)cc2[nH]1 73750,C(=O)(C(F)CC(C)C)N(C1CCCN(C(Cc2c(C)ncs2)=O)C1)C 73751,C1(C(=O)NCCC(CNC(c2ccn(CCOC)n2)=O)OC)CCC(CO)CC1 73752,C1(C)(COC)CCN(C(C2(CO)CCN(C(C3CCCCO3)=O)C2)=O)CC1 73753,C(=O)(CCCCCCCC)N1CC(CNC(C(CC#C)(C)CC)=O)C(O)C1 73754,c1(C(=O)NCCC(=O)NCC(N(C(=O)COCc2ccco2)C)C2CC2)cccs1 73755,C12(N(C)C)CCC(C(=O)NC3CC(C(=O)NCc4ccon4)C3)(CC1)CC2 73756,N1(C(C(F)=CC)=O)CCOC2(CCN(C(c3cscn3)=O)C2)C1 73757,C1(NC(C(F)=CCC)=O)CC12CCN(C(=O)CN1CCCNS1(=O)=O)CC2 73758,C12CCCN(C1C)C2.c1(-c2cc(OCC)ncc2)cc(F)cnc1OC 73759,N#Cc1ccc(N2CCCC(C(N3CC(O)C(C#N)C3)=O)C2)nc1 73760,c1(OC)c(C(=O)NC2CC(CNC(=O)C(C)n3ccnc3)C2)csc1C 73761,CN1CC(O)CC1(C)C(=O)NCC1(CCNC(C2CNC(=O)C2)=O)CC1 73762,C#CCCC(O)C(=O)NCC(C1CC1)NC(c1ccoc1C(F)(F)F)=O 73763,C1(OC)CC(F)CN(C(c2cnn(C3CCOCC3)c2)C(=O)NC(C)(C)C)C1 73764,CCCCC(CNC(=O)C(CC(F)F)N(C(=O)CN1CC2CC2C1)C)CCC 73765,N1(C(c2c(C)noc2C)=O)CC(C)(C)OC2(C1)CN(C(=O)CCN1CCCC1)C2 73766,N1(C(C2C(CC)C2)=O)CCN(C(=O)C=Cc2cccc(F)c2Cl)C2CCC12 73767,CCC(C)C(C)N=c1[nH]c(=NCC2(c3cnccn3)CC2)[nH]c2c1COCC2 73768,C=CCC(C(=O)NCC(CNC(c1cccc(C)c1[N+](=O)[O-])=O)OC)C(C)(C)C 73769,C(=O)(CS(=O)(=O)CCOC)N1CC(CC(=O)NC2C(OCC)CCC2)OCC1 73770,N1(C(C2(COC)CCC2)=O)CCC(NC(C2CCCC2(C)C)=O)C(C)C1 73771,c1(C(=O)NC(CCOC)CNC(=O)C(C)NS(C)(=O)=O)c[nH]c(=S)cn1 73772,c1(CC)nc2ccccc2c(C(=O)NC2CN(C(=O)C(C)(C)C)C2)c1C 73773,C1(NC(CSCCCC)=O)C=CCN(C(=O)COC(C)=O)C1 73774,N1(C(C(CC(=C)C)NC(=O)Cc2ccon2)=O)CCN2C(=O)OCC2C1 73775,c1(CCCC(=O)NCC2CCN2Cc2ccccc2Br)ccccc1Cl 73776,c1(OC)ccc(Cl)nc1C(N1CCC(CN(C)C(C2OCC2(C)C)=O)C1)=O 73777,C=C1CC2(C1)CC(C(=O)NC(C1CCCN(C(c3cc(N)cc(F)c3)=O)C1)C)C2 73778,C1(NC(c2ccc(C)cc2)=O)CCCC12CN(C(C1(C)CSC1)=O)C2 73779,c1(C(=O)NC(C2CCCC2)CNC(C2CC(OC)C2)=O)sc(SC)cc1C 73780,c1(OC)cccc(OCC(=O)NC(C)CNC(c2cn(CC(F)F)nc2C)=O)c1 73781,c1(CCC(=O)NCC(CC)NC(C(F)=CCC)=O)c(C)ncnc1O 73782,Cc1cnc(Cl)c(S(=O)(=O)Nc2ccc(C(=O)Nc3nccc(Br)c3O)nc2)c1 73783,c1(C(N(CCCNC(Cc2nnc(C)o2)=O)C2CC2)=O)cc(F)c(F)cc1F 73784,Cc1ccc(C(O)C(N2CCC(CCC(=O)N(CCC(C)C)CC(C)C)C2)=O)cc1 73785,c1(C(=O)NCC(c2ccc(F)cc2)NC(CC=CC)=O)ccc2nc(O)[nH]c2c1 73786,c1(NC(c2cncc(NC(c3c(C)cccc3)=O)c2)=O)ccc([N+](=O)[O-])c(Cl)c1Cl 73787,C1(CC(C)NC(C2CC(OC)(OC)C2)=O)CCN(C(=O)CC2CC=CCC2)CC1 73788,N1(C(C(C=C)(C)CC)=O)CCN(C(=O)C(CCC)N(C)C)CC(C)(F)C1 73789,N1(C(c2c(CC)cccn2)=O)CCC(NC(=O)COCCC(C)C)C(C)C1 73790,Cc1[nH]cnc1C(=O)NCc1ncoc1C1CN(C(C2CC(CF)C2)=O)C1 73791,CCCCC(CNC(c1cncc(OC)n1)=O)NC(=O)C(CC)n1ccnc1 73792,C1(NC(C(C=CCCC)O)=O)CCN(C(c2ccncc2)=O)C12CCC2 73793,n1(CC)cc(CC(=O)N(C2(C(=O)NC3CCN(C(C)=O)C3)CC2)C2CC2)cn1 73794,CCCCCC(C)(C)C(=O)NCC(C(N1CCOCC(C(C)C)C1)=O)OC 73795,Cc1cc(C#N)ccc1S(=O)(=O)N(C)C(C1(S(C)(=O)=O)CC1)C 73796,N1(C(C2(C#N)CC=CC2)=O)CC2CCN(C(=O)CC3CC3c3ccccc3)C2C1 73797,C(=O)(CC(C)CC(C)(C)C)N1CC(NC(Cc2cc(OC)c(O)c(OC)c2)=O)C1 73798,c1(C(N2C3C(C(N(C4(CCO)CC4)C)=O)C(C3)C2)=O)cc(O)nc(O)n1 73799,N1(C(C(=O)NCCCOC)c2cccs2)CCC(C)C(O)C1 73800,C=CC(C)CCN=c1nc(-c2ccccc2)[nH]c(=NCC(C)(C)n2ccnc2)[nH]1 73801,c1(C(=O)NC2C(NC(c3cc[nH]n3)=O)CCC2)ccnc2ccncc12 73802,N1(C(C2CC3CN(C(c4n(C)c(Cl)nc4)=O)CC2C3)=O)CCN2C(=O)OCC2C1 73803,C12(CSC)CC(C(=O)NCC(C(C)C)NC(=O)C=Cc3cncs3)(CO1)C2 73804,FC(F)=C1CCC(c2nnnn2CC(F)F)(NCC2CCC2CO)CC1 73805,c1(NCCNC(C)=O)ccc(S(=O)(=O)Nc2nc(Br)co2)cc1Cl 73806,CC(C)(CCC(=O)N1C2CCC1CC(C(=O)NCc1cnccn1)C2)[N+](=O)[O-] 73807,CC(C)C(C#N)C(=O)NCCCC(=O)NCC1CCC(F)C1 73808,C(=O)(C1Cc2ccc(F)cc21)NCC(CNC(C1(CCOC)CCCC1)=O)(C)O 73809,C1(O)(CCNC(C2CC(C)(O)C2)=O)CCN(C(=O)C2=CCCCO2)CC1 73810,C(CC(C)C)(C(=O)N1CC(C)CCC1CO)NC(C(C)NC(C)=O)=O 73811,C1(CNC(Cc2cc(C)no2)=O)CN(C(C2CCCC(=O)CC2)=O)CCCO1 73812,c1(C(=O)NC2CCCC(N(C(=O)CCC#N)C)C2)ncc2cc(Cl)ccn12 73813,CON=CC(=O)NC(C)C(=O)NCC(=O)OC(C)C 73814,Cc1nn(C)c(C)c1CC(N1CCC(F)(CC(=O)O)CC1)=O 73815,C(=O)(C(C)(C)C(C)C)NCCCC1OCCN(C(c2c(C)[nH][nH]c2=N)=O)C1 73816,N1(C(C(c2ccc(F)c(Cl)c2)=O)=O)CC2CC1CN(C(c1coc(C3CC3)n1)=O)C2 73817,N1(C(C=C(COC)C)=O)CCC(NC(c2csc(-c3cnc[nH]3)n2)=O)C(F)C1 73818,N1(Cc2ccc(COCC)o2)CC2CN(C(c3ccccc3I)=O)CC2C1 73819,c1(C(=O)NC(c2n(C)ncc2)C(=O)NCCn2ccnc2)ncnc(O)c1F 73820,CCCCCCC(C)C(=O)NC1CC(C)(NC(=O)CCCN=[N+]=[N-])C1 73821,c1(C(=O)Nc2cccc(CNC(C(C)CC(N)=O)=O)c2)cnn2c(N)ccnc12 73822,C1(NC(CN(C)C(c2ccsc2)=O)=O)CC2CC(NC(=O)Cn3nccn3)C1C2 73823,N1(C(C(COC)C)=O)CCC(NC(=O)Cc2csc(-c3ccco3)n2)C1C(C)C 73824,N1(CCNC(C(C)OCC2CCCO2)=O)CCN(C(=O)CC=C(Cl)Cl)CC1 73825,N1(C(c2c(OC)scc2)=O)CC2(CCN(C(=O)C(F)C(C)C)CC2)CC1C 73826,c1(C(=O)NC(CSC)CO)coc2cc(O)ccc12 73827,c1(CSC)noc(CCC(=O)NC2CC2CNC(=O)CC2CCCCO2)n1 73828,N1(C(c2snc(COC)n2)=O)CCC(c2n[nH]cc2N)CC1 73829,C(C(C(=O)NC1CC=CCC1)C(C)C)NC(c1c(C)ccn1C)=O 73830,CS(=O)(=O)c1ccc(C(O)CNC(=O)NCc2c(O)cccc2Cl)cc1 73831,CC12CCC(CNC(N3CCCOC(CCO)C3)=O)(CO1)C2 73832,c1(C(=O)OCC)cnn(C)c1NC(C1CC1c1ccncc1F)=O 73833,c1(CC(C)NC(=O)CCOC2COC2)ccc(CNC(C2CCC(=O)N2)=O)cc1 73834,C=CCC(C)C(=O)N1CCC(N(C(c2ccc(N(CCCC)C)s2)=O)CC)CC1 73835,c1(CC(=O)NCC(C)N(C(c2ccsn2)=O)CC)nnc(C)o1 73836,C1(NC(COCCN(C)C)=O)CCCC(NC(=O)C2=COCCO2)CC1 73837,C1(C(=O)NCC23CCC(NC(CSC)=O)(CC2)CO3)CCCC2(CCCCC2)C1 73838,c1(OC)cccc(C(CNC(=O)C(Cl)=CCl)NC(=O)Cc2c[nH]nc2O)c1 73839,c1(CN2C(CC)CN(C(c3ccc(=O)n(C)n3)=O)CC2)ccc(C)c(F)c1F 73840,N1(C(C2CCN(C(CC)=O)C2)=O)CCC(F)(CNC(c2ccn(CCF)n2)=O)C1 73841,c1(C(=O)NC2C(C(=O)NCC3CN(CC)C(=O)O3)CCC2)ccn2ccccc12 73842,c1(OC)cc(C(N2CC3CC(C2)N3C(C)=O)=O)cc(SC)c1.c12nccc-1n2 73843,c1(C(N(CC(CC)NC(CC(=O)OCC)=O)C)=O)cc(SC)cc(Cl)c1 73844,c1(CN2C3C(C(=O)Nc4ccc(Cl)c(Br)c4)C(C3)C2)ccc2c[nH]nc2c1 73845,N=c1[nH]c2c(s1)CCCC2C(=O)NC1(CNC(C2CC(S(N)(=O)=O)C2)=O)CC1 73846,C#CCCCCCC(=O)N(CCCCC(=O)N(C)Cc1ncnn1C)C 73847,CC1(C)COC(C(=O)NCCC2CN(C(=O)COC3CCCCCC3)C2)C1 73848,c1(CCN(CC(=O)NCC(O)CNC(=O)COCc2nccs2)C)ccccc1 73849,c1(OC)cnc(C(=O)N(C(C)C(=O)NCc2sccc2C)C)cn1 73850,C1(NC(C2C(C(=O)OC)CCO2)=O)C2CC1CN(C(C1CCCCO1)=O)C2 73851,Cc1cc(Cl)ccc1OCC1(NC(=O)Nc2ccsc2CN)COC1 73852,C1(C(N2CC(n3nnnc3C(C)C)C2)=O)(CC)CCN(Cc2noc(C)n2)C1 73853,C1(CNC(=O)C(=CC2CCCCC2)F)C2CC1N(C(C1C(F)(F)C13CC3)=O)C2 73854,c1(CC(N2CCC(C(CNC(C(C=C)OC)=O)C)CC2)=O)ccc(C#N)cc1 73855,c1(C(=O)OC(c2ccccc2)COCC(C)C)cncc(Br)c1 73856,C(=O)(C(C)=NOCC#N)N1C(C(=O)NCCC(=O)NCC)CC1C 73857,C(CNC(=O)Cc1ccn(CC(C)C)n1)(CC)(CC)NC(C1CCN(CC)C1)=O 73858,N12CCCOC(C1)C(=O)NC1(CC1)C2=O.C1(NC(=O)OC)CC(F)(C(=O)NC)C1 73859,N#Cc1cc(Cl)c(C(=O)NC2CCN(C(C3CN(C4CCC4)C3)=O)CC2)s1 73860,CC1(C(=O)NCc2ccccc2OCC#N)CC12CCN(c1ncccn1)CC2 73861,C1(C(N2CC(CCn3cc(-c4nc(C)sc4)nn3)C2)=O)CC1C1CC(F)(F)C1 73862,c1(N(C(C2N(c3ncc(C(=O)OCC)cn3)CCC2)=O)CC)ccnc(Cl)c1C 73863,N1(C(C(C)C2(O)CCC2)=O)CCC2(CC1)CC(C(=O)Nc1ccc[nH]1)CO2 73864,N1(C(COCCC(C)C)=O)CCS(=O)(=O)C(CCNC(C2CC3(CC3)CO2)=O)C1 73865,c1(C(N2CCCCC2CF)C(=O)NCCCOC)cc(Cl)c(Br)cn1 73866,CC(O)CCCN=c1ccc(S(=O)(=O)N2CCC(C#N)CC2)c[nH]1 73867,N1(C(CCSC)=O)CCC2C(NC(=O)CSCc3cscn3)C2CC1 73868,N1(C(C2CC(=O)N(CCO)CC2)=O)CCC2C(C1)CN2C(c1ccns1)=O 73869,c1(C(=O)NCCCN(C(C(C(C)C)NS(N)(=O)=O)=O)C)csc2cnccc12 73870,c1(C(N2CC(CC(=O)NC(C#C)C3CCC3)OCC2)=O)cnn2c1OCC2 73871,c1(CC(C(=O)NCc2ncco2)NC(C(C)Cn2ccnc2)=O)cnn(C)c1O 73872,C1(NC(CCCCN(C(C(CC)(C)O)=O)C)=O)CCCC(C)CC1 73873,C(c1ccccc1C#N)=CC(=O)NC(C1(CNC(C2CCC(=C)CC2)=O)CC1)C 73874,n1(CCC(=O)N(C2CCN(C(=O)OC(C)(C)C)C2)C)nnc2ccccc2c1=O 73875,CC(C)CC(CNC(=O)CC1(O)CCCCC1)NC(=O)CCc1cn[nH]c1 73876,C1(NC(=O)C#CC2CC2)CCN(C(C2CCC([N+](=O)[O-])CC2)=O)C12CCCC2 73877,c1(CNC(c2n(CCC)nnn2)(C2CC=CC2)C)ccc(OC)c(OC)c1 73878,C1(NC(=O)CSc2cccc(F)c2)CN(C(C2CCC3(CC3)C2)=O)CC2CC12 73879,c1(C(=O)NCC2C3CN(C(C4CC(C)OC4)=O)CC32)cc2ccccc2n1C 73880,C12(C(N3CC4(C(C(N5C(C)CCC5C)=O)C4)C3)=O)CCC(CC1)CC2 73881,N1(C(CCCOC(C)=O)=O)CCCC1(C)CNC(C1CC1(c1ccccc1)C)=O 73882,C1(C(N2CCC(C)(NC(c3ccc(CO)nc3)=O)C2)=O)(OCC)CCOCC1 73883,C1(NC(c2cc(OC)ncn2)=O)CCN(C(c2cnc(Cl)s2)=O)CCC1CO 73884,N1(C(CN(CC)CC)=O)CCC(N=[N+]=[N-])(C(=O)NCC(C)(C)C)C1 73885,c1(C(=O)NCC(C(C)(C)C)NC(=O)CCc2ccco2)nnn2c1CCCC2 73886,C(=O)(CCCCCN(C)C)NCCCCNC(C(C)NC(c1ccco1)=O)=O 73887,c1(OCC)nc(C)ccc1C(=O)NC(C1CCOC1)CNC(=O)CCC(C)C 73888,c1(C(N(C2CCC(NC(=O)CC34CCCC3C4)CC2)C)=O)ccc(CCO)cc1 73889,C1(CNC(C(c2scc(C)n2)(F)F)=O)CCN(C(C2(C)CC2C)=O)CC1 73890,c1(C(N2C(CNC(c3coc(C)c3)=O)CC(OC)C2)=O)ccc(N)cc1O 73891,C1(C)(CNC(C(c2n(C)ccc2)=O)=O)CCCN(C(c2cnncc2O)=O)C1 73892,N1(C(c2cn(CCC=C)nn2)=O)CCC(CNC(=O)CN(C)CCO)CC1C 73893,C1(C(=O)NCCN2C(C)CCC2)CC(F)CN1C(=O)CCCN(C)C 73894,N1(C(CCOCC#C)=O)CCCCC(C(=O)NC2CC(C(F)F)C2)C1 73895,N1(CC)CC(C(N2CCOC(CNC(C3CC4CC(=O)C3C4)=O)C2)=O)CCC1=O 73896,c1(NC2C3CN(C(C=CCC4(C(=C)F)CCC4)=O)CC32)nc2ccc(Br)cc2s1 73897,c1(C(=O)NC(CC)CNC(=O)CSC(C)C)cc([N+](=O)[O-])cc2c1OCCO2 73898,C1(C(N2C(CC)CC2)=O)CCCCCCN1C(=O)C=CC(=O)OCC 73899,N1(C(CC2C(C)(C)OCC2)=O)C2CCC(C(=O)NCC3CC(CF)C3)C1CC2 73900,N1(C(c2c(CC)nccn2)=O)CC(O)CC1(C)C(=O)NCc1nnc(O)o1 73901,C=CCC(C)(C)CC(=O)N1CCCCCC1C(=O)NC1(CO)CC(F)C1 73902,N1(C(CC(C=C)(C)O)=O)CCC(F)(F)C(CNC(=O)CC(C)(C)OC)C1 73903,C1(C2CCC(=O)NC2)(C(N2C(CC)C(NC(=O)C(F)(F)C(F)F)CC2)=O)CCC1 73904,N1(C(CCC(=O)N(C)C)=O)CC(NC(c2cnc(N)cn2)=O)CC12CCCCC2 73905,Cc1cc(C#N)nc(=NC(C)CC(C)NC(=O)CC(CC(N)=O)c2cccs2)[nH]1 73906,N1(C(c2ccc(C)o2)=O)CC2CC(NC(=O)COc3ccc(F)c(F)c3)C(C2)C1 73907,c1(C(N2CCN(C(C3CC(=C)C3)=O)CC2CC)=O)cccc2c1CCCC2 73908,C1(NC(c2cncc(OC)c2)=O)CC2CN(C(c3cc(C)ccc3Cl)=O)CC2C1 73909,N1(C(Cc2c(C)n[nH]c2C)=O)CCC2CCCC12C(N1CC(CO)C(C)(C)C1)=O 73910,c1(CNC(CS(=O)(=O)NCC)=O)n[nH]c2c1CN(C(c1cnccn1)=O)CC2 73911,c1(C(N2C(C(C)NC(C3(C(F)F)CCCC3)=O)CCC2)=O)cccc(=S)n1O 73912,S(=O)(=O)(c1cccnc1N(C)CCSC)NC1CCN(CC)C1 73913,C(CCCOCC)(C(=O)NC(C)Cc1cnc[nH]1)NC(CNC(CC#C)=O)=O 73914,N1(c2ncnc(N3CCC(C=C)C3)c2C)CCc2oc3ccccc3c2C1 73915,C(=O)(CCCCCCNC(=O)C(O)C1CCCC1)NCC(C(C)(F)F)Cl 73916,C(CCC)(C(=O)N1CCC(C(C)(C)NC(C23CC(C#N)(C2)C3)=O)C1)=CCC 73917,C(=O)(C(C)(C)C(=O)NC1CC1CNC(=O)CNC(c1ccccn1)=O)NC 73918,N1(C(C(Cc2ccccc2)NC(C)C)=O)CCN(Cc2cn[nH]c2)CC1C#N 73919,N1(C(C(=O)NCCCOC)c2cocn2)CCc2nn(C)c(=O)cc2C1 73920,CCCC(C)CCCNC(C1CCCCC1)C1CCC1 73921,CN=c1nc(N2Cc3cnc(C(C)C)nc3C2)[nH]c(=NCCC2CC2(Cl)Cl)[nH]1 73922,Cc1ncc(C(=O)N(CC(C)(C)CNC(=O)CC2CCCC2O)C)cc1N 73923,C=C(Br)CCC(=O)NC1CCN(C(c2cc(C(N)=O)ccn2)=O)C1 73924,C12(NC(c3cn(C)nn3)=O)CCC(CNC(C3(C4CC4)CC=CC3)=O)(CC1)OC2 73925,c1(C(N2CC(CCCCNC(C(C)CCN(C)C)=O)C2)=O)cc(Cl)ccc1F 73926,C1(C2(O)CCOC2)(C(N(CC(C)CNC(=O)CN2CCCC2=O)C)=O)CC1 73927,C(C(C)(O)C(=O)NCC1(C)CCCN1C(C1CCC(C)C1)=O)OC 73928,c1(C(CC(=O)NC2C(NC(CCCC)=O)CC2)C)c[nH]c2ccccc12 73929,C1(NC(C(C#C)(C)C)=O)CC2CCC(C1C)N2c1ccnc(-c2nccs2)n1 73930,N(S(=O)(=O)NC1CC1)(CCC)CC1OCCC1C(C)C 73931,N1(CC(=O)NC(CNC(C2(C(=O)NC)CCC2)=O)(C)C)CCC(=O)NC1=O 73932,c1(NC(Cc2nc(NC(c3[nH]cc(COC)c3)=O)sc2)=O)cc(C)cnc1Cl 73933,C1(C)(CC)CCCN(C(=O)C(C2CC2)N(C)C(c2cc(C(C)=O)c[nH]2)=O)C1 73934,N1(C(C(CO)OC)=O)CC(NC(=O)CCCC2CCC2)CC12CCCCC2 73935,N1(CC)CCOC(C(=O)NC2CC2CNC(C2(COC)CCCC2)=O)C1 73936,C1(CNC(CSCC#C)=O)C2CN(C(=O)Cc3ccnc(Br)c3)CC12 73937,Cc1ccc(C(F)(F)F)cc1C(N1CCCC(CNC(=O)C2=CCSC2)CC1)=O 73938,C(CCCS(=O)(=O)CCO)NC(=O)NCC1CN(CCC)CC1C 73939,C1(NC(C(C(C)(C)C)SC)=O)CN(C(=O)CC2(O)CCCC2)CC(C)(C)C1 73940,C1(C(c2nnnn2CCCF)NCc2ccc(SC)cc2)CC2(CCCO2)C1 73941,Cc1ncc(N)cc1C(=O)NCCC1CCN(C(=O)C(C)c2ccsc2)C1 73942,C(=O)(C1COCc2ccccc21)N(C)CC1(O)CCN(C(CCCCC=C)=O)C1 73943,c1(OC)cccc(CC(=O)NCC(CO)NC(=O)Cc2cccc(Cl)c2F)c1F 73944,N1(C(CCN(C(=O)Cc2cn(C)nc2C)CC)=O)CC(N(C)C)C(C)(C)C1 73945,C12(CNC(CCC(=C)Cl)=O)CCC1CCN2C(c1ccnc(C)c1)=O 73946,c1(NC(C)=O)cccc(C(=O)N(CC(C)NC(=O)Cc2csnn2)C)c1 73947,C1(C(N(C2CC3CC3C2)C)=O)CC2(CC(NC(=O)Cc3cccnc3F)C2)C1 73948,Cc1ccn2c(C(N3CCC(C(=O)O)CC3)=O)nnc2c1C 73949,c1(C(=O)NCC(c2cccs2)O)n[nH]c2c1CN(C(=O)Cc1cccc(F)c1)C2 73950,C1(NC(c2ccc(COC)cc2)=O)C(C)CN(C(=O)CCCC2CCC2)CC1C 73951,C1(OCC)(CNC(=O)Cc2cccnc2)CCN(C(=O)CC2CCCOC2)C1 73952,C1(CNC(CN(C(=O)Cn2[nH]cnc2=N)CC#C)=O)CCCC(C)(C)O1 73953,c1(C(=O)NCCCC(C)(C)NC(c2ccc[nH]2)=O)cc(Br)cc([N+](=O)[O-])c1 73954,c1(C(=O)NC(C)C(C)NC(c2cccc(CF)c2)=O)cccc(N2CCCC2)c1 73955,C(=O)(C1=CCCCCC1)NCC(CNC(C(C(C)C)NS(C)(=O)=O)=O)F 73956,O=C(CCCC(F)(F)F)NCC1(F)CC(CNC(C2(N3CCOCC3)CC2)=O)C1 73957,c1(C(N2CC(O)(CCNC(CC(C=C)C)=O)C2)=O)nc(C)ncc1Br 73958,N1(C(C2C(C)C2)=O)CCc2cc(CNC(=O)Cc3cncc(Br)c3)ccc2C1 73959,c1(C(=O)NCCCOCCNC(=O)CCCC2CCCO2)ccc(O)cn1 73960,Cc1c(C(=O)NCC=CC(N2CCCC3CC23)=O)cnn1C 73961,c1(CC)c(C(=O)NCC2(C)CCCN2C(=O)CCCCNC(C)=O)nnn1CC 73962,Cc1noc(-c2cn(CCC(=O)N(c3ccn(C)n3)C3CCC3)cn2)n1 73963,N1(C(c2ccc(C)nc2C)=O)CCN(C(C2CCCN2C2CC2)=O)CC(C)(C)C1 73964,Fc1cccc(Cl)c1CN1CCC(C2OCCO2)C1 73965,CC(CN(C)C)C(=O)NCCCN(C(=O)CC(O)c1ccccc1)C 73966,C1(C(N2CC(CNC(c3c(CC)ocn3)=O)C3C2C3)=O)CCC(C)(C)CC1 73967,c1(C(N2C3(CNC(c4cccc(F)c4F)=O)CC(C2)C3)=O)nccn2ccnc12 73968,c1(C(CC(=O)N2CCC3CC23)NC(C)=O)ccccc1F 73969,c1(CN2CC(c3cn(CC(F)(F)F)nc3)C(O)C2)cnc2c(Br)cc(Cl)cn12 73970,C(C(C)C(C)C(=O)N(CCNC(=O)C=CC(N1CCOCC1)=O)CC1CC1)OC 73971,N1(C(C(=O)NCC(=C)C)C(C)C2CCCCC2)CCOC(C)(CC)C1 73972,c1(C(N2CCSCC2c2nc(C)cs2)C(=O)OCCCCCC)cncc(OC)c1 73973,C1(C)(CNC(C(C)(C)n2cccn2)=O)CC(F)(F)CN1C(=O)CC1CC(F)C1 73974,C1(NC(=O)NCC(CC)(C)O)CC(F)CN(C(=O)OC(C)(C)C)C1 73975,N1(C(C(COC)Oc2ccccc2)=O)CCN(C(=O)C(C)(C)OC)C(C)C1 73976,c1(OC)ccc(C(c2nnnn2C)NCC=CCSC)cc1C#N 73977,C1(NC(=O)C=CCC2CC2)CCCCC1NC(C1CCOCC1)=O 73978,CC1COc2ccccc2C1C(=O)NC1CC(NC(=O)COc2cnn(C)c2)C1 73979,C1(NC(C(COC)(F)F)=O)CC2CCC1N(C(=O)Cn1ccc(O)nc1=O)C2 73980,c1(CN(C2CCOC2C)CCOC)ccc(SC)s1 73981,Cc1c(F)ccc(Cl)c1C(N1CCN(C(=O)C=Cc2ccco2)C(C2CC2)C1)=O 73982,C(=O)(CS(=O)(=O)C(C)(C)C)NCCCC(C)(C)NC(c1n(CCC)ncc1)=O 73983,Cc1ncc(S(N)(=O)=O)cc1C(=O)NC1(CNC(=O)C(C)CF)CCOC1 73984,C1(CO)CCC(NC(c2cc(Br)c(Br)o2)c2nnnn2C2CC2)CC1 73985,C1(NC(CC(=O)NC2CC2)=O)COC2(CCN(C(=O)CCOC3CC3)C2)C1 73986,c1(OCCN(C(C(=O)NCC)CC2CCCO2)C(C)C)cccc(Cl)c1 73987,c1(C(N2CCC(N(CCC)C)C2)C(=O)NCCSC)cccc(Cl)n1 73988,CCC(CC(=O)NC(CNC(C1(C)CCC1)=O)CCOC)C(C)C 73989,CCCCC(CC(=O)NC1C=C(C)CCC1)NC(=O)Cc1cc[nH]n1 73990,C#Cc1cc(C(=O)NCC(O)CNC(=O)C(C)(CCC)OC)cc(N)c1 73991,Cc1cc(C(=O)NC2CCC(CCC(N3CCCCC3C(F)F)=O)C2)cnc1C 73992,c1(OC)cncc(C(=O)N(C(C)(C(=O)NCC(c2ccncc2)C)C2CC2)C)n1 73993,CC1CCCc2cc(C(=O)NC3(C)CCN(C(c4cc(C#N)no4)=O)CC3)nn21 73994,C1(NC(C(c2n(C)cnc2)O)=O)CC1C1CCCN(C(c2ccc(Cl)s2)=O)C1 73995,c1(C(=O)NC(C(C)C)CNC(=O)Cc2ccccc2)cnc2ccsc2c1 73996,C1(C(N2CC3(C2)CN(C(=O)CC2CCC=CCC2)C3)=O)(COC)CCCCCC1 73997,C1(C(=O)NC2CCC(N(C)C(c3cnnn3C)=O)CC2)CC2CCCC(C1)C2 73998,N1(C(COCCCC(C)C)=O)CCC(NC(=O)Cn2cnc(Br)c2)C1C 73999,C1(C)(NC(C2C(C)C2)=O)CCN(C(c2ncccn2)=O)C1 74000,c1(C(=O)NC2CC3(CN(C(C4(CC#C)CC4)=O)C3)C2)cc(S(N)(=O)=O)cnc1C 74001,C(=O)(CC1=NNC(=O)C1)NCC12CC(NC(CCCNC(=O)OC)=O)(C1)C2 74002,C1(CNC(c2c(CC)nc(C)[nH]2)=O)CC2CN(C(c3csc(COC)n3)=O)CC12 74003,CCCCC(C)C(=O)NCC1CC(NC(=O)Cn2nnnc2C2CC2)C(O)C1 74004,N1(C(C=NOC)=O)CCC(NC(c2cn3c(n2)CCC3)=O)C(CO)CC1 74005,N1(c2ncnc(NC3CCCC(SC)C3)c2C)CCC2(CCC2)CC1 74006,C1(C)(CNC(c2c(C)nsc2)=O)CCN(C(=O)C=Cc2cccc(Cl)c2)CC1 74007,C1(COC)(NC(=O)C(C)=CC2CC2)CCN(C(=O)CS(=O)(=O)N(C)C)C1 74008,N1(C(CC(CC)C)=O)CC2CCN(C(c3cccn3C(C)C)=O)CC(C2)C1 74009,c1(C(=O)NC2COCCN(C(C3(COC)CC3)=O)C2)c(Br)ccc(C)c1F 74010,Cn1c(Cl)c(C(c2nnnn2CCC2(C)CC2)NCc2nncs2)sc1=O 74011,c1(CNCCCCNc2c(OCCC)cccc2)ccc(Cl)cc1F 74012,C1(C(N(CCNC(C(CCC)N(C)C)=O)CC2CC2)=O)CCn2cnnc2C1 74013,N1(C(CC2ON=C(CC)C2)=O)CCC(CC(N2CCC(F)(CF)C2)=O)C1(C)C 74014,c1(C(=O)NC(CNC(CN(C(C)C)C)=O)C2CC2)cc(F)ccc1C(F)F 74015,c1(NC(c2c(CC)cccc2)CC)ccc(S(=O)(=O)NC(C)CO)cc1C#N 74016,N(C(=NCCCF)NCC1(CC(C)C)CC1)CC1CC(C(C)C)C1 74017,C(c1cc[nH]c1)=CC(=O)NC1(CCNC(c2ccoc2Cl)=O)CCC1 74018,C=CC(C)(O)CC(=O)N(C1CCN(C(=O)C(=O)NCC2CC2)CC1)CC 74019,C1(NC(C(COC)OC)=O)CN(C(=O)CNS(=O)(=O)N(C)C)CCC1C 74020,c1(C(N)=O)cn(C2CN(C(C3CC3c3csc(Br)n3)=O)C2)nn1 74021,c1(C(=O)NCCCN(C(C2CCCC3C2C3(F)F)=O)CC)[nH]nc2ncccc12 74022,N1(c2nc(COC)nc(N3CC4CC4(CO)C3)c2)CCC2(CCCCC2)CC1 74023,c1(C(=O)NC(CNC(CC(C)(C)OC)=O)CO)ccc2cccc(Br)c2n1 74024,C1(C(N2CCC(C(C(=O)N(C)Cc3c(C)ncs3)F)C2)=O)COC(=O)N1C 74025,c1(CC(=O)N(CCCCCNC(C2(C)CC(C)C2)=O)C)ccc(Cl)nc1 74026,O=C(CCCC(F)(F)CO)NC1COCC1NC(C1OCC2CCCC12)=O 74027,c1(CC(C)(C)NCC2(O)CCCNC2)nc2ccccc2s1 74028,c1(C(=O)NC(CNC(c2c(C(C)C)nns2)=O)(C)C(C)C)ccc(S(C)=O)cc1 74029,C1(C(N(C2CCN(C(CCSC)=O)CC2)C)=O)CCCCC(=O)N1 74030,C1(O)(CN(C(CC2C(C)CCO2)=O)C)CCN(C(=O)Cn2cnnn2)CC1 74031,C1(C(=O)NC2C(CNC(CCCNC(N)=O)=O)CCCC2)CCCC(F)(F)CC1 74032,C(CCCCC(=O)NCc1ccc(CNC(=O)C(C)(CC)CO)cc1)OCC 74033,C1(CNC(c2cccc(C)n2)=O)CC(C)(C)CN1C(C1OCCCO1)=O 74034,N1(C(CCC(=C)C)=O)CC(C)(C)OCC1CNC(c1scc(Cl)c1Cl)=O 74035,C1(CC=C)(C(N2CCCC2CC2CC2)=O)CCN(C(c2ncccc2N)=O)C1 74036,Cc1cc(CC(N2CCC(O)(C(C)CNC(c3cncc(Cl)c3)=O)C2)=O)n(C)n1 74037,CC1OCCCC1C(=O)NCc1ccc(C(=O)NC2CC3CC3C2)s1 74038,N1(c2nccc(OCC)n2)CCC(C(=O)Nc2n[nH]c(CC)c2C)C(F)(F)C1 74039,CCCC(O)(CCC)CC(=O)NCC(CN(C(=O)CC(C)(C)CC)CCOC)(C)C 74040,n1(CC(=O)NCCN(C(=O)CNC=O)C)cnc(C(F)(F)F)c1 74041,C12(C(=O)NC(C(N3CC(CC)(OC)C3)=O)C3CCC3)CC1CNC2=O 74042,CCCCC(CC)CC(C(=O)NC1CCOCC1)N(C)CC1CC(O)C1 74043,c1(CC(=O)NC(CNC(=O)CN2CCCC2)C2CCC2)ccsc1Br 74044,c1(CNC(c2cc(CNC(c3cnc(CC)s3)=O)ncc2)=O)nnc2n1CCC2 74045,CC#CCCC(=O)NC1C2CC1N(C(=O)CCCN1CCOC1=O)C2 74046,c1(CN(C(c2cccnc2)C)CC2(C(=O)OC)CNC2)ccc(C#N)cc1C 74047,N1(C(C(C)C2CCC2)=O)CCN(c2cc(CNC(=O)C#CC3CC3)ccn2)CC1 74048,N1(C(C(C)(Cl)Cl)=O)CCC(NC(c2ccc(C(=O)C3CC3)cc2)=O)C(C)(C)C1 74049,N1(C(COC)=O)CCOC2CN(C(=O)CC3(OCC#C)CCOCC3)CC12 74050,c1(CNC(C(c2csc(C(F)F)c2)N(C2CCCCC2)CC)=O)cccc(Cl)c1 74051,C(=O)(CCCC(C)(F)F)N1CC(NC(CC2CC(OCC)C2)=O)C(C)(C)C1 74052,N1(C(=O)Cc2ccc(Cl)nc2)CC2CN(C(=O)C(CO)c3ccccc3)CC2C1 74053,CC1C=C(C(=O)NC2CCN(C(c3cc(C(F)F)cs3)=O)C2)CC1 74054,N1(C(CC2(C)CCN(C(CC(C=C)C)=O)C2)=O)CCCCCCCCC1 74055,Cn1ccc2c(-c3cncc(F)c3C(N3CCC(C)(C#N)CC3)=O)cccc12 74056,C#CCCC(=O)N(CCCNC(=O)COCc1ccccn1)Cc1ccccc1 74057,O(NC(=O)CC(C(C)OC)NC(=O)CCC1CCCN1C)CCCCC 74058,C1(NC(c2c(CC)onc2)=O)CN(C(=O)COCc2scnc2C)CC1C 74059,C1(S(=O)(=O)c2ccccc2)(CN=c2[nH]cc(CCNCCOC)s2)CC1 74060,C1(NC(C(C2N(C(c3n(CC)ncc3)=O)CCC2)(C)C)=O)CC(C)N(C)CC1C 74061,N1(C(C=CCN(CC#C)C)=O)CCC(NC(=O)Cn2ccc(C(=O)OC)n2)C(C)C1 74062,c1(N2CCC(NC3C(OCC)CN(C(=O)NC)C3)C2)cccc(C)c1C 74063,c1(CC(=O)N(CC(CNC(c2ccnc(C)n2)=O)O)C)ccc(Cl)c([N+](=O)[O-])c1 74064,C1(NC(c2c(OC)c(C)cs2)=O)CC2(C1)CC(CNC(=O)CC1(C#N)CC1)C2 74065,c1(NC(C(CCSC)NC(c2cc(CC)oc2C)=O)=O)cccc2c1OCC2 74066,C1(NC(CNS(NC)(=O)=O)=O)CCCC12CCN(C(c1cnc(C3CC3)s1)=O)C2 74067,N1(C(COC(C)C)=O)CC(C(N2CCC(CCCO)C2)=O)C(C2CC2)C1 74068,C(=O)(C1=CC2CCCC12)NC1C(C)(C)N(C(=O)CCn2cc(Cl)cn2)CC1 74069,Cc1cc(F)ccc1NC(C1CCCN1C(=O)COCCN(C)C)=O 74070,C1(C(=O)NCC(CNC(c2ccc(N(C)C)cc2)=O)CO)CN2CCC1CC2 74071,Cc1cc(C(N2CCC(O)(CN(C)C(C3CCCN3C=O)=O)C2)=O)nc(C)n1 74072,C1(C2CC2)(CO)CCN(CC2CCC23CC(F)(F)C3)C1 74073,c1(NC(c2c(NC(C=CC)=O)cccn2)=O)ccc2cc[nH]c2c1 74074,Cc1ccc2nc(C)cc(C(=O)NC(C)CN(C)C(c3ccc(F)cc3)=O)c2c1 74075,C1(C(C)C)CC(C)CN(C(=O)NC2CC(c3ccc(O)cc3)C2)C1 74076,N1(C(c2n[nH]c(C)c2C(F)(F)F)=O)CCC(NC(c2nncs2)=O)C(C)C1 74077,C(=O)(C(F)(F)C(C)O)N1CC(CNC(CC(c2ccc(N)cc2)C)=O)C1 74078,N#Cc1ccccc1CCCC(=O)NC1CCCCN(C(c2ccncc2)=O)C1 74079,N1(C(c2cccc(C3CC3(F)F)c2)=O)CCN(C(c2ccccc2)=O)C(CO)C1 74080,S(=O)(=O)(CCC(=O)NC(C)(C)CCNC(c1c[nH]nc1-c1ccncc1)=O)NC 74081,C1(CNC(COCCCOC)=O)CN(C)CCN1C(=O)Cn1cccnc1=O 74082,N1(C(C(C)c2ccon2)=O)CC(NC(c2ccsn2)=O)CCC1C 74083,N1(CCC(c2cnn(C(F)F)c2)=O)CCCC(C(=O)O)C1.C12CC(C1)NNC(=O)C2 74084,C1(NC(C2CC(OC)(OC)C2)=O)CC(C(=O)N(C)Cc2nc(C)no2)C12CCC2 74085,c1(N2CCN(c3c(N)c(Cl)ccn3)CC2)ccc2nncn2n1 74086,c1(C(N(CC(C)NC(C2CCCN(CCC)C2)=O)C)=O)c(Cl)ccc(C)c1O 74087,c1(C(=O)NC2C(NC(c3cnc(CC)s3)=O)CCC2)cc2c(cc1Cl)NCC2 74088,C(CC)(CCC(=O)NCC1CCCC(C)(C)C1)NC(c1cccc(SCC)n1)=O 74089,C1(NC(c2ncccn2)=O)C2COCC1CN(C(c1sccc1Cl)=O)C2 74090,N1(C(c2c[nH]nc2OC(C)(C)C)=O)CCOCC1NC(c1cc[n+]([O-])cc1)=O 74091,c1(C(N2CC(C(C)NC(C3CCC(OC)C3)=O)C2)=O)cc2sccc2n1C 74092,CCC(O)C(C)(C)C(=O)N1CC(NC(c2c(Cl)n[nH]c2C)=O)C(O)C1 74093,c1(C(=O)NCC23C(CN(C(c4n(CC)cnn4)=O)C2)C3)ccc(=O)n2c1CCC2 74094,Cc1nc(-c2ccc(Cl)cc2)oc1C(N1CCSC(C(N)=O)C1)=O 74095,C1(C(N2CC(C)N(C(=O)CCF)CCC2)=O)CC(C2CCOCC2)=NO1 74096,CC(C)C(C)C(=O)NC(C1CN(C(C2CN(C)C2)=O)C1)C 74097,C1(C(N(C2CC2)CC)=O)CCCCC1NC(c1cc(C)nn1-c1ccncc1)=O 74098,C1(C(=O)N(CCCCNC(c2ccc(Cl)cc2)=O)C)(CC)CCCCO1 74099,N1(C(C2(F)C(C)OCC2)=O)CC2(C1)C(NC(=O)C(O)C1CCCC1)CCS2(=O)=O 74100,C#CC1(N(C)C)CN(C(C2CC=CCN2C(=O)CC2COCC(C)O2)=O)C1 74101,N#CC1(C(=O)NCC2CC(NC(c3ccc(CO)nc3)=O)C2)CCOC1 74102,c1(C(=O)NC(CNC(C2CC=CCC2)=O)CO)ccc(-c2cnc[nH]2)cc1 74103,CC1Cc2cc(C(N3CCNC(=O)CC3)C(=O)NCC3CCOCC3)ccc2O1 74104,Cc1[nH]nc(C(N2CC(O)CC2C(=O)NC(CO)C2(C)CC2)=O)c1O 74105,C(N=c1[nH]c(C)ncc1C)C1CN(C(C(c2ccc(Cl)cc2)OC)=O)C1 74106,CC1(C)CCCCC1C(N1CCC(F)(CNC(=O)CCCC(F)F)C1)=O 74107,c1(C(=O)NCc2cccc(NC(C(C(C)C)F)=O)c2)c(F)ccc2nc[nH]c12 74108,CC1CCN(C(C2(N(C)C(c3ccc(O)nc3)=O)CC2)=O)C(C)C1 74109,C1(O)(CNC(C2CCC2C(N)=O)=O)CN(C(=O)COc2nc[nH]n2)C1.CC(F)(F)F 74110,CCC(C)(C)C(C)CC(=O)NC1CCC(NC(=O)C=CCOC2CCOCC2)C1 74111,CCC(CC(=O)N(C1CN(C(c2ccno2)=O)CC1(C)C)C)C(C)(C)C 74112,CC1CN(C(C)C(=O)NC(C(=O)NC(C2CCCC2)C)c2ccoc2)C1 74113,n1(CCCCNC(c2ccc(C#C)o2)=O)c(C)cc(C(=O)O)c1C 74114,c1(C(N(C)CC2CC(NC(=O)CC3(C)CC3)C2)=O)ccc(F)c(F)c1 74115,CCC(O)(CNCCCCCOC(C)(C)C)C(F)(F)F 74116,CCC(CCC(=O)NC1CC(NC(=O)CSCC(=O)OC)C1)OC 74117,C(=O)(C1=CNC2=NCCC2=C1)N1CCC(CCNC(CSc2n(C)cnn2)=O)C1 74118,c1(C(N2CC3C(CNC(C(C)=C4CCCC4)=O)C3C2)=O)cnc(O)c(Br)c1 74119,N1(C(C(C)N(C)C)=O)CCC(OC2CN(C(=O)C=Cc3ccoc3)C2)CC1 74120,Cc1c(Br)cc(C(=O)NCC2(O)CN(C(C3C4COCC34)=O)C2)c(=O)n1C 74121,C1(NC(C2C(C)OCC2)=O)CC12CC(NC(c1csc(Cl)c1Cl)=O)C2 74122,CC(CC(F)(F)F)C(=O)NCc1nc(CNC(c2ccn3nccc3c2)=O)cs1 74123,N1(C(COCCCOC)=O)CCCC2(C1)CN(C(C1CCCCC1(C)C)=O)C2 74124,CCC(C)C(O)C(C)C(=O)NCc1cncc(C(=O)NOC2CCCCC2)c1 74125,c1(C(N2CCN(C(CCc3scc(C)n3)=O)CC2CF)=O)c(C)cc(F)cc1C 74126,Cc1cc(C)c(CN2CCOC(CC(=O)Nc3cccc(Cl)c3Br)C2)cc1C 74127,Cc1nc(C)c(C(=O)NCC(CC(F)(F)F)NC(=O)C=CC2CCOC2)c(C)n1 74128,C1(C(=O)Nc2c(C)nsc2)N(C(=O)CN(C)C(=O)C2CC2)CC12CCCC2 74129,c1(CC)ccc(CN2CCC(NC(=NC)NCCOC)C2)cc1 74130,C1(NC(C2C(C)=CCS2)=O)C=CCC(C(=O)N(CC(C)(C)O)C)C1 74131,CCCCCC(O)C(C)C(=O)N1CCN(C(c2ccc(Cl)s2)=O)CC(C)C1 74132,c1(OC)cnc(F)c(C(=O)NCC2(CCNC(c3nccs3)=O)CC2)c1 74133,c1(-c2nnc(COC(c3cncnc3-c3ccccc3)=O)o2)cccc2nonc12 74134,C1(C(=O)NC2C(NC(Cc3cn(C)nc3C(F)(F)F)=O)C2)CCCS(=O)(=O)C1 74135,c1(SCC)cnccc1C(=O)NCCC1CN(C(=O)C(O)C2CC2)CCO1 74136,C1(C(=O)NCC23CCC(CC2)C3)CC(O)CCN1C(C1CC12CCOCC2)=O 74137,CCCCCC(C(=O)NCC1=CCN(C(C2CCC(C)O2)=O)CC1)C(C)C 74138,CCC(CC(F)F)C(=O)N1CCN(C(=O)C=Cc2ccc(C)cc2)C(COC)C1 74139,c1(C(=O)NC2CCCN(C(CC3(C=C)CC3)=O)C2)cnc(N)c(CO)c1 74140,N1(CCNC(c2c(C)cccn2)=O)CCCN(C(C2(C)CCOCC2)=O)CC1 74141,Cc1nc(C(=O)NC(C)(C)CNC(=O)C(O)Cc2cn(C)cn2)c(C)n1C1CC1 74142,C(C(F)(F)CC(O)CO)NC(N(C)Cc1cccc(Cl)c1Br)=O 74143,c1(C(=O)NCCN(C(=O)C(C)(F)C(F)(F)F)C)cc2ccc(Cl)cc2s1 74144,CC1(C)C2CN(C(C3CCOCC3NC(C3CC3C(N)=O)=O)=O)CC12 74145,n1(CC)ccc(C(=O)NCC2CCCN2C(=O)Cc2ncc(F)cc2F)cc1=O 74146,n1(CC(N2CC3C(NC(c4ccc(CC(C)C)s4)=O)(C3)C2)=O)cnc([N+](=O)[O-])c1 74147,N1(C(CC=CCC)=O)CCN(C(c2cnc(C)nc2CC)=O)CC1CC(F)F 74148,c1(OC)ccc(C(C)C)c(NC(N2CC3(NC(=O)C(O)C4CC4)CC2C3)=O)c1 74149,Cc1cc(C)n2ncc(C(=O)NC3C4CC3N(C(=O)C(O)c3cnc[nH]3)C4)c2n1 74150,c1(C(C(=O)NC2COC2)N(CC(C)SC)C)c(Cl)nc2sccn12 74151,CS(=O)C=CC(=O)N1CCN(C2CN(C(C3C(F)(F)C34CC4)=O)C2)CC1 74152,C1(C(=O)NCC2CC(NC(=O)CC3(O)CCOC3)C2)CN2CCCN1CC2 74153,c1(C(=O)NC(CC)C)n[nH]cc1CNC(=O)CN(C)C1CC1 74154,c1(C(N2CCC3(NC(CSCC#C)=O)C(C2)C3)=O)c(F)ccc(N)c1F 74155,N1(C(CCc2ccc(OC)cc2)=O)CCN(C(c2ccc(F)o2)=O)CC(CO)C1 74156,c1(OC)ccc2cc(C(=O)NCCCNC(=O)C(C)N(C)C(C)=O)ccc2c1 74157,C(=O)(CC(C)(C)COC)NCCN(C(=O)C(c1cccc(O)c1)C)CCC 74158,Cc1ccc(-c2cn(-c3ccc(C(=O)NC4(CCO)CCC4)cc3)nn2)c(F)c1 74159,c1(N2CC(C(=O)Nc3cc(O)ccc3F)SCC2)ncnc2n[nH]cc12 74160,CC1CC2CC(C(N3CCOCC(NC(c4ccco4)=O)C3)=O)(C2)O1 74161,N1(C(c2ccn(C)c2)=O)CCOC2(COCCN(C(c3ncsc3Br)=O)C2)C1 74162,C1(CNC(Cc2ccc(C)o2)=O)CN(C(c2cc(CO)[nH]n2)=O)C2(CCC2)C1 74163,C1(C(=O)NCC(C(C)C)NC(c2ccncc2F)=O)CCC2(CCOCC2)O1 74164,CC(C)C(C)C(CNC(=O)C(F)n1cccn1)Nc1ncc(O)cn1 74165,Cc1c(C(=O)NCC2CC3CCC(C2)C3)c[nH]c1C#N 74166,C1(C(=O)NCC2C(NC(c3c(CC)c(C)sc3)=O)C2)COc2ccc(Cl)cc2O1 74167,CN1CCCN(C(=O)CC(C(F)F)NC(C2(C)CCN(C)C2)=O)CC1=O 74168,N1(C(c2c(C)cn(C)n2)=O)CCN(C(=O)CCCc2ccc(Cl)cc2)CCC1C 74169,c1(N2CC3(CCN(C(CC(=O)N(C)C)=O)C3)C2)nc(Cl)nc2[nH]cnc12 74170,c1(NC(C2C(NC(C3CCC(=C)CC3)=O)C2)=O)ccc2ncsc2c1Br 74171,C(CC1CC1)(C(=O)NOCCF)NC(C(C(C)O)N(C)C)=O 74172,C1(NC(c2n(CCSC)nnn2)c2ccn(C(F)F)n2)CNC(=O)OC1 74173,C1(NC(CN(C(CN(C(C)=O)C)=O)CC2CC2)=O)CN(C)C2(CCC2)C1 74174,Cc1ccc(F)cc1CC(N1CC=CC(NC(c2oc(C(F)F)cc2C)=O)C1)=O 74175,Cc1ccc(C=CC(N2CC(F)(F)CC2C(N2CC3C(C(N)=O)C3C2)=O)=O)cc1 74176,C1(C(N(CCC)CCNC(C2(C(=O)OCC)CC2C)=O)=O)CNC(=O)N1C 74177,c1(SCC2(c3ccc(O)nc3)CC2)nc2ccc(Br)nc2[nH]1 74178,c1(CC)cc(C(=O)NCC2CN(C(=O)C(C)n3cccc3)CC2C)cn(C)c1=O 74179,n1(CC(=O)NC2(CN(C(c3ncn(CC)n3)=O)C)CC2)cnc2sccc2c1=O 74180,C1(CCCNC(Cn2c(C)cnc2)=O)CCN(C(c2[nH]ncc2C#N)=O)CC1 74181,CC(=O)C(C)CC(C)C(=O)NC1CC2(NC(=O)C(C3CCCCC3)O)COC1C2 74182,c1(NC(C)=O)ccc(C(=O)NCC2CCN2C(C2CCCCC2F)=O)cc1 74183,C1(C(N2CCC(C(=O)NC)C2C)=O)C2CCC(C2)N1C(c1cc[nH]c1C1CC1)=O 74184,c1(C(=O)NCCNC(CC(CCSC)O)=O)c[nH]c2ccc(Cl)cc2c1=O 74185,C1(C(C)NC(=O)Cc2ccnn2C)CCN(C(C2(F)CCOC2)=O)CC1 74186,Cc1nc(C(C)C)[nH]c(=NC2CC(NC(=O)C(C(C)C)c3cccnc3)C2)c1Br 74187,C1(NC(C(=O)NCC(C(=O)OC)C)=O)CC2(CCCC2)C1 74188,c1(CC(CNC(CCC)CO)O)cccc(F)c1 74189,C1(NC)CCN(N(C)CCCCc2ccc(Cl)cc2)CC1 74190,N(C)(C(=NCC(O)c1ccccc1Br)NCc1ccnn1C)CCCC 74191,N1(C(C=CSC)=O)C2CCC1CC(N(C)C(c1ccc(C3CCC3)cc1)=O)C2 74192,c1(CCC)nc(C(=O)NCC(C2CCCN2C(=O)C(C)=C2CCC2)(C)C)cs1 74193,C1(C)(CNC(COCC#C)=O)CCC(NC(=O)COCc2nc[nH]n2)C1 74194,C1(C)(OCC(=O)NCCCN(C(c2cc(CC)no2)=O)C(C)C)CCOCC1 74195,N1(C(CC2N(CC)CCC2)=O)CCC(O)(CCNC(=O)C=CC(C)C)CC1 74196,c1(C(N2C(c3c(C(=O)OCC)[nH]nn3)CCC2)=O)cc(C(F)(F)F)c(Cl)cn1 74197,Cn1ccc2c(CC(=O)NCC34CCC(CC3n3cc(CO)nn3)C4)cccc12 74198,NC(=O)CCC(=O)NC1CCCC(CNC(c2coc(-c3ccccc3)n2)=O)C1 74199,N1(C(c2nc(C)n(C(F)F)c2)=O)CCC(C)(NC(=O)C(C)C(F)(F)F)CC1 74200,C1(=CC(=O)NCCCNC(=O)C2=CC(O)CCC2)CCCCCC1(F)F 74201,c1(C(N2CC(C(C=O)OC)C2)=O)nnc(S)n1C.N1CC(F)(CF)C1 74202,CC(CC(C)(F)F)C(=O)N1CC(O)CC1CNC(c1cc(=O)cc[nH]1)=O 74203,C1(CC=C)(NC(=O)CCc2nc(O)n[nH]2)CCN(C(c2cn(C)nc2O)=O)C1 74204,C#Cc1cnncc1C(=O)NCC1(C)CCN(C(=O)C(C(C)C)SCC)CC1 74205,N1(C(C2C(CC)C2)=O)CCN(C(=O)C(n2ccnc2C)C)CC2(CC2)C1 74206,C1(NC(c2c(OC)cc(Cl)cc2)=O)CC(C)(C)C12CCC2 74207,C(=O)(C(O)CC(C)(C)C)N(C(C(=O)NCCC=CCCC)C)C1CC1 74208,N#CC1CCC1C(=O)NC1CCCC1CC(=O)NC1(CO)CC(O)C1 74209,[SH](=O)(=O)c1ccc(S(N)(=O)=O)c(F)c1.C1(N(C)C)CCS(=O)(=NC(=O)C)C1 74210,CC(C(=O)OCC(=O)NC1CCN(Cc2ccc(Cl)cc2)C1)C(C)(F)F 74211,C1(CNC(c2c(C)csc2)=O)(NC(=O)Cc2ccc(Cl)c(Cl)c2)CCCCC1C 74212,CCCC(C)(CC)C(=O)N1CCC(Cn2cc(CCS(=O)(=O)N(C)C)nn2)C1 74213,c1(C(=O)NC(c2ccn(C)c2)=O)coc(C)c1.c1(C(CCCC)O)ccccc1 74214,c1(OC)cc(C)c(NC(C2CCCC(NC(=O)CC(C)(C)CSC)CC2)=O)cn1 74215,c1(CC)cccc(OCC(N2CC(O)(CCNC(=O)C=CC(C)CC)C2)=O)c1 74216,N1(C(C2C(CNC(=O)COc3cccnc3)OCC2)=O)CC2CCC2C1 74217,C(=O)(C1=CCCSC1)NCC(C)(O)CNC(=O)CNC(c1c(F)cccc1F)=O 74218,c1(C(=O)NCC2(CNC(C(CC)OCC)=O)CCCC2)c[nH]c2cccc(Cl)c12 74219,N1(C(C(CC)(C)O)=O)CC2CCC2(CNC(=O)Cc2ccnnc2O)C1 74220,CC1CN(C(c2ccccc2NC2CC=CC2)=O)CC(C)N1CC=CCO 74221,C(C)(C)(CC(=O)NCC1CCC(NC(=O)CSc2n[nH]c(=N)s2)C1)N(C)C 74222,C1(CC(=O)NC)CN(C(c2ccc(C)nc2)=O)CCN1C(=O)C#CC1CCC1 74223,c1(SC(C)C(=O)NC2CCC(CNC(=O)CCF)C2)ccccn1 74224,C(C(CC(=O)NCC1(C#N)CC1)C1CCC1)NC(c1c(C)[nH]cc1)=O 74225,c1(NC(C2(F)CN(S(c3ccc(C)nc3)(=O)=O)C2)=O)c(C)cc([N+](=O)[O-])cc1Br 74226,C(=O)(CS(=O)(=O)N(c1ccccc1O)CC)OC1COCC1n1cc(CN)nn1 74227,C1(C(=O)NC(C)CCNC(C2CC2(F)F)=O)C2CC1N(C(=O)OC(C)(C)C)C2 74228,c1(C(N2C(CNC(c3cn(CC)nc3)=O)CCC2)=O)cc(N)cc2c1OCCO2 74229,C1(C(=O)NCC(CNC(C2OCCN(C)C2=O)=O)O)(OC2CC2)CCC(C)(C)CC1 74230,N1(C(CSc2ccc(C(C)C)cc2)=O)CC2CC(C1)C2NC(C1(C)CCOC1)=O 74231,C(N=c1[nH]cnc2c1CCC2)c1ccc(C)nc1-n1cc(Cl)cn1 74232,c1(C(N2C(COC)(CNC(=O)C3=CCCC3)CCC2)=O)ccc2cccnc2c1 74233,C1(CNC(COc2c(C)cccc2)=O)N(C(=O)C(C)NC(N)=O)CCC1(C)C 74234,N1(C(CC(C)(C)C2CC2)=O)CC2CCC(C(=O)NCC3COC(=O)N3)(C2)C1 74235,C1(NC(C)=O)CCC(CC(=O)NCC(C2CCN(C(=O)C(C)(Cl)Cl)CC2)C)CC1 74236,C(=O)(C)NCCCNC(C)(C)C1(C(=O)OC)CC1 74237,C(=O)(C1=NNC(=O)CC1)N(CC(C)(C)NC(c1ccns1)=O)C 74238,C1(C(N2CC(CC(C)(C)C)N(C(=O)CCC(F)F)CC2)=O)CCCCC(F)(F)C1 74239,N1(C(Cn2ncc(C)c2)=O)CC2CC2(C(N2CC(Cc3ccoc3)C2)=O)C1 74240,C(=O)(C(CC)C(=O)NCC1CN(C(=O)C(C)(Cl)Cl)CC12CC2)OCC 74241,C1(NC(C2CSCCS2)=O)CN(C(C2CC(O)C2)=O)CC1n1cccn1 74242,c1(NC(C(C(C)NC(C2CC(C)(C)CCO2)=O)(C)C)=O)ccc2ccoc2c1 74243,CCCCC(C(=O)NCC(C(C)(C)C)OC)NC(c1cc(C)c(C)[nH]1)=O 74244,c1(OCC)cc(N2CCC(NC3CC3CC(C)C)C2c2ccccc2)ncn1 74245,Cc1nc(C(N2CC(CNC(=O)C(=Cc3c[nH]cn3)F)C2)=O)nn1C 74246,C1(C(=O)NCC2CN(CC)C(=O)O2)CC(C)NC2=C1C(=O)CCC2 74247,N1(C(CSCCCC)=O)CC(NC(c2cc(O)nc(C3CC3)n2)=O)CC(F)C1 74248,N1(C(C(C)(C)C#N)=O)CC2(CCC(CNC(C3CCC4CC34)=O)O2)C1 74249,C(CC(C)(O)CNC(C1(CNC(=O)COCc2nc[nH]n2)CCCO1)=O)OC 74250,CC1CCCn2c(CC(N3CCC34CN(C(C3(C)CCCN3C)=O)C4)=O)cnc21 74251,C(CCC(C)C)(C(=O)NCCC(C)(C)C)NC(c1c(C)cccn1)=O 74252,c1(CCC(=O)NCC(C(C)C)NC(c2c[nH]c(=N)o2)=O)cc(F)cc(F)c1 74253,Cc1nc(N(C(C)C(F)(F)F)c2ccccc2)ccc1C(F)(F)F 74254,n1(CCOC(C)C)nc(-c2cccc(N)n2)nc1-c1cnncc1O 74255,c1(C(N2C(=O)CCC(C(=O)OCC#C)C2)=O)[nH]c2cc(C)ccc2c1C 74256,N1(C(C(C)N(C)C)=O)CCC(NCc2cnn(C)c2)C1 74257,c1(NC(=O)NC(c2ccc(OC)cn2)C)nc2c(s1)CCc1ccccc1-2 74258,C1(NC(C2(NC(=O)OC(C)(C)C)CC(C)C2)=O)CN(C)CCO1 74259,C1(C(=O)NCc2c(C(=O)NC(CC=C)CC=C)scc2)CC2(C1)CC2(F)F 74260,c1(C(=O)NCCC2(O)CN(C(c3cc[nH]n3)=O)C2)cc(Br)ccc1Cl 74261,c1(C(=O)NC2C(CNC(c3n(CC)nc(C)c3)=O)CC2)cn2nc(C)sc2n1 74262,CCCCC(CC(=O)NCCC1(CO)CCCC1)NC(=O)C(C)(C)C.C1(=O)NC1 74263,S(=O)(=O)(c1ncn(S(=O)(=O)N(C)C)n1)NCC(=O)N(C1CNCC1(C)C)C 74264,C1(CC(=O)NC2(CCNC(CCCC=C)=O)CC2)Sc2ccc(Cl)cc2NC1=O 74265,CCC(C)(C(=O)N1CCC(NC(=O)COC2CC(F)(F)C2)CC1)OC 74266,N1(C(CCCOCC=C)=O)CCCC(O)(CCNC(=O)CCC(C)(F)F)C1 74267,C(=O)(C(O)C(C)SC)N(CCCNC(=O)Cc1ccc(Cl)s1)CC 74268,N1(C(CC2(C)CCN(C(c3noc(CC)c3C)=O)C2)=O)CC2(C1)CC2(F)F 74269,C1(C)(CNC(CNC(C)=O)=O)CN(Cc2ccc(Cl)cc2Cl)CCO1 74270,Cc1ccc(F)c(CC(=O)NC2CCN(C(=O)C(C)CC(N)=O)CC2O)c1 74271,N1(C(CC2ON=C(CC)C2)=O)CCC2CN(C(c3cncnc3CC)=O)CC2C1 74272,C(C(CC)(CC)CO)NC(C1N(C(C(CC)CN(C)C)=O)CCCC1)=O 74273,CN1CCN(C(=O)CNC(=O)Cc2cncnc2)C(CNC(=O)Cc2ccco2)C1 74274,c1(C(CC(=O)N(CCC(CC)O)Cc2ccccc2)NC)ccc(F)nc1 74275,N1(C(CNC(C=C)=O)=O)CCN(C(c2cc(-c3ccc(C)cc3)no2)=O)CC1C 74276,O(P(=O)(OCC)C(c1ccccc1)NC(c1cccnc1O)=O)CC 74277,c1(C(=O)OC)cc(NC2CC(C(F)F)C2)cc(Cl)c1 74278,N1(C(Cn2c(C)nnn2)=O)CCCC12CCC(NC(=O)C(CO)N(C)C)CC2 74279,CN1CC2CCN(C(=O)C(CCC3CCC3)NC(=O)CCC3CCOC3)CC2C1 74280,Cc1cn(C)cc1C(=O)NC1CC(CNC(=O)CC2(C)CCCO2)C1 74281,c1(OC)cc(OC)cc(C(F)(F)C(=O)N(C)CCNC(C2CCCNC2=O)=O)c1 74282,c1(OC)ncccc1C(N1CCC(OCCNC(c2csnc2OC)=O)C1)=O.NCC 74283,N1(CC(c2ccc(C)cc2C)(F)F)CCc2ccc(N(C)C)cc2C1 74284,c1(C(N(C(C)CNC(=O)C(C(C)C)n2ccnc2)CC)=O)snc(O)c1Cl 74285,c1(C(CNC(c2cc(Br)cn2C)c2n(CCCOC)nnn2)O)cccc(Cl)c1 74286,c1(CC)nc(O)c(C(N2CCC(NC(=O)C(C)OCCN(C)C)C2)=O)cc1C 74287,C1(n2cc(CNC(C)=O)nn2)CN(C(c2ccc(C(C)C)cn2)=O)CC1C 74288,N1(C(CCN(C(C2CC(OCC)C2)=O)C(C)C)=O)CCOCC1C1(C)CC1 74289,C=C(C)C(C)(C)C(=O)N1CCC(O)(CN(C(=O)CNC(C2CCCC2)=O)C)CC1 74290,c1(CC(=O)Nc2ccc(NC(c3cocn3)=O)cn2)c(F)cccc1F 74291,C(=O)(CC1C(=O)Nc2c(F)cccc21)NCC1(F)CN(C(CC2CN(C)C2)=O)C1 74292,Cc1ccc(S(=O)(=O)Nc2ccc(C)c(Cl)c2)cn1 74293,C1(O)(CC(=O)N(CC(C)NC(=O)CNC(=O)C2CC2)C)CCOCC1 74294,c1(OC)cc(C)c(S(=O)(=O)N(c2ccccc2C)CCOC)c(C)c1 74295,c1(OC)cc(Br)c(OC(c2scc(C(COC(C)=O)=O)c2)=O)c([N+](=O)[O-])c1 74296,O=C1CC2(CCC2)C(CNc2ccc(C(=O)O)cc2Cl)N1 74297,c1(N(CCC(C)NC(C(c2cccc(C)c2)(F)F)=O)C)nc2ccc(Cl)cc2s1 74298,c1(NC(CCC)=O)nc(=NC2CCCC(N(C)C)C2)nc(OC)[nH]1 74299,c1(OC)cccn2ncc(C(N3CCN(C(=O)C(CSC)OC)C(CF)C3)=O)c12 74300,c1(SC(C(N2C(c3c(OC)cc(Cl)cc3)CCC2)=O)C)nc2ccc(C)cc2s1 74301,C(=O)(CC(C)(O)COC)N1CCC(NC(c2ncc(OCC)nc2)=O)C1C 74302,C12(NC(C(F)=CCC)=O)CCCCC1CN(C(c1[nH]nnc1C1CC1)=O)C2 74303,N1(CC2(CS(C)(=O)=O)CCN(C(=O)OC(C)(C)C)C2)CCOC2(CCOC2)C1 74304,Cc1ccc2cccc(C(N3CCC(NC(=O)C(F)C4CCC4)C34CC4)=O)c2n1 74305,CC(C(=O)N1CCCCC(CNC(=O)C(CO)NC(N)=O)C1)S(C)(=O)=O 74306,C1(C(N2CC(CCC#C)C2)=O)CCCC1CNC(C1SCCS1)=O 74307,N1(C(CCCCC=CC)=O)CC2(CCCCN(C(c3ccnc(OC)c3)=O)C2)C1 74308,C1(C(N(CCCCCC)CCO)=O)CC2CCCC2N1C(=O)Cc1ccc(C)o1 74309,c1(C(N2C(CNC(c3nccc(C)n3)=O)C(C)CC2)=O)cnn2c1NCC(C)C2 74310,N1(C(C(C(CC)C)N)=O)CCCC12CN(C(c1cccc3occc13)=O)C2 74311,C1(C)(CNC(c2n(CC)ncc2)=O)CC(F)(F)CN1C(=O)CCOC(C)C 74312,N1(C(C(N2CCOCC(NC(C=CCOC)=O)C2)=O)C)CCc2ccccc2C1 74313,c1(C(C)C)ccc(C(=O)NC2(C)CC(NC(=O)Cc3cncnc3O)C2)cn1 74314,c1(CC(N2CCC(NC(C=C(CC)C)=O)C(O)C2)=O)ccc(S(=O)(=O)NC)cc1 74315,c1(CC(=O)NC(CN(C(COCCC#C)=O)CC)C)cnn(C(C)C)c1 74316,C1(NC(COC2CN(C(C3CC(=C)C3)=O)C2)=O)CCC(C2CC2)CC1 74317,C1(C(N(C(CNC(=O)CC(C)(C)C#N)C2CC2)C)=O)CN(CP(C)(C)=O)C1 74318,C1(CNC(c2ccc(Br)s2)=O)CCCC(NC(C2SCCS2)=O)C1 74319,N1(C(C2(C)CCOC2)=O)CC2CC(C(=O)NCC3(CO)CC3)C(C2)C1 74320,CCCC(C(=O)NC(C)CC(C)NC(c1ncccc1F)=O)c1ccccc1 74321,C(C(C)(C)CC(=O)N1CCOC(CO)C1)NC(CCC=CC(C)C)=O 74322,c1(C(=O)NCC2(OC)CCN(C(=O)C(C)S(C)(=O)=O)C2)csc2c1CCC(C)C2 74323,N1(C(C=COCC)=O)CCCOC(CCNC(=O)C(C)N2CCC2)C1 74324,C1(C(N2CCC(C(=O)N(C3CC4CCC3O4)C)C2)=O)(OC)CCCCC1 74325,c1(C(N2C(C(N(CC)CC)=O)CCC2)=O)ccc2cc(Br)ccc2c1 74326,c1(SCC(=O)NCC2COCCN2C(=O)CCc2cc[nH]n2)ccc(F)c(F)c1 74327,c1(OCC)ccc(C(N2CC(C(=O)NCC(C)(C)C(N)=O)C(F)C2)=O)cc1 74328,c1(C(N2CC(CC(=O)NCCC#C)OCC2)=O)ccc2cc(Br)ccc2c1 74329,c1(C(=O)NC(C)CNC(C2C=CCCC2)=O)ccc2c(c1)C(=O)CCN2 74330,N1(C(CN(C(COC)=O)C)=O)CCC2(CC1)CC2CNC(c1cc(SC)n[nH]1)=O 74331,C(C1=NOC2CN(C(=O)CNS(N)(=O)=O)CC12)NC(Cn1c(C)nnn1)=O 74332,CCC(C)C(O)CC(=O)N(C1CCCN(C(c2cccc(CN(C)C)c2)=O)C1)C 74333,c1(N2CCN(C(c3c(C)snc3)=O)CC2C)ncnn2cccc12.c1(CN)ccccc1 74334,C1(C(=O)NCCC2CN(C(C3(OC)CCOC3)=O)C2)C2(CC2)C12CC2 74335,N1(C(=O)COCCF)CCN(C(c2c(O)cc(F)cc2F)=O)CC2(CC2)C1 74336,N1(C(c2c(C)c(N)cnc2)=O)Cc2ccc(CNC(C3C(C)C3C)=O)cc2C1 74337,c1(-c2cc(C(=O)NC(CN(C(C(CC)OC)=O)CC)C)n[nH]2)ccc(C)c(C)c1 74338,N1(C(C2(OCC)CCOC2)=O)CCN(C(C2CC(OC3CC3)C2)=O)CC(O)C1 74339,c1(OC)ccccc1C(O)C(=O)NC1CC(CNC(=O)C(CO)OC)C1 74340,N1(C(C(n2c(C)ncc2)C)=O)CC(N(C(=O)Cc2cncn2C)C)C(O)C1 74341,C1(n2cccn2)(NCCn2c(C(C)C)ncc2)CCOCC1 74342,c1(CC)ccc(C(C)(C)C(=O)N(C(C)CNC(=O)Cc2ccnn2C)CC)cc1 74343,Cc1cc(Cl)c(Cl)cc1C(=O)Nc1nc2ccccc2[nH]1 74344,CC1(O)CON(C(=O)C2CSCCS2)C1 74345,c1(CC(N2CCC(N3CCN(C(=O)C4=COCC4)CC3)C2)=O)ccc(F)c(F)c1 74346,C1(C(=O)Nc2c(-n3c(C)ncc3)cccc2)CC(F)(F)CN1S(=O)(=O)C(F)(F)F 74347,c1(CNC2CC3(CC(C(N(CCCCC)CCO)=O)C3)C2)cc2ncccc2[nH]1 74348,N1(CC(=O)N(C)CC2CCN(C(C(CC)(C)CC)=O)CC2)CCc2ccccc21 74349,C(c1cc(C)cc(C)c1)=CC(N1CC(O)(CCNC(C(CCSC)OC)=O)C1)=O 74350,c1(C(=O)NC2C3(CC(NC(C(C(=O)NC)(C)C)=O)C3)C2)cnc2sc(C)nc2c1 74351,c1(C(C)(C)C)csc(C(N2CCCC2C(=O)OC(C)(C)C)C(=O)NC2CCOC2)n1 74352,N1(CC=C)C(=S)NC(c2ccc(Cl)cn2)C2=C1CC(C)(COC)NC2=O 74353,c1(C(=O)NCC2C(CNC(CSc3n(C)nnn3)=O)C2)nn2ccccc2c1Br 74354,c1(C(=O)NC2CCCC2NC(C2CC2C(F)F)=O)cc2scc(Cl)c2[nH]1 74355,CC1CCN(C(C2(CNC(=O)Cc3ccoc3)CC=CC2)=O)C1C 74356,N1(C(C(C)=C(C)C)=O)CC2CCOCC2(NC(=O)CCOCC2CC2)C1 74357,c1(C(N2CCC(C(=O)OC)C2(C)C)=O)ccc(S(=O)(=O)NC(CCCCC)=O)cc1 74358,C1(CNCc2ccn(CC(F)F)n2)CCCCC12CCC2 74359,N1(C(c2cnc(-c3cn(Cc4cnccc4C)nn3)s2)=O)CC(O)CC1SC 74360,C1(CCNC(c2n(C)nnc2)=O)COCCN1C(c1cc(-c2ccns2)on1)=O 74361,c1(C(=O)NC(CCN(C(C=CCC)=O)C)C(C)C)cc(C)cc2cccnc12 74362,c1(C(=O)NCC(CO)NC(=O)C(F)F)cccc(-c2scc(C)n2)c1 74363,CC(CC(=O)NC1CC(F)(CNC(=O)Cc2cncnc2)C1)C1CCCO1 74364,CCC(C)C(CC(=O)NCCCn1cnnc1)NC(=O)COC1CC1 74365,c1(C(=O)NC2(CCC)CCN(C(C3CCSCC3)=O)CC2)cccc2c1NCC2 74366,CC(C)(CCCO)C(=O)N1CCOCC(CNC(c2coc(C3CCC3)n2)=O)C1 74367,N1(C(C2CCC(N(C)C)CC2)=O)CC2CC(C1)N(C(c1cc(Cl)ccc1O)=O)C2 74368,C(=O)(CCC(F)(F)F)NCC=O.C1(C)(OCC)CN(C(=O)C(c2ccnn2C)N)C1 74369,c1(C(N2CCC(F)(CF)C2)C(=O)NCCCF)cnc2n1CCC2 74370,c1(N2CCC3(C)C(C2)C3(F)F)nc2c(c(=NC3CC3)[nH]1)COC2 74371,N1(C(c2cnc(CC(C)C)[nH]2)=O)CCN(C(=O)CC2(O)CCOC2)CC1CCO 74372,N#Cc1ccc(C(=O)NC2CCN(C(c3ccc4n[nH]cc4c3)=O)C2)cc1Cl 74373,c1(CC(N2CCN(C(c3cnc(C)o3)=O)CC2)=O)ccc(C)c(Br)c1 74374,N1(c2cc(NC(CC)COCCOC)nc(C)n2)CCCC(C)(OC)CC1 74375,c1(OC(C)C(=O)N(CC(C)(C)CNC(=O)CC(C)C(F)F)C)ccc(F)c(F)c1 74376,C1(NC(=O)OC(CC(C)C)C)CC(F)(F)C1(C)C 74377,N1(C(C(C)C2CCCC2)=O)CCCC(C)(CNC(C2CCOC(C)(C)C2)=O)C1 74378,CC1(C)CCC(CNC(C2CNC(=O)N2)=O)N(C(=O)CC2(C)CC2)C1 74379,C1(C(NOCC(C)O)=O)CCCCC1NC(=O)OC(C)(C)C 74380,CC1(C)CC(C)(NC(=O)CSCCNC(c2ncncc2Cl)=O)C1 74381,CCCCC(CN(C1CCS(=O)CC1)C)CC 74382,N1(C(c2cn(CCC)nc2)=O)CCC2(CCN(C(C3CC(=O)NC(=O)C3)=O)C2)C1 74383,C1(OC)CC2CC(C(=O)NCC#CCNC(c3ccc(C(C)(F)F)cc3)=O)CC12 74384,CC(C(F)C(=O)NCC1(C(=O)O)CC1)C(F)(F)F 74385,C1(C(=O)NC2CCN(CCOC3C(C)CCCC3)CC2)CCCC12CCOCC2 74386,c1(SCC(=O)N(C2CCN(C(c3cccnc3C(F)F)=O)C2)C)ccccc1Cl 74387,c1(CC)cccc(CC(=O)NC23CC(NC(=O)Cc4n[nH]c(=N)s4)(C2)C3)c1 74388,c1(N2CC(C(N(C3CC(NC(CC(=O)N(C)C)=O)C3)C)=O)C2)ccc(F)cc1Cl 74389,c1(C(N2CCCC2CC2CC2)C(=O)NCCCOC)c(C)cnn1C 74390,c1(C(N(CCC2N(C(C(COC)C)=O)CCCC2)C)=O)cc(Cl)cnc1O 74391,N1(C(C2CC(C)(C)C2)=O)CC(NC(c2cn(CCCF)nn2)=O)CC12CCC2 74392,N1(C(=O)NC2CCCC(C(c3ccc(O)nn3)=O)C2)CCC(CC(=O)NC(=C(C)C)CC)CC1 74393,C1(C)(CC(=O)NCC2(C)CCCO2)CCS(=O)(=O)N1 74394,N1(C(C=NOC)=O)CCC(OCCNC(=O)CC(C)C(=O)NCc2ccco2)CC1 74395,c1(C(=O)NC(CC)(CNC(C2CC(OC(C)C)C2)=O)CC)ncc(C#N)cc1C 74396,C(=O)(NN1CCCC(C(=O)O)C1)C1N(C(C2CC(C#N)C2)=O)CCC1 74397,c1(CNC(C2C(C)CCO2)=O)ccc(CNC(c2nc(C3CC3)cs2)=O)cc1F 74398,c1(C(=O)NC(C2(O)CN(C(C(=O)NC(C)C)=O)C2)C)cc(F)cc2nccnc12 74399,O=C1CCC2(CN1)CN(C(=O)CCC1CCCCN(C(c3cncc(F)c3)=O)C1)C2 74400,C(CC(C)P(C)(C)=O)N1CCCC(CN(C)CC)C1 74401,c1(C(=O)NC2CCC(CNC(Cc3nc(C)[nH]n3)=O)C2)ccc(C)c(F)c1 74402,C1(NC(c2cn(CCC)nc2)=O)CN(C(C2(COC)C=CCC2)=O)CC2(CC2)C1 74403,N12CCCC(C1)NC(=O)C(c1csc(C)n1)N(C)CC2=O.C(COC)OC 74404,CC(CS(C)(=O)=O)C(=O)N1CC(N2CCN(C(C3(C#N)CCCC3)=O)CC2)C1 74405,c1(OCC)cc(C(N2CCC(NC(=O)Cc3cc[nH]n3)C2)=O)cc(Cl)c1O 74406,C=Cc1ccc(C(=O)NC2CCCN(C(=O)C(Cc3ccsc3)NC=O)C2)cc1 74407,Cc1cc(C)c(C(N2CCC(NC(c3ccc(CO)c(Cl)c3)=O)CC2C)=O)cn1 74408,c1(N2C3CN(C(c4cc(C(C)C)no4)=O)C(C3)C2)ncnc2n[nH]c(Br)c12 74409,C12(C(=O)NCC(C3CC3)NC(COC(C)(C)C)=O)CCC(OC(C)(C)C)(CC1)C2 74410,c1(C(N2C3CC(CNC(C4CC(F)(F)C4)=O)C2CC3)=O)ccc2c(c1)SCCN2 74411,CC(=O)CCCC(=O)NC(C(=O)N1CCC(OC2CC2)C1)C(C)(C)C 74412,N1(C(=O)NC2CC(=O)N(C)C2c2ccccc2)CC(C)(CO)CC1(C)C 74413,N1(C(c2ncn(C)c2)=O)CCC2CCCC12C(=O)NCCN1CCC2CC12 74414,N1(C(c2c(C)n(C)nn2)=O)CC2CCCC2C1C(N1CC2(CCOC2=O)C1)=O 74415,c1(C(=O)NC(CC=C)CNC(c2cc[nH]c2C)=O)nn(C)nc1C(F)(F)F 74416,c1(OCC)nc(C)ccc1C(=O)NCC1CCC(NC(=O)CCn2cncn2)C1 74417,C(CCCC(=O)NCc1cc(C(=O)NCCn2cnnc2C)n[nH]1)(OC)OC 74418,C1(CNC(=O)C=Cc2cnc[nH]2)CN(C(=O)CC2CC3CC3C2)C2CCCCC12 74419,C1(NC(Cc2c(C)con2)=O)CC12CCN(C(=O)CC1CC3CCC1C3)C2 74420,C1(C(=O)OCC)(C(=O)NCC(=O)NCC2(Cc3cnn(C)c3)CCC2)CCCC1 74421,Cc1ccc(C(=O)N(CCCCC(=O)N2CC(CO)(CO)C2)C)c(O)n1 74422,C(CC(C)C)(C(=O)NC1(CCCCNC(=O)Cn2nc(C)oc2=O)CC1)OC 74423,c1(N2CCC(OCC)C2)nc(N2CC=C(C)CC2)nc2sccc12 74424,c1(C(N2CCC(N(c3ccccc3)C(C3(OC)CC3)=O)C2)=O)c(C)nn(C)c1N 74425,c1(OC)cc(C=CC(=O)N(C2CCN(C(=O)C3CC3)C2)Cc2ccccc2)sn1 74426,C1(NC(c2ncn(C)c2)=O)CC2CC(C1)N(C(=O)CC1COC(C)(C)CO1)C2 74427,c1(C(=O)NC2CC(CF)C2)ccc(Sc2nncs2)cc1 74428,C1(NC(CCOCCOC)=O)CCCC(C(=O)N(C(C)CCO)CC)CC1 74429,N1(C(C(C(C)C)NC(C(CC=C)OC)=O)=O)CCN(C)C(CO)C1 74430,C(N=c1[nH]c2ccc(F)cc2o1)C1CN(C(C(C)SC)=O)C(C)C1 74431,C(=O)(C(C)C(CC)CC)NCC1C(C)CCN(C(c2c(CC)nn(C)c2)=O)C1 74432,N1(C(C2(NC(C(COC)C)=O)CCC(C)(C)C2)=O)CCn2nc(C)cc2C1 74433,N1(C(CCC)=O)CCC2(CCN(C(c3c[nH]cc3COC)=O)C2)C1 74434,CC1(C#N)CCC(OC(C23CC2CS(=O)(=O)C3)=O)CC1 74435,Cc1cc(C(=O)NC2CCN(C(c3ccc(-c4ccc(Cl)cc4)s3)=O)C2)[nH]c1C 74436,c1(C(N2C(CNC(C(CC=CC)C)=O)CCCCC2)=O)cc2c(nn1)CCCC2 74437,CC#CC1CN(C(C2CC(NC(=O)CC3CN(C(C)=O)C3)C2(C)C)=O)C1 74438,C1(CNC(CCc2cnc(C)s2)=O)CN(C(c2cc3c(s2)CCC3)=O)C(C)(C)C1 74439,C1(NC(Cc2c(C)cccn2)=O)CC12CCN(C(c1cnc(C)c(C)c1)=O)CC2 74440,CC1OCCC1CN(C(=O)Cn1nnc(C2CC2)n1)C 74441,C#CCC(CC#C)C(=O)NC1CN(C(=O)C(F)Cc2ccccc2)CC1OC 74442,C1(C(=O)NC2CC(C)(NC(C3CC(C)(CC)C3)=O)C2)CC12CCCC2 74443,c1(OC)ccc(Br)cc1CCNC12CC(C(=O)OCc3ccc[nH]3)(C1)C2 74444,C1(C(N(CC)CC2CCCC2)=O)CCN(C(=O)C=C2CCC2)C(C)C1 74445,C(C(C)CC(=O)N(CCC(=O)NCC1(C)CCCS1)CCCO)OC 74446,C1(NC(C2CC(=O)NC2)=O)CCCC12CCN(C(=O)CCc1csc(O)n1)CC2 74447,C(=O)(C(C)C1=CCCC1)NCCCN(C(C1CCc2c[nH]nc2C1)=O)CC 74448,C1(C(=O)NCCCCCC)CN(C(c2c(C)cnn2C)=O)CC1(F)F 74449,C1(O)(C(C)NC(=O)CCc2cccnc2)CCN(C(=O)C=Cc2ccnn2C)C1 74450,n1(CC(=O)NC(CCCNC(C2(CC(C)C)CCC2)=O)C)cc(S(N)(=O)=O)cn1 74451,c1(OC)ccc2c(C(N3CCCC(c4cncn4C)C3)=O)ccnc2c1 74452,N1(C(C(C(COC)C)C)=O)CC(C2CCCN(C(=O)CCCC3CCC3)C2)C1 74453,N1(C(CCCC#C)=O)CCCCC(CNC(=O)Cc2ccc(C)nc2)CC1 74454,N1(C(C=Cc2c(C)ncs2)=O)CCCN(C(c2cncc(C(N)=O)c2)=O)CC1 74455,C=Cc1ccccc1-c1ccc(C(C)(C)NC(c2ccc(Cl)cc2C)=O)cc1 74456,N1(C(CC(CCCCC)O)=O)CCC2CN(C(C3CC(=O)N(C)C3)=O)CC2CC1 74457,C#Cc1cc(NC(=O)C(N2CC3CCC2CC3OCC)=O)cc(F)c1 74458,C(=O)(CC(O)C(C)C)NC1C(C)(CNC(C)=O)CCC1 74459,N1(C(C2N(C(C(CC)CN(C)C)=O)CC(O)C2)=O)CC(F)(F)CC1C 74460,N1(C(CCSCC)=O)CCCC(C(C)(O)CNC(c2ccc(F)o2)=O)C1 74461,N1(C(c2c(C)cc(CC)o2)=O)CCCC2CCN(C(C3(SC)CC3)=O)CC12 74462,c1(NC(N(CCOC)CC2CCCCC2)=O)c(CN(C)C)ccnc1SC 74463,C1(C(=O)NC(C2CN(C(=O)C(F)=CC3CC3)C2)C)CSCN1CC(F)(F)F 74464,S(=O)(=O)(c1cnc(O)c(F)c1)N1CC(CCC(N)Cc2ccccc2)C1 74465,N1(C(C2(CC)CC2)=O)CCC12CCN(Cc1ccc(O)cc1O)CC2 74466,c1(C2C(NC(C(C)(c3cn(C(C)C)nn3)NC(C)=O)=O)C2)ccccc1F 74467,C1(CC(=O)NCCC2CC(NC(c3n(CCCC)ncc3)=O)C2)CC2CCC1O2 74468,C(CC(C)(O)C1CC1)NC(CN(CCOC)C(c1coc(CO)c1)=O)=O 74469,N1(C(C2C(C)(C)CC2)=O)CC(NC(c2ccc(O)nc2Cl)=O)CC(O)C1 74470,Cc1cccc(Cl)c1OCC(=O)NC1CCCCC1NC(=O)CN1CCC(C)C1 74471,c1(C(C2COCC2(C)C)N(C)C(=O)NC(C)(C)C)cc2ccccc2n1C 74472,C=CCC(C)(C(F)F)NC(=O)C(C1CCN(C(c2cn(C3CC3)nn2)=O)CC1)C 74473,C1(CN(C(c2cnn(C)n2)=O)CC)CCN(C(=O)CCC2CCCOC2)CC1 74474,C1(CNC(C2(C)CC2Br)=O)CCCC1NC(=O)CCCC1CCC1 74475,c1(C(N(CC(=O)NCC2(C(C)O)CC2)CC2CC2)=O)ccc([N+](=O)[O-])o1 74476,C#CCC(C(=O)NCc1ccccc1CNC(=O)Cn1cnccc1=O)C1CC1 74477,c1(C(N2CC(CCCCNC(C3CCCC(O)C3)=O)C2)=O)cccc(F)c1 74478,CC1CN(C(=O)NCC2CCCCC2)CC1CCNC(=O)CC1COCCO1 74479,C(=O)(CCCC(=O)NCCN(C)C(c1ncc(C)cc1C)=O)OC 74480,CC1(C)CN(C(C2CC23CCC3)=O)CC(CNC(c2csc(C(F)(F)F)n2)=O)O1 74481,C#CCC(CC(=O)NCCCN(C(=O)C(C)S(N)(=O)=O)C)c1ccccc1 74482,c1(C(=O)NCCC(C(N2CC3C(CC)(C3)C2)=O)O)cn2c(n1)CCC2 74483,CC1COCC(CC(N2CC=CC(C(=O)Nc3ccccc3CN(C)C)C2)=O)O1 74484,C1(NC(c2nnc(C)s2)c2nnnn2C2CC(F)(F)C2)CCSC2(CCC2)C1 74485,Cc1cc(N2CCCC(C(=O)Nc3ccccc3C#N)C2)n2nc(C)cc2n1 74486,N1(C(c2cn(CC)nc2)=O)CC(NC(=O)C(=Cc2ccco2)C)CC2(CC2)C1 74487,C1(CNC(C2OCCC2c2ccccc2)=O)C2CN(C(C3CCCC3)=O)CC12 74488,c1(C(=O)NCCN(C)C(C2(O)CCCN2)=O)ccc(OC2CCCCC2)cc1 74489,CCCC(CCCNC(c1cnc(C)nc1C)=O)NC(C1CCC1(OC)OC)=O 74490,c1(C(C)NC(=O)Nc2c[nH]nc2Cl)cc(F)ccc1O 74491,Cc1ccccc1COCC(=O)NC(C1CCCN1C(C1COCCO1)=O)(C)C 74492,c1(-c2cn(CC)nn2)cccc2c1N(C(C13CC(CCOC)(C1)C3)=O)CC2 74493,C(=O)(C(CO)C(F)(F)F)N(C(C1CN(Cc2ccccc2)CCO1)C)C 74494,CCCCC(C(=O)NC1CN(C(c2cc(C)nc3ccnn23)=O)CC1C)C(C)C 74495,c1(N(C)CCOCC2CC2)cc(NCC2(C)CC2Br)ncn1 74496,c1(C(=O)NC2CCN(Cc3ccc(F)cc3O)CC2F)c[nH]c2c(Cl)cccc12 74497,N1(S(CC(C)C)(=O)=O)CCOCC(NC(=O)Cn2cc([N+](=O)[O-])cn2)C1 74498,CC1CN(c2cccc(F)c2)CCN1S(=O)(=O)Cc1c(Br)cncc1Br 74499,c1(CN(CCNC(C(CC)Cc2ccccc2)=O)CC)ccc2c(c1)CCCC2 74500,N1(C(C2CC(C#N)C2)=O)CC2CCC(C1)C(NC(=O)C(c1ccc(F)cc1)O)C2 74501,CCC(C)C(C)C(=O)NCC1CC(NC(c2ncccc2N(C)C)=O)C1 74502,c1(C(=O)OC)cc(C(N2CCC(C(C)NC(=O)C=C(C)C)CC2)=O)n(C)n1 74503,C1(S(N)(=O)=O)(C(=O)NC2CC(c3cn(CC4C(COC)C4(C)C)nn3)C2)CCC1 74504,N1(C(c2[nH]cc(S(=O)(=O)NC)c2)=O)CC2CCN(C(=O)C(C)OC)CC2C1 74505,N1(CC(=O)NCC(C(C)C)NC(=O)C(C)(O)C2CC2)CCCCC1C 74506,C1(NC(c2n(CCSC)nnn2)c2cnnn2C2CC2)C2CCCOC12 74507,C1(NC(C(C)NS(CCC)(=O)=O)=O)CCCC(CNC(=O)Cc2nnc(O)s2)C1 74508,C(=O)(C1=CCCOCC1)NC1(CN(C(=O)CC2(C)OCCO2)C)CC1 74509,CCCC(CCC)=CC(N1CCC(C)C1CNC(=O)CCCC1CCOCC1)=O 74510,C(=O)(C(CC(C)C)NC(=O)CC1CN(C(c2cccc(=O)n2C)=O)CC1C)NC 74511,CCC(CNC(=O)C#CC1CC1)(CC)C(=O)NCc1cc(C(C)C)no1 74512,N1(C(c2c(CCC)n[nH]c2)=O)CCC(NC(C23CCCC2CCC3)=O)C(O)C1 74513,c1(C(N2CCN(C(=O)CO)CC2Cc2ccccc2)=O)cnn2ccncc12 74514,CCCS(=O)(=O)C(C)C(=O)N1CCCC(CNC(C2C3C4CCC(C4)C23)=O)C1 74515,C12(CNC(C3(CCCC)CC3)=O)CCCC(CN1C(=O)CCc1cnc[nH]1)C2 74516,c1(C(=O)NCCOCCC(=O)NCC(C)OC(F)F)cc(Cl)n(C)n1 74517,c1(OC)ccc(SCCCC(=O)NC2CC(NC(c3ncoc3C)=O)C2)cc1 74518,c1(OCC)cc(NC2CC3CCC2N3C(=O)CSc2ccccn2)nc(C)n1 74519,C(=O)(NNC(=O)CCCS(C)(=O)=O)C1CC(C(=O)OC(C)(C)C)OC1 74520,c1(C(=O)NC(CC)CNC(C23CCC(CC2)C3)=O)cc2c(cn1)COCC2 74521,CC(F)CC(=O)NCC(c1ccccc1)NC(=O)Cc1cc(Cl)cs1 74522,O=C(CC(CNC(=O)CCC1CCCCC1)C1CCC1)NCC(CO)C1CCC1 74523,C12(C(=O)OC)COC(C1)C(NC(=O)C(c1cccc(Br)c1)F)C2 74524,c1(CNC2C(SCC)CCCC2)c(Oc2ccccc2)cccc1Br 74525,c1(CC(C(=O)NCC(CNC(c2ccc(C#C)o2)=O)(C)O)O)cc(Cl)cc(Cl)c1 74526,N1(C(c2c(CCC)n(C)nn2)=O)CCCC(n2ccnc2)CC1 74527,Cc1ccnc(C(C)NC(=O)C(C)N(C(=O)C2=NOCC2)C)n1 74528,C(=O)(C(C(=O)N1CCC(COC(=O)CCC2CC2)C1)OC)OCC 74529,N1(C(Cc2ccn(CC)n2)=O)CCC(O)(CN(C(=O)C2=C(Cl)CC2)C)C1 74530,C1(C(=O)OC)CC(n2cc(CN3CCOC3=O)nn2)CN1C(=O)C(O)C1CC1 74531,CC1CC(C)(C(=O)NCC2CN(C(c3c[nH]cc3Br)=O)CCC2(F)F)CC(C)O1 74532,CC(C)C(F)(F)CC(=O)NCCCCCC1CCN(C(c2csnn2)=O)CC1 74533,C1(CNC(=O)COc2ccc(Cl)cc2)CC2CCCC2N1C(C1CCC1)=O 74534,C1(NC(C(C)SC(C)C)=O)CC(C2CCN(C(=O)CC34CCC(CC3)OC4)C2)C1 74535,N1(C(C(c2cccnc2)C)=O)CCCC2(NC(c3ccnnc3Cl)=O)CC2C1 74536,C(=O)(C(C)C(C)C)NC1(C(CNC(C2(CCOC)CCCC2)=O)O)CC1 74537,c1(C(=O)NCC2(C)CCC(NC(c3cnc(CC)s3)=O)C2)cc2cc[nH]c2cn1 74538,c1(C(COC(C=CSC)=O)NC(=O)C(O)CN2CCCC2)cncc(OC)c1 74539,O=C1CN(C(C2CC(F)(CF)C2)=O)C(C(N2CCC3CCCC23)=O)CN1 74540,N1(C(C(c2cn(C)nc2)O)=O)CCN(C(C2(C)CCCCC2)=O)CC12CC2 74541,C(=O)(CCCCSC)N(CC)CC1CCCN1C(c1cc(C(C)C)on1)=O 74542,C1(CC(=O)N(C(C)CNC(C2CC(C)C2)=O)CC)CC1(C)C 74543,C1(NC(=O)COCCc2ccc(Cl)s2)CC2CC1N(C(=O)CCC1CCCO1)C2 74544,c1(OC)ccc(Br)c(C(=O)NCC(CO)NC(c2cc3sccc3[nH]2)=O)c1 74545,c1(C(=O)NCC2CCCN(C(c3c(C)con3)=O)C2)ccn2nncc2c1 74546,CCC(C(=O)NCC1(CCNC(=O)C(C)Cc2ccco2)CC1)NC(C)=O 74547,N1(C(C(C2CCC2)OC)=O)CC2(NC(c3cn(C)nc3C)=O)CCC1CC2 74548,CC1CN(CC2CCN(C(=O)CNc3ccc(C(C)(C)C)cc3)C2)CC(C)O1 74549,c1(OCC(N2CCC(C(=O)NCC(c3ccoc3)O)CC2)=O)ccc(Cl)c(Cl)c1 74550,Cc1cc([N+](=O)[O-])cc(C(=O)NCCCOCCNC(C2CC(C)(C)C2)=O)n1 74551,c1(NC2C(C3C(C)C3)C2)nc2c(c(=NCc3ncnn3C)[nH]1)CCC2 74552,N(C(=NCCNS(C)(=O)=O)NCc1ccc(C2CC2)o1)C1CCCC(OC)C1 74553,c1(C(=O)NCC(C(C)C)NC(C2CC(N(C)C)C2)=O)ccc2c(c1)N(C)C(=O)C2 74554,c1(C2(C(=O)NCC3(C(C)(C)OC)CC3)CCCCC2)ccc2c(c1)OCCO2 74555,C1(C(=O)NC2CN(C(c3cscn3)=O)C3CC23)CN2CCCN1CC2 74556,c1(CNC(C2CCN(C(c3cnc(N(C)C)o3)=O)C2)=O)cccc(I)c1 74557,c1(C(N2CCC(Oc3ccc(C(C)=O)cn3)C2)=O)cccc(N)c1.CCCC(=O)NC 74558,N1(C(C2CC=CCC2)=O)CC2CC(N3CCC(F)CC3)C1C2 74559,C12(CC(=O)NC3CC(N(C(C(C)N(C)C)=O)C)C3)CC3CC(C1)CC(F)(C3)C2 74560,c1(C(N2C(C(N(CCCO)CC)=O)CSCC2)=O)ccc(O)c(C)c1 74561,c1(OC)ccccc1CNC(=O)C(C1CCC(C)(C)C1)N(CC(F)F)C 74562,C1(OC)CC2CCC1CC2C(=O)Nc1cccc(C(N2CCOCC2)=O)c1 74563,C(=O)(C(C)(O)CC(C)C)NC(c1c(C)cccc1Br)C(=O)NCC=CC1CC1 74564,C1(C(=O)NCC(C)N(C(C(c2ccc(F)cc2)CC)=O)C)CC2(C1)CC(O)C2 74565,N1(C(c2c(C)nc(C)o2)=O)CC(C(N2CCCC(CC3CC3)C2)=O)OC(C)C1 74566,C1(C(=O)NC2CC(C(C)O)C2)CC12CCN(C(C1(C(N)=O)CCC1)=O)C2 74567,C1(CNC(C2CCC(C)C2)=O)CN(C(C2CCS(=O)(=O)C2)=O)CCN1C 74568,N1(C(CC2(COC)CC2)=O)CC2(C(=O)NCc3cc(Cl)no3)CC1CO2 74569,C1(NC(COC2CCN(C(C(C)CCN(C)C)=O)C2)=O)CC12CCOCC2 74570,c1(C(=O)NC2CN(C(CC3CC(OC)C3)=O)C(C)CC2)c(F)ccc(Cl)c1N 74571,c1(NC(=O)NCC(Cc2cccc(C)c2)CO)ccc2c(c1)OC(C)(C)O2 74572,Cn1cccc1C(=O)NCC1(CCNC(c2n[nH]cc2CN(C)C)=O)CC1 74573,c1(C(N2CCC(CO)(NC(c3ccnc(F)c3)=O)CC2)C)ccc2ccccc2c1 74574,C(CCC(=O)NC(c1cn(C(C)C(=O)OC)nn1)C)=CCC=C 74575,C12(CNC(c3cnsc3)=O)CN(C(C3CC4(CC4)CO3)=O)CC1CCO2 74576,c1(CC)nc(C)ccc1NC(C1COCCC1NC(=O)CCCCC1CC1)=O 74577,C12(C(N3CC(CC)OCC3)=O)COCC1CN(CCc1[nH]cnc1C)C2 74578,c1(C(N2CC(O)(CNC(C(C(CC)O)C)=O)C2)=O)cc2sccc2n1C 74579,c1(C(N2C3CC(NC(C(C4CC4)OCC)=O)C2CC3)=O)c(F)cccc1[N+](=O)[O-] 74580,C1(CC(=O)NC(CC)CNC(C2CCCCS2)=O)CCC2(CC1)CC2 74581,C1(CN(C)C(C2CCCN(C(N)=O)C2)=O)CCN(c2ncncc2Cl)CC1 74582,c1(N2CC(C)C(CS(N)(=O)=O)C2)nccc(=NCc2cncn2C2CC2)[nH]1 74583,C=CCCCCCC(=O)N(C1CC(NC(=O)CCNC(=O)NC)C1)C 74584,Cc1ncnc(C)c1C(N1CCN(C(=O)CC(=O)NCC(F)(F)F)C(C)C1)=O 74585,c1(C(=O)NCC(CN(C(=O)C(O)c2ccsc2)C)O)cc(N)c(F)c(O)c1F 74586,Cc1cc(CC(=O)NC2(CNC(c3nocc3C)=O)CCC2)cc(F)c1 74587,C1(C(=O)OCC)(CC)CCN(CC(=O)NC(C)CNC(C2CCOC2)=O)CC1 74588,c1(C(=O)NCCOCCNC(=O)C(O)c2cnc[nH]2)cc(Br)ccn1 74589,N1(C(C=CCN(C(=O)C(c2ccccc2)F)C)=O)CC2CCC(C1)C(=O)O2 74590,c1(OC)ccc(O)cc1CNC(=O)CCn1cc(CN(C)CCO)nn1 74591,C1(O)(CNCC(COc2ccc(CCOCC)cc2)O)CCCCCC1 74592,C1(C(=O)NCC(N(OCC)C)=O)CCCCCC1NC(C1CC2(CC2)C1)=O 74593,N1(C(c2c(C)scn2)=O)CCCC(C2CCCCN2C(c2sccc2Cl)=O)C1 74594,N1(C(C2(OC)CC2)=O)CC2CCN(C(c3cc(C(C)=O)c(C)o3)=O)C2C1 74595,CCCC(C(O)C(=O)NOC1CCCN(CC)C1)NC(=O)C(C)(C)C1CC1 74596,C(=O)(CC(c1ccccc1)N(C(c1ccc[nH]1)=O)C1CC1)NC(c1cccs1)C 74597,C1(CC#C)(C(=O)NC2CCN(C(=O)C=CC3CC3)C2)CCCCO1 74598,N1(C(c2cccc(CCC)c2)=O)CCC2(N(C(C3CCC3)=O)CC)CC2C1 74599,c1(C(=O)NC(C)C)ccc(CNC(C2CN(C(c3cccc(Br)c3)C)C2)=O)cc1 74600,c1(C(=O)NC(CNC(c2n(CCC)ncc2)=O)CO)ccc(C(C)C)nc1 74601,C1(CCNC(Cn2nc(C)c(Cl)c2)=O)CN(C(=O)CC(C)F)CCCO1 74602,c1(C(=O)NCC2(O)CCN(C(CC(CC)OC)=O)C2)cccc2nsnc12 74603,Cc1noc(C(=O)O)c1Br.c12sccc1NC(=O)CC1(C)CN(C1)C2 74604,CN1CC(C(=O)NCC2(NC(=O)C(CN(C)C)N(C)C)CCCCC2)CC1=O 74605,C(=O)(C(CCC1CC1)NC(=O)C(Cl)Cl)NCc1n(C)ncc1 74606,N1(c2ncc(C(=O)OC)nc2)CC2(CN(C(=O)C(F)C3CCOC3)CC2CO)C1 74607,N1(C(C2N(C)CCC2)=O)CCC(O)C2(CCN(C(c3c(I)cnn3C)=O)CC2)C1 74608,CC1=C(C)CC(CNC(C2C3(CC(NC(=O)CC4(C)CCCCC4)C3)C2)=O)CC1 74609,C12(NC(CCCn3c(C)ncc3)=O)CCCC1N(Cc1ccccc1)CC2 74610,C1(CNC(Cc2cncc(C)c2)=O)CCCCN(C(c2cccnc2O)=O)C1 74611,c1(C(=O)NC2(CCC(N3CCN(C(=O)OC)CC3)=O)CCC2)c[nH]c(C#N)c1C 74612,Cc1ccnc(C(=O)NCC2CCN2C(C2CCCN2Cc2ccccc2)=O)c1 74613,c1(OC)cc(Cl)c(Br)cc1C(C(=O)NCCCF)N(CCC#N)CCOC 74614,C1(CC(=O)NCCN2CCN(C(C3CCC(O)CC3)=O)CC2)CC2CCC(C1)C2 74615,CC1OCCCC1C(=O)NCC(C)(C)NC(=O)CCC1CC1(Cl)Cl 74616,C12(C(=O)OC)CC(C(=O)NCCC(O)CNC(=O)CN(C)C3CC3)(C1)C2 74617,N1(C(C2CCN(C(CNC(=O)OCC)=O)C2)=O)CCSCC1C 74618,C(=O)(C(C)(C)C(F)(F)F)NCC1C(CC)CN(C(=O)CN2CCC(F)CC2)CC1 74619,C1(NC(N2CCC(c3ccccc3)(OC)C2)=O)Cc2ccccc2OC1C 74620,C1(O)(CNC(CC2CN(C)C2)=O)CCCN(C(C2CCCSC2)=O)CC1 74621,c1(C(C(N2C(c3cn(CCCCCC)nn3)CC2)=O)O)ccccc1OC 74622,N1(Cc2ccc(CCC(=O)OCC)cc2)CCC2(CC1)CS(=O)(=O)CCO2 74623,c1(C(=O)NCC(CC=C)NC(C2CC2C(C)C)=O)cc(N)cc(O)c1 74624,c1(CCC)cc(NC(C2CC(N(C)C(C3CCCN3C(C)=O)=O)C2)=O)n(C)n1 74625,N1(C(C2C(C)CCOC2)=O)CCN(C(c2ccnn2CCF)=O)CC1C1CCC1 74626,c1(-c2n(C(CC)C)nc(COc3ccc(OC)cc3)n2)nccn2nc(C)cc12 74627,CCCCC(CC(=O)NCC1(CO)CC2CC2C1)NC(c1ccc(C)nc1O)=O 74628,C(=O)(CC(O)C(=O)NC1CC1NC(c1ccc(C2(C)CC2)cc1)=O)OC(C)(C)C 74629,c1(C(=O)NC2CCC(N(C(c3c(COC)nn[nH]3)=O)C)C2)nccc(Cl)c1O 74630,c1(CC(N2CC(CC=C)(NC(C3CC3C)=O)C2)=O)cnn(C)c1C 74631,N1(CC(C)Oc2cccc(F)c2)CCC(=O)N(CC2CCC3(C2)OCCO3)C1=O 74632,C1(CNC(=O)CCC2CCOC2)CCCC(NC(=O)CC2COC(=O)C2)C1 74633,C1(C(N(C2CCN(C(CC(C(=C)C)O)=O)CC2)CCO)=O)Cc2ccccc2O1 74634,c1(C(C)(C)NC(=O)CCOCC2CCCO2)cn(Cc2ccoc2C(=O)O)nn1 74635,Cc1cc(Br)cc(C)c1CC(=O)NC1(CCNC(C2CC2(F)F)=O)CC1 74636,CC1CCC(CNC(c2cc(O)ncn2)=O)N(C(=O)COCP(C)(C)=O)C1 74637,C12(NC(C3C(COC)C3)=O)CC(C1)N(C(c1ccccc1OC)=O)C2 74638,c1(NC(=O)OC)cc(CNCC(C2CCC(F)(F)CC2)O)ccc1F 74639,N1(CCCCN2CC(C)OC(C)C2)C(=O)C2COC3(CCC3)CN2C1=O 74640,C=C=CCCNC(=O)C(C1CCOC1)NC(=O)CNC(=O)C1CC1 74641,c12nccc(c1C)N2.C(C1C(=O)N1)OC.C(C)(C)(C)OC(=O)C1CC1 74642,c1(C(=O)NCCN(C(=O)C(F)(F)Cl)CCC=C)cnn(CCO)c1 74643,C1(NC(c2ccc(C(N)=O)[nH]2)=O)(NC(C2(C(N)=O)CN(CC)C2)=O)CCCC1C 74644,c1(C(N2CC(C)N(C3CCN(C)CC3)CC2)=O)cc2c(Cl)ccnc2s1 74645,C1(NC(CC(C=C)C)=O)CC2(CCN(C(=O)Cn3nc(C)oc3=O)C2)C1 74646,c1(C(=O)NC2C(OC)CN(C(CCCOCCC)=O)C2)cnn2ccn(C)c12 74647,CCCCCC(O)C(=O)N1CCC(C)CC1C(N1CCC1C(=O)NCC)=O 74648,N1(C(CC(=O)NCC)=O)CCOCCC1C(=O)NCC1CC(C(N)=O)=NO1 74649,C1(O)(C(c2n(C(C)(C)C)nnn2)NC2CN(c3ccccc3)C2)CCCCCC1 74650,N1(C(c2c(C)snn2)=O)CC2CCC1C(NC(c1n[nH]cc1[N+](=O)[O-])=O)C2 74651,C(CC(C(=O)NC1(C(=O)NCC(O)COC)CCCC1)OC)OC 74652,N1(C(C(COC)N(C)C)=O)CCOCCC1C(=O)NCC1CC2(CCCO2)C1 74653,CC1(C(N2CCC(O)(CNC(C3CC(F)(CF)C3)=O)C2)=O)CCC2CC2C1 74654,C(C(N=[N+]=[N-])C(=O)NCCCC(C)NC(=O)CCc1ccsc1)OCC 74655,C1(NC(C(C(C)C)OC)=O)CC2CCC1CN(C(C1(O)CCCCCC1)=O)C2 74656,C(=O)(C(C)(C)C1CCCN1C(=O)CCN(C)C)NC1(C(C)C)CC1 74657,Cc1nsc(N)c1-c1cn(CC(=O)NC(C2(O)CCC2)C2CC2)nn1 74658,C1(CNC(CNC=O)=O)CC2(CN1C(=O)C=CC1CCCCC1)CC2(F)F 74659,C1(NC(c2c(CC)nco2)=O)CCCCC1CNC(=O)C(O)CC1CCCC1 74660,C1(C2CCN(C(=O)C(F)(F)F)C2)(OC(C2CCN(CC(=O)NCC)C2)=O)CC1 74661,Cc1cc(C(N2CCCC(CNC(=O)CCN3CCC(F)C3)CC2)=O)cnc1O 74662,CC(C)C(C(=O)NC1COCC1NC(C1CC(O)(C(F)(F)F)C1)=O)C(C)C 74663,C(C(O)CC(=O)N1CC(N(C)CCO)C1)NC(CSCC=C)=O 74664,C(=O)(C1=CC2CCCCCC12)NCC1CC(NC(C2OCCN(C)C2)=O)C1 74665,Cc1noc(Cl)c1CC(=O)NC1CCC(CNC(C2(C)CCOCC2)=O)C1 74666,c1(OC)cc(-c2nnc(C(C)OC3CCCCO3)n2C)cc(OC)c1OC 74667,c1(-c2onc(-c3cncc(CCc4cccc(Cl)c4)c3)n2)csc2ccccc12 74668,C=C(Cl)C(C)(C)C(=O)NC(CNC(=O)C(c1ccc(Cl)cc1)(C)O)C1CC1 74669,n1(CCCC(=O)NCC2CCN2C(C2CCCCCC2)=O)ccccc1=O 74670,CC#CCCC(=O)NCCC1CC(CNC(=O)C(CCSC)NC(=O)CCC)C1 74671,N1(C(c2c(C)cc(C)o2)=O)CCC(NC(=O)C=CI)C(C)(C)C1 74672,N1(C(C(C)C)=O)CCC2CN(C(C3CCN(c4ccccc4F)C3)=O)CC2C1 74673,CC(=O)CCCC(=O)N1CCCC(NC(=O)C(C)CC2CCCC2)C1 74674,c1(N2CC(c3ccccc3)=C(C)C2)nc(C)c2ncn(-c3cccc(F)c3)c2n1 74675,C(=O)(C#CC1CCOC1)NC(CCCC)CNC(=O)CC1(NC(C)=O)CC1 74676,c1(C(N2CC(CC=C)(NC(C3CCC(F)C3)=O)C2)=O)c(Cl)cnn1C 74677,C(=O)(C1=CS(=O)CCC1)N(C1CCCN(C(CCn2ncc(C)c2)=O)C1)CCO 74678,CC1CCN(C(c2c[nH]c(=N)o2)=O)CC1NC(=O)CC1CC(=O)NC1=O 74679,n1(CC(=O)NC2(CO)CCN(C(=O)C(c3ccc(F)cc3)F)C2)ccccc1=O 74680,C(=O)(CCCCCF)NCC(C1CC1)NC(=O)CSCc1ccccc1Cl 74681,Cc1cc(C(=O)NCC2C3CC2N(C(c2cccc(Cl)c2)=O)C3)cc(=O)n1C 74682,CCC1CNC1=O.c1(-c2cn(CCCOC)nn2)cc[nH]c1C(=O)O 74683,c1(C(=O)NC(C2CCCO2)CC)cncc(CNC(=O)C(C)c2ccco2)c1 74684,C1(NC(CC2(CC)CCCC2)=O)CCCN(C(=O)Cc2ccc(Cl)cc2C)C1C 74685,Cc1cc(C)c([N+](=O)[O-])c(C)c1CN1CCN(CCC2COC2)CC1 74686,N1(C(c2nc(C(C)OC)sc2)=O)CCC(CCNC(=O)CCC2CC2C)CC1 74687,N1(C(c2ccc(=NC)[nH]c2)=O)CCCC2CCCC(O)C12 74688,C(CC(C)C)(C(=O)N(C(C)CN(C)C(c1ccncc1C)=O)C)OC 74689,CC(C)(C)CS(=O)(=O)NCCC1(O)CC2CCC1C2 74690,C1(CCOC)(NC(c2cn(CCCC)nn2)=O)CCN(C(C2CC(=O)CO2)=O)C1 74691,N1(C(c2c(CC)noc2)=O)CCn2ncc(CN(C)C(C3OCC3(C)C)=O)c2C1 74692,Cc1cccc2c1CCN(c1ccc(CNc3ccccc3)nn1)C2 74693,c1(C(=O)NC(C2(O)CN(C(C=CCC)=O)C2)C)cccc(OC2CCCC2)c1 74694,c1(C(=O)NC2C=CCN(C(=O)CC34COC(CF)(C3)C4)C2)cnc(F)c(F)c1 74695,C(c1ccccc1Br)=CC(=O)NCC1(C)CCC(NC(c2ccc[nH]2)=O)C1 74696,Cc1ccc(C=CC(=O)NCC2(NC(C3CCN(C)C3)=O)CCC2)nc1 74697,N1(C(C=CCC)=O)CC(C)(C)C(NC(c2cc(CO)[nH]n2)=O)C(C)(C)C1 74698,c1(C(N2C(CN(C(=O)C(C)O)CC)CCCC2)=O)ccc(C)c(F)c1N 74699,Cc1cc(C(N2CCC(C)(NC(c3cc(O)nc(O)c3)=O)C2)=O)c(Cl)cc1F 74700,CCCCC(O)C(C)C(=O)NC(C(=O)NC1CC(C)N(C)CC1C)C1CCC1 74701,N1(C(CC2(COC)CC2)=O)CCC(C(=O)N(C2CCC2(C)C)C)CC1 74702,c1(OC)cc(C(C)NC2CCCN(c3ccncn3)C2)ccc1OCCO 74703,c1(C(=O)NC2(CCC(=O)NC3C(C)CCC3)CCCC2)cc2ccccc2[nH]1 74704,c1(OCC)ccc(C=CC(N2CC(CNC(C3(F)CC3)=O)CC2C)=O)cc1OC 74705,c1(CC(=O)NC(CNC(c2c(C)ncs2)=O)C)cccc(Cl)c1F 74706,C1(CC(C)NC(C2CCCN2C)=O)CCN(C(C2C3COCC23)=O)CC1 74707,C(=O)(C(C)C(C)CC)N(CC(=O)NC1(CO)CCC(C)C1)CC#C 74708,N1(C(c2cnsc2)=O)CCN(C(C2CC(=C(F)F)C2)=O)CC1c1ccccc1 74709,C1(CC(C)NC(c2c[nH]nc2F)=O)CCN(C(c2ncoc2C(C)(C)C)=O)CC1 74710,c1(C(N2CCC(N(C(CC(CC)SC)=O)CCO)C2)=O)ccc(C)nc1C(C)C 74711,N1(C(c2c(C)nc(O)[nH]2)=O)CC2CCC1CC2NC(C1CCCO1)=O 74712,S(=O)(=O)(c1ccc(Cl)c(Cl)c1)NCC(=O)NCC(N)C(F)(F)F 74713,C1(NC(C(C)(C)OC)=O)CCCN(C(c2sc(-c3ccsc3)nc2C)=O)CC1F 74714,C(CN=c1nc(O)c(C)c[nH]1)c1ccc(CNC(c2c(C)ccs2)=O)cc1 74715,N1(C(C2CCC(C)(O)CC2)=O)CCC2CN(C(=O)CC3CCC(=O)NC3)CC2C1 74716,N1(C(CCC(C)=O)=O)CCN(Cc2cc(Cl)ccc2Br)CC1C(F)(F)F 74717,N1(C(C2(c3cc(C)no3)CC2)=O)CC2CC(NC(=O)CN(C3CCC3)C)CC2C1 74718,Cn1c(C(=O)NC2CCC(CCNC(c3c[nH]c(=N)s3)=O)C2)cc(Cl)c1Cl 74719,N1(C(C2CC(C)OCC2)=O)CCCC2(C1)CN(C(=O)Cc1cncn1C)CCO2 74720,c1(NC(c2ccc(C)cc2C)c2n(CC)nnn2)ccc(OCCOC)cc1O 74721,CN1CCCCC(C(N2CCOC(CNC(C34CCC(C3)C4)=O)CC2)=O)C1=O 74722,C(=O)(CCN(OC)C(=O)c1cnnc(C)c1C)NCC(CC)(C)C 74723,c1(CC)cnc(O)c(C(N2CC(NC(=O)CCc3ncco3)CC(C)C2)=O)c1 74724,c1(C(=O)NCC2(C)N(C(C(=Cc3cn[nH]c3)C)=O)CCC2)cncc2n[nH]cc12 74725,O=S(=O)(c1cc(F)cc(F)c1)NCCNc1nc2c(s1)CCCCCC2 74726,c1(C(=O)NC(CCNC(C(CC=CCC)C)=O)(C)C)ccc(=O)n(CCOC)c1 74727,c1(-n2cc(CN3Cc4c(nc(C)s4)C3)nn2)ccc2c(c1)NCCC2 74728,Cc1ccc(C(N2CC(O)(CNC(c3ccsc3Cl)=O)C2)=O)c(N)n1 74729,N1(CC)CCN(C(=O)C(C(C)C)NC(=O)C(CSC)OC)CC1 74730,C1(N)CN(C(=O)CNC(N2CCOC(C(=O)NCC)C2)=O)CCC12CCC2.OC 74731,C=C(Cl)C(C)(C)C(=O)NC(CNC(=O)CSc1ccc(C)cc1)C(C)C(C)C 74732,C12(CNC(CC(C=C)C)=O)CC(CC)(CN1C(=O)C(CCSC)NC=O)C2 74733,c1(C(=O)NCC(C2CCCC2)NC(c2ccoc2Cl)=O)ccc2oc(O)nc2c1 74734,C1(CC(=O)N(CCC(c2cccs2)NC(CCNC(C)=O)=O)C)CCOCC1 74735,c1(C(=O)OC)nc(C(N2CCCC2C(C)(C)NC(=O)C(C)(C)C)=O)cs1 74736,CC1CC(NC(c2cncn2-c2ccccc2)=O)CN1C(=O)C=CC1CCCC1 74737,N1(C(C)=O)CS(=O)(=O)CC1C(=O)NCC(C)(C)CN(C(=O)CCCCC1CC1)C 74738,C(=O)(C1OCCn2ccnc21)NC(C)CCCNC(c1csnn1)=O 74739,c1(C(=O)NCCCOCCCNC(C(CC)(C)C)=O)cn2c(n1)C(C)CCC2 74740,C1(C2CN(C(c3ccc(C(F)F)s3)=O)C2)(NC(=O)COC2CCCCCC2)CC1 74741,C(=O)(CCCC(F)(F)CO)NC1CCCN(c2cn(C)nc2)C1 74742,c1(C(=O)NCC2(O)CC(NC(COCCOC)=O)C2)c(C(F)(F)F)cccc1F 74743,C1(O)(CCNC(C2C(=C)C2)=O)CCCN(C(=O)Cc2csc(S)n2)C1 74744,N(C1CCCn2nccc21)C(CC1N(C(CCC(CC)C)=O)CC2(CC2)C1)=O 74745,Cc1ccnc(O)c1C(N1CC2C(C(=O)N(C(C)C(C)C)C3CC3)C2C1)=O 74746,c1(NCC2(NC(c3n(C)ccn3)=O)CCCC2)cc2cc(F)ccc2s1 74747,c1(C(=O)NCC23N(c4nccc(OCC)n4)CC(C2)C3)nc(O)nc(O)c1OC 74748,N(C1CCc2c(Br)ccc(Cl)c21)C(C1C(C)(C)S(=O)(=O)C1)=O 74749,c1(OC)ccc2cc(C(=O)NC(C3CN(C(c4oncc4C)=O)C3)C)ncc2c1 74750,c1(CNC(CC(COC)NC(c2n[nH]cc2C)=O)=O)c(C)cccc1C 74751,CC(N=c1[nH]c2c(c(=NC3CC(C4CC4)C3)[nH]1)COC2)C1CCC1 74752,c1(C(N2CCN(C(COCCOC)=O)CC2CCO)=O)cn2nc(C)sc2n1 74753,c1(CCNC(=O)NC2CCOC2c2ccccc2)cccc2cccnc12 74754,C1(CNC(C(C)(C)n2cnnn2)=O)COCC2(CCN(C(C3COC3)=O)CC2)O1 74755,C(=O)(C1=CC(C)(C)C1)N1CCC(NC(c2cn(CCC)nc2)=O)(COC)C1 74756,c1(NCCCSC)ccc(S(=O)(=O)NCC2(CCN=[N+]=[N-])CC2)c(Br)c1 74757,C1(C(=O)NCc2ccc(OCC=C)cc2)(NC)CCOC(C)(C)C1 74758,CC1Cn2nccc2CN1C(=O)C1=CCCN(C(=O)COCCCF)C1 74759,N1(C(C(C)OCC=C)=O)CC(O)CC1CNC(=O)C1=COCC1 74760,c1(CC(N2C(CNC(C3C(C(C)C)C3)=O)CC2)=O)cnc2ccccc2c1 74761,C1(N(C(c2c(C)nn[nH]2)=O)C)CCCN(C(C2(Cc3cnn[nH]3)CCC2)=O)CC1 74762,Cc1cc(NC(C2CCN(C(=O)OC(C)(C)C)C2C)=O)c(C)n1CC1CC1 74763,C(=O)(C(C)C(O)C(C)C)NCC(CNC(C1(COC)COC1)=O)S(C)(=O)=O 74764,c1(SCC)cccc2[nH]c(C(N3CC4CCCC3C4NC(=O)C=NOC)=O)cc12 74765,C1(F)(CC)CN(C(=O)CC2CCN(Cc3ccc(OC)c(Cl)c3)C2)CC1C1CC1 74766,c1(C(=O)NCC2CCCN(C(C(C(C)C)C)=O)C2)c(F)ccc(Br)c1F 74767,CC1CCN(C(=O)CCSc2ccccc2)C1CNC(=O)CCCc1cncs1 74768,CC1C(NC(=O)CC2(C)CCCO2)CCN1C(c1cccc(Cl)n1)=O 74769,CC(Cc1cnc[nH]1)C(=O)N(CCNC(C1CCOC1C(N)=O)=O)C1CC1 74770,C1(NC(c2c(CC)cns2)=O)CC(O)CN(C(c2cnccc2Cl)=O)C1 74771,c1(N(C)Cc2ccc(-c3c(OCC)cccn3)s2)ccc(S(=N)(=O)CC)cc1 74772,C(C1=NOC2CN(C(=O)Cc3cnc[nH]3)CC12)NC(C1CC2(C(OC)CC2)C1)=O 74773,C1(C(C(=O)OC)C)C(N(C2CC3(CC3)C2)C(C)=O)CCCN1Cc1ccccc1 74774,C1(CC)CC(C(=O)NC(CO)C2CC2)CCN1C(=O)CCc1cscn1 74775,CC(C)CC(CNC(C1(NC(=O)C(c2ccnn2C)C)CCOCC1)=O)CO 74776,c1(NC2C(NC(c3cccc(Br)n3)=O)CCC2)ncnc2occc12 74777,N1(C(c2c(Cl)ccc(NC)c2)=O)CCC2CCCC(C1)N2C(=O)C(C)SC 74778,C1(C(=O)NC2CCN(Cc3onc(CCCCC)n3)C2)CCc2nncn2CC1 74779,c1(C(N2CCC(N(C(=O)CC#N)C)C2)=O)ccc(=O)n(-c2ccccc2)c1 74780,N1(C(c2cc(C(C)C)nn2C)=O)CCC(NC(=O)C(=C2CCCCC2)F)C12CC2 74781,N1(C(C(=O)NCCCCCC)CC2CC2)CCCN(Cc2ccsc2)CC1 74782,n1(CCC)c(C(=O)Nc2ccncc2SC(C)C)cc2ccccc12 74783,C1(CNC(c2c(C(C)C)nco2)=O)CCCCN(C(=O)CCC2CC(F)(F)C2)C1 74784,C(N=c1nc(C)c(Br)c[nH]1)C1(O)CN(C(CSc2nc(C)cc(C)n2)=O)C1 74785,C1(C(N(CCC#C)CCOC)=O)C=CCN(C(c2ccc(C(N)=O)[nH]2)=O)C1 74786,C1(OCC)CC2(C1)CC2C(=O)NCC1CCN(c2nnc(C(C)(C)CC)o2)CC1 74787,C1(Cc2n(-c3n(C)ccn3)nc(C(F)F)n2)CCc2ncsc2C1 74788,C1(CNC(C2(COC)CCC2)=O)CCCCCN1C(c1ccc(O)nn1)=O 74789,N1(C(c2ccc(SC)s2)=O)Cc2ccc(-c3ccc(O)cc3C)cc2C1 74790,C1(CCOC)(NC(COCCC=C)=O)CCN(C(c2snnc2CC)=O)C1 74791,C1(CNC(CCCc2ccc(C)cc2)=O)C(C2CC2)CCN1C(c1cnco1)=O 74792,C(=O)(C(CC)CC(F)F)N1CCN(C(C2C(CC)CCC2)=O)CC1CC12CC(C1)C2 74793,C(=O)(CCCN=c1nc(N(C)C)cc(C)[nH]1)NC1CC(NC)C1(C)C 74794,N1(S(c2ccc(N(CC(C)O)C)nc2)(=O)=O)CC2(CCOCC2)CC1C 74795,c1(SC)ccccc1CC(N1CC(NC(=O)C(F)(F)CN(C)C)C1)=O 74796,Cc1cc(C(=O)NCc2ncoc2CCNC(C2CCC(=O)C2)=O)c(Cl)cc1F 74797,CC1Oc2ccccc2C1NC(=O)C(=O)NCCOCC(F)F 74798,CC(C)CC(F)C(=O)NC1(C)CN(C(C23CC4CC2C3C4)=O)C1 74799,c1(C(N2CC=CC(NC(C=C(C)Cl)=O)C2)=O)cc(F)cc2nccnc12 74800,C1(C(=O)NC2CN(C(C(CC(C)C)=O)=O)C(C)CC2)CCOC2(CCC2)C1 74801,Cn1ccc2cc(C(=O)NC3CC(NC(=O)CSC4CC4)CC3O)ccc12 74802,c1(C(=O)NCCN(C(CC2CCC(C)O2)=O)C)cccc2[nH]ncc12 74803,C1(CCC)(NC(=O)C(CCC2CCC2)NC(=O)C(CCOC)OC)CCNC1=O 74804,C1(NC(c2c(C)c(N)ccc2)=O)CC2CC1CN(C(C1CC1C(N)=O)=O)C2 74805,c1(C(=O)NCC(CN(C(C2(CC)CCCCO2)=O)C)C)ccc2c(c1)ncn2C 74806,C1(OC)CCN(C(C2CCN(C(=O)CCc3cc(C)on3)C2)=O)C1C 74807,C1(C(N2CC(CCNC(=O)Cc3ccc(C(F)F)cc3)C2)=O)CC2(C1)CC(F)C2 74808,Cc1ccc(C(N2CC3C(N(C(=O)Cn4cnnn4)C)C3C2)=O)cc1S(C)(=O)=O 74809,C(CCCC(C)NC(=O)CC1(CO)CC1)NC(c1c(C(=O)OCC)con1)=O 74810,c1(OC)c(C(N2CC(NC(c3cc(C)c(C)[nH]3)=O)C(C)(C)C2)=O)cc(Cl)cc1Cl 74811,C1(C(C)C)OCCC1CNC(=O)C(CO)NC(=O)CC(C)n1cccn1 74812,C(=O)(CCN(OC)C(=O)C1CN(C)CCO1)NC(CC)C(N)=O 74813,c1(OC)ccc(CC(=O)NCCC(C)NC(c2cnc(C(C)(C)C)s2)=O)cc1 74814,C(=O)(CC(CC)CC)OC(CCC)CN1C2CCC1COC2 74815,C1(NC(C2N(C(C)=O)CCC2)=O)C=CCN(C(=O)CSc2cnn(C)c2)C1 74816,C1(NC(CC(COC)C)=O)CN(C(c2conc2C(C)C)=O)Cc2ccnn2C1 74817,C1(NC(CC=C)=O)C2CCN(C(=O)C(c3ccc(F)cc3)(F)F)CCC12 74818,C1(CC(=O)N(CCNC(=O)CC(O)c2ccccc2)CC)OCCC1(C)C 74819,C1(N(CCOC)C(c2ccoc2C2CC2)=O)CCN(C(=O)CC2CCC2)CC1 74820,c1(C(C)C)ncncc1C(=O)NC1CN(C(=O)C(O)CN(C)C)CC1C 74821,N1(C(C(c2ccn(C)c2)C)=O)CCC(C(=O)NC2CC23CCCCC3)C(O)C1 74822,CN1CCn2ncc(C(N3CC4(C3)CN(C(c3nnn(C)c3N)=O)C4)=O)c2C1 74823,C1(C(=O)NCCOCC(=O)OC)CC(NC(=O)CCc2cnco2)C1(C)C 74824,N1(C(C(F)=CCC)=O)CCC(C)C1CNC(=O)C(C)Oc1ccccc1F 74825,c1(N2CCC(N(C)C(C3CCc4nnnn4CC3)=O)C2)c(Cl)cncc1[N+](=O)[O-] 74826,Cc1ccnc2c(C(N3CC(OCCNC(=O)CCCCCF)C3)=O)cccc12 74827,CC1=C(CNC(c2ccc(C(C)(C)C)cc2O)=O)SCCO1 74828,N1(C(=O)NC2CC(F)C2)CCCC1c1ccc(Br)s1 74829,c1(N(C2CC3CC2CN3)C(c2cc(C)nn2C)=O)ccc2ncnn2c1 74830,C1(NC(c2ccc(C(F)(F)F)nc2)=O)CCN(C(C2CCCOCC2)=O)CC1F 74831,N1(C(Cc2c(C)ccs2)=O)CCC2(CCCCN(C(=O)C(O)CC(N)=O)C2)C1 74832,N1(C(CNC(=O)OC)=O)CCCC(CO)(NC(c2ccc(N)nc2F)=O)C1 74833,CC(Cc1cnco1)C(=O)N(CCNC(=O)C(F)C1CCC1)CC1CC1 74834,C1(C(C)C)CN(C(c2n[nH]cc2-c2ccc(OC(F)(F)F)cc2)=O)CCO1 74835,c1(C(C)C)ccccc1C(=O)NC1CCCC1NC(=O)CCC1CC(C)OC1C 74836,c1(C(=O)NC2C(CNC(C3(Cl)C(C(C)=O)C3)=O)CCC2)ccc(C)nn1 74837,N1(C(c2c(Cl)cn(CCC)n2)=O)CCC(NC(=O)C2=CC(O)CCC2)C(C)(C)C1 74838,N1(C(C(C)N2CCC2)=O)CC2(CCCC2NC(=O)CC2CCC3CC23)C1 74839,N1(C(C=CCC)=O)CCN(C(c2ccccc2-c2nc(C)no2)=O)C(CC)C1 74840,c1(C(=O)NC(C2CCN(C(=O)CC3NC(=O)NC3=O)C2)C)cc(Cl)nc(=N)[nH]1 74841,C(CC1(C)CC1)(C(=O)NCC1CCC1)N(C(C)C)C1CC1 74842,C1(NC(c2c(C)ccc(C)n2)=O)CC2CC(C1)N(C(c1ccc(=O)oc1)=O)C2 74843,C1(CC(=O)NCc2c(C)ccs2)CN(C(C23CC(C)(CCO2)C3)=O)CCC1C 74844,c1(C(N2CC3C(NC(c4ccc(C(C)=O)o4)=O)(CC3)C2)=O)cc2n(n1)CCCC2 74845,c1(CCNCC(C2CCCOC2)OC)cn(C)c2cc(Cl)ccc12 74846,N1(C(C(CCC)NC(=O)CCN(CC)CC)=O)CC2CC1C1CC21 74847,CCCC(CNC(=O)CC1CCCOC1)NC(c1ccoc1CC)=O 74848,C1(CNC(C(F)OC)=O)CN(C(c2cnn(C3CCCC3)c2)=O)CCC12CCC2 74849,CON(C)CCNC(=O)C(C1CCN(C(=O)CN2CSCC2=O)C1)C 74850,N1(C(C2CN(C(C)=O)C2)=O)CCC(CNC(=O)C(C2CCCCC2)O)C(C)C1 74851,C12(C(=O)NCCNC(CC)=O)CCC(CC1NC(=O)C(C(C)C)NC(C)=O)C2 74852,C(=O)(C(C)(C)C(C)NC(=O)C(C)=C1CCC1)N1CCC(N(C(C=CC)=O)CC)C1 74853,c1(C(=O)NC2CC3CC(NC(C(CCCOC)C)=O)CC32)cccc(F)c1C#N 74854,Cn1cc2c(n1)CCC(COC(C1CCCC(CC(F)(F)F)C1)=O)C2 74855,CN1CCOC(C(=O)NC2CN(C(=O)Cc3coc(-c4cccs4)n3)C2)C1 74856,C(=O)(C1OCCn2ccnc21)NCCC(C)NC(c1cn(CCC2CC2)nn1)=O 74857,N1(C(CCC(=C)Cl)=O)CCC2(C1)CN(C(C1CCCC(C)O1)=O)CCO2 74858,c1(OC)cc(-c2cnc(OC)c(C(=O)NCC(F)F)c2)cc(F)c1F 74859,N1(Cc2ncc(OC)nc2)CCN(C(=O)C=Cc2ccc([N+](=O)[O-])o2)C2(CC2)C1 74860,N1(C(C(C)NC=O)=O)CC(C(N2CCC3(CCSC3)C2)=O)CCC1(C)C 74861,C(=O)(C(O)CC(C)(C)C)N1CC(C)C(CNC(=O)CCN2CCC(O)CC2)CC1 74862,c1(C(=O)NCCC(=O)NC2CCC(NC(=O)CCCSC)C2)ccc(F)cc1.C=O 74863,C1(CC(NOC(C)C)=O)CN(C(c2csc(F)c2)=O)C(C)(C)C1 74864,C1(OC)CC2(C1)CC(C(N1CC(NC(=O)C=CC3CC3)C(F)C1)=O)C2 74865,C(=O)(CC1=CCCCC1)NC1(COC)CN(C(C2CC(C)CC(C)C2)=O)C1 74866,Cc1ocnc1CC(=O)NCC(c1ccccc1)CNC(C1CC(C)(C)C1)=O 74867,CC(C)(F)C(=O)N1CCCC1C1(O)CN(C(=O)CSCC2CCCCO2)C1 74868,c1(OC)cccc(C(N2CCC(C)C(NC(=O)C(F)C(F)(F)F)C2)=O)c1F 74869,C1(NC(c2n[nH]c(C)c2C)=O)CCCC12CN(C(=O)C#CC(C)(C)O)C2 74870,CN1C2CCC1CC(=CC(N1CCC(NC(=O)C(N)=O)C(CO)CC1)=O)C2 74871,Cc1cc(CCC(=O)NCCC(C)NC(c2cccc(CS(C)=O)c2)=O)c(C)o1 74872,CC1CCC(CNC(c2cc(Cl)c(Cl)s2)=O)N(C(c2cnn(C)n2)=O)C1 74873,N1(C(=O)CC2(CO)CCCC2)CCCC2(CCCN2C(c2nocc2Cl)=O)C1 74874,CC(C)(CC1CCCN(C(=O)NCCC2CNC(=O)C2)C1)C(N)=O 74875,N1(C(c2ccc(SC)s2)=O)C2CCC1CC(N(C(=O)Cn1ccc(C)n1)C)C2 74876,C1(C(=O)NC(C=C)COC)(CNC(C2CCC(C)O2)=O)CC(C)(C)C1 74877,C1(CNC(C(C)SCC)=O)CC2CCC(C1)N2C(=O)CCC1CC1(C)C 74878,N1(C(c2cc(C#C)cc(F)c2)=O)CCC(C2CCN(C(=O)CC3CC3)CC2)CC1 74879,c1(CC(=O)NC23CC(C(N(C(C)(C)C)CCN)=O)(C2)C3)cc(F)cc(Br)c1 74880,c1(CNC(c2cnns2)=O)ccc(CCNC(C2CCO2)=O)cc1 74881,Cc1ccnn1C(C)C(N1CCCC1C1(C(=O)NC2(C(C)C)CC2)CC1)=O 74882,N1(C(COCCC=C)=O)CCC(CCNC(=O)C(C(C)O)N(C)C)CC1 74883,c1(C(=O)NC2CC3CN(C(c4c(OC)ccs4)=O)CC32)csc2c1CCC(C)C2 74884,C1(C(N(C(C)CNC(=O)Cc2nc(C)c(C)o2)CC)=O)CCC2(CCC2)CO1 74885,N1(C(C2N(C(Cc3c(C)ocn3)=O)CC(F)C2)=O)CCC12CCSCC2 74886,CC1(CNC(=O)CC2CCCO2)CCCN(C(=O)CN2CCC(O)CC2)C1 74887,CCC(O)C(F)(F)C(=O)NCC=CCNC(C1CC(=O)N(c2nccs2)C1)=O 74888,C1(C(=O)NCC(COC)NC(c2csc(C)c2C)=O)CCCCC(=O)N1 74889,N1(C(c2n(COC)ncc2)=O)CCC2(CCC2)C(CNC(c2ccon2)=O)C1 74890,N1(C(C(C)(C)OCC)=O)CC2COCC2(C(=O)N(C)CC2(COC)CC2)C1 74891,Cc1noc(C)c1C(=O)N(CC(CO)(CO)NC(c1cnc[nH]1)=O)C 74892,CC(C(=O)OC1CC1)S(=O)(=O)NC(=O)C1=CCNC1 74893,C1(C(=O)Nc2c(C)nn(CCF)c2)CCCCN(C(C2CCC3(CCC3)O2)=O)C1 74894,N1(C(C(C(=O)OCC)F)=O)CCC(CNC(c2cccc(Cl)c2OC)=O)C12CC2 74895,C12CCCC(C1)CNC2=O.c1(NC(C=NOC)=O)ccnc(-c2ccco2)c1 74896,C1(C(=O)NCC2(OC)CCN(C(c3c(C)nsc3C)=O)C2)CC(S(C)(=O)=O)C1 74897,CC1(C)CCN(C(=O)Oc2cccc(CNC(=O)OC(C)(C)C)c2)CC1 74898,C1(CCC)CCCN1C(=O)COc1nncs1 74899,c1(C2(C(=O)NCC3CN3)CC2)ccccc1.C12(CC1)CN2.CC(C)=CCOC 74900,N1(c2ncc(C(=O)OC)cn2)CC2CCC1C(NC(C1CCN(C)C(=O)C1)=O)C2 74901,C1(CNC(C=C(C)Cl)=O)CN(C(=O)C(c2ccc(F)c(Cl)c2)C)CC(C)(C)O1 74902,CC(C(=O)NCC(C1CCCC1)NC(c1nccs1)=O)C1CCCC1 74903,N#Cc1ccnnc1NCC1(NC(C2CCCCO2)=O)COC1 74904,N1(C(CNC(=O)OCC=C)=O)CCCC2C1CCCN2C(=O)CN1CSCC1=O 74905,N1(C(COCc2onc(CC)n2)=O)CCC2CCN(C(=O)CC(C)(F)F)CC12 74906,CCCC(C)(O)CC(=O)NCC1(OC)CCN(C(C2CCN(C(N)=O)CC2)=O)C1 74907,c1(-n2c(Cc3cn(C(C)C)nc3)nc(C3CCCO3)n2)ccc(S(C)(=O)=O)cc1 74908,CC1CCC(NC(=O)CCc2cnccn2)CN1C(c1cc(Cl)cnn1)=O 74909,c1(C(=O)NC2C(NC(c3ccc(CC)o3)=O)CCOC2)ccnc(OC)c1F 74910,C1(C(N2CCC(CCNC(CSCCC(C)C)=O)C2)=O)CC2CCC(C1)C2F 74911,C1(CCC)(NC(c2ccc(F)cc2Cl)=O)CCCN(C(=O)CC2(N(C)C)CC2)C1 74912,N1(C(C(C2CC2)OCC)=O)CCN(C(c2ccc(CC)[nH]2)=O)C(C2CCCC2)C1 74913,c1(CN(CC(COCC)O)C)ccc(C(F)(F)F)c2c1OCCO2 74914,Cc1cc(C)c(C(=O)N(CC(O)CNC(c2ccc(C(C)(C)C)nc2)=O)C)s1 74915,c1(CC(=O)NC2CCC(CNC(CCC=C)=O)CC2)c[nH]c2ncccc12 74916,N1(C(CC(C)N2CCCC2=O)=O)CCN(C(C2C3CC4C(C3=O)C24)=O)CC1CO 74917,Cc1cc(C=CC(N2CCN(C(C3CC(C)(O)C3)=O)CC2)=O)ccc1F 74918,C1(CC)CCC(C)CN1C(c1cc(CNC(C2CC(CC)(CC)C2)=O)ccn1)=O 74919,N1(C(CCN(C(CSC(C)(C)C)=O)CC2CC2)=O)CCN2CCC1CC2 74920,S(=O)(=O)(c1ccc(NC2C3CCCC23)c(F)c1)NC(c1nc2ccccc2s1)C 74921,C12(C(=O)NCCC3N(C(c4ncc(OC)cn4)=O)CCCC3)CCCC1C2(F)F 74922,c1(OCC(=O)NCCCCN(C(C(C)OCC(C)C)=O)C)ccc(F)cn1 74923,N1(C(C(CCSC)NC(=O)CN2CCCCC2C)=O)CCCC(C)C1CO 74924,C=CC(C)(O)CC(=O)N1CCCCC(C(N2CCC(OC3CC3)C2)=O)C1 74925,CC1CCN(CC(=O)N(C2CCCC(N(C(=O)Cc3ccno3)C)C2)C)CC1 74926,c1(C(C(=O)N(C(C)(C)CC)C)N(CC=C)C2CC2)cc(C2CCC2)[nH]n1.C(CO)O 74927,c1(C2(C(=O)NC(CNC(C3(OC)CCSC3)=O)CO)CCC2)ccc(Cl)c(F)c1 74928,C1(C(C)NC(CC=C)=O)CN(C(=O)CCC2CCC(=O)N2)CCO1 74929,C(CCC(C)C(=O)N1CCCCC1CCNC(c1cnn(C(C)C)c1N)=O)OC 74930,N1(C(c2ccc(OCCCC)cc2)=O)CCN(C(C2CCCSC2)=O)C(CF)C1 74931,C1(C)(C(=O)NC2CCC(NC(CCCCCOCC)=O)CC2)CC(C2CC2)=NO1 74932,CC1CN(C(=O)C=Cc2cncs2)CC1n1cc(COCCOCCO)nn1 74933,N1(C(CCCSC)=O)CCN(C)CC1CNC(=O)Cc1ccco1 74934,c1(CC)ccc(C(C)=CC(N2CC(NC(C3CCOCC3)=O)C(O)C2)=O)cc1 74935,C1(CC(=O)N(c2cccnc2)CC2CC2)CCN(C(=O)CC(O)C2CC2)C1 74936,Cc1nnn(CC(=O)NC2CCCC2CNC(c2cc[nH]n2)=O)n1 74937,c1(NCCC2CCCN(NC(=O)OC(C)(C)C)CC2)nc2c(cc1Cl)C(=O)OC2 74938,C1(C(N2CCC(C(C)NC(c3cnn(C4CCC4)c3)=O)C2)=O)CC2CC2CC1C 74939,c1(OC)nc(=NCCN(C)C(c2cccc(F)c2Cl)=O)nc(OC)[nH]1 74940,C1(C(N(C(C)Cc2cccs2)C)=O)CCCC1c1nn[nH]n1 74941,C12(C(N3CCCC(C(=O)NC4CC5CCC4O5)C3)=O)CCC(CC1)CC2 74942,N1(C(c2ccc(C3C(N)C3)cc2)=O)CC2(CO)CCCC2(F)C1 74943,c1(OCC(=O)NCC2(NC(c3c(CC)con3)=O)CCC2)c(Cl)cccc1Cl 74944,C(CS(=O)(=O)c1cc(Cl)ccc1Cl)N(CCC)Cc1cccc(Br)c1 74945,c1(CN)cc(N2CCCC(C=O)C2)nc(C)c1.C1(C(=O)OC(C)C)(COC)CC1 74946,n1(CC)cnc(Cl)c1C(C(=O)NCC1CC(F)(F)C1)N(C)CC1(F)CCC1 74947,c1(NC)ncccc1C(=O)NC(C(=O)NCC12CC(CCO1)C2)C(C)C 74948,C(=O)(C1CCc2ccccc21)N1C2CCC(NC(=O)CCSC(F)(F)F)(CC2)C1 74949,Cc1cc(C)n(Cc2cccc(NC(=O)NCCC(C)Sc3ccccc3)c2)n1 74950,C1(NC(C#CC(C)C)=O)CCN(C(=O)C(C)Oc2cccnc2)C1(C)C 74951,N1(C(C2(NC(N)=O)CCCCC2)=O)CCOCC(NC(=O)C2=CCCC2)C1 74952,N1(C(c2c(CC)c[nH]c2)=O)CC2CCCC2(NC(c2occc2CC)=O)C1 74953,N1(C(c2c(CC)nn(C)c2)=O)CCC2CCN(C(=O)C(C)CS(C)(=O)=O)CC12 74954,C(CN=c1cc(C)nc(S(C)(=O)=O)[nH]1)C1(OC)CN(C(=O)Cn2ccnc2C)C1 74955,C1(C)(CNC(C=CCOC)=O)CN(C(C2C=CCC2)=O)C(C)(C)C1 74956,N1(C(C2C(OC)CCC2)=O)CCC(C(=O)NC(c2ccncn2)C)CC1 74957,c1(C(=O)NC2(CCCNC(c3occ4c3CCC4)=O)CC2)ccc2cncn2c1 74958,N1(C(C=CC)=O)CCN(C(=O)Cc2ccn3cncc3c2)C2CCC12 74959,C1(C)(CC)C=C(C(=O)N2CC(CC(C)NC(C3CC3F)=O)C2)C1 74960,C1(C(F)F)(OC)CCN(C(=O)NC2CCC2C(F)(F)F)CC1 74961,N1(C(c2n(CC)ccn2)=O)CC=C(CCNC(C2(OC)CCSCC2)=O)CC1 74962,c1(NC(C2CC(=O)OC2)=O)cc(-c2cnn(CC(N3CCCC3)=O)c2)ccn1 74963,c1(OCC)cccc(CC(=O)N(C)CC2CC(O)C2)c1 74964,N1(C(C(C)OCC)=O)CC2CCCN(C(=O)CCc3c(C)n[nH]c3C)C2C1 74965,c1(NCC(C=C)OC)cc(=NCC(C(C)(C)C)OC)[nH]c(C)n1 74966,C12(C(=O)NCc3ccco3)CCC(NC(C3CCS(=O)CC3)=O)(CC1)C2 74967,Cc1ccc(C(N2CCN(C(=O)C(C)N(C)C)C(c3ccccc3)C2)=O)c(C)c1 74968,CC(O)C(C(=O)N1CCC(C(C)(C)NC(=O)CN(C)S(N)(=O)=O)C1)N(C)C 74969,c1(N(CCC)C)ccc(NC(=O)CCN2CCOC2=O)cc1 74970,C1(NC(c2cn(CCNC(=O)CCC3CC3(F)F)nc2)=O)CC2(CCOC2)C1 74971,CC1CCC(C)(C)CN1C(C1CN(C(C2C=CC=CC=C2)=O)CCC1(C)C)=O 74972,C#CC1CN(C(C2CN3CCCN2CC3)=O)CCN1C(c1cc2scnc2[nH]1)=O 74973,c1(C(=O)NCC(C)(C)NC(c2cnc(C(C)C)[nH]2)=O)ccc(-c2ncc[nH]2)cc1 74974,N1(C(C2CC(C)(O)C2)=O)CCC(O)C(NC(C2CCN(CC(F)(F)F)CC2)=O)C1 74975,Cn1c(C(N2CC(CNC(C3SCCCS3)=O)C2)=O)cc2ccsc12 74976,C(=O)(CCCCCOC(C)(C)C)OC(c1n[nH]cc1-c1ccncc1)C 74977,C=CC(CCC)CC(=O)NC1CC(NC(=O)C=Cc2ccccc2Br)C(O)C1 74978,c1(C(N2CC3COCC3C2)=O)nc(-c2ccc3nccnc3c2)c2ccccn12 74979,c1(C(C)(C)C)ncc2c(n1)CCN(N(Cc1ccco1)Cc1ccccc1)C2 74980,C12(CNC(C(C)S(N)(=O)=O)=O)CCCC(CN(C(C3(P(C)(C)=O)CC3)=O)C1)C2 74981,C12(C(=O)NCC(C)NC(c3cc4ccccn4c3)=O)CCC(C)(CC1)CO2 74982,Cc1cc(CN(C2CN(C(C3CCCCO3)=O)C2)C)nn1C 74983,c1(NC(=NC)NCCc2ccccc2)ccc(C(c2ccccc2)C)cc1 74984,c1(C(=O)NC(C)CNC(=O)Cc2cnccn2)c(C(F)F)cccc1C(F)F 74985,C1(C(C)NC(=O)C(F)Cc2ccccc2)CN(C(=O)Cc2ccccc2)CCO1 74986,N1(C(COC)=O)CCN(c2ccc(C(F)(F)F)cn2)CC1.N12CCCC1C2=O 74987,CCCC(C)(C)CC(=O)OC(c1nnco1)C 74988,CCC(C(=O)N(CCCOCCNC(c1ccccc1N(C)C)=O)C)C(C)C 74989,C1(NC(c2ccc(F)cn2)=O)CN(S(=O)(=O)C(Cl)(Cl)Cl)CC(F)(F)C1 74990,C#Cc1ccc(C(N2CCC(=CNC(C3CCCN(C(N)=O)C3)=O)CC2)=O)nc1 74991,n1(CCOC)ccc(=NC(=O)C(CC2CCC2)NC(C2CCCN2C(C)C)=O)[nH]1 74992,N1(CCNC(c2nnnn2CCC2CC2)C2(C(=O)OC)CC2)C(=O)CCC1=O 74993,C1(C)(C(=O)NCCCCNC(c2cc(CCC)n(C)n2)=O)CCOC12CC2(F)F 74994,C1(NC(c2c(C)snn2)=O)CCCN(C(=O)C=Cc2ccc(C3OCCO3)o2)C1 74995,O(NC(=O)CCCCCCNC(c1ccc2cccnn12)=O)CC(=C)C 74996,C=CCC(CC)C(=O)NCC(c1ccccc1F)NC(C1(N(C)C)CC1)=O 74997,C1(C(N2CCC(CNC(C(CC)C#N)=O)C2)=O)COC2COCC12 74998,Cc1ccc(C#N)cc1C(=O)NC1CS(=O)(=O)CC1NC(=O)CC(C)(F)F 74999,c1(C(=O)NC2CN(C(C34CC(F)C3C4)=O)CC23CC3)cc(Cl)c2n[nH]cc2c1 75000,c1(OC)cc(C(=O)NCC2CCC(NC(=O)CC3CCC(=O)NC3)C2)ccc1F 75001,Nc1cnc(Cl)c(C(N2CCOCC2CNC(C2CNC(=O)N2)=O)=O)c1 75002,c1(NC(C2CCCN(C(=O)OC)C2)=O)cc(I)ccc1O 75003,C(=O)(CCCS(C)(=O)=O)NC1(CC=C)CCCN(C(c2cc(F)ccc2F)=O)C1 75004,C=CC(CCC)CC(=O)N1CCC2(C1)CN(C(=O)C(C(C)C)NS(C)(=O)=O)C2 75005,C1(CNC(C2(C=C)CC2)=O)CCC(CNC(=O)CSc2nnnn2C2CC2)C1 75006,C=C1Cn2c(C(=O)NC3CCCC3CNC(=O)Cc3cnsc3)nnc2S1 75007,CC(C)C(CO)NC(=O)CC(C1CC1)NC(=O)CC1CCCOC1 75008,CN1CC(CC(=O)NC2(C)CC(NC(C3(O)CCCC3)=O)C2)CCC1C(F)(F)F 75009,C(CCCC(=O)N1CCC(O)(C(C)CNC(C2(n3cccn3)CC2)=O)C1)SC 75010,CCCCC(O)CC(=O)N1CCC(C(=O)Nc2cc(F)ccc2C)(CC)C1 75011,N1(C(C=NOC)=O)CCCC(C(=O)Nc2nc(C3CCCCC3)c(C)s2)C1 75012,N1(c2ccnc(NCc3scc(C(C)C)n3)n2)CC(C)OC2(CCCOC2)C1 75013,c1(CC)ccc(CNC(C2OCCC2CNC(=O)CC(C)(C)C)=O)nc1 75014,C(CC(=O)N(CCC(F)(F)F)C)(C(C)CC)NC(C(CCCC)NC(N)=O)=O 75015,c1(CNC(c2ccc(C(=O)O)cn2)(C)C)ccc(N)c(Br)c1 75016,c1(C(C)(C)C)ccc(C(=O)CN(C(=O)CC2C=CCCC2)C2CC2)o1 75017,CC1(C)CN(C(=O)NC2CCN(C(C3CCCCC3)=O)CC2)C2COCC12 75018,C(=O)(C(O)P(C)(C)=O)NCC1(C)CC(NC(c2cn(CCC)nc2C)=O)C1 75019,C=Cc1ccc(C(=O)NCC(C)CNC(=O)CC2CCN(C)C2)cc1 75020,N1(C(=O)CSC(F)(F)F)CC(C2CCCCN(C(=O)CCC3CCCO3)C2)C1 75021,C1(C(=O)NCCNS(N)(=O)=O)COC2CN(CCC(=O)O)CC12 75022,c1(C(=O)NCCC(C)NC(c2cscc2C(F)(F)F)=O)n[nH]cc1C(C)(C)C 75023,c1(CNC(C(C)CO)=O)n[nH]c2c1CN(C(=O)C(C)NC(c1ccco1)=O)CC2 75024,C(=O)(CCC(C)NC(C1(C)CCCO1)=O)NCCOCCCC 75025,C(C)(CCn1cccn1)(c1nnnn1CCC1(C)CC1)NC(COC)C1CC1 75026,C1(NC(c2cc(Cl)ccn2)=O)C2CCC1CN(C(c1csnn1)=O)C2 75027,C1(C(=O)NC2C(CC)CN(C(c3ncccc3C)=O)CC2)CC2CCCCN2C1 75028,C1(CNC(c2cnc(SC)nc2O)=O)CC2(CO1)CN(C(c1oncc1C)=O)C2 75029,Cc1c(C(=O)NCCC(C(C)C)NC(=O)C(F)C(C)(C)O)sc2ccsc12 75030,C1(CNC(N2CC(OCC)C(NC(=O)OCC)C2)=O)CC2(CCO1)CC(F)(F)C2 75031,N1(c2nnc(C#N)s2)CCC2(CNC(c3cccc4[nH]ncc34)=O)CCCCC12 75032,c1(C(=O)OCC)cc(C(N2CC(C)(NC(c3nccn3C)=O)C2)=O)on1 75033,N1(C(=O)CC(=O)OC)CCC2(CO)CN(C(c3cc(COC)cn3C)=O)CC2C1 75034,C1(NC(Cc2cc(C)[nH]n2)=O)CCC(CC(=O)NC(C(O)CO)C2CC2)CC1 75035,c1(C(=O)NC2C3CN(C(c4ccc(C#C)cn4)=O)C2CC3)cccc2ncnn12 75036,C1(C(=O)NCC2C(NC(c3n(C)cnc3)=O)CCC2)CCC(C(F)(F)F)CC1 75037,Cn1cc(Cl)c(C(=O)NC23CC(CNC(C4CCCNC4=O)=O)(C2)C3)n1 75038,C1(C#C)(C(NOCCCC#C)=O)CCN(C(=O)CC2C(=O)NN=C2C)C1 75039,C12(NC(c3cc(F)c(O)c(Br)c3)=O)COCCC1CN(C(=O)CCF)C2 75040,C12(NC(CCOC)=O)CC(CNC(=O)C(C)OCCOC)(C1)OC21CCOCC1 75041,Cc1c(C(N2CC(C)(C)C2C2CCN(C(=O)C3=CCCO3)CC2)=O)ccn1C 75042,c1(CN(C(C2COC(CNC(=O)CC(C)OC)C2)=O)CC)ccncc1 75043,CC1CC(C(=O)NC2CC3CN(C(=O)CCCCCF)CC3C2)CCS1(=O)=O 75044,CS(=N)(=O)c1ccc(S(=O)(=O)CC(=O)NCCCCCCCCO)cc1 75045,c1(C(=O)NC2CCC(NC(C3CC(=O)N(C4CC4)C3)=O)CC2)ccnc(Cl)c1F 75046,C(c1ccc(Cl)cc1)=CCN(CCN(C)C)C(C1(O)CCCNC1)=O 75047,c1(OCCCNC(C(=O)NC(COC)CN)=O)cc(Cl)cc(Cl)c1 75048,C(=O)(CC(O)C(Cl)(Cl)Cl)N1CC(SC)C(NC(c2oc(C)cc2C)=O)C1 75049,C1(CN(C(=O)Cc2csc(=N)[nH]2)C)CCCN(C(C2(C(F)F)CCCCC2)=O)C1 75050,N1(C(c2nc(N(C)C)sc2)=O)CC2OCCN(C(=O)C(c3cccn3C)=O)C2C1 75051,c1(C(=O)NC(C(=O)NCC(C)NC(=O)OC)C2(C)CC2)cnn(C)c1C 75052,c1(CC(N2CCC(CNC(C(c3cncnc3)C)=O)C2)=O)noc2ccccc12 75053,c1(C(C)=O)ccc(C(=O)NC2CC(CNC(=O)CCc3nccs3)C2)[nH]1 75054,N1(C(CSCCC(C)C)=O)CCN(C(C2CCC=CCC2)=O)CC1C1CCC1 75055,c1(C(=O)NC(CC(C)NC(=O)COCc2nc[nH]n2)C)ccc(C2CC2)cc1 75056,N1(C(=O)Cc2ccc(Cl)cc2)CCC2C(CCN2c2ncc(Br)cn2)C1 75057,C(=O)(CCCCC(C)C(C)(c1nnnn1C1CC1)NCCC(F)F)OC 75058,CC(CN(C)C)CCC(=O)N(C)CCOCCN(C)C(c1ccnc(CO)c1)=O 75059,c1(OC)c(C)cc(C(=O)NC2CCC(NCc3ccc(C)c(Cl)c3)C2)cc1C 75060,C=CCCCCCC(=O)NCC1(NC(=O)C(C)(COC)c2ccccc2)CC1 75061,c1(C(N2C(CCC)CN(C(=O)CC3CCCOC3)CC2)=O)cccc2nc[nH]c12 75062,CS(=O)(=O)c1cc(C(=O)NCC2CC(NC(c3ncc[nH]3)=O)C2)ccc1F 75063,N1(C(c2c(SC)cccn2)=O)CCN(C(=O)C=CC2CCCCCC2)CC1CF 75064,c1(C(=O)NC(C(C)NC(c2c(OC)ccc(C)c2)=O)C)cnc2sccn2c1=O 75065,C1(C(N2C(C(C)C)C(NC(=O)C=C3CCN(C)C3)CC2)=O)CS(=O)(=O)CC(=O)N1 75066,c1(CN2CC(CC(=O)NC3CCCCC3O)OCC2)ccc([N+](=O)[O-])cc1O 75067,C#CCCC(O)C(=O)NC(C1CCN(C(=O)CNC=O)CC1)C 75068,C1(CCCC)CCC(C(=O)NCCCCNC(c2cc(C3CC3)nn2C)=O)CC1 75069,N1(C(c2ccncn2)=O)CCN(c2nc(C(F)(F)F)ns2)CC(O)C1 75070,CCCC(O)CC(=O)NC1CC(CNC(c2cccc(NC3CCC3)c2)=O)C1 75071,c1(C2(C(=O)NCC(CN(C(C=CC)=O)CC)(C)C)CC2CO)cccc(Cl)c1 75072,C1(OCC)CCN(C(C2C3CC3CN2C(C2CC23CCCC3)=O)=O)CC1 75073,c1(C(=O)NCC2(CNC(c3c(C)ccn3C)=O)CCCC2)noc2ccccc12 75074,C1(N(C(c2occ(C)c2C)=O)C)CC2CCC(C1)N2C(=O)C(C(C)C)N(C)C 75075,N1(C(C(F)=CCC)=O)CCCN(CCNC(=O)CNC(=O)CCCCC)CC1 75076,CC(C)(C)C(CO)C(=O)NC(C)(CNC(=O)CC1CNC(=O)O1)CO 75077,C1(NC2CC2)CCN(C)CC1.c1(C2N(CC(C)C)C(=O)C(=O)N2)ccccc1 75078,c1(C(=O)NC(CNC(C(C)NC(CC)=O)=O)(C)C2CCC2)cc(O)ccc1F 75079,C(CC(C(C)(C)C)NC(=O)CC(C1CC1)C1CC1)N(C(c1c(CC)cco1)=O)C 75080,C1(NC(C(C)NC(C)=O)=O)COC2(C1)CN(C(=O)C(c1ccc(Cl)cc1)(C)C)C2 75081,c1(CC(=O)NC2C(CNc3nc(C)nc(Cl)c3)CCCC2)c[nH]c2ncccc12 75082,c1(CC)ccccc1C(NC(=NCc1ccco1)NCC1CCN(C)C1=O)C 75083,C1(C(N2CCC(OC)C2)=O)CCCCC1(C)NC(c1ccnc(OC)c1)=O 75084,C1(CNC(C2CCC(=O)N2)=O)COCCN1C(c1coc(C(F)(F)F)c1)=O 75085,C(=O)(CCCCCC#N)N1CCN(C(C2CCC(N(C)C)C2)=O)C(CCO)C1 75086,c1(NC(=O)C(C2CC23CCCCC3)N2CCC(F)CC2)ccc2c(c1)CCC2 75087,N1(C(C2N(C)C(=O)CCC2)=O)CCOC2CCN(C(c3nccnc3N)=O)CC12 75088,c1(C(N(C2CCN(C(c3cnc(C)cc3Cl)=O)C2)CCC)=O)c(Cl)cncc1Cl 75089,C12(COC)CCC(C(=O)NCCN(C)C(c3ccc(CF)cc3)=O)(CC1)CO2 75090,C(=O)(CCC(F)(F)C(F)(F)F)N1CC(OCC)C(CNC(=O)CCOC(C)C)C1 75091,Cn1nc(C(=O)NC2CCCC3CC23)c2cc(Br)ccc12 75092,C1(C(N(C(C#C)C2CCC2)C)=O)OCCC1N(C(C1CCOC1)=O)CC 75093,c1(CNC(c2ccc(OCC=C)cc2)c2nnnn2CC)ccc2cncn2c1 75094,N#Cc1cnc(N2CCC(CF)(NC(c3cccc(-n4cccn4)c3)=O)C2)s1 75095,CC(CN(C)C)CCC(=O)NCCC1(C(=O)NCC(c2ccco2)O)CC1 75096,C(C(CC(=O)NCc1noc(C(N)=O)n1)NC(=O)C(C)Cn1ccnc1)OC 75097,N1(C(c2ccc(C#C)nc2)=O)CCC2CN(C(=O)CC(C)CCC)CCC12 75098,C1(COC)(CNC(=O)CP(C)(C)=O)CCCN1C(=O)C=Cc1ccsc1 75099,N1(C(C(CSC)(C)NC(c2cc(Cl)ns2)=O)=O)CC(C)(C)C2CCCC12 75100,C1(C(C)NC(=O)C=CC2CCOCC2)CCCCN1C(=O)Cc1cc(C2CC2)on1 75101,N1(C(c2nc(CC)[nH]n2)=O)CCn2ncc(CNC(=O)C(F)=CC3CC3)c2C1 75102,c1(C(=O)NCC(CO)NC(C2CCOCC23CCC3)=O)cc2cc(F)ccc2s1 75103,c1(C(N2CCC3(NC(Cc4c(C)ccnc4)=O)C(C2)C3)=O)cc(C#N)ccc1Cl 75104,c1(C(=O)OC)ccc2c(c1)CC(NCC1CC(c3ccc(Cl)cc3)(O)C1)C2 75105,C1(NC(=O)CNC(=O)C2CC2)CC2CN(C(=O)Cc3ccc(F)cc3F)CC2C1 75106,C1(NC(c2cc(C)no2)=O)CN(C(=O)C(C)CC(F)F)C2(CCCC2)C1 75107,CCC(C)(C)C(C(=O)N1CCCN(C(=O)C(F)CC(C)C)CC1)OC 75108,c1(C(N(C)CCC2CCCCN2C(C2CC3CC3C2)=O)=O)cc(F)ccc1N 75109,CCC(CC)C(=O)NC(CC)C(=O)NCCN1CCC(OC)C1 75110,C(C)(C(=O)N1OC2CCC1C2)N(C(=O)C(F)CCC(C)(C)C)CC 75111,CCC(CO)C(=O)NCC(C)N(C)C(C1CCCN1C)=O 75112,CCCCCCC(F)C(=O)N1CCCC(N(C)C(c2c(C)ncnc2C)=O)CC1 75113,c1(C(c2n(C(CC)(C)C)nnn2)NC2CC(Cl)(Cl)C2)ccc(N(C)C)cn1 75114,c1(OC)ccc(C(N2CC(O)(C(C)NC(=O)C(C3CC3)N(C)C)C2)=O)cc1O 75115,c1(C(N(CCCNC(C2CCC(C)NC2=O)=O)C2CC2)=O)cnc([N+](=O)[O-])n1C 75116,C1(NC(C(c2cn(CC)nc2)(F)F)=O)CN(C(=O)CCn2cccn2)CC2CC12 75117,N1(C(C(=O)NC(c2nnnn2CC(F)(F)F)C)=O)CCOC(CF)C1 75118,Cc1cc(C(=O)NC(C)(CNC(C2(C)CCCN2C)=O)C2CC2)cc(C(F)F)c1 75119,C(CNC(=O)CNC(c1cscn1)=O)(C(C)(C)C)NC(c1cc(CC)no1)=O.S 75120,c1(CNC(CC2C(C)(C)C2)=O)ccc(CNC(C2CCC23CCC3)=O)c(F)c1 75121,c1(C(=O)NC(C(=O)N(CCC)CC)CCN(C)C)cc[nH]c2nccc1-2 75122,c1(C(=O)NC2CC(C)(NC(CC(C)c3cnn(C)c3)=O)C2)cc2n(c1)CCSC2 75123,c1(C(N2CC(O)(C(C)NC(CC)=O)C2)=O)cc([N+](=O)[O-])ccc1OC 75124,c1(CNC(C(C)OCCC=C)=O)nc2c(s1)CN(C(C1CC(C#N)C1)=O)CC2 75125,N1(C(Cc2n(C)cnn2)=O)CCOC2(CCN(C(C3CC3CF)=O)C2)C1 75126,N1(C(Cc2cc(C)no2)=O)CC(F)CC1CNC(c1sc(Cl)cc1Cl)=O 75127,CCCC(CCC)C(=O)OCC(C1CCCC1(C)C)=O 75128,C1(CN(C(C(C)SC)=O)C)CCC(CNC(=O)CN2CCC(C)(C)C2)CC1 75129,N1(CC)CCC2(CC2C(=O)N(C)OCC(=O)OC)C1.N12CC(C1)CC2=O 75130,Cc1ocnc1C(N1CC(N(C(=O)C=CSc2ccccc2)C)C1)=O 75131,C12(C(=O)NCCCOCCN(C(C3CC(CC)C3)=O)C)CCCC(=O)N1CCC2 75132,CON(CC1CCCCC1)C(=O)C(C)C1CCN(C(c2cncc(C)c2)=O)CC1 75133,N1(C(c2n[nH]c(C)c2Cl)=O)CCCCC(N(C)C(C2CCCO2)=O)C1 75134,Cc1oc(Cc2nnc(C(C)(C)C)o2)cc1C(=O)NC1CCN(S(C)(=O)=O)C1 75135,C1(NC(c2cnc(C)o2)=O)CCC(C)N(C(c2cn(C3CCCC3O)nn2)=O)C1 75136,c1(C(=O)NC2CCC(CNC(C(CC)C(C)(F)F)=O)C2)cccc2c1CNC2=O 75137,CCC(C(C)C)C(C(=O)NCCSC)N1CCCC(C(F)F)C1 75138,c1(C(N(CC#C)CC)=O)cccc(SC2CCCC(C(=O)O)O2)c1 75139,CC(C(CO)NC(=O)C(F)(F)C1CCCC1)NC(C1C(C)C1C)=O 75140,C=CC(C)(C)CC(=O)N1CC(C)(OCC(=O)NCC2CN(C)CCN2C)C1 75141,c1(OC)cc(Cl)cc2[nH]c(C(=O)NC(C)CCNC(=O)Cc3cncnc3)cc12 75142,CCC(C)CC(=O)C(=O)N1CC(O)CC1C(=O)NOCCN(C)C 75143,CCCC(CNC(=O)CC1CCSC1)NC(=O)COCCOC 75144,Cc1cc(C)c(C(N2CC(NC(c3cnc[nH]3)=O)CC(O)C2)=O)c(S)n1 75145,c1(CC)cc(CC)nc(N2CCCOC(CNC(=O)CC3(C)CC3(Cl)Cl)C2)n1 75146,Cc1ccc(CC(=O)NC(C2CN(C(=O)CNC(=O)C3CC3)CCO2)C)cn1 75147,C1(OC)CC(NC(c2ccn(C)n2)=O)CN(C(C2CC3(CC3)C2)=O)C1 75148,Cn1nc(C(F)F)c2cc(C(=O)OCC3CC3(F)F)sc12 75149,Cc1ccc2c(=O)c(C(=O)NC3CC3NC(=O)C=Cc3cnc[nH]3)c[nH]c2c1 75150,C1(C(=O)NC(CC#C)CC(N)=O)(NC(=O)OC(C)(C)C)CC2CCC(C2)C1 75151,O(NC(=O)C(CNC(C1CCC(=O)N(C)C1)=O)CC(C)C)CCCOCC 75152,c1(C(=O)NC2C=CC(CNC(=O)C3CC3)C2)ccc(-c2cscn2)nc1 75153,c1(CC(=O)NC(C2CCCCC2)C(C)NC(C(C)=C2CC2)=O)nonc1C 75154,C(=O)(C#CC1CCC(=O)CC1)N1CCCC(N(C(c2c(CC)ccs2)=O)C)CC1 75155,c1(C(=O)NCC2CCC(NC(CC(C)NC(N)=O)=O)CC2)cc(F)ccc1Cl 75156,N(C(=NCC1CC1)NCc1cc(C)on1)CC(C1CCC1)OCC 75157,C1(C(N(C)Cc2ccncn2)=O)CC2CC2N1C(=O)CCc1ccccc1 75158,Cc1nn(-c2cccc(F)c2)cc1C(=O)N(C)CCNC(=O)CC1(C2CC2)CC1 75159,C1(C2(O)CCOCC2)(C(N2CCC(NC(C3(C)CCC(=O)N3)=O)C(F)C2)=O)CC1 75160,c1(C(N2C3CC(C(=O)NC(CCC)CC)C2CC3)=O)nccc2cc[nH]c12 75161,c1(C(=O)NCC2CCCC(NC(C(C)C3CCC3)=O)C2)ccsc1S(C)(=O)=O 75162,C1(C(N(CCCCNC(C(N2CC(C)C2)C)=O)C)=O)CCOC(C)(C)C1 75163,C1(CCNC(c2cc(C)c(C)[nH]2)=O)CN(C(=O)C=CC(F)(F)F)CCS1(=O)=O 75164,C(=O)(CCCC(C)(C)NC(=O)CNc1ccccn1)NC1C(N(C)C)CCCC1 75165,C1(C(F)(F)F)(C(=O)NCC(C)N(C(c2cn(CCOC)nn2)=O)C)CCN(C)C1 75166,c1(C(N2CC(NC(C(C)n3cncn3)=O)C(C)C2)=O)cccc(O)c1Cl 75167,N1(C(C(C)(CO)OC)=O)CCCN(C(C2CC3(CCO2)CC3)=O)CC1 75168,C(=O)(C(F)(F)C(F)F)NCC(c1cccc(C)c1)NC(C12CCCCC1C2)=O 75169,CC(C)C(C)C(CNC(=O)Cn1ccc(C(F)F)n1)NC(c1nnc(S)n1C)=O 75170,C#CCCCC(=O)NCC(CNC(C1CCN(CC(C)C)C1)=O)OC 75171,C(CCN=C(NCc1cccn1C)NCC1(C(C)C)CCCC1)OC(C)C 75172,C1(NC(CSC(c2n[nH]c(=N)s2)C)=O)(CO)CC1(C)C 75173,c1(C(=O)NCC2C(NC(CCC(C)C)=O)CCCC2)ccc([N+](=O)[O-])c(C#N)c1 75174,N1(C(CNC(=O)NC)=O)CCCC2(CCN(c3cc(C)nc(C(C)(C)C)n3)C2)C1 75175,C(=O)(C(F)CCC(C)(C)C)N1C(CC(=O)NC2(C(COC)O)CC2)CCC1 75176,CC(F)(F)C(=O)NC1CCN(C(c2cc(C3CC3)no2)=O)C1 75177,C1(CC)CCC(C)N(C(c2c[nH]nc2CCNC(c2ccc(C(C)C)o2)=O)=O)C1 75178,C1(C(=O)OC)(NC(c2nnnn2C2COC2)Cc2ccc(C)cc2)CC(C)(C)C1 75179,C1(CNC(CCOCC#C)=O)CCN(C(c2ccc(F)c(F)c2)=O)CC1C 75180,CCCCCCC(=O)N1CCC(C(C)C(N2CC(C(=O)OC)C(F)C2)=O)C1 75181,Cc1c[nH]c(C(=O)NCC(CO)NC(=O)C=Cc2cccs2)c1 75182,N1(C(c2cn(C)nc2)=O)CCC(C)(C)C1CNC(c1n[nH]c2c1CCC2)=O 75183,c1(C(=O)NC2CCCN(C(=O)CCCCCO)C2)nc(Cl)ccc1F 75184,N1(C(CC(C(C)C)OCC)=O)CC2CCCN(C(=O)CC(O)CC(C)C)C2C1 75185,CC1(C#CC(=O)NC2(CNC(=O)CSCCN(C)C)CCOC2)COC1 75186,Cc1ccnc(O)c1C(=O)NCCOCCCNC(=O)C(F)=C1CCC1 75187,c1(C(=O)NCC2CC(CNC(C3CN(C)C3)=O)OC2)cc2c(s1)CCC2=O 75188,C=CCC(C(=O)NCc1ccc(CC)o1)NC(=O)CC1CCCCO1 75189,c1(C(=O)NC(CC=C)CNC(=O)Cc2ccccc2C)cncc([N+](=O)[O-])c1 75190,c1(C(=O)NCC(CO)NC(CCC(=C)C)=O)cccc2c1CCO2 75191,C1(CNC(CC2(C(=O)OC)CC2)=O)CN(C(=O)Cc2cccc(F)c2F)CC12CC2 75192,C(C(C)C(C)C(=O)NC(C)(C)CN(C(=O)COC1(C)CCCC1)C)OC 75193,Nc1c(C(=O)NCCNC(c2c(Cl)cncc2Cl)=O)ccc(Cl)c1Cl 75194,N1(C(C(CC)n2ccnc2)=O)CCC(NC(c2sc(C)cc2C)=O)C(F)C1 75195,c1(C(=O)NCC(C)NC(c2cn(CC)nc2)=O)cccc(OC(F)F)c1 75196,c1(C(=O)NCCc2cc(Cl)ccc2Br)cc2nccn2c(O)n1 75197,N1(C(c2oc(CC)c(C)c2)=O)CCC(C)(C)C1C(=O)NC1CCOC(C)(CC)C1 75198,N1(C(C(CC#C)C2CC2)=O)CCC(C)N(C(c2ccc3ncccn23)=O)CC1 75199,c1(OC)n[nH]c(C(N2CC3CC3(CNC(=O)CN(S(C)(=O)=O)C)C2)=O)c1Cl 75200,C1(CNC(C2CCCO2)=O)CC(NC(c2cc(C3CCOCC3)no2)=O)CC1O 75201,N1(C(CSCC(C)C)=O)CCC2(CC1)CN(C(=O)CC1CCOC(C)(C)C1)C2 75202,C(=O)(C(C)C(C)(C)C)N(CC(=O)NC1CN(C)NC1=O)C(C)C 75203,c1(C(N(CCNC(C(C2CCC(C)CC2)CC)=O)C)=O)cc(C)c(=O)n(C)c1 75204,Cc1cc(C(=O)NC2CCC(NC(C3CC(F)C3)=O)C2)ccn1 75205,C(CN=C(NCC(F)(F)C(C1CC1)OC)NC(c1ccccc1)CF)OC 75206,C(=O)(C(C)(C)c1nccs1)N(CCNC(=O)CCSCC(C)C)CC 75207,n1(CC(=O)N(C(CNC(Cc2ncc(C)[nH]2)=O)C)C)cc(C#N)cn1 75208,C1(N(C(Cc2c(C)n(C)cn2)=O)C)CCN(C(c2cc(Cl)ccc2N)=O)CC1C 75209,c1(OC)ccc2cnc(C(N3CC(CNC(=O)C4=CCC4)CC3(C)C)=O)cc2c1 75210,C(CC1=CCCCC1)N(C(CN1CC2C(CNC(C)=O)C2C1)=O)C 75211,C12(NC(C(c3ccc(F)cc3)CC)=O)CCCC(NC(C3CCN(C)C3)=O)(C1)C2 75212,C1(C)(CNC(CCCOCC)=O)COCCN(C(C2(NC(C)=O)CCC2)=O)C1 75213,C(c1cccc(C)c1)=CC(=O)NC1CCC(C(=O)NC(C#C)COC)C1 75214,C1(CCNC(C(c2ccc(Cl)cc2)(C)C)=O)CSCCN1C(C1(F)CCC1)=O 75215,N1(C(C(C(C)C)NC(C)=O)=O)CC(C(=O)Nc2c(C)ncnc2C)CCC1(C)C 75216,C(C(CC(F)(F)F)NC(=O)CC(C)n1cccn1)NC(CC=CCC)=O 75217,c1(CC)cccnc1C(N1CCCC(CN(C)C(C2(CF)CCC2)=O)C1)=O 75218,Cc1nc(O)nc(C)c1CCC(N1CCC(O)C(NC(c2n[nH]cc2F)=O)C1)=O 75219,CN1Cc2ccccc2CC1C(=O)NC1CCCN(Cc2cocn2)CC1 75220,C1(CNC(=O)COC(F)(F)F)CC(O)CN1C(=O)COCCN(C)C 75221,CC(C)CC(C(=O)NC(CCO)C1CCCC1)NC(c1cc(C)n(C)n1)=O 75222,c1(C(N(CCCNC(c2sc(OC)nc2Cl)=O)CC)=O)cc(F)ccc1O 75223,C1(C(N2CCC(O)(C(C)NC(CCOCC#C)=O)CC2)=O)CCc2c[nH]nc2C1 75224,c1(C(=O)NC2(CC=C)CN(C(=O)C(=O)NC(C)C)C2)cc(OC)ccc1F 75225,N1(C(C=CC(C)(C)NC(c2cc(OC)ns2)=O)=O)CCCCCC1CO 75226,c1(C(N(C2CCN(C(C3SCCCS3)=O)C2)CC)=O)cc(C(C)=O)n(C)c1 75227,c1(CC)ccc(C(N2CCC(NC(c3cn(C)nc3C)=O)C(F)C2)=O)cc1F 75228,N1(C(C(C)C(C)O)=O)CC(C)(C)OC2(C1)CN(C(c1ccsc1Br)=O)C2 75229,Cc1nc(C(=O)N(C(C)CNC(c2cnc(C(N)=O)s2)=O)C)cn1C(F)F 75230,C1(C(=O)NCC2(C(N)=O)CN(C(CC(CC)C3CC3)=O)C2)CC2CCC(C1)C2=O 75231,C(=O)(C(CC(=O)NC1CC(CNC(c2cc3occc3s2)=O)C1)C(C)=O)OCC 75232,N1(C(C2(O)CCSC2)=O)CCC2(C1)CN(C(C1(O)COC1)=O)C2 75233,c1(CNC(C(CCC#C)O)=O)nn(C)c2c1CN(C(=O)C(C)N(C)C(C)=O)CC2 75234,Cc1nc(Br)c(Br)n1CC(=O)NC(c1ccnn1C)CO 75235,C1(CNC(CSCC=C)=O)CN(C(c2cccc3c2NCC3)=O)C2COCC2O1 75236,c1(NC(N2C(C(=O)NC)C(C)CC2)=O)cc(C)cnc1OC 75237,c1(C(=O)NC(CNC(CC(n2c(CC)ncc2)C)=O)CO)sc(C)c(C)c1C 75238,CCC(C)C(O)C(C)C(=O)NC(C(=O)NCCc1ccncc1C)c1cccs1 75239,C(C(=O)NCC1(S(C)=O)CC1)(C(C)(C)C)NC(C1CCC(C)CC1)=O 75240,c1(C(=O)NCC(CN(C(C2CCS(=O)(=O)C2)=O)CC)(C)C)ccccc1C 75241,C(=O)(C(F)(F)CCn1cccn1)N(CCC1CC(NC(=O)CC(F)(F)F)C1)C1CC1 75242,N1(C(c2cc(C)ncn2)=O)CCC(CNC(C2COC(=O)N2)=O)C1(C)C 75243,C(CCC(C(=O)N(CC(C)(C)C)C)NC(=O)CC1CCCC(=O)N1)OC 75244,C1(NC(c2c(C)cn(C)c2)=O)C(C)CCN(c2ncns2)C1C 75245,N1(C(c2cc(C)cc(F)c2)=O)CCCN(C(C2CC=CCC2)=O)CC1CO 75246,N1(C(c2cn(CC=C)nn2)=O)CCC2CN(C(=O)Cc3ccc(Cl)s3)C(C)C12 75247,C(=O)(C1CCCc2sccc21)N1CC(C)(NC(c2cc3ccccc3nn2)=O)C1 75248,N1(C(CC2CC(=C)C2)=O)CCN(C(c2ncn3ccccc23)=O)CC2(CC2)C1 75249,C(C(COC)C(=O)NC1(O)CC(C(N2CCC(CCCO)C2)=O)C1)OC 75250,N1(C(C(C=C)OC)=O)CC2(CC(C(=O)N(C(C3CCC3)C)CC)CO2)C1 75251,c1(C(=O)NCC(CNC(=O)C2=NOCC2)F)cnc2[nH]c(O)nc2c1 75252,C1(C(=O)NCC(C(=O)NC2CN(C(C)C)C(=O)C2)O)CCC(O)CN1C 75253,CCC1=C(C(=O)N2CCCCC2CNC(=O)C(CC)CC(C)C)CCCO1 75254,C1(N=c2[nH]nc(C(F)F)o2)(CNC(C(C(C)O)C)=O)CCCCCC1 75255,C1(OC)CN(C(c2nc[nH]n2)=O)CC1C(=O)NC1CCN(C)C1 75256,C1(CC(N2CCN(CC3CN(C(C4C(C)C4)=O)C3)CC2)=O)CCCC(F)(F)C1 75257,N1(C(CSCC)=O)CC2CCCC2(CNC(=O)C(C)Cc2ccc(C)cc2)C1 75258,C(=O)(C1CCc2c[nH]nc21)NCCCN(C(=O)CCn1cncn1)CCC 75259,Cc1ncc(C(=O)NCC2(CN(C)C(c3cc(C)sn3)=O)CC2)s1 75260,C(=O)(C(C)CCC(C)(C)C)N1CC(O)CCC(NC(C=CCCC(C)C)=O)C1 75261,c1(CC(=O)NC2CCCC(CNC(C)=O)C2)ccc(F)cc1[N+](=O)[O-] 75262,N1(C(CCOCCCOC)=O)CCCC(CO)(NC(c2c[nH]nc2C)=O)C1 75263,N1(C(c2ccc(F)s2)C(=O)NCC)CCc2c(cc(F)c(F)c2F)C1 75264,c1(OC)ccncc1C(N1CCCC(N(C(=O)C(C2CC2)OC)CCF)C1)=O 75265,Cc1ccc(C#N)c(NCC(c2ccccc2)NC(C2CCS(=O)(=O)N2)=O)n1 75266,c1(C(N2CCC(O)(CN(C(C3CCC(=C)CC3)=O)C)C2)=O)cc2ccsc2n1C 75267,C1(O)(CNC(c2cn(CCOC)nn2)=O)CCCN(C(c2scnc2C)=O)CC1 75268,C12(C(=O)NCCCNC(=O)OC)C(NC(=O)Cc3cnns3)C3CC1C2C3 75269,Cc1c(C(=O)NC(C2CCN(C(c3occ4c3CCC4)=O)CC2)C)cncc1Cl 75270,c1(C(=O)NCCC(CNC(c2c(C)n(C)nn2)=O)O)cc(C(F)(F)F)ccc1F 75271,c1(COCC)nc(-c2ccn(C(C)CC(C)C)n2)n(-c2ccccc2)n1 75272,n1(C(C)C)cnc2c(NCC3(C)CS(=O)(=O)C3)[nH]c(=NC3CCCCC3C)nc12 75273,C1(S(C)=O)(C(=O)OC)CCN(C(c2nnc3n2CCCC3)=O)CC1 75274,Cn1c(=O)sc2cc(S(=O)(=O)NCc3ccc4c(n3)NCCC4)ccc12 75275,C(CNC(C1CCCN(C(C)=O)C1)=O)(CC(C)C)NC(c1ccc(CCC)s1)=O 75276,c1(CC(C(=O)NCC2CCN(C(C(C)n3cncn3)=O)CC2)=O)ccc(Cl)cc1 75277,c1(SC)nc(Cl)cc(=NC2CC3CN(C(=O)COCc4ccc(C)cc4)CC23)[nH]1 75278,C1(SC)CCCN(C(=O)CCCC(C)c2ccccc2)C1C 75279,O=C(C1CCc2ccccc21)NCC1CCCC1NC(C1CCCS1(=O)=O)=O 75280,c1(C(N2C(CNC(CC(C(=C)C)O)=O)CC2)=O)ccsc1S(N)(=O)=O 75281,N1(C(C2C3N(C(c4ccc(C)cn4)=O)CC(CC3)C2)=O)CCCC(F)C(F)(F)C1 75282,c12cc(cc(C(=O)NN3CC4CCC3C4)c1)NC(=O)N2.C1(COCC)CC1CC 75283,C1(C(N2CC(OCCCCC)C2)=O)C=CCN1C(=O)C(n1ccc(C)n1)C 75284,C1(NC(c2ccc(C(CC)(C)C)cc2)=O)CCN(C(=O)C(C)C(C)C)C12CCC2 75285,C1(OC)CN(C(=O)CC2(O)CCCC2)CC1NC(=O)C(C)Sc1ccccc1 75286,CCC(C(=O)NCC(C1CC1)NC(C1CN(S(C)(=O)=O)C1)=O)n1nccc1C 75287,N1(C(c2c(CC)ccs2)=O)CCC(C(N2CCCCCC2)=O)C1C(C)C 75288,c1(NC(C23C(CN(c4nc(SC)c(F)cn4)C2)C3)=O)cc(F)c(C#N)cc1F 75289,C=C(Cl)C(C)(C)C(=O)N1CCC(O)(CNC(c2c[nH]c(-c3ccccc3)c2)=O)C1 75290,c1(C(=O)NC2C(NC(CCSC)=O)CS(=O)(=O)C2)ccc2ncn(C)c2n1 75291,C1(CC)CN(C(=O)CCCN(C)C)CCC1NC(C1(F)CCCC1)=O 75292,C1(CCNC(COCCC=C)=O)CN(C(c2cnc(N(C)C)s2)=O)CCO1 75293,N1(C(C=CCN(C)C)=O)CCC2CCC(C1)N2C(c1cc(N)ccc1O)=O 75294,N1(C(c2cc(OC)cc(F)c2)C(=O)NCCC#N)CCCc2c(C)cccc21 75295,C(C(C)(C)CCC#N)(c1n(CCCC)nnn1)NCc1cc(OC)ccc1C 75296,n1(CCC)ncc(C(=O)NC2C3CC(NC(c4nocc4C(C)C)=O)CC23)c1C 75297,C1(CC=C)(NC(C2CCCO2)=O)CCN(C(c2ccc(N)c(Br)n2)=O)CC1 75298,C(=O)(CC(F)(F)C(F)F)NC(CC(C)NC(c1c(C)nc(C2CCCC2)s1)=O)C 75299,C1(C(=O)NC(c2nc[nH]n2)C)(CNC(c2nonc2N)=O)CCCCC1 75300,C(=O)(CC(C(F)F)n1cccn1)N1CC(C)C(CNC(c2cnsn2)=O)C1 75301,n1(CC)nc(C)c(NC(=O)CC(CNC(=O)CC(C)(F)F)OC)c1C 75302,C(c1ccc(OC(F)F)cc1)=CC(=O)NCCn1ccnc1.C=CC 75303,N1(C(C(CC)CC2CCCCC2)=O)CC(C)(CNC(C2(O)CC2)=O)CC1(C)C 75304,C1(C(=O)NCC2CC(C(=O)OC)C2)CC12CCN(C(=O)C1=CCN(C)C1)C2 75305,N1(C(CC(C#C)O)=O)CC(C)(C)CC(C)(C)C1 75306,C1(F)(C(=O)NCCc2c(CNC(CC(C)OC)=O)nco2)CCS(=O)(=O)C1 75307,C1(CNC(C(C=C)O)=O)CCN(C(c2nc(OC)c(C)s2)=O)C1(C)C 75308,N1(CC)CC(C(N2CCCC2C(=O)NCCCCCCC2CC2)=O)CC1=O 75309,CCCC(C(C)(C)C)NC(=O)CCC1CCN(C(=O)Cc2csnn2)CC1 75310,N1(C(C)C)CC(C(=O)N(C)CC2(NC(C3CC(CF)C3)=O)CC2)CCC1=O 75311,C1(CC(=O)NC2CC(N(C)C(C3CC4CCC3C4)=O)C2)CCC(F)(F)CC1 75312,c1(NCC2(NC(C(C)C3CCCC3)=O)CCCC2)ncc(Cl)cc1[N+](=O)[O-] 75313,N1(C(C(C=C)OC)=O)CC(O)CC1C(=O)NCCOC1CCOC1 75314,N1(C(c2ccoc2Cl)=O)CCCC1C1CCCN1C(c1c[nH]nc1Br)=O 75315,c1(C(N(C2CCN(C(C(CC)O)=O)C2)CCO)=O)c[nH]c(=N)c2[nH]ccc12 75316,C=CCC(CC(=O)NC(C)C(=O)NC1CC1)NC(=O)COC1(C)CCC1 75317,C(=O)(CC(c1ccccc1)NC(C1CC12CC2)=O)N(C)CC1CCCN1C(N)=O 75318,c1(C(=O)NC2CCN(C(C(C)NS(CC)(=O)=O)=O)C2)cc(N)ccc1O 75319,C(CCCCC(=O)NC(C)CO)NC(C(=CC1CCCC1)C)=O 75320,Cc1cnc(C)c(NC(C2CC2c2ccccc2OC(F)F)=O)n1 75321,c1(CNC(C2(C(F)F)CC(=C)C2)=O)ccc2c(c1)CN(C(C1CC1F)=O)C2 75322,C(=O)(CC1=NNC(=O)C1)NCC1CC(NC(c2c(OC)ccs2)=O)C(O)C1 75323,C1(C(C(=O)NC(CC)C)N(CCCCO)C)C2CCOCC12 75324,N1(C(C(F)OC)=O)CCCC1C(C)NC(=O)C(C)(C)NS(C)(=O)=O 75325,C(C(C)(C)S(C)(=O)=O)n1c(-c2cc(C(F)F)[nH]n2)nc(CCN(C)C)n1 75326,CC(C)(C#Cc1cn(-c2ccc(F)nc2)nn1)NC(c1nsc2ccccc12)=O 75327,N1(C(c2c(OC)c[nH]n2)=O)CCN(C(c2ccc(F)cn2)=O)C(C2CCC2)C1 75328,C1(CC(=O)NCC(COC)C)CC2(C1)CN(C(=O)C(C)C(F)(F)F)C2 75329,c1(C(=O)NCC23CC2CN(C(=O)C=Cc2ccoc2)C3)nsc2c(Cl)cccc12 75330,C1(F)(CNC(C(CC(C)C)N(C)C)=O)CCCN(C(=O)OC(C)(C)C)CC1 75331,N1(C(c2cn(CC=C)nn2)=O)CCC(F)C(NC(c2cc(C3(C)CC3)n[nH]2)=O)C1 75332,CCC(C)(C(=O)NC1CN(C(c2ccccc2NC2CCC2)=O)CC1OC)OC 75333,c1(OC)cccc(C(C)N(C)Cc2ccn(C(F)(F)C(F)OC(C)(C)C)c2)c1 75334,c1(C(=O)NCC2CC(CC)CN2C(c2cc(=O)n(C)cn2)=O)ccc(F)c(O)c1 75335,CCCCC(CNC(c1ccnc(NC(=O)C(C)OCC(C)C)c1)=O)NC(C)=O 75336,Cn1cc(C(C(=O)NCCC#CCO)NC(CCNC(N)=O)=O)nn1 75337,c1(NCC)cc(Cl)ccc1C(N1CCCC(C)(CNC(=O)C=CSC)C1)=O 75338,N1(C(=O)CC2=CCCC2)CCOC2(CCN(Cc3cc4cnccc4[nH]3)CC2)C1 75339,CCC(CC)C(C)NC(C1OCCC1NC(=O)C(C)(C1(C)CC1)OC)=O 75340,Cn1ncc([N+](=O)[O-])c1N(C12CCCCC1OCC2)CC1CCCN(C(N)=O)C1 75341,c1(C(=O)NCCC(C(C)C)NC(c2c(CC)nc[nH]2)=O)cccc2oc(O)nc12 75342,c1(OC2CC(NC(CCn3cc(CCCC(C)O)nn3)=O)C2)ccc(F)cc1 75343,CCCC(O)C(=O)N1CCC(C2N(C(=O)C=CC3CC3)CC2(C)C)CC1 75344,C1(NC(C2C(C(=O)OC)C2(C)C)=O)CCC(C)N(C(c2ccc(F)c(F)c2)=O)C1 75345,C1(C)(C(=O)NC(C2CCN(C(=O)C(C3CCCO3)C3CC3)C2)C)C=CCC1 75346,c1(CC)cc(C(N2CCOCC2CC(=O)NC(C)Cc2cnc[nH]2)=O)ncn1 75347,C(C(C)C(C)C(=O)NCC1(O)CN(C(=O)C(O)C2CCC2)C1)OC 75348,C1(NC(C2(CC(C)C)CCCC2)=O)CC2CC(NC(c3ccc(Cl)cn3)=O)C2C1 75349,c1(C(=O)NCC2CCN(C(c3cnc(CC)[nH]3)=O)C2)c(C)cc(C)nc1O 75350,Cc1cc(N)c(C(=O)NC(C)(CNC(=O)C(C)(C)c2ccccc2)CO)cc1C 75351,O=C(C#CC1CC1)NCC12CC1CN(C(C1CC(=O)N(CC3CC3)C1)=O)C2 75352,N1(C(C2CC(CC)(CC)C2)=O)CC(NC(N2CCCC2CN(C)C)=O)CC1(C)C 75353,c1(C(=O)NCC(C)N(C)C(c2ncncc2Cl)=O)c[nH]cc(Cl)c1=O 75354,CC1CC(=O)NCC1C(N1CCCC1(C)CNC(C1CC(O)C1)=O)=O 75355,c1(OC)ccc(Br)nc1CN1CCCC(C)(C(=O)Nc2nc(Br)ccc2Br)C1 75356,Cc1cnoc1C(=O)N(C(C)CNC(=O)CC1(N2CCOCC2)CC1)CCO 75357,C#CCC(C)(CC)C(=O)NC1C2CC3C1C3C2C(=O)NCC(C#C)OC 75358,CCCCCCCCC(=O)N(C1CCCN(C(=O)CC2CCCCC2O)C1)C 75359,CCCC(CCC)=CC(=O)N(CC)Cc1cn(-c2cc(C)sc2C)nn1 75360,C1(C(N2C(C)CCC2C(=O)Nc2ccc(F)nc2)=O)CC2CCCC2C1 75361,c1(C(=O)NCCCN(C(C(CC)OC)=O)C2CCCC2)ccc(C)n1C 75362,c1(COC)ccsc1C(=O)N(C1CCN(C(=O)CCC=C(C)C)C1)CCO 75363,C12(NC(C)CNC(=O)C(c3ccccc3)O)CCC1CNC2 75364,CC1CC(C(=O)N(C)CC2CCCC2(C)C)N(C(C2(C(N)=O)CCC2)=O)C1 75365,c1(C(=O)NCC(C)C)ccc(N2CCN(C(=O)C=Cc3ccsc3)CC2)cn1 75366,C(C(=O)NNC(=O)C1=CS(=O)CCC1)(c1ccccc1)OC 75367,Cc1cc(C(=O)NC2CC(CNC(c3cc(C4CC4)n(C)n3)=O)C2(C)C)cn1C 75368,C(=O)(CC(C)(C(F)F)N(C)C)N1CCN(C(c2c(C)[nH]c(C#N)c2)=O)CC1CO 75369,N1(C(CC(=O)NCC#C)=O)CCN(C(C)CNC(c2cnns2)=O)CC1 75370,c1(C(N2CC(N(C(C(C)CC3CC3)=O)C)C(O)C2)=O)cc(C(F)F)ccc1Cl 75371,N1(C(c2nc(C)c(C)s2)C(=O)NCC)CC(C)C(C)C1C 75372,c1(N(CC)CC)ccc(CCC(=O)NCC(CC)NC(C2CCC2(C)C)=O)cc1 75373,CC(C(=O)NC1CN(C(C2(C3CCC3)CC2)=O)CCC1C)S(N)(=O)=O 75374,C1(C(=O)NC2CC(CNC(c3ccsc3C)=O)C2)(OCC)CCSCC1 75375,C1(F)(CNC(CC2(OC)CN(C(=O)Cc3cc(C)on3)C2)=O)CCN(C)C1 75376,Cc1cc2[nH]c(C(=O)NC3CC4(CCN(C(C56CC(CO5)C6)=O)C4)C3)cc2o1 75377,N1(C(C2(CNC(CCC(=O)NCC)=O)CCCCC2)=O)CC(O)C(O)C12CCC2 75378,C(C)(C)(CC(=O)NCc1ccoc1C(=O)NCCCC(O)CO)N(C)C 75379,c1(C(=O)NC(C(=O)N(CC)Cc2cnn(C)c2)c2ccoc2)cc(OC)n(C)n1 75380,N1(C(CC2CCCN(C(C=CCC)=O)CC2)=O)CC2CCCC2C12CC2 75381,CC1CCN(C(c2ccc3c[nH]nc3c2)=O)C(C)C1NC(c1ccc(F)nc1)=O 75382,C1(NC(c2cc(C)nc(C)n2)=O)CC2CCC(C1)N2C(=O)C(O)c1cnc[nH]1 75383,c1(C(=O)NC2CCC(F)(CNC(C)=O)C2)ccc(Nc2ccncc2)cc1Cl 75384,c1(C(=O)NC2C(C)CN(C(=O)Cc3ccon3)CC2)c(Cl)ccc(F)c1F 75385,C(=O)(C(F)(F)C(F)(F)C(F)F)N1CC(NC(C2CCc3n[nH]cc3C2)=O)(CO)C1 75386,CCC(O)C(F)(F)C(=O)NCCCC1CCN(C(=O)CC(C)C(C)(C)C)CC1 75387,N1(C(C)=O)CCC2(CO)CN(C(c3coc4cc(F)cc(F)c34)=O)CC2C1 75388,Cc1cc(C)c(C(=O)NCCN(C(=O)CC2CC2C)C)c(C)c1 75389,N1(C(C(CCOC)NC(=O)CC(F)(F)F)=O)CCC(F)(F)C(F)C1 75390,C#Cc1ccc(OCC(=O)NCC2CCN(C(=O)C(C)CCO)CC2)cc1 75391,O=C(C1CCc2ccccc21)NC1CN(C(C2CCC(CO)CC2)=O)CC1F 75392,CN=c1nc(N2CCOc3cccc(Cl)c3C2)[nH]c(=NC(C)C2CCN(C)C2)[nH]1 75393,C1(N(C(=O)Cc2ccsc2Cl)C)CC2CC1N(C(c1ccncc1F)=O)C2 75394,C1(C(=O)NC(CNC(C2C(COC)C2)=O)CO)Cc2cccc(OC(F)F)c2O1 75395,C(=O)(CCCC(F)(F)C(F)(F)F)N1CCC(O)(CNC(C(CC=CC)CC)=O)C1 75396,c1(C(N2CCN(C(CCOCC#C)=O)C(COC)C2)=O)cnc2n1CCC(C)C2 75397,C1(C)(C(=O)Nc2c(C(=O)OC)n[nH]c2)COCCN1C(=O)CC1NC(=O)NC1=O 75398,Cc1ccc(C(=O)NCC2(NC(C3CCCCN3C)=O)CCCCC2C)c(N)c1 75399,N1(Cc2c(C)nccc2)CCc2cccc(C(N3CC4COCC4C3)=O)c2C1 75400,C1(C)(CC(=O)NC(COCC)C)CCN1C(=O)CC1(C)OCCO1 75401,C1(C(N2CCC(C(C)NC(c3cscn3)=O)C2)=O)CC1C1CC1C 75402,N1(C(c2ccccc2Cl)C(=O)NCC)CCn2c(CC)nnc2C1 75403,Cc1ccc(Cl)cc1-c1cn(C2CN(C(c3csc(CC(C)C)n3)=O)C2)nn1 75404,CC1(C)CCCCC1C(=O)NC1C=CC(C(=O)NCC2CC(O)C(O)C2)C1 75405,N1(C(c2cc(C)on2)=O)CCC(F)(C(=O)NC(C2CCCOC2)(C)C)CC1 75406,N1(C(C(CCC)OCC)=O)CCCC(C2CN(C(=O)COc3cccc(Cl)c3)C2)C1 75407,N1(C(C2=CCCN(C(=O)OC(C)(C)C)C2)=O)CCC2(C1)CS(=O)(=O)C2 75408,C1(CC(N2CCC(N(C(c3ccsc3C)=O)CC)C2)=O)CC(C)(C)OC1=O 75409,C(C(C)(C)CC(=O)NCC(C1CC1)NC(C1CC(C)(C)CO1)=O)N(C)C 75410,c1(C(=O)NCC2CC(NC(C34CCC(CC3)OC4)=O)C2)cc2cc(Cl)ccc2o1 75411,C1(O)(CNC(C2(CSC)CCC2)=O)CCN(C(=O)Cc2ccc(O)cc2Cl)CC1 75412,N1(C(CSCC=C)=O)CCCC2CN(C(=O)CCc3cnn(C)c3)CCCC12 75413,c1(C(N2CC(CC)C(NC(c3ccncc3)=O)CC2)=O)cc2nc(Cl)ccc2s1 75414,C1(C(=O)NC(CCC)(C)CC)CCC2(CC2)N1C(C1CCCOCC1)=O 75415,c1(CC)ncccc1C(N1CCCC1C(C)(C)NC(c1ccnnc1)=O)=O 75416,N1(C(c2c(C)cnnc2)=O)CCc2cccc(C(N3CCS(=O)CC3)=O)c2C1 75417,C1(C(=O)NCc2ccsn2)CN(C(=O)C(c2cccc(Br)c2)O)CCC1(F)F 75418,CC1CC(CN2CCCC2Cc2ccncc2)CCO1 75419,CCCCC(O)CC(=O)NCC1(O)CC(NC(=O)CCOc2ccc(C)cc2)C1 75420,C1(C)(NC(C=CCN(C)C)=O)CCN(C(=O)Cn2cnccc2=O)CC1 75421,c1(C(=O)NC2CC3(CN(C(CCCCC)=O)C3)C2)c(Cl)ccc(OC)c1N 75422,Cc1cc(=NCC(CNC(=O)C(F)CC(C)C)C(F)(F)F)[nH]c(C)n1 75423,N1(C(C(C(CC)C)O)=O)CCCC2(C1)CN(C(=O)C1=NNC(C(F)(F)F)C1)C2 75424,C1(C(N(CC(C)NC(=O)CCC(=O)c2ccc(F)cc2)C)=O)CCC2CCC1O2 75425,C1(C(=O)NC(C2(c3ccccc3)CCCC2)C)CC(=O)C12CC2 75426,N1(C(C2(O)CCN(C(C3CN(CC)C(=O)C3)=O)CC2)=O)C2CCC1C(N)C2 75427,Cc1cc(NC2CC(CNC(c3cc(C(N)=O)[nH]n3)=O)C2)nc(CC2CC2)n1 75428,C1(CNC(C=C(C)C2CC2)=O)(CNC(=O)C(C)OCC2CCCO2)CCCC1 75429,C1(CNC(c2cnc(C)s2)=O)CCN(C(=O)CC2CC(C)(C)C2)C1(C)C 75430,c1(C(C(=O)NCCC#N)N(C(CCSC)CO)C)ccc(CF)cc1 75431,C12(C(N3CCC(COC(C)=O)C3)=O)CCCC1CCN2C(=O)C1=CC2C=CC1C2 75432,N1(C(C(CC=CC)C)=O)CC(C(=O)NCC2CC23CCCCC3)C2(CC2)C1 75433,C1(C(=O)NCC2COCCN(C(c3cc(OC)n[nH]3)=O)C2)Cc2ccccc2O1 75434,C1(NC(c2cc(C)oc2C)=O)CNC(C)(C)COC1 75435,CC1CC(NC(=O)CNC(=O)OC(C)(C)C)CN(C(c2ncccc2Br)=O)C1 75436,c1(CC)cc(NC(N2CCCC2CC(c2ccccc2)O)=O)n(C)n1 75437,N1(C(c2ccc(CNC(c3occ(C(N)=O)c3)=O)o2)=O)CC(O)CC12CCC2 75438,N1(C(C(CC)n2ccnc2)=O)CCC2OCCN(C(c3nc(=O)n(C)[nH]3)=O)C2C1 75439,CC1CCCCC1(CNC(=O)CNC(c1cnn(C)c1)=O)NC(=O)C(F)=CC1CC1 75440,c1(OC)cc(C)c(C(C(=O)NCCCOC)N(CCC(O)CO)C)c(C)c1 75441,c1(C(N2CC(NC(C3(F)CCC3)=O)C(F)C2)=O)ccc(Br)c(Cl)c1Cl 75442,C1(S(C)(=O)=O)(C(N2CCC(F)(CNC(c3cc(C)sc3)=O)C2)=O)COC(=O)C1 75443,Cn1ncc(=NC(=O)C2CN(Cc3ccc4nccn4c3)CCC2O)[nH]1 75444,N1(C(c2n[nH]c(CC)c2C)=O)CCOCC(C(=O)N(CC(C)C(=O)OC)CC)C1 75445,C12(CNC(c3cn(CCOC)nc3)=O)CC1CN(C(c1ccn(CCF)n1)=O)C2 75446,C(=O)(CCC(C)(F)F)NC1(C)CC(NC(CN(C2CCC(=O)NC2)C)=O)C1 75447,C(CCOCC)(C(=O)N1CC(c2nc(=O)o[nH]2)C1)NC(C(C=C)O)=O 75448,CC1=C(C(=O)N2CCCC(C)(C(=O)NCc3ccc(C)n3C)C2)CCO1 75449,Cc1ccn(CCC(=O)NC2CC(C)(CNC(=O)Cc3n[nH]c(C)n3)C2)n1 75450,C1(C(=O)NC(C2CCCC2)CNC(c2cc(C#N)sc2)=O)CC2C=CCC(C1)C2 75451,C1(C(N(C(C)CNC(C2(CO)COC2)=O)C)=O)CC(=O)N(Cc2ccccc2)C1 75452,c1(C(C)NC(=O)C(N2CCS(=O)(=O)CC2)=O)ccc2ncsc2c1 75453,Cc1c(F)ccc(Cl)c1C(N1CC2CC(NC(=O)C(C)c3cccs3)C2C1)=O 75454,Cc1c(C(=O)NC(C2CCOC2)CNC(c2cncs2)=O)cccc1Br 75455,N1(C(c2nc(C(C)N)oc2)=O)CCC2(CC1)CN(C(=O)C=CCF)C2 75456,N#Cc1ccc(NC(c2n[nH]cc2NCc2c(Cl)ccnc2Br)=O)cc1Br 75457,C1(C(=O)NCc2cc(C(N(C)CC3(COC)CCC3)=O)n[nH]2)CCC(O)CN1C 75458,C(=O)(CC(C)C1CC1)NCCCCN(C(C1(CC)CCC1)=O)C 75459,C(=O)(C(=O)N=S(C)(C)=O)NCCC1(CNC(C(C)CC2CC2)=O)CC1 75460,Cn1nc(O)cc1C(=O)NCC(c1ccccc1)NC(c1nnsc1N)=O 75461,C12(NC(C(C)=C3CCCC3)=O)CCC(CC1)N(C(=O)C=Cc1ccncn1)C2 75462,CCCC(CC)C(=O)N1CC(F)CC1CNC(c1cc(N2CCCC2)cc(Cl)c1)=O 75463,N1(C(C2CC(C(C)C)C2)=O)CCC(CCNC(c2ncn(C)n2)=O)CC1 75464,c1(C(=O)NCC(C)CNC(C2CCOC(C)C2)=O)ccccc1-n1ccnn1 75465,C#CC1CN(C(=O)C(C2CCCO2)NC(=O)CCN2CCOCC2)CCO1 75466,c1(SC(C(=O)NCC(C)NC(C=CCCC=C(C)C)=O)C)nc2ccccc2[nH]1 75467,N1(C(C(C)OCCOC)=O)CCC2(CCCN(C(=O)CCCC3CC3)C2)CC1 75468,n1(CC(=O)NC2C(F)CCN(C(CC3(C)CCCCC3)=O)C2)cc2ncccc2n1 75469,Cc1ccc(C(=O)C(N2CCC(CCNC(c3ccc[n+]([O-])c3)=O)C2)=O)cc1 75470,C1(C)(C(=O)NCC(C)(CO)CO)CCCN(C(=O)COCC2CCOC2)C1 75471,c1(NC(C2CCC(NCc3cnn(CCC)c3C)CO2)=O)cc(F)c(Cl)cc1F 75472,c1(NC(C(C)(C)C2CCN(C(=O)CC3(C)CCC3)C2)=O)ccc2nccn2c1 75473,C(C)(C(=O)NCC1(C(=O)NCCCOCC(C)C)CCC1)OCC(C)C 75474,C1(NC(C(C2CC2)OCC)=O)CN(C(=O)Cc2ccc3c(c2)CC3)CCC1(F)F 75475,C1(C(N(C2C(C)(C)C2)C2CCC2)=O)CCC=CC1NC(c1cnncc1O)=O 75476,c1(N2CCN(Cc3onc(C(C)OCC)n3)CC2)ncc(C(=O)O)cc1Cl 75477,N1(C(c2[nH]ccc2CNC(C2(O)CCSC2)=O)=O)CCC(F)(F)C(O)C1 75478,C(CNC(C1CC1(C)C)=O)(CO)NC(CSCC)=O 75479,C1(NC(c2n(C)ncc2)=O)CN(C(c2cnccc2Cl)=O)C2(CCCC2)C1 75480,C1(CNC(C23OC(C)C(CC2)C3)=O)CC2CCC(C1)N2C(c1cc(F)c[nH]1)=O 75481,C1(CNC(C2N(C(CC)=O)CSC2)=O)CN(C)CCN1C(C1CCC(=O)N1C)=O 75482,C1(O)(CNC(C2=CC(C)(CC)C2)=O)CCCN(C(c2cc[nH]c2)=O)CC1 75483,C(=O)(C1CCCc2nc[nH]c21)NCC(C(C)(C)C)NC(c1cc(Br)no1)=O 75484,Cc1cnc(NC(C2CC2C(=O)Nc2cccc(I)n2)=O)c(C)c1 75485,CC1CC(NC(C2CC2C2CCC2)=O)CN(C(=O)Cc2nn(C)cc2Cl)C1 75486,C1(C)(NC(CN2C(C)CCC2)=O)CCCCC1C(=O)NCC1(ON)CCCOC1 75487,c1(C(C(C)NC(=O)C(=O)NCc2cc(C3CC3)[nH]n2)OC)ccc(Cl)cc1 75488,C(=O)(C1CCCc2nc[nH]c21)NCC1CN(C(c2nc(SC)sc2)=O)CC1C 75489,C1(CNC(C(C2CN(C(C3CCC(CO)C3)=O)C2)OC)=O)CCCN(C)C1 75490,c1(CC(=O)NC2CC(CNC(C3(CN(C)C)CC3)=O)C2)cc(F)c(F)cc1F 75491,C(=O)(C1=CN=C2N=CNN2C1)NC1CC(C)N(C(=O)C=Cc2nccs2)CC1 75492,N1(C(C(=O)NC(C)CCCNC(C2CCCO2)=O)C)CCCCCC1 75493,c1(OC)cc(Br)cc(CN2CCN(C(c3cnc(Cl)cc3C)=O)C3(CC3)C2)c1O 75494,C1(COC)(NC(C2CC23CCC3)=O)CCN(C(C2(C)CCCCO2)=O)CC1 75495,C(CC(C)C(=O)NCCC1CCCN1C(c1cc(-c2ccc(C)s2)[nH]n1)=O)OC 75496,Cc1cccc(C(N2CCC2CNC(=O)C(c2ccc(C#N)cc2)C(C)C)=O)c1O 75497,c1(C(=O)NC(CCCNC(CC=C=C)=O)C)c(NC(=O)N(C)CC)cccc1F 75498,c1(CC)c(OC)cccc1C(=O)NC1CN(C(=O)Cn2ccc(C)n2)CC12CC2 75499,CN1CCCC12CCN(C(c1nc(Cl)c(Cl)s1)=O)C2 75500,N1(C(CCNC(=O)OC)=O)C(C(=O)NCCCCO)CCC1C(C)C 75501,C(CC(F)(F)C(C)C)NC(C(C1(C)CC1)NC(C(C(=O)OCC)OC)=O)=O 75502,C1(C(N2CCC(C(=O)NC)C2C)=O)N(C(c2nc(C)sc2C)=O)CCCC1(C)C 75503,N1(C(C2C(C)CC2)=O)CCN(c2ccc(CCNC(=O)CC3(C)CC3)cc2)CC1 75504,C(=O)(CS(=O)(=O)CC(C)C)NCC1C(C(F)(F)F)CCN(C(CSCCCC)=O)C1 75505,c1(C(=O)NCC2(NC(C3(COC)CC3)=O)CC2)cnc(C(F)(F)F)s1 75506,CC1(C(N2CC3C(CNC(c4ccc(CC5CC5)s4)=O)C3C2)=O)CC2CC2C1 75507,S(=O)(=O)(CCNC(C1(c2ccccc2)CC1(C)C)=O)N1CC(CC)C1 75508,C1(NC(c2cn(CC(=O)OCC)nn2)=O)CCCCN(C(=O)C(C)C2CC2)C1 75509,Cc1cnc(CC(=O)NC2CN(C(c3cnnn3C3CCOCC3)=O)C2)o1 75510,C1(SC)CC(CC(=O)N(C(C)C(=O)NCCCC2CC(C)C2)C2CC2)C1 75511,c1(C(N(C2CCCC2)CCNC(C=COCC)=O)=O)cnn2c1CC(C)CC2 75512,N1(C(CS(CC)(=O)=O)=O)CC2COCC2(C(=O)NOCc2cccc(C)n2)C1 75513,c1(C(N(c2c(C(=O)NC)onc2C)C)=O)cc(C(=O)OC)cc(Br)c1 75514,CC(C)CC(C)NC(C1(NC(=O)CCn2cncn2)CC1)=O 75515,C1(C(=O)N(C2COC2)C2CCC2)CN2CCC1CC2.Cn1ncc2c1CNC2=O 75516,Cc1cn(-c2ccccn2)[nH]c1=NC(=O)N1CCC(c2cccs2)C1 75517,N1(C(CCOCC)=O)CCC(CN(C(=O)CC(CC)C2CC2)C2CC2)CC1 75518,c1(C(C)=O)ccncc1C(N1CC(O)CC1CNC(=O)CCN1CCOCC1)=O 75519,c1(NC(C2CC=CCN2C(C2CCCOCC2)=O)=O)ccc(CCF)cc1 75520,Cc1ncc(C(N2CCC(N(C(=O)CC3CCOCC3)CCO)C2)=O)[nH]1 75521,CCCCC(O)CC(=O)N1CCC(NC(=O)CCc2cnoc2)C12CCC2 75522,C1(C(N(C(C2CCC2)C)CC)=O)CC12CC(NC(=O)Cn1ccc(C)c1)C2 75523,c1(C(N2CCOCC2c2ccc(Br)nc2)=O)cc2c(Cl)c(Cl)ccc2[nH]1 75524,S(=O)(=O)(c1ccc(=NCCCCn2cnnc2)[nH]c1)NC1CCCC(CC)CC1 75525,c1(CC)ncncc1C(=O)NCC=CC(=O)NCC(=C1CCCCC1)F 75526,c1(NC(C2CC23CCNCC3)=O)nc(=NCC2CCCC2)[nH]cc1Br 75527,N1(C(=O)CC2C=CCCC2)CC(NC(C23CCC(F)(CC2)C3)=O)C2(CC2)C1 75528,C1(NC(Cc2nc(CC)sc2)=O)CC2CCC1CN(C(C1CC1F)=O)C2 75529,O=[N+]([O-])c1ccn(CCSc2ccc(C(=O)NOCC=CCl)cc2)n1 75530,Cc1ccc(C(N2CCCC2C2(C(N3CC(CO)C(C)(C)C3)=O)CC2)=O)cc1O 75531,C(=O)(CCCF)N(C(C)C)C(=O)NCC(=O)OC(C)(C)C 75532,c1(C(N(CCCC(=O)NC(C=C)(C)C)C)=O)ccc(C#N)n1C 75533,C1(NC(c2c(C)ncc(CC)c2)=O)CCOC2(CCS(=O)(=O)CC2)C1 75534,CN1CCOCC1C(=O)NC1(CCC(=O)NC2(C)CC2)CCC1 75535,C1(OCC#C)CCN(C(=O)CC2CCC(NC(C3CCCC3O)=O)C2)CC1 75536,c1(CC(=O)NC(C2CCN(C(=O)Cc3cnc[nH]3)CC2)(C)C)ccc(=N)[nH]c1 75537,C(C(CC)(CC)C(=O)N1CCC(OCC(N)=O)C1)NC(Cc1cn(CC)nc1)=O 75538,N1(C(C(CNC(C=C(CC)CC)=O)N(C)C)=O)CCS(=O)C(C)C1 75539,c1(CC)ccc(Cl)c(C(=O)NC2CCC(NC(=O)CN(C)C)CC2)c1 75540,Cc1ccc(C(N)=O)cc1C(=O)NC1CCC1NC(=O)Cc1cc(Cl)sc1Cl 75541,c1(C(=O)NC(C(C)NC(C(CCCC)(C)F)=O)CO)cnc2c(cnn2C)c1N 75542,N1(C(CCCCCCCNC(=NC)NC2CCCC2)=O)CCS(=O)(=O)N2CCCC12 75543,C(N=c1[nH]c(N(C)Cc2ccc(Cl)nc2)nc2cc[nH]c12)C1(CCC)CCC1 75544,N1(C(CCC(=C)C)=O)CCC2(C1)CN(C(C1C(C)=NOC1C)=O)C2 75545,C1(NC(c2c(C)cc(C)o2)=O)CC2(C1)CN(C(=O)Cc1cn3ccsc3n1)C2 75546,CCC(CC)(C(=O)N1CCC(C(F)C(=O)NC2CC(C)(C)OC2=O)C1)OC 75547,C1(CC)C(C(=O)NCCCOCCN(C)C(c2ccc(CC)[nH]2)=O)CCN1C 75548,c1(C(=O)NC2CN(C(CC(=O)NCC#C)=O)C2)c(Cl)c([N+](=O)[O-])nn1C 75549,C(=O)(C(C#N)C(C)C)N(CCNC(=O)C(O)COc1ccccc1)CC 75550,c1(C(C)C)cccc(F)c1C(=O)OC=CCC1CCN1C(c1cc(Cl)no1)=O 75551,CCCC(C(=O)NC12CCCN(C(=O)Cc3cccc(O)c3)CC1C2)S(N)(=O)=O 75552,N1(C(COC(CC)C)=O)CCC2(CC1)CN(C(c1cc(Cl)c(Cl)[nH]1)=O)C2C(C)C 75553,C1(O)(CCNC(CNC(CC)=O)=O)CCN(C(=O)CCC2CCCOC2)C1 75554,C1(NC(=O)CSC2CC2)CCN(C(=O)C(O)CC(F)(F)F)CC12CCC2 75555,C1(NC(C(CCC)=CCC)=O)CCC2CC1CN2C(c1ncccc1OC)=O 75556,Cc1nc2ccc(F)cn2c1C(N1CCN(Cc2ccc(Cl)nn2)C(CO)C1)=O 75557,C#CC1(O)CCN(C(C2CC2C2CN(C(=O)CC3CCOC3)C2)=O)C1 75558,Cc1cc(C(=O)N(CCCOCCNC(=O)CC2CC2(C)C)C)nnc1O 75559,C#CCC(C)C(=O)N(C1CCN(C(=O)CC2(C)CC2(F)F)C1)C 75560,c1(OC)cc(C(=O)NC2CCCC2CNC(=O)CCCN(C)C(C)=O)ccn1 75561,Cc1ncc(F)c(NC(C2CCN(Cc3cccc(CN(C)C)c3)CC2)=O)n1 75562,C1(CC(=O)NCCCC(C)NC(C(F)=CC)=O)CCC(C(N)=O)CC1 75563,Nc1nccnc1C(N1CCCC(CNC(c2csc(-c3cn[nH]c3)n2)=O)C1)=O 75564,c1(C(=O)NC2C(NC(=O)CCc3ccoc3)COC2)cc2c(Cl)cccn2n1 75565,C1(NC(Cc2cn(CC)nn2)=O)C=CCN(C(C2(CC3CC3)CC2)=O)C1 75566,C(=O)(C(C)(C)CCOC)N1CC(CNC(C(C)OCC)=O)C(N(C)C)C1 75567,C1(C(=O)NCC(CNC(CCNC(C)=O)=O)C)CCc2cc(Br)ccc2O1 75568,c1(CC)n[nH]c(=NC2CCCC(CNC(=O)C(C)CF)C2)s1 75569,c1(C2(C(N(CCN(C)C(c3cnsn3)=O)C)=O)CC2)ccn(C)n1 75570,C12(NC(c3cc(C)ncc3)=O)CCN(C(c3nc(C)ncc3Cl)=O)CC1C2 75571,c1(C(=O)NCCC2CN(C(c3ccccc3)=O)CC(C)O2)cccc2nncn12 75572,CCCC(C(=O)NCC(O)CC1CCC1)NC(=O)C(C)NC(C)=O 75573,Cc1ccc(C(=O)N(CC(C)NC(C2CC(O)C2)=O)C)c(-c2cnn(C)c2)c1 75574,C1(C)(CNC(C(CCC)C)=O)CC(F)(F)CN1C(=O)C(C(C)C)SCC 75575,c1(C(N2CC(NC(c3n(CC)nnc3)=O)C(C)C2)=O)nn(C)c(=O)cc1C 75576,Cc1ccccc1CN(C(=O)C(O)CCNC(=O)C=CCCC(C)C)C 75577,C(C)(N=c1cc(C)nc(CC)[nH]1)C1CCCN(C(c2ccnc(SC)c2)=O)C1.CO 75578,C#Cc1ccc(NC(C2CCCN2C(C2CCN(C)C2=O)=O)=O)c(C)c1 75579,c1(C(=O)NCC2C(NC(CCn3c(C(C)C)ncc3)=O)C2)cccn2ccnc12 75580,N1(CC(=O)NCC(=O)NC(C2CCOC2)C#C)CC(C(F)(F)F)CCC1=O 75581,C1(C#N)(C(N2CC(N(C)C)C2)=O)CC2(CC2)C1.C(=O)(CCC(=O)c1ccc(Cl)s1)N 75582,c1(OC)ccc(CC(N2CCC(NC(C3(N4CCOCC4)CC3)=O)C2)=O)cc1Cl 75583,N1(C(c2nc(C(=O)OC)oc2)=O)CCC2(C1)CN(C(c1ccc(Cl)cc1F)=O)C2 75584,c1(C(C)=O)ccc(Br)cc1NC(c1ccnc(-c2ccoc2)c1)=O 75585,CCC(CN=c1[nH]c(=NCCCOCCO)[nH]c2cc[nH]c12)C(C)(F)F 75586,n1(CCNC(CNC(=O)OC)=O)ccc(C(=O)NCC2CCC(C)C2)c1 75587,c1(C(=O)NC2CC(C(=O)NC(c3ccnn3C)CC)C2)cccc(F)c1C 75588,N1(C(CN(C)CC)=O)CC(NC(=O)CCC(=O)c2cc(C)sc2C)C(C)C1 75589,N1(C(CC(CCC)CC)=O)CCOC2(CCCN(C(=O)Cn3cnnn3)C2)C1 75590,c1(C(c2ccccc2)NC(C2CCCN2C(=O)C2CC2)=O)ccnc(F)c1 75591,C1(CNC(C2N(CC)CC2)=O)CN(C(=O)CC2COC(=O)N2)CC1C1CC1 75592,C1(CNC(CNC(C)=O)=O)CC(F)(F)CN1C(=O)COC1CCCC1 75593,N1(C(c2ccc(-c3cn(C)nc3)o2)=O)CC2CC2(NC(=O)CCc2cc[nH]n2)C1 75594,CC(CC(C)(C)C)C(=O)N1CCCC(N(C(=O)CCn2ccccc2=O)CCF)C1 75595,c1(-c2nc(-c3ccc(F)cc3)nn2CC2CCCOC2)cncc2cnccc12 75596,Cc1nc(O)c(C(=O)NCC23CC(CN2C(=O)CC(O)C(C)C)C3)nc1C 75597,CC1(C)CCCC1(CO)NC(=O)NCCCC1CCCCO1 75598,c1(C(=O)NC2C(NC(C=CCOC)=O)CCCC2)ccc(N)cc1C 75599,N1(c2nnc(C3(C)CCCNC3)n2CCN2CCCC2)CCOC2COCC12 75600,N(C1COCc2ccccc21)C(C1N(C(=O)C(c2ccccc2)O)CCC1)=O 75601,c1(C(N2CCC(OC)(CNC(C3CSC3)=O)CC2)=O)ccc2c(c1)COB2O 75602,N#Cc1nc[nH]c1C(=O)NCC1CC1NC(C1(C(F)(F)F)CCCC1)=O 75603,S(=O)(=O)(c1c[nH]c(C(=O)NC2CC(NC(C3CC(OC(F)F)C3)=O)C2)c1)NCC 75604,n1(CC(=O)NCCN(C(C2CC=C(C)CC2)=O)C)nc(C)c2cccnc12 75605,c1(C(=O)NCC(C)N(C)C(c2cccc(N)c2N)=O)cc2sccc2cn1 75606,c1(C(=O)NC2CC(CNC(c3c(C)nccc3)=O)C2)cn2ncccc2n1 75607,C1(c2n(CC)cnn2)CN(C(C2CCCN(C(=O)C(=O)NC)C2)=O)CCO1 75608,c1(CC)cc(C(N2C3CCC2(CNC(=O)C(C)C(C)CC)CC3)=O)cn(C)c1=O 75609,c1(C(=O)NC(CC=C)CNC(c2nccnc2N)=O)cn(C)c(=O)cc1C 75610,N1(C(C(C)NC(=O)CC(F)(F)F)=O)CCC(C2(NC(=O)CNC=O)CC2)C1 75611,N1(C(=O)COC2CC2)CCC2CC12C(=O)NCC1(CC2CC2)CCC1 75612,C(=O)(C(CO)C(C)(C)C)NC1CCC(NC(C(C)(C)N(C)C)=O)C1 75613,C1(C(=O)N(CCCC(C)C)C)CCn2cncc2C1.C1=CCNC1=O 75614,c1(SCC)nccnc1C(=O)NC1CC(C)N(C(=O)CC2CCC(C)C2)C1 75615,C1(C2CCN(C(c3ccccc3Cl)=O)C2)(NC(=O)Cc2ccns2)CC1 75616,C1(C(N2CCN(CCNC(C3(C)CCC3)=O)CC2)=O)CCCS(=O)(=O)N1 75617,Cc1nc(N2CCC(c3ccccc3)C2C)cnc1N 75618,C1(CN(C(=O)CCOc2ccccc2)C)C2CN(C(=O)CC3(O)CCCOC3)CC12 75619,c1(C(=O)NC(C2CC(NC(c3nocc3C3CC3)=O)C2)C)cncn(C)c1=O 75620,CC(C)(C(=O)NCC12CC(NC(=O)Cc3coc(C(F)F)n3)(C1)C2)C1CCC1 75621,c1(C(=O)NCCN(C(CC2C(OCC)CC2)=O)C)cc(C(C)(F)F)on1 75622,N1(C(C2(C#C)CC2)=O)CCN(C(C)CNC(=O)C(C)C#N)CC1 75623,CC(C(=O)NC1CCCC(CNC(c2ncc[nH]c2=O)=O)C1)C(F)F 75624,CC1CN(C(=O)CC(C)(C)N(C(=O)C(C)(Cl)Cl)C)CCC1N(C)C 75625,C(=O)(C(CN(C)C)SC1CCCO1)NCC(=O)OCC(=O)NC(CC)C1CC1 75626,CC1CC(=O)NC1C(=O)NCC(C)(C1CC1)NC(=O)CCN1CCOC1=O 75627,C(=O)(C1CCCc2ncc(C)n21)NCC(CNC(c1cc(C(N)=O)c[nH]1)=O)OC 75628,C12(CNC(=O)C(O)C3CCC3)CC(CO1)N(C(C1(c3ccncc3F)CC1)=O)C2 75629,CS(=O)(=O)c1cnc(N2CCC(N(C3CCC3)C(C3(S(C)(=O)=O)CC3)=O)C2)c(Cl)c1 75630,Cc1cccc(NNC(=O)NCCCN(C)C(C)C)c1C 75631,Cc1cc(C(N2CC3(C2)CN(C(c2cc(C4(Cl)CC4)n(C)n2)=O)C3)=O)cc(O)n1 75632,N1(C(C(C2CC2)SC)=O)CCC(C2CC(NC(c3c[nH]c(=N)s3)=O)CCO2)CC1 75633,c1(OC)cc(C(=O)NC23CC(C2)N(C(C2(CC4CC4)CCCO2)=O)C3)ccc1Cl 75634,C(CC(C)C)(C(=O)NC(C)CCN(C)C)NC(CC=CCCCCC)=O 75635,Cc1cccc(C)c1C(=O)NC1CCCN(C(c2cnc(C3CCC3)s2)=O)CC1 75636,C1(C(F)F)(NC(CC2(C#N)CC2)=O)CC(NC(=O)CC2CCCSC2)C1 75637,CCCC(C#N)C(=O)NCC1CCN1C(c1ccc(CN(C)C)nc1)=O 75638,CC1(C)CCC(C)(NC(C2CCCN(C(c3[nH]nnc3C3CC3)=O)CC2)=O)C1 75639,c1(CC)cccc(C(=O)NCCC(CC)(CC)NC(C2CCOC2C)=O)c1N 75640,c1(NC(C)=O)ccc(F)c(C(=O)NC2(CNC(c3cc(Br)co3)=O)CCC2)c1 75641,c1(OC)ccc(CN=C(NCC(=O)NC(C)C)N(C)CC2CCCS2)cc1O 75642,c1(CC(N2CCC(C(C(=O)NC3CC(CC)C3)C)C2)=O)coc2ccccc12 75643,C(=O)(C1=CCCCO1)N(CCCC(=O)N(C(C1CCC1)C)C)C 75644,C1(NC(C2C(C=C)C2)=O)CC(C)CN(C(c2cc(C)cc(O)n2)=O)C1 75645,C(CC(C(=O)N1CCC(O)(N(C(=O)CSCCN(C)C)C)C1)N(C)C)SC 75646,c1(OC)c[nH]c(C(=O)N(C)CC2(O)CCN(C(=O)CC3CCC3(F)F)C2)cc1=O 75647,N1(C(C(SC)SC)=O)CCC(C(=O)Nc2cn(CO)nc2C#N)CC1(C)C 75648,c1(CC)nc(=N)[nH]cc1C(N1CCC(CF)(NC(c2cnns2)=O)C1)=O 75649,C1(C)(C(=O)OC)CC(C(=O)NC(C)(CNC(=O)C(C)N2CCCC2)CO)C1 75650,C(=O)(CC(CCCC)NC(c1ccoc1C1CC1)=O)NCC(C=C)O 75651,N1(C(C(C)(C)F)=O)CC2CCN(C(=O)CC3CCCCC3(C)C)CC2C1 75652,C(=O)(C(F)(F)C(O)C1CC1)NC(C1(O)CCN(C(C2CC(n3cccn3)C2)=O)C1)C 75653,C(=O)(C(C)(CC)C(N)=O)N(CCCNC(C1(c2ccccc2)CCOC1)=O)CC 75654,C1(NC(=O)CCN2CCC(F)C2)(CF)CCN(C(C2CC(CC3CC3)C2)=O)C1 75655,CC1(C)CN(C(=O)Cc2csc(Cl)c2)CC1NC(=O)CC1CCOC1=O 75656,C1(NC(C(CCOC)C)=O)CCC2(CC1)CC(NC(=O)CSc1cccs1)C2 75657,C1(Cc2cnc(C)cn2)C(C)CCCN1C(=O)NCC=CCSC 75658,N1(C(CCn2ccc(C)n2)=O)CCC2(CCC2)C(NC(=O)C(C)CC2CC2)C1 75659,N1(C(c2oc(C)c(Br)c2)=O)CCC(NC(C2CC23CCC3)=O)C12CCC2 75660,c1(OC)cncc(C(N2CCC(C(N3CCC(C)(CCO)C3)=O)(OC)C2)=O)c1 75661,Cc1nc(C(=O)NC(CNC(C2CC2C2CCC2)=O)CO)ccc1[N+](=O)[O-] 75662,N1(C(C2(C#C)CCC2)=O)CCCN(C(=O)C(C)C(C)C)C(CO)C1 75663,Nc1cc(Cl)nc(C(=O)NC2CCC(CNC(c3cccnc3S)=O)C2)c1Cl 75664,c1(CC)cc[nH]c1C(=O)NCCOCCCN(C)C(C1(C)CC1(Cl)Cl)=O 75665,CC1(NC(c2ccco2)=O)CN(C(=O)CCCNC2(c3ncco3)CCC2)C1 75666,Cc1cc2ccc(C(=O)NC3CC(C)CN(C(c4sc(C)nc4C)=O)C3)cn2c1 75667,c1(C(=O)NCC2CC(NC(=O)C(=C3CCCCC3)F)C2)cnc2ncccc2c1 75668,N1(C(=O)NCC=CC=CC)Cc2nc(O)nc(O)c2C1 75669,C1(CC)CN(Cc2cc(O)ccc2Cl)c2ccccc2O1 75670,N1(C(C(C(C)(C)C)=O)=O)CCCC(O)(CNC(=O)CCC2CCCO2)CC1 75671,C12(NC(C(N3C(CC)CCC3)=O)=O)CCCC1(F)CN(C(c1cncn1C)=O)C2 75672,N1(C(C2(CCC)CC(=O)C2)=O)CCCC(C(C)C(=O)NCc2ccc(C)cc2)C1 75673,CN1CCN(CCc2nc(-c3cccs3)nn2CC2CCOCC2)CC1 75674,Cc1cccc(NNC(=O)C2(n3cc(N(C)Cc4ccccc4)nn3)CC2)c1Br 75675,c1(C(=O)NC2(C3N(C(C(C)OCC)=O)CCC3)CC2)ccc(CC)c(O)c1 75676,n1(CC(C)OC(=O)Nc2ccccc2)cc(COC(=O)C(C)OC(C)(C)C)nn1 75677,N1(C(C(C)CCO)=O)CCC(C)(NC(=O)COc2cccc(F)c2)CC1 75678,C1(N(C(=O)CS(C)(=O)=O)C)CN(C(=O)CSCCC#N)CC12CC2 75679,N1(C(=O)C=CC(=O)NF)CC2CC1CCC2NC(C1(Oc2ccccc2)CC1)=O 75680,N1(C(C2(COC)CCCCC2)=O)CC(C2CCCN(C(=O)C(C)S(N)(=O)=O)C2)C1 75681,C1(C(N(C2CCN(C(C(CC)(C)C)=O)CC2)C)=O)(CF)CC2(CCC2)C1 75682,c1(C(=O)NCC(CNC(=O)CCc2ccoc2)F)ccn(-c2ccncc2)n1 75683,C(=O)(CCC(C)c1ccccc1)N(CCCN(c1snc(CC)n1)C)C 75684,c1(N(C(CNC(C(C)CC(N)=O)=O)C)C)nc2c(cc1C#N)CCC2(C)C 75685,N1(C(CCC(C)OCC)=O)CC(NC(c2cc(OC)n[nH]2)=O)CC(C)C1 75686,CC1CCC(C)(C)N1C(=O)CC1CC(NC(C2CC2C(C)(C)C)=O)C1 75687,C(=O)(CC1=NNC(=O)C1)NC1C(CNC(C(C)CC2CCC2)=O)CC1 75688,N1(C(C2C(C)CC2)=O)CCOC(C(N2CCCC2C(N)=O)=O)C1 75689,CC(C)CC(CNC(=O)C(c1cccnc1)O)NC(c1cccc(C(C)C)c1)=O 75690,CC(C)(CNC(=O)CNC(c1cscn1)=O)Cn1cccn1 75691,c1(C(N2CC3(CCN(C(C(C)N(CC)CC)=O)C3)C2)=O)nc2nccc(C)n2n1 75692,C(CN=c1[nH]c2c(c(=NCc3conc3C3CC3)[nH]1)CCCC2)c1nc(C)sc1 75693,c1(OC)cc(C(F)(F)F)nc(N2CC(NC(=O)CC3CC(C)OC3C)CC2C)n1 75694,Cc1cc(=NCC(CC(C)C)ON2CCCC2)[nH]c(Cl)n1 75695,C1(CNC(c2oc(CC)c(C)c2)=O)COC(C)(C)CN1C(=O)CN1CCCC1=O 75696,N1(C(C2C(C)(Br)C2)C(=O)NCC2CC2)CCC23CCCCC2(C1)C3(F)F 75697,c1(C(NC(=NCCCC)NCCCC2(O)CCC2)C)ccc(S(=O)(=O)CC)cc1 75698,C1(C(=O)NC(C)CCN(C)C(c2cnsc2)=O)C2CC2CN1C(=O)OC(C)(C)C 75699,C1(CNC(c2ccco2)=O)CCC12CCN(C(=O)Cc1ccc(F)cc1)CC2 75700,CC(CS(C)(=O)=O)C(=O)N(C)CC1CCCN(C(c2csnn2)=O)C1 75701,C1(CNC(CCC(C)SC)=O)CN(C(=O)Cc2ccnn2C)C2CCCCC12 75702,Nc1cc(C(=O)NCC23CC(NC(=O)C(O)CN4CCCC4)(CO2)C3)ccc1F 75703,C(=O)(CC(C)C(C)(C)C)N1CCC(C(C)CNC(=O)Cn2cnc(C(F)(F)F)n2)C1 75704,CC1CN(C(c2ccc(Cl)[nH]2)=O)CCN1C(C1CC(CC(F)F)C1)=O 75705,C1(NC(COC)=O)CC2(C1)CN(C(=O)CNC(c1ccc(Br)cc1)=O)C2 75706,c1(C(=O)NCC2N(C(c3cccc(C)c3C)=O)CC(O)C2)cc2c[nH]cnc-2n1 75707,Cc1cccc(C(CNC(=O)CCCn2ccnc2C)NC(C2CCO2)=O)c1 75708,C(=O)(CC(O)CC(C)C)N1C(CC)C(NC(=O)CCCC(F)F)CC1 75709,c1(CNCc2nc(C(C)(C)C)sc2)cc(I)ccc1F 75710,C12(CNC(C(C)(C)SC)=O)CC(CCO1)N(C(=O)Cn1cnnc1O)C2 75711,C1(NC(C2(C=C)CCN(C(=O)C(CCC)OCC)C2)=O)CN2CCC1(F)CC2 75712,C(c1cccs1)=C(C)C(=O)N(C(C)CNC(=O)CCn1ccnn1)C 75713,N1(C(C2=CCCCC2C)=O)CCN(C(=O)CCc2cncnc2)C2(CCC2)C1 75714,Nc1nc(C(=O)NCC2CC2CNC(c2cc(Cl)ns2)=O)ccc1[N+](=O)[O-] 75715,N1(C(CCCC#CC)=O)CC(NC(c2ccc(OC)nc2C)=O)CC12CCOC2 75716,Cc1nnc2n1C(C(=O)NC1(CCNC(=O)Cc3ccc(F)c(F)c3)CC1)CC2 75717,N1(C(Cc2cccc(OC)c2)=O)CCCC(NC(C2CC(N(C)C)C2)=O)CC1 75718,Cc1ccc(NC(=O)CN(C(=O)CNC2CC(=O)N(C)C2=O)C)cc1C 75719,c1(OC)cc(=O)n(C)cc1C(=O)NCC1(F)CN(C(C2CC3CCC(C2)C3)=O)C1 75720,C1(NC(=O)CC2CC(F)(F)C2)CC2CC1CN(C(c1cccc(CO)c1)=O)C2 75721,N1(C(CC2N(C)CCCC2)=O)CC2CCCC1C2CNC(=O)CCCC1CCC1 75722,N1(C(C(COC)C)=O)CCC(CO)C(NC(c2ncc(F)c(OCC)n2)=O)C1 75723,C1(CNC(=O)CC2CCCC2(F)F)CC2(CO1)CN(C(c1cccc(=O)o1)=O)C2 75724,C1(C(=O)NC(C2CN(C(=O)C(n3ccc(C4CC4)n3)C)C2)C)CCCC1(F)F 75725,c1(CO)ncnc2c1CCCC2.C12CC3CC1N(C3)C(=O)c1ccc(o1)C(=O)N2 75726,CCCC(C)(C)CC(=O)NC1CC2CCC1CN2C(=O)C=CC1CCOCC1 75727,N1(C(c2nn(CC)c(C3CC3)c2)=O)CC(NC(c2ccnnc2)=O)CC2(CC2)C1 75728,N(C1CCc2ccccc21)C(CC(C)CNC(c1nsnc1O)=O)=O 75729,C1(C(=O)NC(CNC(c2cnc(C(C)OC)s2)=O)(C)C)CCc2n[nH]c(C)c2C1 75730,CS(=O)(=O)C1CC(CN)C1.C1(=O)C(F)(F)C2(CCC2)N1 75731,c1(C(C)C)cccc(F)c1C(=O)NCCC(C)NC(c1cnc(Cl)[nH]1)=O 75732,C1(CNC(C2C(C)(C)CC2)=O)(NC(C2CCC=CCC2)=O)CCOCC1 75733,c1(C(=O)NCC2C(NC(c3ccc(Cl)s3)=O)CCC2)coc2c1C(O)CCC2 75734,c1(N2CCC(CN)CC2)nc(N2CCN(c3ccncn3)CC2)c2c(n1)CCS2 75735,C(=O)(C(C)(C)COCC)NC12CC(NC(CCC)=O)(C1)C2 75736,C1(NC(c2cnn(CCN(C)C)c2)=O)CCCN(C(C2(CF)CC2)=O)CC1 75737,C1(CC(=O)N(C)CC2N(C(CCC(=O)N(C)C)=O)CCCC2)CCCCC(=O)N1 75738,N1(C(C2(C)CCCN(C)C2)=O)CCC2(C=C(C(=O)NC3CCCC3C(N)=O)C2)C1 75739,Cc1cn2nc(C(=O)NCCCNC(c3n[nH]cc3C)=O)cc2c(=O)[nH]1 75740,N1(C(CC2N(CC)CCC2)=O)CCN(C(C2(F)CCC2)=O)CC1c1nccn1C 75741,CC(CN=c1[nH]c2c(c(=NCCn3cc(Br)nn3)[nH]1)CCC2)c1ccc(Br)cc1 75742,c1(CS(=O)(=O)CC)ccc(Cl)c(OC)c1F.C12CCC(C)N(C1)CC2=O 75743,c1(CCC(=O)NC(C)(CNC(=O)C=Cc2cn[nH]c2)CO)cccc(O)n1 75744,Cc1ccc(C(=O)NCC(=O)NC(C)CCNC(C2CC(=C3CC3)C2)=O)c(F)c1 75745,C(=O)(CC1=NNC(=O)C1)N(CCCCCCNC(c1c(OC)cc(Cl)cc1)=O)C 75746,c1(C(=O)NCCCCCN(C(C(C(C)C)C)=O)C)ccnc2ncnn12 75747,Cc1cncc(C=CC(=O)NCC2(CNC(=O)Cc3ccsc3)CC(F)(F)C2)c1 75748,CC(C)C(O)CC(=O)NCC1CCN(CCOc2c(Cl)cccc2Cl)CC1 75749,C1(C2CCN2)(NCSC23CCC(C(CCC)CCC)C2C3)CCCN1.N1CCC1 75750,c1(N(C2CC3CCC(C2)N3)CC2(S(C)(=O)=O)CCC2)ncnc2[nH]cnc12 75751,C(N(Cc1ccccn1)N1CC2CC1C1OC(C)(C)OC21)C1N(C)CCCC1 75752,C1(NC(c2cnc(CC(C)C)[nH]2)=O)CCCC12CN(C(c1cc(Cl)ccn1)=O)C2 75753,C12(NC(C(C)S(N)(=O)=O)=O)CCCN(C(c3cnn(C4CC4)c3)=O)CC1C2 75754,C1(C(N2C3CC(CNC(C4CN(C(C)C)C4)=O)(OC3)C2)=O)CCCCCS1(=O)=O 75755,Cc1ccc(F)c(C(=O)NCC2(CO)CCCN(C(c3cc(C)c(C)o3)=O)C2)c1 75756,N1(c2c(OC)cncn2)C2CCC1CC(NC(=O)C=Cc1scnc1C)C2 75757,c1(C(N(CCN(C(=O)CC(C)C2CCCO2)C(C)C)C)=O)nc2cnccc2s1 75758,c1(C(=O)NCCC2(NC(C(CC=CCC)C)=O)CC2)ccc(Cl)nc1OC 75759,C1(CC(=O)NCC(CCOC)NC(C(C)SCC)=O)(COC)CCOCC1 75760,C(=O)(C1SCCc2sccc21)N(CC(C)(C)CNC(=O)CCc1nccs1)C 75761,c1(C(N2CCN(C(C(CC)SC)=O)CC2)=O)ccc2nc[nH]c2c1 75762,C1(C)(C(C)C)CN(C(C2COCCN(C(C3(N=[N+]=[N-])CC3)=O)C2)=O)CCO1 75763,C=CCCCCC(=O)N1CC(CCNC(=O)CN2CCC(C)C2)C1 75764,C1(NC(C(N2CCN(C)CC2)C)=O)CCN(C(=O)CCCC2CC2)C1C1CC1 75765,c1(CN2C(C(N3CCCC3c3ccc(Cl)s3)=O)CCC2)ccc2ncsc2c1 75766,C(=O)(CC(C)C(=O)NC1CN(C(c2cn(CC(F)(F)F)nn2)=O)CC1(C)C)OC 75767,Cc1c(CC(=O)NC2CCCC(NC(=O)C=CC(C)C)C2)nnn1C1CCOC1 75768,c1(N2CCC(CC)(CO)C2)ccc(Br)c(S(=O)(=O)NC(C)C(C)(C2CC2)OC)n1 75769,C1(C)(C(N2C(C3(NC(C4C(C=C)C4)=O)CC3)CCCC2)=O)CCN(C)C1=O 75770,N1(C(C(C(C)C)O)=O)CCN(C(C2CCC(O)CN2C)=O)C(CCO)C1 75771,c1(NC(C2C3CN(C(c4ccc(O)c(O)c4Cl)=O)CC23)=O)cc2cccnc2[nH]1 75772,C(N=c1[nH]c(N2CC=C(C)CC2)nc2c1CCCCC2)c1c(OC)c(Cl)ccc1 75773,C(C)(C)(CCN=c1[nH]c(N(C)Cc2nccn2C(F)F)nc2c1SCC2)OC 75774,C1(F)(CNC(=O)CCc2ccncc2)CCC(CNC(C2(F)CCOC2)=O)C1 75775,N1(C(c2c(OC)nccc2)=O)CCC2CN(C(=O)COC3CCCC3)C2C1 75776,C1(Cn2cc(C3CCCN(C(c4c(C)ccs4)=O)C3)nn2)CCCCC1(F)F 75777,N1(C(=O)NCC#C)CCC(N(CC(O)CC)C)C1 75778,c1(C(N2CC(O)(CNC(C(CSC)O)=O)C2)=O)ccc(Cl)cc1O 75779,C12(C(N3C(C)CN(C(=O)CN4CCC(O)CC4)CC3)=O)CCN(C1)S(=O)(=O)C2 75780,c1(C(=O)NCCC2CC(NC(=O)CC3=CCCC3)C2)c(F)cccc1[N+](=O)[O-] 75781,c1(CNC2C(C(=O)NCC3(C)CCCC3)CCCC2)ccc(OCF)nc1Br 75782,C(=O)(C(F)CC(C)(C)C)NCc1nn(C)c(C(N2CCC(c3ncc[nH]3)C2)=O)c1 75783,N1(C(C(c2ccnn2C)NC(C(CC)O)=O)=O)CCCC(C2CC2)CC1 75784,C=C(C)CC(=O)NCCC(C)NC(C1CC(OC(F)(F)F)C1)=O 75785,C(CC(C)(C)CNC(=O)C(C)CNC(=O)CC1CCC(=O)N1C)OC 75786,C1(C(=O)NC(C)(CNC(=O)CC2CCCCC2)CO)CCCCS1(=O)=O 75787,Cn1ncc(CNC(=O)CCc2ccccn2)c1C(=O)NC(CC1CCC1)CO 75788,N1(C(C2CC(OC)(OC)C2)=O)CC2COCC2(C(=O)NC2CC(F)(F)C2)C1 75789,c1(CC)c(C(=O)NCC=CCNC(=O)C(c2cccc(F)c2)(C)C)ccn1C 75790,C(=O)(C1=CC2CCC(C1)C2)N1CCCN(C(C(CCC)c2ccccc2)=O)C(C)C1 75791,c1(-c2nc(CNC(C(C)OC)=O)sn2)ccc(Br)cc1 75792,C1(NC(=O)OC(C)(C)C)CC(Cc2cn(CN3CCNC3=O)nn2)C1(C)C 75793,C1(NC(C2OCCCO2)=O)CN(C(c2ccc(C(F)(F)F)o2)=O)CC12CCC2 75794,CN1CCN(C(c2ccccc2C2CCC2)=O)C(CNC(c2c[nH]nc2Cl)=O)C1 75795,c1(NC(C(CO)NC(c2cnc(OC)nc2)=O)=O)ccc(C#N)cc1O 75796,S(=O)(=O)(c1nc(N2CCC(COC)C2)ccc1Br)NC1(CC=C)CC1 75797,c1(C(=O)NCC2N(C(c3[nH]c(=NC)sc3)=O)C3C(C2)C3)ccc2c(c1)CCOC2 75798,c1(NC2CC(CNC(C3=NOC(C)C3)=O)C2)c([N+](=O)[O-])cnn1C 75799,C12(C(=O)NCc3c(C4CN(C(c5ccn(C)c5)=O)C4)ocn3)CCC(CC1)C2 75800,CC(C)CC(CNC(=O)Cc1ccsc1)NC(C12CC(CC(F)F)(C1)C2)=O 75801,C(CN=c1nc(NCc2ccc(Cl)s2)c2c([nH]1)c(C)nn2C)c1ccc(C)cn1 75802,c1(CCC(=O)NC(C(=O)N2CC(C(C)OC)C2)CO)cccnc1 75803,c1(C(N(CCC(C)NC(c2ccc(CCC)s2)=O)C)=O)ccn(C)c1C1CCC1 75804,C(=O)(C1=NN(C(C)C)C(=O)CC1)NC1CCN(C(C(CC#C)O)=O)C1CC 75805,C(=O)(C(C)(C)CNC(C1CCN(C(=O)COC2(C)CCC2)C1)=O)NC 75806,CCC(C)(CCC(C)C)C(=O)N1CC(O)CC1C(=O)NCc1cccc(Cl)n1 75807,N1(C(C2(CCOC)CC2)=O)CC(CNC(=O)CC2CCCO2)OC(C)(C)C1 75808,C(=O)(CCC(C)C)NCCCN(CCCNC(c1c(CCC)nns1)=O)C 75809,c1(C(N(C)CC2OCCN(C(C=NOC)=O)C2)=O)cccc([N+](=O)[O-])c1NC 75810,C1(CC=C)(C(=O)NCC2(CO)CCCO2)CCCN1C(=O)C(C)CC#N 75811,c1(C(=O)NC(c2ccccc2Cl)C)nc2ccccn2c1-c1ccoc1 75812,Cc1cc(C(=O)NC2C3CC(NC(=O)C(O)c4ccsc4)CC23)nc(C)c1 75813,CC1Cc2ccc(F)cc2C1Nc1ccnc2[nH]cc(Cl)c12 75814,C1(NC(C(Cc2ccsc2)NC=O)=O)CCOC(CNC(c2cc(Cl)no2)=O)C1 75815,N1(C(C2C(c3onc(C(C)C)n3)C2)=O)CCC(F)C(F)C1 75816,N1(C(c2c(OC)scc2)=O)CC(NC(=O)COCC2CC2)CCC1C 75817,C1(C(=O)Nc2ccnnc2O)CN(Cc2cccc(Br)c2Cl)CCC1O 75818,c1(C(N2CC(NC(C3ON=C(CC)C3)=O)C(C)C2)=O)cccc2c1CCC(=O)N2 75819,S(=O)(=O)(c1cnc(NCCCOc2cncc(Cl)c2)cc1C)NCCC(=O)NC 75820,N1(C(=O)Cn2cncn2)CC2CCN(C(=O)C3=CS(=O)CCC3)C2C1 75821,C(=O)(C(O)CC(C)C)NC1N(C(C2CC(OC)C2)C(=O)NCC(C)C)CC1 75822,c1(C(N2CCN(C(CC3(C=C)CC3)=O)CC2CCC)=O)ncn2c1COCC2 75823,c1(CC(C)OCC)noc(CS(=O)(=O)CC2CC2(Cl)Cl)n1 75824,C1(O)(CNC(C(CC2CC2)OC)=O)CCCN(C(c2ccc(C)cc2)=O)C1 75825,N1(C(=O)OC(C)(C)C)CCCC(NC(=O)Cc2cn[nH]c2)C1.C12CCC(C1)N2 75826,N1(C(=O)Nc2ccc(C)cc2I)CC2(CCCC2)C1C(C)C 75827,C1(CNC(CCC#C)=O)CC2CC1CN2C(c1ccnn1CCN(C)C)=O 75828,Cc1ccc(C(N2CCCC(C(=O)NC3(C)CC(C(=O)O)C3)C2)=O)c(Cl)n1 75829,C(=O)(C(C)(O)CC(F)(F)F)NCC1OCCN(C(CCCCC(C)C)=O)C1 75830,C(=O)(C(C)(C)CC(C)(C)C)Nc1scc(C)c1.N12CCC(C1)OCC2=O 75831,c1(C(=O)NC23CN(C(c4cc(C)cc(F)c4)=O)C(C2)C3)ccc2nc[nH]c2c1 75832,c1(CC(N2CCC2)SCC)ccccc1.C(=O)(CN(CC(=O)NC)C)NC(C)C 75833,Cn1cnc2c(C(N3CCC(CNC(C4CCC5CC45)=O)CC3)=O)[nH]nc2c1=O 75834,N1(C(C2C(C)C2)=O)CCCC(CCNC(=O)CS(=O)(=O)Cc2ccccn2)CC1 75835,Cc1c(N(C)CCN(c2ccccc2Cl)C)ncnc1N1CCCC1 75836,C1(C(=O)NCC2CCCC(OC)C2)N(C(c2n[nH]cc2C)=O)CCC1(C)C 75837,c1(C(=O)NC(CC)CNC(c2cc(C(F)F)[nH]n2)=O)cnccc1C1OCCO1 75838,Cc1ccn(CC(=O)N(CCCCNC(=O)CSC(C)C)C)n1 75839,N1(C(=O)Cc2ccoc2)CC2CC1CCN2C(=O)C(O)Cc1ccccn1 75840,c1(OCC)ncccc1C(=O)Nc1cccc(NC(C2CC(O)C(F)C2)=O)c1 75841,Cc1ccsc1C(=O)NCCCCN(C(=O)C(c1cccnc1)N(C)C)C 75842,c1(C(=O)NCC(C(C)C)NC(c2cn(CC)nn2)=O)nc2nc(C)cc(C)n2n1 75843,Fc1ccc2c(c1)N(Cc1ccc(Cl)[nH]1)CCO2 75844,Cc1ccc(C(=O)NC2CN(C(C3(CCF)CCC3)=O)CC23CC3)cc1O 75845,c1(C(N2C(CNC(C(C)(C)OC)=O)CCC2)=O)cccnc1I 75846,C1(OCC)CCCC1C(=O)NCC(F)(F)Cn1cc(CCS(N)(=O)=O)nn1 75847,c1(N(c2n(CC=C)c(-c3scnc3C)nn2)C)ccc(OCCCC)c(Cl)c1 75848,N1(C(C=CC)=O)CCN(C(=O)C=CC2CCC2)C2CCCCC12 75849,N1(C(C2C(C)C2)=O)CC2CC1C2CN(C(c1ccccn1)=O)Cc1ccccc1 75850,C1(C(=O)NC2CCN(C(Cc3n(C)ccn3)=O)C2)CCc2ccccc2C1O 75851,C1(N(CCCCC(N2CCCC(C)C2)=O)CCC#N)COC2(CCCCC2)C1 75852,C1(CCN(C)Cc2nnsc2Cl)CCN(C(=O)CCCC2CCCC2)CC1 75853,C1(C(N(C(C)CN(C(=O)CCC2CCCC2)C)C)=O)CCC(=O)N1C1CC1 75854,c1(C(=O)NC(CCCNC(CCCCOC)=O)C)cc(Cl)cc(Cl)c1N 75855,c1(CC(=O)N(CC(C)(C)NC(=O)CC2CC2(Cl)Cl)C)ccccc1OC(F)F 75856,Cc1ccc(CC(N2CCN(C(=O)C(C)Cc3ccccc3)CC2C)=O)cc1F 75857,c1(CC)ccccc1CC(=O)NCC1(NC(C2CCCCC2O)=O)CC1 75858,N1(C(c2ccc(C)cc2O)=O)CC(F)(F)CC1(C)CNC(=O)C(C)C(C)(C)C 75859,Cc1ccccc1CC(=O)NCC(O)CNC(=O)C=Cc1csc(Br)c1 75860,C(=O)(C(O)CCC(C)C)NC1CN(C(C2(c3c(C)cccc3)CC2)=O)C1 75861,c1(CC)cc(C(N2CC(CCn3cc(-c4ccc(Cl)s4)nn3)C2)=O)n[nH]1 75862,c1(NC(=O)Cc2ccns2)ncnc2c1CCC2.C12CCCCC1CNC2=O 75863,c1(C(=O)NC(CCOC)CNC(=O)C=C(Cl)Cl)cn(C)c(=O)c2ccccc12 75864,C1(CC(=O)N(CCN(C(=O)CC(C)n2cccc2)CC)CC)CCCC(F)(F)C1 75865,Cc1c(C(N2CC(C3(NC(=O)CSCCN(C)C)CC3)C2)=O)cncc1Cl 75866,N1(C(CSCC=C)=O)CCC2OCCN(C(c3cc(C)cnc3C)=O)C2C1 75867,Cc1ccc2cccc(C(=O)Nc3ccnc4ncnn34)c2n1 75868,N1(C(CCCCNC(N)=O)=O)CC(C2CCCN(C(c3ccc(F)cn3)=O)C2)C1 75869,c1(C(CNC(C2(F)CCC2)=O)NC(c2coc(Cl)n2)=O)ccccc1F 75870,Cc1nc(C)n(CCC(N2CCC(N(CCO)C(C3CC(C)(C)O3)=O)C2)=O)n1 75871,C1(NC(CC2(CC(=O)OC)CC2)=O)CCCN(C(c2ncc(OC)cc2F)=O)C1C 75872,C1(OC2(C(N3CC(OCC)C3)=O)CCN(C(=O)CC3CC3)C2)CN2CCC1CC2 75873,C1(COC)(NC(C2CCC2C(=O)OC)=O)CCN(C(=O)CSc2ccncc2)C1 75874,C1(C(N2CC(C(C)C)OCC2)=O)CC(C)CN(C(=O)C(C)(C)CC#N)C1 75875,c1(C(=O)NCCCCN(C)C(C2CC(N(C)C)C2)=O)[nH]nnc1-c1ccnn1C 75876,N1(C(C2(SC)CCC2)=O)CCCN(C(C2CCN2S(C)(=O)=O)=O)C(C(C)C)C1 75877,N1(CCNC(C=CCN(C)C(c2cnc(Cl)s2)=O)=O)CCCOC1=O 75878,C#CCC(CC(=O)NCC1(CCO)CCCC1)NC(C1(C)C=CCCC1)=O 75879,Cc1n[nH]c(=NCC2CC(C)N(C(c3cc[n+]([O-])cc3)=O)C2)s1 75880,S(=O)(=O)(c1cc(C(C)C)cc(Br)c1)Nc1ncc(-c2ccc(C)cc2)s1 75881,Cc1cc(Br)c(F)cc1CN1CC2C(C1)N2C(=O)C(C)(C)CCl 75882,C1(CC)CN(C(=O)CC2CC3(CC3)CO2)CCC1NC(=O)CS(=O)(=O)NC 75883,c1(C(=O)NC(C)CCCNC(C2(O)CCSC2)=O)ccc(CCNC(N)=O)cc1 75884,Cc1ccc(C(c2nnnn2CC(F)F)NCCCCc2ccccc2)cc1Br 75885,c1(C(=O)NCC2(CCO)CN(C(C3CC3C3CCCO3)=O)C2)cc(COC)on1 75886,n1(CC(C)NC(C(c2ccccc2)OC)=O)cc(C(C)NC(C)=O)nn1 75887,CC1CCCC(N(C)C(c2ccc(CNC(=O)CCCC3CCC3)s2)=O)C1 75888,N1(C(CC=C=C)=O)CC2CCC1CN2C(=O)CCc1cc(F)c(F)c(F)c1 75889,N1(C(C(C)=CC2CC2)=O)CC(CNC(c2c(C)ncnc2C)=O)CC(C)(C)C1 75890,Cc1cnc(-c2nc(COc3cc(F)cc(F)c3)nn2CCCCO)cc1Cl 75891,C=CC(C)(C)C(=O)NCCN(CC(C)O)C(C1CC1C)=O 75892,c1(C(N(C(CCNC(c2nn(CC)c(=O)cc2)=O)C)C)=O)cc[nH]c2nccc1-2 75893,C1(NC(CCC2C(C)(C)C2)=O)CCC(NC(=O)C(O)C2CCCC2)CC1 75894,C1(C(=O)NCC2N(C(C(C)OC3CCCC3)=O)CC2)CCCN1C 75895,c1(C(N2CCC(NC(C(F)=CCC)=O)C(F)C2)=O)c(C)cc(Br)cc1C 75896,c1(C(N(CCC)CCNC(C2(C)CCCC2)=O)=O)ccc(CCN(C)C)cc1 75897,Cc1cccc(C(=O)N(CCCC(N2CCN(C)C(=O)C2)=O)C)c1C#N 75898,N1(C(C(C(C)C)SCC)=O)CC(C)(C(=O)N(CC(=O)NC)C(C)C)CC1(C)C 75899,C1(C)(C(=O)NC2C(OC)CN(C(c3cc(C4CCC4)on3)=O)C2)CCCNC1=O 75900,N1(C(CC2CC(CC)OCC2)=O)CCN(C(c2ccc[nH]2)=O)CC1CCO 75901,C(=O)(CC(CNC(=O)CC1(C)CCOCC1)C1CCC1)NCc1c(C)csc1 75902,CC1(NC(C2CC2c2ccco2)=O)CCN(C(c2cocc2Br)=O)CC1 75903,S1(=O)(=O)c2ccc(cc2)N1.N1(C(C)CO)CC2(CCC2)C1C(=O)NC1CC1 75904,C(C(C(C)C(C)C)NC(c1cccnc1C(F)(F)F)=O)NC(CNC(C)=O)=O 75905,c1(C(=O)NCc2cccc(NC(C3(C)C(C)OCC3)=O)c2)ccc(CO)c(Cl)c1 75906,Cc1cc(C(=O)N(CCCCN(C(=O)CCOc2ccc(F)cc2)C)C)c(C)[nH]1 75907,CC(C)(CCCN=c1nc(N2CCC(C3(O)CC3)CC2)cc[nH]1)N1CCOCC1 75908,N1(C(CCC=CCC=C)=O)CCCN(C(=O)Cn2ccc(C(=O)OC)n2)C(C)C1 75909,C1(C(=O)NC(C=C)C)CN(C(=O)CC(C)CCC)CC12CC2 75910,c1(SC)cc(C(=O)NCC(C)CNC(c2ccc(C(C)C)o2)=O)ccc1F 75911,c1(C(c2nnnn2C)NCc2cnc(C)s2)ccc(Cl)c(C(F)(F)F)c1 75912,Cc1n[nH]c(=NCC2CCN(C(=O)CCCOc3cccnc3)CC2C)o1 75913,C1(C(=O)NCc2c(C(=O)NCC3CCC=CO3)occ2)CC2(CCC2O)C1 75914,c1(C(=O)NCC(CC)NC(=O)CC2CCn3cncc3C2)cc(Cl)c(O)cc1C 75915,C1(O)(CCNC(CC2C(C)C2)=O)CCN(C(c2ccc(N)cn2)=O)CC1 75916,c1(C(N2C(CN(C(CC(=C=C)C)=O)C)CCCC2)=O)ccc2c(c1)CCO2 75917,C=C(Cl)C(C)(C)C(=O)N1CCCCC(NC(=O)C(C(C)C)NC(=O)COC)C1 75918,Cc1csc(C(=O)NCC#CCNC(C2(n3cc(Cl)cn3)CC2)=O)c1 75919,N1(C(c2c(C)nn[nH]2)=O)CC(NC(C2CCCN2c2nccs2)=O)C2CC2C1 75920,c1(C(=O)NC2CC(F)(CNC(C3=NNC(=O)CC3)=O)C2)[nH]cc2c1CCS2(=O)=O 75921,c1(C(N2CCC(CN(C)C(c3ccn(CC#N)n3)=O)C2)=O)cc2cnn(C)c2s1 75922,C1(C(N(C(CC)C(=O)NCCCNC(C)=O)C)=O)CCC(C)(C)C1 75923,C1(NC(c2c(CC)nc[nH]2)=O)CC2CC1N(C(=O)CC(O)c1cnc(Cl)s1)C2 75924,c1(C(N(CC(C)NC(c2c(Cl)ccc(C)c2)=O)C)=O)cccc2cnnc(O)c12 75925,c1(CC(N2CCN(C(C(COC)C)=O)CC2CO)=O)c(C)oc2ccccc12 75926,c1(C(=O)NC(C)(C)CNC(c2cc(C3CC3)[nH]c2C2CC2)=O)cc2n(n1)CCO2 75927,C(c1c(C)noc1C)=CC(=O)NC(CC)(C)CCNC(=O)C(C)=C(C)C 75928,c1(C(N2C3C(NC(C(CC=C)C)=O)C(C3)C2C)=O)cc(C)c(F)cc1F 75929,C1(CNC(c2scc(C)c2C)=O)CN(C(=O)CCc2nc(O)n[nH]2)CCC1(F)F 75930,c1(CNC(=O)COC(F)F)cnn2c1CN(C(=O)CC1C=CCCC1)CC2 75931,c1(C(N2CC(F)CC(NC(CSCC=C)=O)C2)=O)ccnc(S(N)(=O)=O)c1 75932,C(=O)(C(O)C1=CCCCC1)N(C1CC(NC(c2ccc(OCC)nc2)=O)C1)C 75933,c1(CNCC2(NC(=O)Cn3ccnn3)COC2)c(F)cc(I)cc1F 75934,N1(C(c2oc(CC)c(C)c2)=O)CCC2(CC1)CC2CNC(c1csnc1OC)=O 75935,N1(C(c2c(C)cc(C3CC3)nc2)=O)C2CCC1CN(C(C1CCCC(C)C1)=O)C2 75936,c1(NC(C(C(C)C)CNC(C2CCC(=O)NC2)=O)=O)ccc2c(c1)COC2 75937,C1(C(=O)NCCCN(C)C(C2(CC3CC3)CC2)=O)CCCCC1c1nncn1C 75938,C1(C(N(C2CCC2)C(C)C)=O)CC(C)N1C(=O)CCc1cncnc1 75939,C1(CCNC(Cn2c(C)ccn2)=O)CC(F)(F)CN1C(c1c[nH]nc1Br)=O 75940,C(c1cccc(F)c1F)=CC(N1CCC(O)(CNC(C(C)(F)F)=O)C1)=O 75941,C(=O)(CCCCC(C)C)NCC1(F)CC(NC(c2cccc(CC)c2N)=O)C1 75942,c1(OC)cccc(C2CCN(C(C3CCCSC3)C(=O)NC3COC3)C2)c1 75943,c1(C(=O)NCC(CNC(CCc2ccc(C)o2)=O)F)cc(C)c2[nH]nnc2c1 75944,CC12CCC(C(=O)NCC3(O)CN(C(=O)CC4CCCC45CC5)C3)(CC1)C2 75945,C(CCC(C)C)(C(=O)NC1CCC2CC1CO2)NC(C(C(CC)C)=O)=O 75946,CC1CC(NC(c2cnoc2)=O)CCN1C(c1cnns1)=O 75947,CC(CNC(C1C(C)C1C)=O)C(=O)NC(C)C(C)F 75948,CCC(C(=O)OC)C(=O)N1CCC(NC(c2cc(C)no2)=O)C12CC2 75949,N1(C(CC=CCC)=O)CC(NC(=O)C(C(C)C)N2CCCC2=O)C2(CC2)C1 75950,c1(CC(N2CC(C)C(CCNC(c3ccc(Cl)o3)=O)C2)=O)ccc2n[nH]cc2c1 75951,C(=O)(CCCC(C)(F)F)NC1(CNC(c2nn(C)c(=O)cc2)=O)CCOCC1 75952,c1(C(N2CCCC(NC(C(c3ccc(C)s3)C)=O)C2)=O)cc(Cl)nc(=N)[nH]1 75953,CC1(C)CC(CNC(c2cn3cnnc3cn2)=O)CN(C(=O)COC(C)(C)C)C1 75954,c1(C(=O)NCC(CCCC)NC(=O)CC2CSCCS2)cccc2scnc12 75955,c1(C(N2CC(CC(=O)Nc3nccc(Br)c3Cl)OCC2)=O)cc(F)c(F)cc1O 75956,N1(C(C(C)=C2CCC2)=O)CC(O)CC1C(=O)NCC(c1ccccc1)C1CC1 75957,CC1CC(NC(C2(Nc3ccccc3)CC2)=O)CCN1C(C12CCCC(C1)OC2)=O 75958,CCC(C)C(O)C(C)C(=O)N(C1CCN(C(c2cccc(C3CC3)c2)=O)C1)C 75959,c1(C(N(CCNC(C2CC(=O)N(C)C2)=O)CC)=O)cnc2c(C)cccn2c1=O 75960,N1(C(CC2(C)CCN(C(c3ccccc3)=O)C2)=O)CCC2CCCC(C2)C1 75961,C12(C(=O)NC(C)(CNC(C3CC(CCO)C3)=O)C3CCC3)CCC(C1)C2(C)C 75962,c1(C(N2C(CCNC(c3ccc(C)o3)=O)CSCC2)=O)ccc2c(c1)OCO2 75963,C1(CC(=O)NCCOCCOCCNC(C2(F)C(C)C2)=O)COc2ccccc2O1 75964,N1(C(c2cncc(Br)c2)C(=O)NCC=C)CC(C)(C)c2ccccc21 75965,CC1C(NC(=O)C(C)O)CCCN1C(=O)CCC1OCCO1 75966,N1(C(C(CC(=C)Cl)NC(=O)CCC2CCC2)=O)CCNC(=O)CC1C 75967,c1(C(N2CC=CC(NC(c3c(C)onc3Br)=O)C2)=O)ccc(Cl)c(N)c1 75968,c1(C(N2CC(C(C)(F)F)OCC2)=O)c(F)cccc1I 75969,CC1COC2(C1)CN(C(=O)C(Cn1cncn1)NC(C1COCC1(C)C)=O)C2 75970,CC1=CCSC1C(=O)NCCC1CCCN1C(=O)CC1CNC(=O)O1 75971,C#Cc1cc(C(N2CC(C)(NC(=O)C3=C(C)CCCC3)C2)=O)cc(N)c1 75972,C1(NC(C#CC(C)C)=O)CC2CC1CC2C(N1CCOC(CF)C1)=O 75973,c1(-n2cc(CC(N3CCOCC3C3CCCC3)=O)nn2)ccc(C(=O)O)cc1F 75974,c1(OC)cc(C(=O)NCC2(O)CC(CNC(C3(OC)CCSC3)=O)C2)cc(Cl)c1 75975,Cc1cc(Cl)c(C(=O)N(CC(O)CN(C)C(c2cnc(O)c(F)c2)=O)C)cc1F 75976,C12(C(=O)NCC3CN(C(C4(C(=O)OCC)CC4)=O)C3)CCOC1CC(=O)NC2 75977,c1(C(C(=O)NCC(C)NC(=O)C=Cc2ccoc2)O)ccc(Cl)c(Br)c1 75978,C=CCCCCCNC(=O)CN1CCN(C(=O)CCc2cn(C)cn2)CC1 75979,c1(C(=O)NC2CC3CC(NC(=O)C4CC4)C2C3)cc(Cl)c2[nH]c(O)nc2c1 75980,c1(C(=O)NC2C(C)N(C(c3nc(O)sc3C)=O)CC2)ccc2c(c1)nc(O)n2C 75981,c1(CNC(=O)CN2CCOCC2)ccccc1CNC(c1cc(Cl)c[nH]1)=O 75982,N1(C(CN(CC)CC)=O)CCCCC1C1CCCN1c1ncnc2c1cnn2C 75983,C(=O)(CC1=CCCCC1)NCC1(O)CC(CNC(C(C)(F)c2ccon2)=O)C1 75984,CCCCC(CNC(=O)CN1CCN(C2CC2)C1=O)NC(=O)CC1CC(OC)C1 75985,CC1CCc2[nH]c(=NCC(C)(C)CC(F)(F)F)[nH]c(=NC3COCC3N(C)C)c2C1 75986,C(CC(=O)N(C)CCNC(C12COCC1C2)=O)(C1=CCCC1)OCC 75987,N1(C(c2cc(C)[nH]n2)=O)CCC2(CC1)CC2NC(=O)C(C1CC(F)(F)C1)O 75988,Cn1cc(C(=O)NCC2(NC(=O)CC3CCC(C#N)C3)CCC2)c2ccccc12 75989,C1(C(=O)NCCN(C(c2cnc(C)cc2Cl)=O)CC)CCC2(CCOCC2)O1 75990,N1(C(C(C2CCOCC2)C)=O)CCC(C(F)CNC(C2(C)CS(=O)(=O)C2)=O)CC1 75991,c1(CC(N2CCN(C(C(C)OC3CCOCC3)=O)CC2)=O)c[nH]c2ccccc12 75992,N1(C(CC(CCC)(C)O)=O)CCC2CCC(C1)N2C(C1(C)CCOC(C)C1)=O 75993,C#Cc1ccc(C(N2CCCC(CCNC(C3(CCO)CC3)=O)CC2)=O)nc1 75994,c1(COC)ncc(C(=O)NC2(C)CC(NC(=O)C(C)(C)c3ccno3)C2)c(=N)[nH]1 75995,c1(C(N2CCC(NC(=O)C=Cc3nc[nH]n3)C2)=O)cnc2cc(O)ccc2c1 75996,C(=O)(CCCC1CCNCC1)OCC(=O)NCC(C)C 75997,C1(NC(c2cnc[nH]2)=O)CC2CN(C(=O)CCc3ncc[nH]3)CCN2C1=O 75998,N1(C(CCCC(C)C)=O)CCCC2C(CCCN2C(c2ccnn2CCF)=O)C1 75999,C(=O)(CCC(C)N1CCOCC1)N1CCC(N(CCC)C(c2ccoc2Cl)=O)C1 76000,c1(C(=O)NC2(C)CN(C(C3C(C)CC3)=O)C2)cc([N+](=O)[O-])ncc1Br 76001,N1(C(C(C)n2cncn2)=O)CCC2CN(C(C3CC4(C3)CC(O)C4)=O)CC2C1 76002,Cn1ncc(NC(C2CCC(NC(c3csc(Br)n3)=O)CC2)=O)c1C(N)=O 76003,C(=O)(C(C)(C(C)C)NC(c1cc(Cl)cc(C(F)(F)F)n1)=O)OCC 76004,C1(CC(=O)N(C)CC2CCC(NC(c3cncs3)=O)CC2)CC2(CCC2)CO1 76005,N1(C(CCOc2c(C)cccc2)=O)CC2CC1CCN2C(C12CC(C1)C2)=O 76006,CCCS(=O)(=O)CC(=O)NCCCN(C(C1(C2CCCO2)CCCC1)=O)C1CC1 76007,c1(C(=O)NC(C2CCN(C(=O)CSS(C)(=O)=O)C2)C)c[nH]c2cccnc12 76008,Cc1cc(OC(=O)CC2CCN(CC(F)(F)F)C2)ccc1OC(F)F 76009,c1(OC)noc(C)c1C(=O)NCCCC(C)NC(C12CCCCC1C2)=O 76010,N1(C(CN(C)S(N)(=O)=O)=O)CCC(C)(C)C(NC(C2CNC(=O)C(C)(C)C2)=O)C1 76011,C(=O)(C#CC(C)(C)C)NC1(C(=O)NCCOCC(F)(F)F)CCN(C)C1 76012,C(=O)(C1=CCCCCC1)NC(CCN(C(c1ccc(OC)c(Br)n1)=O)C)C 76013,C#Cc1ccc(C(=O)NC(C(=O)N2CC(OC)C2)C2CCCO2)cc1 76014,C#CCC(CC(F)F)C(=O)NCC(C)(C)OCC(=O)NCC1(c2ccsc2)CC1 76015,c1(CSC)cc(C(=O)NC(C)CC2CN(C(=O)CCC3CCCCO3)C2)sc1C 76016,C12(c3onc(C(N4C(CS(N)(=O)=O)CCCC4)=O)n3)CCC(CC1)CC2 76017,C1(NC(=O)C=CC2CCCC2)CCCCC1NC(C1C(F)(F)C12CC2)=O 76018,N#Cc1cc(C(N2CC(F)CC2C(=O)Nc2cnn(CCO)c2)=O)ccc1Br 76019,c1(C(=O)NC2CCC(C)N(C(=O)CC3CCCCC3)C2)cc2cccnn2c1 76020,C1(OC)CCN(C(=O)CC(C(C)C)NC(C2CCCN2C(C)C)=O)CC1(C)C 76021,c1(C(C(N2C(C)CC(NC(c3cnc(Cl)s3)=O)C2)=O)=O)c[nH]c2ccc(F)cc12 76022,c1(C(=O)NCC2CN(C(C3COC(=O)O3)=O)C2)ccncc1Br 76023,Cn1cc(C(=O)NCC2(NC(C3CC4C=CC3C4)=O)CCC2)c(C2CCCO2)n1 76024,C12(CC)CN(C(=O)Cc3nonc3C)C(CNC(c3cc(C)nc(O)n3)=O)(C1)C2 76025,N1(C(C2ON=C(C)C2)=O)CCN(C(c2ncn3ccccc23)=O)C2(CCC2)C1 76026,c1(C(=O)NCC(CN(C)C(C2CCSCC2)=O)O)ccc2c(O)nnc(O)c2c1 76027,Cc1nccnc1-c1cn(C(=O)C(C)(O)c2ccccn2)nn1.C12CN(C1)C2 76028,C12(C(N3CCCC(NC(=O)C=C4CCCC4)CC3)=O)CCCCC1C2(F)F 76029,CC(C)(C)CC(F)C(=O)Nc1ccoc1C(=O)NCCN1CCCC(O)C1 76030,C=Cn1nccc1C(N1CC(F)CC1CNC(c1ccccc1)=O)=O 76031,C(=O)(CCCS(=O)(=O)N1CCCC1)N1CC(NC(c2cc(O)ncn2)=O)C2C1C2 76032,CCC(C)(C)CC(=O)NCC1CC(NC(=O)C(c2ccccc2Cl)O)C(O)C1 76033,N1(C(C2(C)CCC(=O)C2)=O)CCCCC(NC(c2ncc(Cl)cc2Cl)=O)CC1 76034,n1(C(C(CCC)=O)C)nc(C)ccc1=O.C12(N)CCC(C1)N(C(C1(S(N)(=O)=O)CC1)=O)C2 76035,c1(CN2CC(NC(C(C)(C)O)=O)C(F)(F)CC2)c[nH]c2ccc(F)cc12 76036,N1(C(CCN(C(c2cnc(CC)o2)=O)CCO)=O)CC2CCC1C2 76037,CCCCC(O)C(C)C(=O)NCC1OCCC1C(=O)Nc1cc(CC)ccc1C 76038,c1(C(=O)NCC2(C)CCN(C(C(CN(C)C)(F)F)=O)C2)ccnc2c1CC(=O)N2 76039,C(CN=c1[nH]c2c(c(=NCCOc3ccncc3)[nH]1)CSC2)C1(C)CCCO1 76040,N1(C(c2c(C)n(C)nn2)=O)CCC2C(C1)CN2C(c1cc(C(C)(C)C)nn1C)=O 76041,C1(CC(=O)NCC2CCN(C(=O)CC3CS(=O)(=O)C3)CC2)CCCCC12CC2 76042,Cc1cc(O)ccc1C(=O)NC1CC(NC(=O)CSc2ccncc2)CC1O 76043,Cc1c(CC(=O)NCC(C)NC(C2CCCN2C)=O)ccc(Cl)c1Cl 76044,C(=O)(C1=CCCCC1P(C)(C)=O)N(C(CNC(c1cc(OC)c(C)cc1)=O)C)C 76045,C(=O)(C(CCC1CC1)N1CC2CC2(c2ccccc2C)C1)NC1CC(C)(CC)C1 76046,c1(C(=O)NC2CN(C(C3CC3(Cl)Cl)=O)CC2C(F)F)cnc(O)c2ncccc12 76047,c1(C(=O)NCC(CC=C)NC(=O)CCCCOC)cc(O)cc(F)c1F 76048,N1(C(C(C)NC(CC)=O)=O)CC2(C1)CN(C(C13COC(CS(C)(=O)=O)(C1)C3)=O)C2 76049,N1(C(c2ccc(SC)o2)=O)CCC(F)(CNC(=O)CC2CCOC2=O)CC1 76050,c1(CC(C)=CC(=O)NCCOCC(N2CCOCC2)=O)ccc(C)c(C)c1 76051,[N-]=[N+]=NCCCC(=O)NCC1(C(N2CCC(N3CCCC3)C2)=O)CC12CCC2 76052,C1(CC(=O)NCC(C)N(C(=O)CCc2ccccc2F)C)CCOC1(C)C 76053,C(CNC(=O)C1=CSCS1)(C(C)(C)C)NC(C(C)OCC)=O 76054,N1(C(C(CO)NC(N)=O)=O)CC2(CCCN(C(c3cc(C4CC4)cs3)=O)C2)C1 76055,C#Cc1ccc(OCC(N2CC(NC(c3cnc(C)cc3C)=O)CC2C)=O)cc1 76056,c1(C(N2CCC(NC(c3cn(C(C)C)nn3)=O)CC2C)=O)cccn2ccnc12 76057,c1(C(=O)NC2CCC(CNC(c3c(C)oc(Cl)n3)=O)C2)cc(O)cc([N+](=O)[O-])c1 76058,c1(NCC(=O)N(CCNC(C)=O)C)cc([N+](=O)[O-])c(F)cc1NCCCF 76059,C(CCCCCC(=O)NCC(C)N(C)C(c1ccc(C(F)(F)F)c(F)c1)=O)SC 76060,Nc1c(C(N2CC3C(CNC(=O)CCSC(F)(F)F)C3C2)=O)cc(F)c(F)c1F 76061,c1(NC(C2CCC(C(CC)(C)C)CC2)=O)cc(C)cc(Br)c1C 76062,C1(C(=O)NC2CCN(CCNC(C(C)c3cc[nH]n3)=O)CC2)CC2CCCCC12 76063,c1(C(=O)NCC2COCCN2C(C2COC2)=O)ccn2ncc(Br)c2c1 76064,c1(N(CC(N)=O)CC2(C)CCN2)ccc2ccccc2c1 76065,c1(C(=O)NCCC(C)NC(c2c(C)noc2C)=O)ccc2nc(O)[nH]c2c1 76066,C1(CNC(C(C)NC(C)=O)=O)CCN(C(=O)Cc2ccccc2Br)CC1 76067,C12(C(=O)NCC3C(C)CN(C(=O)Cn4cc(Cl)cn4)C3)CCOC(C)(C1)C2 76068,c1(C(N2CCN(C(=O)NC3CCCC(C(N)=O)C3)CC2)=O)c(F)cc(F)cc1Br 76069,C1(C(=O)NCCCCC(C)NC(=O)C=CC2CCC2)CCc2ccccc2N1 76070,c1(C(N2CCC(Cc3ccnn3C)C2)C(=O)NC)ccc(S(C)(=O)=O)s1 76071,c1(OC)nsc(C(=O)NC2CC3(C2)CC3NC(C2CC2(C)C)=O)c1Br 76072,C#Cc1cc(C(=O)NC2CS(=O)(=O)CC2NC(=O)C(C)CC(F)(F)F)ccc1C 76073,c12nc3n(c1Cl)CCN(C3)C2.C(C(C(=O)OCC)NC(=O)OC(C)(C)C)SCC 76074,c1(OC)cccc2c(CCNC(C3(c4ccc(F)cc4)CC(C)(C)C3)=O)c[nH]c12 76075,N1(C(c2ccc(NCc3cnccc3C)cc2)=O)CCCC2C1CCN2OC 76076,C(=O)(C(C)CS(C)=O)NCC1(CNC(c2c(C)n[nH]c2C)=O)CC1 76077,C(CCC(C)C(=O)N(C1CCN(Cc2csc(Cl)n2)C1)C)OC 76078,C1(C(=O)NCC(CC(C)C)(C)C)CCN(C(=O)CCC(C)(C)F)O1 76079,CCC(O)C(C)(C)C(=O)NCC1(CN(C)C(c2cc(O)nc(Cl)c2)=O)CC1 76080,C=Cc1cncc(C(=O)NC(Cn2cncn2)C(=O)N(C2CCOC2C)CC)c1 76081,CC(C)C(O)C(=O)N1CCC(C(C)(O)CNC(=O)C(F)=C2CCCC2)CC1 76082,C1(C(=O)NC2CC(C)(NC(c3nc(C(C)OC)sc3)=O)C2)CC12CC(F)(F)C2 76083,C(CC(CNC(=O)CN1CCCCC1)NC(=O)C=C1CC(C(C)(C)C)C1)OC 76084,CC(C)(CC(F)(F)F)C(=O)N1CCCC(NC(C2Cc3nncn3C2)=O)CC1 76085,N1(C(c2cc(C(C)=O)oc2C)=O)CCCN(C(c2csnc2Br)=O)CCC1 76086,C1(C(=O)NCC(=C)C)CC(N(C(=O)CCC2CCC2)C)C1 76087,N1(C(C2CC2c2cccc(F)c2)=O)CC2CC1CN2C(C12CCC(CC1)C2)=O 76088,N1(C(C(=O)NCCc2cnn(C)n2)=O)CCCCCC1C(F)(F)F 76089,c1(C(=O)OC)c(C)[nH]c(C)c1C(=O)C(C)ON(C(C)CO)C 76090,CCCCC(CNC(=O)C(OCCCC(C)C)NC(=O)CC1CC(F)(F)C1)OC 76091,N1(C(C(CC2CCC2)NC(Cn2cnc(=N)[nH]2)=O)=O)CC2CC1CS2=O 76092,c1(C(=O)NC2C(SC)CN(C(C3(C#N)CC3)=O)C2)nn2cccnc2c1Br 76093,C12(NC(C(CC)NC(C)=O)=O)CCC(CC1)N(C(=O)C=C1CCCCC1(C)C)C2 76094,C1(C(N2CCC(N(C)C(c3coc(C(N)=O)c3)=O)C2)=O)(OCC)CCOCC1 76095,c1(CC(=O)NCC(N2CCN(C(C(C(C)O)C)=O)CC2)=O)ccc2ccoc2c1 76096,c1(COCCNC(=O)NCC(O)C2CC2)ccco1 76097,c1(C(=O)NCC2C(NC(CC(CC)OC)=O)C2)cc(-n2ccnn2)ccc1F 76098,N1(c2cc(OC)nc(OC)n2)CCC2CN(C(c3cc(SC)nn3C)=O)CC2C1 76099,C1(C)(C(N2CC(OC)(CO)C2)=O)CC(O)CN1C(=O)C=C(C)C(C)C 76100,N1(C(c2c(C)nsc2)=O)CC(NC(=O)CSCc2nc(=N)[nH][nH]2)CC1C 76101,C(C(C)C(C)N=c1nc(N2CCC(CCO)CC2)c2cc(Cl)ccc2[nH]1)OC 76102,C1(C(N2CCC(C(N(CC)CC)=O)C2)C(=O)NC2CC2)CC(C)OC1C 76103,CC1CCN(C(=O)COC(=O)CO)C1CNC(=O)CCCC1CC1 76104,c1(CNC(C(=O)NC(c2cccc(C)c2)CC)=O)cn2cccnc2n1 76105,C1(NC(=O)C2=CCCSC2)CC(C2CCN(C(c3csc(C(F)F)c3)=O)C2)C1 76106,Cc1cccc2[nH]cc(C(=O)NCCN(C(=O)C(C)n3ccnc3)CC(C)O)c12 76107,C1(OC)CC(CNC(=O)C2=CCCS2)N(C(=O)CC2(C)CCCCC2)C1 76108,C1(NC(c2cn[nH]c2)=O)CN(C(c2cncc(-n3ccnc3)n2)=O)CCC1CO 76109,N1(C(CC)=O)CCC(N=c2nc(N3CCC=CC3)c3c([nH]2)CCC(C)C3)C1 76110,N1(C(C2(CO)CC(C)(C)C2)=O)CC2CC(NC(=O)CCC3CCC3)C1C2 76111,c1(CCC(=O)N(CCC(C)NC(C(CC)(C)O)=O)C)nnc(O)nc1O 76112,Cc1cc(Cl)c(Br)cc1S(=O)(=O)N1CCc2scnc2C1 76113,c1(C(CNC(C(C)OCC=C)=O)NC(=O)CCN2CCCC2=O)ccccc1F 76114,N1(C(c2nnc(C)s2)=O)CC(O)C(O)C1CNC(=O)Cc1ccc(F)cc1F 76115,n1(CC(=O)NCC2CC(C)N(C(=O)C(C3CC3)C3CC3)C2)nc(O)ccc1=O 76116,c1(C(=O)NCC2C(C)(C)CN(C(C3CC4C=CC3C4)=O)C2)nnc2ccccn12 76117,c1(CC)sccc1C(=O)NC(C1CCCN1C(c1cnco1)=O)C 76118,N1(C(C2N(C(C3CCN3CC(F)(F)F)=O)CCC2)=O)CCC(CO)C(F)C1 76119,CC1CN(CC#N)CCN1C(=O)Cc1nc(C2CC2)cs1 76120,N1(C(c2cnc(CC)nc2)=O)CCC(NC(=O)Cc2ccn(CC)n2)C12CC2 76121,c1(C(=O)NCC2CCCC2Nc2cc(C(F)(F)F)ncn2)cn2c(n1)COCC2 76122,c1(OC)ccc(C(N2CC(CO)(NC(=O)COCCSC(C)C)C2)=O)cc1Cl 76123,Cn1cc([N+](=O)[O-])c(=NCC2(NC(c3cncn(C)c3=O)=O)COC2)[nH]1 76124,c1(OC)ccc2[nH]c(=NCC(C)NC(c3cc4c(C)cc(C)nc4s3)=O)sc2n1 76125,N1(C(C2(CCOC)CC2)=O)CC2CCCC(C1)N2C(C1CCCC1S(C)(=O)=O)=O 76126,Cc1csc(=O)n1CCCC(=O)NC1CC(N(C)C(c2cc(Cl)cn2C)=O)C1 76127,N1(CC)CCC(NC(=O)C(C2CC2)NC(=O)C(C)COC(C)=O)C1 76128,C12(CNC(=O)CCn3cccn3)CCC1CCN2C(=O)CNc1ncccn1 76129,c1(CNC(C2CC2c2cnn(Cc3ccccc3)c2)=O)coc(C(F)(F)F)c1 76130,c1(C2(C)CCO2)ccccc1C(N1CC2C(NC(C3(CC4CC4)CC3)=O)C2C1)=O 76131,[N-]=[N+]=Nc1ccccc1C(=O)NC1(CF)CCN(C(=O)Cn2cccn2)C1 76132,C1(NC(C(CC)OCC)=O)CCC2CN(C(=O)C(C)Sc3ncccn3)CC2C1 76133,C1(NC(CCC(=C)C)=O)CCN(C(C2CCC(=O)C2)=O)CC(O)C1 76134,c1(C(N(CC(CNC(c2ccn(C(C)C)n2)=O)C)C)=O)ccc2c(n1)CCCC2 76135,c1(C(=O)NCC2C=CCN2C(c2sccc2Cl)=O)ccc(OC(F)(F)F)nc1 76136,C#CCC(C)(C)C(=O)NCC(C1(O)CCN(C(c2ncncc2N)=O)C1)C 76137,C1(NC(c2c(C)ncn2C)c2nnnn2CC(F)F)CCCCCCCCC1 76138,C12N(CC1(C)C)C(=O)CC1CCCC(C1)NC2=O.c1(COC)cccnn1 76139,N1(C(C2(S(N)(=O)=O)CCCC2)=O)CCC2(CC1)OCCC2NC(C1CCCC1)=O 76140,c1(C(N2C(CNC(=O)CC3CC4(CC4)C3)CCC2)=O)cc(O)ncn1 76141,C1(CNC(c2cc(C)on2)=O)CCCCN1C(c1cocc1C(N)=O)=O 76142,N1(C(Cc2nc(C)[nH]n2)=O)CCCCC1CCCNC(=O)C(F)CC1CC1 76143,C(=O)(CS(=O)(=O)C(C)C)N1CC(OC)CC1(C)CNC(=O)C=Cc1ccoc1 76144,N#CC12CCCCCC1CN(c1ccn3nccc3n1)C2 76145,N1(C(c2c(CC)nnc(C)c2)=O)CC(NC(C2CN(CC)C2)=O)CC12CCOC2 76146,c1(C(=O)OCC)cnc(NC2(CNC(c3cccc(Cl)c3F)=O)CCC2)nc1C 76147,c1(-c2cc(C(=O)NC3C(CNC(C(COC)C)=O)C3)no2)ccc2c(c1)CCO2 76148,CC1(C)NC(=O)CC1C(N1CC(C(=O)NC2CCCN(O)C2=O)C(F)(F)C1)=O 76149,CC(Cc1ccco1)C(=O)NCC1(O)CN(CC2CCC(C)O2)C1 76150,Cc1cc(C(=O)NC2CN(C(=O)Cc3cscn3)CCC2F)cnc1O 76151,Cc1c(C(=O)NCC(CNC(=O)Cc2nc[nH]n2)CO)sc2nnc(S)n12 76152,C1(N(C(c2c(COC)cccn2)=O)C)CN(C(C2CN(C(C)C)C2)=O)CC12CC2 76153,N#CC1CCC(C(=O)NC2CC(CNC(=O)Cc3cnn(C(F)F)c3)C2)CC1 76154,C1(C(N2CCC(CC#C)CC2)=O)CN(C)CCN1C(C1C2COCC12)=O 76155,c1(CN(C(C(c2cn(C)nn2)NC(Cn2c(C)nnn2)=O)=O)C)ccccc1F 76156,C12(CC)CN(C(=O)CC(C)OC)C(CNC(=O)CC3C(=O)NN=C3C)(C1)C2 76157,N1(C(CC=CCNC(CC=C(C)C)=O)=O)CCC(COC(C)C)CC1 76158,c1(C(=O)NC2CCC(NC(C3(Cl)CC34CCC4)=O)C2)csc2cccnc12 76159,c12ccc(nc1)C(=O)NC2.n1(CC)ccnc1NC(=O)CC1CSCCO1 76160,N1(C(C(C(CNC(c2ccnc(OC)n2)=O)C)F)=O)CCc2nc(O)[nH]c2C1 76161,C(N=c1cc(NCc2cccc(Cl)c2F)nc[nH]1)C1C(CCOC)C1 76162,C1(C)(C(=O)NCC2CC(C(=O)NC(c3nc(C)on3)C)C2)CNC(=O)C1 76163,C(=O)(C(C)CS(C)(=O)=O)NCCC(C)CF 76164,CCCCCCNCC1CN(C(N)=O)C1.c1(C(COC(C)(C)C)N)nnnn1C(C)C 76165,Cc1oc(C(C)C)nc1C(=O)NC1CCCCC1NC(=O)CNC(=O)C(C)(C)C 76166,Cc1ccnc(C(=O)N(C2CCC(NC(c3sc(Cl)cc3Cl)=O)C2)C)n1 76167,CC1C(C)N(C(c2ccc(N(C)C)cc2)=O)CCN1C(=O)CC(O)CCN(C)C 76168,Cc1cccc(NC(N2CCN(Cc3cc(C(=O)O)cc(Br)c3)C(C)C2)=O)c1C 76169,N1(C(CN2C(=O)COCC2)=O)CCC2CCC(C1)N2C(=O)CN1CCSCC1 76170,N1(N(CC(=O)OC)CCOC)Cc2ncsc2C1.C1(C=O)CC(NC)C1 76171,Cc1cc2cc(C(=O)NCC3CC3CNC(C3CCC3)=O)oc2cc1C 76172,c1(C(N2C(C)CC(NC(C3CC(=C)C3)=O)C2)=O)ccc2c(c1)OCCC2 76173,c1(C(N(CCNC(=O)CC2(CC)CCOCC2)CC)=O)nc(OC)ccc1Cl 76174,N1(C(C)=O)CCCC1(C)C(=O)N(CCCNC(C1(CC(C)C)CC1)=O)C 76175,C12(NC(=O)CC3CCC34CCC4)CCCC(CN(C(c3cnsn3)=O)C1)C2 76176,CN1C(=O)C2CN(c3cc(C#N)ncn3)CC2C1=O 76177,C1(C(=O)NCC(O)CNC(C2(CC=C)CC2)=O)(CC)CCNC1=O 76178,C1(N(CC#C)C(c2ccc(COC)o2)=O)CCN(C(=O)CCN(C)CCC)CC1 76179,CCCC(O)C(=O)N1CCC(C(=O)N(C)CCOC)C1 76180,C1(CC(N2C(CNC(C3CCCC(OC)C3)=O)CC2)=O)CCn2cncc2C1 76181,N1(C(C(C)(C)n2cccn2)=O)CC(NC(=O)CCc2cc(Cl)cs2)C(C2CC2)C1 76182,N1(C(c2cc3ccoc3cn2)=O)CCCC2C1CCN2c1ncc(Cl)cn1 76183,C(=O)(C1c2[nH]cnc2CCN1C(=O)C(CC1(C)CC1)c1ccccc1)OC 76184,C1(C(=O)NCCCCO)CN(C(=O)CC2CCOC2=O)CC12CC2 76185,C1(=CC(=O)NCCC2(NC(C(C)OCC3CC3)=O)CCCC2)CN2CCC1CC2 76186,Cc1cc(NC(=O)CC2(C)CCN2C(C2(C)CC2)=O)c([N+](=O)[O-])cc1Br 76187,CC(O)C(C(=O)N(CCCNC(=O)CCC1CCCCCC1)C)NC(=O)C1CC1 76188,C1(CCNC(c2cc(C(=O)OC)[nH]c2)=O)CC(F)(F)CN1C(c1ccc(Cl)o1)=O 76189,C1(NC(C(CCCC)NC(N)=O)=O)CN(C(=O)CC2(C)CCCC2)CCC1(C)C 76190,C1(C(N(CCCn2cc(CCCS(N)(=O)=O)nn2)C)=O)CCOC2(CCCC2)C1 76191,C1(F)(CC(=O)NCCNC(C(n2nnc(-c3ccccc3)n2)C)=O)CCCOC1 76192,N1(CC#C)CCc2nc(C(=O)N(CCn3cc(C)cn3)C(C)=O)cn2CC1 76193,C(=O)(CCCC(=O)N1CC(O)(CNC(=O)CCc2ccncn2)C1)N(CC)CC 76194,C=C(C)C1CCC(C)(O)C(NC(C2(c3cccc(C(F)(F)F)c3)CCC2)=O)C1 76195,c1(CC(=O)N(C)Cc2onc(C)n2)csc2nccn12 76196,C(c1cncn1C)=CC(=O)NC1CC(C(C)NC(=O)CC2CCOC2)C1 76197,C1(N(C(C2CN(CC(C)C)C2)=O)C)CCCC(NC(c2ccc(=O)oc2)=O)C1 76198,C1(C(=O)NCC(C)(C)OCC(=O)N(C2CCCC2C#N)C)CCCCCC1 76199,C(C(C)(CC(C)C)NC(c1cc(C(N)=O)on1)=O)NC(C(C)=CC1CC1)=O 76200,c1(C(N2C(CC(=O)N(C(C=C)C)C)CC2)=O)cnn2ccccc12 76201,CN=c1[nH]cc(C(N2CCC(O)(C(C)CNC(c3cn(C(C)C)nn3)=O)C2)=O)o1 76202,c1(NC(C2N(C(C(CC)(C)O)=O)CC2)=O)ccc(=O)n(CCOC)c1 76203,CC#CC1CCN(C(=O)C=CCC2(NC(=O)Cc3ccn(C)c3)CCC2)CC1 76204,N1(c2nccc(SC)n2)CCC(C2CN(c3cc(C)ncn3)C2)CC1 76205,N1(C(CCCCC=CC)=O)CCC(C2CCN(C(C3CC3(F)F)=O)CC2)C1 76206,N1(C(C(CC)(C)COC)=O)CCC2(C=C(C(=O)NCC3CSCCO3)C2)C1 76207,NC(=O)CCC(N)C(=O)N1C(C(=O)NC2COC(=O)C2)CC2CC12 76208,C=CCC(CC(C)C)C(=O)N1CCCOCC1c1ccccc1OC 76209,Cc1c(-n2nc(Cc3ccccn3)nc2CCCCS(N)(=O)=O)cccc1Cl 76210,C=C(C)CCCC(=O)N1CCCCCC1CNC(=O)CC1CCCCN1C 76211,N1(C(c2cnc(C)nc2)=O)CCC2CN(C(c3cncnc3C3CC3)=O)CC2C1 76212,c1(C(=O)Nc2ccc(C(N3C(CCC=C)CCC3)=O)nc2)cnnc(C)c1C 76213,C(=O)(C1c2c[nH]nc2CN1C(C1CCCCN1C)=O)N(CCC(=O)NC)CC 76214,C1(NC(C=C(C)C(C)C)=O)(CO)CCCN(C(C23CCCC(C2)OC3)=O)C1 76215,C1(C(=O)NC(CCNC(C=C(CCC)C)=O)(C)C)CC2CCC(C1)C2O 76216,C1(CCC)(NC(C(CC=C)C)=O)CCCN(C(c2ccc(C)c(O)c2)=O)C1 76217,C1(C(=O)NCC2(C)CC2)CC12CCN(Cc1cccc(Br)n1)CC2 76218,Cc1cnn(CC(=O)NCC(CO)NC(=O)CNC(=O)CCc2ccccc2)c1 76219,C1(C(=O)Nc2ccc(CNC(=O)ON)cc2)CC2CCCC2C1 76220,C1(C)(C(N(CCOC)CCn2cc(C3(CCO)CC3)nn2)=O)CC(C#N)C1 76221,c1(C(=O)NC2COCCN(C(C=CC(CC)C)=O)C2)cc2c(cn1)OCO2 76222,C#CC1(C(=O)NCCC(=O)OCC)CN(C(=O)CCC2CCOC2)C1 76223,C(=O)(CC(F)(F)C(F)(F)F)NCCC(C(C)C)NC(=O)C(=O)NCC1CC1 76224,C1(OCCCC(=O)ONC(COCC)C2CC2)CCCC1 76225,CCC(CC1CCCC1)C(=O)NC1CCCCC1NC(C1OCCCO1)=O 76226,N1(C(C)C)CCC(CC(=O)N(C)CC2CCN(C(C3C(C)C3(F)F)=O)C2)CC1 76227,C12(C(N(CC=C)CCO)=O)CCC(CC1NC(c1ncn(C)n1)=O)C2 76228,Cc1cc(C(=O)NCCN(C(=O)Cc2ccco2)C)n(C2CCC2)n1 76229,c1(C(C)C)cc(C(=O)NC2(CNC(=O)CC3CCCC34CC4)CCOC2)nn1C 76230,C(=O)(C1=CCN(C(c2cscn2)=O)CC1)NCC1C(C)CCCC1 76231,c1(NC2C(C)CN(C(=O)CCCC(=O)N(C)C)C2)ncc(Br)cc1[N+](=O)[O-] 76232,C(c1cn(C)nn1)=CC(=O)NC(C(=O)NC(CC=C)CC)CC1CC1 76233,c1(C(=O)NCC2C(CC(=O)NCc3ncsn3)C2)cc(Cl)n[nH]1 76234,N1(C(C(C)CN(C)C(c2ccco2)=O)=O)CCCCCCC1C 76235,c1(CCCC(=O)N(CC(C)NC(=O)Cc2ccon2)C)ccc(Br)cn1 76236,N1(C(C(C)N(C)C)=O)CC2CC(NC(c3ccsn3)=O)CC1C2 76237,N1(C(C(=O)Nc2ccc(C)cc2)=O)CCCN(C(c2cc(C)c(C)cn2)=O)CC1 76238,C(=O)(CCCC(=O)N1CC(CNC(=O)CCC(=O)c2cccc(Cl)c2)C1)N(C)C 76239,Cc1cnc2cccc(C(=O)N(C(C)CNC(=O)CSCC(C)C)C)n12 76240,N1(C(c2cn(CC=C)nc2)=O)CCC2(CC2C(N2CC(CSC)C2)=O)C1 76241,N1(C(C2C(=C)CC2)=O)CC(C)OC2(CCN(c3nc4cc(C)ccc4o3)CC2)C1 76242,C1(NC(Cc2n[nH]c(=NC)s2)=O)CC2CC(C1)N(C(C1(O)CCC1)=O)C2 76243,C=CCC(C)C(=O)N1CCC(C(F)F)(CNC(=O)CN(c2ccnc(Cl)n2)C)C1 76244,c1(C(=O)NCc2c(C)n(-c3ccccc3)nc2)cc2c3ccccc3n(C)c2s1 76245,C(CC(C)(C)C(=O)NCC(CNC(=O)C(N1CCC(O)CC1)C)OC)OC 76246,C1(C(=O)NC(c2ccccc2)C(=O)NCC(CC)C#N)CCOCC1(C)C 76247,c1(C(=O)NC2C(C(=O)Nc3cncc(CC)c3)CCC2)ccc([Si](C)(C)C)cc1 76248,N1(C(C(CC)(C)O)=O)CCOCC(CNC(=O)CCc2ccn(C)n2)C1 76249,CCC(CN(C)C)CC(=O)NC1(C(=O)NC2CC(Cl)(Cl)C2)CC1 76250,c1(CC)cccc(C(N2CCCC(NC(C3CCC4(CCC4)C3)=O)CC2)=O)c1O 76251,CN=c1[nH]cc(-c2cnc(NCC3CCO3)c(C(=O)OC)c2)cc1C#N 76252,c1(Cn2cc(C(C=C)(C)O)nn2)ccc(CNC(c2ccc(C(F)F)o2)=O)cc1 76253,C1(N(C(c2cn(C)nc2)CO)C(=O)CNC(=O)Cn2cccn2)CCC(C2CC2)C1 76254,O(NC(=O)C(F)C1(O)CN(C(c2cn(C)c(C)n2)=O)C1)CC(=C)Cl 76255,C1(C(N(CC(=O)NCC)C)=O)CCCCCN1C(C1CC(=O)N(OC)C1)=O 76256,Cc1cc(C(F)(F)F)nc(NC(c2ccc(Cl)cc2)c2ccccc2)n1 76257,c1(C(N(C2CCN(C(C(C(C)C)OC)=O)C2)C)=O)cc([N+](=O)[O-])c(C)cc1C 76258,c1(-c2nc(-c3ccc(OC)cc3)nn2C2CC2)cnc(OC)c(Cl)c1 76259,c1(CC)ccc(C=CC(=O)NC(C)C(C)(C)NC(c2ccc(O)nc2)=O)cc1 76260,C1(NC(C(c2ccccc2)N(CC)CC)=O)CC2CC2N1C(C1CC1C#N)=O 76261,c1(C(=O)NC(C(C)C)C(C)NC(c2ccc(N(C)C)nc2)=O)cn(C)c(=O)n1C 76262,c1(N(C)Cc2cccc(OC)n2)ncccc1S(=O)(=O)NC12CCN(CC1)CC2 76263,C12(C(=O)NCC(C)(CNC(=O)C(C)(C)OC(C)=O)OC)CCC(F)(CC1)CC2 76264,Cc1c(C(=O)NCC(CNC(=O)C(F)(F)CN(C)C)CO)cc(C(C)(C)C)n1C 76265,c1(C(=O)NC(C(C)(C)C)CNC(C2C3CCCC23)=O)cnn2ccccc12 76266,c1(OC)noc(C2CC2)c1C(=O)NCCC(C)NC(=O)C(C(C)C)NS(N)(=O)=O 76267,c1(CCNC(CCOCCN(C)C(C2CC2F)=O)=O)cccnc1 76268,N1(C(Cc2c(C)noc2)=O)CC(O)CCC1C(=O)NCC(C)(C)C1CCCC1 76269,CCC(C)(C(=O)OC)NC(=O)C(CNC(c1c[nH]nc1OC)=O)OC 76270,N1(C(C(C(C)C)n2cccc2)=O)CCCN(C(C2CC3(F)CC2C3)=O)CC1 76271,C1(C(=O)NC2CCC(CNC(C(C=C)(C)O)=O)C2)CCc2cncn2C1 76272,N1(C(=O)Cc2cnn(C(F)F)c2)CC2CCCC(C1)N2C(C1CCC2CC12)=O 76273,C(CSC)(CCC1(NC(=O)CSCC(N)=O)C(C(=O)OC)CC1)OC 76274,c1(C(N(C2CN(C(c3cc(C)c(C)s3)=O)CC2O)C)=O)cc2scnc2[nH]1 76275,Cc1cn2cc(C(=O)N(C)CC3CCN(C(=O)C(C)(C)C)C3)nc2s1 76276,C1(O)(CNC(C2(C#C)CCC2)=O)CCCN(C(=O)Cc2ccccc2SC)C1 76277,c1(C(=O)NCCCN(C(C2CC(C)N(C)C2)=O)C)ccc2nc(O)cc(O)c2c1 76278,C(=O)(C1=CCCC1)NC1CCC(NC(c2ccc(COC)s2)=O)C1 76279,c1(C(=O)NC(CCNC(C2ON=C(C)C2)=O)C)ccc(C)c2c1NCCC2 76280,Cc1cc(=NCCc2cnc(C)s2)[nH]c(N2CC3CC2C2CC32)n1 76281,c1(NC(C(C2CCN(C(C3C(CCC)C3)=O)C2)F)=O)ccc(NC(C)=O)cc1 76282,N1(C(CCC(N)=O)=O)CCN(C(C2CC2F)=O)C(c2cn[nH]c2)C1 76283,C(=O)(C(CC)C(C)C)N(CCCOC1CCN(C(C2C(CCC)C2)=O)CC1)CC 76284,c1(C(=O)NC2(C)CC(NC(=O)CC3=CCCC3)C2)cnc2ccsc2c1 76285,C(C)(CC(=O)NCC(c1cccs1)O)NC(CNC(C)=O)=O 76286,c1(C(=O)NC(C(N2CCC3(CC(F)C3)C2)=O)C2(C)CC2)ncc2ccccn12 76287,Cc1cc(=NCC(F)c2ccc(C)c(C)c2)[nH]c(NC2CCCn3ncnc32)n1 76288,C1(NC(c2ccccc2)C)CCOC1c1ccccc1 76289,C(C)(C(=O)OC(C)(C)C)(C(=O)N1CCC(N(C(=O)C(C)CSC)C)CC1)OC 76290,CCCC(C)(CCC)C(=O)NCCN1CCN(C(=O)C(C)(F)C(=O)OC)CC1 76291,C1(CNC(C(C)CN(C)C)=O)CN(C(c2cnc(N)c(N)c2)=O)CC(C)(C)O1 76292,C1(CC(=O)N(CCCCC)C)CCCC1NC(=O)Cc1nccn1C 76293,C(=O)(CCC(C)(C)O)N1CCCC(N(C(C(CC)OCC)=O)CC)C1 76294,C1(=O)C(CC(C)C)OCNC(=O)CCN1CC=C.C1(CC)CCCCC1O 76295,c1(C(N2C3C(NC(C(C)CC4CCCC4)=O)C(C3)C2)=O)c[nH]nc1S(N)(=O)=O 76296,N1(C(CCC(C)OC)=O)C2CCC1C(CNC(c1cn(C)nc1C(F)(F)F)=O)C2 76297,CC(C)C(C)C(=O)NCCCN(C(c1cccc(C2CC(F)(F)C2)c1)=O)C(C)C 76298,C1(CNC(CC(CC)(F)F)=O)Cc2ccccc2CN1C(=O)CC1CC(C)=NO1 76299,C(CS(=O)(=O)CC(=O)OCc1nnn(C)c1C(F)(F)F)OC 76300,C1(CNC(CCCC#C)=O)CN(C(c2cc(C)ccn2)=O)CCC12CCOC2 76301,N1(C(=O)COCC2CCOCC2)CC2(CCC(CO)O2)C1.C12CC(F)(C1)NC2=O 76302,Cc1nccc(C(=O)NCC(O)CN(C(=O)COc2c(C)occc2=O)C)c1N 76303,c1(C(=O)OC(CCC)(C)C)ccc(C(C)C)cc1 76304,C1(NC(c2ccc(C#C)cn2)=O)(CNC(C2CCCN2C)=O)CCC(C)(C)CC1 76305,c1(C(=O)NC(c2cccnc2)C(N2C(C)(C(=O)OC)CC2)=O)n[nH]c(C)c1C 76306,c1(C(N2C(CNC(=O)CCC(N)=O)CCC2)=O)cccc2[nH]ncc12 76307,N1(C(c2ccccc2)=O)C2CN(Cc3ccncc3-c3sccc3CO)CC12 76308,CCCCC(CC(=O)NC1CCC1)NC(C1CCCC(C#N)C1)=O 76309,Cc1sc(Cl)nc1C(N1CCN(CCNC(C2CCC2)=O)CC1)=O 76310,N1(C(CC=C=C)=O)CCCC1C1CCCN1C(c1nc(OC)ccc1OC)=O 76311,N1(C(CCCCOCC)=O)CCC2CN(C(=O)CC(O)CN(C)C)CC12 76312,N1(C(Cc2nc(C)sc2C)=O)C2CCC1CC(N(C)C(c1ns[nH]c1=O)=O)C2 76313,C1(C(N(C)CC2CCCN2C(C2(CO)CCCCC2)=O)=O)CCC2(CCC2)O1 76314,C1(NC(C2CCC2C(=O)OC(C)(C)C)=O)CCC(CC(=O)NC(=O)NC2CC2)C1 76315,C1(C(N2CCC(O)C2)=O)(CC)CCCN1C(=O)C=CCOC 76316,C1(C(CO)NC(Cn2c(C)nnn2)=O)CCN(C(C2C3CCC(=O)C23)=O)CC1 76317,C1(CNC(=O)CCc2ccccc2)CN(C(=O)CCC2OCCO2)CCCO1 76318,C1(C(=O)NCC(=O)NOC)(OC)CCN(C(=O)C(C)n2ccnn2)C1 76319,C(=O)(C#CC1CCCCO1)NC(N1CCCC(c2nnc(O)o2)C1)=O 76320,N1(C(c2cc(C)c(Br)cc2)=O)CCC2CN(C(C3CC=CCC3)=O)CC2CC1 76321,c1(C(C(=O)NCC2(NC(CCOCC)=O)CC2)C)ccn(C)c1 76322,CCCCC(C(=O)N(C)CCOCCN(C(=O)C(n1cc(Cl)cn1)C)C)C(C)C 76323,C1(C(N2CCCC(C)(C(N)=O)C2)=O)CCC2(CN(Cc3cc(O)cc(Br)c3)C2)O1 76324,c1(C(=O)NC2CCC(Cn3cc(COC(=N)O)nn3)C2)cccc2cnsc12 76325,C1(C(N2CCC(NC(C3Cc4cscc4C3)=O)C2)=O)CC2(CCC2O)C1 76326,[N-]=[N+]=NCC(F)CC(C(=O)O)NC(=O)C=Cc1cn[nH]c1 76327,C=CC1CN(C(=O)CN(C)C(=O)C2CC2)CC1NC(=O)Cn1cc(CC)cn1 76328,C1(C(N(C)CCC2CCCCN2C(=O)CCn2cccn2)=O)CC12CC(F)(F)C2 76329,c1(C(=O)NC(CC(C)NC(Cc2nnc(C)o2)=O)C)ccc2nc[nH]c2c1 76330,C1(CNC(c2cn(CCO)nn2)=O)CC2CC1CN2C(c1cc(Br)co1)=O 76331,c1(C(N2CCC(NC(CSC)=O)CC2C)=O)cc(S(N)(=O)=O)oc1Cl 76332,C(CC(C)(C)C(=O)N1CCC(O)(CCNC(=O)C(F)C2CCOC2)CC1)OC 76333,C(=O)(CC1CCc2ccccc21)N1C2CCC(NC(CCNC(C)=O)=O)(C2)C1 76334,C(=O)(CC1NC(=O)c2ccccc21)N1CC2CC3C(NC(C=NOC)=O)C1C2C3 76335,n1(SCC)nc(CS(C)(=O)=O)nc1C(C(N)=O)=CC(=O)OC 76336,c1(C(=O)NC2C(NC(Cc3c(C)cc(Cl)cc3)=O)COC2)cc(C)n(C)c(=O)c1 76337,C(=O)(C(C)(C)CC(C)C)NCCN(C(=O)CCCSc1ccc(Cl)cc1)CCC 76338,C=CCC(F)(F)C(=O)NC(CNC(c1ncc(F)cc1F)=O)C(C)C 76339,c1(C(=O)NCC(C)CNC(c2c[nH]nc2C2CCOC2)=O)cnn(C)c1C(F)F 76340,N1(C(C(C2CC2)OC)=O)CCC(C)N(C(c2cc3ccsc3s2)=O)CC1 76341,C(C1c2ccsc2CCN1C(=O)C(C)OCC1CC1)NC(C(C)OCC#C)=O 76342,c1(C(=O)NCC2C(C(N3C(C(=O)NS(CC)(=O)=O)CCC3)=O)C2)cc(C#N)cs1 76343,c1(OC)ccc(Cl)c(CC(=O)NC2CC(NC(=O)C(=C3CCCCC3)F)C2)c1 76344,c1(CNC(=O)NCC(C2CCC(F)(F)CC2)O)cccc([N+](=O)[O-])c1 76345,c1(OC)ccc(OC)c2[nH]c(-c3nc(-c4cc(C)cc(C)c4)no3)cc12 76346,N(C(=NCCOc1ccc(Cl)cn1)NCC(F)F)CC1CCN(C)CC1 76347,c1(CC(=O)NCC)nncn1C(N1CC2CC1C2)C(=O)NCCCOC 76348,C12(CNC(c3csnc3C3CC3)=O)CCC(F)(CC1)C2 76349,N1(C(c2cscc2C(F)F)=O)CCc2[nH]nc(CNC(C3(F)CCOC3)=O)c2C1 76350,C=C(C)CC(C)C(=O)NCC12CC(NC(c3cccc(CC)c3F)=O)(CO1)C2 76351,N1(C(C(CC)=CC)=O)CC2(CC(C(N3CCC(CC(N)=O)CC3)=O)C2)C1 76352,c1(C(=O)NC(C)CNC(C2CC2C(C)(F)F)=O)cccn2ncc(Br)c12 76353,CN1CCN(C(=O)Cc2csc(S)n2)C(CNC(C2(n3cccn3)CCC2)=O)C1 76354,N1(C(C2(CC=C)CC2)=O)CCC(NC(c2coc(C(C)OC)n2)=O)C(F)C1 76355,N1(C(CS(CC)=O)=O)CCC(CNC(=O)CCCOC)C1(C)C 76356,C1(C(N2CCC(C(=O)NC3C=CCC3)(CC)C2)=O)CCC2(CCC2)O1 76357,c1(OC)ccc(NC2CCN(c3ccnc(SC)n3)CC2C)c(O)c1 76358,Cc1ccc(C(=O)NC(C)CCN(C)C(C2(C(F)(F)F)CCN(C)C2)=O)nc1C 76359,N1(CC(C)C)CCN(C(=O)C(=O)NCCSc2ccccc2)C(C)C1=O 76360,C1(CNC(c2c(C)nsc2Cl)=O)CC2CCC(C1)N2C(=O)C(F)C1CCC1 76361,N1(C(c2c(C)scn2)=O)CC(CNC(C2(C)CC3(CCC3)C2)=O)CC12CCC2 76362,N1(C(C(=O)NCCC(C)N(C(CCN(C(C)=O)C)=O)C)C)CCCCCC1 76363,C1(OC)CC(C(=O)NCCC(C)SC)N(C(=O)CC23CCC(CC2)C3)C1 76364,C=CC(CCC)CC(=O)NCC1CC(C(=O)NCC(F)(F)C(F)F)CO1 76365,c1(C(=O)NCC2CC(NC(C(CC)(C)COC)=O)C2)ncnc2c1cnn2C 76366,c1(C(=O)NC2CCC(N(C(=O)CCc3cnc(O)[nH]3)C)C2)cc2cc(Cl)ccn2n1 76367,c1(C(=O)NC2CC(CNC(C3CC3(F)F)=O)C(O)C2)nc2ccccn2c1F 76368,c1(C(=O)NC(C)CCCNC(=O)CN2CCS(=O)CC2)cnn2c1OCC(F)C2 76369,O=C1CCC(NC(C2(O)CCCN(Cc3cnc(Br)s3)C2)=O)C(=O)N1 76370,c1(CCC)sc(C(=O)NCC2(NC(C3CC=CCC3)=O)CCOC2)cc1CC 76371,c1(C(=O)NCCc2cc(C(NOC(C=C)C)=O)no2)cncc(C=C)c1 76372,O(N(CC)C(=O)C1(F)CN(C(C2CC(CC)=NO2)=O)C1)CC 76373,N1(c2snc(CC)n2)CCCC2C(NC(=O)Cc3cnn(C(C)C)c3)C(C)(C)C12 76374,C1(NC(=O)Cc2ccccc2)CC2(CCN(C(C3CCS3(=O)=O)=O)C2)C1 76375,N1(Cc2c(C)nc(-c3ccccc3N(C)C)o2)CC=C(C2(C(=O)O)CCC2)CC1 76376,Nc1cc(-c2cn(C3CCCC3C3CC(C4CC4)=NO3)nn2)cc(F)c1 76377,C1(CNC(CN2C(C)CCCC2)=O)CCCCCN1C(=O)CC1(C)CC1 76378,C(=O)(C1=CCCN(C)C1)N(c1ccc(C#N)nc1)c1ccc(C)cc1.C(CCCl)O 76379,Cc1cc(C(=O)NCC2(CN(C)C(C3CCCC3C)=O)CC2)cc(C)c1C 76380,c1(C(=O)NC2C3CC(NC(C4CCCCS4)=O)CC23)nc2c(s1)COCC2 76381,c1(C(N2C3CC(NC(CCCOC(C)=O)=O)(C3)C2)=O)c(Cl)cncc1Br 76382,CC1CC(C(=O)N(C)CC2(NC(=O)C(F)C(F)(F)F)CC2)=NO1 76383,N1(C(c2c(CC)c[nH]c2)=O)CC(C)CN(C(=O)Cc2csc(C3CC3)n2)C(C)C1 76384,Cc1ccc(Cl)c(OCC(=O)N(C(C)CNC(=O)CCN2CCC(C)CC2)C)c1 76385,c1(C(=O)NCC(CCC)NC(=O)COCC2CCCOC2)cccn2cnnc12 76386,N1(C(C2(C)C(CC)CCC2)=O)CC2CCC(C1)N2C(C1(CC2CC2)CCCC1)=O 76387,C(C)(C)(CCCCNC(C(c1ccc(C)cc1)F)=O)NC(C1CC1C1CCCO1)=O 76388,CCCCC(CC)CC(=O)N1CCC(N=[N+]=[N-])(C(=O)NCCC(C)(C)F)C1 76389,c1(C(=O)NCC2CC(CNC(c3n(C)ncc3)=O)OC2)cnc2cnn(C)c2c1 76390,c1(CC(N2CC(C)(NC(C3CCC4C3C4(F)F)=O)C2)=O)noc2ccc(F)cc12 76391,C1(NC(Cc2c(C)cc(Cl)nc2)=O)CN(C(=O)C(C)SC(C)C)CCC12CCC2 76392,N1(C(C(=O)NCCOC)=O)CC(NC(=O)Cc2nc(C)sc2Cl)C2(CC2)C1 76393,C1(OC(=N)O)CN(C(=O)CCOCCNC(C2CSC2)=O)C1 76394,N1(C(C(CCOC)OC)=O)CCC2CCCC12C(=O)NCCC1CC(O)C1 76395,Cc1sc(=O)n(CC(=O)NCC=CCNC(=O)C(Cl)=CCl)c1-c1ccccc1 76396,N1(C(CN(C)CC)=O)CC2CC(C1)N2C(C1CC1Cl)=O 76397,N1(C(CC(C)N(C)C)=O)CC(NC(c2ccc(SC(F)(F)F)o2)=O)CC12CCC2 76398,N1(C(CN(C(=O)CCc2cnoc2)CCC)=O)CCC(CN(C)C)(OCC)C1 76399,O=C1CCC(C(=O)NCC23CCC(NC(=O)C4=CCCSC4)(CO2)C3)=NN1 76400,N1(C(C(C)O)=O)CCC2CCN(C(=O)COc3ccc(Cl)nc3)CC2C1 76401,S(=O)(=O)(CCC(F)(F)C(C)(F)F)NC(=O)CN(CC(F)(F)F)CC#C 76402,c1(C(N2C(C(CNC(CC=CC)=O)(C)C)CCC2)=O)cc2occc2n1C 76403,C1(CNC(C(C)(O)c2ccccn2)=O)C2CN(C(=O)Cc3ccc(Cl)s3)CC12 76404,C1(NC(=O)CCc2cnco2)COC2(C1)CN(C(c1ccc(O)cc1Cl)=O)C2 76405,C(=O)(C(CC(C)C)C(C)C)N(CCNC(=O)C(C)N(C)C)CC 76406,C(C1CCCN1C(=O)C=Cc1ccco1)=CC(=O)N(CCOC)CCO 76407,c1(C(=O)NCC2N(C(=O)Cn3ccnn3)CCN(C)C2)ccc2oncc2c1 76408,N1(C(CC=C=C)=O)CCC2(CCCN2C(=O)Cc2cncc(O)c2)C1 76409,N1(C(CC(C)N(C(=O)C#CC2CC2)C)=O)CC2(CNC(=O)N2)C1 76410,CCC(CC)(CC)C(=O)NC1CC2CN(C(=O)Cn3ccc(C)n3)CC2C1 76411,c1(C2CCN(C(C(C)CC(=O)c3ccc(F)cc3)=O)C2)ccc(S(N)(=O)=O)cc1 76412,CC1CC(NC(=O)CCCc2ccc(N)cc2)CN1C(c1cc(Cl)no1)=O 76413,C12(NC(c3c(C)cc(C)nc3)=O)CCCCCC1N(C(c1cn[nH]c1)=O)CC2 76414,c1(NC2(CNC(c3cccc4[nH]ccc34)=O)CCCC2)ncc2c(n1)COC2 76415,C#Cc1ccc(C(N2CCCC2CN(C(=O)C(C)OCC)CC)=O)c(F)c1 76416,C1(C(N(CCC)CCNC(=O)COCC2CCCO2)=O)CCCC12CCOCC2 76417,c1(C(C)NC(=O)N(C)CC2CCCN2C)c(F)cccc1I 76418,C(CC(CCC)CCC)NC(C(CCCNC(CSCCC=C)=O)O)=O 76419,C1(C)(C(=O)NCCCCN(C)C(C2(CC(F)(F)F)CC2)=O)CCCCO1 76420,c1(OC)ncnc(C)c1C(=O)NC1CCCC1NC(C1CC12CCOCC2)=O 76421,C(=O)(C(O)CNC(=O)C(F)CC1CN(C(C2CC(CC3CC3)C2)=O)C1)OC 76422,C(=O)(C1=CNC2=NCCCN12)NC(C)CN(C(=O)CN1CCCCC1=O)C 76423,Cc1c(N)ccc(C(N2CC(N(C(=O)CSC(C)C)C)C(O)C2)=O)c1Cl 76424,c1(OC)cc(C(N2CCCC(C(N3CCCC(O)C3C)=O)C2)=O)cc(C)c1 76425,c1(OC)c(Cl)cc(C(N2CC3(CC3)CC2CNC(=O)C(C)C)=O)nc1Cl 76426,c1(NC(=O)OC)ccc(C(=O)NC(C)(C)CCNC(=O)CC(C)CF)c(C)c1 76427,C(C)(C)(C(C)CC(=O)N(C)OC1CCCC1)NC(CC(CC)C1CC1)=O 76428,CCCCC(C(=O)NC(C)(C)CN1CCN(C(C2CSC(C)=N2)=O)CC1)C(C)C 76429,C(=O)(C1=CCCCC1)N1CC2C(CNC(Cn3ccc(C)n3)=O)C2C1 76430,c1(CC)ccccc1C(CNC(=O)C(O)CCSC)NC(=O)C(O)CCSC 76431,C1(C2CCN(C(=O)NCC3C(C)=NO3)C2)OC(C)(C)C(C)(C)O1 76432,c1(C(N(C(CNC(c2cn(CCCC)nn2)=O)C)C)=O)cc(S(=O)(=O)NC)cs1 76433,c1(CNC(CC2CC(=C)C2)=O)cc(C(=O)NCC2CC(COC)C2)cs1 76434,c1(C(=O)NCC2C=CCN2C(=O)C=CBr)ccc2nc[nH]c2c1F 76435,c1(OC)ccc(OC)c(C(=O)NCCC(C)N(C)C(C2OCCOC2C)=O)c1 76436,Cn1c(O)nc2cc(C(=O)NCC3CC(NC(C4CCCCC4F)=O)C3)ccc12 76437,c1(C(=O)NCC2CCC2NC(C2(Br)CC2)=O)ccc2ncnn2c1 76438,C(=O)(C(CC)C(=O)N(C1CN(C(c2cc(C(C)C)ccc2C)=O)C1)C)OCC 76439,N1(C(c2n(CC)cnn2)=O)CC2CC2(CNC(=O)C(C)Cc2ccco2)C1 76440,C1(OC)CC(C(=O)N(C)CC=C(C)C)N(C(=O)CC=CC(C)(C)C)C1 76441,N(C)(C1CS(=O)(=O)c2ccccc21)S(c1c(C)ccc(Br)c1F)(=O)=O 76442,c1(C(=O)NC(C2CCN(C(c3c(Cl)cn(CC)n3)=O)CC2)C)nccc(Cl)c1O 76443,C1(CNC(C2CC3CCC3C2)=O)CN(C(=O)CC2(CO)CC2)C2(CCC2)C1 76444,C=C1CN2C(=O)CCC2(C(N2CC(NC(=O)CS(=O)(=O)C3CC3)C2)=O)C1 76445,C12(CNC(C3C(C)(C)NC(=O)C3)=O)CCCC1CN(C(=O)Cc1cnccn1)C2 76446,c1(C(=O)NC2CN(C(=O)CCNC(c3ccccc3)=O)C2)cc(Cl)cc(Cl)c1 76447,C1(CC)CC(C(=O)NC2CC(CCNCc3ncccn3)C2)CCO1 76448,S(=O)(=O)(c1ccc2oc(O)nc2c1)Nc1ccnc(C(C)C)n1 76449,n1(CC)nc(C(=O)NC2C=CCN(C(C3CC(O)CN3C)=O)C2)ccc1=O 76450,c1(OC)ccc(C(=O)NCC(CO)NC(C2CCOC(=O)CC2)=O)cc1N 76451,C1(CC(N2CC(N(CCOC)C)C2)=O)CCCN1C(=O)CC(C)c1ccco1 76452,C#CCC(C)(CC)C(=O)N1CC(OC)C(C(=O)NCC(C)(C)C(C)(C)C)C1 76453,CCCCC(C(=O)N(C)Cc1nc(=O)o[nH]1)NC(c1cocc1C(N)=O)=O 76454,CC1(C)OC2OC(CN3CC(=O)N(CC4CC4)C3)C(O)C2O1 76455,N1(Cc2cccc(C(=O)OC)c2)CCC(C#N)(NC(C2CCCS2)=O)C1 76456,C1(CC(=O)NC2(CN(C(Cc3c(C)n[nH]c3C)=O)C)CC2)CCCC(C)(C)C1 76457,C(=O)(N=c1[nH][nH]c2cc(Cl)ncc12)C12C(CN(Cc3c(OC)nc(Br)cc3)C1)C2 76458,c1(OC)ccccc1CC(C)NC(=O)NNC(=O)Nc1nc(-c2cccs2)cs1 76459,C1(COC)(CNC(=O)C(O)C2CC2)CCN(C(=O)CN2CC=CC2)CC1 76460,C1(C(=O)NCC(CN(C(=O)Cn2ncc(Br)n2)C)O)CC2CC2C1 76461,C1(CNC(CC(C)n2ccnc2)=O)CC2CCCCC2N1C(C1CC(=O)C1)=O 76462,N1(CC(C)O)CCN(C(C2CCC(NC(=O)CC3CSCCO3)CC2)=O)CC1 76463,S(=O)(=O)(c1cccc(=NC2C=CCC2)[nH]1)NCCc1c(C)nn(C)c1C 76464,c1(CCNC(c2ccc(C(=O)OCC)nc2)=O)ccc([N+](=O)[O-])cc1Cl 76465,c1(CN(C)Cc2ccc(N3CCC(O)CC3)cc2)ccc(I)cc1F 76466,CC1CN(C(c2cc(C3CC3)ns2)=O)CCN1C(=O)CCCn1cc(CO)nn1 76467,c1(C(N2CC(c3nc4ncccn4n3)C2)=O)cc(Cl)cc(Cl)c1F 76468,C(C1CCOCC1)=CC(=O)NC(C(=O)NCCP(C)(C)=O)CC1CCCC1 76469,Cc1cc(F)ccc1CC(=O)NCC1CCCC1NC(C1C2CCCC12)=O 76470,c1(-c2onc(C(c3ccco3)C)n2)cscc1C#N 76471,c1(C(C)C)ccc(-c2cc(CN3CCC(C)C3c3cccc(F)c3)[nH]n2)cc1 76472,C1(C2CN(C(C(N3CCOCC3)C)=O)C2)CN(C(=O)CN(C2CCC2)C)CCO1 76473,Cc1ccccc1C=CC(=O)NCC12CC(NCS(=O)(=O)C3CC3)(C1)C(C)O2 76474,N#Cc1cccc([N+](=O)[O-])c1N1CC(OCCC(N2CC(O)CC(O)C2)=O)C1 76475,Cc1csc2c(C(N3CCN(C(=O)CS(N)(=O)=O)CC4(CC4)C3)=O)ncnc12 76476,CC(CS(C)=O)N=c1cccc(S(=O)(=O)N2CCCn3cc(Br)cc3C2)[nH]1 76477,N1(C(C(C)=C2CCC2)=O)CCC2(C1)CN(C(C1(Br)CC1(F)F)=O)C2 76478,C1(C)(C(N2CC(CNC(c3ccc(OC)s3)=O)C(F)(F)C2)=O)CCC(C)C1(C)C 76479,c1(CC)nnc(N(C)CCOc2ccccc2)n1CCOC1C=CCCC1 76480,C(C1(C)CCOCC1)=CC(=O)N(C)CC1CCCN1C(=O)CC1CC1(C)C 76481,C=C1CCN(C(=O)C(CC)C(C)C)C(C(=O)NC(C)C)C1 76482,C(CCC(CC)CC)N(C(C1C(CC)N(C(=O)C(C)N(C)CC2CC2)CC1)=O)C 76483,C(=O)(CC(C)(C)CC(F)F)N1CCC(N(C(C(C)SC)=O)C)C2(C1)CC2 76484,N12CCc3ccc(cc31)NC2=O.N1(CC)CCCC(C(=O)OC)C1COC 76485,c1(C(=O)NC2CC2CNCc2cccc(F)c2)cccc(N2CC=CC2)c1 76486,c1(C2(C(N3CCCC(NC(C4CC5CCC4O5)=O)C3)=O)CC2)ccccc1F 76487,c1(C(=O)O)cc(Cl)c(S(=O)(=O)N2CCC3CC(O)CCC3C2)c(Br)c1 76488,c1(CN2C(C(=O)Nc3ccc(OC)cc3OCC)CC2)cnn2cccnc12 76489,c1(C(=O)NCCNS(CC)(=O)=O)[nH]ccc1CNC(=O)Cc1cnc[nH]1 76490,C(=O)(C1=CCN(C(=O)Cn2ccc(C)c2)C1)NCCOCC(=O)NC 76491,C(CCCC(=O)N(C1CCN(C)C1)C)N(C(C(C)=CCC)=O)C 76492,c1(C(=O)NCCC2CCC(NC(C=CCOCCOC)=O)C2)nccc(Cl)c1C 76493,c1(C(=O)NC2(CNC(C3(OC)CCC(C)C3)=O)CCC2)ccc(C)cc1C 76494,C1(C(=O)NC2(CC)CCN(C(=O)C(F)(F)C(C)(C)O)CC2)CCn2ncnc2C1 76495,c12ccc(cc1)S(C)(=O)=NC(=O)NC1CCCc3c1cnn3C2=O.CN 76496,Cc1nn(C)cc1CC(N1CCC(NC(=O)C=Cc2ccccc2)C1C(C)C)=O 76497,N1(S(CCC)(=O)=O)CC2CCC(C1)C2Nc1ncncc1C 76498,C#CCCCCCC(=O)NCC1CCN(C(=O)C2=CCCO2)CC1C 76499,c1(CC)ccc(C(=O)NC(C)(CNC(=O)C(O)Cc2cnc[nH]2)CO)c(C)n1 76500,c1(NC(C)=O)cccc(CC(N2CC3CC2C3NC(=O)Cn2cccn2)=O)c1 76501,C1(NC(c2cc(SC)c(C)o2)=O)C2CC(O)C1N(C(=O)CC(C)(C)C1CC1)C2 76502,c1(OCC(N2CC(NC(C3CC(SC)C3)=O)C(C)C2)=O)c(C)occc1=O 76503,c1(OCC(=O)Oc2ccc(C(=O)NCC)cc2)cccc2c1CNC2=O 76504,Cc1[nH]c(C)c(C(=O)NC2CCC(NC(c3ccc(C(F)F)cc3F)=O)C2)c1C 76505,CCCCCC(F)C(=O)N1CCC(C)C1C(N1CC(C(C)OC)C1)=O 76506,C12(NC(c3occ4c3CCC4)=O)CCCCCC1N(C(C1COC1)=O)CC2 76507,N1(C(C2C(NC(C3C(CCC)C3)=O)C2)=O)CCSCC1.C(C)(=O)O 76508,C1(CNC(Cc2c(C)ccs2)=O)CCCC2(CCN(C(c3cnns3)=O)CC2)O1 76509,N1(C(C2(N(C)C)CCC2)=O)CCC(CNC(C(C2CCOC2)OC)=O)C1 76510,C(=O)(CCCCCCCCCO)NCCCN(C(=O)Cn1ccc(O)nc1=O)C 76511,C(=O)(CC1=CCN(C)CC1)N1C(C)CCC(CNC(C2CC(F)(F)CS2)=O)C1 76512,N1(C(c2cc(C)nc(C)c2)C(=O)NCCOC)CCn2c(C(=O)OC)cnc2C1 76513,c1(C(=O)NCC2CC3CCC2N3C(=O)CCc2ccoc2)cnc2[nH]cncc1-2 76514,N1(C(C(c2ccccc2)=O)=O)CCN(C(c2cc(C(F)(F)F)c[nH]2)=O)C2CC12 76515,c1(C(=O)OCc2cnn(CC)n2)ccc2oc(CC(F)(F)F)nc2c1 76516,C1(OC)CN(C(C2CC(C)N(C)C2)=O)CC1NC(=O)Cc1nn(C)cc1Cl 76517,N1(C(c2cccc(C)c2O)=O)CC2CC(C)N(C(C3CCN(C)C3=O)=O)C2C1 76518,CCC(CNC(C1C=C(C)CS1)=O)(CC)NC(=O)Cc1csnn1 76519,C1(NC(c2cn(C)cc2C(F)(F)F)=O)CCCC(NC(=O)C2=CCCC2)CC1 76520,CCCCC(O)C(=O)NC1(CO)CN(C(=O)Cc2ccc(C)c(O)c2)C1 76521,c1(N2c3c(scn3)C(=O)N3C(C4CC3CC4F)C2=O)cccc2c1CCO2.CO 76522,c12ccc(cc1OOCCC)C(C)N2.C1(CNC)CCCN(C(C)C)C1 76523,O=C(C1COc2ccccc21)NC1(CCCNC(=O)C(F)(F)C2CC2)CC1 76524,CC1(C)CC(C(N2CCC3(CC3NC(=O)CCc3cnccn3)C2)=O)C(C)(C)O1 76525,C(=O)(CC(C)(CN(C)C)C(F)(F)F)N1CC(F)(CNC(CC=C)=O)C1 76526,CC(C(F)C(=O)N1CCC(CCNC(=O)CCc2nncn2C)CC1)C(F)(F)F 76527,c1(NC(C2N(C(N(CC)Cc3ccccc3)=O)CCC2)=O)ncccn1 76528,N1(C(c2cc(C(C)C)nn2C)=O)CCC2(CCC(NC(c3cscc3Cl)=O)C2)C1 76529,C1(N=[N+]=[N-])(C(N(C(C)C)CCF)=O)CCN(C(=O)OC(C)(C)C)C1 76530,C1(F)(CNC(c2c(OC)cccc2)=O)CC2CCC(C1)N2C(C1CCC2CC12)=O 76531,C1(n2cc(NS(C)(=O)=O)nn2)CN(C(=O)C(C)NC(c2ccoc2)=O)CC1O 76532,N1(CC)CCN(CC(N2CCCC2C(C)NC(C2(OC)CCSC2)=O)=O)CC1 76533,c1(C(=O)NCC(n2cc(COCC(=O)N(C)C)nn2)C)cc(Cl)cc(Cl)c1F 76534,C1(C)(COC)CCN(C(N2CCN(C(C#N)C(C)C)CC2)=O)C1 76535,N#Cc1c(CCCNC(C2CCC3CC3CC2)=O)[nH][nH]c1=N 76536,CC1(CNC2CC23CCOC3)CCCN(C(c2ccc(Cn3ccnn3)o2)=O)C1 76537,C1(C(=O)NC(C)CNC(c2ccc(CS(C)(=O)=O)cc2)=O)CC(S(C)(=O)=O)C1 76538,c1(CN2CC(C(=O)NCCCOC=C)SCC2)c(F)cc(O)cc1F 76539,c1(C(=O)NC2CCN(C(Cc3cccc(C)c3)=O)C23CC3)ccn2ncccc12 76540,Cn1nc(C(=O)NC2(C)CCN(C(C3CC4(C3)CC(C)(C)C4)=O)C2)c2c1CCC2 76541,C1(CC)CCN(c2ncnc(NCc3cc(Cl)n(C)n3)c2C)CC1C 76542,C1(C(N2CCC(C(CC)CC)C2)=O)C=CCN(C(=O)CN(C)CC)C1 76543,c1(CC)onc(-c2ccccc2)c1C(=O)NC1CCCC1NC(=O)CCC#N 76544,C1(NC(=O)CSC2CC2)CCC2(CCN(C(C3CN4CCC3C4)=O)C2)C1 76545,C1(CNC(C2N(CC)CC2)=O)CN(C(C2OCCO2)=O)CC1C(F)(F)F 76546,N1(CC)CCCC(C(N2CC(N(C(=O)C=C(C)C(C)C)C)C(O)C2)=O)C1 76547,C1(C(=O)NC)CCCN(C(=O)CC2CCN(Cc3ncc(C)s3)C2)C1 76548,CCC(C)(CNC(C1OC2CCC1C2)=O)C(=O)NC(c1cscn1)C 76549,N1(C(C2(O)C(C)(C)OCC2)=O)CCC(C(=O)NC2CCCC(O)C2)=C(F)C1 76550,C1(NC(=O)Cc2nncs2)CCC2CC1CN2C(C1C(C(F)(F)F)C1[N+](=O)[O-])=O 76551,N1(C(C)C)CCOC(C(=O)NC23CC(CNC(=O)CC4CCCOCC4)(C2)C3)C1 76552,N1(C(c2cc(OC)nn2C)=O)CCN(C(c2cccc(OC(F)F)c2)=O)C2CC12 76553,c1(C(=O)NC2(CNC(=O)C(O)C(F)F)CCCC2)nccn2ccnc12 76554,C(C)(C)(CCC(=O)N(C)CC1(O)CCN(C(C2CCC(OC)CC2)=O)CC1)OC 76555,CP(C)(=O)CC(=O)NC1CC(CC(=O)NCc2cc(C(N)=O)co2)C1 76556,CC(=O)C1=C(c2ccc(F)cc2)N(CC(F)F)C(=S)NC1c1cccc(O)c1F 76557,C1(NC(=O)CSC(F)F)CCN(C(=O)C2=NOCC2)C(C2CC2)C1 76558,Cc1ccccc1CC(CNC(=O)C(F)(F)C1(O)CCC1)CO 76559,c1(C(=O)NC(C(C(C)C)NC(c2cc(O)cs2)=O)C)ccc2ccn(C)c2c1 76560,C1(NC(=O)CCC(F)F)CCN(C(=O)CC2CCCC23CC3)CC1O 76561,C1(CCCC)CN(C(c2csnn2)=O)CCN1C(=O)CC1CC(N(C)C)C1 76562,Cc1cc(C(=O)NC2(CCNC(=O)C=Cc3cn(C)cn3)CC2)cc(=O)n1C 76563,Cc1noc2nc(C(C)C)cc(C(=O)NCC(C)CNC(=O)Cc3cnoc3)c12 76564,C(C(CC(=O)N1CC(C)(C)CC1CNC(c1ncccc1O)=O)C(F)F)N(C)C 76565,C#CCC(O)C(=O)N1CC(F)(CNC(c2ccc(-c3ccccn3)s2)=O)C1 76566,CC1(NS(=O)(=O)CCCN2CCNC2=O)CCCNC1 76567,CN1CCCC(C)(CNC(C2COCCC2NC(C2CC(F)(CF)C2)=O)=O)C1 76568,N1(C(C(c2ccccc2)NC(C2=C(C)CC2)=O)=O)CC2CCC2(C)C1 76569,C1(NC(C(Cc2cn[nH]c2)NC(c2n[nH]cc2Cl)=O)=O)C=CCCCC1 76570,c1(OC)ccc2cc(C(=O)NC3CCN(C(c4cnc[nH]4)=O)C3(C)C)sc2c1 76571,N1(CC)C(=O)COC(C(=O)N(c2ccnc(OC)c2)C)C1c1nccn1C 76572,N1(C(CN(CCOC)C)=O)CC2(CC(NC(=O)CCSC)c3nccn32)C1 76573,C1(O)(CC(=O)N(C2CCN(C(CCc3scc(C)c3)=O)C2)C)CCCCCC1 76574,c1(CNC(=O)CC2OCCCO2)cc(C2CCCC2)ccn1 76575,CCC(C(=O)NC1CC(F)CN(C(c2cc(C(F)F)cs2)=O)C1)C(C)C 76576,S(=O)(=O)(c1cc(Br)c(Br)s1)NC1CC2(CN(C(c3nc(Cl)ccc3F)=O)C2)C1 76577,N1(C(C(CC)(C)O)=O)CCC(CCNC(=O)CCc2ncco2)C(F)(F)C1 76578,n1(CC(C(=O)NC(c2scc(C(=O)OCC)n2)C)C)nnc2ccccc12 76579,CN1CCCCC(C(=O)NCCC2(CNC(C3COCCN3C)=O)CC2)C1=O 76580,Cc1ccc(C(C)C(=O)N(CC(O)CNC(c2csc(Br)n2)=O)C)s1 76581,C(=O)(CC(C(F)(F)F)NC(c1cn(C2CC2)nn1)=O)NC(C)Cn1cnnc1 76582,C1(C(N(CC(C)NC(c2ccncc2F)=O)C)=O)C2CCC1(c1ccco1)C2 76583,c1(C(=O)NCC2CN(c3ccnc(Cl)n3)CCCO2)ccc2c(c1)CCO2 76584,C(=O)(CC(=O)N1CCC1CNC(C1CCCCO1)=O)NCC#C 76585,c1(-n2c(C(C3CCC3)O)nc(CCCC)n2)ccc(Br)cc1OC 76586,N1(C(c2ccc(CO)cc2)=O)CC2(CCCN2C(c2coc(Cl)n2)=O)C1 76587,CC(C)CC(CC(C)C)C(=O)NC(C1CCCCC1)CNC(C1CCC(O)C1)=O 76588,N1(CC(=O)NCC(C)N(C)C(C2(SC3CCCCO3)CC2)=O)CCN(C)CC1 76589,c1(C(C)NC(C2C(CNC(C3(SC)CC(=O)C3)=O)CCC2)=O)ccc(C)nc1 76590,N1(C(=O)Cn2cncn2)CCC2(CC1)CC2NC(C1(C2OCCO2)CC1)=O 76591,C12(COC)CC(NC(C)=O)(CN1C(=O)Cc1ccc(OCC(C)C)cc1)C2 76592,C1(C(=O)NC)CCCN(C(C2C3CN(CC(N4CCCCC4=O)C)CC23)=O)C1 76593,C12(NC(CCC=CC)=O)CCC(CC1)N(C(c1cc(C)c(Br)cc1C)=O)C2 76594,c1(C(=O)NCC(CC)(CC)NC(c2ccnc(C)n2)=O)ccc2nc(S)[nH]c2c1 76595,N1(C(C2(NC(CCC(=O)NC)=O)CC2C)=O)CCCC(C)(N(C)C)C1 76596,c1(CC)nocc1C(=O)N(C(C)CN(C(=O)Cc1ccnn1C)C)C 76597,c1(OC)ccc(Br)c(C)c1C(N1CC(C)(CNC(c2oncc2C)=O)C1)=O 76598,C(c1cc(OC)cc(C(=O)OC)c1)=CC(N1CCC(C)(COCC)C1)=O 76599,CC(C)C(O)C(C)C(=O)NCCC(C)(C)NC(c1ccncc1Br)=O 76600,CC1(C)COC(=O)C1NC(=O)CC1(NC(=O)CCC(N)=O)CC1 76601,C(=O)(C1=C(Cl)CCCC1)NCC1C(NC(COCc2n(C)ccn2)=O)CC1 76602,Cc1ncc(CCC(=O)NCCC2CC(NC(c3ccccc3C)=O)C2)c(O)n1 76603,Cc1cc(CC(=O)NCC(C)(C)CN(C(=O)CCC2CCC(C)O2)C)ccc1Cl 76604,c1(C(C)(C)C)nccn2cnnc12.C12C3CN(CC13)C(=O)C=CCSCC(=O)N2 76605,c1(C(N(CCCN(C(=O)CC2(C)CCCO2)C)C)=O)cnn2c(=N)[nH]cnc12 76606,C1(CN(C2CCN(Cc3ccccc3)C2)C)CCCCN1C(=O)CCCC1CC1 76607,C1(O)(CN(C(C2C(C=C)CC2)=O)C)CCCN(C(c2ccc(C)c(OC)c2)=O)C1 76608,N1(C(C2CCC(C)(N3CCC3)CC2)=O)CC2CCCC(C1)C2(O)C(F)(F)F 76609,N1(C(c2nccc(C)c2O)=O)CCN(C(c2ccc(Cl)o2)=O)C(C)C1C 76610,c1(CC(=O)OC)cscc1C(=O)NC(C)C(C)NC(c1ccsc1)=O 76611,c1(C(=O)OC)cccc(NC(=O)CN2CCC(C(N)=O)(N(C)C)C2)c1 76612,c1(C(=O)OC)cc2cc(C(N3CCN(C(=O)C(C(C)C)N(C)C)CC3)=O)sc2[nH]1 76613,N1(C(C=Cc2c(C)noc2C)=O)CC2CCC1CN2C(=O)Cc1sccc1Cl 76614,C(=O)(CCC(CF)CF)NC1CC2CC(NC(=O)C=CCF)C2C1 76615,c1(C(N2CCN(C(c3ccc(CC(F)F)cc3)=O)CC2)=O)c[nH]c2ccccc12 76616,c1(C(C(=O)NCC2(O)CN(C(C(CC)N(C)C)=O)C2)CC)ccc(F)cc1 76617,c12ccc(C(=O)OC)cc1NC(=O)C2N1CCC(OC)CC1.CCOC 76618,C(=O)(CCC(N)=O)N1C(C(C)NC(c2cnoc2C2CC2)=O)CCC1 76619,c1(C(=O)NC2(CO)CCCN(C(CN(CCOC)C)=O)C2)ccn2cccc2c1 76620,N1(C(c2cc(OC)c(F)cc2)=O)CCc2sc(-c3ccc(C(C)N)cc3)cc2C1 76621,C1(NC(CN(C(C(C)C)=O)C)=O)C(C)CN(C(=O)CCCn2cncn2)CC1C 76622,N1(C(c2nc(C(=O)OC)oc2)=O)CCCCC(NC(=O)Cc2nocc2C)C1 76623,c1(C(N2CCC(O)(CCNC(c3ccc(Cl)s3)=O)C2)=O)cnc(C2CC2)nc1O 76624,CC1CCC(NC(=O)CC2CS(=O)(=O)C2)CN1C(=O)CNC(N1CCCC1)=O 76625,N1(C(COCC(=C)C)=O)CCC(C(=O)NCC2CC(O)C23CCC3)CC1CC 76626,C#CCCCCCC(=O)NCc1nc(C(N2CCOC(CC)C2)=O)c(C)o1 76627,C1(NC(C2(CC)CCCN2C(=O)CC(C)COC)=O)CC2(CCOC2)C1 76628,N1(C(C2(c3ccccc3)CCN(C)C2)=O)CCC(NC(=O)C2CC2)C(C)(C)C1 76629,c1(NC)snc(C)c1C(=O)N(C(C)CNC(C1(C)CCC(=O)C1)=O)C 76630,c1(C(N2CCN(CC(=O)NCC3(C)CCCC3O)CC2)=O)ncn2c1CCC2 76631,C(=O)(C(CN=[N+]=[N-])NC(=O)C(C)N1CCCC1)NCCc1nc(C)[nH]n1 76632,C=CCCC(C(=O)NC1CN(C)CC1(C)C)NC(=O)C(n1ccc(C)n1)C 76633,c1(C(N2C(CCNC(Cc3c(C)nsc3)=O)CCC2)=O)cnc2c(c1)OCCN2 76634,CCC(O)(CNC(=O)Nc1ccc(F)nc1)CCC(F)(F)F 76635,CC(CN=c1[nH]c(=N)[nH]c(=NCCC(=O)N(C)C)[nH]1)Sc1ccccc1 76636,N1(C(C(C)(C)OC)=O)CCC(NC(C2CCC2)=O)C(CO)CC1 76637,C(=O)(C(C)C(O)C(C)C)NC12CC(NC(C3(CC#C)CCCC3)=O)C(OC1)C2 76638,C(=O)(C(C)C(O)C(C)C)N(CCC(=O)NCCOCC)CC 76639,C(C)(CCCC(=O)NCc1ccc(CC)s1)NC(COCCCC#C)=O 76640,C1(C(=O)NCC(CNC(C(C)SC)=O)C)CC(Br)(Br)C1 76641,CCC(C)C(O)C(=O)NC1CCC(CNC(c2cccnc2N2CCCC2)=O)C1 76642,C1(OC)CN(C(C2C(C)(C)C2(F)F)=O)CC1NC(c1cc(C)c(C)s1)=O 76643,c1(CCC(=O)NCCN2CCC(NC(C3CC4CCC34)=O)CC2)ccccc1O 76644,c1(C(=O)NC2CCC(C)N(C(C3CNC(=O)N3)=O)C2)cnc2c(c1)C(=O)CCC2 76645,C=CCCC(C)(C)C(=O)NCCCC(O)C(=O)NCCC(C)CCC 76646,C12(C(=O)NCc3ccc(CNC(C(C)C)=O)cc3F)CCOC1CCOC2 76647,C(CCN(C)C(c1cccc(N(C)C)c1)=O)(C(C)C)NC(C(OC)OC)=O 76648,c1(C(=O)NCCN(C(CCC)=O)C2CCCC2)nnn(C)c1C(F)(F)F 76649,C(CCNC(=O)CC1CC(OC)C1)(C(=O)NCCC1OCCC1(C)C)OC 76650,NC(=O)CCCCC(=O)NC1CCN(C(C2(N3CCOCC3)CC2)=O)CC1O 76651,C12CCC(CC1)NC2=O.C=CCCC(=O)NC1CCC1NC(=O)C1CC1 76652,CC(C)CC(CN=c1[nH]c(C2CC2)nc2[nH]ccc12)NC(C1CC2(CC2)CO1)=O 76653,N#Cc1cc(S(=O)(=O)NCC2CN(Cc3ncco3)C2)ccc1Br 76654,C1(O)(CNC(c2ccc(Br)o2)=O)CCCN(C(C2CCC(CO)CC2)=O)C1 76655,CC1COC2(C1)CN(C(=O)CC1CN(C(c3cnc(=N)[nH]c3)=O)C(C)(C)C1)C2 76656,C12(CC(=O)N(C3CCC3)CC(CO)OC)CCC1CN(C(c1cc(O)ncc1F)=O)C2 76657,C(=O)(C(C)(C)CCCOC)N(CCNC(c1nn(CC)nc1C)=O)C1CC1 76658,C1(CC(=O)N(CCCC(C)C)C)CC2(C1)CN(C(=O)C(O)C1CCC1)C2 76659,Cc1noc(C)c1S(=O)(=O)N(c1c(N)ccc(F)c1F)CCC1=CCCCC1.C1C(=O)N1 76660,c1(-c2ncc(C(=O)NCC3CC(NC(=O)C(O)CF)C3)s2)ccccc1F 76661,c1(C(C(=O)NC(C(=O)OC)C)N(C2CC2)Cc2cncnc2)nnc(C)n1C 76662,c1(C(=O)NC2CN(C(c3scc(C)c3)=O)C3C2C3)c(F)ccc2n[nH]cc12 76663,C#CCC(C)(CC)C(=O)NC1CCCN(C(=O)C=Cc2c[nH]c(=N)c(C)c2)C1 76664,C(=O)(C1=CNS(=O)(=O)N=C1C)NC1C(CNC(C2(COC)CCCCO2)=O)CC1 76665,N1(C(C2N(CC)CC2)=O)CCC(O)(CNC(=O)C(Br)=C(C)C)CC1 76666,N#Cc1cccc(F)c1CC(N1CCCOC(CNC(C2(CCO)CC2)=O)C1)=O 76667,c1(NC2CN(C(=O)OC(C)(C)C)CC2CO)cc(N=S(C)(C)=O)ccn1 76668,Cc1ccc(C(=O)NCC2CC(NC(=O)C(C)Cn3ccnc3)C2)cc1Br 76669,C1(N(C(=O)CCn2cccn2)C)CCN(CC(=O)N2CCC2)C1.NC1CC1 76670,c1(C(=O)NCC#CCNC(C2C(C(N(CC#C)C)=O)C2)=O)ccncc1C 76671,C1(CNC(c2[nH]c(=N)sc2)c2nnnn2CC2CCCO2)CCCC2(CCC2)O1 76672,N1(C(c2nc(CCC)sc2)=O)CCC(NC(c2ccnnc2S)=O)CC1 76673,c1(C(=O)NCC(C)CN(C)C(c2nccn2C)=O)ccc(F)c2c1CCC2 76674,c1(C(c2nnnn2CC2CC2)NCC=CCOC)ccc(C(F)(F)F)s1 76675,Cc1n[nH]c2cnc(C(=O)NC(C(C)NC(=O)C(C)(C)C(C)(F)F)C(C)C)cc12 76676,N1(C(C(CC)(C)OC)=O)CCC2(C=C(C(=O)N3CCC(N4CCCC4)C3)C2)C1 76677,c1(C(N2CCC3(CC3C(N3CC(O)(CO)C3)=O)C2)=O)cccc2c1CCC2 76678,C#CCC(C(=O)OC)NC(=O)CCC1CCCN1C(c1cnn(CC2CC2)c1)=O 76679,C1(CNC(C2(C)CCCC2O)=O)CC2CCC1N2C(=O)Cn1cncn1 76680,C(=O)(C(CNC(=O)C(C)CCOC)C(C)(C)C)NC(c1nn[nH]n1)CC 76681,C1(NC(C2CCN(C(=O)OC(C)(C)C)CC2)(C)C)CSC2CCCC12 76682,c1(C(=O)NC(CNC(CC(C)c2ccccc2)=O)CO)ccncc1Cl 76683,Cc1cc(CCC(=O)NCCCCNC(=O)C(C)c2ccsc2)ccc1Cl 76684,O=S(=O)(c1ccc(Br)cc1N1CCC2(CCSC2)C1)NCCc1cccc(Cl)c1 76685,c1(C(N2CC3=C(CN(C(C=CC(=O)O)=O)C3)C2)=O)csc2c(Cl)cccc12 76686,CC(C(=O)OCC1(O)CCC(C)(C)CC1)C(C)S(C)(=O)=O 76687,Cc1ccc(COCCC(=O)NCC2CN(C(=O)CCSC(=N)N)CCO2)cc1 76688,C1(C)(C(=O)NC(C)(C)CF)C=CCN1C(C1CC1(F)Cl)=O 76689,S(=O)(=O)(CC(=O)N1CCCC1CCCNC(C1CC2(CSC2)C1)=O)N(CC)CC 76690,O=C(N=c1[nH]nc2ccc(Br)cn12)N1CCc2cc([N+](=O)[O-])ccc21 76691,C1(CNC(CCc2onc(C(C)C)n2)=O)CCCCN(C(c2coc(Br)c2)=O)C1 76692,C1(CCNC(C2(C#C)CC2)=O)C(C)CCCN1C(c1cccc(NC(C)C)c1)=O 76693,C1(NC(C(CC)N(CC)CC)=O)CN(C(=O)CC2COCCOC2)CCC1F 76694,C1(C(N2CC(C(=O)N(C3CSC3)C)(CC)C2)=O)CCNC(=O)C1 76695,c1(OC)ccc(C=CC(=O)NCC(Cn2cc(C3CC3)nn2)OC)cc1Cl.CCO 76696,c1(C(=O)NCC(C)CN(C)C(c2cc3n(n2)CCC3)=O)cncc([N+](=O)[O-])c1 76697,c1(C(=O)NCC2CCCCC2F)c[nH]cc(Br)c1=O 76698,N#Cc1ccc(F)c(C(=O)NC2CC2CNC(c2cc3sccc3s2)=O)c1 76699,C=CCC(CC(=O)N(C1CC2CC2C1)C)NC(=O)C(O)c1ccco1 76700,C1(NC(C(C)C2CCCO2)=O)C2CC(NC(=O)CP(C)(C)=O)CC12 76701,N1(C(C2CC(C#N)C2)=O)CC2CC(NC(c3ccoc3)=O)CC2C1 76702,C1(NC(C(CC)CN(C)C)=O)COCCN(C(C2CN(C)CCN2C)=O)C1 76703,c1(C(N2CC(NC(C#CC(C)(C)C)=O)C(CO)CC2)=O)cc2ccc(F)cc2s1 76704,c1(C(=O)NC2CN(C(c3ccc(C)c(N)c3)=O)CC2C)ccc2[nH]nc(O)c2c1 76705,N1(Cc2ccc(C)nc2)CCC(O)C(C(N2CC3C(C(=O)O)C3C2)=O)C1 76706,C=CC(C)(CCOC)C(=O)N1CCOC(CN(C)C(C2CC(O)(C#N)C2)=O)C1 76707,C1(CNC(C(c2ccn(C)n2)C)=O)CC(C)N(C(=O)CC2CC3(CCC3)C2)C1 76708,c1(C(N2CC(NC(C(C3CCCOC3)OC)=O)(CO)C2)=O)ccc(N(C)C)cn1 76709,C12(NC(c3ccc(O)nn3)=O)CC(C1)N(C(c1cncc(F)c1)=O)C2 76710,C(CC(C(C)(C)C)NC(c1nsnc1O)=O)N(C(Cc1ncc(C)s1)=O)C 76711,N1(C(C(C)(C)SC)=O)CC2CCOC2(CNC(c2n[nH]c3cccnc23)=O)C1 76712,C1(C(=O)NC(CC)C(C)C)C=CCN(C(c2ccn(CC)c2C)=O)C1 76713,C1(O)(C(=O)NCc2c(C(=O)NCc3c(C)noc3)n(C)nn2)CCC(C)CC1 76714,N1(C(C(CC(C)C)=O)=O)CCCC12CCN(C(=O)C1CCCc3ncnn31)CC2 76715,C1(NC(CC(C)(C)F)=O)CC2CCC(C1)N2C(c1ccc(Cl)c(N)c1)=O 76716,C(CCCCCNC(=O)C(C)(C)CNC(C1C=CCC1)=O)OC 76717,Cn1c(C(N2CC3CC(NC(C4(C(C)(C)O)CC4)=O)CC2C3)=O)cnc1[N+](=O)[O-] 76718,O=C(C#CC1CCOC1)NCC(c1ccccc1Br)NC(CC(O)CO)=O 76719,c1(-n2c(C3CCCN(S(C)(=O)=O)C3)nc(CS(C)(=O)=O)n2)cc(Cl)nc(Cl)c1 76720,c1(C(c2nnnn2C)NC(c2c(F)cccc2F)C)cccc(F)c1Cl 76721,c1(C(N2CCCC(C)(NC(C3C(OC)CCC3)=O)C2)=O)cc(O)cc(F)c1F 76722,CC1CC(C(=O)NCCOCCC2CC2)CCN1C(C1CC2CC(=O)C1O2)=O 76723,C1(N(C(=O)Cc2cnccn2)C)CC2CCC(C1)N2C(=O)Cc1nn(C)cc1Cl 76724,N1(C(Cc2scc(C)c2)=O)CCCC(C2CCN(c3cncc(Cl)n3)CC2)C1 76725,C1(C(=O)NC(C2CN(C(C3CC(=O)N3)=O)C2)C)CCCCC12OCCO2 76726,C1(C(=O)NC2CCC(CC)CC2)CCC2(CN(Cc3cnc(Cl)s3)C2)O1 76727,N1(C(C(C)=CC)=O)CC2(CCNC(=O)CSc3nnc(S)s3)CCC1C2 76728,c1(CC(N2CC=CC(NC(C3(CC)CCC3)=O)C2)=O)c(C)cccc1C 76729,Cc1nn(C)cc1C(N1CC2C(NC(C3(C)CC3(Cl)Cl)=O)C2C1)=O 76730,C1(CC(=O)NC(C)CN2CCCC2)CCN(C(=O)C(C)OC(C)(C)C)C12CCC2 76731,c1(C(=O)NCC2CCSCC2)ccc(-c2cc3sccc3s2)c2cc[nH]c12 76732,c1(C(=O)NC(C(C)C)CCN(C(=O)CC(C)(C)F)C)cccc2nc(O)n(C)c12 76733,n1(CC)cc(C(=O)NCC(O)CCNC(c2cnc(C(C)(C)C)[nH]2)=O)c(C)n1 76734,CCCC(CC)C(=O)NC1CCC(NC(c2ccc(Br)cc2N)=O)CC1 76735,c1(CNC(c2ncc(-c3cnn(C4CCCC4)c3)s2)=O)ccc(OC(F)F)c(F)c1 76736,C#Cc1ccc(C(=O)NC2CC(CO)N(C(c3ccnnc3C)=O)C2)c(F)c1Cl 76737,C1(NC(C2CC23CC3)=O)CC2CCC1N2C(c1cc2[nH]ccc2s1)=O 76738,CC(CC1CC1)(CO)CN=c1nc(N2CCCc3ccccc32)c2sccc2[nH]1 76739,c1(C(N(CCCN(C(=O)CCC(F)F)C)C)=O)cnc2ccoc2c1 76740,C1(CNC(C(C)c2ccco2)=O)CC2CN(C(=O)C=Cc3ccc(Cl)s3)CC12 76741,c1(C(=O)OC)cc(C)c(C(N2CCCCC2Cn2cc(CCCSC)nn2)=O)o1 76742,c1(NC(C(CC2CCCC2)NC(CC(C)(C)O)=O)=O)ccc(O)c(CO)c1 76743,C1(N(C(=O)C2CC2)CC)CCN(C(=O)CCCNC(c2ocnc2C)=O)CC1 76744,c1(NC(C2C(C(=O)Nc3cc(F)c(OC)c(F)c3)C2)=O)nc2cc(Br)cnc2[nH]1 76745,C1(C(=O)NCCN(C(C(C=C)O)=O)CCOCCO)CC2(CCOCC2)CO1 76746,ClCCCN=C(NCCN1CC2CCC1C2)NCc1ccc(Br)cc1 76747,C(CC(CO)NC(=O)CC1CC(NC(C2CC2c2cccs2)=O)C1)SC 76748,N1(C(C)=O)CC(C2CC2C(=O)N(CCOC2CCOC2)C2CC2)C1 76749,Cc1cc2c(=O)n(C3CCN(c4ccc(Br)cc4)C3=O)cnc2cc1F 76750,C1(C(N(CC(=O)N(C(C)C(=O)NCC)CC)CCC)=O)COCC1(C)C 76751,Cc1cn2c(C(N3CC4(C3)CN(C(C3(C)CCC3C(N)=O)=O)C4)=O)c(C)nc2s1 76752,CCCC(C(=O)N(C(C)CC(=O)NCC1(Cl)CC1(F)F)C)NC(C)=O 76753,N1(C(C2C=CC(NC(C(C)c3ccccc3)=O)C2)=O)CCCC12CCNC2=O 76754,C#CCC(O)C(=O)NCC1(CN(C)C(c2cscc2Cl)=O)CC1 76755,c1(C(N(C(c2ccccc2)CC)C)=O)sc(NC(c2occc2Br)=O)nc1C 76756,N1(C(C(=O)NC2C(N3CCC(C)(C)CC3)CCC2)=O)CCCC(O)(C(F)F)CC1 76757,Cc1cc(CCC(=O)NCC2CC(NC(=O)C(F)C(F)(F)F)C2)ccc1Cl 76758,c1(OC)cnc(C(=O)NCCNC(C2CC(=O)CCO2)=O)cn1 76759,CC1CN(C(c2cn(C)cn2)=O)CC(CCNC(=O)C(C)N2CCCC2)O1 76760,N1(C(C(F)=CC)=O)CCCC(O)(CN(C(=O)C(C)(C)CC)C)C1 76761,C(=O)(C(C(C)C)NC(=O)CC)NC(c1cn(CCCCC=C)nn1)C 76762,c1(C(N2C(C(N(C(C(=O)OC)C)C)=O)CC2C)=O)cc(C)ncn1 76763,C1(NC(c2cc(C)nc(C)n2)=O)CCC12CCCN(C(=O)C=CC1CCCC1)C2 76764,c1(C(=O)NC2CN(C(C3(CCC=C)CC3)=O)CC2F)cccc2c1C(F)(F)CC2 76765,C(CSC)(C(=O)N=S(C)(=O)c1cnn2c1CN(C(=O)C=C1CC1)CC2)OC 76766,C(=O)(CCCN(C)N=O)N1CC(COC)(CNC(=O)C(C)C(C)C)C1 76767,N1(C(COCCOCC)=O)CCCC(O)(CCNC(c2c[nH]c(=N)cc2C)=O)C1 76768,C1(NC(C(CCCOC)C)=O)CC2CCC(C1)N2C(c1cc2occc2s1)=O 76769,C1(C(=O)NCCN(c2cnc(C#N)cn2)CC)CS(=O)(=O)CC(=O)N1 76770,Cc1ccnn1CC(N1CCC(C2CCCN2C(c2ccc(Br)o2)=O)C1)=O 76771,N1(C(CC2N(C)CCC2)=O)CC2(CCCC2NC(c2cn3ncccc3n2)=O)C1 76772,c12cc(ccc1F)C(=O)NC2.C(C)(C(C)(C)SC)NC(=O)CSC(C)(C)C 76773,C(=O)(CS(=O)(=O)C(C)C)NC(C(C)NC(c1n(OC)cnc1C)=O)CO 76774,CCCCCCC(=O)N(C1CCCN(C(c2c(CC)cnn2CCO)=O)CC1)C 76775,N1(C(CCCC#C)=O)CCN(C(=O)CCc2csc(Br)c2)CC1CC 76776,Cc1cc(NCC2CCC2(F)F)ncc1S(=O)(=O)NC(CO)C1CC1 76777,c1(CC)cc(CN2CCC(C(=O)NC3CCCN(C(C)=O)C3)CC2)ccc1F 76778,C1(NCc2c3nc(C)oc3ccc2)CC2CC3(CC2C1)OCCO3 76779,C1(=CCNC(C(C2CCC(=O)N2)C)=O)CCN(C(=O)CCF)CC1 76780,C12(C(=O)Nc3cncc(C#C)c3)CCCC1N(C(=O)CN1CCNC1=O)CC2 76781,C12(CNC(CCC=C)=O)CC1CN(C(c1cc(C(=O)C(C)C)c[nH]1)=O)C2 76782,C(=O)(CC(C(F)F)NC(=O)CC1(NC(C)=O)CC1)NCC(=C)C(F)(F)F 76783,Cc1c(C(=O)NC(C)(C)CCNC(C2(C)CCCC2O)=O)cnn1CCC#N 76784,C1(NC(=O)CCN2CCCC2)CC2C1CCN2C(C1CCOC(=O)CC1)=O 76785,c1(C(=O)NCC2(C)CCC(NC(C(C)C3CCC3)=O)CC2)cccc2c1CCC2 76786,C1(C(C)C)(CO)CCN(C(C2CC(C)N(C(=O)CSCCC#N)C2)=O)C1 76787,C1(CNC(C=CCC)=O)CCC(NC(=O)C(F)(Cl)c2ccccc2)CC1 76788,C(=O)(C1c2ccccc2C2CC1C2)NCC1(C)CC(NC(C=CC=CC)=O)C1 76789,Cc1ccc(-c2ccc(C3CCN(Cc4ccnc(Cl)c4Cl)CC3)cc2)c(F)c1 76790,c1(OC(C)C(=O)NC2CC2NC(=O)Cc2ccccc2)ccc(Cl)c(F)c1 76791,c1(N(CCOCC)CC)nc(NC(C2CCCCC2)CO)c2c(ncn2C)c1 76792,CC(O)C(C)(C)C(=O)N1CCN(C(=O)CCN(C)C(C2CCCC2)=O)CC1 76793,CC1(CNC(c2cc3occc3s2)=O)CCCN(C(C2C(F)(F)C23CC3)=O)C1 76794,c1(C(=O)OC)cc(Cl)cnc1NCC1NCCC1C1CC1 76795,c1(OC)cc(N(C)C)ccc1C(=O)NCC(C)(C(C)C)NC(=O)CC(C)F 76796,c1(CC(=O)NCC#CCNC(C2CCC(C)C2)=O)cc(Cl)ccc1[N+](=O)[O-] 76797,N1(C(c2c(C)nc(O)nc2C)=O)CCC2(CCOC2)C(CNC(=O)CNC=O)C1 76798,C1(NCCN2CC(N(C)C)C2)CC12CCN(Cc1ccccc1)C2 76799,CC1(C)OC(=O)NC1C(=O)NCC1CC(NC(=O)COc2ccc(C#N)cc2)C1 76800,C1(C2CC2)(CNC(CC2C(C)(C)CCCC2)=O)CCN(C(C2SCCCS2)=O)C1 76801,c1(OC)ccc(C(=O)NC2CN(C(=O)CCCCN(C)C)CC2C)c2[nH]ncc12 76802,c1(C(=O)NCC(CNC(C2CCOC2)=O)OC)ccc(C)c(Cl)c1 76803,C12(NC(c3c(C)cc(=N)[nH]c3)=O)COCCC1CN(C(c1c(Cl)n[nH]c1C)=O)C2 76804,c1(C(N(C)C)C2CC2)cn(CCC(N2CCCC2C(N)=O)=O)nn1 76805,N1(C(C(CC)N(CC)CC)=O)CC(NC(=O)CC(CC)C2CC2)C(C)C1 76806,N1(C(C2C(CNC(CN3CCN(C)CC3)=O)CCC2)=O)CCOC(C)(C)C1C 76807,n1(CC)ncc([N+](=O)[O-])c1C(=O)NC1CCCC(NC(c2csc(C)n2)=O)C1 76808,CC1(C)CN(CC(=O)NCCCCNC(c2cnc(-c3ccccc3)s2)=O)C1 76809,C(=O)(C1=NN(CC(C)C)C(=O)CC1)N1CC(N(C(C(CC=C)(C)N(C)C)=O)C)C1 76810,C12(NC(c3c[nH]c(=NC)o3)=O)CCCC(NC(=O)COc3ccccc3Cl)(C1)C2 76811,c1(C(=O)NC2CCC(NC(c3cc(C(C)=O)sc3)=O)C2)ccc2c(c1)ncn2C 76812,N1(C(C(C2CCC2)OCC)=O)CC2CCC1C2NC(c1nccnc1CC)=O 76813,c1(OC)ccnc(C(N2CC(NC(C3OCC4CCCC34)=O)C(SC)C2)=O)c1F 76814,C(C(C(F)(F)F)n1cncn1)NC(=O)Nc1cccc(OC(F)(F)C(F)F)n1 76815,c1(C(CO)N(C(=O)CC2(CN)CCOCC2)C)ccc(F)cc1 76816,c1(N2C(CC)CN(C(=O)Cc3cccc(SC)c3)CC2)ncc(C#N)cc1Cl 76817,C1(CNC(c2cnc(C(C)OC)s2)=O)C2CN(C(=O)Cn3nnc(=N)[nH]3)CC12 76818,c1(OC(C)C)cccc(C(N2CCCCC2C2CCN(CC#N)C2)=O)c1 76819,Cc1ccc2c(c1)CCN2C(c1ccc(NC(=O)Cc2nncn2C)cc1)=O 76820,c1(CNC(C(C)N(CCN(C)CC)C)=O)ccc(F)c(OC)c1 76821,Cc1ncoc1C(=O)NCC1CCCC1NC(=O)C(C)c1ncco1 76822,C=CCCN=C1NN2CCC(N1)CC=NC=C2.C1(C)CCN(CC(F)(F)F)CC1 76823,Cc1ccc2cc(C(N3CCN(C(c4cnc(O)o4)=O)CC3C)=O)[nH]c2c1 76824,C1(C(=O)OCC)CN(C(=O)C(CC)NC(=O)CSc2nc[nH]n2)CCC1O 76825,C1(NC(C2(CNC(C(CC)C)=O)CC2)=O)CC(=O)N(COC)C1 76826,C1(CNC(CCC#CC)=O)CCCC2(CCN(C(=O)CNC(=O)NC)CC2)O1 76827,C1(C(=O)NC2(C3CN(C(c4[nH]cc(C(C)=O)c4)=O)C3)CC2)CCCC(C)(C)CC1 76828,C1(C(=O)NCC(C)C(=O)NCc2ccoc2)C(C)(C)C1(C)C 76829,C1(CNC(CCOCCOCCCCC)=O)CN(C(c2cc(C)sn2)=O)CCO1 76830,c1(CNC(C(COCC)NC(=O)C=CC(C)CC)=O)ccc(F)cc1F 76831,c1(N(C(C(C)Cc2ccc(Cl)cc2)=O)C)ccc([N+](=O)[O-])nc1 76832,c1(C(=O)OC)cc(NC(c2ccc(NC(C3CC(O)C3)=O)cn2)=O)n(C)n1 76833,C#Cc1cc(F)c(C(=O)NCC(C)N(C(c2cc(C)c(F)cn2)=O)CC)c(F)c1 76834,C=C(C)CC(C(=O)N)OC.C1C(=O)N(C)CCN(C)CCO1.C1CS1 76835,c1(CNC(N2CC(N(C(=O)CC3(C)CCC3)C)C2)=O)cc(Cl)ccn1 76836,c1(C(N2CCC(N(C)C)C2)C(=O)Nc2ccc(Cl)cc2F)ccc2occc2n1 76837,N1(C(CCCCN(C)C(c2cc(C#N)c[nH]2)=O)=O)CC2C(C1)C2(F)F 76838,C1(C(N2CC(C(C)NC(=O)COc3cccc(F)c3)C2)=O)CCc2nc[nH]c2C1 76839,c1(C(c2n(CCC)nnn2)NCCCN2CCCCC2)ccnc(C)c1 76840,C(CC1CC1)(C(=O)NCc1csc(C2CC2)n1)NC(C(C)n1cncn1)=O 76841,C1(NC(C)=O)CC(CNC(=O)CCc2c(F)cccc2F)C12CCC2 76842,CC(C)(C)CCCCC(=O)NC1CCCCN(C(C2C(Cl)(Cl)C23CC3)=O)C1 76843,C1(CC(=O)NCC(C)(O)C2CC2)CCCCN1C(=O)CN1C(=O)CNC1=O 76844,Cc1noc(Cl)c1CC(=O)NC(C1CN(C(=O)CC2(CSC)CC2)CCO1)C 76845,C1(NC(c2c(COC)cco2)=O)CN(C(=O)CCc2nc(C)c(C)[nH]2)CC1SC 76846,C1(NC(C(C)C2CCC2)=O)CC2CCC(C1)N2C(=O)CCCN(C)C(C)C 76847,c1(OC(C)C(=O)NCC(O)CNC(=O)C=CC=C(Cl)Cl)cccc(N)c1 76848,C1(F)(CNC(CCOCC#C)=O)CCN(C(c2ccnnc2O)=O)C1 76849,c1(CC(=O)NC(CN(C(C2C(OC)C2)=O)C)C)ccc(C(N)=O)nc1 76850,C1(CC(N2CCN(C(c3csc(Cl)c3)=O)C(CO)C2)=O)CCC2(CCC2)O1 76851,C1(CC)CC(C(=O)NCC(C2CCCCC2)O)CCN1C(=O)C(C(C)(C)C)OC 76852,c1(CCN2CC(OCC)C(O)C2)oc2ccccc2c(=O)c1C.N1(C)CCN(C)CC1 76853,N1(C(CC(C)NC(C2(CO)COC2)=O)=O)CC2OC(=O)N(C)C2C1 76854,c1(C(=O)NC(CCC(=O)NCC2C(C(=O)OC)C2)C)cnc(O)c(F)c1 76855,c1(C(=O)NCC(CC)NC(C=CC=CCCCCC)=O)ncc(F)cc1F 76856,c1(C(CC)Nc2cc(OC)ccc2OC)cc(C)cc(Br)c1OC 76857,CC1CCCN(C(c2cn(C)nc2C2CC2)=O)C1CNC(C1CC2CC1C1CC21)=O 76858,N1(C(C(C)Cc2ccco2)=O)CCCCC1C1(NC(C2CCCSC2)=O)CC1 76859,C1(N(CCC)C(C2CC2(C)C)=O)CCN(C(=O)Cn2ccc(Br)n2)C1 76860,C(=O)(C1=C(CCl)N(CC(F)F)C(=S)NC1c1nccc(Cl)c1Cl)OC(C)(C)C 76861,CC1CC2CC2CC1C(=O)N(CCNC(c1csc(=N)[nH]1)=O)CC1CC1 76862,C(=O)(CC(C)(C)CN(C)C)NC1(C)CN(C(C2N(C(C)=O)CSC2)=O)C1 76863,C=C(I)CC(=O)NCC1(NC(=O)CN2CCCCC2)CC1 76864,C(=O)(C1=NOC(C)(C)C1)NC(CNC(c1csc(C)c1N)=O)C1CC1 76865,C1(C(N2CC(C)C(NC(=O)C(c3ccc(Cl)cc3)=O)C2)=O)CCCCN1N=O 76866,c1(C(=O)NCCN(C(COCCC)=O)CCc2ccccc2)cccn(C)c1=O 76867,C1(C(=O)NCC=C(COC)C)(CN(C(CC(=O)CC2CC2)=O)C)CCCC1.C1(SC)CC1 76868,c1(CC)cc(C(=O)NCC(C)(C)OCCNC(=O)C(C)CC2CCCC2)c(C)o1 76869,C1(C(=O)NCCCN(C(C(C)NS(CC)(=O)=O)=O)CCO)Cc2ccccc2S1 76870,N1(C(C(C)=C(C)C)=O)C(C(=O)NCc2ccc(C)nc2)CCC1C(C)C 76871,N1(C(C2CCN(S(C)(=O)=O)C2)=O)CCOCC(C)(CN(C(=O)C=C2CC2)CCO)C1 76872,Cc1ccc(F)cc1C(=O)NCC1(CNC(=O)CCOCC(C)C)CCCC1 76873,c1(C(=O)NC(C2CCOC2)C2CC2)cc(C2CC2)ncn1 76874,N1(C(C(COC)OC)=O)CC2(CC(NC(c3cnnc(C)c3C)=O)CO2)C1 76875,CC1CC=C(C(=O)NC(C(=O)NCCc2ncon2)c2cccs2)CC1 76876,C(=O)(CCC[N+](=O)[O-])N1CC(N2CCN(C(C3C(C=C)CC3)=O)CC2)C1 76877,C1(CNC(CC(CN(C)C)O)=O)C2CCCC1N(C(c1csc3nnsc13)=O)C2 76878,C(=O)(CCCCc1cnc[nH]1)NC(C)CC(C)NC(C1CCC(F)C1)=O 76879,C(=O)(C1=NNC(=O)CC1)NCC1C(NC(C(CCC)NC(C)=O)=O)COC1 76880,C(C(C)C(=O)NC(c1cn(C)nn1)C(=O)NCCC1(O)CCOC1)SC 76881,Cc1cccc(OC(C)C(=O)NCCCNC(C2(C3CCCO3)CCCC2)=O)c1 76882,C1(O)(C(=O)NCC)CCN(C(C2CCCN(c3ccc(Br)cc3)C2=O)=O)CC1 76883,CC1CN(C(=O)CC2(NC(c3ccc(F)s3)=O)CCCCC2)CC1F 76884,CC(O)C(C)(C)C(=O)N(C)CC1CN(C(c2ccc(CN(C)C)cc2)=O)CCO1 76885,c1(C(N2CC3CCCC(C2)N3C(c2cnc(Cl)[nH]2)=O)=O)cc2c(s1)CCCCC2 76886,N1(C(COCCOC)=O)CC2(CCN(C(=O)CN3CCCCC3=O)CC2)CC1C 76887,C(C(=O)NOCC1CC1)N(C(=O)C=Cc1cc[nH]c1)CC#C 76888,c1(NC(C2C(C(=O)NC)C2)=O)cc(Br)cn2ccnc12 76889,N1(C(C)=O)CCCCC1C(=O)NCCCCC(C)NC(=O)Cc1ccc(F)cc1 76890,C(=O)(C1CCCc2cncn21)NC1CC(NC(Cc2ccc(C#N)cc2F)=O)C1 76891,c1(C(=O)OC)cccc(Cl)c1Cl.N1(N2c3ccccc3OC2)CCN(C)C(C)C1 76892,c1(C(CNC(c2c(C)cns2)=O)NC(=O)CCOC2CC2)ccccc1F 76893,C(=O)(C(C)C(O)CC(C)C)NC(C(=O)NCC(COC)C)CC1CCOCC1 76894,Cc1nc2ccncc2cc1C(=O)NC1CCN(C(=O)C=CC(C)C)CC1F 76895,c1(N2CC3C(CNC(c4cc(OCC)no4)=O)C3C2)ncnc2c1cnn2C 76896,c1(C(=O)NCC(CC=C)NC(C2CC(Cl)(Cl)C2)=O)cnn2ccccc12 76897,N(C(=NCc1cc(-c2ccco2)on1)N1CCC(OC)C1)C1CCN(CCC)C1 76898,C1(NC(C(=C(C)C2CC2)F)=O)CC(C)N(C(=O)Cn2cncc2C)C1 76899,Cn1ncc2c(SCC(=O)NCc3cccc(Cl)c3)ncnc12 76900,c1(CNC(C2CCCC2NCC2CCC(F)(F)C2)=O)cc(Br)c(Br)s1 76901,C1(CCCC)CCCN(N(Cc2cccc(C)c2)CC(F)F)C1 76902,C(=O)(C1=CC(O)C(NC(C2(CCF)CCC2)=O)C1)Nc1c(CC)noc1 76903,N1(C(CC(C)CNC(c2ccc3c(c2)CC3)=O)=O)CCC2(C=CCO2)C1 76904,C1(C2N(C(c3c(C)noc3)=O)CCC2)CCCN(C(=O)CC(=O)N(C)C)C1 76905,N1(C(c2c(CC)con2)=O)CC2CCC1C(CNC(C13CC(OC)C1C3)=O)C2 76906,C#Cc1ccc(C(=O)NC2CCN(C(=O)CN(C3CCC3)C)CC2O)c(OC)c1 76907,CC1CCCC1(C)NC(C1CC2CC2N1C(c1ccc(CF)cc1)=O)=O 76908,c1(C(N(CC(C)N(C(c2c(CC)noc2)=O)C)C)=O)nc(C)c(C)nc1O 76909,N12CC3CC1CN3C2=O.c1(SCCCNS(C)(=O)=O)ccccc1 76910,N1(C(C2CN(C(C)=O)C2)=O)CCC(CNC(=O)CC2CC3(CC3)C2)C(O)C1 76911,C1(C(=O)OC)CN(C(=O)C(N2CCC(NC(=O)NC)CC2)=O)C(C)CO1 76912,c1(C(N2C(C(=O)NC(C)C(=O)NCC(C)C)(CC)CCC2)=O)cn(C)c(=O)cn1 76913,C=CCCCCCCC(=O)NCc1nnn(C)c1C(=O)NCC(O)CN(C)C 76914,Cc1cc(C(N2CCC(CO)(NC(=O)Cc3cncnc3)CC2)=O)c(C)cc1Br 76915,C(=O)(C(O)CCCc1ccccc1)NC1C(C)CN(C(c2ccnnc2O)=O)C1 76916,c1(C(N(CCC)CCNC(C2(F)CC2)=O)=O)cc(F)c(O)c(F)c1 76917,c1(CCC(=O)NCC2C(NC(CNC(CCC)=O)=O)CC2)ccn(C)n1 76918,C1(N(CC(F)CCOCC2(SC)CC2)C)CCC(COC(C)(C)C)O1 76919,C1(O)(CN(C(c2cnc(C(C)C)[nH]2)=O)C)CCCN(C(C2CC23CC(O)C3)=O)C1 76920,C1(C(N(C2CCCC2)CCNC(c2ccc(C3CC3)o2)=O)=O)CC2(C)CC1CO2 76921,CCCC(C(=O)NCCC1CN(C(c2nc(Cl)sc2Cl)=O)CCO1)NC(N)=O 76922,c1(C(N2CCCC(NC(c3nccc(C)c3)=O)C2C)=O)cnc2c(F)cccn12 76923,C=CCCC(C)(c1nnnn1C(C)(C)C)NCC1(C=C)CCC1 76924,N1(C(c2c(CC)nccn2)=O)CC(NC(C2CCSC2)=O)C(C)(C)C1 76925,N1(C(CCC)C)CC2C(C(=O)NCc3noc(-c4ccccc4)n3)C2C1 76926,Cc1cc(Br)ccc1C(=O)NCCC1CN(C(=O)C(C)NC(N)=O)C1 76927,c1(NC(N)=O)csc(C2CCCN2S(=O)(=O)CC2CNC2)n1 76928,C1(CNC(c2cc(OC)no2)=O)CN(C(C2SCCS2)=O)CCCO1 76929,C1(C(=O)NC23CC(C(=O)NCc4cncs4)(C2)C3)CCC=CCC1 76930,c1(C(=O)NCc2ccc(C(=O)OCC)cn2)c(C(F)(F)F)nn(C)c1C 76931,CCC(C)(COC)C(=O)NCC(C)N(C(=O)Cc1cccc(C(N)=O)c1)C 76932,c1(C(CNC(C=C(C)C)=O)NC(=O)CC2COCCO2)cccc(Cl)c1 76933,C12(CNC(c3cnns3)=O)CC1CN(C(=O)C(C1CCCCCC1)O)C2 76934,c1(NC2CCN(C)C2)cc(NCc2cc[nH]n2)ncn1 76935,C(CCC(=O)NCC(F)CNC(=O)CNC(c1ccsc1)=O)N(C(C)=O)C 76936,c1(OC)c(CNC(CCC=C(C)C)c2ccccc2)ccc2ccccc12 76937,C(=O)(CC1=NNC(=O)C1)NC1CC(CC)(CC)N(C(C2(F)CCOC2)=O)C1 76938,c1(CC(=O)N(C)CC2COCCN2C(C2CCSCC2)=O)ccc(F)c(Cl)c1F 76939,C1(C(C)CC(=O)NCC(C)(C)C)CCCN(C(=O)OC(C)(C)C)C1 76940,C(C(=O)NCCCN(C)C(C1(CO)CCCCO1)=O)(C(C)C)NC(=O)OCC 76941,C#Cc1ccccc1CC(=O)NC1CCN(C(c2ccc(I)nc2F)=O)CC1O 76942,Cc1oc(C#N)cc1C(N1CCC(NC(c2ccn(C)c2)=O)C(CO)C1)=O 76943,[N-]=[N+]=NC1CC(C(N2CC(N3CCOC3=O)C2)=O)N(C(=O)CC2CC(=O)NC2=O)C1 76944,C(=O)(CC(C)CC(C)(C)C)N1C(CNC(CCC#CC)=O)CC(O)C1 76945,C(=O)(C1CCCc2sccc21)NCCC(C)NC(=O)CN1CCN(S(C)(=O)=O)CC1 76946,C1(OCC(=O)NCC(CC)N(C(=O)CC2CCN(C)CC2)C)CCN(C)CC1 76947,c1(NC(=O)NCC2CCC(NC(C(C(C)C)O)=O)CC2)cccc(S(C)(=O)=O)c1 76948,N1(C(CCOCCN(C)C)=O)CC2CC(C1)N(C(c1ccc(N(C)C)nn1)=O)C2 76949,C(=O)(N=c1cc2n([nH]1)CCOC2)NC1CN(C2CC(OC(C)(C)C)C2)C(=O)C1 76950,c1(NC(C2CC(C)CN2C(=O)CCc2cccc(O)c2)=O)nc(Cl)nc(Cl)n1 76951,Cn1ccc(S(=O)(=O)N2CCC(NC3CCCC4CC34)CC2)c1 76952,C1(CC(=O)NC(c2cscn2)C)CC2(CC2)CN1C(c1cccc(F)c1N)=O 76953,c1(C(=O)NC2CCC(CNC(c3csnn3)=O)C2)c(F)ccc2n[nH]cc12 76954,CCCCCCN(C)CCN(C1CCN(C(c2nocc2C)=O)C1)C 76955,c1(C(=O)NC2(CF)CCN(C(CCC(=O)OC)=O)C2)cc(C)cc(Br)c1F 76956,c1(NCC(C2CC(F)(F)C2)OC)ncccc1S(=O)(=O)N.C1(C)C2COCC12 76957,C(CC)(C(=O)NC1CC(c2cn(CCOC(F)(F)F)nn2)C1)OCC 76958,CC1=NOC(C(N2CC(NC(=O)C(C)COc3ccccc3)C2)=O)C1 76959,N1(C(C=CCOCCOC)=O)CC2CC2(CNC(C2CCOC2C2CC2)=O)C1 76960,C1(NC(C=C2CCC(C)C2)=O)COCCC1NC(=O)C=CCO 76961,C1(C)(C(=O)NCC(CN(C(c2c(C)n[nH]c2C)=O)C)C)CC(C2CC2)=NO1 76962,C1(C(=O)NC(C(C)C)CNC(=O)C(C)(C)N(C)C)Nc2ccccc2C1(C)C 76963,c1(OC(C)C(=O)NC(C)(CNC(=O)CS(C)(=O)=O)C2CC2)ccc(F)cc1Cl 76964,c1(C(=O)NCC2N(C(CC3CC(=O)C3)=O)CCCC2)ccc(Br)c(F)c1 76965,c1(C(=O)NCC(CC(C)C)NC(CNS(CC)(=O)=O)=O)ccc(O)c2ccccc12 76966,N1(C(Cc2nc(NC(=O)Nc3ccnc(O)c3)sc2)=O)CCCC(F)(CO)C1 76967,C1(CCC)CN(C(c2c(N)sc(C)c2C)=O)CCN1C(c1cnn2c1OCC2)=O 76968,N1(C(C(=Cc2cccs2)C)=O)CCC(C2CC2)C1CNC(c1ccoc1C)=O 76969,C1(C(N2CC3C(CO)C3C2)=O)C(O)CCN1C(c1cccnn1)=O 76970,Cc1nc2nccc(N(C(C)CNC(c3cc(F)cnc3O)=O)C)n2n1 76971,c1(OC)cc(C)cnc1C(=O)NCC1(OC)CN(C(C2CCC2)=O)C1 76972,CCC(C#N)C(=O)NCC(C)C(=O)NCCc1cnco1 76973,[nH]1cc(C#N)c(=NC(=O)c2cc3ccc(-c4c(O)cccc4O)cc3s2)[nH]1.CCCO 76974,C12(C(=O)NCC3OCC(CNC(C4(OC)CCOC4)=O)C3)C3C4C1C1C2C3C41C 76975,c1(C(N2CC(C(C)NC(C(C=CC)O)=O)C2)=O)coc2cc(C)c(C)cc12 76976,N1(C(C2(CSC)CCC2)=O)CC(C(=O)NC(c2cncs2)C)C2(CC2)C1 76977,c1(CC(C)C(N2CCCC(CNC(=O)CCC(N)=O)C2)=O)ccc(Cl)c(Cl)c1 76978,N1(C(c2ncccc2Br)=O)CCC2CCN(C(C3(F)CC3)=O)C2C1 76979,Cc1ncccc1CC(N1CCOCC1CC(=O)N(C1CCN(C2CC2)C1)C)=O 76980,c1(-c2ccc(OC)cc2)ccc(NC(=O)Nc2cnccc2Br)cc1F 76981,CC(C)C(C)C(=O)NC(=O)NN1CC1.C(=O)(C1CC1)O.C1(C)CC1 76982,C1(C(N2CCOCC2)=O)CCN(C(=O)CO)C1.C(=O)(CN)N(C)CC1CC1 76983,C1(C(=O)NC(C2CCN(C)C2)C)(CC)CC(C)(C)C1.C12CC(C1)C(=O)NCC2 76984,N1(C(C2C(CCOC)C2)=O)CCN(C(c2ns[nH]c2=O)=O)C(c2ncc[nH]2)C1 76985,CC1(C(N2CC(OCCC(=O)NCC3CCCS3)C2)=O)CC2C=CC1C2 76986,CCC(F)C(=O)N(C)CC1(CNC(C2(C(=O)NC(C)C)CCC2)=O)CC1 76987,c1(C(=O)NC2CCC(C(N3CCC(C(C)(C)O)CC3)=O)C2)cccc(I)c1F 76988,CC(O)C(CO)NC(=O)COC1CN(C(=O)C(O)c2ccsc2)C1 76989,N1(C(C=CC(CC)C)=O)CC=C(CC(=O)N2CCN3CCCC3C2)CC1 76990,CC1CC(=O)NCC1C(N1CC2(CCN2C(c2nscc2Br)=O)C1)=O 76991,C(=O)(C(CC(C)C)NC(=O)C(N1CCOCC1)C)N1CC(CCO)(CC)C1 76992,CN1CCN(C(C2(NC(N)=O)CC2)=O)C(CNC(c2cnc(C(C)(C)C)o2)=O)C1 76993,Cn1cncc1C(O)C(=O)N(C1(C(=O)NC2CC(C(F)(F)F)C2)CCC1)C1CC1 76994,c1(C(C)(C)C)csc(C(C(=O)N(CCC#N)C(=O)C2CC2)N2CCCC2)n1 76995,c1(OC)csc(C(=O)NCCCC(C)NC(=O)CC2(C)CC2)c1 76996,C1(C)(CNC(c2nc(C(C)C)sc2)=O)CCN(C(c2ccn(CCF)n2)=O)CC1 76997,N1(C(c2c(C)ncc(Br)c2)=O)CCC2CN(C(c3ccc(F)c(F)c3)=O)CC2C1 76998,C1(CCNC(C(CC)=CC)=O)CN(C(=O)C(C(C)C)c2ccccc2)CCO1 76999,CCC(C)C(C(=O)NC(CC(N)=O)C(=O)NCC(C1CC1)SC)N(C)C 77000,c1(CN(C(CC)CC)C)cn(CC(O)Cc2ccccc2)nn1 77001,n1(CC)cc(C(N2CCCCC2C(CO)NC(=O)CCCNC(C)=O)=O)c(C)n1 77002,CC(C)CC(Cc1ccccc1)C(=O)N(C)Cc1ccn(C)c1 77003,c1(OCC)nc(Cl)ccc1C(=O)NCC1CC2CC2N1C(=O)C(O)C(C)(C)C 77004,Cc1cc(C)c(C(=O)NCCC(O)CNC(=O)Cc2ncccc2C)c(S)n1 77005,c1(N(C2CCN(C(C3CCCCC3O)=O)C2)C)ncccc1S(C)(=O)=O 77006,N1(C(CC#C)=O)CCC2(CC2C(N2CCCC2(C)C(=O)OCC)=O)C1 77007,c1(C(=O)NC2C3CN(C(CN4C(C)CCC4)=O)CC32)cccc2c1CCC2=O 77008,N1(C(c2ccc(CC)s2)=O)CC(NC(=O)C(C)(O)C2CC2)C(SC)C1 77009,N1(C(C(=O)NCC(CC(C)C)(C)O)=O)CC2CC(N)C(C2)C1 77010,CCCCC(CC)C(=O)N1CCCC1C1(NC(c2nncs2)=O)CC1 77011,N1(C(C2C(NC(=O)CCc3ccncc3)C=CCC2)=O)CCCC2(CCCO2)C1 77012,c1(CC)cc(C(N2CCC(C(F)F)(CNC(C3CCCC(O)C3)=O)C2)=O)ncn1 77013,C1(C(N(CC(C)N(C(c2c(C)nc(C(C)C)o2)=O)C)C)=O)Cc2nccnc2C1 77014,c1(C(=O)NCCC2CC(NC(C3C(C)CC3)=O)C2)cncc(N(C)C)c1 77015,N1(C(C(C(=O)OC)(C)F)=O)CC2CC(C(=O)Nc3cnc(N(C)C)nc3)CC2C1 77016,C(=O)(C(C)C(O)C(C)C)N1CCN(C(C(CCC)(C)C)=O)CC1CF 77017,C1(CN(C(C2(NC(CN(C(=O)OC)C)=O)CCC2)=O)C)CCOC1C 77018,C(=O)(C#CC1CCOCC1)NC1C(C(=O)NC(C(=O)NCC)C)OCC1 77019,N1(C(C(CC)CC)=O)CC2OCCN(C(=O)CC3CCCC34CC4)C2C1 77020,CCCCCCCc1cn(C2(C(=O)N(c3ccc(Cl)cn3)C)CC2)nn1 77021,CN1CCN(N2CCCC2C2CCCO2)CC1NC(=O)OC(C)(C)C 77022,CC(C)CC(C(=O)N1CCN(C(c2ccc(F)o2)=O)C(CC(F)F)C1)N(C)C 77023,c1(CC)noc(C)c1C(=O)NCC1(F)CCC(NC(=O)CC23CCCC2C3)C1 77024,O=C1CCN(CC2CCOCC2)C(=O)N1CCOCc1nc2ncccn2n1 77025,c1(OC)ccc(CC(N2C3CN(C(C4(C#N)CC4)=O)CC23)=O)c(Br)c1 77026,C=CCC(C)C(=O)NCC1CCN1C(=O)C(=Cc1ccccc1)C 77027,c1(OC)cccc(CCC(N2CCN(C(c3cncc(N)c3)=O)CC2)=O)n1 77028,C(=O)(CCCCC(=O)NCC1(OC)CN(C(=O)C(c2ccccc2)SC)C1)OC 77029,c1(C(=O)NCC(CCNC(=O)CCc2nncs2)OC)cc(F)c(F)cc1O 77030,c1(OCCCC)ccc(C(C)Nc2ccc(I)cn2)cc1OC 77031,c1(C(=O)NC2CN(C(C3C(CC)CCO3)=O)CC2C)ccc(OC)c(OC)c1Cl 77032,c1(C(=O)NC2C(CNC(c3c[nH]c(C(F)(F)F)c3)=O)COC2)ccc(O)cn1 77033,c1(C(N2CCC(NC(c3cnc(Cl)s3)=O)C(F)C2)=O)ccc2nc[nH]c2c1F 77034,C1(O)(CNC(CC(OCC)OCC)=O)CCCN(C(c2cscc2Cl)=O)C1 77035,C1(C(=O)NCc2c(C(=O)NCC3(CC(C)C)CC3)cco2)CC(=O)CCO1 77036,N1(C(C(n2c(C)cc(C)n2)C)=O)CC2(CCC2NC(c2cc(=O)n(C)cn2)=O)C1 77037,C1(NC(=O)CCC2CCCC2)CN(C(=O)C#CC2CCCCC2)C2(CCOC2)C1 77038,c1(C(N2C(C3CCCN(C(C(=O)N(C)C)=O)C3)CCCC2)=O)cc([N+](=O)[O-])n[nH]1 77039,C(C(=O)NCC1(CNC(=O)C(F)F)CCOCC1)(C(C)C)N(CC)CC 77040,c1(CC(=O)NCC23CC2CN(C(C2CCSC2)=O)C3)ccc(Cl)c([N+](=O)[O-])c1 77041,c1(N(C(C=CC(=O)NC(c2c(C)ncs2)c2ccccc2)=O)C)ccc(F)cc1 77042,C(=O)(CCCCCN(C(=O)CSCCC#N)C)N1CCC(C(C#C)C)CC1 77043,CN1CC(NC(=O)C#CCNC(c2cc[nH]c2C2CC2)=O)C(F)(F)C1 77044,CCC(C)(CCC(C)C)C(=O)N1CC2CC(C1)C2(C)C.N12CC(CC1=O)n1nnnc12 77045,N1(C(CSCCCC)=O)CCCC(CC)(NC(=O)C(C)NC(=O)C(C)(C)C)C1 77046,c1(-c2cc(CNC(N3CC(C(=O)O)(COC)C3)=O)sc2)ccc(C(N)=O)cc1 77047,C1(CNC(=O)Cc2ccoc2)CCCN(C(c2ccccc2-n2cncn2)=O)C1 77048,C1(NC(c2c(OCC)oc(C)n2)=O)(CO)CCCN(C(c2cc(C)ns2)=O)C1 77049,c1(SC)nc(C)cc(=NC(C)CCN(C(=O)CNC(=O)CC(C)(C)C)C2CC2)[nH]1 77050,C1(NC(=O)CCc2sccc2Br)CCCN(C(c2cn[nH]c2)=O)CC1 77051,C(=O)(CC(C)CC(C)C)NC(CNC(C(CC)N1CCCC1=O)=O)(C)C 77052,c1(N(C)Cc2nc(C)sc2)nnc(CCO)n1CC1CCCO1 77053,C1(NC(CC2(COC)CC2)=O)CC(CO)N(C(c2nc(O)sc2C)=O)C1 77054,c1(C(=O)NCCCCN(C(C2C(OC)CCCC2)=O)C)cnc2cc(C)[nH]c2c1 77055,N1(C(C2(C(=O)OCC)CC2)=O)CC(C2(NC(=O)CCC3CCCC(O)C3)CC2)C1 77056,N1(C(COCC(C)C)=O)CCCC(C2CN(C(=O)Cc3cccnc3Br)C2)C1 77057,c1(CC(=O)NCC(CC)NC(c2cc3nccnc3[nH]2)=O)ccc2ncsc2c1 77058,c1(CC(=O)N(C2CCCN(C(CC=C)=O)C2)C)coc2cc(O)ccc12 77059,Cc1nnc(=NCC(CC(C)C)NC(=O)CC(C(F)F)n2cccn2)[nH]c1C 77060,c1(CC(=O)NC2CC(F)(CNC(C(C)N3CCC3)=O)C2)cncc2ccccc12 77061,C1(C(N2C(CNC(C(C)(C)C3CCCC3)=O)CC(O)C2)=O)CC2(C1)CC2(F)F 77062,C(=O)(C(C1=CCCSC1)N1CCC(NC(=O)OCC)C1C)NCC=C 77063,N1(C(CC(=C)C)=O)CCC(CN(C(=O)CN2CC(=O)NC2=O)C2CC2)CC1 77064,C(C(C)(O)CC(=O)N1CCC(C2CCCCN2C(C23CC2C3)=O)C1)OC 77065,C(CC)(C(C)(F)F)NC(C(CC1CCC1)NC(CNC(CC)=O)=O)=O 77066,c1(CN(C(=O)CNC(=O)C(=Cc2ccc(C)cc2)C#N)CC)c(F)cccc1F 77067,C1(CNC(c2ccc(SC(F)F)cc2)=O)CN(C(=O)NCc2ccccc2)CCO1 77068,CCCCC(CNC(c1ccsc1C(F)(F)F)=O)NC(c1cnsc1C)=O 77069,CC(CN(C)C)CC(=O)NC1(C(=O)NC(C)CCc2cn[nH]c2)CCC1 77070,N1(C(Cc2c(OC)cccc2)=O)CC(OCc2ccccc2)CCC1C 77071,N1(C(C2C(=C)CC2)=O)CCC(CC(N)=O)(NC(C23CC2COC3(C)C)=O)CC1 77072,C(C(CC)(CC)C(N)=O)N(C(CCC(CC)C)=O)CCNC1(CC(=O)OC)CC1 77073,CCC(F)(F)CC(=O)N(C(C)CCNC(c1snnc1C1CC1)=O)C 77074,c1(C(=O)NCCNC(=O)Cc2csc(-c3ccc(O)cc3)n2)ccn2nncc2c1 77075,N1(C(CCN(CCC)C)=O)CCCCC1CCC(=O)NCCCc1cccnc1 77076,C12(C(N3C(CC(=O)NC)CC3)=O)CC(CCO1)N(C(=O)C=CCF)C2 77077,c1(C(N2CCC(C)(CCNC(c3c(C)occ3)=O)C2)=O)cc(F)ccc1N 77078,C1(C(=O)NC(CC)Cn2cncn2)CCOCCN1C(=O)CC1COCC(C)O1 77079,N1(C(C2(C)C(C)C2)=O)CC2(CCCN(C(C3C=CC(=O)N=N3)=O)C2)C1 77080,C1(C(=O)OCC)CCCN(C(=O)C(CN(C)C)NC(c2ccncc2)=O)C1 77081,C1(NC(Cc2n(C)nnc2)=O)CC(CNC(=O)CC(C)(C)c2cccs2)C1(C)C 77082,C1(C(N)=O)(CNC(C2CC2C(N)=O)=O)CN(C(=O)C(C)Sc2ccccc2)C1 77083,Cc1noc(C(F)F)c1C(=O)NCCC1CCN(C(=O)C=Cc2cc[nH]n2)C1 77084,C(CC(C)(C)CC(=O)NCC(C1CCN(C(=O)CCCCCF)CC1)F)OC 77085,c1(C(=O)NCC(CSC)OC)ccc(CNC(C2CC(CN(C)C)C2)=O)s1 77086,c1(OC)cnc(C(=O)NC2CCC2NC(C2(C)CC3CC3C2)=O)c(F)c1 77087,S(=O)(=O)(c1ccc(N(C)Cc2ccc(Br)o2)cc1Cl)NC1(CC)CCOCC1 77088,CCCCC(C(=O)NC1CCCN(C)C1=O)NC(c1cnnn1CC)=O 77089,C=CC(C)C(=O)NC(c1ccccc1)C(=O)NCc1nn[nH]c1C1CC1 77090,C1(C(=O)Nc2cc(C#N)sc2)Cc2ccccc2CN1C(c1ccon1)=O 77091,C12(NC(C(COC)C)=O)CCCC1N(c1ncnc(O)c1Br)CC2 77092,C(=O)(C#CC(C)(C)CNC(C1C2CCC(F)C12)=O)N(C1COC(C)(C)C1)C 77093,c1(C(=O)NCC(N2CC(C)CC(C)C2)(C)C)cncc(C2=CCNCC2)c1 77094,Cc1nc(=N)[nH]cc1C(N1CCC(CNC(c2ccc(F)o2)=O)C1(C)C)=O 77095,C(=O)(C1COc2cc(C)c(C)cc21)N1CCCCCC(NC(CCC(=C)C)=O)C1 77096,C(C1CCCC1)=CC(=O)N(CCN(C(C(n1ccc(Br)n1)C)=O)C)C 77097,c1(OCC(C)C)cccc(C(=O)NC2CN(C(=O)C(=O)NCC(F)F)C3CC23)c1 77098,CC1(C)CN(C(c2c[nH]c(Br)c2)=O)CC1NC(c1cccc(C(N)=O)c1)=O 77099,c1(NC2CCC(CC(=O)NCCCOc3ccccn3)CC2)cccc(F)c1I 77100,c1(CC(=O)NCC2CCCN(C(C(CC)OC)=O)C2)ccc(S(C)(=O)=O)cc1 77101,C1(C)(NC(CC(CC)C2CCC2)=O)CCCN(C(=O)CC(C)(C)O)C1 77102,C1(C#N)(SC)CN(C(=O)C(CCC2CCC2)NC(=O)C(=O)N(C)C)C1 77103,c1(NCC(CC)(C)OC)cc(NC2C=CC(CO)C2)ncn1 77104,CCC(C)(C1CC1)NC(=O)OC(C)(C)C.C(Cc1nccs1)CO 77105,c1(CNCc2ccc(-c3cc(C)[nH]n3)nc2)ccc(F)c2ccoc12 77106,CCC(C)C(O)CC(=O)NC1(CCC(N2CCC(F)(C#N)C2)=O)CCC1 77107,N1(C(C(CCC)CNC(=O)CC2CC(C)C2)=O)CCC(C2(C)CC2)CC1 77108,C(=O)(C1Cc2ccccc21)NCC1(NC(C=Cc2ccc(OC)c(OC)c2)=O)CC1 77109,C1(O)(CCNC(CC2N(C)CCOC2)=O)CCN(C(=O)C=Cc2ncc[nH]2)CC1 77110,n1(CC)c(C(=O)NCC2CCN(C(C34CC(C3)C4)=O)C2)cc2ccccc12 77111,c1(CNC(C2N(Cc3ccc(SCC)o3)CC2)=O)cccnc1N1CCCCC1 77112,N1(C(C2C(C(=O)OC)C2)=O)CCC(NC(=O)Nc2cccnc2I)CC1 77113,C1(NC(c2ccc(COC)cc2)=O)CCCCN(CSc2ccc(C)cc2Cl)C1 77114,CCCCCCCCCC(=O)N1CCCC12CN(c1ccncn1)C2 77115,CC1CN(C(=O)Cc2cccc([N+](=O)[O-])c2)c2ncc(Br)cc2O1 77116,C(C(C)(O)CC(=O)N1CCC(NC(c2cccc(NS(C)(=O)=O)c2)=O)C1)OC 77117,C1(CS(C)(=O)=O)CN(C(c2c(F)cccc2Cl)=O)CCN1C(=O)C(O)C1CCC1 77118,c1(C(=O)NC(CNC(C(COC)C)=O)C2CC2)ccc(N2N=CCC2=O)cc1 77119,C1(NC(c2nc(C)c(C)s2)=O)(CO)CCCN(C(C2CC3(CCOC3)C2)=O)C1 77120,c1(C(=O)NC23CC(NC(Cn4c(=O)ccc(C)n4)=O)(C2)C3)ccn2ccccc12 77121,N1(C(C2N(C(C)=O)CCCC2)=O)CC2CCC1C2NC(=O)C=Cc1cccnc1 77122,c1(C2C(=O)NC(=O)N2C)ccc(Br)s1.CC(C)CSCCOC(C)(C)C 77123,Cc1ccc(Cl)c(NC(N2CCC(c3nc(C)c(C)[nH]3)CC2)=O)c1Cl 77124,C1(OC)CC(CNC(c2cc(N3CCCCC3)ncn2)=O)N(C(=O)C(C)CO)C1 77125,c1(NC(C2CCCC2NCc2ccc(OCC(=O)O)cc2)=O)ccc(Cl)cc1F 77126,c1(CC(=O)NCCNC(c2c(CC)con2)=O)cc(Br)cnc1F 77127,N1(C(c2c(C)cc(C)[nH]2)=O)CCCC(NC(=O)C(F)(F)c2nccs2)C(F)C1 77128,N1(C(c2cc(C)oc2)=O)CCC(NC(c2cc(O)no2)=O)C1(C)C 77129,C(CCCCCNC(c1cccc(O)c1)=O)N(C(C1(CN(C)C)CC1)=O)C 77130,C(=O)(C(C(C)(C)OC)Nc1ncnc(N2CCCCC2CO)c1C)OC 77131,c1(NC(c2c(-c3c(C)cccc3)cccn2)=O)cc(Br)ccc1Cl 77132,N1(C(C(CC2CC2)NC(c2cnc(CC)o2)=O)=O)Cc2ccc(C#N)cc2C1 77133,N1(C(C(C(C)(C)C)NC(C(C(CC)CC)F)=O)=O)CCC2(CCC2)C(O)C1 77134,C(C)(CNC(c1cc(OC)no1)=O)(C(C)C)NC(Cc1nc(COC)sc1)=O 77135,C1(NC(CC=CCC)=O)CCCC(CN(C)C(c2cc(C(=O)OC)nn2C)=O)C1 77136,c1(NC(=O)Nc2ccc(N3CC(C)OC(C)C3)nc2)cccn2nncc12 77137,c1(C(N2C(CN(C(C(C)n3cccn3)=O)C)COCC2)=O)ncc2[nH]ncc2n1 77138,N1(C(c2cccc(OC)c2N)=O)CCN(C(=O)Cc2cncnc2O)CC(O)C1 77139,c1(N(C2CCCN(C(C3ON=C(C)C3)=O)C2)C)ncc2c(n1)COC2 77140,C1(NC(CN2CC(CC)C2)=O)CC2CC1CN(C(=O)C#CC1CCC1)C2 77141,c1(C(N2CCC(CCNC(C3OCCN(C)C3)=O)C2)=O)ccc(N)c(Cl)n1 77142,Cc1cc(NC(C2(O)CCN(C(C3CCOCC3)=O)C2)=O)ccc1C(F)(F)F 77143,CC(Cc1ccccc1)C(c1nnnn1C)NCC1(F)CCCC1 77144,N1(C(C2C(CCOC)C2)=O)CC(N(C(=O)Cn2ncc(Cl)c2C)C)C(C)(C)C1 77145,c1(C(=O)NCC2N(C(CCN(C)CCO)=O)CCC2)cc2ccccc2c(O)n1 77146,C(=O)(C1=NOC(C)C1)N1CC(O)(CNC(COCCCCCC)=O)C1 77147,c1(C(C)(C(=O)N2CC(F)(CN(C)C)C2)NC(C)=O)c(F)cc(Br)cc1F 77148,CCCC(C(=O)N1CCCC1C1(NC(=O)Cc2ccsc2Cl)CC1)OCC 77149,C(=O)(C(F)(F)C(O)C1CC1)NC1CCC(CNC(=O)CC2(O)CCCC2)C1 77150,C1(NC(=O)C(c2ccc(Cl)cc2)O)CCCCC1NC(C1(CO)CCOCC1)=O 77151,C(=O)(C(O)C(F)(F)F)NC(CCCCNC(c1c(C)[nH]nc1Cl)=O)C 77152,N1(CC)CCCC2C1CCCN2Cc1ccc(-c2ccccc2C=O)s1 77153,C1(C(=O)NCc2ccc(C(N)=O)o2)(NC(C2(CC)CC2)=O)CC1(C)C 77154,C#CCC(C(=O)N1CCC(C(F)(F)F)C1)NC(=O)CCc1cccnc1 77155,C(C(=O)NC1CC(CCNC(C2CC2(Cl)Cl)=O)C1)(C(C)(C)C)NC(C)=O 77156,CCCCCC(=O)N(CCCNC(=O)CN1CCN(C)CC1)CCO 77157,C1(CNC(C(C=C)C)=O)CN(C(c2n[nH]c(C)n2)=O)C2CCN1C2 77158,Cc1cc(CNC(c2oc(CNC(C3(CO)CCOC3)=O)nc2C)=O)c(C)s1 77159,C(=O)(C1=NNC(=O)CC1)N1CC2C(CNC(c3c(C)ncnc3)=O)(C2)C1 77160,N1(C(C2CC(C(F)F)(OC)C2)=O)CCC2(CC1)CC(C)N(C(=O)C(C)SC)C2 77161,N1(C(CCc2nc(=N)[nH][nH]2)=O)CCCC2C1CCN2C(c1ccn(C(F)F)n1)=O 77162,C1(CC)C(C(=O)NCC(C)(CNC(=O)CC2CCC(=O)N2C)OC)CCN1C 77163,c1(CN(C2CC2)Cc2ccc(OC(C)C)cc2)ccc2c(c1)OCCO2 77164,CC1CC(NC(=O)CSS(C)(=O)=O)CN1C(=O)Cc1cc(C2CC2)no1 77165,C1(NC(C2(N(C)C)CC2)=O)CCCC1NC(=O)CCOCC(F)F 77166,C#CC(CC)(CC)NC(C1(C(C)C)CCN(C(C2CCSC2)=O)C1)=O 77167,C(=O)(C#CC1CCCC(C(=O)OC(C)(C)C)C1)N(CCCC(=O)OC(C)(C)C)C 77168,N1(C(C2(NC(c3cc(C)sc3)=O)CCSC2)=O)CCCC2(CC(O)C2)C1 77169,C1(C2(N)CCC2)(C(=O)NCCn2ncc(C(C)=O)c2)CCC1 77170,n1(CC)nnc2c(NCC(C)CNC(=O)C(C)(C)N3CCCCC3)ncnc12 77171,CCCS(=O)(=O)NC(C)C(=O)N(CCCNC(=O)C(F)CC1CC1)C1CC1 77172,c1(C(=O)NC2CN(CCc3c(C)[nH]nc3O)CCS2)n[nH]c2c(F)cccc12 77173,c1(NCc2ccc3[nH]c(C)c(C)c3c2)[nH]c(=NC2CSCC2C)nc2scnc12 77174,C1(CCC)CN(C(=O)C2=C(Cl)CCC2)CCN1C(=O)CC1(c2ccon2)CCC1 77175,c1(NC2C(O)CN(Cc3cccc(F)c3Cl)C2)ncnc2c(F)cccc12 77176,CCS(=O)(=NC(=O)C1(CCC(C)(N)Cl)CC1)c1ccc(C)cc1 77177,CCCCC(C)C(=O)N1CCN(C(C2CC(C)(C)C2C(F)(F)F)=O)CC1C 77178,O=C(CCCC(=O)C1CC1)NCCC1CSCCN1C(C1CC1c1ccco1)=O 77179,C1(NC(CN(C(C(CC=C)NC(C)=O)=O)C(C)C)=O)CC2CCCC2C1 77180,O=CN1CCOCC1C(=O)NC1CCCCN(C(=O)C2=NOCC2)C1 77181,C1(C(=O)NCC(C)C(C)(F)F)CC12CCN(C(C1COCC1C(N)=O)=O)C2 77182,n1(CC(=O)NCC2=CCN(C(CC3(C)CC3F)=O)CC2)ccc2cc(F)ccc12 77183,C(CSc1ccccc1)(C(=O)N(C1CCN(C(=O)C(C)(C)C)C1)C)NC(=O)OC 77184,CC(C)C(C(=O)N1CC(NC(=O)CNC(c2cc(Cl)no2)=O)C1)NS(C)(=O)=O 77185,c1(CCC(N2CCC(N(CCC)C(C)=O)C2)=O)ccc(F)cc1F 77186,N1(C(C2N(C(C(CCC)NC(C)=O)=O)CC(F)(F)C2)=O)CCCC2(COC2)C1 77187,N1(C(=O)C=CC(=O)NC2CC2)CCC(CNC(C=C2C(C(C)(C)C)C2)=O)C1 77188,C1(NC(c2[nH]cc(C#N)c2)=O)CCCCCCC1NC(=O)CC1CNC(=O)O1 77189,N1(C(Cc2n(C)ncc2)=O)CCSCC1C(=O)NC1CC(O)C1O 77190,C1(C(=O)NCC(C)NC(=O)CSCC(=O)OC(C)(C)C)CC(F)(CO)C1 77191,N1(C(c2n[nH]c(CC)c2Cl)=O)CC2CCN(C(=O)Cc3ccc(F)cc3)C(C2)C1 77192,Cc1cc(C(=O)N(CCCNC(=O)CS(=O)(=O)C2CC2)C(C)C)c(O)cc1F 77193,c1(C(=O)NC(C)C(N2CCC(O)CC2C)=O)cnccc1C#N 77194,c1(OC)cc[n+]([O-])c(C(=O)NCCC2(NC(C3CNC(=O)C3)=O)CC2)c1 77195,C1(CNC(CC(CC)(C)C)=O)CCC2CN(C(=O)C3=CCCOCC3)CCC2C1 77196,N1(C(c2ccc(C)nc2O)=O)CCn2cnc(-c3ccc4c(c3)OCC4)c2C1 77197,Cc1cncc(C(=O)NC(C2CCN(C(c3cc(=O)cc[nH]3)=O)C2)(C)C)c1 77198,C=CCCCC(C)(C)C(=O)NCC1CCC1NC(=O)C(=Cc1cccnc1)C 77199,c1(CNC2C(C)CCC(C)(C)C2)ccc2cc(Cl)ccc2n1 77200,C12(C(=O)NCC3CC(O)(CNC(c4ccc(O)nn4)=O)C3)CCN(CC1)C2 77201,c1(C(N2CCC(OCCNC(C3(C=C)CC3)=O)C2)=O)c(C)cc[nH]c1=N 77202,C1(CC(=O)NCC2N(CC)CCC2)CC(C)(C)CN1C(c1cnc(C2CC2)o1)=O 77203,N1(C(C2C3CN(C(C(CCC(C)C)F)=O)CC32)=O)C2CCC1CC1(CC1)C2 77204,c1(C(C(=O)NCC=C)N(C)CC=CC(C)(C)C)ccc(-n2cccn2)cc1 77205,C1(CNC(C(Cc2c(C)nc[nH]2)O)=O)C2CCC(C2)N1C(=O)C1=NNC(=O)C1 77206,N1(C(CC(C)(C)C)=O)CC2CCCC2(NC(c2ccc(N)cc2F)=O)C1 77207,Cc1cccc(C)c1CNC(=O)C(C)NC(c1cocc1C(N)=O)=O 77208,N1(CC(O)C)CC23CCCC2(C1)C3.c1ccccc1OC(F)F 77209,c1(C(N2C(C(=O)Nc3c(C#C)nccn3)CC(OC)C2)=O)ccc(O)c(O)c1Cl 77210,n1(CC(=O)N(C(=O)CNS(=O)(=O)c2cccs2)C)nc2c(n1)CCCC2 77211,CC(C)(F)CCC(=O)NCC(CNC(c1ccnc(C(F)(F)F)n1)=O)CO 77212,c1(C(N2CCN(C(c3cc(C)ncn3)=O)CC2)=O)c2c(nn1C)CCC2 77213,C1(C(N2C(C)CN(C(c3cnnn3C)=O)CCC2)=O)COc2ccccc2C1 77214,CCN=c1ccc(C(N2CC(O)(CNC(=O)CCc3nnc(C)n3C)C2)=O)c[nH]1 77215,c1(CC)[nH]c(=N)sc1C(N1CCCCC1CCNC(C1CC1CC)=O)=O 77216,Cc1cccc(C(=O)NCC2CCC(NC(=O)C(C)S)CC2)c1Cl 77217,C1(NC(CNC(C2CCCCC2)(C)CO)=O)CC2CCCC(C1)N2 77218,C1(C(N2C(CNC(c3ccn(CC)n3)=O)CCC2)=O)CCCN(C(=O)C2CC2)C1 77219,C12(CNC(c3cc(C)cc(C)c3)=O)CC(CCO1)N(C(=O)C(C)CC(C)(C)C)C2 77220,N1(C(CCCNC(C)=O)=O)C(C(=O)NCC2CC23CCCCC3)CC2CCCC12 77221,Cc1cc(C(=O)NCC(C)NC(C2(C(C)C)CC2)=O)nc(C2CCC2)n1 77222,N1(C(CSCC(N)=O)=O)CCC2CCC(NC(c3ccc(C(N)=O)c(Cl)c3)=O)C12 77223,c1(CNC)cccc2ccnn12.Cc1cnc(N2CC(C(N)=O)(NC(=O)N)C2)nc1 77224,C1(CNC(c2c(CC)ocn2)=O)(CNC(=O)C(C(C)C)SCOC)CC12CCC2 77225,C(=O)(C(F)(F)CCn1ccnn1)NCC(C)NC(C(c1c(OC)cccc1)O)=O 77226,N(C1CCCc2c1cnn2CCO)C(C1CCCCO1)C 77227,C(=O)(C(C)CCCOC)NCC12C(CN(C(c3nn(CC)c(C)c3)=O)C1)C2 77228,C(=O)(CCCCCCNC(C1CCOCC1)=O)N1C(C)(C)C(CO)C1 77229,N1(CCNC(C(C)OC)=O)CCCN(C(c2sc(Br)nc2C)=O)CC1 77230,C#CCCCC(C)C(=O)NCC1CCC12CCN(C(=O)CSC(F)(F)F)CC2 77231,CC1(C)Cc2nc(NC(=O)Cc3cc(Cl)cc4ccccc34)sc2C(=O)N1 77232,C1(O)(C(=O)NC(CC)CNC(=O)C(C)(C)CC(F)F)CCc2ccccc2C1 77233,N1(Cc2nc(CC)sc2)CCC(O)C1C(=O)Nc1sccc1C(=O)OC 77234,N1(C(Cn2nc(C)oc2=O)=O)CC2(CC2)CC1CNC(C12CCC(CC1F)C2)=O 77235,C1(CNC(=O)Cc2cncs2)CC2CC1CN(C(=O)COC(=O)CO)C2 77236,CC1CC=C(C(=O)N2CC3(CC(NC(c4ccccc4OCCF)=O)C3)C2)CC1 77237,Cc1cc(C(N2CCCC2CC(=O)N(CC(C)(C)N(C)C)C)=O)co1 77238,C#Cc1ccc(CC(N2CCCC2(C)CNC(C2(C)CC(F)C2)=O)=O)cc1 77239,C=CCCC(F)(F)C(=O)NC1CN(C(=O)C(C)N(CC(F)(F)F)C)CC1(C)C 77240,c1(C(=O)NC2C(CNC(C34CC(OC)C3C4)=O)CCC2)cc(S(C)(=O)=O)oc1C 77241,c1(OC)ccc(C2CCN(C(c3c(C)n[nH]c3C)C(=O)NC(C)C)C2)cc1 77242,N1(C(C2C(CC)N(C(=O)C(F)F)CC2)=O)CCCN(C)CC1C 77243,CC(CC(C)(C)C)C(=O)N1CC2C(C(=O)NC3CN(C)CC3(F)F)C2C1 77244,N1(C(C(CCC)OC)=O)CCC(C2CC2)(CNC(c2cccc(F)c2CC)=O)C1 77245,C=CCCC(C)C(C(=O)NCCCF)N(CC(=O)OCC1CC1)C1CC1 77246,N1(C(c2cc(C#N)sc2)=O)CCC(CNC(=O)CC2CCCC2O)C(F)(F)C1 77247,C1(NC(CCc2cnc(C)o2)=O)COCCC1NC(=O)CCc1cnc[nH]1 77248,c1(C(=O)NC(C2CCN(C(C3CN(C)CCN3C)=O)C2)C)ccnc2[nH]ncc12 77249,N1(C(C=C(CC)C)=O)CCC(C2CCN(C(=O)CCn3nc(C)cc3C)C2)C1 77250,c1(C(COC(C2C(C(=O)OCC)CC2)=O)F)ccc(F)cc1F 77251,N1(C(C(CC)NC(N)=O)=O)C2CCC1CC(NC(c1c(O)nnc(C)c1C)=O)C2 77252,CC1(C)CCC(C)(C(N2CC(CO)(NC(c3cncc4nc[nH]c34)=O)C2)=O)CC1 77253,c1(CCC(=O)NCC(C2CCOC2)O)ccc(Cl)c(F)c1 77254,C1(NC(CN(CC(C)(C)C)C)=O)CC2C1CCN2C(c1cnn(C)c1Cl)=O 77255,N1(C(C(COCC)(C)C)=O)CC(C)CN(C(=O)Cc2ccc(O)c(Cl)c2)C(C)C1 77256,c1(CCC(=O)NC2COCC2CNC(C2(N(C)C)CCC2)=O)nnc(S)nc1O 77257,N1(C(C(CC)C)=O)CCN(C(c2cc(C(=O)OC)on2)=O)CC1CC(F)F 77258,c1(C(N(C2CC2)CC2N(C(C(CSC)C)=O)CCC2)=O)cnn2ccsc12 77259,N1(C(C2N(C)C(=O)CC2)=O)CCCN(C(=O)CCCCC#N)CC1CC(C)(C)C 77260,c1(C(=O)NCC(C(C)C)NC(c2cccc3nn[nH]c23)=O)ccnc2[nH]ncc12 77261,C1(N(C(c2ncccc2Br)C(=O)NC(C)(C)C)C)CCC(F)(F)C1 77262,C(=O)(C(C)(C)CCCC=C)NC(C(N1C(C#C)CC1)=O)COC 77263,Cc1c(F)ccc(C(=O)NC2(CNC(C3CCCCO3)=O)CCOC2)c1O 77264,CCC(C)CCCC(=O)NCC(N1CC(CO)C2(CC2)C1)=O 77265,N1(C(c2c(COC)noc2)=O)CCC(N=c2cc[nH]cc2C#N)CC1C 77266,N1(C(c2scc(OC)c2)=O)CC2CN(C(c3cc(C4CC4)on3)=O)CC2C1CO 77267,c1(NCC(=O)NC2CN(C(C=C(C)C(C)C)=O)C2)cccc(C#N)c1 77268,C1(CC(=O)N(C(CNC(C2COC(=O)N2C)=O)C2CC2)C)CCCCC1(C)C 77269,C1(CNC(C2CN(CCOC)C(=O)C2)=O)(CO)CCN(C(=O)CSC)CC1 77270,C=CC(C)C(C)C(=O)NCc1ccc(C(=O)NCCNC(=O)OC)cc1 77271,C1(C(N)=O)COCCC1C(N1CCC(N(C(C2CCCC2O)=O)CC2CC2)C1)=O 77272,C1(C)(CNC(C2CC(COC)C2)=O)COCCN(C(=O)CNc2ccncc2)C1 77273,CCC(CC)CC(F)C(=O)NC1CC=C(C(=O)N(C2CCNC2=O)C)C1 77274,C1(CNC(C(F)=C(C)C)=O)CN(C(=O)CSCC2CCCO2)CC(C)(C)O1 77275,C(=O)(CCC(=O)C(C)(C)C)N1C(C(=O)NCCN(C(C)C)C(C)C)CNC(=O)C1 77276,c1(N(C)Cc2ccc(OC(C)C)cc2)cc(Br)c2ccccc2c1 77277,C(=O)(C(C(=O)NC1CCCN(C(=O)C(N2CCSCC2)C)CC1)C(C)C)OCC 77278,C1(O)(CNC(C2(COC)CCC2)=O)CCCN(C(=O)C(=O)NCC(F)(F)F)CC1 77279,N1(CC(C)(C2CCC2)N(C(C)(C)C)CCC#N)CCCC(C)C1C 77280,C1(CSC)CCN(CC(=O)N(CCN2CCOCC2)CC2CCCC2(C)C)CC1 77281,CC(C)C(F)(F)CC(=O)NC1CN(C(c2c(F)cncc2Cl)=O)CC1(C)C 77282,CC(C(C)C(=O)N1CC2CC1CS2)NC(=O)CCNC(N)=O 77283,Cc1ccc(COCC(=O)NCC2(F)CC(NC(=O)COc3ncnn3C)C2)cc1 77284,Cn1[nH]c(C(=O)NC(C)(CNC(C2CCN(CCF)CC2)=O)CO)nc1=O 77285,C1(C(=O)NCC2(CC(=O)Nc3cn(CC#C)nc3)CC2)CC(=O)OC1(C)C 77286,c1(C(=O)NC23CC2CN(C(C2CCC4CC4CC2)=O)C3)c[nH]c2cccc(F)c12 77287,c1(CNC(C2CCC(CNC(C3CN(C(=O)NC)C3)=O)O2)=O)nc(O)ccc1C 77288,c1(OC2CCN(C(C)=O)CC2)cccc(C2CC2NC(c2[nH]c(C)nc2C)=O)c1 77289,c1(OC)ccc(CN(c2ccccc2)C(=O)CNc2ncc(F)cn2)cc1 77290,c1(C(N2CCN(C(=O)CSc3ccccn3)C3CC23)=O)cc2c(cn1)OCCO2 77291,C1(NC(c2c(C)cno2)=O)CN(C(C23CCC(CC2)CO3)=O)CC2(CCC2)C1 77292,N1(C(C(CC)n2cncn2)=O)CC2(CCCN(C(=O)C(F)CC(C)(C)C)C2)C1 77293,C1(N(C(C(C)OCc2ccccc2)=O)C)CCC(NC(c2sccc2F)=O)CC1 77294,C1(F)(C(N2CC(F)(CNC(Cc3cc(C)[nH]n3)=O)C2)=O)CCN(C)CC1 77295,c1(C(N2CCCC(C(C)NC(=O)C(F)=CC3CC3)C2)=O)[nH]nc([N+](=O)[O-])c1Cl 77296,c1(C(=O)NCC(N(C(C=C(C)C(F)F)=O)C)C2CC2)cnc2ccccc2c1C 77297,c1(C(N(C2CCN(C(c3nccn3C)=O)CC2)CC)=O)nc[nH]c2ncc(Br)c1-2 77298,N1(C(C(C)=CC2CC2)=O)CCC2CN(C(=O)Cc3cnccc3C)CC2CC1 77299,c1(C(=O)NCC2CC(NC(CSC)=O)C2)ccc(Nc2ccc(Cl)nn2)cc1 77300,c1(CNC2CC(CNC(=O)COCc3ccccc3)C2)ncc([N+](=O)[O-])cc1F 77301,CC1CN(c2ccc(CNC(=O)CN(C)C)cn2)CC(C)CN1 77302,Cc1cccc2cc(C(=O)NCC(C)Nc3ccc([N+](=O)[O-])cc3C(F)F)sc12 77303,c1(C(=O)NCC(CNC(C(C)c2ccco2)=O)O)ccn(C)c1 77304,N1(C(C(C)NC(=O)CN)=O)CCN(C)C(C(C)(C)C)C1 77305,N1(C(=O)CNc2ccccn2)CCC2(CCN(C(=O)C(F)CC3CCCC3)C2)C1 77306,c1(OC(C(CC)(Cc2ccc(OC)cc2)CC)=O)ccc2c(=O)[nH]ccc2c1 77307,c1(C(N2CC(NC(C3(COC)CCCC3)=O)C(F)C2)=O)cc(C)nnc1C 77308,C1(C(=O)NCC2CCN(C)C2)(OC)CCN(C(=O)Cc2cc(C3CC3)no2)CC1 77309,c1(C(=O)NC2C(NC(c3c(CC)oc(C)c3)=O)CC2)cc(C)c(OC)c(C)c1 77310,CCCC(C)(C)C(=O)NC(CNC(=O)C(C)S(C)(=O)=O)Cc1ccccc1 77311,Cc1ncnc(C)c1C(=O)NCC(C)CNC(C1CCOC1C)=O 77312,N1(C(COCCC#C)=O)CC(C(=O)NCC(C)C(C)O)C(CC)C1 77313,c1(C(N2C(C(N(C)C)=O)C=CC2)=O)cc2cc(Br)ccc2o1 77314,C1(NC(C2N(C(C)=O)CCC2)=O)CCN(C(=O)C(C)Sc2ccccc2)C1(C)C 77315,N1(C(C(C)OCC#C)=O)CC2(CC(CC(N3CC4(CC=CC4)C3)=O)C2)C1 77316,O(C=CC(=O)N(C)CC1(NC(=O)Cc2ccco2)CC1)CC 77317,N1(C(C2NC(=O)OC2)=O)CC2CCCC(NC(c3cc4ncccc4s3)=O)C2C1 77318,c1(-n2c(-c3ccc(C(F)F)cc3)nc(C)n2)ccc(-n2cnnc2)cc1[N+](=O)[O-] 77319,c1(C(=O)NC(C)CN(C(=O)C(Cc2ccccc2)N(C)C)C)c(O)cncc1F 77320,c1(C(N(CC(CC)NC(c2cnn(C)c2N)=O)C)=O)ccn(C)c1C1CCC1 77321,c1(OC)ccccc1C(C)N(C)C(C1CCN(C(c2cnn(C(C)C)c2)=O)C1)=O 77322,N1(C(C=CC)=O)CC(NC(=O)CC2(C#N)CCC2)CC1CO 77323,N1(C(C(C(C)(C)C)OC)=O)CCCC2(C1)CN(C(c1cc(C)c(C#N)cn1)=O)C2 77324,Cc1c(C)n(C)c2ccc(C(=O)NC3CCOCC3NC(C3CC(O)C3)=O)cc12 77325,C=CC1OCCCC1C(N1CCC(OCCNC(c2nn(C)c(C)c2Cl)=O)C1)=O 77326,c1(OC(CNC(C)=O)(C)C)ccc(C)nc1CNC(c1c[nH]c(=N)o1)=O 77327,N1(C(CN2CC(C)(OC)C2)=O)CCc2sccc2C1CNC(=O)CNC1CCC1 77328,C1(N(C(C(C)NC(CC)=O)=O)C)CCCN(C(c2cnn(C)c2COC)=O)C1 77329,C1(NC(c2ccc(C)o2)=O)(CNC(=O)C=CC2CC2)CC(F)(F)C1 77330,C1(CC)CN(C(c2ccc(Cl)nc2)=O)CCN1C(=O)CCc1cccc(OC)n1 77331,c1(CCCC)ccc(CC(=O)NC2CC2NC(=O)C(C)OCCOC)cc1 77332,C1(CNC(CC(COC)(C)O)=O)CCN(C(=O)CCNC(=O)NC)CCC1(F)F 77333,c1(NC(C2(C)CN(C(=O)NCC(=O)OCC)C2)=O)cc(F)cc(F)c1C#N 77334,C=CCC(C)C(C)(c1nnnn1C1CCC(F)(F)CC1)Nc1cnc(CC)nc1 77335,CC(C)(C)C(CNC(C1CN(CC(F)F)C1)=O)C(=O)NC(CCO)C(C)(C)C 77336,N1(C(Cc2c(C)cccc2F)=O)CCN(C(C2(S(C)(=O)=O)CC2)=O)CC12CCC2 77337,C(=O)(CC(CC1CCCCC1)NC(c1[nH]nnc1-c1ccccc1)=O)OCC 77338,C1(F)(C(N2CC(OCCOC)C2)=O)CCCN(C(=O)CC2CCCSC2)C1 77339,Cc1cc2c(C(=O)NCC3(C)CCCN3C(=O)Cc3cnc[nH]3)nccn2n1 77340,N1(C(C(CCC)C(C)C)=O)CCN(C(=O)CC2CCCCC2(F)F)CC(C)(C)C1 77341,S(=O)(=O)(c1cccc(N2CCOC3(CCC3)CC2)n1)NC1CC(C)SC1 77342,N1(C(c2cncnc2)C(=O)NCC=C)CCc2cnn(-c3ccccc3)c2C1 77343,N1(C(C(CCC)C)C(=O)NC2COC2)CCc2c(C(N)=O)cccc2C1 77344,c1(C(=O)NC(C)CCO)cccn1Cc1ccncc1 77345,C1(C(=O)NCC2CN(C(CCN(C(C)=O)C)=O)C2)CCCC(C(F)(F)F)O1 77346,C(=O)(CCC(C)OCC)NC(C1N(C(C(C=C)O)=O)CCC1)(C)C 77347,C12(NC(COCC=C)=O)CCC(CN(C(=O)C(CC)C3CCOCC3)C1)C2 77348,N1(C(CCC)=O)CCC(C(=O)NC2CC(C)(NC(C3CCCN3CC)=O)C2)CC1 77349,C#CCC(CC(=O)NC1(C(O)COC)CC1)NC(C1(CO)CCOC1)=O 77350,c1(C(C)=O)nc(C(=O)NC2CC2NC(c2cnn(-c3ccccc3)n2)=O)cs1 77351,c1(C(N2CCC(Cc3ccc(NC(C)=O)nc3)C2)=O)ccc(C#N)c(Cl)c1 77352,N1(C(c2cnc(C(C)=O)s2)=O)CCC(NC(=O)CCSC2CCCC2)C(C)(C)C1 77353,CC#CCCC(=O)NCC1COC(CNC(c2c(C3(NC)CC3)noc2C)=O)C1 77354,c1(OC)cc(C(=O)NCC2CCC2NC(=O)CN2CC(C)C2)cnc1OC 77355,C12(NC(c3ccc(CCC)[nH]3)=O)CC1CN(C(=O)C(CC)n1cccn1)C2 77356,C1(C(c2n(Cc3c(OC)cccc3)nnn2)NC(C)C)CC2CCC(C1)O2 77357,c1(C(=O)NC(CC)CN(C)C(C2(C(N)=O)CC2)=O)cn(C)c(=O)c2cncn12 77358,c1(OC)ncc(C)cc1NC(=O)NC(CC1CCCCC1)C(C)(C)C 77359,C1(C(=O)NCC(COCC)O)CC(NC(=O)Cc2cccnc2O)CCO1 77360,c1(C(=O)NCC2(NC(c3onc(OC)c3Br)=O)CCC2)ccc2c(c1)CCC2 77361,N1(C(COCC)=O)CC2COCC(C1)C2NC(=O)CCC1CCC(=O)N1 77362,c1(NC(C2C(C)(C(=O)OCC)C2)=O)ccc(-n2cccc2)nc1 77363,C1(C(=O)NCCCOCCOCCNC(C(C)C)=O)CC=CCC1 77364,N1(C(C2(C)CC2)=O)CC2(CCN(C(C3C4CCC3(c3ccc(F)cc3)C4)=O)C2)C1 77365,C=Cc1ccc(C(N2CCC2C(=O)Nc2ccc(C(F)(F)F)nc2)=O)cc1 77366,c1(CC)ccc(C)cc1C(=O)NCC(CNC(c1cc(C)ns1)=O)S(C)(=O)=O 77367,c1(CNC(C(=O)N(C2CCC(C#N)C2)CC2CC2)=O)coc2c1COC2 77368,c1(C(=O)NCC2(C(N(CCCN=[N+]=[N-])C)=O)CC2)cncc(Cl)c1 77369,C(=O)(C(F)CC(C)(C)NC(=O)Cc1ccc(F)cc1)NC1C(C)SCC1 77370,c1(NC(C2CCN(Cc3c(Br)ccnc3Cl)C2)=O)cccc2nsnc12 77371,N1(C(C(C)CCN(C)C)=O)CCC2(CCC(NC(=O)Cc3nccn3C)CC2)C1 77372,c1(C(C(=O)NC2COC2)N(C(CC)CC)C(C)CC)cc2c(cc1OC)CCC2 77373,C1(NC(Cc2n(C)ccc2)=O)CCN(C(=O)CCc2ncco2)CC12CCC2 77374,N1(C(C2C(CNC(c3ccc4c(c3)CC4)=O)C2)=O)CCN2C(=O)OCC2C1 77375,C#CCC(CC#C)C(=O)NCC1CCN(C(=O)CCc2cccc(F)c2)C(C)C1 77376,C1(C(N(C)CC2(O)CCCC2)=O)(NC(C2CCCC2F)=O)CCC(C)(C)C1 77377,N#Cc1c[nH]cnc1=NC1COC2(CCN(C(=O)C3=CCCCO3)CC2)C1 77378,C1(c2nnnn2C2CCCC2)(Nc2ccc(CC)cc2C)CC2COCC2C1 77379,c1(NC(c2c(C)nc(C)o2)=O)cnc2c(c1)CN(C(=O)CC#N)CC2 77380,CC1(C)C(CNC(c2c(O)cccc2F)=O)CCN1C(=O)CC1CCCOC1 77381,C12(NC(c3c(OC)c(=O)cco3)=O)CCCC1CN(C(c1cc(=O)cc[nH]1)=O)C2 77382,CCC(C)C(=O)C(=O)N1CCC(F)(C(=O)NC2CC2c2ccn(C)n2)CC1 77383,N1(C(C2(Cl)C(C(C)=O)C2)=O)CCOC(c2cn(-c3cccc(C)n3)nn2)C1 77384,C12(NC(c3c(=N)[nH]cnc3)=O)CCN(C(=O)CCOC3CCC3)CC1C2 77385,C1(CC(=O)NC2(CF)CCN(C(C(C)n3ccnc3)=O)C2)CC(=O)NC(=O)C1 77386,C1(C)(C(=O)OC)CN(C(c2cc(CNC(=O)CC3CC(F)(F)C3)[nH]n2)=O)C1 77387,CC(C)C(C)CC(=O)N(C1CC(C(=O)NC(C)CS(C)(=O)=O)C1)C 77388,O=S1(=O)CC2CN(c3nnc(-c4ncnc5[nH]cnc45)n3CCCCF)CC2C1 77389,c1(C(=O)NCC2C(C)CN(C(=O)Cn3ncnn3)C2)csc2cc(Cl)cnc12 77390,CCCC(C(=O)N(CC(C)(C)NC(C1CC(SC)C1)=O)C)OCC 77391,c1(NC(N2CCC(c3ccc(SC)cc3)CC2)=O)ccc(Br)c(Br)c1 77392,N1(C(CCC)=O)CCC(C(=O)NCC2(F)CC(C(=O)OC)C2)CC1 77393,c1(C(=O)OC)cccc(C(N2CC3CC2C3C(=O)NCc2ccncc2F)=O)n1 77394,c1(CCC(N2CCC(NC(c3cccc(C)c3)=O)C2)=O)c(F)cccc1Cl 77395,N1(C(CCOCCN(C(C(CCC)=CCC)=O)C)=O)CCCC(CO)C1C 77396,CS(=O)(=O)c1cnc(CCNC(c2cccc(OC(F)F)c2)=O)nc1 77397,CC1CCC(C)C1NC(=O)CC1CCCC1NC(=O)Cc1cnns1 77398,c1(C(=O)NC2CC(F)(CNC(C=C(C)C)=O)C2)cc2scc(C)c2[nH]1 77399,c1(OCC(=O)NCCCN(C(C#CC(C)C)=O)C)cc(Br)ccc1F 77400,C(=O)(CC(C)(C)C(=O)OC)NCC(C1CCC(=C)CC1)ONC(=O)c1cn[nH]c1 77401,C(=O)(CC(COC)NC(C1(C)CNC(=O)N1)=O)NCc1ncc(CC)[nH]1 77402,C(=O)(C(C)CC(C)(C)C)NC1(CC(N2CCC(COCC)CC2)=O)CCOC1 77403,c1(C(=O)NC(CNC(C2(CC)CC2(F)F)=O)(C)CO)cnc([N+](=O)[O-])n1C 77404,C1(C(=O)NC2CCCC2CNC(=O)CCc2ccncc2)(COC)CCCC1 77405,Cc1onc(CC(=O)NCc2ccc(CC(=O)O)cc2)c1-c1nn[nH]n1 77406,c1(C(=O)NCC2N(C(CC(C(C)C)O)=O)CCC2)nccc2c(Cl)cccc12 77407,c1(C(=O)NC(C(C)NC(c2cccc(CO)c2)=O)C)ccc(O)c(N)n1 77408,n1(C(C(=O)NC2CN(C(c3cc(C)on3)=O)C2)C)c(=O)oc2ccccc12 77409,N1(C(C2(F)CCN(C(c3ccc(O)nc3Cl)=O)C2)=O)CC(O)C(O)C(O)C1CO 77410,c1(C(N2CCC(F)(CNC(C3C(C)C3)=O)C2)=O)cc(-c2ccccn2)cc(F)c1 77411,C(=O)(C(c1cccs1)N(C)C(C)C)NCCSC 77412,C1(C(=O)NCCc2c(CNC(C(C=CC)O)=O)nco2)CCCC(CF)C1 77413,C(CNC(=O)C(C)C(F)(F)F)(CC(F)(F)F)NC(c1cccc(C(C)C)c1)=O 77414,Cc1ccc(Br)c(C(=O)NC2(C)CCN(C(c3c(C)cccc3O)=O)C2)c1 77415,c1(NC(C(C2(C)CC2)NC(CC2C(C)(C)C2)=O)=O)cnc2ccnn2c1 77416,C1(NC(CN(CC)CC)=O)CN(C(c2cccnc2NC2CCC2)=O)CCC1O 77417,c1(C(=O)NC2C(C(N(CC(F)(F)F)C)=O)C2)ccc2cnccc2n1 77418,C(=O)(C(F)CCC(C)(C)C)NC(CN(C)C)C(N1CCC(CO)C(C)(C)C1)=O 77419,S(=O)(=O)(c1nc(N2CC(CO)C(C3CC3)C2)ccc1Br)N(CCF)CC 77420,CC(CC(C)(C)O)NC(=O)C(Cc1ccccc1Br)NC(=O)C=Cc1cscn1 77421,C(CCCCC(=O)NC1CCCCCC1C(=O)NCCC(C(C)C)OC)OCC 77422,C(=O)(C1=CC2CC=CCC12)N(C)Cc1cccc(CNC(C2(CSC)CC2)=O)c1 77423,Cc1c(C(=O)N(CCCNC(C2CC(C(C)(C)C)C2)=O)C(C)C)nnn1C(C)C 77424,CCC(CC(F)F)C(=O)NCC1(F)CN(C(C2(C3CCCCC3)CC2)=O)C1 77425,N1(C(C2C(C)(CC)C2)=O)Cc2nccn2CC(NC(=O)C(c2cnn(C)c2)C)C1 77426,Cc1cc(C(=O)NCCN(C(=O)C(F)F)C2CC2)n2ncnc2n1 77427,C#Cc1ccc(C(=O)N(CCCNC(c2cc(C)n(CCO)n2)=O)CC)c(C)c1 77428,CN1CCC(C(C(=O)NCCCOCC2CC2)N(C2CCOC2)C2CC2)CC1 77429,N1(C(CSCCN(C)C)=O)CCCC(C2CCCN(c3nnc(C#N)s3)C2)C1 77430,c1(NC(C(=O)N(CC(=O)NC)C(C)C)C)cccc2c1NC(=O)CO2 77431,C(=O)(C(C)(O)C(F)(F)F)N(CCCNC(c1c(O)ncc(SCC)c1)=O)C1CC1 77432,C1(NC(c2cccc(O)c2F)=O)CN(Cc2c[nH]c3cccnc23)CC(F)(F)C1 77433,CCCC(CC(=O)NCCC(C(C)C)OC)NC(C1C=C(C)CS1)=O 77434,C1(CNC(C(C(C)C)NC=O)=O)CCN(C(=O)C(C)C#N)C1(C)C 77435,Cc1cc(C)c(C(N2CCOCC(C(=O)NCC(C)O)C2)=O)c(Cl)n1 77436,N1(C(C2N(C(CC(C)(C)OC)=O)CC=CC2)=O)CC2CC1C(F)(F)C2 77437,c1(NCC(=O)NC(CC2CN(C(C(CC)C)=O)C2)C)cccc(Cl)c1 77438,c1(C(CN(C)C)NC(C(CC)NCc2cccs2)=O)ccccc1C 77439,n1(CC(C)C)cc(CN(CCCN(C)C)C)c(CC2CCC2)n1 77440,C1(C(CN(C)C(c2cc(F)ccn2)=O)=O)CCCCC1(F)F 77441,N1(C(CCc2c(C)n[nH]c2C)=O)CCC2(CCCN2C(=O)CC2CSCCS2)C1 77442,CCCCCCC(C)C(=O)NC(CNC(=O)C(CC)n1cncn1)CC 77443,N1(C(C(CCC#C)O)=O)C2CCC1CC(C(=O)NCCOc1cc(Br)no1)C2 77444,C1(CC)CCN(C(=O)C(C)Cc2cnco2)C1CNC(C)=O 77445,CCC(CC(F)(F)F)C(=O)NCCC(C)N(C)C(c1cc(C(C)C)[nH]n1)=O 77446,CS(=O)(=O)C1(C(=O)NCC2CC(NC(C3CC(N(C)C)C3)=O)C2(C)C)CCOCC1 77447,CC(C)(C)C(CNC(c1nsnc1O)=O)NC(C1C=CCCC1)=O 77448,CN1CCOC(C(=O)NC2CC2CNC(=O)CC2CCC(C)(C)O2)C1=O 77449,N1(CCNC(CCCOC)=O)CCC(NC(=O)C(C)Sc2ccccc2F)CC1 77450,c1([SH](c2ncc(-c3cccc(C)c3)[nH]2)c2ccccc2)nc(=NCC(C)C(C)C)[nH]c2ccsc12 77451,N1(Cc2n(CC)ncc2)CCCC(CN(C)C(c2ncccc2Cl)=O)C1 77452,CC(C)CC(C)(C)C(=O)N1CCCC1CN(C)C(c1cncnc1C(C)C)=O 77453,C1(CNC(C2CCC(NC(C3(CCC)CC3)=O)CC2)=O)CC2(C1)CC(O)C2 77454,C1(COC)(NC(=O)CC2CC(C)C2)CCN(C(C2CCC(=O)O2)=O)C1 77455,n1(CC)cc(NC(=O)CC2CCN(C(c3ncccc3F)=O)C2)ccc1=O 77456,c1(C(=O)NCC)cc(NC2CC2C(=O)Nc2cccc(OC3CC3)c2)cc(C)n1 77457,N#CC1CN(C(c2cccc3c2OCO3)=O)CCN1C(c1ccccc1)=O 77458,C(C(C)(COC)C(=O)N1CCCCC1CNC(c1cnn(C)c1)=O)OC 77459,CCCC(CC(C)C)C(=O)N1CCC(C(=O)NCCC2CCN(C)C2=O)CC1 77460,c1(C(N(C(CNC(CC(C)c2ccco2)=O)C)C)=O)ccnc(-c2ccco2)c1 77461,N1(CC)CCCN(C(C2CCC(C)CC2)C(=O)NCCCF)CC1=O 77462,N1(CC(=O)NCCCN(C(=O)C=CC2CCOCC2)C)CCN(C2CC2)C1=O 77463,c1(C(N(C(C)CCNC(c2nnsc2C(F)F)=O)C)=O)nc2ncccn2n1 77464,C(=O)(C(C)(O)c1ccccc1)NCC(CC)NC(=O)Cc1csnn1 77465,c1(C(N2CCOC3(CCC3)C2)C(=O)Nc2c(C)cccc2)ccc(C)c(C)c1F 77466,c1(OC(C(=O)NC(C(C)NC(COCCCC#C)=O)C)(C)C)ccc(Cl)cc1C 77467,CN1C(=O)NC2(CCC(NC(C3CCCCC(O)CN3)=O)CC2)C1 77468,C(=O)(CC(F)(F)C(F)(F)F)N1CC(C)(C)C(NC(C2CC3(C2)CC3F)=O)CC1 77469,N1(C(C2CC(=C)C2)=O)CC(C)CCC1CNC(c1ccc(C(C)C)c(F)c1)=O 77470,C(=O)(C(O)C(C)(C)CC)NC1CC(C(N(CC(CCC)O)C)=O)CC1O 77471,CN1Cc2ccc(C(=O)NC3CCCCC3N(C(=O)COCCF)C)cc2C1 77472,C1(CC(=O)NCCN(C(=O)C=C(C)C(F)F)CCOC)CNC(=O)C1 77473,O(P(C)(=O)CNC(=O)CC1(C)CCN1C(C12CCC(C1)C2)=O)CC 77474,c1(C(=O)NC2CCC(CCNC(C3N(CCC)CCC3)=O)C2)ccc(F)c(O)c1 77475,c1(C(=O)NCC23C(CN(C(C4C(CC)CCO4)=O)C2)C3)cccc([N+](=O)[O-])c1.CCO 77476,CC(CNC(=O)CCC1CCCCN1C(=O)CCCC1CC1C)C(C)(C)C 77477,C1(CNC(=O)CNC(c2nncs2)=O)CCCCN1C(C12CCCC1C2)=O 77478,c1(OC)ccc(C(=O)N(CCCN(C)C(C2CCC(C)C2)=O)C)n2nccc12 77479,c1(C(N2C(C#C)CCC2)C(=O)Nc2ccccc2CC)cccc([N+](=O)[O-])c1C 77480,c1(C(=O)NC2C(NC(C(COC)N(C)C)=O)CCC2)ccn(C)c1C 77481,c1(CC)nnc(O)c(C(=O)NCC23CCCNC2CCC3)c1CC 77482,c1(C(=O)NCCCN(C2CCCC2)C(c2on(C)c(=O)c2)=O)cc(F)cnc1O 77483,C(=O)(C(C)(C)C(=O)OC)NCC(CC=C)NC(=O)CC1(C)CC1 77484,c1(CC)c(C(N2CCCC(NC(C3CC(C)(F)C3)=O)C2)=O)cnn1C(C)(C)C 77485,C1(CC=C)(C(=O)N(C(C)CC)C)CN(C(C2CCC(=O)C2)=O)C1 77486,C1(N(C(=O)CCCF)CC)CCCN(C(c2cn(C(C)C)nc2Br)=O)C1 77487,C1(C(=O)NC)CCN(C(=O)CCN(C(=O)CN2CCCC2C)C(C)C)C1 77488,C12(NC(c3cn(CC)nc3)=O)CCCC1N(C(c1c(C)cc(O)nc1C)=O)CC2 77489,N1(C(C(CC)OCC)=O)CCCCCC(NC(c2cnn(C(C)(C)C)c2C)=O)C1 77490,C1(NC(NC(CC)CC)=NCc2snnc2C)CCC(=O)N(C)C1 77491,c1(C(N(CCN(C(C2C(CC)OCC2)=O)CC)CC)=O)ccn2cc(C)nc2c1 77492,c1(OC)ccccc1C(=O)NCC1(CCNC(C2(CO)CCCO2)=O)CC1 77493,CC(N=c1nc2scnc2c(NCCS(=O)(=O)CCO)[nH]1)c1cn(C)nn1 77494,c1(C(=O)NC(C)C2=CCN(C)CC2)cccc(P(C)(C)=O)c1 77495,C(=O)(CCCC(C)(C)C#N)N1C2(C(N(CC(CC)O)C)=O)CC(C1)C2 77496,C(C1(C)OCCc2ccccc21)NC(C1CN(C)CCO1)C 77497,N1(C(=O)CC(F)(F)F)CCC(C2CN(C(C3(C(F)F)CC3(F)F)=O)C2)CC1 77498,c1(C(=O)NCCN2CCCC(c3nc(C4CCN4)no3)C2)ccc(Cl)c(NC=O)c1 77499,N1(C(C(CC)CO)=O)CCN(C(c2cccc(Cl)c2N)=O)CC1C(C)C 77500,CC(C)CCC(C(=O)NCC1(F)CC(CO)C1)NC(=O)CC=CC(C)(C)C 77501,C(=O)(C1=CC2C=CC(C1)C2)N1CC(C(=O)NC(c2ccn(C)n2)C)CC12CCC2 77502,c1(C(N(CCC(C)=O)C)=O)ccc(-c2cn(CCCCCO)nn2)o1 77503,c1(C(=O)OC)cc(C(N2CC(NC(=O)CN=S(C)(C)=O)CC(F)C2)=O)cc(C)c1 77504,S(=O)(=O)(c1ccc2nc(N3CC4CC=CC3C4)sc2c1)N1CC2C(C)(CC2)C1 77505,N1(C(C2(NC(c3c(C)n(C)nn3)=O)CC2C)=O)CCOCC(O)C1 77506,Cc1c(N)ccc(C(N2CCC(=CCNC(C3CCCC3(F)F)=O)CC2)=O)c1C 77507,Cc1nc(C(N2CCN(C(=O)CNC(C3CSC3)=O)CC2)=O)ccc1C#N 77508,C1(CCC(N2CCC(CN(C)C(C3(F)CC3)=O)C2)=O)CC(C)(C)CO1 77509,N1(C(c2onc(C)n2)=O)CCCC2(CNC(=O)C(C)O)CCCCC12 77510,CC1(C)CC(NC(N2CCOCC2CO)=O)c2cccc(Br)c2O1 77511,c1(C(N2CCCC(NC(C3(C)CCC(OC)CC3)=O)C2)=O)cc(C)n(C)c(=O)c1 77512,CCCC(CC(=O)NCc1c[nH]nc1C1CCC1)NC(=O)OC(C)(C)C 77513,c1(C(=O)NC2(CNC(C(CC(C)C)(C)O)=O)CCC2)ccc2c(c1)C=CS2(=O)=O 77514,N1(C(c2c(CCC)[nH]cc2)=O)CCC(C(C)NC(=O)C(C)(C)CC)CC1 77515,c1(C(N(CCC)CCNC(=O)C(CC)C(F)(F)F)=O)ccc([N+](=O)[O-])c(C)c1 77516,c1(OC)ccccc1CN1CCC(C)(NC(=O)COc2ccc(CO)cc2)C1 77517,C12(N(CCC(=O)NC(C)=O)C(=O)CCC3CC3(F)F)CCC(C1)OC2C 77518,C1(NC(C(CC)C(C)C)=O)C2CCCN(c3cc(Cl)c(O)nn3)C2C1(C)C 77519,CC(O)C(C)(C)C(=O)N1CC2CC1(C(=O)NCCCn1cncn1)C2 77520,c1(COC)ccc(C(=O)NC2CC(CNC(C3CCC(=O)C3)=O)C2)cc1F 77521,C1(CNC(c2ccc(C(C)O)cc2)=O)CCC(C)CN1C(=O)CCc1nncs1 77522,C=CC(C)(O)CC(=O)N(CCC(=O)N1CCC(O)C1CC)OC 77523,c1(C(=O)NCC=CCNC(C2CCC(C)O2)=O)c[nH]c2nc(Br)ccc12 77524,c1(C(N(CCCCCNC(C2CCC(C)CC2)=O)C(C)C)=O)cc([N+](=O)[O-])ccn1 77525,c1(NC(C(N2C(CCC(=O)NC)CCCC2)=O)=O)cnc2[nH]cnc2c1 77526,C(=O)(C(O)CC(N)=O)NC1CC(CCNC(CCCOc2c(C)cccc2)=O)C1 77527,C1(C(N(C2CN(C(C3(C(F)(F)F)CCCCC3)=O)C2)C)=O)CCC12CCCO2 77528,c1(C(N(C2CCC2)CC)=O)coc(C)n1.C(=O)(C=CC(=O)N(C)C)NC 77529,CCCS(=O)(=O)N1CCCC1C(C12CC(n3cc(CC4CC4)nn3)C1C2)NC 77530,c1(CNC(C2(CC)CCC2)=O)nc(CNC(C2CC(C(F)(F)F)C2)=O)cc(O)n1 77531,CC(C)C(F)C(=O)NC1C=CC(C(N2CCN(C(=O)CO)CC2)=O)C1 77532,N1(C(CNC(=O)NC)=O)CCC(C2CC2)C1CNC(c1n[nH]c2c1CCOC2)=O 77533,C1(C)(CNC(COc2cccc(C)c2)=O)CN(C(=O)C(C)N(C)C)C(C)(C)C1 77534,n1(CCC)nccc1C(C(=O)NC(C)C)N(C)CCn1ccnc1 77535,c1(C(=O)NCC(CC=C)NC(c2cc(C#N)c[nH]2)=O)nc2sccn2c1C 77536,N1(C(c2cc(COC)oc2C)=O)CC2(CC2)CC1CNC(C1(C)CC(OC)C1)=O 77537,N1(C(C(C=C)O)=O)CCC2CCCN(C(=O)COc3ccc(F)cc3)C2C1 77538,CC1CC(=O)NC(C(=O)NCC(O)CNC(=O)C(=O)NCCC(N)=O)C1 77539,c1(CNC(C2CCC(F)(F)C2)=O)cccnc1CNC(C1CCCOC1)=O 77540,CCCC(CC1CCCC1)C(=O)NCc1cc(C(=O)OC)co1 77541,CCC(C)(C)C(O)C(=O)NCC1CN(C(C2(C(N)=O)CC2)=O)CC1(C)C 77542,CN1CCn2nc(C(NC3CCc4ccc(CC(=O)O)cc43)=O)cc2S1(=O)=O 77543,c1(C(=O)NCC(CC)NC(=O)C(C)N2CCC2)ncc(Br)cc1F 77544,CC1CC(CNC(c2ccnc(C(F)(F)F)c2)=O)CN1C(=O)Cn1cnnc1O 77545,c1(C(=O)NCC2CC(NC(=O)C=CC3CCC3)CC2O)cc2c(nc1O)CCC2 77546,c1(C(=O)NCCN(CCC)C(C2(C)CC2C)=O)ccc(-n2ccnc2)c(C)c1 77547,Cc1n[nH]c(=N)n1C1CCN(C(=O)C(=O)NCc2csc(C(F)F)n2)CC1 77548,C(=O)(C1OCCn2ccnc21)N1CCC(CN(C)C(c2ccc3c(c2)CC3)=O)C1 77549,CCCCC(CNC(=O)CCC(C)=O)NC(c1csc(C)c1)=O 77550,c1(N(C(c2ccc(C)cc2)c2ccccc2)CC)nc2ccccn2c1[N+](=O)[O-] 77551,N=c1ccc(C(N2CCC(CNC(c3coc(O)n3)=O)C2)=O)n[nH]1 77552,C1(C)(C(N2C(C(N(C3CCC(F)(F)C3)C)=O)CCC2)=O)CCC2CC2C1 77553,C1(C(=O)NCCn2cc(CNC(C(C(C)C)C)=O)nn2)CCCCNC1=O 77554,Cc1cc(Cl)c(C(N2CCCN(C(c3n[nH]c4c3CCOC4)=O)CC2)=O)cc1C 77555,C1(C)(CNC(C(C)OCCCC)=O)CCN(C(c2cc(N)cc(F)c2)=O)CC1 77556,C(=O)(CCC(C)(C)[N+](=O)[O-])NC1CCN(C(CNC(=O)NC)=O)CC1C(F)(F)F 77557,c1(C(=O)NC2(C)CN(C(c3ccc(CO)cc3)=O)C2)ccc(N)c(O)c1 77558,c1(C(=O)OC)ccc(-c2nncn2C(C)(C)C)c(F)c1.N12CCOC(C1)C2 77559,CCC(CC)C(c1nnnn1Cc1cccs1)NCC1COCC1(C)C 77560,N1(C(C2(OC)CC2)=O)CCCCC(CNC(C23CC(CC(F)F)(C2)C3)=O)C1 77561,Cc1cc(C(N2CC(NC(c3cc(Cl)ccc3N)=O)CC(F)C2)=O)c(Cl)cc1F 77562,CCCC(C(=O)N1CCC(NC(=O)COC2CN(C(C)=O)C2)C1)NC(C)=O 77563,C1(C(=O)N(C(C(N)=O)C2CC2)C)(CC)CN(C(=O)CCc2cccnc2)C1 77564,C1(=O)C(N(C)C)CN1.C1(CC(=O)N(CCC2CC2)CC)OCCCOC1 77565,C1(=CC(=O)NCCN(C(C(c2c(F)cccc2F)OC)=O)C)CCC(C)(C)CC1 77566,c1(NC(CCC(=O)OCCCC(C)=O)=O)ccc(C)c(OCCF)c1 77567,C1(CC=C)(C(=O)NC(CCCC)c2ccccc2)CN(C(C2CC=CC2)=O)C1 77568,c1(OCC)cc(C(=O)NC2(CNC(C3CCC3(C)C)=O)CC2)on1 77569,c1(OC(C(=O)NC(C2(NC(N)=O)CC2)C)C)ccccc1N(C)C 77570,N1(C(C(C)SCC)=O)CCC2CN(C(c3cnc4cccnc4c3)=O)CC2CC1 77571,CC(C(F)F)=CC(N1CCC1CNC(=O)COCCOCCO)=O 77572,c1(CNC(c2cnn(C)c2C)c2n(C(CC)C)nnn2)cc(F)ncc1C 77573,C(=O)(C(C)S(C)(=O)=O)NC(C(C)NC(C=C(CCC)CCC)=O)(C)C 77574,c1(OC)ccc(CNC(=O)CC2CCCN2S(=O)(=O)Cc2ccccc2)cc1O 77575,CN1CCN(C(=O)CC2CSCCO2)CC1C(=O)NCC1(C)NC(=O)NC1=O 77576,c1(OCCC(=O)N(C(C)CCNC(=O)CC2CCCN2C)C)ccccc1F 77577,N1(C(C(C)CC2CCCC2)=O)CCC(N(C(=O)CC(C2CC2)C2CC2)CCO)CC1 77578,N1(C(CCCC2C(C)C2)=O)CC(C(=O)NCCNC(=O)CO)C2(CC2)C1 77579,C(=O)(CCC(=O)NCC(CC)NC(C1CCCCC1OC)=O)NCCC 77580,C1(CC#C)(C(=O)NCC(C)(CC)NC(c2cncc(Cl)c2)=O)CC=CCC1 77581,c1(C(=O)NCC2(CCNC(c3cc(C(C)C)no3)=O)CC2)cc(C#N)c[nH]1 77582,c1(C(N(C)CC2CCCN(C(C3(C)ON=C(C)C3)=O)C2)=O)cc(N)c(Cl)cn1 77583,C(=O)(CC(C)(C)CNC(=O)C(C)(F)C(=O)OC)NCC1OCCN(CC)C1 77584,c1(C(C(=O)NCCCOC(C)C)N(CC=C)C)cccc(Cl)c1 77585,CC1C(NC(C2CCCCCC2)=O)CCN1C(c1cccc(-n2ccnc2)c1)=O 77586,N1(C(C2(SC)CCOCC2)=O)CCC2(CC1)CCN(C(=O)Cc1n[nH]c(C)n1)C2 77587,N1(C(C(N(C(CNC(CN(C)C)=O)=O)C)C2CC2)=O)CCC(CCCO)C1 77588,CC(C)CC(C)C(=O)N1CCCC(F)(C(=O)NCCCc2cc[nH]n2)C1 77589,N1(C(CN2CCOCC2Cc2ccn(C)n2)=O)CC2CC1(C(=O)NOC(F)F)C2 77590,c1(COC(C23CCC(C2)C3)=O)cc(Br)sc1Br 77591,c1(C(N(CCNC(C2C(CC)CCC2)=O)CCOC)=O)c(C)nc(C)n1O 77592,C1(CNC(C(C)SC)=O)N(C(=O)CCn2cccn2)CCC1(C)C 77593,c1(OCC(=O)N(C)CC2(NC(CCC(=O)OCC)=O)CC2)ccc(CC)c(O)c1 77594,c1(C(=O)NCC(CN(C(C2CC2F)=O)CC)(C)C)ncccc1Br 77595,C1(NC(CN(C)C(N)=O)=O)(CNC(=O)CC2CCCOCC2)CC(F)(F)C1 77596,c1(OC(C)(C)C(=O)NCCC(=O)Cc2ccc(F)cc2)cc(F)cc(F)c1 77597,C1(CNC(COCCCOC)=O)CC2CCC(C1)N2C(=O)C(C)(C)C(C)C 77598,Cc1ccc(O)c(C(=O)NC2CC3(C2)CC3C(=O)NC(C)CC(C)C(F)F)c1 77599,c1(CC)nn(C)c(Cl)c1C(=O)NCCCC1(NC(c2cccc(C#N)c2)=O)CC1 77600,N1(C(c2c(C)n(C)nn2)=O)CC(CNC(c2ncc[nH]c2=O)=O)CC(C)(C)C1 77601,C1(NC(C2(CC=C)CCOC2)=O)CCN(C(=O)Cc2cccc(C)c2Cl)C(C)C1 77602,c1(C(N2CC(C)N(C(C3CCc4cncn4C3)=O)CC2)=O)cc2n(n1)CCCO2 77603,NS(=O)(=O)c1ccc(C(=O)NC2CCCC23CN(C(c2cnns2)=O)C3)o1 77604,Cc1nn(C2CC2)cc1C(N1CCOC(C2CCOCC2)C1)C(=O)OC.C1(C)(N)CC1 77605,c1(C(N2CCC(CCNC(C3=CCCC3C)=O)C2)=O)ccc(Cl)c(Cl)c1N 77606,n1(CC(N2CC(CNC(c3ccc(OC)s3)=O)C2)=O)ccc(C)cc1=O 77607,C1(CC(C)NC(=O)Cc2cn(C)nc2Cl)CCN(C(=O)CN2CCCC2=O)CC1 77608,c1(N2CC(C)C(CO)CC2)nc(=NCc2ccncc2F)[nH]c2c1COC2 77609,C(=O)(CCC(=O)NCC1(C)CCN(C(=O)CC(CC)SC)C1)NCC 77610,C1(CNC(CSCC#C)=O)CN(C(c2cccc(F)c2CC)=O)CCC1(C)C 77611,c1(N2CCC(CCOC)(NC(c3cc(C#N)c[nH]3)=O)C2)ncnc(C)c1F 77612,N1(C(C)=O)CC=C(CNC(=O)CNC2CCCN(CCN3CCCC3=O)C2)CC1 77613,CCC(CNC(c1ncccc1F)=O)(CC)C(=O)NC1CC1C(C)C 77614,N1(C(C(CC)F)=O)CCOC2(CCC(NC(c3cc(C#N)ccc3C)=O)CC2)C1 77615,CC1CN(C(=O)CC2CCN(C(C3CC4C(C3)C4(C)C)=O)CC2)CC(C)O1 77616,C1(CC(N2C(C(C)(C)NC(CSCCC)=O)CCC2)=O)Cc2ccccc2N1 77617,N(C(=NCCF)NCC12CC(C1)C(C)(C)O2)C1C(C(C)C)C1 77618,c1(OC)cccc(OCCC(N2CC3(NC(=O)Cc4ncoc4C)CC2C3)=O)c1 77619,c1(N2CCC(CC=C)(NC(=O)CN3CCOCC3)C2)ncnc2c1CCC2 77620,N1(C(c2c(N)ccc(C)c2)=O)CCCC12CCN(C(=O)CCCCCF)C2 77621,C1(C(=O)NCC(=O)N(CC(C)(C)NC(C=CCCC)=O)C)CC(=O)NC(C)C1 77622,c1(NC)ccc(CNCC2=CCCOC2)cc1[N+](=O)[O-] 77623,C(=O)(C1CCCn2c(Br)cnc21)NCC(N1CCN(C(CC(=C)C)=O)CC1)=O 77624,Cc1cc(N2CCN(C(C3CCCC4(CC4)C3)=O)CCC2C)n2ncc(C)c2n1 77625,C1(O)(COC)CCN(C(C2CC(CNC(=O)C(C)(F)c3ccon3)C2)=O)C1 77626,N1(C(C2C(CNC(CCNC(C)=O)=O)C2)=O)C2CCC1CC(C(N)=O)C2 77627,C1(OC)CC(NC(=O)C2=C(Cl)CC2)C12CCN(C(=O)C(C)(C)C(F)F)CC2 77628,c1(CC(=O)N(CCCNC(c2nc(C)sc2C)=O)C(C)C)cc(F)ccc1Cl 77629,C(=O)(C(O)CC1CC1)NCCN(C1CCCCC1)C(C(C)n1cnnn1)=O 77630,c1(OC)ccccc1C(CNC(C)=O)NC(C1(C(N2CC2)=O)CC1)=O.C(=O)C=CF 77631,C1(N(C(C2C(C)OC(=O)N2)=O)C)CCCN(C(=O)CC2CCCCC2(C)C)CC1 77632,C1(OC)CCCN(C(C2CC(O)CN2C(c2ncncc2N)=O)=O)CC1 77633,c1(SC)nc(O)nc(C)c1C(=O)NC1CCCCC1NC(=O)C1=CCCCC1C 77634,C1(C(N(CCNC(C(C(C)c2ccccc2)O)=O)C2CC2)=O)CC2C=CC1CC2 77635,Cc1ccc(C(=O)NCC(C2CCN(C(C3(O)CCOC3)=O)CC2)F)nc1 77636,n1(CC)cnc2[nH]c(=NCC3CCCC3O)nc(N3CCCC(COC)C3)c12 77637,N1(C(C2NC3CCC2C3)=O)CCOC(Cn2cc(-c3ccoc3)cn2)C1 77638,C1(NC(c2ccc(C(C)=O)cn2)=O)CCC(C)N(C(C2CCOC2)=O)C1 77639,C1(C(=O)NCCn2ncc(C)c2)CCCN(C(c2scnc2C(C)C)=O)C1 77640,N1(C(C(=O)NC(C2C(COCCOC)CCC2)=O)=O)CC2CCCN2CC1CO 77641,C1(C(N2CCC(CF)(NC(c3cnco3)=O)C2)=O)(CC)CCNC1=O 77642,c1(CN(C(c2nc(C)sc2)=O)C(C)C)cccc(NC(=O)C(C)C2CC2)c1 77643,c1(-n2ncc(C(C(=O)NC)N(C(C)CCC(=O)OC)C)c2)cccc([N+](=O)[O-])c1 77644,c1(OC(C(=O)NC(c2c(C)noc2C)C(F)(F)F)CN(C)C)cc(Cl)cc(Cl)c1 77645,N1(C(CSCC#C)=O)CCN(C(=O)C=C2CCC(C)CC2)C(CC(F)F)C1 77646,c1(CNC(C(CO)NC(CC2CCC(=O)NC2)=O)=O)cc(O)ccc1F 77647,CCCC(CCCNC(C1CC1F)=O)NC(=O)CCOCc1csc(C)n1 77648,C#CCC(C(=O)NN1CCCC1C(N1CC(c2cnccn2)C1)=O)C1CC1 77649,c1(C(N2C(C(N(CCC#N)C3CC3)=O)CC(F)(F)C2)=O)cc(O)c(O)c(O)c1 77650,C1(NC(c2cnc(CC)s2)=O)C2CCN(C(c3ccc(NC=O)cc3)=O)CCC12 77651,C12(NC(COC3(C)CCOCC3)=O)CCC(CC1)N(C(=O)C=Cc1ccc[nH]1)C2 77652,c1(C(N2C(CNC(CC(C)C)=O)C(C)CC2)=O)c[nH]c2ccc([N+](=O)[O-])cc12 77653,N1(C(c2c(C)nc3sccn32)=O)CCCC2(CCCN2C(c2ccnn2C)=O)C1 77654,C1(NC(CCCCOC)=O)CC2CCC1N2C(=O)C(C)Cc1cccc(Cl)c1 77655,C#CC1(OCC(=O)NCC2CCN(C(=O)C(CO)c3ccccc3)C2)COC1 77656,C(N=c1cccc(S(=O)(=O)NC2CCC=C2Br)[nH]1)C1CC(C)(C)OC1 77657,C=CC1(C(=O)NOC(C)C)CCN(C(=O)CC2C=NN(C)C2=O)C1 77658,c1(CC(=O)NCC2CCN2C(c2cc(C(F)F)no2)=O)ccccc1Br 77659,c1(C(=O)NC2CCCCN(C(CCC=C)=O)C2)cc(S(N)(=O)=O)c(F)cc1OC 77660,C(=O)(C1=CS(=O)CCC1)N1CC=CCC(NC(=O)CC2(Sc3ccccc3)CC2)C1 77661,c1(C(N2CC(NC(=O)Cc3cccnc3Cl)CC(C)C2)=O)c[nH]c2ccccc12 77662,N1(C(c2cnc(C)[nH]2)=O)CCN(c2ccc(CNC(C3CN(C)C3)=O)cc2)CC1 77663,c1(Cc2c(N)cnn2CC)ccc(F)cc1F.C1(c2nnnn2CC)(CC)CCSC1C 77664,N1(C(c2c(CNC(CCc3ncn(C)c3)=O)c[nH]n2)=O)CCCC(N=[N+]=[N-])CC1 77665,CC1CN(C(C2C3CCC(C3)C2NCc2ccc(F)cc2)=O)C(C)(C)C1 77666,C1(C(N(C)CC2(NC(c3c(COC)scc3)=O)CC2)=O)CCS(=O)(=O)N1 77667,C1(C(=O)NCC(C)(C)C2CCC2)C=CCN1C(=O)COCCN(C)C 77668,C1(CNC(c2n(CC)cnn2)=O)CCCCN1C(C1OCCOC1C(F)(F)F)=O 77669,c1(C(C)NC(=O)OC(C)(C)C)ccc(OC(F)F)nc1.C12CC(C)(C1)NC2=O 77670,C(=O)(C(C)N=c1[nH]c2ccccc2s1)NC1CC(CNC(CCCCC#C)=O)C1 77671,CC(C)(C)CCNC(N1C(C(=O)Nn2cc(C#N)cn2)COCC1)=O.C1CC1 77672,Cc1cc(SCC(N2CC3(C2)CN(C(=O)CC(C)(C)CN(C)C)C3)=O)ccc1F 77673,CN1CC(CC(N2CC(F)(CNC(c3csc(C(F)(F)F)n3)=O)C2)=O)CC1=O 77674,C1(CC(=O)NC(C)CN(C(=O)C(N2CCC(O)CC2)C)C)Cc2ccccc2O1 77675,N(C1CCC(N=c2[nH]nc(C#N)s2)c2ccccc21)Cc1c(C)nc(N(C)C)s1 77676,C1(CNC(COCCC=C)=O)CCC2CN(C(=O)CC3CCSC3)CC12 77677,c1(C(N2CCC(NC(c3ccc(OC)s3)=O)(CF)C2)=O)cc2sc(C)nc2[nH]1 77678,C1(C(N(CCCNC(CNS(CC)(=O)=O)=O)C)=O)CC(F)(F)C1(F)F 77679,Cc1ccc(OCC(=O)N(CCNC(C2(C(C)C)CNC(=O)C2)=O)C2CC2)cc1 77680,C(N=c1[nH]cc(Br)c2ccc(Br)cc12)C1C(O)COC1 77681,c1(C(=O)NC(c2cccnc2)C(=O)NCc2[nH]nc(C(C)C)n2)ncncc1Cl 77682,C1(NC(C2(OC)CCN(C(c3cnc(OC)s3)=O)C2)=O)CCCCC1(C)C 77683,Cc1cc2c(C(N3CC(NC(C4CC4(C)C)=O)C4(CCC4)C3)=O)nccn2n1 77684,N12CC(C)(CC1(C)C)C2.CS(=O)CCCCN(c1scc(CC(=O)OC)n1)C 77685,N1(C(C(=O)NC(C)C)=O)CCC2(NC(=O)CC3(O)CCCCC3)CCCCCC12 77686,C(=O)(C#CC1(C)CC1)NC(CC)CNC(=O)CSCC1CCCO1 77687,CCCC(O)CC(=O)NC1CC2CC1N(C(=O)CC(COC)COC)C2 77688,C12(C(=O)NCc3c(CC)noc3)CCN(C(=O)Cc3ccccc3)CC1C2 77689,CC1CN(C(=O)CS(N)(=O)=O)CC(C)CN1C(c1nccc(Cl)c1O)=O 77690,c1(C(N(C)C)=O)nnc2ccccn12.C1(=O)C#CC(=O)NCC23OCC(C2)(C3)CN1 77691,Cn1nc2c(c1C(N1CC(NC(C3CCOC3)=O)C(C(F)(F)F)C1)=O)CCC2 77692,C1(N(C(Cn2c(C)ncc2)=O)C)CN(C(C2CC(F)(CO)C2)=O)CC1O 77693,c1(C(=O)NC2CCC(C(N3CCC(C)(O)C3)=O)C2)ccc2c(c1)OCO2 77694,C1(CC=C)(C(=O)NC2CCCSCC2)CCN(C(C2CC(F)C(=O)N2)=O)C1 77695,C1(N(C(C2CC2C)=O)CC)CCC(NC(C2CC(C)=NO2)=O)CC1 77696,c1(NCc2nn(CC)nc2C)cc2c(I)cnn2cn1 77697,C(=O)(C(F)(F)CC(C)C)NC(CN(C(c1cnc2ccnn2c1)=O)CC)C 77698,O=C(CCC(F)(F)F)NCC1C(O)C(O)CN1C(=O)C(O)CN1CCCC1 77699,N1(C(C2(CC)CCCC2)=O)CCC(C)C(N(C(=O)CCC2(C)CC2)C)C1 77700,N#CC1(C(N2CC3CC3(CNC(=O)CCc3cnc(O)[nH]3)C2)=O)CC12CCC2 77701,c1(C(=O)OCC)cc(C(=O)NC(CNC(=O)Cc2nccn2C)CC)ns1 77702,c1(NC(C(C2CCCO2)NC(CNC(CC)=O)=O)=O)ccc(O)c(F)c1 77703,CC1=C(CNC(=O)C(C2CCN(C(=O)CC3CCC(=O)C3)CC2)C)CCC1 77704,c1(C(=O)NC(C2N(C(c3cc(C)sn3)=O)CCCC2)C)c(N)c(F)cc(F)c1F 77705,c1(C(=O)OC)cc(C(N2CCCC(C(C)(C)C)C2)C(=O)NCCCF)c(C)s1 77706,C=CC(CC)CC(=O)N1CCOCC1CN(C)C(c1cn(C(F)F)cn1)=O 77707,CC1(CNC(=O)CC2CC(O)CN2C(=O)COC2CC=CC2)CCCCCC1 77708,C1(N(C(c2sc(CC)c(C)c2)=O)C)CN(C(C23CCC(C2)C3)=O)CC12CC2 77709,c1(C(C)N(CCNC(=O)N(C)C)Cc2ccnc(Cl)c2)cccc(F)c1 77710,CC(C)C(O)CCNC(=O)C(CCOCCO)NC(c1cc(O)nn1C)=O 77711,c1(C(=O)OC)c(C)cc(C)nc1NC(C)CCNC(C1(C2CCOCC2)CC1)=O 77712,C1(CC(=O)N(C)CC2CCN(C(=O)CS(N)(=O)=O)C2)CCC2(CCC2)O1 77713,CC1CC(NC(c2ccco2)=O)CN1C(C1CCCC(O)C1)=O 77714,c1(OC)ccc(CCC(=O)N2CC(NC(=O)CCc3c(N)cnn3C)C2)cc1F 77715,C1(NC(c2cc(CC)[nH]n2)=O)CCN(C(c2nc(-c3cccs3)no2)C)CC1 77716,c1(CCC(=O)NCC2C(CNC(=O)Cc3cccs3)CC2)csc(C(F)(F)F)n1 77717,Cc1cc(C)c(C)c(C(=O)NCC2(O)CN(C(c3coc(CO)c3)=O)C2)c1C 77718,c1(OC(C(=O)NCCCC(C)NC(C2(C=C)CCC2)=O)C)cccc(C)c1C 77719,C1(NC(CCCOCC)=O)CC12CCC(NC(=O)CCNC(C1CCC1)=O)CC2 77720,C(=O)(CN=c1cc[nH]cc1)N1CC2C(CNC(=O)C(F)=CC3CC3)(C2)C1 77721,c1(C(N2CC(N(C)C)C(C)(C)C2)C(=O)NC)cc(Br)cnc1OC 77722,N1(C(C(C)Cc2ccc(F)cc2)=O)CC2CC(NC(=O)C3CC3)CC1C2 77723,N1(C(CSCCN(C)C)=O)Cc2ccccc2C1C(=O)N(C)C 77724,c1(CC)cc(C(=O)NCCCCC(=O)NC(c2ncn(C)n2)C)c(C)o1 77725,C1(C(=O)NC2CCC(CC(N3CCC(C(=O)OCC)C3)=O)C2)CCCC(C#N)C1 77726,C(=O)(C1=CCC2CCC1N2C(=O)C(C)(C)CC(F)F)NCC(C(C)C)(C)O 77727,CC(=O)CCC(=O)NCC(C(C)(C)C)NC(c1ccc(-c2ccccc2)o1)=O 77728,C(CC(C(=O)NCC(C)OC(F)F)OC(F)F)NC(C(C)NC(C(C)C)=O)=O 77729,C1(C)(CNC(c2cnn(CC)c2C)=O)CCCN(C(c2c(C#N)cnn2C)=O)C1 77730,Cn1nnc(CNC(=O)C(C)(C)C#N)c1C(N1CC(CO)C1(C)C)=O 77731,N1(C(C(C#C)(C)C)=O)CCOC2(CCC(NC(=O)CCCCN(C)C)CC2)C1 77732,c1(CC(=O)NCC(CC)NC(CC(C=C)C)=O)nn(C)c(=O)c2ccccc12 77733,c1(CNC(=O)CCC2CC2)csc(CNC(C2C(C(=O)CSC3CC3)C2)=O)n1.CN 77734,N1(CCC#C)CCC(C(=O)NC2CCCC(CNC(=O)C(COC)CC)C2)CC1 77735,CCC(C(=O)NCCCC1CCCN1C(=O)C(c1ccc(C)o1)C)N(C)C 77736,c1(NS(C)(=O)=O)ccc(C(N2CCCC2CNC(=O)C2=CCC2)=O)cc1 77737,c1(-n2cc(CN3CCC(COC)(CO)C3)nn2)cc(Br)cc(F)c1O 77738,CC1CN(C(c2c(Cl)ncn2C)C(=O)NCC2CCOC2)CCN(C)C1 77739,NC(=O)CCC(=O)NC1CCCC1NC(c1ccc(Br)o1)=O 77740,C1(C(=O)NC2(CSC)CCC2)CCCCN1C(=O)Cn1cccc1 77741,C12SC3C=CC1CC3CN(C(=O)OC(C)(C)C)CC(F)CCCOC2=O 77742,C1(CNC(C2CCN(CCC#C)CC2)=O)CC2CCC1N(C(=O)C(C)C1CC1)C2 77743,N1(C(CCCCCNC(c2n[nH]c(CC)c2C)=O)=O)Cc2ccncc2C1 77744,c1(NC(C(N2CCC3(C=CCO3)C2)C)=O)nc2ccc(F)cc2s1 77745,N#Cc1ccncc1N1CCN(C(=O)CCc2nncs2)CC1 77746,c1(C(=O)NC2C(C)CCN(C(c3scc(C)c3Cl)=O)C2)cnc(O)c([N+](=O)[O-])c1 77747,c1(-n2cc(C(=O)NC(C3CN(C(=O)Cn4cncn4)C3)C)nn2)ccccc1Br 77748,c1(C(N2CC(NC(c3cn(C)c(=O)n3C)=O)C2)=O)ccccc1S(C)=O 77749,C(=O)(CCCCC(F)(F)F)N1CC(N(C(COC(CC)(C)C)=O)C)C2(C1)CC2 77750,C1(C(N(CC(C)(CO)CO)C)=O)CCN(C(=O)C2CCCS2)O1 77751,C#Cc1cncc(CNC(c2ncc(OC)cc2F)=O)c1 77752,C(c1cscn1)=CC(=O)NC1CC1CNC(c1coc(C2CCC2)n1)=O 77753,C(=O)(C1=CCN(C(=O)CN2C(=O)CCCC2=O)CC1)Nc1c(CC)cccn1 77754,N1(C(Cc2ccc(OC)c(O)c2)=O)CC2CCC(NC(=O)CC3CC3)CC2C1 77755,C1(C)(CC(N2CC(C)C2(C)C)=O)CCN(C(=O)CC2CCCC(C)O2)CC1 77756,c1(C(=O)NCCC2CCCN2C(=O)CCC=CBr)cnc2c(c1)CCOC2 77757,CC(C(=O)NC1(CNC(c2cn(CC(N)=O)nn2)=O)CCOCC1)S(N)(=O)=O 77758,C1(C)(C(N(CC(C)(C)NC(C2C(C(=O)OC)CC2)=O)C)=O)CCOC1 77759,CC1CN(C(=O)CCOCCN(C(=O)C(c2ccn(C)n2)C)C)CC1C 77760,c1(C(c2nnnn2C2CCCC2)NC2(C)CCCC2)cc2ccccc2nc1O 77761,c1(C(=O)NCCn2cc(C(CC)N(C)C)nn2)cc(C)c2nc(C)nn2c1 77762,c1(C(=O)NC2(CCNC(C(COC)OC)=O)CCC2)cn2cnnc2cn1 77763,Cc1cc(=NC(=O)C(=O)NC2CC3CN(C(=O)CCc4ncc[nH]4)CC3C2)[nH]o1 77764,Cc1cc(=NCc2nc3ncccc3o2)[nH]c(N(C)Cc2ccc(Br)cc2C)n1 77765,C(C)(CC(=O)O)(c1n(C(C)C)nnn1)NCC1(c2cnn(C)c2)CCCO1 77766,C#Cc1ccccc1CC(=O)NCCN(CCc1ncc(C(F)F)cn1)C1CC1 77767,Cc1ccc2c(c1)C(C(=O)N1CCN(C(c3cc(=O)cc[nH]3)=O)CC1CCO)C2 77768,c1(NC(C2CSCCN2Cc2ncc(Cl)cc2Cl)=O)ncc(Br)cc1I 77769,N1(C(CC2CC(C)C2)=O)CCC(C(C)C)CC1CNC(=O)Cn1cccnc1=O 77770,N1(C(c2cn(C)nn2)=O)CCN(C(=O)C=CC2CC2)C(c2ccnn2C)C1 77771,N(C1CC2(CCCC2)c2ccccc21)C(C(CC)NC)=O 77772,c1(C(=O)NCCC2(CNC(C3(C#N)CCCO3)=O)CC2)cnn2c1CC(F)(F)C2 77773,c1(CC2CC2)nc(N(C)CCN(C(=O)C(F)C2CCC2)C)c2ccsc2n1 77774,C1(CNC(C2ON=C(C)C2)=O)(CNC(c2[nH]ccc2C2CC2)=O)CCCCC1 77775,C1(C(N(C2(C)CCCC2)C)=O)CN(C(C2CC(C3CC3)C2)=O)CCO1 77776,C1(NC(c2cc(F)c(OC)c(F)c2N)=O)C(C#N)CCC12CCOCC2 77777,n1(CCOC)nc(C(=O)NC(CNC(=O)CC2(O)CCCC2)C2CC2)ccc1=O 77778,N1(C(CCCC)=O)CC2(CCCC2)C1C(N1CCC2C(C(N)=O)C2C1)=O 77779,C(C(C)(C)CCNC(c1csc(CC(C)C)n1)=O)NC(Cc1c(C)ncs1)=O 77780,c1(OCC)cccc(CC(=O)NCCCC(C)NC(c2c[nH]ccc2=O)=O)n1 77781,C1(CNC(C(C)NC(COC)=O)=O)CC2CCC1N(C(C1CC=C(C)CC1)=O)C2 77782,N12CCCC(C3CN(C3)C(=O)C3(CC3)C1=O)C2.C1(COC(C)C)C2CCCCC12 77783,c1(CC(=O)NCC(CC)N(C(c2c(CC)c[nH]n2)=O)C)cncc(C)c1 77784,CCCC(C)C(=O)NCc1cc(C(=O)NCC2(CO)CC2)ccn1 77785,C12(CC(=O)N(C)CC3(C)CC3)CCC1CN(C(C1(C3CC3)CC(=O)C1)=O)C2 77786,CC(C)C(C(=O)NCCn1cc(C2(O)CCOC2)nn1)n1cc(Br)cn1 77787,C(C(CNC(c1n[nH]c2c1CCC2)=O)S(C)(=O)=O)NC(C1OCC(C)(C)C1)=O 77788,N1(C(C(c2cn(C)nc2)=O)=O)CCC2(NC(=O)CC(F)(F)C(F)F)CCCCC12 77789,N1(C(c2cc(CNC(c3c(C)ccnc3O)=O)no2)=O)CCC(C2CCOC2)C1 77790,C12(C(N3C(C(C)NC(=O)C(C)(C)O)CCC3)=O)CCOC(C)(C1)C2 77791,c1(C(N2CCC(NC(C3N(C)CCC3)=O)(CF)C2)=O)cc(Cl)cc(Cl)c1F 77792,C(=O)(C(O)CC(F)F)N1CCCC(N(C(c2ccccc2)=O)CCO)C1 77793,c1(-c2nc(C(CC)O)nn2-c2ccc(Cl)cc2)ccc2ncccc2c1 77794,C1(C)(CNC(C(CCC)C)=O)CCCN(C(=O)C(CC)N2CCCC2=O)C1 77795,c1(CC(=O)N(C2CC(CCNC(CN(C)CS(CC)(=O)=O)=O)C2)C)nnc(C)s1 77796,c1(C(=O)NCCC2(NC(C34COCC3C4)=O)CC2)nccn2ccnc12 77797,n1(CC)ncc2c(C(=O)NCC3(CNC(=O)CO)CCC3)cc(SC3CC3)nc12 77798,c1(C(C)=O)cn(C)nc1C(=O)NC(c1ccc(C)cc1)CNC(c1cnsc1)=O 77799,Cc1ccc(CC(=O)NC2C=CCN(C(=O)CCOC3COC3)C2)c(F)c1 77800,N1(C(c2c(C)nc(OC)s2)=O)CC(C(=O)NC2CCC2(C)C)OC(C)C1 77801,CC(C)(F)C(C)(F)C(=O)NCC1(O)CC(CNC(c2cc(O)nc(Cl)c2)=O)C1 77802,c1(CCC)n[nH]cc1C(=O)NC(COC)C(=O)NC(C)CO 77803,n1(CC)c(C2CCCN(C(C3C4CC3(c3ccco3)CO4)=O)C2)nc2ccccc12 77804,c1(CC2C(OC)CN(C(c3cnncc3N)=O)C2)ccc(C)c(F)c1 77805,c1(CNC(CCC2CCC(NC(C3CCC(CC)O3)=O)C2)=O)cc(C)nc(O)c1 77806,N1(C(C(C)(C)C2CCCC2)=O)CCC(C)(CC(=O)N(CCCO)C2CCC2)C1 77807,c1(C(=O)NC2CN(C(CC(C)F)=O)CC2(C)C)c2ccccc2nn1C 77808,c1(C(=O)NCC2(S(N)(=O)=O)CC2)c[nH]c2ccc(C3=CCOC3)cc12 77809,N1(C(C(C(C)SC)O)=O)CCC(C)(CNC(=O)CCN(C2CCCCC2)C)CC1 77810,c1(C(C(=O)NCCOCC)N(C)CCC2CCCCC2)c(Br)cnn1C 77811,Cc1cc(C)n(C(C)CC(=O)NC2C=CCN(C(=O)CSc3cn[nH]c3)C2)n1 77812,Cn1nc([N+](=O)[O-])cc1C(=O)NCC1CN(C(C2CCS(=O)(=O)CC2)=O)C2CC12 77813,C1(N(C(=O)CCn2cc(C3CCCCO3)nn2)C)CNC(=O)C12CC2 77814,S(=O)(=O)(c1ccc(F)c(C(F)(F)F)c1)N1CCC(O)(C(=O)NCc2cc[nH]n2)C1 77815,c1(CC(=O)OC)cccc(C(=O)NCCCNC(=O)C(c2ccc(Cl)s2)C)c1 77816,C(=O)(CC(CC(C)C)NC(=O)C(F)(F)CCCC)NCC(CC#C)(C)C 77817,Cc1cc(C)n(CCNC(=O)C(CC2CC2)NC(=O)COc2cnn(C)c2)n1 77818,c1(C(N2CCCN(C(C(C=C=C)C)=O)CC2)=O)cc(OC)c(OC)cc1F 77819,Cc1cnc(C(N2CCC(C)(CNC(c3cncc(N)n3)=O)C2)=O)cn1 77820,N1(C(C(=O)NC(C)C)=O)CC2CCN(C(c3ccn4nccc4c3)=O)CC2C1 77821,N1(C(c2c(SCC)cccn2)=O)CCCC(C2CCN(C(=O)CCOC)CC2)C1 77822,c1(NC(=O)NC2CN(C(=O)OC(C)(C)C)C2)conc1C1CC1 77823,C1(CNC(c2c(SC)snn2)=O)CC2(CO1)CN(C(C1CC=CC1)=O)C2 77824,N1(c2c(C(C)=O)c(C(F)(F)F)ncn2)CCCC1C1CCCCN1NC(=O)C(C)C 77825,C1(CC(=O)NC(C)CCN(C(=O)COCC2CC2)C)CCC12CCC2 77826,Cc1ncnc(C)c1OCC(=O)NC1CCC(NC(C2CS(=O)(=O)CCO2)=O)C1 77827,N1(C(CC2C(C)CCO2)=O)CCCC(C)(C)C1C(N1CCC2(CC1)N=N2)=O 77828,O=C1NC(C2CCOC2)C(=O)N1CC1CC2CCC1CC2 77829,c1(OC)oc(C)nc1C(=O)NC(C)CC(C)NC(c1c[nH]nc1C(C)(C)C)=O 77830,CCC(C)(C#N)C(=O)N(C)CC=CC(N1CCC(C)CC1C)=O 77831,C1(C2CN(C(=O)Cc3ccc(C#N)s3)C2)(NC(C2(c3ccn(C)n3)CC2)=O)CC1 77832,Cn1cc(Cl)c(C(=O)NCc2ccc(CC(C)NC(C34CC(F)C3C4)=O)cc2)n1 77833,C1(CC(=O)NCC2C(CNC(C(C)CC3CCC3)=O)C2(F)F)CC(O)C12CCC2 77834,C1(CNC(C(=O)NCc2nccc(-c3ccccc3)n2)=O)CNCCC1(F)F 77835,Cc1ccc(CNc2cn(C3CC4(C(N5CCCNCC5)=O)C3C4)nn2)nc1 77836,N1(C(c2c(OC)csc2)=O)CCC(CO)(CNC(c2cncnc2C2CC2)=O)C1 77837,Cc1[nH]c(-c2ccco2)nc(=O)c1C(=O)NCCN(C(=O)CCCF)C1CC1 77838,c1(C(=O)NC2CCN(C(c3ccc(OC)nc3F)=O)C2)c[nH]c2nc(F)ccc12 77839,C(=O)(CCCC(C)CC)N1C(C)CC(CC(N2CC(C(=O)OC)C2)=O)C1 77840,N(C(=NCCCCC)N1CCc2c(cc(F)c(F)c2F)C1)C(C#C)CCCOC 77841,CCCCC(C(=O)NC)NC(=O)C=CC(C)(C)NC(c1cn(C)cc1C)=O 77842,N1(C(CCN(CCC)C)=O)CCCC12CCN(C(=O)CC(=O)N(C)C)CC2 77843,n1(CC)nc(C)c(C(=O)Nc2c(N(C(COC(=N)O)C)C)ncnc2Cl)c1C 77844,c1(C(=O)OCC)cn(C)nc1C(N1CC(NC(=O)CN2CCC2C)C(F)C1)=O 77845,CCC(C)(C)CC(=O)NC(C)CC1CN(C(c2ccc(F)c(CC=C(C)C)c2)=O)C1 77846,c1(CC(=O)NCC(C2CC2)NC(=O)CCn2ccnc2)ccc(Cl)nc1F 77847,c1(C(=O)NCC(C)N(C(=O)C(C)CC(F)F)CC)ccnc2[nH]c(C)nc12 77848,Cc1cc(C(=O)NCC(CNC(=O)CC#N)CO)n(C(C)(C)C)n1 77849,n1(CC)ccnc1C(C(=O)NC(Cn1cncn1)C(=O)OC)N(CC(=O)OCC)C 77850,c1(C(=O)NCC2CCN(C(C3NC(=O)OCC3)=O)C2)csc2ccc(F)cc12 77851,c1(CN(C(=O)C(C)OCCC(C)C)CC(C)NC(CSC)C)ccccc1 77852,n1(CCC)ccnc1C(F)(F)C(=O)N(CC(C)NC(=O)CC(C)C1CCCC1)C 77853,CCC(C)CC(CO)Nc1ncc(CN(C)C)cc1Br 77854,C1(C(=O)NCC(CC)NC(c2ncc(C(F)F)s2)=O)COCC1(C)C 77855,CCCCC(O)C(=O)NCCC1CCCN(C(c2ccc(C)c(OC)c2)=O)CC1 77856,N1(C(C2CCC(=C)CC2)=O)C(C(=O)NCCCCc2cnc[nH]2)CCC12CC2 77857,CCS(=O)(=O)C=CC(=O)N1CCN(C(=O)Cc2cccc(C)c2)C(C)C1 77858,c1(C(=O)NCC2CN(C(c3cnn(CCC)c3C)=O)CC2C)cnc(C)c(N)c1 77859,c1(C(=O)OC)cccc(CNC(N2C(COc3ccc(SC)cc3)CCC2)=O)n1 77860,N1(C(=O)OC(C)(C)C)CCC2CC1CN(NC(c1ccnn1-c1ccccc1)=O)C2 77861,c1(-c2onc(CNC(=O)NC3CCCC=C3Br)n2)cccc(F)c1 77862,N1(C(C(c2cscn2)N(C)C)=O)CCN(C(c2cnn(C3CC3)c2)=O)CC(O)C1 77863,C1(CNC(C(C)n2ccnc2)=O)C2CN(C(=O)CCOCC3CCC3)CC12 77864,n1(CCC(N2CCC(N(C(C(CC)N(C)C)=O)C)C2)=O)ccc2cc(C)ccc12 77865,CC1CN(C(=O)CCC2(C)CC2)CC2(CCN(C(C3CCCN3C)=O)CC2)O1 77866,c1(C(N2C(C(C)NC(C(CC)c3ccccc3)=O)CCC2)=O)cc(C)nc(C)c1 77867,N1(C(c2c(C)nsc2)=O)CCCCC1CCCNC(C1CC1C)=O 77868,S(=O)(=O)(c1nc(C)cs1)NC(c1cccc(OC)c1)CO 77869,N1(C(CC=CC)=O)CCCC2CCN(C(C3CC4(CSC4)C3)=O)CC12 77870,N1(C(CCC2N(C(C3CCSCC3)=O)CCC2)=O)CC(CO)C2(CC2)C1 77871,N(C(=NCC(C)CO)NCc1ccnn1C)Cc1cc(C)no1 77872,C(CC(C(=O)NC1CC(=O)N(C)C1)NC(=O)C(CC1CCC1)OC)OC 77873,c1(C(C)C)c(C(=O)N(CC(C)NC(=O)CC2COC(=O)N2)C)cnc2ncnn12 77874,C1(NC(C2CCN(c3ncccn3)C2)=O)C=CCN(C(c2cnccc2Cl)=O)C1 77875,Cc1cc(C(=O)NCC2CCCC(NC(C3CC3F)=O)C2)cc(S(C)(=O)=O)c1F 77876,CC1(C)CC(C(=O)N2CC(C(C)(C)O)(CNC(C3(Cl)CC3(F)F)=O)C2)=NO1 77877,CCCC(CCC)C(=O)N1CCOCC1CCNC(=O)CSCCN(C)C 77878,CCC(C)C(O)CC(=O)NC1(CNC(=O)Cc2ccc(F)c(Cl)c2)CC1 77879,C1(c2n(CC=C)nnn2)(NC2CC3CCC(C2)O3)CC2(CCOCC2)C1 77880,C(C)(CCN=c1[nH]cnc2cc(C3CC3)nn12)NC(C1C(C)C1)=O 77881,c1(CC(=O)NCCCCn2cc(-c3ncn(C)c3)nn2)[nH]nc(C(F)(F)F)c1Br 77882,C(C(C)(C)C(=O)NCC1CC(CF)C1)NC(C1CCC(C)C1)=O 77883,N1(C(C(C2CCN(C(CC3C(C)OCC3)=O)CC2)C)=O)CC2CCC2(C)C1 77884,C(c1cscn1)=CC(=O)NCCSCC(=O)N(CC#C)Cc1ccco1 77885,Cc1[nH]c(=N)nc(O)c1CC(N1CCC(C)N(C(C2CCC2CF)=O)CC1)=O 77886,N1(C(C2(C)N(C(C3C(OC)(OC)CC3)=O)CC=C2)=O)CCC(C)(C(C)C)CC1 77887,N1(C(C2CC(OC)C2)=O)CC2CC(O)C1C2NC(c1cccnc1N)=O 77888,Cc1ncc(CC(=O)NC2CC(NC(=O)CSc3nnnn3C3CCCC3)C2)o1 77889,N1(C(C2(OCC)CCC2)=O)CC(C(=O)OCC(C)CC(C)C)CCC1(C)C 77890,c1(C(C)NC(=O)C(C)(C2CC2)N(C)C(c2cn(C)cn2)=O)cccc(O)c1 77891,c1(CNC(N(CCCC(C)C)C)=O)nnc2c(Cl)cccn12 77892,C1(n2cc(-c3cccc(C)c3)nn2)CON(C(=O)C2CC(n3ccnc3)CO2)C1 77893,c1(NC(=O)OCC)ncc(C(C(=O)NC2CC2)N(C)CCCC(=O)NC)s1 77894,C(=O)(N1CCC(CC(C)(C)C)O1)C1N(C(C2C(OC(C)=O)C2)=O)CCC1 77895,C1(N(C(=O)CNC(=O)C2CC2)C)CC12CCN(C(C1(n3ccnc3)CCCC1)=O)C2 77896,c1(C(=O)NCC(C)N(C(C2CC3CC3C2)=O)CC)ccc(Cl)c2c1OCCO2 77897,CC(CCC(F)(F)F)NC(C1C2CCC1(c1ccco1)C2)=O 77898,C1(NC(CCCSC)=O)(CO)CCN(C(=O)CC2CC(F)C2)CC1 77899,Cc1nc(O)sc1C(N1CCC(CN(C(=O)C=Cc2ccncc2)C)C1)=O 77900,N1(C(C2C(=C)C2)=O)CCC2(CCCN(C(=O)CC3(CO)CCCC3)C2)C1 77901,C1(CC(C(=O)NC(C)CC)N(C)CC2(OC)CCCC2)COC(C)(C)O1 77902,c1(OCCC)ccc(C(=O)NC2CN(C(=O)C(C)C(C)O)C2)c(OC(C)=O)c1 77903,C1(C(=O)Nc2cccc(CC)c2F)CC(C)(C)CCN1C(=O)C(C)c1cc[nH]n1 77904,c1(CC(=O)NCC2CC(NC(=O)Cc3cnc(C4CC4)[nH]3)C2)cncc(F)c1 77905,N1(C(Cc2cc(C)no2)=O)CC(NC(c2cc(=O)c(Br)c[nH]2)=O)CC12CCC2 77906,Cc1cc2c(cc1C)C(NC(=O)C(C1CCCCC1)O)CCS2 77907,c1(C(=O)NC(C2(O)CN(C(c3cc(F)ccc3N)=O)C2)C)ccc2occc2n1 77908,c1(CNCCC(C)CC(C)(C)C)cc2nc(Cl)ccc2s1 77909,N1(C(C2(CC=C)CCCN2C(C23CCCC2C3(F)F)=O)=O)CCC2(CC1)CSC2 77910,C(=O)(C(O)CCCNC(=O)CCc1cccnc1)NC(CCC)c1nn[nH]n1 77911,C=C=CC(C)C(=O)N1CCCC1C(C)(C)C(=O)Nc1cnc(N(C)C)nc1 77912,C1(C(=O)NC(C(C)C)CCN(C)C(c2cnnn2C)=O)OCCN(C)C1=O 77913,C1(CNC(c2csc(C)c2C)=O)CN(C(C2(O)CC2(C)C)=O)CC(C)(C)C1 77914,C1(NC(C2(C=C)CCC2)=O)CC(O)CN(C(c2ccc(OC)c(C)c2)=O)C1 77915,c1(C(=O)NCCCN(C(CNS(CCOCC)(=O)=O)=O)C)ccc(C)cc1CC 77916,C1(NC(C2CC=CCN2C(=O)Cn2cccnc2=O)=O)CC12CCCCC2 77917,c1(C(=O)NC(CCCNC(COC(CC)C)=O)C)nccc(Br)c1O 77918,c1(OC)cc(C(N2CCCC(C(C)(O)CNC(=O)C=CCO)C2)=O)c(N)c(C)c1 77919,c1(NC2CCN(C(=O)Sc3n(C)nnn3)C2)cccnc1O 77920,N1(C(c2n[nH]c(C)c2C)=O)CCC(C)(CNC(C2CC2C(=O)NCCO)=O)CC1 77921,N1(C(Cn2ncc(CC)c2)=O)CC=C(CNC(C2CCN(C(N)=O)CC2)=O)CC1 77922,C1(CNC(CCC)=O)CN(C(=O)C(O)C2=CCCCC2)C2CCCC2O1 77923,C(=O)(C(F)CC(C)(C)NC(=O)C(C)C1CC1)Nc1cccc(C#C)c1 77924,C1(CCC=C)(C(=O)NCc2cnn(C)c2)CN(C(C2CCO2)=O)C1 77925,Cc1[nH]c2ccccc2c1CCNC(=O)C(C)SCC1CCCO1 77926,c1(C(N2CCC(NC(C=COCC)=O)CC2C)=O)cccc2c1C(F)(F)CC2 77927,c1(C(N(C)CC2COC(C)(C)O2)=O)ccc(Cl)cc1N=[N+]=[N-] 77928,C1(C#N)(C(=O)NCc2c(C(N(CC(C)(C)CO)C3CC3)=O)n[nH]c2)CCCO1 77929,C=CCCCCC(=O)NC(C)CCCCNC(C1CCCN1c1cnccn1)=O 77930,NC1CC2(CC(CNC(C3(O)CCCNCC3)=O)C2)C1 77931,C1(C)(CNC(Cn2nnc(C(C)(C)C)n2)=O)CN(C(=O)CC2CC(F)C2)CC1C 77932,C(=O)(C1=C(Cl)CCC1)NCC1(F)CC(NC(=O)CCC(=O)c2ccc(O)cc2)C1 77933,Cc1cc(C(N2CC(CNC(C3COC3)=O)CC2C)=O)c2nc(C)n(C)c2n1 77934,CCC(C)(O)C(=O)NC(CNC(=O)CCc1ccc(Br)cc1)C1CCC1 77935,c1(COC)ccsc1C(N1CCC(NC(c2ccc(C(C)(C)C)[nH]2)=O)C1)=O 77936,c1(OC)c(NC(=O)C(F)C2CC(NC(C3CC4(CC4)CO3)=O)C2)cccc1F 77937,c1(NC(C2C(C)(C(=O)OCC)C2)=O)ccc(Br)cc1Br 77938,C(=O)(CC(C)CC(=O)NCC1(NC(c2ccc(Br)cc2C)=O)CCOC1)OC 77939,c1(C(=O)NCC23OCC(NC(CC(C(C)C)O)=O)(C2)C3)cc(Cl)c(F)cc1F 77940,CC1CC(C)(C)CN1C(=O)COC1(C)CN(C(=O)C=Cc2cc[nH]n2)C1 77941,c1(CC(=O)NCCC2CCC(NC(CC(C=C)C)=O)C2)cn2cccc(C)c2n1 77942,Cc1noc(C)c1CCNC(C1CCCC1CNC(c1cnn(C)c1N)=O)=O 77943,C(=O)(CCC(F)(F)C(F)(F)F)NCC1CN(C(c2c(C)cc(O)nn2)=O)C1 77944,N1(C(c2cc(SC)oc2)=O)CC(C2CCN(C(C3CCOC(C)(C)C3)=O)CC2)C1 77945,C(CC(=O)CCN(CC)CC)NC.C(C(=O)NC(C)COC)NC 77946,C1(C(NOC(C)(C)CO)=O)CC1C1CN(C(C2CCCCCC2)=O)C1 77947,CC(CC(=O)NCCCC1CCCN1C(=O)CCN1CCCC1)P(C)(C)=O 77948,C(CC(C)CCCC(C)C)NC(c1n(CCCC)nnn1)c1ccnn1CC 77949,c1(C(=O)NC2CCC(C(N3C(C#C)CC3)=O)C2)ccc(F)cc1F 77950,N1(C(c2ncc(OC(C)C)nc2)=O)CCC2(NC(c3c[nH]c(=N)o3)=O)CC2C1 77951,C(C(N=[N+]=[N-])C(=O)Nc1nc(OCC)ccc1Cl)OCC 77952,C#CCC(CC(=O)N(C)CC1(N(C)C)CCC1)NC(=O)CC(C)C(F)F 77953,C#CC1(CNC(=O)CC2CCC(NC(C3CC4(CCO3)CC4)=O)C2)CCOCC1 77954,c1(C(N2CC3C(CNC(CC4N(C)CCCC4)=O)C3C2)=O)cc(N)c(O)c(F)c1 77955,C1(NC(C2CCCC2)=O)CC2CCC1CN2C(c1cc(O)ncc1F)=O 77956,N1(C(COCC#C)=O)CCC(CO)(NC(c2coc(C(N)=O)c2)=O)C1 77957,C1(CCC)CCCN(C(=O)C#CCNC(C2CC(=O)N(C)C2)=O)CC1 77958,CS(=O)(=O)C1CC(C(=O)NCCCCNC(C2CCN(S(C)(=O)=O)C2)=O)C1 77959,C(=O)(C(C)(C)C(C)(F)F)NCC(C1(O)CN(C(C2(C)CCOC2)=O)C1)(C)C 77960,C1(C)(CC)CCCC1C(=O)NC(=O)C(N1CCC(NC2CC2)C1)C 77961,C1(C(C(=O)NCCC=C=C)C)CCN(C(=O)Cc2noc(C)n2)CC1 77962,c1(CC)nnc(CNC(C2C(NC(=O)C(COC)OC)COC2)=O)o1 77963,C1(C(N2CCN(C(CSCCCC)=O)CC2CF)=O)COC2CCCCC12 77964,c1(C(N(CCOCC#C)C)=O)coc(CNC(C2CCC(=O)C2)=O)n1 77965,c1(C(=O)NC2(CC)CCCC2)ncnc2c1ncn2CC(=O)N1CC(C)CO1 77966,c1(C(N2CCC(N(C(C3COC(=O)O3)=O)CCO)CC2)=O)cc2cc(Cl)cnc2o1 77967,CN1CCC2(CCN(CC3CC(N)C3)C2)C1=O 77968,C1(NC(C(C)n2ccnn2)=O)CC(CNC(C2(C3CC3)CC2)=O)C1(C)C 77969,N1(C(c2ccncc2)=O)CCC(CCN2CCN(C(c3cnsn3)=O)CC2)CC1 77970,c1(C(N(C2CCN(C(=O)CCc3ccc(C)s3)C2)CC#C)=O)nc(CC)oc1C 77971,Cc1cc(N)cnc1C(=O)NCC1CCN(C(C2CCC3CC3C2)=O)C1(C)C 77972,C(=O)(CC(CC)C(C)(C)C)NC(c1cccnc1)C(=O)N(C)CC1CC(=C)C1 77973,C(=O)(C(C)(C)C(=O)NCCCCCCNC(C1CCN(C)S1(=O)=O)=O)OC 77974,N1(C(c2c(OC)nccc2)=O)CC(NC(=O)CCc2ccn(C)n2)CC12CCC2 77975,C(C)(CN=c1[nH]c(N2C3CCC2CC(CC(F)(F)F)C3)nc(=N)[nH]1)OCC=C 77976,c1(CC)nc(C)cc(=NC(CNC(=O)C(F)C(C)C)C2CC2c2ccccc2)[nH]1 77977,C1(CCCNC(Cc2cc(C)no2)=O)CCCCN1C(c1c[nH]nc1C)=O 77978,Cc1cc(F)cnc1-c1cn(CCCN(C)Cc2nc(CC(=O)OC)sc2)nn1 77979,C1(CCC(N2CCC(CCC(=O)NC(C)(C)C)C2C)=O)(CC)CCC(=O)N1 77980,c1(C(N(C)C)=O)cccc(CN2CCCCC2CNC(=O)CC2CC(=O)N2)c1 77981,c1(CC(C)C(=O)N(C)CCOCCNC(C2CCC(=O)N2)=O)cccc(F)c1 77982,C1(F)(CNC(C(CC)F)=O)CCN(C(=O)CCCc2csc(C)n2)C1 77983,N1(C(C(C)(C)NS(C)(=O)=O)=O)CCCCC(CC(=O)O)C1 77984,c1(NC2C(CC)C2)ncccc1S(=O)(=O)NCc1nc2ncccn2n1 77985,C(CCCC(C)(C)NC(=O)C(C)NS(C)(=O)=O)NC(CC1CC(OC)C1)=O 77986,c1(C(=O)OC)ccc(NC2CC(F)CN(Cc3ccc(Br)o3)C2)c([N+](=O)[O-])c1 77987,c1(C(N(C(CNC(C(CC=C)C)=O)C)C)=O)c[nH]c2cccc(Cl)c12 77988,CC1(C)CNCCC1N1CCN(Cc2cc(Cl)ncc2Cl)CC1 77989,c1(C(N2CC(C(C)NC(c3cc(CF)on3)=O)OCC2)=O)cc(Cl)c(O)c(Cl)c1 77990,C1(O)(CNC(CC(C)F)=O)CCCN(C(c2ccc(C(F)F)cc2F)=O)CC1 77991,CCC(CC)C(C)N=c1nc(N2CCC(CCCO)C2)c2[nH]ccc2[nH]1 77992,CC1CN(C(=O)C(C)N(C)C(C2CC(=O)OC2(C)C)=O)C(C)C1C 77993,N1(C(=O)OC(C)(C)C)CC2CC2(C(=O)NC2CCN(Cc3cccnc3)CC2)C1 77994,c1(C(N2C3C(NC(=O)C=CC4CCC4)CC(C3)C2)=O)ccc2ccncc2n1 77995,c1(N2CCN(C(=O)Nc3cc(C)ncc3Cl)CC2)cccc2nsnc12 77996,C=Cc1cncc(C(=O)NC2(CO)CCCN(C(=O)CN(C)C)C2)c1 77997,N1(C(C2C(CC)CCC2)=O)CC2C(CNC(C3CCC(=O)N3C)=O)C2C1 77998,N1(C(C2CCN(CC)C2)=O)CCOC(CCCNC(=O)CSC2CC2)C1 77999,N1(C(CCc2c(C)noc2Cl)=O)CCC2(CCN(C(=O)CCn3ccnc3)C2)C1 78000,N1(C(c2c(C)ncnc2)=O)CC2CCC(C1)C2NC(C1(C)CC2CCC(C1)S2)=O 78001,c1(NC(c2n(CCC)nnn2)(C)CCOC)ccc2c(c1)OC(F)(F)O2 78002,c1(CC#N)cccc(C(=O)NC2CC(C(=O)NCC3NC(=O)NC3=O)C2)c1 78003,N1(C(c2cc(C)on2)=O)CCCC(O)(CN(C)C(c2ccc(C(C)C)nc2)=O)C1 78004,C(=O)(C(C(=O)c1ccccc1)NC(=O)OC(C)(C)C)OC1(CCCC)CC1 78005,C(=O)(C1=CC2C=CC1C2)NC(C1CCCN1C(c1cc2ccccn2n1)=O)C 78006,c1(OCC(=O)NCCN(C(c2[nH]c(C)cc2C)=O)CC)ccc(Cl)nc1 78007,C(=O)(CC(O)CC(C)C)NC(C(=O)NC(CC(=O)OC)C)COC(C)C 78008,c1(C(N(CC(C)C)CCC)=O)cccc(CNC(=O)CSCC(=O)OC)n1 78009,CCC(C)C(O)C(C)C(=O)NCCCCCC(=O)NCC(F)(F)Cl 78010,CCC(CC(F)(F)F)NC(=O)CC(C)N(C(=O)Cc1cncnc1)C 78011,c1(CC(=O)NC(C)CNC(=O)CC2CCCC2)cccc(F)c1O 78012,C(=O)(C(C)CC(C)CC)N1CCC(OCC(=O)NCC(=C)CC)C1 78013,CC1CC2(CCN(C(=O)C(N3CCCC(c4nccs4)C3)=O)C2)CO1 78014,Cc1cc(O)c(Cl)cc1C(=O)NCCCCNC(=O)C(C)CC1CCC1 78015,N1(C(C2CCCN2C(C2CC2Cl)=O)=O)CCc2nnnn2CC1 78016,C1(CNC(C23OC(C)C(CC2)C3)=O)CC2(CO1)CN(C(C1CC(O)C1)=O)C2 78017,C#CC1CCN1C(C1CC(N(C(=O)CN(C)C(=O)OC)C)C1)=O 78018,c1(SC)sccc1C(N1CCCC1CNC(c1ncoc1C(F)(F)F)=O)=O 78019,c1(OC(C)C(=O)NCCN(C(=O)CC2(O)CCC2)C2CC2)ccc2c(c1)CCC2 78020,C1(C(C)C)CC(CNC(C2(CN)CCCO2)=O)CCO1 78021,c1(CC(N2CCCC(NC(C(CC)O)=O)C2)=O)ccc(Cl)c(Cl)c1 78022,C=C(C)C1CN(C(=O)CCNC(C2CC2(C)C(F)F)=O)CCO1 78023,N1(C(c2cccc(C(C)C)c2N)=O)CCC2(CC(NC(C3CC3(C)C)=O)C2)C1 78024,CCCCCC(CC)C(=O)NCC1CN(C(C23CC(C2)C3)=O)CCCO1 78025,c1(C(C(=O)NCC(=C)C)N(CCCCO)C)ccn(-c2cnn(C)c2)c1 78026,Cc1n[nH]cc1C(=O)NC1(C(=O)NCC2(F)CCOC2)CSC1 78027,N1(C(CN(C(=O)C(C)n2ccnc2)CC)=O)CCOC(C)C1C 78028,N1(C(CC=CC=C)=O)CCC(C=C)(C(=O)NCCC(C)CCC)CC1 78029,c1(C(=O)NC2C(NC(CNC(CC3(OC)CCC3)=O)=O)CC2)cc(C)c(C)cn1 78030,CC1CC2CN(C(=O)CCN3CCOCC3)CC2N1C(c1scnc1Cl)=O 78031,C1(CNC(C(=O)NC(CC)Cc2ccccc2)=O)CCC2(CC1)CC(N)C2 78032,CC1(C)CCC(NC(C2(c3ncco3)CC2)=O)C(CNC(c2ccoc2)=O)C1 78033,C1(CC)(CC)CC(O)CN1C(C1CC(CNC(c2c[nH]c(=NC)s2)=O)C1)=O 78034,N1(C(C2(SC)CN(C(=O)OC(C)(C)C)C2)=O)CCC(N=[N+]=[N-])C1 78035,C1(CC)CN(C(=O)C(CCOC)OC)CCN1C(c1ccc(O)c(Br)c1)=O 78036,C1(NC(C(CO)NC(C(CCC)NC(N)=O)=O)=O)CCCC(O)CC1 78037,C1(C(C)C)CCC(C(=O)NC2COCC2NC(=O)CC2COCCO2)CC1 78038,C1(C(N2C3CN(C(c4c(C)ocn4)=O)CC2CC3)=O)C(C)(C)CCCC1(C)C 78039,c1(C(=O)NC2C(CNC(c3cnc(O)s3)=O)CCC2)ccncc1Br 78040,c1(SC)cc(N2CC3(CCN3C(=O)CCc3cncc(C(F)(F)F)c3)C2)nc(C)n1 78041,S(=O)(=O)(c1cccc(=NCC2(C)CC3CC3C2)[nH]1)N(CCCCCO)C 78042,Cc1cc(Cl)ncc1CC(=O)NC(C1CCCCC1)CNC(=O)C1=COCC1 78043,N1(C(CC(C)SC)=O)CC2CC(C(N3CCC(CC4CC4)CC3)=O)CC2C1 78044,C1(N(c2c(Br)cnc(CCC)n2)C)Cc2ccccc2C1O 78045,N1(C(C=NOC)=O)CCN(c2ccccc2CNC(C2(N(C)C)CCC2)=O)CC1 78046,c1(C(N2CCC(CO)C(O)C2)=O)cccc2[nH]nc(C3=COCC3)c12 78047,C(=O)(C(C)(C)C1=CCN(C(=O)C2=CC3(CCOC3)C2)C1)N(C)CC1CCCS1 78048,C=CCC(CC=C)C(=O)NCC(CNC(=O)CCc1c(C)nc(O)nc1O)OC 78049,C#CC1C(C(=O)NCC2COCCN2C(=O)CNC(=O)OCC)C1(C)C 78050,c1(C(C)C)n[nH]c(=NC2CC23CC(NC(=O)C(C)(C)S(=O)(=O)C2CC2)C3)o1 78051,c1(NC(N2CC(C(CO)C(=O)NCc3ccncc3)C2)=O)cc(Br)ccc1CO 78052,C(=O)(C(CO)NC(=O)C(CC1CC1)NC(c1cc(C(C)=O)on1)=O)OC 78053,N1(C(C(C)CS(C)(=O)=O)=O)CCN(C(c2ccc3cnsc3c2)=O)CC12CCC2 78054,Cc1cc(C(=O)NCC=CCNC(c2cc(C)n(C)c2)=O)cnc1C(F)F 78055,C1(C(C)NC(c2cocn2)=O)CN(C(=O)Cc2cscc2Br)CCO1 78056,c1(C(N2CC3CN(C(COCCCCC)=O)C3CC2)=O)cnn2cc[nH]c(=O)c12 78057,c1(C(N2CC3(C(NC(c4cnc[nH]4)=O)CC3)C2)=O)noc2ncccc12 78058,Cc1cc(=NC(=O)C(=O)N(CC(N2CCCC2)C)CC)[nH]n1-c1ccc(Cl)cc1 78059,CS(=O)(=O)CCCCc1noc(C23CC(CN)(C2)C3)n1 78060,C1(CNC(c2snc(C)c2N)=O)C(C)CCCN1C(=O)CCC1CC1(F)F 78061,C1(C(=O)NCCC2CCCC2)CN(C(c2n[nH]c3c2COC3)=O)CC1C1CC1 78062,c1(C(=O)NC2C(CNC(CCn3ccc(C)n3)=O)CC2)ccccc1N(C)C 78063,N1(C(C=C(C)CNC(=O)CC2CCC(C)CO2)=O)CCC2=C(CCCC2)C1 78064,CC1(C)CCN(C(=O)C(F)C2CCC2)CC1NC(c1cc(C2CCC2)no1)=O 78065,C#CCCCC(C)C(=O)NCC(C)CN(C(=O)CNC(C1CCCCC1)=O)C 78066,c1(C(N2CC(C(=O)NC)OCC2)=O)c[nH]c2c(F)cc(OC)cc2c1=O 78067,C1(C(=O)NC(CNC(C2COC(=O)N2C)=O)CO)(CC)CNC(=O)C1 78068,c1(NCC2(C)CC=CCC2)cc(=NC2CCCc3sccc32)[nH]c(C(F)(F)F)n1 78069,C1(CNC(C(C)OCC)=O)(Cn2cc(C3(O)CCOC3)nn2)CC12CCC2 78070,C1(OC)CC(C)CN(C(C2CC(F)C2)=O)C1 78071,c1(C(C)C)c(C(c2nnnn2C)NCC(c2ccccc2)CO)cccc1F 78072,S(=O)(=O)(c1ccc(=NCc2cnn(C)c2Br)[nH]c1)NCc1ncc(C)cn1 78073,C(=O)(C1=NOC(C(C)(C)C)C1)NCCC1(O)CN(C(CP(C)(C)=O)=O)C1 78074,C1(NC(c2ccc(F)c(CO)c2)=O)CCS(=O)(=O)C12CN(C(C1C=CCC1)=O)C2 78075,N1(C(=O)OC(C)(C)C)CCC(O)C(C(N2CC3CC(C(F)(F)F)C3C2)=O)C1 78076,CC1CCC(NC(=O)CCCC2CCCC2)CN1C(=O)Cc1cc(F)ccc1O 78077,c1(C(CC(N2CCC3(CCNC3)C2)=O)Sc2ccccc2)ccc2[nH]ccc2c1 78078,N1(C(C2C3(CCC(C)(C)CC3)C2)=O)CCc2c(Br)ccc(C#N)c2C1 78079,C(C1=CCCOC1)N(C(=O)CC1CCC(NC(c2cnc(C3CC3)o2)=O)CC1)C 78080,N1(C(C2N(CC)CCC2)=O)CCC2CCCC12C(=O)NC(C)C(C)SC 78081,C(CCNC(=O)Cn1nnnc1C(C)C)(C(C)C)NC(CN(S(CC)(=O)=O)C)=O 78082,C(C)(C)(CC(F)C(=O)N1CC(OCCOC)C1)NC(c1c(CC)ocn1)=O 78083,N1(C(C2(SC)CC2)=O)CC2CCC1CN2C(C1(CO)CC1)=O 78084,c1(C(N2CC(CNC(C3(CC#C)CCC3)=O)C2)=O)nccc(C)c1N 78085,c1(OC(C)C(=O)NCCCCN(C(=O)CC2COC(=O)C2)C)cc(Cl)cc(Cl)c1 78086,n1(CCC(=O)NCC(=O)NCCC#C)cc(-c2ccnn2C(C)C)nn1 78087,CC(C)(F)CCC(=O)NCC1CCCC1C(N1CCC(CCO)CC1)=O 78088,c1(C(=O)NCC2(O)CCN(C(C(C=C)(C)CC)=O)C2)cnc2c(c1)CCCC2 78089,c1(C(=O)NC2C(C)CN(C(=O)CC3SC(=N)NC3=O)C2)nc2ccccc2[nH]1 78090,N1(C(C(C(C)C)CN)=O)CC2COC(=O)C2C1 78091,c1(C(=O)NCC(C)(C(C)C)NC(C2N(CC)CCC2)=O)ccc2ncnn2c1 78092,C1(C(=O)NC(c2cccnc2O)C)CC=CCC1NC(=O)CC1COCC1O 78093,c1(C(N(CC(C)N(C(C(C)OCCN(C)C)=O)C)C)=O)cccn1C 78094,C1(CC(=O)NC2(CNC(C3C(C)=C3)=O)CCC2)CCCNC(=O)C1 78095,n1(CC=C)cc(C(=O)N(CCC(=O)NC2(C(O)COC)CC2)CC)cn1 78096,C#CCC(C)(C)C(=O)NCc1ncccc1C(=O)Nc1ccc(C(C)C)cc1 78097,O=C(C1=Cc2ccc(Cl)cc2OC1)NCC(C1CC1)NC(c1cscn1)=O 78098,n1(CC(N2CCC(CCCC)C2)=O)ccc2ccc(F)cc12 78099,c1(C(=O)NC2C(NC(C(CCCC)(C)F)=O)COCC2)cc2ccc(Cl)cc2o1 78100,C(=O)(CCC(C)CC)N1CC(CCNC(C2CC(=C)C2)=O)OCC1 78101,N1(C(CSc2ccc(OC)cc2)=O)CCN(C(C2CCCC2C2CC2)=O)CC1C 78102,c1(C(N(CC(O)CN(C(=O)C(C)(C)O)C)C)=O)cnn(C)c1C(F)(F)F 78103,C(Cc1cccs1)(CC(=O)Nc1cnccc1C(C)=O)NC(C(=C)F)=O 78104,CCC(CCCC(=O)N1CC2(COC(C)C2)C1)NC(=O)C=CC(C)(C)C 78105,N1(C(C2C(=C)CC2)=O)CCC2CN(C(c3c(Cl)ccc(OC)c3N)=O)CCC2C1 78106,CC(C)(CC(=O)NC1(C2CCN(C(=O)C(F)CC3CC3)C2)CC1)C(F)F 78107,C1(O)(C(C)NC(=O)C=C2CCC2)CCC(C)CC1.C12CCN(C1)C2=O 78108,C1(CC)CCCC1(C)C(N1CC(NC(=O)CSc2ccccc2OC)C1)=O 78109,c1(CC)nc(=N)[nH]cc1C(N1CCC1CNC(=O)CC1CC1(C)C)=O 78110,C1(C(=O)NCc2cc(Br)cs2)CC12CCN(C(c1ccc(Br)cc1F)=O)C2 78111,C(C(C(=O)N1CC(OC(C)=O)C1)NC(C1C=C(C)CS1)=O)OC 78112,N#Cc1ccc(NC(c2ccnc(CNC(=O)CCCCCO)c2)=O)cc1C#N 78113,Cc1ncnc(C)c1C(N1CC2C(CNC(=O)Cc3cccc(F)c3O)C2C1)=O 78114,C1(C(=O)NC2CC3(CN(C(C(C)OCCC(C)C)=O)C3)C2)CC2(CCCCC2)C1 78115,c1(C(=O)NCC2OCC(CNC(CC3CC(=C)C3)=O)C2)ccc[n+]([O-])c1 78116,c1(C(=O)NCC(C2CC2)NC(=O)CN2CCCCCC2)cc2c(Cl)cncc2o1 78117,C(=O)(C1=CC2C=CC1C2)N1CC2C(CC(=O)NCC(O)C3(Cl)CC3)(CC2)C1 78118,N1(CCNC(Cc2c(C)nc[nH]2)=O)CCN(C(c2ccsc2)C)CC1 78119,Cc1cccc2c(C(=O)NC3CC4CCC(C3)N4C(=O)C=CC3CC3)csc12 78120,c1(OC)cc(=O)n(C)cc1C(=O)NCCOC1CN(C(=O)C2=CCCCC2C)C1 78121,N1(C(c2cc(C)on2)=O)CCC(NC(c2coc(Cl)c2)=O)C(O)C1 78122,C1(NC(N2CC(N(C(CC3N(CC)CCOC3)=O)C)C2)=O)CC2C=CCC(C1)C2 78123,N1(C(CCC)=O)CC=CC(C(N2CCC(OCCF)C2)=O)C1 78124,c1(C(=O)NC(C2(CNC(CC3CC(=C)C3)=O)CC2)C)sc2ccccc2c1Cl 78125,n1(CCC)ccnc1CNC(=O)NCCC(C)(O)C1(C)CC1 78126,c1(CN(C)C(c2ccccc2F)=O)ccccc1CNC(c1c[nH]nc1Cl)=O 78127,c1(C(=O)NCCC(C)N(C)C(C2C=CCC2)=O)c[nH]nc1-c1ccccc1 78128,n1(CCC#C)c(N2CCC(N3CCOC3=O)C2)nnc1-c1cccn1C 78129,c1(-n2ncc(C)c2)ccc(CNC(N2CCOC(C)(C3CC3)C2)=O)cc1F 78130,N#Cc1cnccc1CN1CC(NC(C2Cc3ccccc3O2)=O)C(F)(F)C1 78131,N1(C(C2CCC(COC)O2)=O)CCSCC1C(N1CCCOCC1)=O 78132,CC(C)CC(C)CNC(C1CCN(CCC2CCCC(C)C2)C1)=O 78133,C1(N(C(C=C(C)C(F)F)=O)C)CN(C(=O)C(CCN(C)C)N(C)C)CCC1O 78134,CCC(=O)CCC(=O)NC(C)CCCC(=O)NC1CCN(CC)C1 78135,N1(C(CC2C(C(=O)OC)C2)=O)CCC2CCN(C(C3CCCCCCC3)=O)CC12 78136,c1(C(N2C(CNC(C(C)Cc3ccccc3)=O)CCC2)=O)nc[nH]c2ncnc1-2 78137,O=C(CC1=CCOCC1)NC1(CNC(c2ccc(C(N)=O)cn2)=O)CCC1 78138,c1(C(=O)NC)ccc(NCC(O)CNC(C2COCCO2)=O)c([N+](=O)[O-])c1 78139,C1(CNC(C2(C(C)(C)OC)CC2)=O)CN(C(c2cc(C)c(C)o2)=O)CC1C 78140,Cc1noc(C(C)NC(=O)CCNC(=O)CNC(C2CC2C)=O)n1 78141,C1(C)(C(=O)OC)CCCN1C(C1(C)CN(C(c2cc(Br)ccn2)=O)C1)=O 78142,c1(C(N2CC(C(C)NC(=O)CC3CC(O)C3(C)C)C2)=O)cc(Cl)c(Cl)cc1O 78143,C1(C)(CNC(CCOC(C)=O)=O)CCN(C(=O)C=Cc2cnn(C)c2C)CC1 78144,Cc1ccc(C(=O)NC2CC2NC(C2COCC2(C)C)=O)c(N)c1F 78145,c1(C(N2C(CCNC(C3C(C=C)C3)=O)CCC2)=O)ccc2c(c1)CCN2C(C)=O 78146,c1(C(=O)NCC2(C(N)=O)CN(C(=O)CC3CCC(=O)C3)C2)ccc(O)cc1O 78147,N1(C(C)=O)CCC2(CC1)CC(NC(=O)C(C)CS(C)(=O)=O)C2 78148,c1(C(N2C(CNC(c3nccc(N)c3)=O)CCC2)=O)noc2ncccc12 78149,C(=O)(C1=Cc2ccccc2C1)N1CCC(CNC(C(CO)N(C)C)=O)C1 78150,C1(CC)CN(C(=O)C(N2CCCC2)C2CC2)CCC1NC(c1ccncc1)=O 78151,N1(C(CCC(=O)N(CC)CC)=O)CCC(NC(=O)C(C)(C)CO)C(C)(C)C1 78152,C1(CN)CN(C(=O)C(=O)Nc2cnn(C3CC3(F)F)c2)CC1(F)F 78153,C(=O)(C(C)CS(C)=O)NCC1(NC(Cc2ccc(CC(=O)NC)cc2)=O)CC1 78154,O=C(C1CCc2snnc21)N1CCCCC(CNC(C2(Cl)CC2)=O)C1 78155,C(C)(C)(CCCNC(=O)C(C)C1CC1)NC(CN(CC)Cc1cccc(Cl)c1)=O 78156,CC1CCCCC1(CNC(C1CCCSC1)=O)NC(=O)C1=CCCOC1 78157,c1(C(=O)NC(CC)CN(C(=O)C(C)(C)F)C)ncc(OC)cc1F 78158,N1(C(C=CC(CC)C)=O)CC(F)(F)CC1CCNC(c1ncccc1C)=O 78159,C#CCC(C)(C)C(=O)NC1C2CN(C(c3ccc(CC(C)C)nc3)=O)CC12 78160,Cc1ccncc1C(=O)NC1(CCNC(c2occc2C)=O)CC1 78161,C1(CNC(c2cnccn2)=O)CCCCCN1C(=O)CC1COCCO1 78162,C1(OC(c2ncc(OC(C)C)nc2)=O)CC(NC2CCS(=O)(=O)C2)C12CCOCC2 78163,C(=O)(C(C)(C)CN(C)C)NCc1c(C(=O)NCCN(C(C)C)C)occ1 78164,C(=O)(CCC(C)SC)N(C(CNC(C1(C=C)CCC1)=O)Cc1ccccc1)C 78165,N1(C(c2cnc(Cl)cn2)=O)CCC2CN(C(c3cccc4sccc34)=O)CC2C1 78166,c1(C(N2CCC(C#N)CC2)=O)cccc2c1CN(C(c1sccc1Br)=O)CC2 78167,N1(C(=O)C(Cl)=CCl)CC(NC(C2(c3cccnc3)CC2)=O)C(F)C1 78168,N1(C(c2cc(C)cc(Cl)c2)=O)CCCC(NC(=O)C(O)CCC(C)C)CCC1 78169,N1(C(CCC)=O)CCCC1C(=O)NC(CNC(=O)COc1ccccc1)C1CC1 78170,N1(C(C(N)=O)=O)CC23CCCCC2(C1)CN(C(c1cc2c(Cl)cccn2n1)=O)C3 78171,C12CN(CCO1)C(=O)NC2.C1(CN(C)C)CCCN(c2ccc(Cl)cc2)C1 78172,n1(CCC)nc(C)cc1C(=O)NC1CCCCC1NC(c1n[nH]c(C)c1C)=O 78173,C1(C(=O)NCCCNC(c2ccc(OC(F)F)cc2F)=O)C2CC3C(C2=O)C13 78174,Cn1ncc2c(NCC3CSC3)nc(N3CCOC(C4CCOC4)C3)nc12 78175,C1(C(=O)NCC(C2CC2)NC(C2CCCN(C)C2)=O)C(C)(C)OC1(C)C 78176,N1(C(CCCCC)=O)CCN(C(c2ccn(CCC(F)(F)F)n2)=O)C(C)C1C 78177,C#Cc1ccc(CCCC(N2CCC(O)C(NC(=O)CC(C)OC)C2)=O)cc1 78178,c1(C(=O)NC2CC(C)(CNC(=O)CC3CCCC(O)C3)C2)cc2ccccn2n1 78179,CCN=C(NCc1noc(C2CCC2)n1)NCC1COC1 78180,C1(C(=O)NCCCCOC(C)C)CCN(C(C2CC2(C)C(F)(F)F)=O)CC1 78181,C(=O)(C1=CC(C)CC1)NCCC(C)NC(c1c(C)occ1C(F)(F)F)=O 78182,C(=O)(C(F)C(C)C(F)(F)F)NC1(C)CN(C(CCOc2cccc(C)c2C)=O)C1 78183,C1(CNC(C2C(C)C(=O)C2)=O)CCCN(C(=O)C=CC(=O)N(C)C)C1 78184,C#Cc1ccc(Cl)c(C(=O)NC2CCCN(C(C3CCC(C(N)=O)C3)=O)C2C)c1 78185,C1(CN=C(NCCCP(C)(C)=O)NC2CCOCC2)CCC2(C1)OCCO2 78186,CN1CC(CC(=O)NOc2ccc(N)c(Cl)c2)CCC1C(F)(F)F 78187,N1(C(c2cnn(CCN(C)C)n2)=O)CCN(C(=O)CCN2CCC(F)C2)CC1 78188,C(=O)(C1=C(C)OCCS1)NC1C(OC)CN(C(=O)CN2CCC(C)(C)C2)C1 78189,C=CC(C)N=C(Nc1cccc(C(C)C)c1)N1CCC(OCCOCCOC)CC1 78190,C(=O)(CC1COCc2ccccc21)N1CC(F)(CNC(C2(C)ON=C(C)C2)=O)C1 78191,C12(C(=O)NC3C(NC(CCc4n(C)ncc4)=O)CCOC3)C3C4C1C1C2C3C41C 78192,C1(O)(CC(N2C(C(N(C)C)=O)COCC2)=O)CCCN(CC2OCCO2)C1 78193,N1(C(c2cnn(C3CCOCC3)c2)=O)CC2(C1)CN(C(C1(Cl)CC1)=O)CCO2 78194,c1(C(N2CCC(O)(CCNC(CC(C=C)C)=O)C2)=O)cc(F)c(C(F)F)cc1F 78195,C1(NC(c2ccc3n[nH]cc3c2)=O)C2CC3CN(C(c4coc(Cl)n4)=O)C1C3C2 78196,CCC(CC(=O)NC(CNC(c1csc(-c2ccc(Cl)cc2)c1)=O)CO)C(C)C 78197,c1(NCCOCCOCCOCCNC(C2CC2C2CC2)=O)nc(O)[nH]c(=O)n1 78198,c1(N(C2(CCO)CCC2)C)ncccc1S(=O)(=O)NCc1n(CC)ccn1 78199,C#Cc1cn(C)nc1C(=O)NCC1CN(C(C2CS(=O)(=O)C2)=O)C1 78200,CC1CC(C(=O)Nc2cc(C3CCCNC3)no2)C(C)O1 78201,C12(CC(=O)NCCC(CC)C)CCC1CN(C(c1cc(CO)on1)=O)C2 78202,N1(C(C2Cc3ccccc3C2)=O)CC2(CCCCN2C(C2CCCS2)=O)C1 78203,c1(OC)cccc(-n2nnc(C(=O)NCC(CO)NC(=O)C(C)C(C)O)c2C)c1 78204,N1(C(C(c2ccc(F)c(F)c2)(C)C)=O)CC2CCC(C1)N2C(=O)CNS(N)(=O)=O 78205,CCC(C)CCCCC(=O)N(CC(=O)NCCN1CC2CC2C1)CC 78206,c1(C(=O)NC2(C)CN(C(C3N(CC(C)C)CCC3)=O)C2)cc2ncccn2n1 78207,C(=O)(C(C(C)C1CC1)N1CCN(c2nccs2)CC1)NCCCOC 78208,N1(C(c2c(C)oc(Cl)n2)=O)C2CCC1C(CNC(c1ccc(Cl)cc1)=O)C2 78209,N1(C(c2c(C)scn2)=O)CC(NC(c2ccnc(N3CCCC3)c2)=O)CCC1C 78210,c1(CCNC(C(=O)N(C)Cc2cccc(Cl)c2)=O)nnc2c(=O)[nH]ccn12 78211,C(=O)(CC(CC1CC1)NC(c1c[nH]cc1C1CC1)=O)N1C(C(N)=O)CC1 78212,C1(NC(CN(CCCCCC)C)=O)(CNC(c2ccsc2Cl)=O)CCCCCC1 78213,C=CCC(CC=C)C(=O)NCc1cc(C(=O)NC2CCCCCC2C)co1 78214,C(=O)(C(C)(C)C1CCCCO1)OC(F)F.CC1CN(C)C(=O)CN1 78215,C(C)(C)(CCCCC(=O)NC1CC2CCC1C(NC(C1CCC(C)O1)=O)C2)OC 78216,c1(C(=O)OC)[nH]c(C)c(C(=O)N(C)CCN(C(=O)CCOCC2CC2)C)c1CO 78217,c1(C(=O)NCC2(F)CC(NC(c3ccc(N)cc3Cl)=O)C2)cnc2ccccn12 78218,c1(C(=O)CC2CCN(C(C3CCCC3)=O)C2)ccc(S(=O)(=O)NCC(=O)O)cc1 78219,C1(NC(=O)C(c2ccc(I)cc2)F)COc2ccccc2C1=O 78220,c1(CNC(CC2(C)CCCO2)=O)ccc(-c2cn(C3CC3)nn2)c(F)c1 78221,c1(C(=O)NC(CN(C(C2(C#C)CCOCC2)=O)C)C)ccc(C)c2c1CCC2 78222,C(=O)(CC(CNC(=O)Cc1cccnc1F)OC)NCc1cc(C(=O)OC)no1 78223,C1(CCNC(=O)Cc2ccccc2)CCCCN1C(C1CC=CCO1)=O 78224,c1(C(=O)NC2C(C(=O)O)CN(Cc3ccccc3)CC2)c(F)c(F)nc(F)c1F 78225,c1(CNC(C(=O)OC)Cc2ccc(F)cc2F)cc(S(C)(=O)=O)ccc1F 78226,c1(C(=O)NC2CN(C(CCC)=O)C3C2C3)c(C)nn(CC)c1C 78227,CCCCC(CC)C(=O)NC1CC(C(F)F)(NC(c2cccc(C)c2Cl)=O)C1 78228,Cc1cc(CCC(N2CCC(C(C)(C)NC(=O)C(F)=CC3CC3)C2)=O)no1 78229,N1(C(C2(CC#C)CCOC2)=O)CCC(CO)(CNC(C2C3CC(=O)CC23)=O)C1 78230,c1(C(N(C(C)C(=O)NCC(O)C2(Cl)CC2)C2CC2)=O)c[nH]nc1C(F)F 78231,c1(-c2c(C(CC)Nc3cncc(C(C)C)c3)cccc2)ccc(C#N)cc1 78232,c1(CNC(c2cccc(F)n2)c2n(CC(=C)C)nnn2)ccc(F)c(C)c1 78233,C(=O)(CCCCCC(C)(C)C)N(C(C)CNC(=O)CCCn1cncn1)C 78234,c1(C(C)NC(N2CCC3(C(C(=O)OC)C3)CC2)=O)cn(C)c2cc(Cl)ccc12 78235,c1(C(C(=O)N(C(C)CNC(=O)Cc2cc[nH]n2)CC)(C)C)cccc(OC)c1 78236,C1(NC(CN2CC(C)(C)C2)=O)CN(C(=O)CC2C=CCC2)CC1(C)C 78237,C#CC(CC(C)C)NC(=O)CCC1CCN(C(C2CCC(=O)NC2)=O)C1 78238,C12(C(N3C4CN(C(c5c(OC)ccs5)=O)C(C4)C3)=O)CCCN1CC(OC)C2 78239,c1(C(N2CC(C)(NC(C=CSC)=O)C2)=O)ccnc(S(N)(=O)=O)c1 78240,c1(OC)ccn2cc(C(=O)NCC3(C)CCN(C(C4CC4F)=O)C3)nc2c1 78241,c1(C(N2CCC(OC)(CNC(c3ccncn3)=O)C2)=O)cc(C)[nH]c(=NC)n1 78242,C1(OC)(CNC(c2nc(Cl)cs2)=O)CCN(C(C2CCC(C)C2)=O)CC1 78243,N1(C(C(C)(C)N=[N+]=[N-])=O)CCC(C(=O)NCC(F)C(C)(C)O)=C(F)C1 78244,N1(C(C(CC=CC)C)=O)CCC2C(C1)CN2C(c1cc(C)cc(OC)c1N)=O 78245,C1(C(=O)NC2(CNC(C34CC(F)C3C4)=O)CCCC2)CC2(CCCCC2)C1 78246,c1(OC(C(CC2CCCCCC2)NC(=O)OC(C)(C)C)=O)ccc(F)c(F)c1Br 78247,N1(C(CC(C)=C(C)C)=O)CCC(c2cn(CCC(=O)N(C)C)nn2)(N(C)C)C1 78248,c1(SCC=C)ccccc1C(=O)NCC1COCC1NC(=O)C(F)(F)C1CC1 78249,n1(CC(=O)NC(CN(C(c2c(CC)c[nH]c2)=O)C)CC)cccnc1=O 78250,C1(C(=O)NCC(CCOC)NC(c2nc(OC)c(C)s2)=O)CC(=O)NC(C)C1 78251,C1(CNC(C=Cc2cn(C)nn2)=O)CC2CCC1N(C(=O)CC1(O)CCCC1)C2 78252,C(CC(C)(C)COC)NCCOC.CCC1C(=O)N1 78253,N1(C(Cc2c(C(=O)OC)nccc2)=O)CCCC(C)C1C(=O)O 78254,c1(C(N2CCC(NC(c3c(C)ncnc3)=O)(CF)C2)=O)cc(C)c2[nH]cnc2c1 78255,c1(OC)ccc2c(c1)OC(C(=O)OC(=O)COC1CCCC(C)C1)C2 78256,C(=O)(CCCN=[N+]=[N-])NCC12CC(NC(C(C)NC(CC)=O)=O)(C1)C2 78257,N1(C(C(C)C2CCC2)=O)CC(CNC(c2c(C(F)F)cnn2C)=O)CC(C)(C)C1 78258,C(=O)(N=c1[nH]onc1-c1ccncc1)C1(Br)C(C)(C)C1C(=O)O 78259,c1(N2CC(CCOC)OCC2)[nH]c(=NCCCc2n[nH]c(=N)s2)nc2scnc12 78260,C1(C)(C(=O)NC(C(=O)NCc2c(C)cccc2)CCF)CC2CCC1C2 78261,Cc1c(Cl)ccc2c1CN(C(C1CC13CCC3)C(=O)NC1CCOC1)CC2 78262,c1(C(Cn2cccn2)NC(c2cnc(C(C)(F)F)s2)=O)ccc(Cl)cc1 78263,C1(CNC(CCC=C)=O)CCN(C(=O)CC2(SC3CCCC3)CCCC2)C1(C)C 78264,c1(-c2nc(CSC)nn2-c2cc(C(F)F)ccc2C)c(C)c2ccccc2n1C 78265,c1(CCC(N2CCCC(C)(c3cn(CC(=O)OC)nn3)C2)=O)cnc2cc[nH]c2c1 78266,c1(CN(C(C(=O)Nc2c(C)n(C3CCOC3)nc2)=O)C)cccc(Cl)c1Cl 78267,C1(C(=O)NCC2CC(NC(C3(NC(C)=O)CCC3)=O)C2)Cc2ccccc2C1C 78268,CC(CN(C(=O)C(C)N(C(c1ncccc1Cl)=O)C1CC1)C)C(F)(F)F 78269,c1(NC2C(F)CN(Cc3cccc(C(F)(F)F)n3)CC2)ncc2sccc2n1 78270,N1(C(c2cnc(C)[nH]2)C(=O)NC(C(=O)OC)C)CCC(CC(F)F)CC1 78271,C(=O)(N1CCCc2nncn21)C1CC(NC(CC2COCC(C)O2)=O)C(O)C1 78272,C#CCCC(C(=O)N(C)Cc1ccoc1)NC(=O)CCOCC(C)(C)C 78273,c1(OC)cccc(C(=O)NC2CCN(C(=O)CCc3c(C)c[nH]c3C)C2)c1 78274,C(=O)(CCC(=O)NC1(C(N2CCC(NC(N)=O)CC2)=O)CCCC1C)N(C)C 78275,CCCCCC(C)(C)C(=O)N1CCCC(C2(NC(c3cn(CC)nn3)=O)CC2)C1 78276,C1(CNC(CCC)=O)CCCCC1NC(=O)C=CCN1CCCC1 78277,N1(C(CCN(C)CCN)=O)CCC2(CC1)C(=O)Nc1cc(Br)ccc12 78278,c1(C(=O)NCC2(C)CCC(NC(c3cn[nH]c3)=O)C2)ccc(N)c(Cl)c1 78279,C(=O)(C#CC1(C)CC1)Nc1ccc(OC(C)C)nc1 78280,c1(OC)c(C(=O)N(C(C)CNC(=O)CNc2ncccn2)C)cccc1C(F)F 78281,N1(C(N)=O)CCC(C(N2CC(O)CC2CNC(C2CC2C(N)=O)=O)=O)CC1 78282,C1(NC(C2(CCCC)CC2)=O)CCN(C(=O)CN2CCC(C)C2)CC(C)(C)C1 78283,N1(C(C)C)CCN(C(c2cc(CNC(C34CCC(CC3)C4)=O)cs2)=O)CC1 78284,c1(NC(C2CC3(CC(NC(C4(Br)CC4)=O)C3)C2)=O)cccc([N+](=O)[O-])c1F 78285,c1(C(=O)NC(=O)NC(CNC(=O)CC2(CC3CC3)CCC2)C2CCC2)cc(O)cs1 78286,c1(C(=O)NC(C)CCN(C)C(C2CCCN(C)C2)=O)cccc(P(C)(C)=O)n1 78287,c1(OC)ccc(S(C)(=O)=O)cc1C(=O)NC1CN(C(c2cn[nH]c2)=O)CCC1F 78288,CCCC(C(=O)N1CCCC(CC(C)(C)NC(=O)CC2(O)CCC2)C1)OCC 78289,C1(NC(CN(C2CC2)CC)=O)CCN(C(c2cc(O)cs2)=O)CC1O 78290,N1(C(=O)OC)CCCC(C(N2CCCCC2c2ccccc2OC)=O)C1.C1CCC1 78291,C1(CCC(=O)NC)CCCCN1C(c1coc(C)c1)=O 78292,c1(C(=O)NCC(C2CC2)NC(C(C)NC(=O)C(C)(C)C)=O)cc2n(c1)CCC2 78293,Cc1c(C(=O)NC(CNC(c2cc(C3CC3)ncn2)=O)C2CC2)ccn1C(C)C 78294,CC12CCC(C(N3CCC3CNC(=O)CNC(C3CCS(=O)(=O)C3)=O)=O)(C1)OC2 78295,CC1(C)CC(CC(=O)NCc2ccoc2)N(C(c2cnn(C3CC3)c2)=O)C1 78296,N1(C(C(CC(=C)Cl)NC(C2CC3CC(=O)C2C3)=O)=O)CC2(C)CC1CCO2 78297,C(CO)(CCCCNC(=O)CN(C)CCO)NC(C(C)=C1CCC1)=O 78298,N1(C(C(C)OCC#C)=O)C2CCC1CC(CNC(c1oc(Br)cc1C)=O)C2 78299,c1(CC(=O)NC2CN(C(C3CCC3)=O)CC2C(F)(F)F)cccc(O)c1F 78300,N1(C(C(C=C)(C)C)=O)CCC2CN(C(=O)COc3cc(F)ccc3F)C2C1 78301,Cc1c(C(=O)NC2CC3(C2)CC3NC(=O)Cc2cccc(O)c2)sc2nccn12 78302,C1(CC)CCCC(NC(=O)CCN(C(=O)Cc2cccnc2C)C)C1 78303,C(C)(CC(C)CC)N(C(C1(CNC(c2c(CCC)nco2)=O)CCCO1)=O)CC 78304,C1(NC(CC2(COC)CCCC2)=O)CC(O)CN(C(C2(O)CCCCCC2)=O)C1 78305,c1(C(=O)NCCCCNC(C2(COC)COC2)=O)n[nH]nc1C 78306,C(=O)(C(C)CC(N)=O)NC(CC=C)CNC(c1cnoc1-c1cccs1)=O 78307,C(=O)(CCCC(C)(C)C)N1CCCN(C(C2N(CC)CCCC2)=O)CC1 78308,CCCC(CC(C)C)C(=O)NC1CCC(C(=O)NC2CC3CC(OC)C3C2)C1 78309,c1(SC)nc(-c2ccccc2)nc(=NC2CN(c3nccc(Br)n3)CC23CC3)[nH]1 78310,N#Cc1ccc(F)cc1C(N1CC2C(C1)N2C(C1CCC2(CC1)CC2)=O)=O 78311,C(=O)(CC(O)CNC(=O)C(c1ccccc1)O)N(CCC)CCC 78312,O=S(=O)(CCO)c1ccc(CNCC2CN(c3ncccn3)CCO2)cc1 78313,C1(C)(CNC(c2c(C)cc(SC)o2)=O)CCCN(C(C2CCC3(CC2)CC3)=O)C1 78314,S(=O)(=O)(CCC(=O)N1CCC12CN(C(C1(C)CCOC1)=O)C2)N(C)C 78315,c1(NC(C(CC2CCC2)NC(c2ccc(CC)o2)=O)=O)ccc(C)nc1O 78316,N1(C(C(CC#C)NC(c2ccn3cncc3c2)=O)=O)CC(=O)N(C)C(C)C1 78317,N1(C(C2CC(C)OC2C)=O)CCC(C2CC2)(CNC(=O)CSC(F)(F)F)C1 78318,c1(SCC)cc(C(N2CC=CC(NC(=O)C(C)N(C)C)C2)=O)ccn1 78319,Cc1ccc(-c2ccc(N3CCCC3=O)cc2)cc1NC(C1CC(C)OC(C)C1)C 78320,C12(CC13CCC3)C(=O)N(C1CC1)C2.CC(C(=O)c1ncc[nH]1)OCCN(C)C 78321,c1(C(=O)NCC2N(C(CCc3c(C)noc3C)=O)CCC2)c(Cl)ccc(Cl)c1N 78322,N1(C(C(Cc2ncn(C)c2)O)=O)CC2(CC(NC(C3(C)CC=CC3)=O)CO2)C1 78323,C(=O)(C1CCCc2nccn21)N(C1CCN(C(C(c2ccc(C)cc2)=O)=O)C1)C 78324,c1(COC)nnc(N2CCCC(C(C)(F)F)C2)n1CCC(=O)OC(C)(C)C 78325,Cc1ncc(C(=O)NC2CCC2NC(c2cnnc(O)c2)=O)cc1C#N 78326,c1(CC(C(=O)N(C2CN(C(C(CC)OCC)=O)C2)C)C)ccc(F)cc1 78327,CCCC(C)(CC)C(=O)NCCC1CCN(C(c2cn(CC)nn2)=O)CC1(F)F 78328,C1(C(=O)NC2(CNC(C(OC)OC)=O)CCCC2)CCn2ncnc2C1 78329,c1(NC(c2cc(Br)nn2C(C)C)c2n(CCCOC)nnn2)cc(Cl)cnc1C 78330,N1(C(c2c(N)cc(F)cc2)=O)CCC2(CCC(NC(c3cnc[nH]3)=O)C2)CC1 78331,c1(OC)cnnc(C(=O)N(CCN(C(=O)C(=O)Cc2ccc(O)cc2)C)CC)c1 78332,c1(C(N(C(C)(C)C)CC#C)=O)cc(C)c(C(c2ccccc2Cl)=O)o1 78333,C1(NC(CN(C)C)=O)CS(=O)(=O)CC1NC(c1ccc(N)c(F)c1)=O 78334,S(=O)(=O)(c1ccc(F)cc1)NCc1ccc(NC(C(C)O)=O)c(F)c1 78335,N1(C(C(C(C)C)NC(CC(=O)OCC)=O)=O)CC(=O)N(C)C(C)C1 78336,N1(C(CC2N(C(Cn3c(C)cc(C)n3)=O)CCCC2)=O)CCCC2(CC1)CC2 78337,n1(-c2c(C(N3CC(CO)OCCC3)c3cccs3)cccc2)nnc2ccccc12 78338,c1(CCC(=O)NCC(CNC(C(COC)(C)C)=O)CO)ccc2ncsc2c1 78339,CN1CC(CNC(C2(C)CCN(C(C3CC(=O)CCO3)=O)C2)=O)CC1=O 78340,C(=O)(C(C)(CC)CCCCC)N1CCC(C(C)NC(C(CC=C)(C)C)=O)C1 78341,CC1(NC(=O)NC(c2cccnc2)CCC2CC2)CCCC1O 78342,Cc1ccsc1C(=O)N(CCc1cn(C2CC2)nn1)Cc1ncoc1C1CCC1 78343,c1(OC)ccc(Br)nc1NC(c1ccc(NC(c2ccccc2SC)=O)cn1)=O 78344,C1(CNC(CCN(C(C)=O)C)=O)CN(C(=O)CN(C2CCCC2)C)CC12CCC2 78345,c1(C(C)C)noc(C(C)NC(=O)CC2CCN(C(C3CNC(=O)N3)=O)C2)n1 78346,c1(C(=O)NC(C2CCCN2C(=O)COC2(C)CCC2)C)ccc(F)cc1F 78347,C1(CCC)CN(C(=O)C(CCOC)OC)CC1C(=O)NCC(C)C(C)O 78348,C1(C2CCN(C(c3cc4c[nH]nc4s3)=O)CC2)(NC(CC(=O)OCC)=O)CC1 78349,c1(-c2c(N(C(C)C)C(=O)Nc3ccc(Cl)nc3)cnn2C)ccc(F)cc1F 78350,c1(CC)oncc1C(N1CCC(CNC(C2CC(C)(F)C2)=O)C1)=O 78351,c1(C(=O)NCC(C)CN(C)C(C2CC2(C)C)=O)cnc2cc(Br)ccn12 78352,C(=O)(C1CCCn2nccc21)NC(CCNC(C(F)=C(C)C)=O)C 78353,N1(C(c2[nH]cc(C(=O)OC)c2)=O)CC2(CCC2)CC1CNC(C1CNC(=O)N1)=O 78354,C12=CC(=NC(=O)N(C)C1)NN2C.C12(C(=O)OC)CCCC1(C(N)=O)C2 78355,N1(C(C2(CNC(=O)Cn3ccccc3=O)CC23CCC3)=O)Cc2c[nH]nc2C1 78356,CC1CS(=O)CCN1C(C1CN(C(C2CNC(=O)N2)=O)CCN1C)=O 78357,c1(C(=O)NC2CCC(NC(C3(CCC)CC3)=O)CC2)cc(F)c2c(c1)CCC2 78358,Cc1cn(CC(=O)NCCCCN(C(=O)C(C)C(F)(F)F)C)c2ccccc12 78359,C1(NC(c2n(CCC)ccc2)=O)CCOCC1C(N1CCC1(C)C)=O 78360,N1(C(C2OCCN(C)C2)=O)CC(C2CC2C(=O)NCCn2cnnc2)C1 78361,c1(C(=O)OC)cc(CCC(=O)N2CC(NC(c3cnc(CC(C)C)s3)=O)C2)c[nH]1 78362,N1(C(CC(C)C)=O)CCC2(CCC(NC(=O)C(N)=O)C2)C1 78363,c1(COC)nc(C(N2CCC(CN(C(=O)C=CCOC(C)(C)C)C)C2)=O)n[nH]1 78364,C(c1cnccc1C)=CC(=O)NC1CC(CNC(c2cncc(SC)c2)=O)C1 78365,CCC(CCC(=O)NCC(C(C)C)OC)NC(C1(C)CC1C)=O 78366,C(c1ccc([N+](=O)[O-])cc1)=C(C)C(=O)NCCN(C(=O)CCCC(N)=O)C(C)C 78367,Cc1cc(C#N)cnc1C(N1CC2(CC2)CC1CNC(C1(O)CCOCC1)=O)=O 78368,N1(C(C(C2CCN(C(c3cc(CO)[nH]n3)=O)CC2)C)=O)CC2(CCNC2=O)C1 78369,c1(NC(C)=O)ccc(C)nc1C(=O)NC(C)CNc1cccc(C)c1C 78370,c1(C(N2CCC(F)(C(=O)NCc3ccsc3)C2)=O)c(F)ccc(C(F)(F)F)c1F 78371,c1(C(=O)NC(CN2CCN(C(c3c(C)cns3)=O)CC2)C)cc(S(N)(=O)=O)co1 78372,N1(C(CC=C(C)C)=O)CC(O)(C2CCN(C(C3(C)CC(C(C)C)=NO3)=O)CC2)C1 78373,N(C(=NCC1CCCS1)NCc1cccnn1)C(C1CCCO1)C 78374,C1(CNC(CCC=CC(C)C)=O)C2CCC(C2)N1C(c1ccc(F)c(F)c1)=O 78375,N12CCC(CC1)C2.Cc1ncc(NC(=O)CCCn2cc(CN(C)C)nn2)[nH]1 78376,N1(C(c2[nH]cc(C)c2)=O)CCC2(CCN(C(=O)CC(C)NC(N)=O)C2)C1 78377,c1(CS(N)(=O)=O)cc(C(=O)N)n[nH]1.n1(C)cc(C2(C(N3CCC3CF)=O)CCC2)nn1 78378,C1(NC(C2(O)CC(C)(C)C2)=O)CN(C(C2CC23CCOC3)=O)C2CCCCC12 78379,C1(C#N)(C(N2C(COC)COCC2)=O)CC12CCC2 78380,CC(C)N(O)C(=O)C(=O)N1CC(C)(C)OCC1CNC(=O)C(C)n1ccnc1 78381,C1(NC(=O)CN2CC3CC3C2)CCCC(NC(C2CCC(F)(F)C2)=O)C1 78382,C1(NC(c2c(C)csc2)=O)CCN(C(=O)CCC2CCCC(=O)N2)C12CC2 78383,c1(C(N2C3CC(NC(c4nccc(C)c4)=O)C3CC2)=O)ccc2c(c1)OCC2 78384,CS(=O)(=O)c1cccc(-c2nc(C3COC(=O)O3)n(C3CCSC3)n2)c1 78385,c1(OC)cc(CCSC)c(OC)cc1C.N12CC(C(CO)C1)NC(=O)C2c1ccsc1 78386,c1(C(=O)NC2C=CC(CNC(C3ON=C(CC)C3)=O)C2)cc(F)c(Cl)cc1F 78387,C1(NC(C2COCCO2)=O)CN(c2ncnc3sccc23)C2CCCCC12 78388,N1(C(C2(C(N(C)C)=O)CC2)=O)CCC(CNC(=O)CCc2nc[nH]n2)C(O)C1 78389,C(N=c1nc2sccc2c(NCc2cccc(N(C)C)c2)[nH]1)c1ccc(C)nn1 78390,c1(SC(C)C(N2CC(NC(C3CCS3(=O)=O)=O)C(C)C2)=O)ccc(F)c(F)c1 78391,N1(C(CC2C(C)(C)C2(C)C)=O)CC2CN(C(C3(C#N)CCCCC3)=O)CCC12 78392,CC(C)(C)C(=O)NCC1CC(CNC(C2CCCSC2)=O)C1 78393,CC1CCN(C(C2N(C(C3CCC(C#N)CC3)=O)CCC2(C)C)=O)CC(C)O1 78394,C1(NC(CC=C(C)C)=O)CC2CN(C(=O)C(C)(C)COC(C)C)CC2C1 78395,N1(C(C(C(CC)C)=O)=O)CC(C(=O)NCCC(O)C(=O)OC)C2(CCC2)C1 78396,N1(C(C2C=C(C)CS2)=O)CC(C2CC2C(=O)NCC2CNC(=O)C2)C1 78397,N(C1CCCn2ccnc21)C(C(CCC1CC1)NC(C1CCCCS1)=O)=O 78398,c1(C(=O)NCC2C(NC(=O)COc3cncc(Cl)n3)C2)cnc2n1CCC2 78399,n1(CC)cc(NC(=O)CC2(C)CCN2C(C2CN(C)C(=O)N2)=O)ccc1=O 78400,N1(C(CCC)=O)CCCC(CCNC(=O)Cc2nn(CC)cc2Br)C1 78401,c1(CC(=O)NC(CNC(C(CC#C)O)=O)CO)ccc([N+](=O)[O-])cc1 78402,c1(CC(=O)NCC2CCN(C(C(COCC)C)=O)C2)cc(Br)ccc1C 78403,N1(C(CC(C=C)(C)C)=O)CC(C)CN(C(c2c(F)cc(OC)cc2Cl)=O)CC1C 78404,c1(NC(C2N(C(C=CC=CCC)=O)CC(O)CC2)=O)cncc([N+](=O)[O-])c1 78405,Cc1ccc(N(C(=O)CCC2NC(=O)NC2=O)C)cc1C 78406,c1(C(C(=O)NCC2CC(F)(CNC(C34CC(OC)(C3)C4)=O)C2)O)ccc(F)cc1 78407,c1(C(=O)NCC(CC)NC(c2cn(C(C)(C)C)nn2)=O)c[nH]c(C)c1 78408,C1(CC(=O)NCCc2ocnc2CNC(=O)C(O)CC2CC2)CC(O)C12CCC2 78409,C1(O)(C(C)NC(c2ccnn2C)=O)CCN(C(=O)C=Cc2cnn(C)c2)CC1 78410,C(=O)(C1CCc2ccc(Cl)nc21)NC1CN(C(C(N)=O)=O)CC1CCO 78411,CC(C)(C)CC(F)C(=O)NC1CN(C(C2CN3CCC2(C)CC3)=O)CC1O 78412,c1(C2C(C)C2)ccc(C(=O)N(C)CCN(C)C(c2csc(Cl)n2)=O)o1 78413,c1(NC(=O)C(C2CC3C=CC2CC3)N2CC=CC2CF)cccc([N+](=O)[O-])c1 78414,C1(CNC(c2cc(CNC(C3C(C)(C)COC3)=O)[nH]n2)=O)CC2CCCC2C1 78415,CC1=C(C(=O)N(C2CCC(NC(=O)CCc3cc(C)cc(C)c3)C2)C)SCCO1 78416,Cc1ncc(C(=O)NC2CN(C(C3C(C)C3(F)F)=O)CC23CC3)cc1N 78417,CC1(C)CCc2ccccc2C1NC(=O)Nc1ccc(OC2CCCCC2)cc1 78418,C1(=CC(=O)NC(C2N(C(c3c(C)oc(Cl)n3)=O)CCCC2)C)CN2CCC1CC2 78419,Cc1ncc(C(=O)NCC2CCN2C(C2CC23CCCC3)=O)cc1CC(C)C 78420,C1(C(=O)NC(C)CCN(C)C)COC(CNC(=O)COCCN(C)C)C1 78421,n1(CC)cc([N+](=O)[O-])c(C(N2CC3CCC(C2)N3C(C2CC(O)CN2C)=O)=O)n1 78422,c1(N2CC(C)C(CNC(c3cc4[nH]ccc4s3)=O)CC2)ccncc1[N+](=O)[O-] 78423,CC1(C)CC(NC(C2CCCS2(=O)=O)=O)CN1C(c1csc2nnsc12)=O 78424,CCCC(C(=O)N(C(CC1CC1)CO)C)NC(=O)C(F)CN(C)C 78425,CC(C(=O)OCCCCOCCCNC(=O)C1=NOCC1)C(C)(C)c1ccccc1 78426,CCCCC(C(=O)NC(C)CNC(C1CCCN(C(=O)C2CC2)C1)=O)N(C)C 78427,C(C)(CSC)(C(=O)NC(CN1CCCC1)CC)NC(C1C(OCC)CC1)=O 78428,N1(C(c2noc(C)c2[N+](=O)[O-])=O)CCCCC(C2CN(C(C3(F)CC3)=O)C2)C1 78429,C(CC(CC)C(=O)NCCNCC(=O)NCC(=O)NC(=O)NC)=CC 78430,N1(C(Cc2ccc(C(=O)OC)nc2)=O)CCCC(NC(=O)C(F)C(C)(C)O)C1C 78431,c1(C(=O)OCCn2ncc(C)c2)csc2ccc(F)cc12 78432,c1(OC)ccc2c(c1)C(N(C)C(c1cc(C)c(Cl)s1)C(=O)NCCCF)CC2 78433,C1(C(N(C2CCCC2)CCNC(C2CS(=O)C2)=O)=O)CCC2CCCCN12 78434,Cc1ccc(C(N2CC=CC2(C)C(=O)NC(C)CF)=O)nc1C 78435,c1(C(C(N2CC3C(CNC(c4cc(C)n(C)n4)=O)(C3)C2)=O)O)ccc(F)c(Cl)c1 78436,C12(C(N)=O)CCCC1(C(=O)NC1CCCC1NC(=O)Cc1nnc(O)s1)C2 78437,C1(C(=O)NCc2ncc[nH]2)COCCC12CN(C(c1ccnc(Cl)n1)=O)C2 78438,N1(C(c2cc(CC)ncn2)=O)CCCC(O)(CCNC(c2ccc(Cl)o2)=O)C1 78439,c1(-c2cnc(C#N)c(F)c2)ccn2cc(C(=O)NC3CCCC(F)(F)C3)nc2c1 78440,N1(C(C=C(C)c2cccs2)=O)CCC(CO)(NC(=O)CCN2CCOC2=O)CC1 78441,C(=O)(C1CCCc2sccc21)N1CC(CNC(c2c(C)cno2)=O)OC(C)(C)C1 78442,C1(OC)CCC(C(N2CC(F)CC2CNC(=O)C(c2nc(C)cs2)C)=O)CC1 78443,c1(C(=O)NCCn2cccc2)cn(C2CCOC2)nn1 78444,C(CC(=O)N(C(C)CN(C(=O)C(C)n1cncn1)C)C)OCCC 78445,c1(OC)ccc(C(C)(C)C(=O)NC(C2CN(C(=O)C(O)CN(C)C)C2)C)cc1 78446,c1(C(N2CCCC(C(C)(C)C)C2)C(=O)NCCC)csc([N+](=O)[O-])c1 78447,c1(CN2CC3(C(CNC(c4ccnc(CO)c4)=O)C3)C2)ccccc1OC(F)F 78448,C(=O)(C(C)(C)CCCF)N1CCC(C2N(C(C3=CC(C)(C)C3)=O)CCC2)CC1 78449,C(=O)(C1CCCn2cnnc21)NCC(CO)NC(c1ccc(OCOC)cc1)=O 78450,c1(C(=O)NCCCC(C)NC(C(COC)C)=O)cc(N2CCNC2=O)ccc1F 78451,c1(N2CC(CNC(c3ccc(OC)c(C)n3)=O)OC2=O)c(C)cc(Br)cc1C 78452,CC1(C)C2CCC(C2)C1C(N1CC(NC(C2CC(O)C2)=O)C1)=O 78453,c1(OC)cc(C(=O)COCC(O)C(=O)N(C)C)ccc1OCC(=O)OC 78454,c1(OC)ccn2cc(C(N3CC=CC3CNC(c3cc(Cl)c[nH]3)=O)=O)nc2c1 78455,c1(C(N2CCC(NC(c3nn(CC)c(O)c3)=O)C(C)C2)=O)c(N)cc(F)cc1Cl 78456,CC(C)C1=NOC(C(=O)NCCCCNC(C2(C)CCC(=O)NC2)=O)C1 78457,C1(NC(c2cnn(C)n2)=O)CCCCC12CCCN(C(=O)CN1CC3CC3C1)C2 78458,c1(CC(N2CC3C(NC(CC(CC)C)=O)C(CC3)C2)=O)ccc(Cl)c([N+](=O)[O-])c1 78459,c1(C(=O)NC2CCC(CNC(C3C(C)(C)C3(F)F)=O)C2)cc(F)ccc1F 78460,c1(N(CC)CC)cncc(NCc2csc(-c3ccccc3OC)n2)c1 78461,C(=O)(C1=CNC2=NCCCC2=C1)N(CC(CO)(CO)NC(CSC(C)C)=O)C 78462,CC1CCC(CC(=O)NC2CCC(NC(=O)CC3COC(C)(C)C3)CC2)OC1 78463,N1(C(c2cc(Cl)ncc2O)=O)CC2CC(C1)N(C(c1coc(O)n1)=O)C2 78464,C1(NC(=O)Nc2ccc(C)s2)CCN(C(C2CN(CC(C)C)C2)=O)CC1C 78465,C1(CNC(C(COC)(C)O)=O)CC2CCC1N(C(c1cnn3c1OCC3)=O)C2 78466,c1(CN(c2ccccc2C(C)C)C(C(C)OCCOC)=O)cccc(C#N)c1 78467,C(=O)(C(F)(F)C(C)(C)O)NCC(=C)CCNC(=O)C(c1ccccc1)F 78468,N1(C(CCSC)=O)CCC2(NC(=O)CCCCC(C)C)CCCCCC12 78469,C1(NC(C(CO)NC(Cc2cc(CC)no2)=O)=O)C=CCCCC1 78470,Cn1cc(C2CC2NC(=O)CCCn2cc(CCC3CCCCC3)nn2)cn1 78471,C1(CC)CCN(C(C)=O)C1C(=O)N(C)CCOC.c1(C(N(C)C)=O)nc(OC)c(C)s1 78472,c1(C(=O)NC2C(NC(c3sccc3C3CC3)=O)CC2)cn2c(n1)CCC2 78473,C#Cc1ccc(C(=O)NCC(C)(C)C(=O)NCC2(COC)CCCC2)cc1 78474,c1(C(=O)NCC2CCN(C(c3c(C)cnnc3)=O)CC2C)ccc(N)c(Cl)c1O 78475,C(=O)(C(F)(CNC(c1cn(C)cc1C)=O)C(C)C)N1C(C)(COC)CCC1 78476,N1(C(Cn2cc(CNC(=O)C=CC3CCCCC3)nn2)=O)CC2CCC(C1)O2 78477,C1(CCN(C(CC(COC)C)=O)C2CCOCC2)CCN(c2cncc(Cl)n2)CC1C 78478,c1(C(N2CC(CCNC(C(C)OC)=O)C(C)C2)=O)csc2cccc(F)c12 78479,CC(C)CCCC(C)CNC(=O)C(F)CC1CN(C(C2CC2[N+](=O)[O-])=O)C1 78480,c1(OC)cccc(CNC(=O)OC(C)(C)C)c1C.C12CCCN(C1)C(=O)C(=O)N2 78481,C(=O)(C#CC1CCCOC1)NCC1(NC(C(COC)CC(C)C)=O)CC(OC)C1 78482,c1(OC)ccc(NC(C2CN(Cc3ncccc3OC)CCS2)=O)cc1O 78483,C(=O)(CC(C)CC(=O)N(C(CC(F)F)C(=O)NCC1=C(C)CCC1)C)OC 78484,N1(C(c2c(C)n3c(n2)scc3)=O)CCC2C1CCCN2C(=O)CC(C)P(C)(C)=O 78485,C12(C(=O)OC)CCNC1CN(C(c1cccc(C3(C)CCO3)c1)=O)C2 78486,CC1CC(=O)NCCN1C(c1c[nH]nc1-c1ccc(Cl)s1)=O 78487,N1(C(C23CC(CC(C)O2)C3)=O)CC2CCCC(C1)N2C(=O)CCn1cncn1 78488,c1(C(=O)NC(CCSC)C)cc(CNC(=O)CCc2nncs2)[nH]n1 78489,C1(NC(C2C(C=C)C2)=O)CC2CCC(C1)N2C(c1ocnc1C(F)(F)F)=O 78490,C1(C(=O)NCCC2CCCN(C(CCCCC#N)=O)C2)CC12CCC1(CC1)CC2 78491,S(=O)(=O)(CCC(=O)NC1CC(NC(c2ccc(Cl)c(N)c2)=O)CC1O)NC 78492,C1(C(N(CCNC(C(F)=CCC)=O)C)=O)CC(CC)=NO1 78493,CCC(C)CC(C(=O)NCc1ccc(O)c(OC)c1)NC(=O)C(C)CC(=O)OC 78494,C1(NC(c2cc(C)c(Cl)s2)=O)CCCN(C(=O)COc2cc(F)cc(F)c2)C1C 78495,c1(NC(CCC2N(C(C3CCC(CC)O3)=O)CCC2)=O)ccc2ccoc2c1 78496,C(=O)(CC(C)CC(C)(C)C)NCC(CC)(CC)NC(C1CC(O)CN1C)=O 78497,N1(C(C(CC)n2cccn2)=O)CCC(NC(=O)CCCn2ccnn2)CC1 78498,C12(NC(=O)C(C3CCOCC3)O)CCCC1N(C(=O)CCc1ccon1)CCC2 78499,N1(C(C23OCC(C(C)C)(C2)C3)=O)CCC2CN(C(=O)C(O)P(C)(C)=O)CC2C1 78500,c1(C(=O)NCCNC(C(C(C)C)SCC)=O)ccc(C)c(C#N)c1 78501,c1(C(=O)OC)cc(NC(=O)NC(C2CCCC2O)C)c2c(c1)CCC2 78502,CC1CCC(NC(=O)C=C2CCCC2)CN1C(c1cc(Br)n(C)c1)=O 78503,c1(C(CNC(=O)NC(CC)C(F)F)CC)ccc(F)c(F)c1 78504,N1(C(c2cc(SC)ncc2)=O)CC2CN(C(c3cccc(C(C)C#N)c3)=O)C2C1 78505,N1(C(CC2(OCC)CCC2)=O)CC(OC)C(NC(=O)Cc2ccccc2)C1 78506,c1(SC)nc(NC2(CNC(C3CCC(O)C3)=O)CCCC2)cc(C)n1 78507,c1(OC)cc(C(N2CCCC(SC)CC2)C(=O)NC2CCC2)ccc1S(C)(=O)=O 78508,C1(N(C(=O)CC2(CO)CCCCC2)CC)CCCN(C(=O)CC(O)CC)C1 78509,C1(CC=C)(NC(=O)CCN2CCCC2)CCN(C(C2(CSC)CCC2)=O)C1 78510,C1(CNC(=O)C=CCN2CCCC2)(NC(C2COC(=O)N2)=O)CCOC1 78511,c1(CC)cccc(C(=O)NC2(COC)CCN(C(C3CC3(C)CC)=O)CC2)c1O 78512,CC1CCN(C(=O)Nc2coc(Oc3ccccc3)n2)CC1Nc1ccccn1 78513,CC(C)CCCC(C)C(=O)NCC1(NC(=O)C=Cc2cocn2)CCCCC1C 78514,CCC(C)(C(=O)Nc1nc(-c2ccc(F)cc2)cs1)OC.C12C=CC(C1)NC2=O 78515,c1(N2C(CNC(C(C)C)=O)CC(F)C2)cc(-c2cccs2)ncn1 78516,c1(C(=O)NCC2CC(OC)CN2C(c2cscc2OC)=O)cc2cnccc2o1 78517,c1(C(=O)OCC)cc(NC(C2CCCN(Cc3cncs3)C2)=O)ccn1 78518,C(=O)(C1=CCCC1C)N(CC(C)O)CCNC(c1ccc(C2CC2)o1)=O 78519,Cc1cc(C)c(CNC(=O)C(C)Oc2ccc(C(C)(C)C)cc2)s1 78520,CC1CN(C(c2cnc(Cl)cn2)=O)CC(C)N(C(c2cc(F)ccc2O)=O)C1 78521,c1(CC)cc(C(N2CC(NC(C3C(C)C3C)=O)C(F)C2)=O)cc2c[nH]nc12 78522,n1(CC(N2CCC(c3c(C(=O)OC)nco3)CC2)=O)cc(C)c(=O)cc1C 78523,Cc1ccc(=N)[nH]c1C(N1CC(NC(=O)C(C)(C)c2cccs2)CC1C)=O 78524,N1(C(C2C(C)C2)=O)CCC2CN(C(c3ncccc3F)=O)CC12 78525,Cc1nn(C(C)C)cc1C(=O)NCC1CC1NC(=O)C(c1ccc(F)cc1)F 78526,C1(NC(C(C)(C)OCC)=O)CCCC(NC(c2cncc(CC)c2)=O)C1 78527,C(CC(=O)N1CC2(C1)CN(C(C13CCC(C)(CC1)C3)=O)C2)(C(F)(F)F)N(C)C 78528,CCC(O)C(C)C(=O)NC1CN(C(=O)CSc2cn[nH]c2)CC1C(F)(F)F 78529,C1(CNC(C(c2ccnn2C)NC(C(C)NC(CC)(C)C)=O)=O)CCC(F)(F)C1 78530,N1(C(C2C(NC(CC(COC)(C)C)=O)CCCC2)=O)CCc2ccncc21 78531,N1(C(C=CC=CCC)=O)CC2(CCC2)CC1CNC(c1cnccc1Br)=O 78532,C(CCC(C)CC(=O)NCCNC(c1cccc(O)c1F)=O)=C(C)C 78533,C(=O)(C1CCCc2nnn(C)c21)N1C(CN(C)C(c2n[nH]cc2Cl)=O)CCC1 78534,C1(F)(CNC(c2n(COC)ncc2)=O)CCN(C(c2nc(=O)n(C)[nH]2)=O)CC1 78535,N1(C(CCCCC)C(=O)NC(C)C)CCC(S(=O)(=O)NC)C1 78536,c1(C(=O)OC(C2CC2Cc2c(OC(C)C)cccc2)=O)c(Cl)cccc1[N+](=O)[O-] 78537,C1(O)(C(=O)NC2CCC(CNC(c3c(C)ccnc3C)=O)C2)CCC(C)(C)CC1 78538,N(C(=NCC(C)(C)OC1CCOCC1)NC1CCC1)C(C)C1CC1 78539,N1(C(c2cc(-c3ccccc3)on2)C(=O)NCCSC)CCC(O)C(O)C1CC 78540,CN1N=C(C(=O)NCC2(CC(=O)NCC3CCCCS3)CC2)CCC1=O 78541,N#Cc1ccc(CC(N2CC3CC2C3NC(c2cnccc2C(N)=O)=O)=O)cc1 78542,C(=O)(C1=CCCC1C)NCC1(COC)CCCN1C(=O)CCS(C)(=O)=O 78543,N1(C(C2N(Cc3cnc(CCCC)[nH]3)C3C(C2)C3)=O)CCOCC1CO 78544,c1(C2(C(=O)NCC3(F)CC(CNC(C4(C)CCCS4)=O)C3)CC2)cccc(F)c1 78545,c1(C(COCCCCC)C)ccc(NC(C2CCC2c2ccc(Cl)cc2)=O)cc1 78546,c1(C(C)C)noc(CCCC(=O)N(C(CNC(c2nccn2C)=O)C2CC2)C)n1 78547,C12(CNC(C3C(C(C)C)(CC)C3)=O)CC1CN(C(=O)CN1CC(=O)NC1=O)C2 78548,c1(CC(C)C)ncc(CNC(C)Cc2cnc[nH]2)s1 78549,N1(C(C2(OC)CC2)=O)CCC(NC(C2(C(F)(F)F)CC3(CCC3)C2)=O)C(O)C1 78550,CC1OC2(C(=O)NC(C)CCN(C(=O)CCc3ccc(C(F)F)cc3)C)CC1C2 78551,c1(CC(N2CCCC(c3cc(OC)c(C)cc3)C2)=O)ccc2occ(C)c2c1 78552,N1(C(C=C(C)CN2CCOCC2)=O)CC2CCN(C(c3cn[nH]c3)=O)CC(C2)C1 78553,C(=O)(C(C1(C)CC1)NC(=O)C(F)OC(F)(F)F)NCC(C1CCC1)OCC 78554,N1(C(c2ccc(C#N)s2)C(=O)Nc2c(C)cc(F)cc2)C2CCC1CC(CO)C2 78555,N1(C(CNC(N)=O)=O)CCC2CCN(C(c3csc(-c4cccs4)n3)=O)CC12 78556,CCCCC(CNC(=O)C(C)Cc1cnc[nH]1)NC(c1cc(C)nn1C(F)F)=O 78557,Cc1ncncc1C(=O)NCC1CN(C(c2ccnc(Br)c2)=O)CCO1 78558,c1(OC)cc(C(N2C3CN(C(c4sncc4C)=O)CC23)=O)cc(OC)c1C 78559,N1(C(C=C(CC)CC)=O)CCC2(CCCC2NC(C2CCS2(=O)=O)=O)CC1 78560,C1(CC=C)(NC(=O)C(C)OCC(C)C)CCCN(C(c2cc(N)nc(Cl)c2)=O)C1 78561,c1(C(=O)NC(c2ccccc2)C(=O)NC(C)Cc2ccnn2C)ccc(C#N)cn1 78562,CN1CC(C(N2CCCCC2C2CCN(C(=O)Cn3[nH]cnc3=N)C2)=O)NC1=O 78563,C1(C(=O)NC(c2nocc2C(=O)N(CCF)C2CC2)C)CC=CCC1 78564,C12(NC(NNC(=O)C(C(F)(F)F)C3CCCNC3=O)=O)CCCN1S(=O)(=O)CC2 78565,c1(CC)c(C)noc1.c1(CC)nn[nH]c1C(=O)NCc1nocc1C(=O)N 78566,Cc1nn(C)c(N(C)C)c1CCCc1ccc(Cl)cc1Cl.C12(F)CC1C(=O)NC2 78567,C1(O)(C(=O)NCC2(O)CN(C(=O)C(O)CC3CC3)C2)Cc2ccccc2C1 78568,c1(C(=O)NCCN(C(CCC=C)=O)CC(C)O)cc(C2(C)CC2)ccc1F 78569,c1(OC)cc(C)cc(C(=O)NCC2(O)CN(C(=O)C3=COCCC3)C2)c1N 78570,c1(SC)ncc(C)c(N2CC3(CC3C(N3CCCC3CN3CCCC3)=O)C2)n1 78571,c1(SCC2(N)CCOC2)cc(Cl)c2cccc(Br)c2n1 78572,C1(C)(N(C)C)CCCN(C(c2cc(C(c3cccs3)=O)cnc2O)=O)C1 78573,C#CC1(C(=O)NCC2(CC)CCCO2)CCN(C(=O)C(O)C(C)C)C1 78574,C(c1csc(C(F)(F)F)c1)=CC(=O)NCCC1N(C(CCC#C)=O)CCC1 78575,C1(CNC(c2c(C)snn2)=O)CC(NC(c2ccc(C3CC3)s2)=O)C(O)C1 78576,N1(C(=O)NC(C(=O)OCC)c2ccns2)C(=O)COCC1(C)C(C)C 78577,C1(C(=O)NC2CCN(CCNC(c3c(C)n[nH]c3)=O)CC2)CC(C)CC(C)C1 78578,C1(CNC(C2CN(C(c3ccc(CC)cc3)=O)CC2O)=O)Cc2ccccc2O1 78579,N1(C(c2cnc(-c3cccc(C#N)c3)s2)=O)CCC2(CC(=O)NC2=O)C1 78580,CC1(C)CCN(C(=O)Cn2nccc2N)CC1CNC(=O)CCN1CCCC1=O 78581,C(N=c1[nH]c(C)c([N+](=O)[O-])cc1Cl)C1OCC(CNC(c2c(CC)ccs2)=O)C1 78582,c1(C(=O)OCC)c[nH]c(=NC)nc1CN(C)Cc1ncc(Cl)n1C 78583,N1(C(c2ncn(C(C)C)n2)=O)CCCC(CN(C)C(c2ccc(F)cc2)=O)C1 78584,C1(CNC(=O)NCC(c2cccc(Cl)c2)C)CCC2C(CC1)C2(F)F 78585,C(=O)(CCS(=O)(=O)N(C)C)NC1(C)CC(NC(c2cc(CC)nn2C)=O)C1 78586,C1(CNC(Cn2ncc(C)c2)=O)CC2(CO1)CN(C(=O)C(N1CCCCC1)C)C2 78587,CC1CN(C(=O)CC2CCC(=O)NC2)CC1CNC(=O)CN1CCCC1=O 78588,C(CC(C)C(=O)NCC1(NC(=O)CCCc2n[nH]c(=N)s2)CCCC1)OC 78589,N1(C(C2C(C)CCO2)=O)CC(NC(=O)Cc2ccccc2Cl)CC12CCOCC2 78590,CC(=Cn1ccnn1)C(=O)NCCC1(NC(C2CCCN2N=O)=O)CC1 78591,Cc1nc2[nH][nH]cc-2c(=NCC=CCNC(c2cc3n(n2)CCNC3=O)=O)n1 78592,C1(C(=O)NC2(C3N(C(C4C(C)C4)=O)CCC3)CC2)CC2(CC2)CN1C 78593,C1(N(C(c2cccs2)=O)CC)CCCN(C(=O)CSc2ccccc2)C1 78594,C(=O)(C(C)(C)CCCOC)NCCN(C(=O)C=CCN1CCCCC1)CCC 78595,c1(C(=O)NCC(C2CCCCC2)NC(C(C=C)O)=O)ccnnc1Cl 78596,N1(C(C2N(C(C(CO)OC)=O)C(C3CC3)CC2)=O)C2CCC1CN(C)C2 78597,C(CCCCC(=O)NC1CCC1CNC(=O)CC12COC(C)(C1)C2)SC 78598,c1(CC(=O)NC2(CNC(C=CC(C)(C)SC)=O)CC(F)(F)C2)ccc(C)cc1F 78599,c1(CC)ccc(OCC(=O)NCC(CC)NC(=O)C(C)C2(O)CCC2)cc1 78600,c1(NC(C(c2ccccc2)C)=O)cccc(NCC(F)(F)F)c1 78601,c1(C(=O)NCC2(F)CC(NC(CCCCOC)=O)C2)cc2n[nH]cc2cc1C 78602,C(=O)(C(O)CCCC)N1CCC(CC=C)(C(N2CC(Cc3ccoc3)C2)=O)C1 78603,c1(C(N2CCOCC(NC(C3(C)C=CCCC3)=O)C2)=O)ccc(C#N)cc1O 78604,N1(C(C2(C(=O)NC)CCC2)=O)CCCC(C2CC2NC(C2CC23CCC3)=O)C1 78605,N1(C(CSSC)=O)CC(CNC(c2cc(C(F)(F)F)ncn2)=O)C(O)C1 78606,c1(C(=O)NCC2(F)CC(NC(=O)CC3CSCCS3)C2)ccc(F)c2ccoc12 78607,C1(C)(C(=O)NCC(C)(C)OCCNC(c2c(C)n(C)nn2)=O)CCC(=O)NC1 78608,c1(NC(C2C(C(=O)NC3CC4(CC4)C3)C2)=O)cccc(I)n1 78609,CCC(CC(=O)NC(C)CNC(=O)CCc1cccc(Br)c1)OC 78610,N1(C(C(C(C)C)N2CCCCC2)=O)CC2CCC1CN2C(c1ccc(F)cc1)=O 78611,Cc1ccc2c(NC(C3(CNC(=O)CC(C)CC(C)(C)C)COC3)=O)cccc2c1 78612,S(=O)(=O)(c1ccc([N+](=O)[O-])cc1Cl)NCC1CCCN(C(C2(C)CCCC2)=O)C1 78613,C1(NC(c2c(C)sc(O)n2)=O)CC(O)CN(C(C2CC(C(F)(F)F)C2(C)C)=O)C1 78614,c1(C(=O)NCCN(C(C23CC(C2)C3)=O)CC)cc(Br)cc2c1CCN2 78615,C1(F)(C(N(CC)Cc2ccccn2)=O)CCN(C(C2SCCS2)=O)C1 78616,c1(C(=O)NC(CCNC(C(CCC)N(C)C)=O)C)cc([N+](=O)[O-])n(C)n1 78617,C12(CC(O)C1)C(=O)N2.CC1CC1C(=O)NCC(=O)NCCCO 78618,Cc1cc(C(=O)NC(CO)CCCCNC(=O)C(C)C(C)(C)C)cc(=O)n1C 78619,c1(C(N2CCN(C(C3CCS(=O)(=O)N3)=O)CC(O)C2)=O)csc2ncnc(O)c12 78620,N1(C(c2cc(C(CC)CC)no2)=O)CC(C2CN(C(C3(CN(C)C)CC3)=O)C2)C1 78621,C1(CC(=O)NCCNC(=O)CC2OCCCO2)CC2CCC1CC2 78622,CC1(CO)CCCC1NC(C1CCC1NC(C1CC1(F)Cl)=O)=O 78623,N1(C(=O)Cc2ccc(Cl)cn2)CC2CCCN(C(C3COC4(CCC4)C3)=O)C2C1 78624,c1(C(N2C(C(C)NC(C3(CF)CC3(F)F)=O)CCC2)=O)ncc2n1CCCC2 78625,C1(F)(C(=O)NCCC(C)CO)CCN(C(=O)C=Cc2cn(C)nn2)C1 78626,C(=O)(CCCCCF)N1C(C(C)NC(c2cc(OC)no2)=O)CCCC1 78627,C(=O)(C1CCc2snnc21)N(C)CC1CCN(C(C(n2ccc(C)n2)(C)C)=O)C1 78628,c1(C(N2CCC(C)(NC(C=CCOC)=O)C2)=O)ccnc2ncsc12 78629,c1(OCC)ncccc1C(=O)NCCCCC(C)NC(=O)COc1ccccc1 78630,C1(C(=O)NC(CC(C)NC(C=CSC)=O)C)CCCCN1C(=O)OC(C)(C)C 78631,c1(C(N2C3(CNC(C(C)SC)=O)CCC2CC3)=O)cccc2c1OC(C)C(=O)N2 78632,Cc1ccc(C(N2CC(NC(c3cncc(N)n3)=O)C(C(F)F)C2)=O)nc1C 78633,N1(C(c2c(Cl)ccc(CC)c2)=O)CCN(C(c2cc(SC)[nH]n2)=O)C(C)C1C 78634,C1(CNC(=O)CC2(CO)CC2)CCCN(C(=O)C(F)(F)c2cscn2)C1 78635,N1(C(c2c(C)nsc2)=O)CCCC2(C1)C(NC(c1cn(C)nc1Cl)=O)CCN2C 78636,N#Cc1ccc(SCN=c2[nH]nc(C3CCCCC3)s2)cc1 78637,N1(C(C(C2CC2)OCC)=O)CCC2C(NC(c3cc(CC(C)C)c[nH]3)=O)C2CC1 78638,Cc1cc(C(=O)NC2CCCN(C(=O)CSC3CC3)CC2)ccc1[N+](=O)[O-] 78639,c1(C(N2CC(NC(C3CCN(C)C3=O)=O)C2)=O)ccc2c(O)n[nH]c2c1 78640,C1(CN(C(CNC(CNC(C)=O)=O)=O)C)CN(C(c2cnncc2O)=O)CCO1 78641,C1(C(N(CC(C)NC(C2CCS(=O)(=O)CC2)=O)CC)=O)(OC)CCCCCCC1 78642,c12ccc(C)c(c1)N(C)C2=O.N1(C(C2C(C)(CC)C2)=O)CCC(NC(C)=O)CC1 78643,C1(C)(CNC(C(C2CN(C(=O)CC3(C)CCOC3)C2)OC)=O)CCCC1 78644,c1(C(=O)NCCCC(C)NC(C2CC3(CC(=C)C3)C2)=O)ccc2sc(=N)[nH]c2c1 78645,C1(N(C(C(C)SCC)=O)CC)CCC(NC(=O)CC2COCCN2C)CC1 78646,C(CCCC(C)NC(c1c(Cl)n[nH]c1C)=O)NC(CC1(CSC)CC1)=O 78647,c1(C(N(C2CCCC(NC(c3occc3F)=O)C2)C)=O)ccc(F)cn1 78648,Cc1nc(CNC(=O)C(O)CNC(C2CC(C3CC3)C2)=O)sc1C 78649,C1(C(=O)NCCN(C(C)C)C(C)C)C(NC(=O)C(C)CO)C1(C)C 78650,Cc1cc2ncc(C(=O)NCC=CCNC(c3ccc(Br)c(F)c3)=O)cn2n1 78651,CC(CC(=O)N1CC(NC(=O)Cc2cc(F)cc(Br)c2)C(O)C1)C(F)F 78652,N1(c2snc(C(=O)OC)n2)CC(CNC(=O)Cc2cnco2)OC(C)(C)C1 78653,N1(C(C2(OC)CS(=O)(=O)C2)=O)C2CCC1CN(C(=O)CCCNC(N)=O)CC2 78654,C1(C(N2C(C)C(NC(C3(C)CC(F)C3)=O)CC2)=O)CC2C(C1)C2(F)F 78655,CCC(C)(COC)C(=O)N1CCC(CNC(c2cnn(C3CCCC3)c2)=O)C1 78656,CCC(CC(C)C)C(=O)N1CC(O)(CNC(c2nc(Cl)sc2Cl)=O)C1 78657,c1(NC(N2CCCC(CCCO)C2)=O)cccc(-c2ccc[nH]2)c1 78658,c1(CC)cc(C(=O)NCC2CC(NC(C3CN(C(C)C)C3)=O)C2)oc1CC 78659,C(=O)(CCC1=CCCCC1)NCCCCCNC(c1nc(N)c(O)cc1)=O 78660,CC1=NOC(CCNC(=O)C(C)(C2CCC2)NC(=O)CC2(C)CC2)C1 78661,c1(C(N(CCC)CCN(C)C)=O)ccc([N+](=O)[O-])c(SC)c1 78662,C1(C)(C(=O)NC(c2cn(Cc3cnc(C)nc3)nn2)C)Cc2ccccc2C1 78663,CCCC(CC)CCC(=O)NC1CC2(C(=O)NC(C)(CO)CO)COC1C2 78664,C12(NC(=O)OC(C)(C)C)CCCC1CCN2C(c1ccc(F)c(N)c1F)=O 78665,C(CNC(=O)CCC(C)N(C)C)(CC(F)(F)F)NC(Cn1c(C)nnn1)=O 78666,C1(C(=O)OCC)CC(C(N2CCC2(C)NC(CCC)=O)=O)C1(C)C 78667,C(C(CN=c1[nH]cnc(Cl)c1Br)CCOOC)NC(c1ccc(OCC)cc1)=O 78668,C(C(O)C(=O)NCC(c1ccccc1)NC(=O)CC1CC12CC2)SC 78669,C(CCC(=O)NCC1=NOC2CCCC12)(C(C)C)NC(c1nc(C)oc1C)=O 78670,N1(C(C(C)(C)C2CC2)=O)CCOC2(CCN(C(C3CC(=O)N(O)C3)=O)CC2)C1 78671,c1(C(N2CCC(N(C(=O)CC3=NNC(=O)C3)CC)C2)=O)ncc([N+](=O)[O-])cc1C 78672,C1(C(N(CC(F)(F)CO)C)=O)CN(C(=O)C(C)(C)n2cncn2)CCO1 78673,CC1C(C(=O)NC2CC(F)C2)C(C(=O)O)C1(C)C 78674,c1(CC(=O)NC2CC(C(=O)NCc3c(C)nns3)OCC2)c(F)cccc1F 78675,C1(O)(CNC(c2cccc[n+]2[O-])=O)CCCN(C(=O)C(Cl)=CCl)CC1 78676,c1(NC(CN2C(Cn3cc(CCS(C)(=O)=O)nn3)C=CC2)=O)ccc(F)c(F)c1 78677,c1(C(=O)NCC(C)NC(c2cc(C(C)(C)C)no2)=O)cn(CCC2CC2)nn1 78678,Cc1cc(C(N2CCC(N(C(=O)CC3COC(=O)C3)C)C2)=O)ncc1CO 78679,N1(C(c2c(C)noc2C)=O)CC2CC1CN2C(=O)CSCC(F)F 78680,C(C)(CNC(=O)CN(C1CCCC1)C(C1(n2nccn2)CC1)=O)(C1CC1)OC 78681,N1(C(c2c(C)cccc2Cl)=O)CC2(CCCC2NC(C2CCC3CC3CC2)=O)C1 78682,c1(C(C)C)ccc(C(=O)NCC(C)N(C(=O)CSc2ccccn2)C)s1 78683,CCC(CNC(=O)CCCN(C(=O)C(C)NC(C)(C)CC)C)CO 78684,CC1(C)CC(C(=O)NCC2CC2(F)F)CN1C(=O)CCc1cccc(O)n1 78685,N1(C(CCN(C(C2CCC(C)(C)OC2)=O)CC)=O)CC(S(N)(=O)=O)C1 78686,c1(C(=O)NC(CC)CC(=O)NCC(C)(C)C2CCCO2)ccnc(C)c1C 78687,c1(C(N2C(C(C)NC(CN3CC(C)(OC)C3)=O)CCC2)=O)ccc(N(C)C)cn1 78688,Cc1ccc(CN2CCCC2CCC(=O)N(C)Cc2ccccc2)c(Cl)c1 78689,c1(NC2(CNC(=O)CSC(F)F)CC2)nc2c(cc1Cl)C(=O)OC2 78690,C1(NC(C(CC)N(CC)CC)=O)CCN(C(=O)C2=CCCCCC2)CC12CCC2 78691,c1(CC)nc(O)c(C(N2CCC3CN(C(C45CCCC4C5)=O)CC23)=O)cc1C 78692,C1(N(C(C(=O)N(CCN(C(C=C(COC)C)=O)C)C)C)C)CCCOC1 78693,C=CCCCCC(=O)N(C)CC1(C)CCCC1NC(c1ccc(C)s1)=O 78694,C1(OC(CNC(C2(CCOC(C)=O)CC2)=O)=O)CCCCC1.C1(=O)CN1C1CC1 78695,N1(C(C(C)C)=O)CCCN(C(=O)C(n2nnnc2C(C)(C)C)C)C(C)C1 78696,c1(OC)ccn2c(C(=O)NCCN(C(c3c(C)ncn3O)=O)C3CC3)cnc2c1 78697,CN=C(NCCc1cc(-c2ccccc2)n[nH]1)NCCN1CCCC1 78698,N1(C(C2CC(N(C)C)C2)=O)CC2C(CC(=O)NCC3(n4cncn4)CC3)C2C1 78699,Cc1ccc2c(=NCC(C)(C)C3CCOCC3)[nH]c(=NCc3cc[nH]n3)[nH]c2c1 78700,C=CC1(CO)CCN(C(=O)C(CCC)NC(=O)CSCC(N)=O)C1 78701,C1(NC(c2cc(C(F)F)ccn2)=O)CC2(CCCCN2C(C2(CO)CC2)=O)C1 78702,C(=O)(CC(O)C(=O)NCC1CCN1C(C12CC(C1)C(C)(C)O2)=O)OC(C)(C)C 78703,S(=O)(=O)(c1cccc(=NCc2cn(C)nn2)[nH]1)NC(c1ccn(C)n1)CO 78704,N1(C(C)=O)CC(O)CC1C(=O)NCC1CCN(C(C2(C)CSC2)=O)C1 78705,C(=O)(CCCCCCCCCO)N(CC(CC)NC(C1(Cl)CC1(F)F)=O)C 78706,Cc1ccccc1C=CC(=O)NC(C(=O)NCC12CCN(CC1)C2)c1cccs1 78707,c1(SC)cccc(C(N2CC(O)CC2C(=O)NC2CN(c3ncco3)C2)=O)c1 78708,c1(C(C(=O)NCCC2CC2)N(C)CC2C3CCCC23)cc(C(C)(C)C)oc1C 78709,N1(C(c2c(CC)nn(C)c2)=O)CCCC2(C1)CN(C(=O)CC1CC1C)CCO2 78710,n1(C(C)C)cnc2c(NCc3cnn[nH]3)nc(N3CCC4(CCCOC4)C3)nc12 78711,C1(N(C(=O)C(N)=O)C)CCCN(C(=O)COCc2nc(C(C)(C)C)no2)CC1 78712,c1(C(=O)NCC(C)CN(C)C(C2CNC(=O)N2C)=O)coc2c(F)cc(F)cc12 78713,O=C(CCCNC(C1CCCS1)=O)N1CCC(NC(=O)OC(C)(C)C)C1 78714,C1(NC(C(N2CC(OC)(COC)C2)=O)=O)CCNC(CC2CC2)C1 78715,c1(OC)ccc(=NC(=O)C23CC2CN(C(c2cc(Br)ncc2F)=O)C3)[nH]n1 78716,n1(CC(=O)N(C2CN(C(c3cnnn3C)=O)CC2(C)C)C)nc(Cl)ccc1=O 78717,N1(C(C23C(C)OC(CO)(C2)C3)=O)CCCN(C(=O)CNS(=O)(=O)N(C)C)CC1C 78718,N1(C(CNC=O)=O)CC2CC1C2CNC(C1(c2ccccc2)CC1(F)F)=O 78719,c1(C(N2CCC(NC(CCC#CC)=O)(CC)CC2)=O)c(O)cnc2ccccc12 78720,C1(CC)(NC(c2ccc(NS(C)(=O)=O)nc2)=O)CCCN(C(C2(C)CC2C)=O)C1 78721,N1(C(C(C)C2CCCO2)=O)CC2(NC(c3ccc(Br)cc3N)=O)CCC1CC2 78722,C1(CNC(=O)C(=O)NC2CC2)CCC2CN(C(c3ccc(O)cc3)=O)CCC2C1 78723,C1(NC(C(C)(C)SC)=O)CC12CCN(C(=O)Cc1ccoc1C)CC2 78724,C(c1cn(C)c2ccccc12)=CC(=O)NCCCN(c1cc(C)ns1)CCO 78725,C(=O)(C(C)N(C(C1CCC1C)=O)C1CC1)NCCN(C(C)C)CC 78726,c1(C(N(CC(CNC(c2n(C(C)C)ccc2)=O)C)C)=O)[nH]ncc1C#N 78727,CCCCS(=O)(=O)NC(C)C(=O)N(C(C)CNC(=O)C=CCN1CCCC1)C 78728,c1(CC(CO)N(C2CC2)CC2C(C(N3CCC3)=O)C2)ccccc1.CC 78729,c1(C(=O)NC(CCCNC(c2nnc(C)s2)=O)C)cccc(CO)c1C 78730,C=CCCN=C(NCC1CC(=O)N(C)C1)NC1CCC(CC)CC1 78731,c1(C(C(N2CC(NC(C3(OC)CCCC3)=O)C2)=O)N(C)C)c(F)cccc1F 78732,N1(C(c2c(CC)[nH]c(=N)s2)=O)CCC2(NC(c3cc(Cl)c(Cl)s3)=O)CCCC12 78733,N1(C(C(CC)(F)F)=O)Cc2occ(C(N3CCC(CCCO)C3)=O)c2C1 78734,Cc1cc(C)n(CC(C)NC(=O)CC(N)Cc2ccc(F)cc2)n1 78735,Cc1ccc(C(F)F)cc1C(=O)NC(C1CCCN(C(C2OCCO2)=O)C1)C 78736,c1(C(C(=O)NC2C(OC)CN(C(C3CN(C)C3)=O)C2)O)ccc(Cl)cc1Cl 78737,Cc1cc(C)c2c(=NC(=O)NCC(F)(F)Oc3ccc(Br)cc3)[nH]sc2c1 78738,Cc1nc2ccc(S(=O)(=O)NC3CCC4CCCCC4C3)cc2o1 78739,Nc1ccc(Br)c(F)c1C(=O)NC(c1ccccc1)Cn1cncn1 78740,N1(C(c2cnn(CC)c2C)=O)CC2CCC2(CCNC(c2csnn2)=O)C1 78741,c1(CCC(=O)NCC2N(C(C(CC)C(C)C)=O)CC2)ccccc1[N+](=O)[O-] 78742,C1(N(C(C(CC)F)=O)C)CN(C(c2ccc(C(=O)NC(C)C)cc2)=O)CC1(C)C 78743,C1(=CC(=O)NCC2COCC2NC(C2CCOC2)=O)C2CC3CC(C2)CC1C3 78744,N1(C(c2cc(CC)on2)=O)CC(NC(c2sc3cncn3c2C)=O)C(C2CC2)C1 78745,C(CCCCCC(=O)N1CC2CCC2(CNC(=O)C(O)C(C)(C)C)C1)SC 78746,C(=O)(CC(C)(C)C(F)F)N1C(CNC(C(CCC)CC)=O)CCC1 78747,c1(C(=O)NCC(C)CNC(=O)CCCC(C)(C)C)n[nH]c2c1CCCCC2 78748,Cc1cc(C(=O)NCC(C)(C2CC2)NC(c2ccn(C)n2)=O)sc1C 78749,C(CC(F)F)(C(=O)N1CCC2C(O)CC12)NC(=O)CCN1CCOC1=O 78750,c1(NC(c2occ(C(C)=O)c2)=O)ccc(NC(C2(O)CCCCCC2)=O)cc1C 78751,C1(N=c2[nH]nc(C(F)F)s2)(NC(C2(C)CCC(C)(C(=O)OC(C)(C)C)C2)=O)CC1 78752,C(=O)(N=c1cc(C)n(C)[nH]1)C1OCCC(NC(CCCOCCC)=O)C1 78753,N1(C(CC2(OCC)CC2)=O)CCCC1C(C)(C)C(=O)NC1CC(F)C1 78754,c1(OCCOC)ccc(C(=O)NC2CCC(NC(=O)C(C)C(C)C)CC2)cc1 78755,C1(C(=O)NCC2CN(C(CSCCOC)=O)C2)CCc2cnnn2C1 78756,N1(C(COCC(C)C)=O)CC2C3CCC(C2C1)N(C(c1ncccc1CO)=O)C3 78757,Cc1cccc(C(=O)OCC(=O)N(C2CC2CNC(c2nn(C)cc2C)=O)C)c1 78758,C1(NC(c2n(CCOC)nnn2)c2ccncc2)CCc2ncccc2C1 78759,c1(CNC(C=NOC)=O)ccc(CC(C)NC(=O)C(CCN(C)C)N(C)C)cc1 78760,Cc1nsc(N)c1C(N1CSCC1C(=O)NCCSCCO)=O 78761,CCCC(C)C(=O)N1CC=CC1(C(=O)NC1CC(C)(C)C1)COC 78762,C(=O)(C1=NOC2(CCOC2)C1)N(CCN(C(c1cn(CC=C)nn1)=O)C)C 78763,Cc1nn(C)c(C)c1CC(N1CC(NC(c2cc(C(C)(C)C)n[nH]2)=O)C(C)C1)=O 78764,N#CC1CCCC(C(=O)NC2CC(C(=O)NC3CCOC3)C2)C1 78765,c1(N2CCC(CC=C)C2)cc(NCC(C)CC(C)C)nc(C(F)(F)F)n1 78766,CC1CC=C(C(=O)NC2COCC2NC(c2cccc3nccn23)=O)CC1 78767,C1(C)(C(C)C)CC1C(=O)N(CCCCN(C(=O)CCc1cn[nH]c1)C)C 78768,CC1(C)CC=C(C(=O)NCC(=O)NCC(=O)Nc2cc(CO)ccn2)CC1 78769,c1(OC)cc(C)c(Cl)cc1S(=O)(=O)N1CCN(C(c2cnc[nH]2)=O)C(C)C1 78770,CC1=C(C(=O)NCC2(NC(=O)CC3CCCN3C(C)C)CCOCC2)CCO1 78771,Cc1ccc2c(c1)C(=O)OC(C)(C(=O)NC(C)CNC(c1sc(C)nc1C)=O)C2 78772,c1(C(CC(=O)O)NC(C2NCCN(CC)C2)=O)cccc(-c2cscn2)c1 78773,N1(C(c2nc(CC)sc2)=O)CC2CC1CN2C1CCN(C(C)C(=O)OC)C1 78774,C=CC1(CC(=O)NC(C)C(C)NC(=O)CC2CSC2)CCCCC1 78775,C1(NC(C(CCOC)OC)=O)CCN(C(=O)Cn2nnnc2C(C)C)C(C)C1 78776,N1(C(c2cc(OC)n[nH]2)=O)CCC2CN(C(=O)CC3CCC=CCC3)CC2CC1 78777,N1(C(COC(C)C)=O)CCC(C)(C)C(NC(=O)COCC2(F)CC2)C1 78778,C1(C(=O)NC(CNC(c2cnn(C(C)C)c2C)=O)CCOC)(CC)CCNC1=O 78779,c1(C(=O)NC2CN(C(c3c(CC)cccc3)=O)CC2F)c(C)nn(CCO)c1C 78780,Cn1cnc(CCNC(=O)C(C2CC2)N(C(=O)CSCC(N)=O)CC2CC2)n1 78781,CCC(C(=O)N1CC(OCC(=O)NC2CCOC2)C1)OC 78782,N1(C(C2CC(=O)NCC2)=O)CC=C(C(=O)NC2CC3CCCCC23)CC1 78783,CC1(C)COCCC1C(N1CCC(CC(N)=O)(NC(C2(CO)CCC2)=O)CC1)=O 78784,C(CCC(F)(F)F)N(C(c1scc(C(C)=O)n1)=O)C 78785,C(=O)(CC(CC)C(C)(C)C)NCC(CC=C)NC(=O)CNS(=O)(=O)C1CC1 78786,c1(C(=O)NC2CCN(C(c3cc4ccnn4cn3)=O)C2)c(F)c(F)cc(F)c1F 78787,c1(-n2c(CC3(CC=C)CC3)nc(-c3ccccn3)n2)cccc2nc[nH]c12 78788,C(=O)(CC(C)(C)CNC(=O)Nc1cc(C(C)(C)C)ccn1)OCC 78789,C1(C(=O)NC(C(NOCC(=C)Cl)=O)c2ccnn2C)CC2(CCC2O)C1 78790,CC(CCCC(=O)NCC#CC#CCO)NC(C1(CCN(C)C)CC1)=O 78791,c1(C(C(=O)C(c2sccc2CO)N2CCCC2CN=[N+]=[N-])C)ccc(N)cc1 78792,c1(C(N(CCC)CCNC(C2CCC3CC3CC2)=O)=O)ccc2n[nH]cc2c1F 78793,c1(C(=O)NC(C)C(=O)NC2CC(CNC(=O)CCCF)C2)ccc([N+](=O)[O-])cc1 78794,C#CCCCCCCCC(=O)NCCN(C1CCCCC1)C(C1(C)CCCO1)=O 78795,CCCCCCCC(=O)NC(C(=O)N1CC(n2cnnn2)C1)C(C)(C)C 78796,C1(C(N(CCCCCNC(C2CC(NS(C)(=O)=O)C2)=O)C(C)C)=O)CCCS1(=O)=O 78797,c1(C(=O)NCC(n2cncn2)C)ccn(CCNC(=O)CCCc2ncco2)c1 78798,C1(C(=O)NC(C2(C(=O)NCC(C)(C)C)CC2)C)CCC2(CC2)C1 78799,N1(C(c2cc(C)c(Br)o2)=O)CC(NC(c2snnc2C)=O)CC(F)C1 78800,C(=O)(CCS(N)(=O)=O)N.CC1(CO)CCN(C(=O)CSCCN(C)CC)C1 78801,c1(CN2CCCC(CNC(c3cccc(OC)c3)=O)C2)cc([N+](=O)[O-])ccc1Cl 78802,C1(NC(=O)CC2COCC2O)C2CN(C(=O)CCCc3ccccn3)CC12 78803,C1(NC(=O)CNC(=O)C2CC2)CC2CCC1(C(=O)NCC1(F)CCC1)C2 78804,C1(N2C(=O)C2)CCN(C(C2CCOC2C(F)(F)F)=O)C1.C(C(C)C)SC 78805,C1(C(=O)NC2C=CC(CC(=O)NC3(c4nc(C)on4)CC3)C2)CCCN1C=O 78806,C1(CNC(CC2C(C)CCO2)=O)CCCCCN1C(c1csc(=N)[nH]1)=O 78807,N1(C(Cc2c(C)occ2)=O)CCOC(CCNC(=O)CC2COCCOC2)C1 78808,Cc1ccc(F)c(C(=O)N(C)CC2(O)CCN(C(=O)CCC3CC3(C)C)C2)c1F 78809,C1(C)(C(=O)NC(C2CCOCC2)CC)CCN(C(c2cc(CO)[nH]n2)=O)CC1 78810,C12(NC(c3snnc3C3CC3)=O)CCCC1CN(C(=O)Cc1ccsn1)C2 78811,C1(NCC(N2CCC(CC(=O)NCc3ccc(O)cc3)C2)=O)CCC2(CCC2)C1 78812,c1(C(N2CC(CC)N(C(C3CC4CC4C3)=O)CC2)=O)ccc2nccn2n1 78813,C1(CN(c2n(CC=C)c(-c3c(C)sc(C)c3Br)nn2)C)CSc2ccccc2O1 78814,N1(C(c2cc(CSCC)on2)=O)CC2C(NC(C3CCCC(C(C)C)O3)=O)C2C1 78815,CCC(CC)(C(C)C)NC(c1cc(CCNC(=O)C(C)=CC(C)(C)C)on1)=O 78816,c1(C(C)NC(CONC(Cc2scc(C)c2)=O)=O)ccc(F)cc1 78817,N1(C(c2c(C)[nH]cc2)=O)CC2C3CCC(C2C1)N(C(C1CC(C)CO1)=O)C3 78818,C1(OC)CC(N=c2[nH]c3c(c(=NCC(F)C4CCCCC4)[nH]2)SCC3)C1 78819,c1(OC)cc(F)c(C(N2CC(O)C(O)C2CNC(=O)C(O)CSC)=O)cc1OC 78820,C1(C(=O)NC2CN(C(C(C)OCCOC)=O)C2)CC2(CCCCC2)S1(=O)=O 78821,c1(C(=O)NC(C)(C)CNC(C2(C)CCCOC2)=O)cc2c(nn1)CCCC2 78822,N1(C(=O)CN2CCCC2)CCC(O)C(N=c2ccnc(Br)[nH]2)C1 78823,c1(C(=O)NC(CC(C)NC(c2ccc(C3CC3)cc2)=O)C)nnc(O)cc1O 78824,C(C)(C(C(=O)N(C1(CCO)CC1)C)C(C)C)NC(C(C(=O)OC)C)=O 78825,c1(CN(C)C)cc([N+](=O)[O-])cc(-c2ccccc2)c1O.C1(=O)NOCC12CC2 78826,C1(NC(COc2cccc(OCC)c2)=O)CCN(C(=O)CC2CC2)CC12CCC2 78827,c1(C(=O)NC2CC(C)N(C(=O)C#CC(C)(C)C)C2)cc2n(n1)CCCO2 78828,N#CC1(C(N2CC(NC(=O)C(N)=O)C(n3cccn3)C2)=O)CCSCC1 78829,Cc1onc(C2CCCCC2)c1C(=O)NCC1(NC(=O)CC(F)(F)F)CCCC1 78830,Cc1ccc(F)c(C(=O)NCC2(C)CC(NC(c3cnc4n3CCS4)=O)C2)c1F 78831,N1(C(C=CC2(C)COC2)=O)CC(C(=O)NCC2C3CCCCCC23)C(C)(C)C1 78832,CC(C)(CC=CC(=O)NC1CCCC1n1cccn1)NC(=O)CC1CCSC1 78833,c1(C(N2C(CC)CN(C(=O)C=C(C)Cl)CC2)=O)cccc2cc(Cl)ccc12 78834,C1(CC)CNC(=O)CN1C(C1(NC(C2CCCCNC2=O)=O)CCCC1)=O 78835,C1(NC(C(C)S(N)(=O)=O)=O)CS(=O)(=O)C12CCN(c1ccn3nccc3n1)CC2 78836,C1(C(=O)NC2CCC(CNC(CCC3C(C)(C)C3)=O)C2)CCc2n[nH]cc2C1 78837,c1(C(=O)NCC(CC)NC(C2(CC)CC(F)(F)C2)=O)cnc(S)n1C 78838,N#CC12CCCCC1(NC(=O)NC1CC1c1cc(Cl)ccc1F)C2 78839,CCCC(O)C(=O)N(C)CC1C2CN(C(=O)CCCCNC(N)=O)CC12 78840,C1(CCOC)(C(=O)NCC(O)CCNC(=O)Cc2ccn(C(C)C)n2)CCCC1 78841,c1(SCC(=O)NCC2CCCN2C(c2ncccc2Cl)=O)ccsc1[N+](=O)[O-] 78842,CC(CNC(C1(CCCF)CC1)=O)CC(=O)Nc1cccc(O)c1 78843,CN=c1[nH]c(=NCc2cncc(C)c2)[nH]c(=NC2CCN(c3cnccn3)C2)[nH]1 78844,Cc1cnc(C(=O)NCC2(CNC(=O)C(c3ccn(C)c3)C)CC2)cn1 78845,C1C(F)(F)C(=O)N1C.O(NC(=O)COC)CC(=O)OCC 78846,N1(C(c2ccccc2[N+](=O)[O-])=O)CC2CCN(C(C3CC3(Cl)Cl)=O)CC2C1 78847,C1(CNC(C=CSC)=O)CCC(C)(C)CN1C(c1sc(C)nc1C)=O 78848,C1(CC#C)CCCN1N(C)C(C)C1CCN(CCSC)C1 78849,C1(NC(CS(=O)(=O)NCC)=O)(CNC(c2ccoc2C)=O)Cc2ccccc2C1 78850,C12(C(N3CCC(OCCNC(CCCOCC)=O)C3)=O)CCCC1CC(=O)CC2 78851,c1(CNC2C(C(=O)NCc3ccc(C)cc3C)C2)cc(F)c(F)cc1O 78852,c1(C(N2C(CNC(C(CC)C)=O)CC(C)(C)C2)=O)ccc(S(N)(=O)=O)cc1F 78853,c1(OC)ccc(CNC(=NCC2CCCOC2)NCC2CCOC2)c(OC)c1 78854,CC1CCNCC1NC(=O)C(=O)NC(c1cccc(F)c1)c1ccccn1 78855,N1(C(C(=CC2CCCC2)C)=O)CCC2(C=C(C(=O)N3CCOCC3C(N)=O)C2)C1 78856,c1(C(C(N2CC(COC)(NC(c3nccnc3N)=O)C2)=O)O)ccc(F)c(Cl)c1 78857,C(CC(C)(C)CNC(=O)C(=O)NCc1ncc(C)o1)OC 78858,C(=O)(CC(C)C(C)(C)NC(=O)CC1CCC(=O)CC1)NCC(NOC)=O 78859,CC1CC2(CCCC2)CN1C(C1CCC(C2CC2)N1C(C1CCCN1C1CC1)=O)=O 78860,CC1CC(NC(=O)CCc2ccsc2Br)CCS1(=O)=O 78861,N1(C(C(C)(C)c2cscc2Cl)=O)CCN(C(=O)C(C)(C)C2CCOCC2)CC1 78862,C(CS(=O)(=O)Cc1cn(C2COCC2n2cccn2)nn1)CNC(c1onc(C)n1)CC 78863,C(C(C)C(F)C(=O)N(C)CCc1cccs1)NC(CCn1ncc(C)c1)=O 78864,C(=O)(C(C)(C)NC(=O)C=CC(C)(C)NC(c1cc[nH]c1)=O)OC 78865,c1(NC(C2N(C(Cc3cccc(C#C)c3)=O)CCC2C)=O)ccccc1C(=C)C 78866,C(=O)(CCCCC(C)=O)N1C(C)CC(C(N2CC(C(CC)C)C2)=O)C1 78867,N1(C(C(CC#CC)NC(=O)CC2=CCCC2)=O)CCCC(N=[N+]=[N-])C1 78868,c1(C(N(CCOCCNC(C(CSC)OC)=O)C)=O)c(C)cc(Cl)cc1C 78869,C(CCC(=O)N1CC(CC2CCCC2)C1)N(C(C(C)=C(C)C)=O)C 78870,CC1CN(C(c2ocnc2C(F)F)=O)CC(C)C1NC(=O)Cn1nnnc1C1CC1 78871,c1(NC)ccc(C(=O)NCC2CCCN2C(c2snnc2C2CC2)=O)nc1 78872,Cc1ncc(C(C)NC(c2cn(CCNC(=O)CC34CCCC3C4)cn2)=O)s1 78873,c1(C(N2CCC(NC(c3ccnnc3S)=O)C2)=O)cc(N2CCCC2)ccn1 78874,CCC(C)C(=O)NCC(=O)N(C(C)CCNC(=O)Cc1cc(C)no1)C 78875,N1(C(c2c(CC)c[nH]c2)=O)CC(N=[N+]=[N-])CC1C(=O)N(C)CC1CCCCO1 78876,Cc1cc(NC(C2(NC(C3CC3(Cl)Cl)=O)CCSC2)=O)cc(CO)c1 78877,N1(CC(C)(C)NC(C(C)=C(C)C)=O)CCN(C(=O)C(C)(C)N(C)C)CC1 78878,N1(C(CN(C(=O)C=CC2CCOC2)CCOC)=O)CC(CO)CC(C)(C)C1 78879,c1(N(C)Cc2nnc(C)s2)nc(N2CCn3nncc3C2)c2c(n1)CSC2 78880,C1(NC(CC2N(C(c3c(OC)cnnc3)=O)CC(O)C2)=O)CCN(C)CC1C#N 78881,N1(C(CNC(CCC(C)C)=O)=O)CC2CCCC1(CNC(=O)Cc1cnoc1)C2 78882,C1(F)(C(N2CCOCC(CNC(c3cnccc3Cl)=O)C2)=O)CC12CCCCC2 78883,CC1(C)CC(NC(=O)C=Cc2cncs2)CN(C(=O)COC(F)(F)F)C1 78884,Cc1cnc(CNC(=O)COCCNC(=O)CN2CCCC2=O)[nH]1 78885,Cc1cc(C(=O)NCCCN(C)C(c2cc(Br)c[nH]2)=O)c(Br)c(C)c1 78886,c1(C(=O)NC2CC3CN(C(CSC(C)C)=O)C(C2)C3)nc2cc(O)ccc2[nH]1 78887,C1(CCC)COCCN1C(=O)CC(C1CC1)NC(C1OC2CCC1C2)=O 78888,N1(C(C2C(=C)C2)=O)CC2OCCN(C(c3cnn(CCOC)c3C)=O)C2C1 78889,Cc1csc2cc(C(=O)NCC(C)NC(c3csc4nccn34)=O)[nH]c12 78890,CC1(C)C(NC(=O)C=Cc2cncs2)CCN1C(C1CC2CC2C1)=O 78891,c1(C(=O)NC2CC(F)(CNC(CC(CC)SC)=O)C2)ccc2c(c1)CC(C)O2 78892,C#Cc1cccc(C(N2CC3(CCN3C(=O)CCc3cc(OC)no3)C2)=O)c1 78893,c1(C(=O)NC23CC(NC(C4C(C)(CC)C4)=O)(C2)C3)cnc2ncc(Cl)cn12 78894,C1(C(C)(C)C)CC(F)CN(Cc2ccccc2C(N2CCC(CO)C(O)C2)=O)C1 78895,c1(C(=O)NCC=CCC(=O)NCc2cc(OC)no2)ncc(N)cc1C 78896,c1(OCC)cc(CNCCS(N)(=O)=O)ccc1OC(C1CC1N)=O 78897,C1(O)(CNC(C2(CCC)CC2)=O)CCCN(C(C23CCC(C)(C2)OC3)=O)C1 78898,C(=O)(CCCC(F)(F)F)N(CC(F)F)C(=O)N(CCSCC(=O)OC)C(C)C 78899,N1(C(CC2CCC(C)CO2)=O)CC(NC(c2nccc(C(F)F)n2)=O)CC(F)C1 78900,CCC(O)C(C)C(=O)N1CCC(CC)(NC(=O)CSc2nncn2C)CC1 78901,c1(C(=O)NC2C(CNC(Cc3n(C(C)C)cnn3)=O)C2)cc(F)ccc1N 78902,c1(SC)cc(=NC(=O)C(C)C(C)NC(=O)C(C)OC(C)=O)[nH]n1C 78903,CC1(C)C2CCC(C(=O)NC3C4CN(C(c5ccc(C(F)F)nc5)=O)CC34)C1C2 78904,C1(c2ncc(CCC(=O)OC)o2)CN(N2CCCC3(COCCO3)C2)C1 78905,Cc1ncc2n1CC(C(N1CCCC(C)(C)C1CO)=O)CC2 78906,C(=O)(CCCCC(F)(F)F)NCCCN(C)C(c1nccc2ncncc12)=O 78907,CC1CCCCC1(CNC(c1ccsn1)=O)NC(C12CCCC1CCC2)=O 78908,C1(C(=O)NC(c2cnn[nH]2)C)COCCN(C(c2ocnc2C(C)C)=O)C1 78909,c1(C(=O)NC23CCN(C(c4c(CC)noc4)=O)CC2C3)ccc2nc(C)cn2c1 78910,CC1=CCC(C(=O)NCC(C)(C)NC(C2CCCN(C(=O)OC(C)(C)C)C2)=O)CC1 78911,N1Cc2ccc(Cl)nc2C1.Cc1nccn1CCC(=O)N(CCO)CCN(C)C 78912,N1(C(C2C(=C)C2C(=O)OC)=O)CC2CN(C(c3cnn4ccsc34)=O)CC(C1)O2 78913,C1(CNC(CN(C(CCCOCCC)=O)CCOC)=O)CC2(C1)CC2(F)F 78914,c1(Cn2cc(CCN(C(=O)C(O)c3ccsc3)C)nn2)cccc(Cl)c1Cl 78915,C(=O)(C(CC(=O)NC(C)(C)C)Cc1ccc(OC(F)(F)F)cc1)OC(C1CCC1)C 78916,Cc1c(N)cc(C(N2CCC(CCNC(=O)C(C)CC(C)(C)C)CC2)=O)cc1N 78917,Cc1cc(NC(c2ccccc2O)=O)sc1C(=O)NC1CONC1=O 78918,C1(NC(C(CC)N2CCCC2=O)=O)CN(C(=O)CN(C(=O)COC)C)CCC1F 78919,C(=O)(C1=NNC(=O)CC1)NCC(C)N(C(=O)CCC1CCCO1)CC 78920,C1(CC)CN(C(=O)CCc2ccccc2OC)CCN1Cc1c(C)noc1C 78921,C(c1ccc(Br)cc1)=CCC(=O)NCC(CNC(C(C)C1CC1)=O)CO 78922,N1(C(C(CCCC)O)=O)CC2CCCC2(CNC(c2ncc(F)c(OC)n2)=O)C1 78923,C1(NC(c2c(CC)n(C)nn2)=O)CCCCCC1NC(=O)CCCn1ccnn1 78924,N1(C(CCCC#C)=O)CCCC(C(=O)NC(c2ccccc2F)CO)CC1 78925,c1(C(=O)NC(C(=O)NCCN(CCCC)C)CC(F)F)c[nH]c2ccccc12 78926,C(C)(CCCNC(=O)NC1CC(N2CCOCC2)C1)(OC)OC 78927,C1(CC)(CNC(c2cc(I)cs2)c2nnnn2C)CCCO1 78928,CC(C)C(N=[N+]=[N-])C(=O)NC(C)(C)C(=O)NC1CC(CO)C12CCC2 78929,C1(NC(C(C)(C)F)=O)CC2(C1)CN(C(C1(Cc3cnn[nH]3)CCCC1)=O)C2 78930,C1(C(N2CC3CC2CCC3NC(C23CC(F)(C2)C3)=O)=O)CC2CCC(C1)S2(=O)=O 78931,Cc1ncc(NC(C2CCN2C(c2cc(Br)cnc2F)=O)=O)c(C)n1 78932,C1(O)(CN(C(c2ccc(COC)s2)=O)C)CCN(C(=O)C2=COCCC2)CC1 78933,C1(C(N2CCC(CCNC(c3cscn3)=O)CC2)=O)CC1C1CC(F)(F)C1 78934,C(=O)(C(F)C(C)CNC(=O)C(C)OCC=C)NCCSCC#C 78935,c1(C(C)C)ccc(C(N2CC(NC(=O)CC(C)c3cccnc3)C(O)C2)=O)nc1 78936,N1(C(c2c(C)snn2)=O)CC2ON=C(CNC(=O)CNC(=O)OC(C)(C)C)C2C1 78937,c1(NC(c2n(CC(=C)C)nnn2)c2cnc(C(C)(C)C)[nH]2)cc(C)cnc1OC 78938,C1(C(=O)NC(c2nc(=O)o[nH]2)C)CC2(CCN1C(C1CC(=O)C1(C)C)=O)CC2 78939,Cc1nc(C=CC(=O)N(C)CC2CCCN2C(=O)C(C)SC(C)C)[nH]c1C 78940,C1(CC)CN(C(c2cc(Cl)n(C)n2)=O)CCN1C(=O)Cc1ncc(C)s1 78941,c1(SC(C)CCN2C(=O)NC(C)C2=O)c[nH]c2ncccc12 78942,c1(CN2C(C(=O)Nc3cnn(C(F)F)c3)CC3CC32)cc(Cl)c(Cl)c(Cl)c1 78943,N1(C(C(CC)C2CCOCC2)=O)CCN(C(C2(C)COC2)=O)C(C)C1 78944,c1(-c2ccn(CC)n2)n[nH]c2cccc(C(=O)Nc3ncc(F)cc3F)c12 78945,CCC1=NOC(C(=O)NC(C2CCCN2C(=O)C2CC2)(C)C)C1 78946,Cc1cc(C(=O)NC(c2ccc(N(C)C)cc2)CNC(=O)C(C)O)ncn1 78947,N1(C(C2CCC(F)(F)C2)C(=O)NCC(C)C)CCN(c2cnccn2)CC1C 78948,CC(C)CCC(C)NC(=O)C(C)NC(=O)C=CC(F)(F)F 78949,O=C(O)CC(C(=O)NC1CCC(c2nc[nH]n2)CC1)C1CC1 78950,C(=O)(CCCCN=[N+]=[N-])NCCCN(C)C(C1(C)C=CCC1)=O 78951,O=C1CCC2(CCCN(Cc3cccc4ccc(C(F)(F)F)cc34)C2)CN1 78952,C1(C(N2CC(CCCCNC(=O)CCc3ncc[nH]3)C2)=O)Cc2ccccc2O1 78953,CC1CN(C(C23CC(CC(F)F)(C2)C3)=O)C(C)CN1C(c1cc(Cl)c(Cl)[nH]1)=O 78954,C12CN(CCC1C)C(=O)C1C(Cl)(C1)N(CCC(F)(F)F)C(=O)C2.C(C)(=O)SC 78955,C12(CNC(c3ccccc3)C(=O)NCCC#C)CCC(CC1)C2 78956,C(C(N=[N+]=[N-])C(=O)NCC1CCCN(C(=O)CCN2CCN(C)CC2)C1)OCC 78957,c1(C(C(=O)N(CCNC(C2CC3(CC3)C2)=O)C2CC2)(F)F)cccc(F)c1F 78958,Cc1cc(C)c(C(=O)NC2C=CCCC2)cc1O 78959,C1(OC)(OC)CC(C2CCN(c3nnc(-c4ncccc4F)n3C3CC3)C2)C1 78960,c1(C(N2CCCC2)=O)ccc(-c2ncno2)cc1.CCCN 78961,Cn1[nH]cnc1=NC(=O)NC1CCN(Cc2ccc(OC(F)(F)F)cc2)C1 78962,C1(CNC(CCCCC=CC)=O)CN(C(=O)C=C(Cl)Cl)CCC12CCC2 78963,N1(C(c2c(C)n(C3CC3)cc2)=O)CCC(C2CCN(C(=O)CSS(C)(=O)=O)C2)C1 78964,O=C(CC1=CCOCC1)N1CC(N2CCN(C(C3CCCC4(CCC4)C3)=O)CC2)C1 78965,C1(ONC(=O)C2CCCO2)COC2(CCN(CC3CC(=C)C3)CC2)C1 78966,C12(C(N(CC(CC)O)CC)=O)COCC1CN(C(=O)CCc1ccncc1)C2 78967,C1(C(=O)NCC(CC)NC(c2snc(C)c2N)=O)CC2CC1C1C2C1(F)F 78968,N1(C(COC)=O)CCN(C(C2CCCC2(F)F)=O)CC(C)(C)C1 78969,N1(C(=O)Nc2c(OC)ccc(-c3cnco3)c2)CC(F)(CO)C2(CCC2)C1 78970,c1(CC)cccc(C(=O)NCC(C)(C)NC(c2cc(C3CC3C)on2)=O)c1 78971,CC1CC(C)CN(C(=O)CN2CCCC2C(C)(C)CN(C)C)C1 78972,CN(C)NC(=O)CCC(=O)NC1CC2(C(=O)NC3CC3(C)C(F)F)COC1C2 78973,N1(C(CCc2ccc(C)cc2)=O)CCN(C(=O)C(F)C2CCCC2)C2CC12 78974,N1(C(C(C2CC2)OC)C(=O)NC2CCOCC2)CCn2c(C(F)(F)F)nnc2C1 78975,C1(CNC(C2CCC(C)O2)=O)C2CN(C(=O)CCNC(N)=O)CC12 78976,C1(CNC(C(C)NC(C)=O)=O)CC2COCC2N1C(c1cncn1C(C)C)=O 78977,c1(C(=O)NC2CN(C(C(CC)COC)=O)CC2C2CC2)cc2cc(F)ccc2[nH]1 78978,N1(C(C2(CC)CCC2)=O)CCC2(CCN(c3ccc(C#N)nc3)C2)C1 78979,c1(C(=O)NCC2(C)CCCN(C(COC(CC)C)=O)C2)cc(S(=O)(=O)NC)cs1 78980,N1(C(C2(C(=O)OCC)C=CCC2)=O)CCN(C(=O)CNc2ncccn2)CC1 78981,N1(C(c2c(C)cco2)=O)CC2CC2(CNC(c2sccc2-n2cccc2)=O)C1 78982,c1(NC(=O)Nc2ncc(C(N)=O)s2)nccc(-n2ccnc2)n1 78983,c1(C(=O)NC(C(CO)NC(C(C)Oc2cccnc2)=O)C)sc2ncccc2c1Cl 78984,n1(C2CN(C(C3CN(C4C(C)C4)C(=O)C3)=O)C2)c(O)nc2ccccc12 78985,CCCCC(F)C(=O)N1CCC(CC(C)NC(=O)C(C)N2CC(C)C2)CC1 78986,C(CCF)(C(=O)N(C)CCC1CCCN1C)NC(C1CC(OCC)C1)=O 78987,CC1(CNC(c2cscn2)=O)CCN(C(C2(C)CCCNC2)=O)C1 78988,c1(CC)cc(CC(=O)NCCC(=O)N(CC(C)OC)C(C)C)on1 78989,C1(NC(C(CC=C)C)=O)(CNC(c2cc(C)nc(OC)n2)=O)CCCCC1C 78990,C(=O)(CC(C)CC(F)(F)F)NC1CCC(C)N(C(C2(O)CCCC(C)(C)C2)=O)C1 78991,C(CC(C)C(=O)NCCC(O)CNC(C1(CCN2CCCCC2)CC1)=O)=CC 78992,S(=O)(=O)(c1ccccc1F)NCCC(N1C(c2ccc(C)cc2)CC1)=O 78993,C1(NC(C=CCC)=O)CC(OC)C12CCN(C(C1CCC=CCCC1)=O)CC2 78994,c1(C(=O)NCC(CNC(C2C(C#N)C2)=O)CO)ccc(OCC2CC2)nc1 78995,C1(CNC(CN(C(C)=O)C)=O)CCCC(NC(c2ccc(OCCO)cc2)=O)C1 78996,c1(OCC)ccc(Br)cc1CN1CCC(NC(c2cc(CC)[nH]n2)=O)C(O)C1 78997,N1(C(C2(CNC(C3C(CC(C)(C)C)C3)=O)CC=CC2)=O)CC2(CCCC2)C1 78998,C1(NC(C(c2ccc(Cl)cc2)(C)O)=O)CN(C(=O)COCC(F)F)CC2(CC2)C1 78999,C12(NC(C(C)CC(N)=O)=O)CCC(CNC(c3cccnc3O)=O)(CC1)OC2 79000,c1(C(=O)NCCCCCNC(C2C(C=C)C2)=O)cc(=NS(C)(=O)=O)cc[nH]1 79001,c1(CNC(c2ccc[nH]2)=O)c[nH]nc1C(=O)NCCC1CCOC1 79002,Cc1ncccc1C(N1CC(NC(=O)COC2CCN(C)CC2)C(C(F)F)C1)=O 79003,c1(C(=O)NC(C2CN(C(c3ccccc3C(F)F)=O)C2)C)nc(=O)n(C)[nH]1 79004,C(CCC(C)C(=O)NC(C)C(C)(C)C(=O)NCc1cc(C)sc1C)OC 79005,c1(OCC)ncc(C(=O)NCC2CCN(C(C3CC(O)CN3C)=O)C2)cc1Cl 79006,N1(C(CCN(CCC)C)=O)CC2CC(NC(=O)C=Cc3ccncn3)CC1C2 79007,C(C(C)(C)C1=CCCC1)NC(C1C2N(C(C(CN(C)C)N(C)C)=O)C(CC2)C1)=O 79008,N1(C(Cn2ncc(C)c2)=O)CC2CCC(NC(=O)CCS(C)=O)CC1C2 79009,c1(C(N2CC(O)(C(C)NC(C3CN(C)C3)=O)C2)=O)ccc2[nH]c(=N)oc2c1 79010,C1(CC)(CC)CC(NC(=O)Cc2nocc2C)CN1C(c1ncn2c1CCC2)=O 79011,c1(OC)cncc(C(=O)NCC2CC2NC(C2CC(n3cnnc3)C2)=O)c1 79012,n1(CC(=O)NCC2N(C(C(CO)N(C)C)=O)CCC2)nnc2ccccc12 79013,CC1CNc2ccc(C(=O)N(C(C)CCNC(=O)C=CC(C)(C)C)C)cc21 79014,CC(=O)CCCC(C)C(=O)NC1(C(N2CCCC2CC(C)O)=O)CC(O)C1 79015,c1(CNC(CC(CC)N(C(C(CCC)OCC)=O)C)=O)cccc(F)c1F 79016,N1(C(CSc2n(C)cnn2)=O)CC(NC(=O)CCONC2CCC2)CC1CO.N 79017,c1(CN(C(C(C2CCCC2)NC(C2CC(=C)C2)=O)=O)C)cccnn1 79018,C1(C(C(=O)NCC(C)N(C)C)(C)C)CCCN(C(=O)CC(=O)NC2CC2)C1 79019,C1(CNC(c2cn(C)nc2)=O)CCC2(CO1)CC(NC(=O)C=Cc1ccco1)C2 79020,CC1CCc2nc(N3CCC(CO)C3)[nH]c(=NCc3ccc(S(N)(=O)=O)s3)c2C1 79021,N1(C(C2COCCN2C(=O)C(F)F)=O)Cc2cccc(O)c2C1 79022,C=CCC(CNC(=O)C(CC)C(=O)OC)C(=O)NC(C)CN(C)C 79023,C1(NC(CCC(C)NC(=O)CN2CCC(F)CC2)=O)CCC(O)C(O)C1 79024,C1(C(=O)NC(C(=O)OC)Cc2cn(CC(C)(C)C)nn2)CCn2cncc2C1 79025,Cc1cnccc1CCNC(N1CCCC1Cc1cnn(C)c1N)=O 79026,C1(NC(CS(CC)(=O)=O)=O)CN(C(c2conc2C)=O)Cc2ccnn2C1 79027,c1(OC)ccc2c(N3CCCN(C(c4cc(C)ccc4Cl)=O)CC3)ncnc2c1 79028,CC1(C(=O)NC2CC2NC(C2(CC3CC3)CCOCC2)=O)CCCCO1 79029,c1(CC(N2C(C)(CNC(=O)C3=NOCC3)CCC2)=O)cc(F)cc(F)c1 79030,CC1(C)Oc2ccsc2C(NC(=O)COc2ccc(F)c(CN)c2)C1O 79031,c1(C(N2CC(C(=O)NCCCCCCO)OCC2)=O)c(I)ccnc1F 79032,c1(CC)c(C(=O)N(C2CCCN(C(=O)CC(C)(C)OC)C2)CCO)cccc1F 79033,C(=O)(C#CC1CCC1)NCC1(C)CCN(C(=O)CCC(=O)c2ccccc2)C1 79034,N1(CC(C)(C)NC(=O)COCCF)CCN(C(=O)C(C)(F)c2ccccc2)CC1 79035,C1(CCCNC(C2CC(OC)C2)=O)CCN(C(=O)Cc2nnc(C)o2)CC1 79036,Cc1cnc(C(=O)NCC2(F)CC(NC(C3CC3C(F)F)=O)C2)nc1 79037,C(=O)(CC(C)(C)CNC(=O)CCCC1CC1C)NCC1(OC)CCOC1 79038,Cc1ccc(CNC(C2CCC(NC(c3ccccc3Br)=O)C2)=O)c(C)c1 79039,N1(C(C)=O)CC2(CC2)CC1C(=O)Nc1ccc(SCCCO)cc1 79040,C1(N(C(c2c(CC)c[nH]n2)=O)C)CCN(C(c2cn(C)nn2)=O)CC12CC2 79041,CS(=O)(=O)c1ccc(F)c(C(N2CCCN(C(=O)C3=CCCC3)C(CO)C2)=O)c1 79042,C1(C)(C(=O)NCC(CNC(C(CC)(C)CC)=O)(C)O)CCCNS1(=O)=O 79043,c1(C(=O)NCCN(C(c2ccnc(O)c2)=O)CC2CC2)c(F)ccc2[nH]ccc12 79044,CN1CCOC(C(=O)NCC2CN(C(=O)CCc3ncc[nH]3)CC2(F)F)C1=O 79045,c1(CC(=O)NC2CN(C(=O)CC3CCCCC3O)C2)ccc(O)cc1Cl 79046,C1(C)(CNC(C(COC(C)C)(C)C)=O)CCCN(C(C2C3C4CCC(C4)C23)=O)C1 79047,c1(NC(c2c(NCc3c(C)c(Cl)ccc3)cnc(Cl)c2)=O)c(Br)ccc(F)c1F 79048,CC1(CC(=O)NC2CCCCC2CNC(=O)C=Cc2cc[nH]n2)CCCCCC1 79049,c1(SC)ncc(C(F)(F)F)c(N(C(C23CC(N)(C2)C3)=O)Cc2ncccn2)n1 79050,N1(C(c2ncn(C)n2)=O)CCCC(NC(=O)Cn2cnc([N+](=O)[O-])n2)C(F)C1 79051,C(C=CC(N1CC(C(C)NC(=O)CNc2nccs2)C1)=O)(CC)=CC 79052,Nc1cc(Cl)ncc1C(=O)NC1CC2CCC1(CNC(=O)Cn1ncnn1)C2 79053,C1(CN(C)C(c2nncs2)=O)COCCN1C(c1c[nH]nc1C1CCOC1)=O 79054,CC(CS(C)(=O)=O)C(=O)NC1CC(CNC(c2ccc(-c3cc[nH]n3)s2)=O)C1 79055,Cc1ccccc1CC(N1CC(NC(c2ncoc2-c2ccon2)=O)C(C)C1)=O 79056,c1(C(N2CC(C)(NC(C(C)OC3CCCC3)=O)C2)=O)ccnc(CC(F)(F)F)n1 79057,O=C(C1=CS(=O)CCC1)NC1CC2CC1N(C(c1cncc3[nH]ccc13)=O)C2 79058,N12CCc3nc(cn3CC1)C2=O.N1(CCNCc2cc(C)on2)CCCCC1=O 79059,CC1(O)CCN(C(C2CCCCC2NC(C2CCCC(C#N)C2)=O)=O)CC1O 79060,C1(CNC(C(CC)C#N)=O)CC2CCCC2N1C(c1ccccc1F)=O 79061,C1(C#N)(C(=O)N(CC)CC)CCN(CC(CO)CO)CC1 79062,c1(CNC(CC2(CC(=O)OC)CC2)=O)ccoc1NC1CC1C(=O)OC 79063,N1(C(C2N(CC)CCC2)=O)CCC(O)CC1C(=O)NC1C2C=CC(C2)C1CO 79064,c1(C(=O)NC(C(=O)N(CCOCCOC)C)CO)ccc(=O)n(C)c1 79065,C(=O)(C1=CCCCCC1)NC(C(=O)NCC(C)O)CN(C)C 79066,C1(C)(C(N2C(CNC(c3ccc(CC)[nH]3)=O)CC2)=O)CCCCCC1 79067,C(c1ccc(C2CC2C)o1)=CC(=O)NCC=CCNC(COC1(C#C)COC1)=O 79068,Cc1cc(C(N2CCC(O)(CNC(c3coc(C(C)C)n3)=O)CC2)=O)cc(O)c1 79069,c1(C(=O)NC2C=CC(CC(=O)NCCCN(C)C)C2)cc(O)cc(F)c1 79070,C1(C=C)(C(=O)NCC(CC=C)NC(c2cc(Cl)ccc2N)=O)CCCCC1 79071,N1(C(C(n2cc(C3(N4CCCC4)CC3)nn2)C)=O)CC(c2ccccc2)C1(C)C 79072,C1(NC(C2C(C)(C(F)F)C2)=O)C=CCC(C(=O)NCc2ncoc2C2CCC2)C1 79073,N1(C(C2(C)CCCCO2)=O)CCOCC(NC(c2c[nH]nc2-c2cccs2)=O)C1 79074,n1(C(C)C)ncc2c(NCCCCC#N)[nH]c(=NCC(C)=C3CC3)nc12 79075,C#CC12CCN(C1)C(=O)OC1CCN(C1)C2=O.C1(C(=O)NC)CN(C2CCC2)C1 79076,Cc1onc(Br)c1C(N1CCC(C(C)NC(c2cccnc2O)=O)C1)=O 79077,CC(C)C(F)(CNC(C1(C)CCCC1O)=O)C(=O)NC12CC1COC2(C)C 79078,c1(C(N2C(CNC(c3c(CC)con3)=O)C=CC2)=O)ccc(C(F)F)c(F)c1 79079,C(CC(O)CC(=O)NC1CC(N(C(=O)CC(C)O)C)C1)SC 79080,c1(N2CCC(CC=C)(NC(C3CC4CCCC34)=O)C2)ncnc(Cl)c1C#N 79081,C1(NC(C2C3CN(C(c4cn(CC)nc4C)=O)CC32)=O)CC2(CCC2)C1OC 79082,CC(C)C(CNC(C1CCC2(CC1)CC2)=O)C(=O)NCC(C)Cc1cn[nH]c1 79083,CCCN=C(NCc1cc(C)cc(Cl)c1)N1CCN(c2ccccc2F)C(=O)C1 79084,CC(C)(C(C#N)OC(c1ccc(C2(C#N)CC2)cc1)=O)c1ccc(F)cc1 79085,c1(C(=O)NCCC(C)NC(CC(C=C)C)=O)ccc(NCCO)c([N+](=O)[O-])c1 79086,c1(OC)cccc(C(N2CCC2(C)C(=O)NCC2CCN(C)CC2)=O)c1O 79087,n1(CC(=O)NCCCN(C(CC(=O)NCC)=O)C2CCCC2)nc(C)ccc1=O 79088,C(=O)(C1=CCCCC1)N(CC(O)CNC(C1CC12CC2)=O)C 79089,C1(CNC(C(C)OC)=O)CN(C(c2cncc(C(=O)N(C)C)c2)=O)CC(C)(C)O1 79090,N1(C(C(C(CC)O)C)=O)CC2CCC(C1)N2C(=O)CN(C)S(N)(=O)=O.C1COS1 79091,C1(CCC)CN(C(=O)CC2CCC(C)(C)C2)CCN1C(=O)C(=O)C(C)(C)C 79092,CC(CC1CCCC1)C(C(=O)NC1(C)CC1)N1CCC(C)(c2ccccc2)CC1 79093,CCC(C)(O)C(=O)NN1CCCC1C(=O)N(CCC1CCCC1C(=O)O)CC 79094,N1(C(c2cc(OC)no2)=O)CC(NC(c2ccc(CCC#N)cc2)=O)C(C)(C)C1 79095,C(=O)(CC(C)n1cccn1)NCC(C)N(C(COCCSC)=O)C 79096,c1(C(=O)NCCCCCN(C(C2C(C(C)C)C2)=O)C)cc2cccc(Cl)c2s1 79097,c1(CC(N2C(CNC(CC(C)(C)O)=O)CCCC2)=O)c(Cl)cccc1Cl 79098,CC(CN(C(=O)C(N1CCC(c2cccc(Br)c2)CC1)=O)C)C(F)(F)F 79099,N1(C(c2c(C)onc2)=O)CCC2(CCC2)C(NC(C2CC3CC2C3)=O)C1 79100,C1(NC(=O)CSc2nncs2)CC2CC1N(C(c1ccc(O)nc1Cl)=O)C2 79101,CC1(C)CCC2(CC1)CC2C(=O)NCC1CCN1C(=O)CCc1nccs1 79102,c1(C(=O)NCCC(C)N(C)C(c2ccc(CO)c(F)c2)=O)cc2cn[nH]c2cn1 79103,C(CCC(O)C(=O)Nc1cccc(F)c1C)NC(C1C(=C)C1C(=O)OC)=O 79104,C1(C#N)(C(N2CC(CNC(c3ccc(COC)cc3)=O)C2)=O)C(C#N)C1(C)C 79105,C(C(C(=O)N1CCOC(COC)C1)C(C)(C)C)NC(C(C=C=C)C)=O 79106,c1(C(N(C2CCN(C(c3sc(C)nc3C)=O)C2)CC)=O)cccc(C(C)(F)F)c1 79107,C1(C)(CNC(Cc2cccc(OCC)n2)=O)CCCN(C(C2OCC2(C)C)=O)C1 79108,N1(C(c2n(CC)ncc2)=O)CC(CNC(=O)C(F)(F)C(O)C2CC2)CC1(C)C 79109,N1(C(c2nc(C)sc2)=O)CC2CCCC2(NC(=O)CN2CCC(=O)NC2=O)C1 79110,N1(C(Cc2c(C)ncs2)=O)CCC(C(N2CCN(C)CC2C)=O)C12CCC2 79111,N1(CC)CC(CNC(=O)C(c2ccccc2)NC(c2cnccc2C)=O)CC1=O 79112,CCCC(CC(=O)NCCC(=O)NC)NC1OCCCC1(C)C 79113,Cc1c(C(=O)NCC2CC2NC(c2cccc(CO)n2)=O)cncc1N 79114,C1(CC(=O)NC2CN(C(c3c(C)oc(C(C)C)c3)=O)C(C)C2)CCCC(C#N)C1 79115,C(CC(C(=O)NC1CCOC1CC)NC(c1oc(C)nc1CC)=O)OCC 79116,Cc1cc(C(N2CCN(C(c3nc(C(C)C)oc3C)=O)CC2)=O)c2occc2c1 79117,C(=O)(CC1OC(=O)c2ccccc21)N(C(C1CC1c1c(C)ccc(F)c1)=O)CCF 79118,CC(C)C(O)C(=O)NCC1CN(C(c2ccnc(-c3ccccc3)n2)=O)C1 79119,C(=O)(CC(CNC(c1ccccc1Cl)=O)C1CCC1)NCC1(CO)C(C=C)C1 79120,c1(-c2cn(C3CCCC(NC(C(COC)OC)=O)C3)nn2)cccc(Cl)c1F 79121,C1(NC(c2n(CC)cc(Cl)c2)=O)CCC(O)CN(C(=O)C(C)O)C1 79122,C1(CNC(c2ncc(C)nc2)=O)CN(C(C2CC3(C2)CC3F)=O)C(C)(C)C1 79123,C1(C(=O)NCC(CNC(c2cnc(NC(C)=O)o2)=O)(C)O)CC12CCCCC2 79124,CON(Cc1ccc(C)o1)C(=O)C1(NC(=O)C(n2nccc2C)C)CC1 79125,N1(C(c2n(CC#C)cnn2)=O)CCOCCC1C(=O)NC1CCCCC1(C)C 79126,C(C(CNC(c1ncnc(C)c1C)=O)C(F)(F)F)NC(c1c(C)coc1)=O 79127,N1(C(Cc2cccc(CC)c2)=O)CCN(C(=O)C(C)CF)CC(C)(C)C1 79128,c12ccc(cc1Cl)o2.c1(C(=O)OC)cnc(C2(NC3C(OC(C)(C)C)C3)CC2)o1.CN 79129,Cc1cc(Br)ccc1C(N1CCC(CN(C)C(c2cccc(Cl)c2F)=O)CC1)=O 79130,c1(C(=O)NC2C(NC(=O)CC3C=CCCC3)CC2)cnc2ccccc2n1 79131,CC1(C)CC2CN(C(=O)C(=O)NCC3CCC(N)CC3)CC12 79132,C1(CC(=O)NCC(=C)CCNC(=O)C(C)c2cccs2)(CO)CCCCC1 79133,C=CCC(CC=C)NC(C1CCOCC1NC(=O)CC(C)F)=O 79134,c1(C(N2CCC(CCNC(CN(C(C)=O)C)=O)CC2)=O)cc(N)c(Cl)c(O)c1 79135,c1(C(N2C(C3CCN(C(COCC)=O)CC3)C(C)(C)C2)=O)cc(N)cc(C#C)c1 79136,CC(=O)CCCCC(=O)N1CCC(C(=O)NCc2ncccc2F)(CF)C1 79137,N1(C(c2c(N)non2)=O)CCCC2(CCCN2C(C2C3CCCOC23)=O)C1 79138,C(N=c1[nH]c2ccc(Cl)cc2s1)C1C(C)CN(C(=O)CC2(O)CCCCC2)CC1 79139,c1(CC(=O)NCC23CN(C(C(C)CO)=O)C(CC2)C3)cn2cc(Cl)cc(Cl)c2n1 79140,c1(CC)ccc(C)cc1NC1(c2nnnn2C(C)C(=O)OC)CC2(CSC2)C1 79141,CCCCCCCCC(=O)N1CCCOC(CNC(C2CCC(O)C2)=O)C1 79142,CCC(C)(CC)C(=O)NCCCN(CCCNC(C1CCC(=O)NC1)=O)C 79143,CC1(C)COCC1CNC(c1ccc(CNC(C2CCC(=O)N2)=O)s1)=O 79144,C=CCC(CC=C)C(=O)NCC1CC2COCC2N1C(c1cc(C#N)on1)=O 79145,CC(C)(CC(=O)NC12CCCC1CN(C(=O)COCC(F)F)C2)CC(F)F 79146,C#CCC(CC(F)F)C(=O)N1CCC(CC)C1C(=O)NOCCC(C)O 79147,c1(C(=O)NC2CCN(C(C(C)OCC)=O)C2C)nc(S(N)(=O)=O)c2ccccn12 79148,CN1CCN(C(C2CN(C(=O)C=Cc3cocn3)CCN2C)=O)C(CO)C1 79149,c1(OC)cccc(Cl)c1CN1CC(CO)(NC(c2cccnc2C(F)(F)F)=O)C1 79150,CC1=C(C(=O)NC2CC(C)N(C(=O)CCCn3ccnc3)C2)CCC(C)(C)C1 79151,C1(NC(=O)Cc2sc(O)nc2O)CCCC12CN(C(C1CCC(C(F)F)O1)=O)C2 79152,C(CCF)(C(=O)NOCC(O)C(C)C)NC(CCCCCOC)=O 79153,Cc1cc(Br)c(N(C)C(C2CCN(c3cccc(Br)c3)C2)=O)c(Br)c1 79154,C1(NC(CS(CC)=O)=O)CCS(=O)(=O)C2(C1)CC(CNC(=O)C=C(C)C)C2 79155,c1(C(N2CC3(CCN(C(C)=O)C3)C2)=O)cc2c(nc1O)CCCC2 79156,CC(CC(F)(F)F)C(=O)N1CC(N(C(=O)CCn2cccnc2=O)C)C(O)C1 79157,C(CC(C)(C)C)(C(=O)NCC1(F)CC(O)C1)NC(C1=CCCC1C)=O 79158,c1(NCCOCCNC(=O)CCC(F)F)ncnc2sc(C(F)(F)F)nc12 79159,N1(C(c2c(C(C)(C)C)[nH]cn2)=O)CC2CCC(CNC(C3CC4CCC3C4)=O)C2C1 79160,c1(N2CCC(CCOC)(NC(C3CCC(C)C3)=O)C2)nccc(S(C)(=O)=O)n1 79161,n1(CCC(=O)NCCN(C(=O)C(C)O)CCOC)c(C)csc1=O 79162,CON=Cc1ccc(C(=O)N(CCCn2cc(C(O)C(C)(C)C)nn2)C)cc1 79163,N1(C(C=CC(C)NC(C(CC(C)C)C(C)C)=O)=O)CCc2ccc(C#N)cc21 79164,N1(CC(=O)N(C(C)C)CC)CCCC(c2nn(C)cc2C(=O)O)C1 79165,C1(C2(C(N(CCOC(C)=O)C)=O)CC2)CCCN1C(=O)CCn1ccnc1 79166,C(C(CC)(CC)C(=O)NCC1C=CCCC1)NC(CCSCCCC)=O 79167,c1(C(=O)NC(C(C)NC(=O)CC(O)CN(C)C)(C)C)ccc(N)c(Cl)n1 79168,C1(CNC(C(CC)CC)=O)CN(C(C2CC3CCC2O3)=O)CC12CCC2 79169,N1(C(C23CN(C(c4ccc(O)nc4)=O)C(C2)CO3)=O)CCN2C(=O)NCC2C1 79170,c1(CNC(=NCCC)N(C)Cc2ccc(OC)cc2)nc2ccc(C)cc2[nH]1 79171,C1(CC)CCCCC1OC.C(C(C)(C)CN(C(=O)COC)C)NC(C=CC)=O 79172,N1(C(CN2C(=O)CNC2=O)=O)C2CCC1CC(NC(C1(F)CCOC1)=O)C2 79173,C(C)(CC(=O)NC12CC(NC(=O)C(C)CC3CC3)(C1)C2)SC 79174,C(=O)(CCCCCCCCCO)N(CCNC(c1cccc(CC#N)c1)=O)CC 79175,CC1CN(C(c2c[nH]nc2-c2cccc(F)c2)=O)CCN1C(=O)C(C)(C)C#N 79176,Cc1nc(O)c(C(=O)NC(C)(C)C(C)NC(=O)C=CC(F)(F)F)cc1Br 79177,C(=O)(C(O)C(F)(F)F)N(CCOCCCN(C(=O)CCc1ccccc1Cl)C)C 79178,C(CCC)(C(=O)NCc1ncc(C)s1)NC(C(C=C)C)=O 79179,N1(C(C(C2CCOCC2)C)=O)CC=C(C(=O)Nc2c(O)cccc2Cl)CC1 79180,CC(C)(C)C(CNC(c1cccc2nccn12)=O)C(=O)N1CC=CC1(C)C 79181,N1(CCCOCC)CC(NC(=O)CSC)CCC1C 79182,c1(NC2C(C)CN(C(C3(O)CCOC3)=O)C2)ncnc2cc(F)c(F)cc12 79183,C1(C)(C(N2CC(COC)(CNC(C3(F)CCOC3)=O)C2)=O)CC2CC2C1 79184,N1(CC)CCCC(C(N2CCCC2C(C)(C)CNC(=O)CC(C)(F)F)=O)C1 79185,CCC(CCCC(=O)N1CCCC1C1(C)CC1)NC(c1cc(C(C)C)[nH]n1)=O 79186,C(=O)(CC(C(N)=O)NC(C)=O)NCCCC(C)NC(C1(CCOC)CCC1)=O 79187,c1(C(=O)NCC(O)CNC(C2COCCC2(F)F)=O)ccc2ccnn2c1 79188,N1(C(C2C(C=C)CC2)=O)CCC2CN(C(c3cccc4cc[nH]c34)=O)CC2C1 79189,N1(C(Cc2c(C)cc(F)cc2)=O)CC(C2CN(C(c3n[nH]c(C)c3O)=O)C2)C1 79190,Cc1cc(C(=O)NC23CCOC(CNC(C4CCCCC4C)=O)(C2)C3)ccc1Cl 79191,c1(C(C(N2CCN(C(c3c(C)nsc3)=O)C(C)C2)=O)(C)C)ccccc1[N+](=O)[O-] 79192,c1(CC)ccc(NC(C2CCCN2C(C2CCCN2C2CC2)=O)=O)cn1 79193,CC(C)C(CNC(C1CCN1C)=O)C(=O)N1CCC1c1ccccc1 79194,O=S(=O)(c1cccc(O)n1)N1CCN(c2ccc(F)nc2)CC1 79195,Cc1ocnc1CC(N1CC(C(C)NC(=O)C=CC2CCCO2)C1)=O 79196,C1(NC(CCCCOC)=O)CC2CCC1N(C(=O)CNC(c1nc(C)no1)=O)C2 79197,CCC(CC)C(=O)NC(Cc1ccoc1)C(=O)N(CC(C1CCC1)OC)C 79198,c1(C(=O)NC2C(C)CCN(C(=O)C=CBr)C2)nccc2ncccc12 79199,N1(C(CC)=O)CCC(NC(=O)CCCc2cc(C)no2)C(O)C1 79200,C(=O)(C1SCCc2sccc21)NC(CCOC)Cc1ccnc2c1CCO2.C(C)(=O)OC 79201,c1(OC(C(=O)NC2(C)CCN(C(c3c(CC)nns3)=O)C2)F)ccc(Cl)c(F)c1 79202,C(=O)(CCCCCC(C)O)NC1C2CN(C(c3nn(CC)c(C4CC4)c3)=O)C1C2 79203,c1(C(=O)NC(CC=C)CNC(=O)C(C)CCC)ccc2c(c1)n(C)c(=O)n2C 79204,Cc1occc1CNC(C1(N(C(C2CCC3CC23)=O)C2CC2)CCC1)=O 79205,c1(C(CNC2CCC(COC)C2)O)c(F)cccc1Cl 79206,C(=O)(CC1=CCCCC1)N1CC2(CN(C(C(CC)OC3CCCC3)=O)C2)C1 79207,N1(C(C(C)SCCCC)=O)CCOCC(C(=O)N(c2cccc(Cl)c2)CC)C1 79208,c1(CCC)cc(C(=O)NC2CC(CNC(C3CC34CCC4)=O)CC2O)nn1C 79209,c1(C(=O)NCC2(CN(C(C(CC)SC)=O)C)CC2)cnn(CCO)c1C 79210,Cc1ncc([N+](=O)[O-])n1CC(=O)NCCCCC(CO)NC(c1n[nH]cc1Cl)=O 79211,c1(NC(C)(CCI)c2nnnn2CC2CCOCC2)cccc2c1CNC2=O 79212,Cc1ccc(S(=O)(=O)NC2CCCNC23CC3)cc1[N+](=O)[O-] 79213,N1(C(C2CCC(C)(F)CC2)=O)CCN(C(=O)C=CCO)CC2CCCCC12 79214,C1(CC(=O)Nc2ccc(C)c(F)c2F)CCN(C(=O)C(C)(C)C)CCC1(F)F 79215,C1(CC(=O)N(CC(C)NC(=O)COCc2nc[nH]n2)C)CCCCCC1 79216,N1(C(c2c(OC(C)C)cncc2)=O)CC2CC(NC(=O)C(F)=CCCF)CC1C2 79217,CC(C)CCCC(=O)N1CC2(CNC(=O)C(O)Cn3cncn3)CC1CO2 79218,N1(C(C2C(CC(C)(C)C)C2)=O)CC=CCC1C(=O)NCC1=CCCC1 79219,c1(C(N2CC(CC)C(NC(=O)C(c3ccccc3)O)C2)=O)cc(C)cc(O)c1 79220,N1(C(C2C(=C)C2)=O)CCC2(COC(CNC(c3sc4cncn4c3C)=O)C2)C1 79221,c1(NC2(C(=O)NC)CCCC2)ccc(S(=O)(=O)NC2CCSC(C)C2)c(Br)c1 79222,C1(C(=O)NC2CCN(C(CCSCCC)=O)C2C)CCC2CC1CO2 79223,N1(C(CCCC)=O)CCN(C(C2C(C)C2C)=O)CC1c1cc(F)cc(F)c1 79224,C1(C(=O)NCC(C(C)(C)C)(C)O)CC2(CCN(C(C3(C)C(C)(C)C3(C)C)=O)C2)C1 79225,Cc1oc(CNC(C2CCCC(F)C2)=O)nc1C(=O)N(C1CSC1)C 79226,c1(C(=O)NCC2CC(NC(C3C(C)(CC)C3)=O)C2)cnc(C)n1C(F)F 79227,C1(CC#C)(C(N2CC(OCC(=O)N(C)CCC3CCCN3C)C2)=O)CCOC1 79228,C1(NC(C(C)OCC)=O)CN(C)CC12CC2.C1=CCNC1=O 79229,c1(CCC)cccc(C(=O)N(C)CC2CCN(C(C34CC(C)C3C4)=O)C2)c1 79230,N1(C(CCC(=O)NC)=O)CCn2nc(CNC(=O)CCC3CCOC3)cc2C1 79231,c1(C(=O)NCCNC(C(C=C=C)C)=O)cc(Br)ccc1N1CCCC1 79232,c1(-c2scc(CC(=O)N(c3ccc(Cl)cn3)C)n2)ccccc1Cl 79233,N1(C(CCn2c(C)ncc2)=O)CCCCCCC1C(=O)N(C)CC1CCOC1C 79234,N1(C(c2c(CC)ocn2)=O)CCC(C)(CC(=O)NC2CCCN(C(C)C)C2)CC1 79235,c1(C(=O)NCC2C=CC(NC(CC3(C)CC3)=O)C2)cnc(C(F)(F)F)c(Cl)c1 79236,C1(NC(C(C2CCC2)NC(C=C(C)C)=O)=O)CC(F)(F)C1(C)C 79237,C1(C(N(CC(O)CNC(c2cscc2Cl)=O)C)=O)Cc2nccnc2C1 79238,C1(C(C(=O)N(CCC(=O)N(C2CC2)CC)C)F)CCCCC1 79239,c1(C(=O)OC)ccc(C(=O)NCCN(C(c2cnns2)=O)C(C)C)cc1Cl 79240,N1(C(c2[nH]cc(C)c2)=O)CCN(C(c2ccnc(C(C)C)n2)=O)C2CCCCC12 79241,C(=O)(CC(C(F)(F)F)NC(=O)C(F)=CC1CC1)NC(CC)COC 79242,C12(CC(N3C(CCNC(CCC)=O)CCC3)=O)COC(C)(C1)C2 79243,C(C1=CCN(C(=O)Cc2ccc(O)cn2)CC1)NC(c1c(SC)n(C)nc1)=O 79244,CC1CCCN(C(=O)CCCCCF)C1CNC(c1cc[nH]c1)=O 79245,n1(CC(CC)O)cc(C(=O)NCC#CCNC(=O)C(C2CCCC2)OC)nn1 79246,c1(C(=O)NCCCCNC(C2C3CCC2(c2cncs2)C3)=O)cccc(Cl)c1F 79247,CC(C)CCCCCC(=O)NCC(C)CNC(=O)C=CC1CCOC1 79248,CCC(C)(C)C(O)C(=O)NCC1(O)CCCN(C(=O)CN2CSCC2=O)CC1 79249,C1(C(N2CC(n3cccn3)C2)=O)CCC2(CC2)N1C(c1cc(F)ccc1F)=O 79250,C=CCCC(CC(C)C)C(=O)N(CCCCCNC(C1CC12CC(C)(C)C2)=O)C 79251,N1(C(=O)CCCCCl)CCC2(CCCC2N2CCC(C(F)F)CC2)CC1 79252,CC1CCN(C(=O)COC2CC=CC2)CC1N(C)C(C1CCOCC1(C)C)=O 79253,C1(CC)(NC(c2ccc(C#N)s2)=O)CCN(C(=O)CCC2CCC(C)O2)CC1 79254,C(c1ccccn1)=C(C)C(=O)NC(C1CCCC1)CNC(C1(C#N)CC=CC1)=O 79255,C(CO)(CCCCNC(=O)C(F)CC1CCCC1)NC(C(c1ccccc1)C)=O 79256,C(c1cccnc1)=C(C)C(N1CCC(=CCNC(=O)CC2(C)CC2(F)F)CC1)=O 79257,CC1COC(CO)CN1C(=O)CCCNC(=O)CC(=O)N(C)C 79258,C1(C)(NC(CN2C(C)CCCC2)=O)CCCN(C(=O)CC2CC3CC3C2)C1 79259,Cc1ccc(C(=O)NCCCN(CCCCNC(=O)C=CCF)C)cc1O 79260,c1(CCC)coc(=NCC2(S(=O)(=O)N(C)C)CC2)[nH]1 79261,C1(NC(c2cn(CC)nn2)=O)CN(C(c2ccn(CC)c2C)=O)C(C)(COC)C1 79262,c1(C(N(CC(C)C(=O)N(C2CCOC2)C2CC2)C)=O)cnn(C)c1Cl 79263,c1(C(=O)NC2(C(F)F)CC2)cnn(-c2ccccc2)c1I 79264,n1(CC(=O)NC(C2CCCN(C(c3cncnc3)=O)C2)C)cc(Br)c(=N)[nH]1 79265,c1(CC(N2CC(C(Cn3cc(C(C)OCC)nn3)F)C2)=O)ccc(O)cc1 79266,c1(NC(C(=O)NCC(C)O)=O)ccc(-c2ncn(C(C)C)n2)cc1 79267,Cc1nc[nH]c1C(=O)NC1(C(=O)NC2CC2CN(C)C(C)C)CC1 79268,c1(CC(N2CC(NC(C(C(CC)O)C)=O)C2)=O)ccc2cccnc2c1 79269,c1(C(=O)NC2CC(CCNC(C(C)OCC=C)=O)C2)nnn2c1CCCC2 79270,C(=O)(C1=COCCC1)NCC1CC(NC(CC2(CS(C)(=O)=O)CC2)=O)C1 79271,C1(C(=O)NC(CNC(C=Cc2cncc(C)c2)=O)CO)CC2(C1)CC(C)(C)C2 79272,N1(C(c2scc(C)c2)=O)CC2(CCC2)CC1CNC(C1COCCN1C)=O 79273,C(=O)(CCCCCC#N)NCC(C)NC(c1cccc(SCCN)c1)=O 79274,N1(C(CCC(CC)NC(=O)Cc2cc[nH]c2)=O)CC2CC3CC2C1C3 79275,N1(C(CC=C=C)=O)CCC2CN(C(=O)CCSc3ccc(Cl)cc3)CCC2C1 79276,c1(NC(=O)OC(CCOC)C(=O)OC(C)(C)C)ccc(Cl)c(F)c1 79277,C(CC(=O)NC(c1ccc(C)nc1)C)(C(F)(F)F)NC(C=CC(CC)C)=O 79278,CC(C)(CNC(=O)C(F)CC1CN(C(=O)CC(C2CC2)C2CC2)C1)C(F)(F)F 79279,CC(CCC(=O)NCC1(NC(=O)CSCc2ncc[nH]2)CCC1)N(C)C 79280,C(N=c1[nH]c(=NCc2ccnnc2)[nH]c2c1CCC2)C1CC(=O)NC1 79281,N1(Cc2c(NC(CC(C)N(C)C)=O)cccc2Cl)C(=O)c2ccccc2C1=O 79282,C1(N(C(CCOCC#C)=O)C)CCCCN(C(=O)CCC2CCCCO2)C1 79283,N1(CCN(C(N(C(c2ccco2)C)C)=O)CCN)CC2CCCCC2C1 79284,C12(NC(Cn3ncn(C)c3=O)=O)CCCC1N(C(c1cc(F)cnc1O)=O)CC2 79285,C1(NC(CCOCCOC)=O)(CF)CCN(C(=O)CN2CCOC2=O)C1 79286,N1(C(c2c(OC)csc2)=O)CC2=C(C1)CN(C(C1(C(F)(F)F)CC3CC3C1)=O)C2 79287,CCCC(C)CC(=O)NCc1cc(C2CCN(C(c3ccno3)=O)CC2)no1 79288,c1(C(N2CCN(C(C3CCS3(=O)=O)=O)C3C2C3)=O)cc2nc(=O)ccn2[nH]1 79289,N1(C(C2CN(CC)C(=O)C2)=O)C2CCCC1CC(NC(=O)C=Cc1cscn1)C2 79290,Cn1c(C(=O)NC2CCCC(CNC(C3CC4(CC4)C3)=O)C2)cnc1S 79291,c1(C(C)=O)ccc(C(N2CC(NC(=O)C(C)NS(C)(=O)=O)CC2C)=O)cc1C 79292,C(C(F)(F)C(=O)NCC1(C)CCCC1NC(=O)CC1COCCN1C)N(C)C 79293,C1(NC(c2cc(COC)on2)=O)CN(C(C2CCOC2C)=O)CCC12CCC2 79294,c1(CNC(CCN(C(CCC(C)C)=O)CCCO)=O)cncc(C#N)c1 79295,c1(C(=O)NCC2(NC(C(CC)SC)=O)CCC2)cc(N(C)C)nc(Cl)c1 79296,C1(C)(CCNC(C(C)=CC2CC2)=O)CCN(C(C2(F)CC2)=O)C1 79297,c1(C(N2CCC(CCNC(c3c(CCC)nco3)=O)C2)=O)c(C)nnn1CC 79298,N1(C(CCOCC#C)=O)CCC2(NC(c3ccc(CSC)cc3)=O)CC2C1 79299,C1(C)(C(N(CCCCN(C(c2cnc(C)s2)=O)C)C)=O)CCCN(C)C1 79300,CC(C)(O)CC(=O)N(CCC(=O)NC1CCCC(O)C1)C1CC1 79301,N1(C(C(C2(O)CCC2)NC(CC(=O)N(C)C)=O)=O)CC(C#N)C2(CCC2)C1 79302,C1(NC(C(c2cccc(F)c2)C)=O)CC(NC(c2cc(C(N)=O)c[nH]2)=O)C(O)C1 79303,C1(NC(C2C(CNC(CC3(N(C)C)CCC3)=O)CCC2)=O)COCC1N=[N+]=[N-] 79304,N1(C(CCC(C)SC)=O)CCCC(NC(=O)C=Cc2cnn(C)c2)CC1 79305,C1(CC)(CC)CC(NC(C2CCCC2CNC(=O)CC(=O)OC)=O)C1 79306,c1(C(N(c2cc(Cl)cc(Cl)c2)CCOC)=O)cccc2c1NC(C)CC(=O)N2 79307,c1(C(=O)NC2C(NC(c3c(N)cccc3)=O)CCCC2)ccc2ncnn2c1 79308,C1(NC(C=CC(C)C)=O)CN(C(C2CC2C2CC2)=O)CC1c1cccc(F)c1 79309,Cn1cc(S(=O)(=O)Nc2ccc(N3CCSCC3)cc2)c2cccc(Br)c12 79310,c1(C(=O)NC(CC)CNC(=O)COCCC(C)C)ccc(O)nc1Cl 79311,C(CNC(=O)CC(C)Cc1cccc(OC)c1)(C(C)(C)C)NC(C1C(CC)C1)=O 79312,N1(C(c2n[nH]c(=N)[nH]2)=O)CC2CC(NC(=O)CCc3cccs3)CC2C1 79313,N1(C(C2C(c3c(C)n(C)nc3)C2)=O)CC(NC(=O)C(C)C(C)C)CC(F)C1 79314,CON1CCC(C(=O)NCC2CCCC2C(=O)N(CC(C2CCC2)OC)C)CC1 79315,CC1CC(=O)CCC1C(=O)NC(C(=O)N(CCC(=O)NC1CC1)C)C1CCC1 79316,N1(C(=O)C=C2CCC2)CC2(C1)CN(C(c1c(Cl)cncc1Br)=O)C2 79317,N1(C(C(CCC)Cl)=O)C2CCC(C2)C1C(N1CCCC(C)C1)=O 79318,C(=O)(C(C(C)C)OC)N(CC(CC)NC(=O)C=CC(C)(C)C)CC 79319,C1(NC(CC(C)C(F)F)=O)CC2CC(C1)N(C(c1ccc(N)cc1)=O)C2 79320,C(=O)(C#CC(=O)N(C)C)NC1CC(NC(c2c(SC)occ2)=O)C1 79321,Cc1nccc(C(N2CCC(O)(CNC(c3cc(Cl)cs3)=O)CC2)=O)c1C 79322,c12cn(nn1)CC(=O)NC2(C)C.c1(C(=O)OC(C)(C)C)csc(Cl)c1 79323,CC1(CC(N2CC3CC2C3NC(C2CCCOCC2)=O)=O)CCCCC1 79324,Cc1nc(C)n(O)c1C(=O)NC(C)CCCCNC(=O)Cn1ccc([N+](=O)[O-])n1 79325,N1(C(C(N2CCOC2=O)C)=O)C2CCC1CN(C(c1cncn1C)=O)CC2 79326,C1(C(N2CCC(F)(CNC(=O)CC(F)F)C2)=O)(OC)CCCCCC1 79327,C(=O)(CCC(F)(F)F)N1C(C)(CC(=O)NC(C(=O)OCCCC)C)CC1 79328,N1(C(C2CCN(C(CCC)=O)CC2)=O)CCCC2(NC(C3CCC3)=O)CC2C1 79329,C1(NC(C2CC(F)(F)C2)=O)CC2CC(C1)N(C(=O)CCc1ccc(Cl)c(F)c1)C2 79330,CC1(C(=O)NCC2(F)CC(NC(c3cn(C4CC4)cn3)=O)C2)CC2C=CC1C2 79331,c1(C(=O)NCC2C(NC(COCCC)=O)CCC2)ccn2c1CCCC2 79332,C12(CNC(c3cnc4nccn4c3)=O)CN(C(=O)CCC(F)F)CC1CCO2 79333,c1(OC(C)C)ccc(C(=O)NCC2CC(C)(C)CN2C(=O)C(C)N(C)C)c(Cl)c1 79334,c1(CCNC(=O)CC2CC2)ccccn1.c1(C2C3CC3C(=O)N2)nc[nH]n1 79335,C1(C(=O)NCCC2C(=O)OCC2)CC(O)CN1C(C1CCO1)=O 79336,c1(C2(NC(C(=O)NCC3(SC)CCCOC3)=O)CCC2)c(F)cccc1F 79337,CCC(C)CCC(=O)NCC1(O)CCCN(C(c2ccnc(NC3CCC3)c2)=O)C1 79338,c1(C(N2C(CN(C(C(C)C3CC3)=O)C)CCC2)=O)cc(C(F)F)cc(Cl)c1 79339,Cc1cc(-c2cccc(CC(=O)N(C)Cc3ccc(O)cc3)n2)cc(O)c1F 79340,CC#CCCCC(=O)NC(c1ccccc1F)CNC(=O)C(C)c1cc[nH]n1 79341,Cc1nn(C)c(N2CCN(C)CC2)c1CNC(=O)CC1CC12CC2 79342,C(=O)(C(O)CC(F)(F)F)N(C(CC)CSc1ccccc1)C 79343,c1(CNC(C2(COC)CCCN2C(=O)C(O)C(C)(C)C)=O)nc(COC)cc(O)n1 79344,C1(NC(c2ccnc(C3CC3)n2)=O)C2CC1N(C(C1CC3CCC1O3)=O)C2 79345,C1(C(N(CCCNC(=O)C2=CCCCC2)CCO)=O)CCCC2CCCN12 79346,c1(CCCC)cc(C(=O)NC2CCCCC2NC(c2n[nH]c(C)n2)=O)c(C)o1 79347,C1(COC)CN(C(C2COCCC2(F)F)=O)CCN1C(=O)CCc1cnn(C)n1 79348,N1(C(c2n(CC)nnc2)=O)CC(NC(=O)C2=CCCC(C)(C)C2)CC12CCOC2 79349,N1(C(C=C(C)C(F)F)=O)CCCC(C)(C)C1CNC(C1CCC2CC2CC1)=O 79350,c1(C(=O)NCCN(C(C2C(C)(C(C)C)C2)=O)C)ccc2c(=N)[nH]cnc2c1 79351,c1(C(C(N2CCC(N(C(=O)CC3CC3)CCO)C2)=O)O)ccc(Cl)c(Cl)c1 79352,c1(CCC(=O)NC2C3CC2N(C(c2cc(Br)no2)=O)C3)n[nH]c2c1CCCC2 79353,C12(NC(CCCNC(c3c(C)nn[nH]3)=O)=O)CC1COC2(C)C 79354,c1(C(=O)NCC2(CNC(CCCOC)=O)CCC2)cccc(C(=O)OC)n1 79355,Cc1c(C(=O)NC2CCC2NC(c2ccn(CC(F)F)n2)=O)ccn1C(C)C 79356,c1(C(c2n(CCCC)nnn2)NCCCCC(C)(C)C)ccc2c(c1)OCCO2 79357,c1(CC)cc(C(=O)NC2(C(N3CCC(n4ccnc4)C3)=O)CSC2)nn1C 79358,c1(CC)c(C(N2CC(NC(C3C4CC4C4CC34)=O)C2)=O)oc2ccccc12 79359,C1(C(=O)NCc2cc(C)no2)(NC(=O)COc2ccsn2)CCCC1C 79360,C1(NC(c2cc(Cl)cc(F)c2F)=O)CN(C(C2(O)CCOC2)=O)CC2(CC2)C1 79361,c1(C(=O)NCC2CN(C(CCNC(=O)NC)=O)C3C2C3)ccnc2c1nnn2C 79362,N1(C(CC(C)(C)N(C)C(C2CC(=O)CC(=O)N2)=O)=O)CC2(CCC(=O)N2)C1 79363,N1(C(C(CC)COC)=O)Cc2ccc(C(C)NC(C3CCCCCC3)=O)cc2C1 79364,c1(C(=O)NCC2C3CN(C(C(CC(N)=O)O)=O)CC32)cccc2nc(O)[nH]c12 79365,Cc1ccc(O)cc1C(=O)NC1CC(OCC(N2CCCC(C)C2C)=O)C1 79366,N1(C(CN(C)C(N)=O)=O)C2CCCC1CC(CNC(C1(O)CCC1)=O)C2 79367,C1(O)(CNC(c2c(C)oc(C3CC3)n2)=O)CCCN(C(=O)CCC2CCOC2)C1 79368,C(C)(C)(CC(=O)N(C)CC1CCCN(C(=O)C(c2ccc(F)cc2)(F)F)C1)OC 79369,N1(C(C(COCC)n2cc(Cc3c[nH]nc3OC)nn2)=O)CCCC(C(=O)O)C1 79370,C1(NC(CC=CCC)=O)CCC2(CCCN(C(c3cnc4n3CCC4)=O)C2)C1 79371,c1(OC)ccc(Cn2nnnc2C(C2(SC)CC2)NC2CC2c2cccs2)cc1 79372,c1(C(N2CC(OCCNC(C3CC3(F)F)=O)C2)=O)ncc(Br)cc1[N+](=O)[O-] 79373,C12(NC(C(C)CN(C)C)=O)CCCC1(F)CN(C(c1ccc3c(c1)CCO3)=O)C2 79374,c1(C(=O)NC2CN(C(CCC(=O)OC)=O)CC(O)C2)cccn2cnnc12 79375,C#CC1(C(=O)N(CCCOC)C)CN(C(=O)CCc2nc[nH]n2)C1 79376,O=C1CC2(CCN(C(C3CNC4(CC4)CO3)=O)CC2)C(=O)N1 79377,CN1C(=O)CN(C(=O)Nc2ccc(=O)n(-c3ccccc3)c2)c2ccc(Br)cc21 79378,N1(C(C2N(C)CC2)=O)CCC(C(=O)NCCC2C=CCC2)C1(C)C 79379,c1(CCOC)cnoc1C(=O)NCC1CC(CNC(=O)CCF)CO1 79380,N1(C(c2c(C)nns2)=O)CC2(C=C(C(=O)Nc3cccc(CCO)c3)CO2)C1 79381,C1(C(NOCCCOC)=O)(COC)C=CCN1C(c1c[nH]c(=O)cn1)=O 79382,CC(C)(C(=O)NCC1(O)CCN(C(c2ccccc2O)=O)CC1)C(N)=O 79383,c1(CCC(=O)NC2CN(C(C=C(C)Cl)=O)C2)c(C)nc(-c2ccccc2)nc1O 79384,N(C)(S(=O)(=O)N1CCC(C(N2CCNCC2)=O)CC1)C(CC)COC 79385,C(CC(C)C)(C(=O)NC1(C)CCN(C(=O)Cc2ccc(C(C)=O)cc2)C1)OC 79386,C(=O)(CCCC(c1nnnn1C(C)(C)C)NCCc1nncn1C)OCC 79387,CC1OCCC1CC(=O)N(C(c1ccccc1)CNC(c1ccsc1)=O)C 79388,C(=O)(CCCN(C)N=O)N1CCC(C)C1CNC(=O)COCC1CCC1 79389,C1(CC)C(NC(=O)C(C2CCC(=O)N2)C)CCCN1C(=O)Cc1ccccc1O 79390,c1(COCC(N2CCCC2Cn2cc(-c3nccs3)nn2)=O)ccccc1Cl 79391,c1(C(=O)NC2CCC(NC(C(CC)(C)O)=O)CC2)c(Cl)cncc1Cl 79392,C1(NC(=O)COCc2nccn2C)CCOCC1.C12CCN(C1)C(=O)COC2C 79393,C1(C(N2CCCC(N(C(Cc3ccc(OC)nc3)=O)C)C2)=O)CC2C(C1)C2(C)C 79394,c1(CC)nc(=N)[nH]c(=NC2CC3CC(C2)N(C(C2CC(=O)N(C(C)C)C2)=O)C3)[nH]1 79395,C1(CNC(c2ccccc2OCc2cccs2)=O)CC2(C1)CC21CC1 79396,C12(COC)CC(NC(=O)CN3CSCC3=O)(CN1C(=O)C(C)C(C)(C)C)C2 79397,CC1=C(C(=O)NCC2CCCCC2NC(=O)C(N)=O)C(C)n2ncnc2N1C 79398,c1(C(c2nnnn2CSc2ccccc2)NCC(CC)(C)OC)c(I)ncn1C 79399,N1(C(CCNC(=O)C=CCl)=O)CCC2(CC(NC(C3CCCCC3(F)F)=O)C2)C1 79400,C(=O)(CCC(C)(C)F)NC(C1CCN(C(c2ccn(C)n2)=O)C1)C 79401,N(C(=NCCCN(C)C)NCC(C)Oc1cccc(Cl)c1)C(C=C)C 79402,c1(N2C3CN(C(c4ccc5nc[nH]c5c4)=O)CC2C3)ncnc2cccc(F)c12 79403,C(N=c1[nH]c(=NCCOCCC2CC2)[nH]c2c1CCCC2)c1c(F)ccc(F)c1 79404,C=CCC(C(=O)NC(CCC)C(O)C(=O)N(C(CC)CC)CCO)C(C)C 79405,c1(CC(=O)N(C(C)C)CCN(C)C(c2c[nH]c(=N)o2)=O)cccnc1Cl 79406,C(N=c1ccnc(N(C)C)[nH]1)C1(OC)CCCSC1 79407,C1(NC(C(CC)C(C)C)=O)CCOC2(CCC2)C1 79408,N1(C(Cc2c(C)cco2)=O)CCCC(C(C)(O)CNC(=O)C2=CCCC2)C1 79409,c1(C(=O)NC2CN(C(COCC)=O)C(C)C2)ccc([N+](=O)[O-])cc1 79410,N1(C(COCc2cc(C)no2)=O)C(CNC(c2ccoc2C)=O)CC2COCC12 79411,C1(C(=O)NCC2(F)CCCC2)CCN(C(=O)c2cc(O)ncn2)O1 79412,C1(C2CN(C(=O)C(C)(C)CF)C2)(NC(c2ccc(CN(C)C)o2)=O)CC1 79413,C1(C(=O)NC(C2CCN(C(c3ccncc3N)=O)CC2)C)Cc2ccncc2C1 79414,N1(C(CC2ON=C(C)C2)=O)CC(NC(c2c(N)cccc2Cl)=O)CC(F)C1 79415,CC1CN(C(c2cc(CN(C)C)on2)=O)CCC1NC(c1csc(C2CC2)n1)=O 79416,CCN=c1cc(-c2cn(CC(F)(F)CNC(c3cn(CC)cn3)=O)nn2)cc[nH]1 79417,c1(NC(=O)CCNc2ncc(Cl)cn2)ccc2c(c1)OC(F)(F)O2 79418,C1(CN)(NCCSC2CC3CCC2C3)CCOCC1 79419,CC(CC1CCCCC1)C(=O)NCCC(F)Cn1cc(C(c2ccccc2)O)nn1 79420,Cc1cn2cc(C(N3CCCC3CNC(C3(C)CCCN3C)=O)=O)cc(F)c2n1 79421,CC(CC(C)(F)F)C(=O)NC(C)(C)CNC(c1cc2n(n1)CC(F)C2)=O 79422,C1(CC(C)NC(=O)C(Cc2ccoc2)NC(=O)CCN(C)C)CCCCC1 79423,S(=O)(=O)(c1ccc(N(C)CCc2ccc(Cl)cc2)c(Cl)c1)NCC(C(C)O)C 79424,C=C(C)CCC(=O)N1CCC(C(C)(C)NC(c2c[nH]cc2-c2ccc(C)s2)=O)C1 79425,c1(C(=O)NC2C(C(NOC(CC)CC)=O)CC2)cc(C(N)=O)c[nH]1 79426,c1(C(=O)NCC2(NC(=O)CC3CC34CC4)CCOC2)nncc2c1CCCC2 79427,N1(c2nc(CC)on2)CCC2(CC1)CC2C(N1CCC2OCC2C1)=O 79428,c1(OC)cc(C2CC2)ccc1C(=O)NC1C2CC1CN(C(=O)C(F)=CC1CC1)C2 79429,Cc1cc(OCCCC(=O)NCCNc2ccccn2)ccc1Cl 79430,N1(C(C(F)=CC)=O)CCCCC2(C1)CN(C(=O)CCn1ccnc1C(C)C)C2 79431,c1(C(=O)OC)cc(C(=O)NCC2(F)CC(NC(=O)C(CCO)N(C)C)C2)c(C)o1 79432,Cc1cc(C(=O)NC2CC=CCC2C(=O)NC(C)C(=O)NC2CC2)c(N)s1 79433,N1(C(Cc2c(OC)nccc2)=O)CCCC(C)(NC(=O)CC2CCCN2C)C1 79434,N1(C(C2C(=O)OCC2)=O)CCC2(CCCCN(C(c3ccc(O)nc3)=O)C2)C1 79435,c1(OC)ccc(C(N2CCN(C(C3CCCSS3)=O)C(C)C2)=O)cc1C 79436,C1(CNC(C2(C#N)CC2)=O)CCCCN1C(C1(C(F)F)CCCCC1)=O 79437,C1(C(=O)NCCCNC(CCCCNC(C)=O)=O)CCC2CC2CC1 79438,c1(N2CCC(c3occc3)CC2)nc2cc[nH]c2c(=NCC2CCCO2)[nH]1 79439,N1(C(C(C=CCCC)O)=O)C2CCCC1CC(NC(=O)C=C1CCC(C)CC1)C2 79440,c12c(OC)cc(cc1Br)NC(=O)N2.C1(C(OC)OC)CC(=O)N(C2CC2)C1 79441,C(C1CN(C(=O)COC2(C)CCCC2)Cc2ccccc21)NC(C(C)(C)CF)=O 79442,C12(CCOCC1)CC(=O)C2.C1(N)CCCCC1NC(C1(CO)CC1)=O.CN(C)C1CC1 79443,c1(C(=O)NC2(CN(C(=O)Cc3cnnn3C)C)CC2)ccc(-c2nnco2)cc1 79444,C1(CC=C)(C(N2CC(OCC(=O)NCCCF)C2)=O)CC=CC1 79445,Cc1cnc(C)c(C(=O)NC(C2CCCN2C(=O)C(C)OC2CCCCC2)C)c1 79446,C(=O)(C(O)C(C)(C)CC)NC1C(NC(c2cc(CC)[nH]n2)=O)C1 79447,CCC(O)C(C)(C)C(=O)N1CCC(C(F)C(=O)N(C2CC3(CCC3)C2)C)C1 79448,Cc1cccc(OCC(N2CCC(C)(c3cn(C4CCOC4)nn3)C2)=O)n1 79449,c1(C(N2CC(O)(CCNC(C3C(C)C3C)=O)C2)=O)cc2ccccc2s1 79450,C(=O)(C(F)(F)CCn1cc(-c2ncoc2C)nn1)N1CCC(C(C)OC)CC1 79451,c1(NC(C(C)C)CNC(C2CCCNS2(=O)=O)=O)ncnn2cccc12 79452,Cn1cc(NC(=O)Cn2cc(Cl)c(C(F)(F)F)n2)ccc1=O 79453,C1(NC(C(COCC)C)=O)C2CC3C1C3C2C(=O)NC1CCC(N(C)C)C1 79454,C(=O)(CCCCC(=O)NC(c1ccccc1)c1nccn1C)NC 79455,C(CC(=O)N=c1cc2ccccn2[nH]1)C1N(C(CC(C(C)C)C)=O)CCCC1 79456,Cc1ccc2c(C(=O)NC(C3(O)CN(C(c4ccnc(O)c4)=O)C3)C)c[nH]c2c1 79457,CC(CC(C)(C)C)NC(c1[nH]ccc1CNC(=O)C=C1CCOCC1)=O 79458,c1(C(N2CC(CN(C(=O)CCCC3CC3)C)C2)=O)cccc2ccncc12 79459,C#CCC(O)C(=O)NC(c1cn(C)nn1)C(=O)N(C)Cc1conc1CC 79460,c1(OCC(N2CCC(CNC(C=CSC)=O)C2)=O)ccc([N+](=O)[O-])cc1 79461,C(=O)(C1CCCc2nc[nH]c21)NCCC1CC(OC)CN1C(C1CCC1(F)F)=O 79462,Cc1nn2cccnc2c1C(=O)NCCCCNC(=O)COC1CCCCC1C 79463,Cn1ncc(C(=O)NCC2(NC(C3CCC(F)CC3)=O)CCC2)c1Cl 79464,C(=O)(C(C)C(F)(F)F)NCCC1CN(C(c2cc(OC)c(Cl)s2)=O)C1 79465,N1(C(Cc2c(C)cnn2C)=O)CCC(NC(C2CCN(C(N)=O)CC2)=O)C(F)C1 79466,Cc1cc(O)cc(C)c1C(=O)NC1CCCC(N(C(=O)Cn2cnnn2)C)C1 79467,Cc1cncc(CC(N2CC(NC(=O)Cn3nnc(C4CC4)n3)C2)=O)c1 79468,C1(C(=O)NCCF)Cc2c([nH]c3ccccc23)CN1Cc1ncccn1 79469,Cc1cc(CCC(=O)NC(C)C(C)NC(=O)CCc2cscn2)n[nH]1 79470,Cc1cc(C(=O)N(CC)CC2CCCCC2n2cc(-c3cnn(C)c3)nn2)c(C)o1 79471,CCCCC(C(=O)NCC1(Nc2cncc(C#N)n2)CC1)ON=C(C)C 79472,C1(C(=O)NCC2N(C(C(C)Cc3cnc[nH]3)=O)CC(O)C2)CC(C)(C)CCO1 79473,c1(C(=O)NC2CCC(NC(C3CCC(C)C3)=O)CC2)cnn2c1N(C)CC2 79474,C12(NC(c3cc[nH]c3)=O)CN(C(=O)CSC3CC3)CC1CS(=O)(=O)C2 79475,C(=O)(CC(C)c1ccccc1)NC(C)CNC(=O)C=CCOCC(F)(F)F 79476,c1(C(=O)NCC(=C2CN(C(c3cc4occc4[nH]3)=O)C2)F)cn2ccccc2n1 79477,C(=O)(CCC(=O)C(C)(C)C)N1CC(C(=O)NCCc2ncn(C)n2)CC(C)(C)C1 79478,C(=O)(C(CCC1CCC1)NC(=O)CCC=C(C)C)NC(C=C)C1CCC1 79479,c1(CCC(=O)NCC(CC(C)O)C)ccnc2ccccc12 79480,N1(C(c2cc(C)n(C)c2)=O)CC(NC(c2conc2C(C)(C)C)=O)CCC1C 79481,C1(CC)CN(C(C2CCOCC2(C)C)=O)CCN1C(=O)C=CSc1ccccc1 79482,C(=O)(C1=CC2C=CC(C1)C2)NC(C1CN(C(Cc2c(C)cccc2)=O)C1)C 79483,C=CC1CN(C(=O)C(C)C2CCCC2)CC1NC(c1cn(C2CCC2)nn1)=O 79484,c1(C(=O)NCC2C(Cn3cc(CC(C)O)nn3)C2(F)F)[nH]c(=N)ccc1Br 79485,C1(C(=O)NC2CC(CNC(c3ccccc3C(N)=O)=O)C2)(OC)CCCC(C)C1 79486,N1(C(c2n(CC)ncc2)=O)CC2CC(NC(c3cnoc3)=O)CC1C2 79487,C1(NC(c2c(CC)cco2)=O)C2CC3CN(C(c4cnc5sccc5c4)=O)C1C3C2 79488,N1(C(CC2CC(CC)OCC2)=O)CCCN(C(c2cnsn2)=O)CCC1 79489,C(C1c2ccsc2CCN1C(=O)C(O)CC1CCCCC1)NC(CCC=C=C)=O 79490,c1(OC)ccc(S(=O)(=O)N(C)C)cc1C(=O)O.c1(C(C(=O)O)N)cscn1 79491,Cc1cc(C(=O)NC2COCCN(c3nnc(C4CC4)s3)C2)nc(Cl)c1 79492,C1(CN(C(CSCC(C)C)=O)C)CN(C(=O)CC2COCCN2C)CCO1 79493,N1(C(c2cc(C)ns2)=O)CCC(CNC(=O)CCC2(C)CC2(F)F)C(F)(F)C1 79494,CC1(CNC(C2CCCC(c3ccccc3)O2)=O)CCCN1C(=O)CS(N)(=O)=O 79495,Cn1nnc2cc(C(=O)NC3(C)CC(NC(c4c[nH]c(=N)s4)=O)C3)ccc12 79496,C1(NC(Cc2ccc(C)cc2)=O)CCN(C(=O)CC2(CSC)CC2)CC1C(C)C 79497,C(=O)(CC1CCc2ccccc21)NCCN(CCC)C(C12CCC1C2)=O 79498,C1(C(N2CC3(N(C)CC3)C2)=O)CN(C(=O)C=CCN2CCC2)CCN1C 79499,C(C(=O)NCCNC(=O)Cc1ccnc(Br)c1)(C(C)(C)C)N(C)C 79500,c1(C(N2C(C(C)NC(=O)C(C)(Cl)Cl)CCC2)=O)ccc2ccoc2c1 79501,CCC(CCC(=O)NC1CC(NC(=O)CC2OCCC2(C)C)C1)OC 79502,c1(C(=O)NC2CN(C(C(C)NC(CC)(C)C)=O)C2)n[nH]c(C)c1Cl 79503,c1(N2CCCC(C=C)C2)nc2ccc(S(=O)(=O)NC3CCC(C)(C)CC3)cc2s1 79504,C1(C(N2C(CN(C(C3CN(C(C)=O)C3)=O)C)CCC2)=O)CCc2nncn2C1 79505,N1(C(c2c(Cl)cc(C)nc2)=O)C2CCCC1CN(C(=O)CC1COC(=O)N1)C2 79506,c1(C(N2CCN(C(C(C)OC)=O)CC3(C2)CC3)=O)cc2c(O)ccc(F)c2[nH]1 79507,c1(OC)c(I)ccc(C(N2CC(c3ccccc3)C(C#N)C2)=O)c1C 79508,c1(-c2ccsc2)n[nH]c(=NC2CCC2C2(C)CCOC2)o1 79509,C1(C(=O)NCC2(F)CCN(C(c3c(C)c[nH]c3)=O)CC2)CC(C)(C)OC(C)(C)C1 79510,C1(C(N2CCC(N(C(=O)Cn3nnc(C4CC4)n3)C)CC2)=O)OC2CCC1CC2 79511,c1(C(=O)OC)ccn(CC(=O)NCCN(CC(C)O)C(c2cnccn2)=O)n1 79512,N(C(=NCc1ccc(OC(F)F)cc1)NCC12CC(CCO1)C2)Cc1c(C)ocn1 79513,c1(C(=O)NC(CCOC)CNC(=O)CC2(NC(C)=O)CC2)ccnc(C)c1N 79514,c1(C(N2C(C(=O)OCC)CCCC2)C(=O)NCCSC)cc2c(cn1)OCCO2 79515,C1(C(N2CC(CCC)C(CO)C2)=O)CCCCC1(C)NC(=O)C(=O)N(C)C 79516,N1(C(CC(C)=C(C)C)=O)CC(C)(C)CC1CNC(=O)CCc1cccnc1F 79517,Cc1cc(C(=O)N(CCC(=O)NCC2CCC(C)(C)O2)CC2CC2)cn1C 79518,C1(C(=O)Nc2cc(O)n[nH]2)CCCC12CCN(Cc1csc(Br)n1)C2 79519,Cc1cc(=NC(CCO)C2CCSCC2)[nH]c(=NCc2cccc(CO)c2)[nH]1 79520,C1(c2ccccc2)(NC(C(CC)NC(C)=O)=O)CCN(C(c2nocc2C)=O)C1 79521,c1(C(=O)NCC2C(NC(c3c(CC)ccs3)=O)COC2)ccc(F)c(C)c1F 79522,C=CC(C)(CC)C(=O)NC(CC(=O)Nc1cnc(N(C)C)nc1)C1CC1 79523,n1(CC)ncc(Cl)c1C(=O)NCC1(COC)CN(C(C2CC(=O)N2)=O)C1 79524,C1(N(C(C(C2CCCC2)OCC)=O)C)CCCCC1NC(c1ccc(C)nn1)=O 79525,Cc1c(C(=O)OCC(=O)NC2CCN(Cc3ccccc3)C2)cccc1O 79526,c1(C(=O)NCCCNC(C(CC2CCCCC2)OC)=O)c([N+](=O)[O-])c(C)nn1C 79527,n1(CC(=O)N(C(CCNC(C(CSC)C)=O)C)C)nc(C(C)(C)C)cc1N 79528,c1(C(=O)NC2C(C)CN(C(c3ccc(C(N)=O)s3)=O)C2)cccc(S(N)(=O)=O)c1 79529,c1(CC(=O)NCC(n2cc(C3(CO)CCN(C)CC3)nn2)C)c(F)cncc1Cl 79530,c1(C(=O)NC2C(CC)N(C(c3ncc(F)cn3)=O)CC2)cc(=O)cc(Cl)[nH]1 79531,C=C(C)CCCC(=O)N(C)CC1CCCN1C(=O)C(N1CCOCC1)C 79532,N1(C(CSCCC)=O)CC(CO)C2(C1)CN(C(=O)C(O)CN1CCOCC1)C2 79533,N1(c2cc(NCc3cnc(C(C)(C)C)[nH]3)nc(C)n2)CC2CCCCC2(CO)C1 79534,c1(C(=O)NC2CCC(CCNC(C3(CC(C)C)CC3)=O)C2)cnn2ccsc12 79535,Cc1cc(C(N2CCC(CNC(=O)CN3CCCC3=O)C(C)C2)=O)c(N)c(Cl)c1 79536,c1(OC)cccc(N(C(=O)COC(C)(C)CNC(c2nc(C)oc2C)=O)C)c1 79537,C(CC(O)C(=O)N(CCCCNC(=O)CCC(C)OC)C)SC 79538,Cc1c(C(=O)N(CC(=O)NOCCF)C2CCOC2)cco1 79539,C(=O)(CS(=O)C(F)(F)F)NCCCCN(C)C(c1cnc2[nH]cncc1-2)=O 79540,c1(C(C)CC(=O)NCC(O)CN(C)C(c2ncn(C)n2)=O)ccc(Br)cc1 79541,N1(C(c2cccc(N(C)C)c2)=O)CCN(C(C2CC(C)(F)C2)=O)C2COCC12 79542,N1(CCCN(S(CC)(=O)=O)CC(=O)O)CCN(C2CCCN(C)C2)C(=O)C1 79543,C12(CNC(CNC(=O)OCC=C)=O)CCC1CN(C(=O)CC1CC(F)(F)C1)C2 79544,c1(NC(C2(O)CCN(Cc3ccccc3SC(F)(F)F)C2)=O)ccccc1I 79545,N1(C(C(=O)Nc2cnc(N3CCOCC3)nc2)=O)CCC(C2CCOC2)CC1 79546,N1(C(c2n[nH]c(C)c2O)=O)C2CCC1C(C)C(NC(c1ccc(CF)cc1)=O)C2 79547,c1(CC(=O)NC(CC)CNC(=O)C(C)n2cnnn2)ccc(C)c(C)c1 79548,N1(C(CSCC(C)=O)=O)CCCC1COC(F)(F)F 79549,c1(C(=O)NC2(C(=O)NC3CC3CN(C)C)C(C)C2)ccc(Cl)cc1 79550,C1(C(=O)NCCC(=C)CNC(=O)CC2=CCOCC2)C2CC3CC(C2)CC1C3 79551,C(=O)(C(F)CCC(C)(C)C)N1CCCC(CN(C(=O)C2=NNC(=O)CC2)CC)C1 79552,C(CCCN=C(NCC1CC12CCC(F)(F)CC2)NC(C)Cc1ccccc1)OC 79553,c1(CC)nc(C)[nH]c1C(N1CCOC(CN(C(=O)C(C2(O)CCCC2)F)C)C1)=O 79554,C1(CC(=O)NCCCCCNC(c2cc(OC)no2)=O)CCC(C)(O)CC1 79555,N1(C(CC2(OC)CC2)=O)CC(C(=O)Nc2cnoc2CCS(C)(=O)=O)OC(C)C1 79556,c1(CN2CCC(CC(=O)NC(c3ccccc3)CCO)C2)c(F)ccc(O)c1F 79557,Cc1nc(Br)cnc1NC(C1CCCN(C(c2cnnn2C)=O)CC1)=O 79558,C1(NC(C=C(C)C(F)F)=O)CCCC(CN(C(=O)Cc2c(C)n[nH]c2C)C)C1 79559,C[Si]1(C)CCCCN(CC(N2CCC(CCS(N)(=O)=O)CC2)=O)C1 79560,N1(C(c2c(C)nc[nH]2)=O)CCC(F)(F)C(C(=O)NCc2ccnc(Br)c2F)C1 79561,N1(C(CN(CCCCCC)C)=O)CCOC(C(C)NC(C2(C(F)F)CCC2)=O)C1 79562,C(=O)(CCCCSC)NCC1(OC)CN(C(=O)COC2CCOCC2)C1 79563,C(=O)(C1=CC2CCC1C2)N1CC(F)(CNC(c2cc(OC)no2)=O)C1 79564,C1(CNC(N2CCC(O)C2c2ccc(Br)cc2)=O)CC(F)(F)C(=O)N1 79565,C1(NC(CSC)=O)CCCN(C(=O)CC2(O)CCC2)CC1 79566,C1(C(N2CCCC(n3cc(CC(O)C4CC4)nn3)C2)=O)CCCC12CC2 79567,C1(OC)(CNC(=O)CS(=O)(=O)N2CCOCC2)CCN(C(=O)C2=CCCC2)CC1 79568,N1(C(CN(C)CCO)=O)CCCC(C)(NC(C23CC(c4ccccc4)(C2)C3)=O)C1 79569,Nc1ccc(C(N2CCCC(O)(CCNC(=O)C=CC3CCCO3)C2)=O)c(Cl)c1 79570,N1(CCC)CCCCC1C(N1CC2CC2(CNC(=O)CSC(F)F)C1)=O 79571,N1(C(CC2C(=O)NC(=N)S2)=O)CC2CC(CNC(=O)Cc3cc(C4CC4)no3)C2C1 79572,c1(NC(C)=O)cccc(-c2cnc(CNC(=O)Nc3cc(O)ncn3)nc2)c1 79573,C(c1cc(Cl)cc(Cl)c1)=CC(N1CCCCC(CNC(C=COCC)=O)C1)=O 79574,C1(C(=O)NC2C3CN(C(CSCC)=O)CC32)CC2(CCC2)CCO1 79575,N12CC(C(=O)O)C(C1)C2=O.C1(CNCC)(OC)CN(C(=O)ON(C)C)C1 79576,C(C)(c1cccs1)=CC(=O)N(CCNC(C1CC(OC)C1)=O)C1CC1 79577,N1(C(CC(OCC)OCC)=O)CCN(C(=O)C(=O)N=S(C)(C)=O)C(C)C1C 79578,c1(C(=O)NC(C2CCOCC2)C(=O)OC)cc(-c2ccc(F)s2)cc2cc[nH]c12 79579,C#CC1(C(=O)NCc2ccco2)CN(C(=O)CN2CCOCC2=O)C1 79580,Cc1cnc(N2CCC(NC(C3CN(C)C(=O)N3)=O)C2C)nc1 79581,c1(CC2(c3ccccc3)CCN(CC(=O)N(CC)CC)C2)cn2ccccc2n1 79582,Cc1cc(Cl)c(C(N2CCC(NC(c3c[nH]c(C(N)=O)c3)=O)C(F)C2)=O)cc1C 79583,c1(-n2c(C(C3CCCCC3)O)nc(CC(CC)C)n2)cccc2c1CCCC2 79584,c1(OC)cccc(-c2nc(Cc3ccno3)n(Cc3cccs3)n2)c1 79585,n1(CC)cnc2c(NCC3(SC)CC3)[nH]c(=NCc3n[nH]c4c3COCC4)nc12 79586,CC1CC(=O)NC(C(=O)NC2CCN(C(C3(N4CCOCC4)CC3)=O)CC2F)C1 79587,C(=O)(N1CC(O)CCO1)NC(C)CS(C)(=O)=O 79588,N(C(=NC)N1CCC(CCOC)C1)CC(CC)OC.c1(OC)ccccc1F 79589,N1(C(C(CC)(C)O)=O)CCC2(CCN(C(c3cc(COC)[nH]n3)=O)CC2)C1 79590,CCCCCCCCNC(C1CCCC1CNC(c1ncoc1C(C)C)=O)=O 79591,Cc1ccc(C(=O)NCC(CO)NC(C2(CC(F)(F)F)CC2)=O)nc1 79592,C(C)(C(=O)N1CC(CCNC(=O)C(O)C2CC2)C1)(C1CC1)OC 79593,C(=O)(CCCN=[N+]=[N-])NC1(CC=C)CCN(C(C2CCCC(=O)N2C)=O)C1 79594,Cc1ccc(C=CC(N2CCC2CNC(C2CC(=O)N(C(C)(C)C)C2)=O)=O)o1 79595,C1(C(=O)NCC(=O)NCC2CC2)CC2(CCN(C(C3CCC4(CCC4)C3)=O)C2)C1 79596,c1(C(=O)NC2C(C)CN(C(c3scnc3C3CC3)=O)C2)csc2nnsc12 79597,C1(NC(c2cnn(CC3CCC3)c2)=O)CCCC(NC(c2csc(S)n2)=O)CC1 79598,C1(C(=O)NCC(C)NC(c2cc(Cn3cccn3)on2)=O)(COC)CC=CCC1 79599,c1(N(CC(=O)NCCC)C)nc(=NC2CCCCC2)[nH]c2ncn(CC)c12 79600,N1(C(CCSCC)=O)CC2CCN(C(c3cc(COC)no3)=O)CCC2C1 79601,N1(C(=O)CC2CCC(C(N)=O)O2)CC2CCCC(C1)N2C(=O)Cc1cccnc1Cl 79602,NS(=O)(=O)c1cccc(C(=O)NC2CCCC2CNC(=O)CCc2cnc[nH]2)c1 79603,c1(C(=O)NC23CN(C(c4n(C)cnc4)=O)C(C2)C3)ccc2c(c1)CC2 79604,c1(C(=O)NC2CCCN(Cc3c(C)ccnc3)C2)cc2cc(Cl)ccc2[nH]1 79605,c1(C(N(CCC(C)NC(c2c(CC)con2)=O)C)=O)csc2ccc(F)cc12 79606,N1(C(C(CC)(CO)OC)=O)C2CCC(C(=O)NCC3CCC3(F)F)C1CC2 79607,c1(CC)cc(C(N2CCCC2(C)CNC(=O)C=CCOC)=O)c2c(c1)CCO2 79608,CC(C)(CO)C(=O)NC1CCN(C(c2cnc(C(F)(F)F)o2)=O)C1 79609,CC1(C)C(NC(=O)C(O)CC2CCOCC2)CCN1C(C1CCS(=O)(=O)CC1)=O 79610,N1(C(CN2C(C)CCC2)=O)CCCC(O)(CN(C)C(c2cccnc2CO)=O)C1 79611,CC1OC2(CNC(C3COC(C)C3)=O)CC1(NC(=O)C=Cc1ccco1)C2 79612,c1(CC(=O)NCC(C)N(C(=O)COCCCF)CC)ccc(C)c(C)c1 79613,N1(C(CSCC)=O)CC2CCC1CN2CCOC1CCCCC1C 79614,N1(C(c2n[nH]c(C)c2O)=O)CCC(NC(=O)CCOCC(C)C)CC(C)(C)C1 79615,C1(N(C(=O)C(C)c2ccco2)CCC)CCN(C(c2cc(CO)[nH]n2)=O)C1 79616,c1(C(=O)NCC(CS(C)(=O)=O)(F)F)cc(Br)cc2c1CCCC2 79617,c1(N2CCC(OC)C(C)C2)ccc(S(=O)(=O)NCCSC(C)C)cc1Cl 79618,C1(C(=O)NCCC(C)(C)NC(c2ccc(CC3CC3)s2)=O)CC(O)(C#N)C1 79619,c1(C(=O)NCc2nc(C(N3CCC4CCCC34)C)on2)cncc2n[nH]cc12 79620,Cc1cc2ccc(C(=O)NCC3CCN(C(=O)CCC4CC4(Cl)Cl)CC3)cn2c1 79621,C1(N(C)C(c2ccc(=O)oc2)=O)CCN(C(=O)Cc2cccc(O)c2)CC12CC2 79622,c1(C(=O)NC(CNC(CC(C)c2ccncc2)=O)(C)C2CCC2)cc(Cl)cn1C 79623,c1(C(N2CCC(NC(C=CC(C)(C)SC)=O)C(F)C2)=O)ccc(N)c(Cl)c1O 79624,N1(C(c2nnn3c2C(=O)NCC3)=O)CCN(C(=O)CC2CCC2)C2COCC12 79625,C1(CNC(C(CC)OCC)=O)CCCC(CNC(=O)C=Cc2nc(C)co2)C1 79626,c1(C(=O)NC2CC(CCNC(c3cc4sccc4[nH]3)=O)C2)cc(Cl)c(F)cc1O 79627,CCC(C(=O)OC)C(=O)NCC(C)(C1CC1)NC(C1CC2(CSC2)C1)=O 79628,c1(C(=O)NC(C(C)NC(c2c(CC)c[nH]n2)=O)C)cc(Br)ccc1F 79629,C1(CNC(C(C)c2cccs2)=O)(CNC(c2ccnn2C2CC2)=O)CC1(F)F 79630,c1(CN2C(C(=O)Nc3c(C(N)=O)ncc(C)c3)CC(F)C2)cccc2ncsc12 79631,C=CCC(CC=C)NC(C1CC1C(C)NC(C1CC2(CC2)C1)=O)=O 79632,C(CCC(C)C)(C(=O)NC(c1ccccc1)CC#N)NC(COC)=O 79633,C12(CC(=O)NCCN(C(=O)COC3CC3)CC3CC3)CCCCC1C2(F)F 79634,c1(OC)c(C(N2CCC(N(C)Cc3ccc(Br)cc3C)C2)=O)cccc1F 79635,N1(C(c2cnn3c2CCCC3)=O)CC(O)(C2CCN(C(C3CC34CC4)=O)CC2)C1 79636,C(=O)(C1=NNC(=O)CC1)N1CCC(NC(C(Cn2ccc(C)n2)C)=O)C1C(C)C 79637,Cc1cc(O)cc(C)c1C(N1CC2(CCC(NCc3cccc(Cl)c3O)C2)C1)=O 79638,c1(C(N2CC(CNC(CCC=C)=O)C3(C2)CCC3)=O)ccc(F)c2ccncc12 79639,n1(CC)cc(C(N2CCCC2C(C)NC(c2cc(Cl)c[nH]2)=O)=O)c(C)n1 79640,c1(C(=O)NC2C(NC(C3=CCCC3C)=O)CCCC2)cccc2c1OCCC2 79641,C1(CC(=O)NCC(C2CC2)NC(=O)C(C)=C(C)C)(CC)CCC1 79642,c1(C(N2CC(CNC(C(CC=C)C)=O)(OC)C2)=O)ccc2[nH]c(=N)n(C)c2c1 79643,N1(C(CC2C(C)OCC2)=O)CC2COCC2(C(=O)NC2(C3CC3)CCOC2)C1 79644,C(C)(CO)(C(=O)NC1COCC1NC(=O)CC(C)O)NC(C)=O 79645,C=CC1(NC(C2CN(C(=O)C(C3CCCC3)OC)CCO2)=O)CCCC1 79646,c1(-c2nc(C(C)O)nn2Cc2ccc(Cl)cc2)oc2ccccc2c1Cl 79647,C1(C(C)NC(C(C)=O)=O)CCN(C(C2CC23CC3)=O)C1 79648,c1(C(N2C(C(=O)Nc3cc(C)c(O)cn3)CCCC2)=O)cc(F)c(C)c(F)c1 79649,C1(NC(C(C)NC(C)=O)=O)CC2CCC1CN(C(=O)C(c1c(C)n[nH]c1C)C)C2 79650,C12(C(N3CC(O)(CCNC(c4ccc(C)c(C)n4)=O)C3)=O)CC3CC1C2C3(F)F 79651,C1(NC(CCOC)=O)CN(C(c2cc(C3CCCO3)n(C)n2)=O)C2(CCCC2)C1 79652,C1(F)(CNC(C(CC)N(C)C)=O)CCC(NC(C2(C)CC(F)(F)C2)=O)C1 79653,CCCC(CCCNC(c1cc[n+]([O-])cc1)=O)NC(C1CCCN(C)C1)=O 79654,C(=O)(C(F)(F)C(F)(F)C(=O)O)N1C2(CCCN(C(c3cc(C)[nH]c3)=O)C2)CC1 79655,Cc1nc2ncnn2c(NC(N2CCc3c(ccnc3Cl)C2)=O)c1C#N 79656,C1(Cl)(C(=O)NCC#CCNC(c2c[nH]nc2C(F)F)=O)CC1(F)F 79657,N1(C(c2ccccn2)=O)CCC2(CCN(S(=O)(=O)c3cccc(Br)c3F)CC2)C1 79658,C1(CNC(c2cc(C(F)(F)F)no2)=O)COCCN1C(c1coc(O)n1)=O 79659,C=CC(C)(CCOC)C(=O)N1CCOC(C(N2CC(c3cc[nH]n3)C2)=O)C1 79660,C#CCCC(O)C(=O)N1CC2(CNC(=O)COC3(C)CCCC3)CCC1C2 79661,N1(C(=O)CCCc2ccccc2)CC2CN(C(c3ccc(Cl)cc3)=O)C2C1 79662,C1(C(=O)NC(c2n(CC)ncc2)C)C=CCCN1C(=O)C(C)N1CCCC1 79663,c1(C(=O)NC(c2ccccc2)CNC(C(C2CCC2)OC)=O)cccnn1 79664,c1(OC)cc(C(N2CCCCC(CNC(C3(O)CCC3)=O)C2)=O)cc(F)c1F 79665,N1(Cc2c(C)noc2C)CCN(C(=O)Cc2ccc(Cl)s2)C2(CC2)C1 79666,c1(CC(=O)NC(CNC(C2CC(=O)NC2)=O)Cc2ccccc2)ccc(F)cn1 79667,CN1CCC(C)(C(=O)NCCNC(c2cc(N3CCOCC3)ccn2)=O)C1=O 79668,S(=O)(=O)(c1cc(C(=O)NCC(C2(C)CCCCC2)=O)n(C)c1)N1CCCC(C)C1 79669,c1(C(N2C(C)(CNC(C3(CCF)CCC3)=O)CCC2)=O)ccn2nccc2c1 79670,C1(CCC)CN(C(c2cn(C)nn2)=O)CCN1C(c1cc(CC2CC2)on1)=O 79671,c1(CN(C(C(Cc2cc[nH]n2)NC(c2cc(CC)sn2)=O)=O)C)cc(C)ccn1 79672,C(CCC(=O)N1CC(c2cn(CC(C)C)nn2)(N(C)C)C1)NC(=O)OCC 79673,C1(NC(CC2(C(=O)OC)CC2)=O)CCN(C(=O)CCc2ccncc2)CC1C 79674,Cc1cc(C)c2[nH]c(C(=O)NC3CC4CC3CN4C(=O)Cc3cscn3)cc2c1 79675,Cc1nc(-c2ncc[nH]2)sc1C(=O)NC1CCN(C(=O)CC2CN(C)C2)CC1 79676,N1(C(c2ccc(C(=O)OC)s2)=O)CC(NC(c2cccc(O)n2)=O)CC2(CC2)C1 79677,c1(CNc2cc(C(=O)OC)sc2)ccc2c(c1)OCC2 79678,C(=O)(C(F)CC(C)(C)C)NCC(C(=O)NCCc1cc(C)ns1)N(C)C 79679,C(CN=c1[nH]c(N2CCCC(N(C)C)C2)nc2c1CC(C)CC2)NC(COC)=O 79680,Cc1cc(Cl)ccc1OC(C)C(=O)NCC(F)CNC(C1(CC(F)(F)F)CC1)=O 79681,c1(C(=O)NC2CC2C(=O)Nc2ccn3ncnc3c2)ccc2cccc(F)c2n1 79682,c1(SCC(=O)NC(c2ccccc2)CNC(C=C(COC)C)=O)ccc(C)cc1 79683,C1(C(C)C)NCC12CCN(C(c1ncccc1N)=O)CC2 79684,C(=O)(C1=CCC(NC(c2ncsc2C)=O)C1)N1CCC(C(=O)OCC)C1 79685,c1(C(=O)NC2C(C(N(CCCC)CCCO)=O)CCC2)cc(C)cc(O)c1 79686,CCC(CC(=O)NCC(N1CCN(C(=O)C(C)(C)OC)CC1)C(F)F)SC 79687,Cc1noc(C)c1CC(C)C(=O)NCC1CC(NC(c2[nH]nnc2C(F)F)=O)C1 79688,c1(C(N(C2CN(C(CNC(C)=O)=O)CC2(C)C)C)=O)cc2ccc(C)cn2c1 79689,Cc1cc(OC(=O)C(C)(C)CCc2cc(Cl)sc2Cl)ccc1Oc1ccccc1 79690,C1(CC)CCC(C(=O)NCC(C(=O)N(CCC(=O)NC)C)N(C)C)O1 79691,S(=O)(=O)(c1ccc(Br)cc1[N+](=O)[O-])C1CCN1Cc1c(CCN=[N+]=[N-])ccc(Cl)c1 79692,C1(CNC(c2c(CCC)cccc2)=O)CC2(CC2)CN1C(C1CCC(C)O1)=O 79693,c1(C(=O)NCCNC(c2ncc(C)cc2F)=O)cc2sc(C)cc2n1CC1CC1 79694,C(=O)(C1=CCS(=O)(=O)C1)N1CC(NC(c2ccncc2)=O)C(CO)CC1 79695,c1(C(=O)NCC2(O)CCN(C(CCCOCCC)=O)C2)c(F)cc(F)c(F)c1F 79696,C1(C(C)NC(=O)NCc2cc(C(N)=O)ccn2)CN(C)CCN1C 79697,C1(NC(CN(S(C)(=O)=O)C)=O)CC1C1CCCN(C(c2cc[nH]c(=N)c2N)=O)C1 79698,c1(C(=O)NCCOCCN(C(C(C)c2ccco2)=O)C)sccc1NS(C)(=O)=O 79699,n1(CC)nnc2c1CCC(C(N1CCN(C(=O)CC(C)C3CC3)CC(O)C1)=O)C2 79700,c1(C(=O)NCCc2cnc(NC(c3c(C)c(Cl)ccc3)=O)s2)cc(F)c(F)cc1O 79701,N1(C(COc2cccc(C)c2)=O)CC=C(CNC(C2(O)CC(C)(C)C2)=O)CC1 79702,N1(C(CCCC#CC)=O)CCC(C2(NC(c3cnc(N(C)C)c(Cl)c3)=O)CC2)C1 79703,C(=O)(C1CCCc2sccc21)NC(CC(C)C)CNC(=O)C(c1ccnn1C)O 79704,C=CCC(C(=O)N1CC(OCCNC(c2nc(C)c(C)s2)=O)C1)C(C)C 79705,c1(C(N2CCN(CC(=O)Nc3ccc(F)c(Cl)c3)CC2)=O)ccc(Cl)cc1Cl 79706,C=CCC(C)(O)C(=O)N1CC2CC1C2NC(c1ccc(C(C)C)cc1)=O 79707,c1(C(=O)NCc2cc(C(=O)NCC3CC(=C4CCC4)C3)sc2)ccc(O)nn1 79708,Cc1ncc(Cl)cc1C(=O)N(C)CCN(C)C(c1cccc(F)c1F)=O 79709,c1(C(=O)NC23C(CCN(C(c4cn(C)nc4)=O)CC2)C3)cc([N+](=O)[O-])ccc1Cl 79710,N1(C(C(C)c2ccsc2)=O)CCOC(CNC(c2ncsc2C(F)(F)F)=O)C1 79711,C1(C(=O)N(C)CC2CCCN2C(c2c(Cl)n[nH]c2C)=O)(OCC)CCCCCC1 79712,CC1=C(C(=O)N2CCC(NC(=O)CN3CCNC(=O)C3)C23CC3)CCO1 79713,c1(C(C)C)ccc(O)c(C(=O)NCCCNC(c2cc(F)ccc2Cl)=O)c1 79714,CC1(CNC(c2ccsc2Cl)=O)CCN(C(c2cnc(Br)s2)=O)C1 79715,C1(C(=O)NC(CC#CC)CO)CN(C(=O)C#CC2CC2)C2(CCC2)C1 79716,N1(C(c2n(C)ncc2Br)=O)CCC2C1CCCN2C(c1cccn(C)c1=O)=O 79717,Cc1cccc(S(=O)(=O)N2C3CN(Cc4cc([N+](=O)[O-])ccc4O)CC23)c1 79718,N1(C(C2CC(C)OC2C)=O)CCC(F)(F)C(CNC(=O)CC(C)C2CC2)C1 79719,C(=O)(C(C(C)(C)C)NC(=O)C(C)=C(C)C)N1CCC(CC)CC1 79720,N1(C(C=CCCC)=O)CCC2CCN(C(=O)CCC3CCC3)C2C1 79721,C1(CNC(C2(N(C)C)CCCC2)=O)CC(C(=O)NCC2CC(O)C(O)C2)=NO1 79722,c1(C(N2CC(C(Cn3cc(CCC(C)O)nn3)F)C2)=O)cc([N+](=O)[O-])cnc1Cl 79723,c1(SC)ncc(C(=O)NCCC2CCCCN2C(C2CN(C)CCO2)=O)c(O)n1 79724,C1(NC(C(CCC)(C)C)=O)CN(C(=O)Cc2cnc(C)o2)C2(CCCCC2)C1 79725,C1(NC(C(CC=C)C)=O)CN(C(C23C(=O)C4CCC2C3C4)=O)CC1C1CC1 79726,C1(C(=O)NC(c2cncs2)C)CCC(C(C)C)N1C(=O)COC1CCCC1 79727,C(=O)(CCC(C)(C)OC)NC(CC#C)C(=O)N(C)CCOCCOC 79728,c1(C(N(CCCCCCNC(C(CC)N(C)C)=O)C)=O)cc(OC)nc(Cl)c1 79729,N1(C(C=CC)=O)CC2(CCOCC2)CC1CNC(c1cc2oc(Cl)cc2[nH]1)=O 79730,C1(NC(CC(COC)(C)O)=O)CN(C(=O)C=C2SCC(=O)N2C)C2(CCCC2)C1 79731,C(C)(C)(C(C)CC(=O)N(C(C)CCCC)CCCO)N(C(C=CCC)=O)CCC 79732,N1(C(C(CC)(F)F)=O)CCC(CNC(C2(C)CCCOC2)=O)C(C2CC2)C1 79733,Cc1cc(C)nc(-c2cccc(NC(=O)C(N3CCC(C)C(CO)C3)=O)c2)n1 79734,c1(CC(=O)NC(CC(C)NC(CNC(C(CC)C)=O)=O)C)sc(C2CC2)nc1C 79735,N1(C(COC(CC)(C)C)=O)CC=CC1CNC(c1cnnn1C1CC1)=O 79736,c1(C(=O)NC2CCCN(C(C(C=C=C)C)=O)C2)ccc2c(c1)NC(=O)CC2 79737,N1(C(C(C)OC)=O)CCC2C(CCCN2C(=O)Cc2coc3cc(C)ccc23)C1 79738,c1(OC)cc(C(=O)NC2CCCC2CNC(C2COC(=O)O2)=O)cc([N+](=O)[O-])c1 79739,c1(C(=O)OC)ccc2c(c1)C(CNC(=O)NNC(=O)C1CCCC1)CCC2 79740,C1(C(N(CCN(C)C)C)=O)COC2CN(C(=O)Nc3cccc4nc[nH]c34)CC12 79741,c1(C(=O)NCC(=C)CCNC(c2ccc(O)c(F)c2)=O)c([N+](=O)[O-])cnn1CC 79742,C1(CC)C(NC(C2C=CCS2)=O)CCCN1C(C1CCCC(=O)N1C)=O 79743,C1(NC(CCCC)=O)CCCC2CN(C(=O)C=Cc3ccc4c(c3)CCO4)CC12 79744,N1(C(C#CC(C)(C)C)=O)CCOC2(CCCN(C(=O)CC3CCCCC3O)C2)C1 79745,C(=O)(CN=c1ccc(Cl)n[nH]1)N1C2C(NC(C3(NC(C)=O)CCC3)=O)C(C2)C1 79746,c1(OCC(C)C)cccc(CC(=O)NC2(C)CCN(C(=O)Cc3cnoc3)C2)c1 79747,CC(C)C(N=c1[nH]nc(O)s1)C(c1ccccc1)NC(c1c[nH]ccc1=O)=O 79748,c1(OC)ccc(C(N2CC(CNC(c3cnc(C)n3C)=O)CC2(C)C)=O)c(Cl)c1 79749,c1(OC)cncc(C(N2CCN(C(=O)CC3(C4CC4)CC3)CC2)=O)n1 79750,C1(C(N2CCC(C(CNC(CN(C)CC)=O)(C)O)CC2)=O)CCn2ccnc2C1 79751,CCC(CCN1CCCCC1)OC.C(CC(C)(C)O)N(C=O)C 79752,C1(NC(c2cc(C)sn2)=O)CN(C(c2ccc(N)cc2O)=O)CCC1C 79753,C1(O)(CNC(C(C)OC)=O)CCN(C(c2cnn(C(C)(C)C)c2)=O)C1 79754,N1(C(C2(OC)CC2)=O)CCC2CCC(C1)N2C(c1cc(Cl)cc(Cl)c1[N+](=O)[O-])=O 79755,CCCCC(O)C(=O)NCC(CC)NC(C1C(C)C1C)=O 79756,N1(CC)C(C)CN(C(=O)CN(C(C2CC2(F)Cl)=O)CC2CC2)CC1C 79757,N1(C(C2C(C(C)(C)C)C2)=O)CC2CCC1C(CNC(=O)CN1CSCCSC1)C2 79758,Cc1ccc(C(=O)NCCC(C)N(C)C(C2CCS(=O)(=O)N2)=O)c(Cl)c1 79759,N1(C(CSCC=C)=O)CCC(F)(CNC(c2cnn(CCC#N)c2C)=O)CC1 79760,CCCCCC(O)C(=O)N1CCN(C(c2n[nH]c(C)c2[N+](=O)[O-])=O)CC(C)C1 79761,c1(NC(C2(C)CCOCC2)c2n(CCCC)nnn2)cccc(S(C)=O)c1 79762,S(=O)(=O)(c1cc(F)cc(Br)c1)N1C2CC(N(c3ccccc3)C)CC1CC2 79763,O(C1CCCc2ccccc21)CC(N1CC(NC(=O)C=CCF)C(C(F)F)C1)=O 79764,c1(C(=O)NC2(COC)CN(C(C3C(CC)CCCC3)=O)C2)ccc(O)cc1F 79765,C1(CNC(c2n(C)ccc2)=O)C(C2CC2)CCN1C(C1C(C)(C)C1(C)C)=O 79766,C(=O)(CC(O)CC(C)C)NC(CC#C)(C)C(=O)N1CC(CC(F)F)C1 79767,c1(-n2ccc(C(=O)NCC3C(C)C3C)n2)ccccc1F 79768,C1(NC(C)=O)CN(C(C2(C(=O)OCC)CCO2)=O)C2CCCCC12 79769,C12CSCCN1C2=O.c1(COC2(CC(=O)NC3CC=CCC3)CC2)ccccc1 79770,C(N=c1[nH]c2c(c(=NCc3cccc(C(F)F)c3)[nH]1)CCC2)c1c(CC)nns1 79771,C(CCN=c1[nH]c2c(c(=NCCSCCC(F)(F)F)[nH]1)CSC2)c1nc(=N)[nH][nH]1 79772,C#CC1(NC(C2(NC(=O)C(CC)OCC)CCN(C)C2)=O)CC2CCCC12 79773,C1(NC(CN(c2ccncc2)C)=O)CN(C(C2CCOC2C2CC2)=O)CC12CC2 79774,CCC(CC)C(F)C(=O)NC(CNC(c1cccc2ccoc12)=O)C(C)(C)C 79775,C1(CC(C)NC(COCC(C)C)=O)CN(C(C2CCC2)=O)C1 79776,CCC(CNC(=O)C(C)(C1CC1)N(C(=O)CC1CCCCC1)C)(CC)C(N)=O 79777,CCCCC(CC(=O)N1CCC=CC1CO)NC(C1(N2CCCC2)CC1)=O 79778,c1(C(=O)NCC2(F)CN(C(C3(C)CCOC3)=O)C2)cc2scnc2[nH]1 79779,c1(C(N(C(C)C)CCNC(c2cnn(C3CC3)c2Cl)=O)=O)cc(F)c(F)cc1Cl 79780,C1(CN(C(c2c(CC)ocn2)=O)C)CCCCN1C(c1ccn(C(F)F)n1)=O 79781,C1(NC(c2cn(CCC3CC3)nn2)=O)COCCN(C(=O)CC23CCCC2C3)C1 79782,N1(CC(=O)NC(c2ccnn2C)CN)CCC(C)(C)CC1.C1(C(=O)C(C)=O)OCCC1N 79783,C(=O)(CC(F)(F)F)NC(C)C(=O)N(CC(O)CN(C(=O)CCc1cnoc1)C)C 79784,CN1CCC(CC(=O)N2CCN(C(=O)C(N)=O)CC23CC3)c2ccccc21 79785,c1(SCC(=O)NC(CNC(c2cn(CCCOC)nc2)=O)CO)ccc(F)cc1 79786,C1(F)(CNC(c2cnc(S)[nH]2)=O)CCC(CNC(=O)C(O)C2CCC2)CC1 79787,C(CCF)(C(=O)NCC(O)CCC1CC1)NC(C1ON=C(C)C1)=O 79788,c1(OC)cc(N)c(C(N2CCCC(O)(CNC(c3ccc(Cl)s3)=O)C2)=O)c(F)c1 79789,c1(N(C)CC)ccc(C(=O)NCCCN(C2CCCC2)C(C2C(C)CC2C)=O)cc1 79790,c1(C(=O)NC(C2CCCC2)CNC(CCSCC(N)=O)=O)cc2cccnc2[nH]1 79791,C1(C(=O)NCC2CCN(C(=O)OC)C2)CC(=O)N(c2cn[nH]c2)C1 79792,C(c1ccc(C(F)F)o1)=CC(=O)NCCC(C)NC(c1cc(Cl)c[nH]1)=O 79793,C1(NC(C=CC(CC)=CC)=O)CCOC2(CCN(C(=O)C(C)(C)SC)CC2)C1 79794,C=CCCC(C(=O)N1CCCC(C(=O)NC)C1)NC(C1CCCSC1)=O 79795,c1(CNC(C2CCSC2)=O)ccc2c(c1)CN(C(C1CCCC(CF)C1)=O)C2 79796,C=CCC(C)(C(=O)N1CC2(C1)CN(C(C1(OC)CS(=O)(=O)C1)=O)C2)N(C)C 79797,C(=O)(CC(C)(C(F)(F)F)N(C)C)OC(c1ccc(F)nc1)C 79798,c1(CC(=O)N(c2ccc(F)cc2)CCCO)c[nH]c2cc(Cl)ccc12 79799,O=S(=O)(c1ccc(Br)c(Cl)c1)N1CC2CN(Cc3cnc4ccccn34)C2C1 79800,c1(CNC(c2n(C)nnn2)C2CC(C)(C)C2)cncc(C(C)(F)F)c1 79801,c1(C(=O)NC2CN(C(c3c(NCC)scn3)=O)CC2SC)c(OC)cccc1O 79802,N1(C(C=CC=CCC)=O)CC(CNC(c2cc3ccsc3s2)=O)C2(CCC2)C1 79803,C(C(CC(=O)N(C1CCC(F)(F)C1)C)NC(C1CC(F)(F)C1)=O)OC 79804,N(C1CN(C(=O)CC2CC3CC3C2)CCc2ccccc21)C(C=CC)=O 79805,c1(OC)ccc(CC2CCN(C(c3ccccc3)=O)CC2)cc1C(F)(F)F 79806,c1(C(=O)NCCCN(C(C(CC)SC)=O)CC)cccc2ncoc12 79807,C12(NC(CCOCC#C)=O)CCCC1N(C(c1cc(C(N)=O)ccc1C)=O)CC2 79808,C1(CC(=O)NCCC2CC(C(=O)NC(C(C)C)C3CC3)C2)COCC1O 79809,c1(N2CCC3=C(CC(=O)N3C)C2)cn(C)c(=O)c2cnccc12 79810,c1(C(N(CCN(C(COCCCCC)=O)C)C(C)C)=O)nccn1C 79811,C1(CCOC)(NC(=O)C=C(C)CN2CCOCC2)CCN(C(=O)CS(N)(=O)=O)C1 79812,C1(CNC(CC2(CSC)CC2)=O)CC(NC(C2(C3CC3)CCC2)=O)C(O)C1 79813,C1(CNC(=O)CC2CCC3CC23)(NC(=O)CSc2cccc(O)c2)CCOCC1 79814,CCC(C)C(C)N(C(=O)C(=O)N(C)CCC1CCCCC1)C1CC1 79815,c1(C(N(CC(=O)NCC2CC2)CCC(O)CO)=O)cnc(C2CC2)o1 79816,C1(NC(C2CNC(=O)O2)=O)C2CC1N(C(C13CCCCC1C3)=O)C2 79817,C(=O)(C(C)CC(C)(C)C)NC12C(NC(C(C(CC)O)C)=O)CC(CC1)C2 79818,c1(CCNCC2C(c3ccc(C(=O)OC)cc3)C2)ccc(F)cc1Cl 79819,N1(C(C(CCC)NC(c2ccc(C#C)cc2)=O)=O)CC(C)(C)CCC1C 79820,C1(C(N(CCNC(c2cn(CC(F)(F)F)nn2)=O)C2CC2)=O)CCC2(CCC2)O1 79821,C12(C(=O)NCC3N(C(CC4C(CC)C4)=O)CC(F)C3)CCCN(CCC1)C2 79822,C1(N(C(C(C)CO)=O)C)CCCCN(C(C2(c3cccnc3Cl)CC2)=O)C1 79823,Cc1ccncc1C(C)NC(c1nc(CNC(c2cc(C)c(C)[nH]2)=O)oc1C)=O 79824,N1(C(=O)NCCOCCCC)CCC(CC#N)C(F)(F)CC1 79825,C(=O)(C1CCCc2sccc21)N1C2C(NC(C3C(CCC)CCC3)=O)C(C2)C1 79826,C(=O)(C1=Cc2ccccc2C1)NCC(CNC(CCCOCCOCC)=O)F 79827,c1(C(N2CCN(C(c3c(C)nsc3)=O)CC2C#N)=O)ccc(Cl)c2[nH]ccc12 79828,Cc1n[nH]cc1C(=O)NC(C)CCN(C(=O)CC1(O)CCOC1)C 79829,C1(C(N(C2CCN(C(C(CN(C)C)(C)C)=O)C2)C)=O)CC2CCC(C1)N2C 79830,c1(CNC(C2C3CN(C(C(C)Cc4ccco4)=O)CC32)=O)cc(F)ccc1[N+](=O)[O-] 79831,c1(C(=O)NCCCNC(C2(Oc3ccc(Cl)cc3)CC2)=O)cccc2c1CCO2 79832,c1(-c2cc(C(=O)Nc3c(SC(C)(C)C)cccc3)no2)ccc(Br)cc1[N+](=O)[O-] 79833,C1(NC(C(C)(C)n2cc(Cl)cn2)=O)CCC(O)CN(C(C2CC2(F)F)=O)C1 79834,C1(S(N)(=O)=O)(C(=O)NCCCCCNC(c2c(SC)cnn2C)=O)CCC1 79835,C(=O)(C(C(=O)N1CCCCC1CNC(=O)CCCCC(C)=O)C(C)(C)C)OCC 79836,Cc1cc(C(=O)NC(C)(C)CCNC(=O)C(C)CS(C)(=O)=O)c2occc2c1 79837,c1(C(=O)NCC(C)(C2CCC2)NC(COCCC=C)=O)c(C)ncn1O 79838,c1(CC)nc(C(=O)NC2CCC(CC(=O)N(C)Cc3cc(=O)cc[nH]3)C2)c(C)o1 79839,c1(SC)cc(C(=O)Nc2cccnn2)co1 79840,N1(C(c2c(CC)nc[nH]2)=O)CCN(C(c2cc(C)on2)=O)C2(CCC2)C1 79841,C1(NC(CCOCCOC)=O)CS(=O)(=O)CC1NC(c1cc(OC)ns1)=O 79842,C(=O)(CCC(C)(C)F)NCC(C)N(C(c1ccc(OC2CCCC2)cc1)=O)CC 79843,N1(C(C(C)(C)OCC)=O)CC2(CC(NC(c3ccc(CO)nc3)=O)CO2)C1 79844,c1(C(=O)NC2CCCN(C(CSCC#C)=O)C2C)ccc2c(c1)N(C)C(=O)CO2 79845,C1(C(N(C(CNC(=O)C2=CC(C)(C)C2)C2CC2)C)=O)CCCN2CCCCC12 79846,Cc1cc(C(=O)NCCC(C)NC(=O)C(F)Oc2ccc(Cl)c(F)c2)cc(O)c1 79847,c1(C(=O)NCC(C(C)C)NC(C2CCCOCC2)=O)n[nH]c2c1CN(C)CC2 79848,CCC(CC(=O)N1CC(C(=O)NC2(c3cc[nH]n3)CC2)C(F)(F)C1)C(F)F 79849,N1(C(C(CC)(C)F)=O)CCC(C2CCN(C(c3cc(C)cc(C)c3N)=O)C2)CC1 79850,N1(CCC)CC(C(=O)NCCCCN(C(=O)CC2CC2(Cl)Cl)C)CC1=O 79851,c1(C(=O)NC2C(NC(C3(C)CC3)=O)COC2)ccnc(OC2CCOC2)c1 79852,N1(C(C)CNC(C2CCCCO2)=O)CCN(C(c2ccncc2Cl)=O)CC1 79853,C1(CC(=O)NCC2C(C)CN(C(=O)CN(S(C)(=O)=O)C)C2)CCCC(C)(C)C1 79854,N(C(=NCCCCl)NCC(Cc1ccccc1F)CO)CCN1CC(=O)NCC1 79855,C1(N(C)C(C2CC(C)(C)C2)=O)CCCCN(C(C2(N(C)C)CCCSC2)=O)C1 79856,n1(CCC)ccc(=NC(=O)C2(F)CCCN(C(C34CCC(C3)C4(C)C)=O)C2)[nH]1 79857,c1(COC(C(=O)NC(C)CN(C)C(c2sccc2F)=O)C)ccc(Cl)cc1 79858,N#Cc1ccc(NC(=O)NC(=O)C(c2ccccc2)Sc2ccc(Br)cc2)cc1 79859,C=C(C)C1CN(C(=O)C(=O)NN(C(=O)OC(C)(C)C)CCC2CC2)CCO1 79860,N1(C(c2c(C)c[nH]c2)=O)CCC2(CC1)COC(C)C2N(CC(F)F)C 79861,c1(C(N(CCC[Si](C)(C)C)C)=O)ccn2ncc(Br)c2c1 79862,c1(OC)cnncc1C(=O)N(C)CC1CCN(C(C2CCNC2=O)=O)C1 79863,C1(NC(c2cc(CC)nn2C)=O)CN(C(C2C=CCC2)=O)CCC1(C)C 79864,c1(SC)ccc(C)c(NC(=O)NCC2(O)CCS(=O)(=O)C2)c1 79865,C1(n2cc(CC(C)C)nn2)CCN(C(c2cn(CCO)nc2C2CC2)=O)CC1O 79866,CCCCCCCCCC(O)CC(=O)N1C2CC1CN(C(=O)C(O)C(C)CC)C2 79867,C(C(=O)N(CCOCCO)CC1CC1)(C1CC1)OC.C1(=O)C(C)ON1 79868,CC1(CNC(C2CC=CCC2C(F)(F)F)=O)CCN(C(c2csc(=N)[nH]2)=O)CC1 79869,C1(C(N2C(CC(=O)NCc3cnc(CC)[nH]3)CCCC2)=O)C2C3CCC(C3)C12 79870,C=C(C)CCC(C)N=c1[nH]c(=NCC2(C)CC2)c2ccc(C)cc2[nH]1 79871,c1(C(=O)NC(C2CCOC2)C)cc2occc2[nH]1 79872,c1(-c2ncc(C(=O)NCC(CO)NC(c3cccs3)=O)s2)ccccc1Cl 79873,C(=O)(CCCNC(=O)C(C)NC(=O)C1CC1)NCC(C)(C)OCC(C)C 79874,Cc1ccnc2c(C(=O)NC(C)CC3CCN(C(=O)CC(C)C)CC3)cccc12 79875,C(=O)(C(C)(C)C(=O)N(CC(C)C(=O)NCc1nc(C#N)cs1)C)NC 79876,N1(C(CC(C)C2CC2)=O)C2CCC1CC(N(C(=O)C(C)(C)C1CCC1)C)C2 79877,N1(C(c2c[nH]nc2C2CC2)=O)CCN(C(C2(C3CCC3)CC2)=O)C2CCCC12 79878,CC1CCC(CC(N2CCCC(CN(C)C(c3nnn(C)n3)=O)C2)=O)CC1 79879,C1(NC(c2cc(C)cc(Cl)c2)=O)CS(=O)(=O)C2CN(C(C3CSC3)=O)CC12 79880,N1(C(C2CCN(C(c3c(CC)con3)=O)C2C(C)C)=O)CCC(C2CCC2)CC1 79881,c1(OCCC(=O)NCC(CN(C(C2(C#C)CC2)=O)C)O)ccc(F)cc1Cl 79882,Cc1cnc(NC(C2CN(C(=O)CCCCCO)CCC2O)=O)c(C)c1 79883,C1(C(=O)NCC(C)(CO)NC(c2ccc(C)c(C)n2)=O)(CC)CCC(O)CC1 79884,CC1CN(C(C2CCC(C)(C)N(C(=O)CC3CSC3)C2)=O)Cc2c[nH]nc21 79885,N1(C(CC(CC)O)=O)CCN(C(c2ccccc2-n2cccc2)=O)CCC1C 79886,c1(OCCCC(=O)NCC(C)NC(=O)CN)ccc(F)cc1.C(=O)(C1CC1)N(CCO)C 79887,C(=O)(C(F)(F)CSC1CC1)N(CCOCCNC(c1c(C)con1)=O)C 79888,n1(CC(=O)NCCC(C)N(C(CC(C)(C)OC)=O)C)cc([N+](=O)[O-])cn1 79889,CCCC(C(=O)NCc1ncccc1C(=O)N(c1cnn(C)c1)CC)NC(N)=O 79890,C(=O)(CC(C(F)(F)F)NC(C12CCC(CC1)C2)=O)N(c1cnc(C2CC2)nc1)C 79891,N1(C(C=CC(C)NC(=O)CC2=NN(C)C(=O)C2)=O)CCOC2COCC2C1 79892,Cc1ncc(Cl)c(-c2nc(CP(C)(C)=O)no2)n1 79893,C1(C(=O)NCCN(C(=O)CC2CC(=O)C2)CC)CC(n2cnnc2)C1 79894,N1(C(C(=O)NCCNC(C)=O)=O)CCN(C(c2coc(O)n2)=O)CC1 79895,c1(CNC(=O)Nc2c(C)c(F)ccc2)cccc2c1cnn2C(=O)NC(C)(C)C 79896,N1(C(C(CCOC)C)=O)CCC(NC(C2CCN2C)=O)C12CC2 79897,N1(C(C2(C)CSC2)=O)CCC(CNC(C2(C)CCC(=O)NC2)=O)C(F)(F)C1 79898,C1(C(=O)NC2CCN(CC)C2)CCN(C(=O)c2cccn2C2CC2)O1 79899,C12(NC(CN(CC)CC)=O)CC(C)(C1)OC21CN(C(c2cc(C)c(C)cc2C)=O)C1 79900,C1(CNC(CCCCN(C(C)C)C)=O)CCC2(CCN(C(=O)C3CC3)CC2)CO1 79901,C1(C)(CC(=O)NC(C)(C)CF)CCN1C(=O)COc1ccccc1 79902,CCCC(C(=O)N1CC(N(C)C(c2ccc(CS(C)(=O)=O)cc2)=O)C1)NC(N)=O 79903,C1(NC(C2CC(OCC)C2)=O)CCN(C(=O)C(C)=CCCN2CCCC2)CC1 79904,c1(CNC(C=CC2N(C(C(CC)CN(C)C)=O)CCC2)=O)ccc(F)cc1F 79905,C1(NC(CNC(=O)OC)=O)CCOC12CCN(C(c1cc(=O)n(C)o1)=O)CC2 79906,Cn1cccc1-c1cn(CCCC(=O)NCC(C(=O)O)C2CCCCC2)nn1 79907,Cc1nnc2cc(NCC3CCCC(CNC(C4(COC(C)=O)CC4)=O)C3)ncn12 79908,N1(C(C(CC)O)=O)CCC(n2cc(NC(=O)CSc3nc[nH]n3)nn2)CC1 79909,CCC(F)(F)C(C)(C)C(=O)N1CC2CCC1CN(C(c1[nH]nnc1C)=O)C2 79910,N1(C(C2(CC)CC2)=O)CCC2C1CCCN2C(=O)C=Cc1ccccc1[N+](=O)[O-] 79911,C12(C(N)=O)COCC1CN(c1nc(-n3cnnc3C3CC3)cs1)C2 79912,c1(C(C(=O)Nc2ccccc2)N(C(C(=O)OCC)CC)C)cc(C)nn1CC 79913,c1(C(=O)NC(c2cnn(C)c2)C(=O)NC(CC(=O)OCC)C)cccc(C)c1O 79914,c1(C(N2CCC(C(C)(C)C)(CNC(CC3(OC)CC3)=O)C2)=O)cc(C)nc(C)c1 79915,CON(C)CCCNC(C1C=CCCN1C(=O)CC1(C)OCCO1)=O 79916,C(CCCCC(=O)NC(C)C(C(C)C)NC(C1CCSCC1)=O)OC 79917,O=C(CC1C(=O)Nc2cc(Cl)ccc21)NC1(CCO)CS(=O)(=O)C1 79918,C(CC(C)C)(C(=O)NC1CC(CNC(=O)Cc2c(C)noc2Cl)C1)NC(C)=O 79919,c1(C(=O)NCC2(COC)CN(C(C3C(C)(CC)C3)=O)C2)c(C)nc(C)n1O 79920,c1(C(=O)NCC2C(NC(=O)Cn3cncn3)C2)c[nH]cc1C1CC1 79921,C1(C)(CNC(C(c2ccc(C)o2)C)=O)CCCN(C(c2cn(C(C)C)nn2)=O)C1 79922,C1(CNC(=O)NCC2CCN(C(=O)OC)C2)CCC=CCCC1 79923,C1(CNC(=O)COc2ccc(F)cc2Cl)CN(C(C2(O)COC2)=O)CCC1(F)F 79924,C1(NC(COC(CC)(C)C)=O)CCCC(C(=O)NCCN(CCCF)C)C1 79925,C1(C(C)(C)O)CCCN(C(C2(C)CN(C(=O)Cc3cccc(Cl)c3)C2)=O)C1 79926,C=C(C)CCCN=c1c(Br)ccc(NC(=O)CNC(=O)C(C)(C)C)[nH]1 79927,C1(NC(C(C(C)(C)C)n2cc(C(CC)N(C)C)nn2)=O)CCC([N+](=O)[O-])CC1 79928,C1(NC(C2C(CNC(c3c(CC)oc(C)c3)=O)CCC2)=O)CC2CC1C(O)C2O 79929,C1(CNC(C(CCCC)O)=O)CCC12CCN(C(c1cnc(C)[nH]1)=O)CC2 79930,N1(C(C=CC2N(C)CCC2)=O)CCN(C(c2cc[nH]c(=N)c2)=O)CC1CC(F)F 79931,C1(CN(C(=O)CNC(c2ncc[nH]2)=O)CC)CC1C1CC1 79932,C1(NC(CC(C)c2ccco2)=O)CN(C(c2cn(C)nc2O)=O)CCC12CCC2 79933,CC1CN(C(c2cn(C)c(=O)n2C)=O)CCC1NC(C1(CO)CCCC1)=O 79934,C1(COC)(NC(=O)CC2CN(C(=O)CSc3nc[nH]n3)C2)CCC1 79935,CCC(O)C(C)C(=O)N(C1CCN(C(C2CC(CN(C)C)C2)=O)CC1)CCOC 79936,C1(NC(C2CC2(F)Cl)=O)CC2CC1CC2C(=O)NC1(CF)CC1 79937,CC(O)C(C(=O)NCCC1CCCN(C(c2csc(Cl)n2)=O)C1)N(C)C 79938,Cc1ccc2c(=NC3CCOCC3)[nH]c(=NCc3nnc(C)o3)[nH]c2c1 79939,c1(CCC)ncc(C(=O)NC2CCC(NC(=O)CSc3nncn3C(C)C)C2)s1 79940,C(=O)(C#CC1CCOC1)N1CCCC(C(=O)NCc2nc(C)c(C)s2)C1 79941,C12(NC(CC=C)=O)CCCCCC1N(C(=O)CNC(=O)NC1CCCCC1)CC2 79942,c1(NC(C(C(C)C)NC(=O)Cc2ccns2)=O)ccc(F)cc1CO 79943,c1(C(=O)NCC(C)N(C(c2ccc(N)c(O)c2)=O)CC)ccc2c(C)[nH]nc2c1 79944,C1(C(N(C)CC2(O)CCN(C(Cn3c(C)csc3=O)=O)C2)=O)C2CCC(F)(F)C12 79945,c1(CNC(=O)NC2CC(C(N)=O)OCC2)cc(O)cc(Br)c1 79946,CC1COc2ccc(C(=O)NC3CCC3NC(=O)CCCc3ccsc3)cc21 79947,c1(CC)cc(C(=O)O)c(C(=O)NCC2(CNC(=O)C=CC3CC3)CCC2)cn1 79948,C1(NC(COCCCC)=O)(CO)CN(C(=O)C(C)C2CCCO2)C1 79949,C1(CC(N2CC(O)(CN(C(=O)C(C)(C)C3CCOC3)C)C2)=O)OC(C)(C)OC1=O 79950,C(=O)(C(C)C(O)CC(C)C)NCC(C)(C)OCC(=O)NCC1CC(OC)C1(C)C 79951,C(=O)(C(CC)(CC)C(C)C)NC1CC2CN(C(C(CC)CN(C)C)=O)C1C2 79952,C1(CCC)CN(C(C2C3CCCOC23)=O)CCN1C(=O)C(O)CC1CCCC1 79953,C1(CCNC(c2ccc(C(C)C)o2)=O)(OC)CN(C(c2cn(CCO)nn2)=O)C1 79954,n1(CC)ccc(NC(=O)CN(C2CCCCC2)C)n1.C12CN(C1)CC(=O)NC2C 79955,C1(CCC)COCCN1C(=O)C(C)C(C)NC(=O)C=C(C)C 79956,C1(NC(c2ncc(F)cn2)=O)CN(C(C2CN3CCC2CC3)=O)CC12CCCC2 79957,C1(CNC(CC(C)C)=O)CN(C(C2CCN(C)CC2)=O)CC(C(F)(F)F)O1 79958,C1(C(=O)NC2CC(CCC(=O)NC(C(=O)NCC)C)C2)COC(=O)N1C 79959,C1(NC(=O)NCC(C2CCCO2)O)CC12CCS(=O)(=O)CC2 79960,N1(C(C(C)C2CC2)=O)CCCC12CCN(C(C1CCOC1)=O)C2 79961,C1(NC(Cc2ccc(C)nc2)=O)CC2CC(C1)N(C(=O)CCC1CCCC1)C2 79962,c1(C(C(=O)NCCCC)N(CCCC=C)C)noc2c1CCC2 79963,c1(C(N(C(=O)CCc2cccs2)C2CC2)=O)nccc(-c2cnccn2)n1 79964,N1(C(CCCCCC)=O)CCN(C(=O)CCc2cccc(C#N)c2)C(C)CC1C 79965,Cc1[nH]nc2cc(CCCC3(NC(=O)C(C(C)C)n4ccnc4)CC3)ccc12 79966,C1(CNC(C2CC2F)=O)COCCN1C(c1cccc(CC2CCC2)c1)=O 79967,c1(C(=O)NC(C(CCC)O)CO)cc2[nH]nnc2cc1OC 79968,C1(C(N(CCCSC)C)=O)CC(=O)CN1C(c1cc(C)[nH]c1C)=O 79969,N1(C(CN2CC(C)C2)=O)CCCC(n2cc(CNC(C3CC3(Cl)Cl)=O)nn2)C1 79970,CCCCCCC(O)CCC(=O)NC1(C)CCCN(C(=O)CC2OCCO2)C1 79971,N1(C(C2NC(=O)OC2)=O)CC2CN(C(c3cc4n(n3)CCCN4)=O)CC2C1 79972,C(=O)(C1=Cc2ccc(Cl)cc2OC1)NCCN(C(=O)C1=C(C#N)CCC1)CC 79973,C1(N(C(=O)C(C)C2CCCO2)CC)CCN(CCOCc2cccc(C)c2)CC1 79974,CN=c1ccc(C(=O)N(C(C)CNC(c2csc(C3CCCO3)n2)=O)C)c[nH]1 79975,C(=O)(C(C)S(=O)Cc1c(Br)cnn1C)Nc1c(C(C)C)cccc1 79976,N1(C(C(CCO)N(C)C)=O)CC(C2CCN(C(C3CC3(C)C)=O)CC2)C1 79977,N(C(=NCCCN1CCOCC1)NC1CCCOC1)CC1CCC(=O)NC1 79978,CC1(NC(c2cc(-c3ccoc3)[nH]n2)=O)CCCN(C(=O)CC2CCC(=O)N2)C1 79979,CCS(=O)(=O)CC(=O)NCC1C(C(=O)Nc2ccc(O)c(C(N)=O)c2)C1(C)C 79980,Cc1cnc(N2CCC(CNC(=O)C(C)C(C)(C)C)C2)nc1S(C)(=O)=O 79981,c1(C(N2CC=CC(NC(=O)CC3CCC(C4CC4)O3)C2)=O)ccnc(Cl)c1Cl 79982,c1(C(=O)NCC(CC=C)NC(=O)Cc2cc(C)cc(C)c2)cc(OC)ccc1C 79983,C(=O)(C1=CCCS1)NC1(CNC(=O)CCC2CCC(C(=O)OC)O2)CCC1 79984,c1(C(N2CC3(C(NC(CS(CC)=O)=O)CC3)C2)=O)c(C)cc(O)nc1C 79985,Cc1cc(F)ccc1NC(C1(C(=O)Nc2csc(-c3ccccc3)n2)CC1)=O 79986,N1(C(C(C2CCCC2)NC(CC2(C)CC2)=O)=O)CCC(CO)C(C)C1 79987,C1(C(=O)NCC(C)N(CC)CC)CCCC1CNC(=O)CC1CSCCO1 79988,C1(C(N2C(CNC(c3cc(Cl)ccc3F)=O)CC2)=O)Cc2ccccc2N1 79989,c1(C(N2C(C(=O)NC3C(CC=C)COC3)C3CC3C2)=O)ccc(C#N)cn1 79990,C12(CNC(=O)CC3=CCCC3)CCCC(CN1C(=O)C(=CC1CCCCC1)F)C2 79991,C(=O)(C(F)CCC(C)C)N1CCN(C(CCCC#C)=O)C(CCO)C1 79992,C=CC1(C(=O)NC(C2CCCCC2)CNC(=O)Cc2n[nH]c(C)n2)CCCC1 79993,C1(CC(=O)NCc2cc(C)ncn2)CCCN(C(c2cc(C3CC3)on2)=O)CC1 79994,c1(C(N(c2nccn2C)CCNC(C(C(=O)OC)C)=O)=O)ccc2nccn2n1 79995,c1(C(=O)NC2CC(NC(C3COCC(C)(C)O3)=O)C2)c[nH]c2c(C#N)cccc12 79996,C(=O)(C(C(C)C)n1cnnn1)NC1C(NC(CC(OCC)OCC)=O)CC1 79997,N(C1CCCc2sccc21)C(CCCc1c(N)cccc1)=O 79998,c1(C(=O)NC2C(C)CN(C(C3CCCO3)=O)C2)cc2cccc(Br)c2[nH]1 79999,C1(C)(CC)C=C(C(=O)NC2(CNC(=O)C(N)=O)CC2)C1 80000,C1(OCC)CC(C(=O)NC)N(C(c2cnc(C)s2)C(=O)NC2CCCC2)C1 80001,Cc1ncncc1C(=O)NC1CN(C(c2occc2CN(C)C)=O)CC1F 80002,C(CC1=CCN(C(C2CC23CC(C)(C)C3)=O)CC1)NC(CCCC(=C)C)=O 80003,N1(C(C(CCC)N(C)C)=O)C2CCC1C(C)C(NC(=O)C1=C(C)S(=O)(=O)CC1)C2 80004,c1(CN2C(CC)COC(C(F)(F)F)C2)ccc2cc(C(=O)NC)[nH]c2c1 80005,c1(C(=O)NCC2N(C(C3CCCC(OC)C3)=O)CCC2C)cccn(C)c1=O 80006,CCC(CC)C(=O)NC(C1(O)CN(C(=O)CCCC2CCCCC2)C1)C 80007,Cc1cc(CC(=O)N(CCCCNC(C2CCSC(C)C2)=O)C)c(C)s1 80008,n1(CC(C)C)cc(NC(c2ccn(C)n2)c2nnnn2Cc2cccs2)cn1 80009,c1(NC(C2C(NC(=O)COCCc3cc[nH]n3)CCC2)=O)cccc(F)c1F 80010,c1(N(C)C)ccncc1CNC(C1CCCC1NC(=O)CC(C)(C)N(C)C)=O 80011,C1(C(C)C)CCc2[nH]nc(C(=O)NC3(CNC(=O)C(O)CCN(C)C)CC3)c2C1 80012,CC1(C)CN(C(c2csc(C(F)F)n2)=O)C(CNC(C2(Cl)CC23CCC3)=O)CO1 80013,C(C(CO)(CO)NC(C1CCN1S(C)(=O)=O)=O)N(C(c1nc(CC)sc1)=O)C 80014,C12(NC(COCCSC)=O)CCCC1CN(C(=O)C(=O)NCC1CC1)C2 80015,N1(C(C=CC)=O)CCC(CO)C(NC(=O)Cc2cccc(C(F)(F)F)c2)C1 80016,N1(C(C(C)SC(F)(F)F)=O)CC2CCC2(CNC(=O)C(F)(F)Nc2cnn(C)c2)C1 80017,N1(C(=O)C=Cc2ccncn2)CCN(C(C2(O)CC2)=O)CC(O)C1 80018,C(=O)(CC(C)CNC(C1(C2CCCN2C(c2nc[nH]n2)=O)CC1)=O)OC 80019,C1(C(NOCCCCC)=O)CC(C)CN1C(=O)C(=O)NOC 80020,Nc1cc2[nH]cnc2cc1C(N1CCC(NC(=O)Cc2csc3cncn23)C1)=O 80021,C(C(O)CC(=O)NCCC1(C)CCOCC1)NC(C(C)OCC=C)=O 80022,C(=O)(C(C)(O)CCC)NC(CN(C(c1c(CC)nccc1)=O)C)CC 80023,C1(NC(C(C)Oc2cccnc2)=O)CN(C(C2CC3CCCC23)=O)CCC1CO 80024,C(=O)(C1=CS(=O)CCC1)N1CCC(NC(c2cn(C(F)(F)CO)nn2)=O)C1 80025,N1(C(CN2CC(C)(OC)C2)=O)CC(CNC(=O)C=CC2CCCC2)CC1C 80026,C12(NC(Cc3scc(C)c3)=O)CCCC1N(C(c1cnc(F)cc1C)=O)CCC2 80027,C(=O)(C1CCc2cc(Br)ccc21)NCCn1cc(C2CCCN(C)C2)nn1 80028,Cc1scc(C(N2CC3C(CNC(c4cc(Br)n(C)c4)=O)C3C2)=O)c1N 80029,c1(C(=O)NC(CCC)CC)ccc(=N)[nH]n1 80030,c1(CNC(c2csc(C)c2C)c2n(CC)nnn2)cccc(F)c1 80031,Cc1cc(C(N2CCC3(CC3C(=O)N(c3cccc(Cl)c3)C)C2)=O)ccc1O 80032,C(C(=O)NN1CCCC1C(N1CCC(F)(F)C(O)C1)=O)c1c(C)n[nH]c1 80033,C(=O)(C1CCCc2ccccc21)NC(C1N(C(Cc2cnc(C)[nH]2)=O)CCC1)C 80034,c1(C(N2CC(O)(C(C)NC(C3CCCN3C)=O)C2)=O)ccccc1Br 80035,C1(NC(C(Br)=C(C)C)=O)CC2CCC1N(C(C1(O)CCC(C)CC1)=O)C2 80036,c1(OCC(=O)NC2C(NC(c3c(CC)non3)=O)C2)ccc(Cl)cc1[N+](=O)[O-] 80037,Cc1cc(C(=O)N(CCC(C)NC(c2ccc[n+]([O-])c2)=O)C)ccc1F 80038,N1(C(Cn2c(C)ccn2)=O)Cc2nccn2CC(NC(=O)OC(C)(C)C)C1 80039,c1(OC)cc(Br)c(C(=O)NC2CC2CNC(=O)CC(F)F)cc1F 80040,N1(C(c2ccn3cncc3c2)=O)CCCC2(CCCN2C(=O)C2=CCC2)C1 80041,C1(NC(C2CC=C(C)CC2)=O)CCN(C(c2ccn(CCO)c2C)=O)C(C)C1 80042,c1(C(=O)NCCCC(C)NC(C2(OC)CCOC2)=O)cccc2cc(F)ccc12 80043,N1(C(C(C)Oc2ccccn2)=O)CC(F)CC1CN(C(=O)CCn1ccnc1)C 80044,CC(C)C(C)(C)C(=O)NCCCNC(C1(C(F)(F)F)CC(O)C1)=O 80045,c1(C2C(C(N3CC(c4cn(CC(C(=O)OC)O)nn4)C3)=O)C2)ccccc1F 80046,CC1CCN(C(C2CC(=O)N(O)C2)=O)CCN1C(c1cc(C2CCCC2)[nH]n1)=O 80047,c1(SCC(N2CCCC(NC(C=C(CCC)C)=O)C2)=O)nc2ccccc2[nH]1 80048,c1(C(=O)NCCN(C(CCc2onc(C(C)OC)n2)=O)C)cnncc1O 80049,C1(C(=O)NCC(CNC(c2ccn(CCN(C)C)n2)=O)O)CC2C=CCC(C1)C2 80050,Cn1nc(Br)c2c(NC3CC(=C4CC4)C3)ncnc12 80051,c1(C(=O)NCC(C(C)C)NC(C2(CC(C)C)CCC2)=O)ncccc1C(C)(C)C 80052,N1(C(=O)NCC(C2CC(F)(F)C2)OC)CCC2(CC1)OCCO2 80053,N1(C(c2cc(C(C)=O)on2)=O)CC2(C1)C(NC(=O)CC(C)C(F)F)CCS2(=O)=O 80054,c1(-c2n(CCOC)ccn2)ccc(OC)c(-c2ccc(=NC)[nH]c2)c1 80055,n1(CC)c(N)c(C(=O)COC(=O)Cc2ccc3c(c2)CCC3)c(O)nc1=O 80056,c1(C(=O)NCc2cc(C)c(C(N3CC(F)C(F)C3)=O)o2)cc2ccncc2[nH]1 80057,O=C(C1=CC2CCC(C1)C2)N1CCC2(CC1)CN(C(c1ncccc1F)=O)C2 80058,c1(C(C(N2CCCN(C(CC(C=C)(C)C)=O)CC2)=O)O)cccc([N+](=O)[O-])c1 80059,CC(O)C(C(N)=O)NC(=O)COC1CCN(C(=O)CC2(O)CCCC2)C1 80060,C1(NC(c2cc(CCNC(CN(C)CC)=O)on2)=O)CC2C(C1)C2(F)F 80061,C1(C(N2CC(SC)C(NC(=O)COCCN(C)C)C2)=O)CC2C(C1)C2(C)C 80062,O=S(=O)(c1cccnc1NCCCN1CCC(O)CC1)NCCC1CC1(F)F 80063,c1(SCC(=O)NC(CCN(C(C(CC)F)=O)C)C)ccc(F)c(F)c1 80064,Cc1cc(C(N2CC(NC(=O)CC3(C)CCCC3)C3(CC3)C2)=O)nc(O)n1 80065,N1(C(C2N(C)C(=O)C(F)C2)=O)CCS(=O)(=O)CC1CCO 80066,c1(OC)ccccc1C1(Cc2ncc(Br)cn2)CC1.c12n[nH]cc1NC2=O 80067,C1(NC(CC(C=C)C)=O)CCCCC12CCN(C(=O)C=Cc1cncn1C)CC2 80068,Cc1nc2ncnn2c(C)c1CC(=O)NC1CC2CC1N(C(=O)C(C)C1CC1)C2 80069,C(c1cccc(Cl)c1)=CC(=O)NC(CC)CNC(C1CC=CCC1C)=O 80070,N1(c2ccnc(C(=O)OC)n2)CCC(C)(NC(=O)CSC2CC2)CC1 80071,c1(N2C3CC(CNC(C4CCS(=O)(=O)N4)=O)CC2CC3)nc2ccc(Br)cc2s1 80072,CCN=C(NCC(c1ccccc1)N(S(=O)(=O)c1ccccc1)C)N1CCCC1 80073,CC(c1ccsc1)=CC(=O)NCC1CC(NC(=O)C(C2CCCCC2)F)C1 80074,C1(C(N2CCN(C(c3c(CC)nn[nH]3)=O)C(CC)C2)=O)CCCC2(CCC2)C1 80075,N1(C(Cc2n(C)ncc2Cl)=O)CCCCC2C1CCCN2C(=O)C(F)CC1CC1 80076,O=NN1CCCC1C(=O)NCCC1CCN(C(C2CC(CF)C2)=O)CC1 80077,n1(CC)nc(C)c(C(N2CCCC(N(C(=O)CC3(C#N)CCC3)C)C2)=O)c1Cl 80078,c1(NCc2c(C)nc(CC)o2)nccc(=NCC2(OC)CCCC2)[nH]1 80079,c1(C(=O)NCC(CN(C(C(CC)F)=O)C)O)ccc(Nc2ncccn2)cc1 80080,Cc1c(C(=O)NCC2(NC(=O)CCSCC(N)=O)CCCC2)c(C(F)F)nn1C 80081,C#Cc1ccc(C(N2CC3CC3(C(=O)NCC3CC(SC)C3)C2)=O)c(C)c1 80082,N1(C(C2CC(=O)NC2)=O)CCCC(C2(NC(c3c(F)cc(F)cc3Cl)=O)CC2)C1 80083,CC1CC(NC(=O)CCc2nc(C3CCCC3)no2)C(=O)N1c1ccccc1 80084,n1(C(C)C)cc(C(=O)NC(C)(CNC(C2CC=CC2)=O)C(C)C)c(Br)n1 80085,c1(CC(N2C3CC(NC(c4cc(Br)co4)=O)(C3)C2)=O)ccc2c(c1)OCO2 80086,c1(-c2nc(SCC(C)C)on2)cccc(OCc2cccc(Br)c2)c1 80087,CC(C)S(=O)(=O)CC(=O)N(CC(O)CNC(=O)CNC(c1cccc(O)c1)=O)C 80088,Cc1ccc(C(C)C)c(OC(C)C(N2CC(C)(C)CC2C(C)(C)C)=O)c1 80089,CCC(C)C(O)C(=O)NCc1nc(CNC(c2ncccc2F)=O)cc(O)n1 80090,CCC(C)(C(=O)N1CC(N(C)C(c2ccn(C)c(=O)c2O)=O)C(C)(C)C1)C(N)=O 80091,c1(-c2cn(CC(=O)NC(Cc3cccc(F)c3)CO)nn2)cccn2ccnc12 80092,Cc1cnc(C(N2CCC(C(=O)NCCCC3CCCC3)C(C)C2)=O)c(F)c1 80093,N1(C(c2cnc(CC)s2)=O)CCC(F)(C(=O)Nc2ccc(F)c(C)c2)CC1 80094,CCC(CC(F)F)C(=O)NC1(CNC(C2NC(=O)CC2C)=O)CC1 80095,c1(C(=O)NCC23CC(NC(CC4CC(C)OC4)=O)(C2)C3)cccc2ccn(C)c12 80096,CC(C)CC(O)C(C)C(=O)N(CCCCNC(c1cc2occc2n1C)=O)C 80097,N1(C(c2ccc(C)cc2)=O)CCC(C(N2CCC(OC3CCC3)CC2)=O)CC1C 80098,c1(C(=O)NC2CCC(NC(C3C(OC)CC3)=O)C2)nc(C(F)(F)F)cn1C 80099,c1(C(c2n(CCCCCC)nnn2)NCC2CC(CF)C2)cnn(CC)c1CC 80100,c1(COC)nc(C(=O)NC(C)CCN(C)C(C2CC23CCC3)=O)co1 80101,c1(CNC(CC2(NC(Cn3c(C)nnn3)=O)CCC2)=O)cc(Cl)ccc1F 80102,C(CN1C(=O)Cc2ccccc21)NC(=O)C(=O)NC1CCCC12CCNCC2 80103,C#Cc1cncc(C(=O)NCC2C3CN(C(c4cnc(OC(C)=O)s4)=O)CC23)c1 80104,N1(C(CC(=C)Br)=O)CC(NC(=O)CCCN(C)C(C)=O)CC1C 80105,C(=O)(C(O)C(C)(C)CC)N1CC(CCNC(=O)CN2CCC(C)(O)C2)(OC)C1 80106,C(CCCCCC(=O)NCC1CC(C)N(C(c2ncc[nH]c2=O)=O)C1)SC 80107,c1(C(=O)NC2CC3CC2N(C(C2CC2(Cl)Cl)=O)C3)cc2n(n1)CCCCO2 80108,C1(C(N(C)C)=O)CCN(C(=NCCCC2CCCCO2)NCc2cccs2)C1 80109,c1(C2C(C(=O)NC3C(CNC(=O)C(c4ccc(Cl)cc4)=O)C3)C2)ccccc1C#N 80110,C1(NC(CCCN(C(C)C)C)=O)CC2CCC(C1)N2C(c1occc1C1CC1)=O 80111,C(CCCC(=O)NCCC(C)NC(c1n[nH]c(C2CC2)c1Br)=O)OCCC=C 80112,O=C(C#CC1CCCOC1)NC1(CNC(c2ccnc(S)c2)=O)CCOC1 80113,c1(N(C)C)cc(N2CCCC(CN3CCOC(Cn4ccnn4)C3)C2)ncn1 80114,CN1CCN(c2nc(Cl)ncc2Cl)C(CNC(C2CC3CCC(C2)S3)=O)C1 80115,C1(F)(CNC(c2ncc(C)s2)=O)CCCN(C(C2(C(F)(F)F)CC2)=O)C1 80116,S(=O)(=O)(c1ccc(N2CC(C)c3ccccc3C2)nc1)NC1C(C=C)OCC1 80117,c1(C(=O)NC2CCN(C(C(CCC)C#N)=O)C2)cnn2c(Br)cccc12 80118,C1(NC(CC(n2c(CC)ncc2)C)=O)CCCCC1NC(c1ccc(F)cc1)=O 80119,C1(N(C(CC(COC)C)=O)CC)CCN(C(=O)CNC(c2ccco2)=O)C12CC2 80120,c1(C(N2CC3(C2)CN(C(C2(CF)CC2(F)F)=O)C3)=O)ccc([N+](=O)[O-])cc1 80121,c1(C(=O)NCC23C(CN(C(C(C(=C)Cl)(C)C)=O)C2)C3)cccc2c1ncn2C 80122,C1(C(=O)NC2CN(C(C(C)NS(CC)(=O)=O)=O)C2)(SC)CC(C(F)F)C1 80123,c1(NCC2CCCCN(C(C(c3ccc(C)s3)C)=O)C2)nc(Cl)nc2sccc12 80124,Cc1c(NCCCOCCC(C)C)ncnc1N1CCC(C)(F)C1 80125,c1(CN(C(=O)C=CC2(C)CCOCC2)C)cc2ccccc2[nH]1 80126,c1(C(=O)NC2CCC(NC(CC(C=C)(C)C)=O)CC2)cc2ccccc2nc1C 80127,c1(C(=O)NCC2N(C(C(C=C)(C)CC)=O)CC2)cc2ccc(OC)cc2[nH]1 80128,O=C(CCCCc1ccc(F)cc1)NCCC1CN(C(C2C3CC3C3CC23)=O)C1 80129,C1(NC(C2C(C(C)O)C2)=O)CCCN(C(c2cncn(C)c2=O)=O)CC1 80130,C1(NC(=O)CCc2ccccn2)CCN(C(c2cc(O)nc(Cl)c2)=O)CC1CO 80131,c1(C(=O)NC(CNC(C2C(C)C2)=O)C)nc(C2CC2)ncc1Br 80132,c1(CC(C)C)ncc(C(=O)NC2CC(CCNC(C3CC3C3CC3)=O)C2)s1 80133,c1(NC(=O)Cc2cccc(Cl)c2Br)cc(Cl)cc2nc(O)oc12 80134,C1(C(C)C)C(NC(=O)CCC2CCOC2)CCN1C(=O)CCCN(C)C 80135,c1(C(N2CCN(C(C(CC)C)=O)C(C)C2)=O)oc2ccccc2c1CO 80136,n1(CC)cc(Br)c(C(=O)NC(C)CC(C)NC(c2scnc2Cl)=O)n1 80137,N1(C(c2c(C)nc[nH]2)=O)CC(NC(=O)CN(C)C(=O)OC)C2(CCOCC2)C1 80138,C1(C(=O)NCC(N(C)C(c2ccnc(S)c2)=O)C2CC2)CCC2CCC1O2 80139,N1(C(c2n(CC)ncc2)=O)CCCCC(N(C(=O)COCc2ccccc2)C)C1 80140,C1(C(=O)NC2CC(n3cc(C(C)(C)C4CC4)nn3)C2)CCC(C2CC2)C1 80141,C(C)(C)(CN(C(=O)C(C1(C)CC1)NC(=O)C(=O)NCC(F)F)C)OC 80142,c1(OCCOC)cncc(C(=O)NC2CCC(NC(C3CC=CC3)=O)C2)c1 80143,N1(C(CC2(COC)CC2)=O)CCOC2CN(C(C3CCSCC3)=O)CC12 80144,N1(C(CCCOCC=C)=O)C(CNC(c2cnn3cc[nH]c23)=O)CC2COCC12 80145,c1(C(N2C(CCNC(CCOCCOC)=O)CSCC2)=O)cnc2ccoc2c1 80146,c1(C(C)=O)sc(NC(=O)CC2CC(NC(c3cnc[nH]3)=O)C2)c(C#N)c1C 80147,CC(C)CCC(=O)C(=O)NCC#CC(=O)NCC1CCOCC1(C)C 80148,C1(C(N2C(CCCC)CCC2)=O)CC(C)CN(C(c2cc(C)cc(Cl)c2)=O)C1 80149,C=CC(C)(CC)C(=O)NC1CCN(C(c2c(C)ccnc2OCC)=O)C1 80150,C12(CNC(C(CSC)(C)C)=O)CCC(CNC(=O)C3=CCCC3)(CC1)CO2 80151,N1(C(CCCNC(=O)OC)=O)CCN(C(C)CNC(=O)Cn2ccnc2C)CC1 80152,C#CCCC(O)C(=O)N1CC2(CC(NC(=O)C(=Cc3ccc(Cl)cc3)C)C2)C1 80153,Cc1c[nH]c(C(=O)O)c1C(=O)NCCC=CCl 80154,C(=O)(CC(CC(C)C)NC(c1cnc(OC)s1)=O)NC(C#C)(C)C1CC1 80155,CCCCCCC(C)CC(=O)NC1CC1CNC(C1(O)CCCCCC1)=O 80156,N1(C(CSCC(=O)OC(C)(C)C)=O)CCC(C)(NC(C2(C#N)CCCO2)=O)C1 80157,CC(C(C)(C)CO)NC(=O)C(c1cn(C)nn1)NC(=O)CC(C)(C)C1CC1 80158,Cc1ccc(C(=O)O)c(CN2CCN(C)C(Cc3ccccc3)C2)c1F 80159,C(CCOCCO)(C(=O)N(C(C)CO)C)NC(Cc1c(C)scc1)=O 80160,CCCN=C(NCc1nnnn1C1CC1)NC(c1ccnn1C)COC 80161,C1(CNC(C2CC(=C)C2)=O)CCCCC1C(=O)NCC(Cl)=CCl 80162,C1(C2CN(C(C3CCCCNC3=O)=O)C2)(NC(c2cncc(NCC)c2)=O)CC1 80163,N1(C(=O)CC2COC3CC2C3)CCC2(CCCN2C(c2cnc[nH]2)=O)C1 80164,n1(C(C)C)cccc(NC(=O)C(C)C(N)C2CC2)c1=O 80165,C=Cn1ncc(C(=O)NCC2CCCN2C(=O)CCc2ccc(C)o2)c1N 80166,CC1(CC(=O)NCCN(C(=O)CCCNS(C)(=O)=O)C(C)C)CC1(Cl)Cl 80167,N1(C(C2CC(OCC)C2)=O)CCCOC(CNC(=O)CCCCC2CCSS2)C1 80168,N1(C(C2C(NC(=O)OC(C)(C)C)C2)=O)Cc2ccnn2CC(COC(F)F)C1 80169,c1(C(=O)NCC(CNC(C2CC(C(C)=O)C2(C)C)=O)F)ccc(F)cc1F 80170,N1(C(C2CC(C#N)C2)=O)CC(CNC(=O)CCSc2ccc(Cl)cc2)C2(CC2)C1 80171,C1(C)(COC)CCN(C(=O)C(C)(C)C2CCN(C(=O)CNC(N)=O)C2)C1 80172,N1(c2n(CCOC)c(C(C3CCCCC3)(C)O)nn2)CCOC2(CCOC2C)C1 80173,C1(OC)(NC(=O)NCCCC(=O)OCCSC)CCC(c2ccccc2)CC1 80174,Cn1nc(C(C)(C)C)cc1C(N1CCOCC1CCNC(=O)Cc1ccno1)=O 80175,C(=O)(C(C)(C)CCSC)NCCN(C(C(CSC)O)=O)C 80176,C(=O)(C1=CCCN(C(=O)CC2CCC3CC23)C1)N1C(C)CC1(C)C 80177,c1(SC)nc(Cl)c(C)c(=NC2CCCC3CN(C(=O)C(O)C4CC4)CC23)[nH]1 80178,C1(C(=O)NC2CC3(C(NC(c4ncn(C)n4)=O)C3)C2)Cc2ccccc2NC1=O 80179,Cc1ccc(CC(N2CCC(=CC(=O)NCC3CC(F)C3)CC2)=O)nc1 80180,Cc1cc(C(=O)NC2CC(CC(=O)Nc3nccnc3Cl)C2)ncc1[N+](=O)[O-] 80181,CC1CCN(C(=O)C(C)CC(N)=O)C(CNC(=O)Cc2cccc(O)c2)C1 80182,N1(C(C2C(C)C2)=O)CC2CC2(NC(c2coc(Cc3ccccc3)n2)=O)C1 80183,C1(OC)CCN(C(=NCCN2CCCOCC2)NCC(N2CCCCC2)=O)C1 80184,n1(C(C(=O)NCC2CCN(C(C(C=C)O)=O)CC2)C)nc([N+](=O)[O-])cc1C 80185,N1(C(c2cn(C)nc2)=O)CCCC2CCN(C(c3cc(C(N)=O)cs3)=O)CC12 80186,C1(NC(C(N2CC(OCCCCC)C2)=O)=O)CCCC(CN=[N+]=[N-])C1 80187,N#Cc1cc(NC(C2CN(C(=O)CC3CCCCO3)CCS2)=O)cnc1Cl 80188,C1(NC(CNC(CC(C)C)=O)=O)CC2CC1CC2C(N1CC(C)C(O)C1)=O 80189,Cc1cc(-n2nc(Cc3cnn(C)c3)nc2CCCc2cnn[nH]2)ccc1Cl 80190,C1(C(=O)NCC2C(NC(c3cc(OC)no3)=O)CCC2)CCCC(=O)O1 80191,C(=O)(C(CC1CCCC1)NC(c1ccncn1)=O)NC(C(=O)N(CC)CC)C 80192,C1(O)(CN(C(CCC(C)SC)=O)C)CCCN(C(=O)C(F)=CC2CC2)C1 80193,N1(C(CC(=O)N(C)C)=O)CCCC1C1CCCN1C(C1CC2(C1)CC(F)(F)C2)=O 80194,N1(C(=O)Cc2cccnc2O)CCN(C(c2ccc(O)nc2)=O)C(C2CCC2)C1 80195,N1(C(c2cnn(CC(F)F)c2C)C(=O)NCCOC)CCC(OC)C(C)C1 80196,c1(NC(CC2CCN(Cc3cnn(CC)c3C)C2)=O)cc([N+](=O)[O-])ccc1CO 80197,N1(C(c2nnn(CC)c2C)=O)CC2(CNC(C3(COC)CCOC3)=O)CC1CO2 80198,Cc1cc(NC(c2nncn2C2CCCCC2)=O)ccc1OC(F)(F)F 80199,c1(C(=O)NC(C2CCCO2)CC)ccc(CNC(C2CC(C)(O)C2)=O)o1 80200,CC(CNC(=O)CNC(=O)NC1CC1)N=c1ccnc(C2CCCC2)[nH]1 80201,N1(C(CC(C=C)CC)=O)CCC(CNC(=O)C2=CCCC2(C)C)C(F)(F)CC1 80202,N(C1CCC(NC(C2CC3CC2C3)=O)c2ccccc21)C(CSC(C)C)=O 80203,c1(NC(c2c(C)cco2)=O)cccc(C(=O)NN2CC(C)C(O)C2)c1 80204,c1(OC)cccc2cnc(NC(C3CCN3C(c3cc(Cl)ccc3C)=O)=O)nc12 80205,c1(CNC(N2CCCCC2CCO)=O)cc(Cl)ncc1Br 80206,C(=O)(NN=c1ccc2nccn2[nH]1)c1c(C)ccc(C(=O)OC)c1O 80207,c1(CC)cccc(CC(N2CCCC2(C)CNC(=O)Cc2cnn(C)c2)=O)c1 80208,C1(C(=O)NOC2CCOC2)(CC)CCCN1C(C1CC(C)(C)CO1)=O 80209,CN(C)S(=O)(=O)N1CC(NC(c2nnnn2CCC2CC2)CC2CC2(Cl)Cl)C1 80210,C1(CNC(C(CC)OC(C)=O)=O)CCCCC1NC(=O)CCOc1ccc(C)cc1 80211,C1(C)(CCNC(C2(N(C)C(c3nc(Cl)cs3)=O)CC2)=O)CCOCC1 80212,c1(C(=O)NCC2C3CN(C(C(C)OC4CCCC4)=O)CC32)nnn2ccccc12 80213,C1(C(=O)NCCCCOC)CCOCC1NC(=O)C(C)(C)C1CC1 80214,N1(C(CC=C(C)C)=O)CCC(CCNC(=O)C=Cc2cscn2)CC1C 80215,Cc1ccc(C)c(CC(=O)NC2CC(C)N(C(C3CCC(N(C)C)CC3)=O)C2)c1 80216,CCCC(F)C(=O)NCC(C1CCN(C(c2ccc(C)cn2)=O)CC1)C 80217,n1(C(CC)C)nnnc1C(c1sccc1Cl)NCC1CC2(CC2)C1 80218,S(=O)(=O)(c1ccc(C(=O)N(C)CCNC(=O)CC2CCC(OC)CC2)o1)NC 80219,Cc1ccc2nc(C(N3CCCCC(NC(c4ccc(Cl)o4)=O)C3)=O)c(N)n2c1 80220,N1(C(c2cncc(OCC)c2)=O)CC(C)(C)CCC1CNC(C1CC1(C)C)=O 80221,N1(C(CC2CC(NC(CCCOCC)=O)C2)=O)CCOCC(O)C1 80222,N1(C(C(CC=CC)C)=O)CCC2(CC1)CN(C(c1cccc(CO)c1C)=O)C2 80223,c1(CN(C(C)(C)CO)CC(=O)Nc2nn[nH]n2)ccccc1F 80224,O=C(C1CCCc2n[nH]cc21)NC1(CF)CCN(C(=O)C(F)(F)C2(O)CCC2)C1 80225,c1(C(=O)NC(C(C(C)C)NC(=O)CSS(C)(=O)=O)C)cncc2nc(O)[nH]c12 80226,NS(=O)(=O)c1n[nH]cc1C(N1CCCC(NC(=O)CC2CC(=O)NC2=O)CC1)=O 80227,Cc1cnc2cc(C(N3CCOCC3CNC(=O)CCc3csnn3)=O)ccn12 80228,C(=O)(C1=CC2(CN(C(=O)C(C(CC)CC)OC)C2)OC1)N(CCC#C)CC 80229,C(=O)(C(CNC(=O)C(OC)OC)C(C)C)Nc1c(CC)noc1C 80230,C1(N(C(=O)COC)CC)CCCN(C(c2cc(COCCC(C)C)[nH]n2)=O)C1 80231,c1(CNC(COC(CC)(C)C)=O)cn(CC(=O)NCC2(C)CCCO2)nn1 80232,Cc1cc(C#N)ccc1NC(C1CCN(c2ncc(Br)cn2)C1)=O 80233,C12(C(N(CCN(C)C(c3cnc(O)s3)=O)C)=O)CCC(CC1)C2(C)C 80234,c1(C2OCCN(C(CC(=O)NC(CC(C)C)=O)=O)C2)ccc2ccccc2c1 80235,C1(NC(C(C(C)C)C(C)C)=O)CCC2(CCN(C(c3cc[nH]c3)=O)CC2)CC1 80236,Cc1cccc(NC(=O)Nc2ccc(C(=O)NC(c3cccnc3)C)cc2)c1 80237,c1(C(N2CCC(c3ccncn3)CC2)C(=O)NC(C)C)cccc2cn(C)nc12 80238,CC1(C)OCCC1C(=O)NC1CCC(NC(C2CC(F)(CO)C2)=O)CC1 80239,C(CCCCCNC(C1(C)CCCCC1)=O)NC(C(C)Cc1ccncc1)=O 80240,c1(C(C)C)ccc(F)c(C(N2CC(NC(c3ccnc(C(C)C)n3)=O)C2)=O)c1 80241,C(=O)(C1=CC2(CCN(C(=O)Cc3ccoc3)C2)C1)NCC(N1CCOCC1)C 80242,C(=O)(CC(CC)C(C)(C)C)NCCN(CCCCCC)C(=O)C(O)CC1CC1 80243,C(C(=O)NCCC1(CNC(=O)CCc2nccs2)CCC1)(c1cccs1)SC 80244,C=CC(C)(C)CC(=O)NC(C)(C)C=CC(=O)NCC1CCCC(OC)C1 80245,c1(C(=O)NC2CCC(CNC(C3(SCC)CC3)=O)C2)cncc2c[nH]nc12 80246,C1(NC(C(C(C)C)O)=O)C2CC1CN(C(c1cc(C#N)c[nH]1)=O)C2 80247,N1(C(C(c2cccnc2)NC(C2CC(C)=C(C)CC2)=O)=O)CC2CCCC(C2)C1 80248,N1(C(C(C(C)C)OC)=O)CCCC2(C1)CN(C(c1cccc(O)c1Cl)=O)CCO2 80249,C12(C(=O)NC3CCN(C(c4n[nH]c(C)c4Cl)=O)C3)CCCN(CC1)C2 80250,CC1(CNC(c2cc(N)ccc2O)=O)CCCN(C(c2c(F)ccnc2Cl)=O)C1 80251,CC1(C)CN(C(c2cc(-c3ccncc3)no2)=O)C(CNC(C2(F)CC2)=O)CO1 80252,c1(C(=O)NCC(C)(C2CCC2)NC(=O)CCCC#N)cc2cncn2c(O)n1 80253,c1(C(N(C2CCN(C(CC(C=C)C)=O)C2)CC)=O)cc2nc(Cl)ccc2s1 80254,c1(N(C)CCn2ccnc2)nccc(N2CCC(CC3CCC3)CC2)n1 80255,C1(NC(CC(CC)C)=O)CCOC12CCN(C(=O)C(C)OC)CC2 80256,C1(NC(c2cc(COC)on2)=O)CC1C1CCN(C(=O)Cc2sccc2C)CC1 80257,c1(C(CO)NC(NNC(c2cccc(OC)c2)=O)=O)ccc(S(C)(=O)=O)cc1 80258,c1(CN2CC(CCCCNC(C3CC(CC)C3)=O)C2)c[nH]c2ccc([N+](=O)[O-])cc12 80259,C12(CNC(C=COCC)=O)CCCC1N(C(c1cncc(NC)c1)=O)CCC2 80260,N1(C(CC(CC)N(C(=O)CN2CCOC2=O)C)=O)CCC(O)C(CO)C1 80261,Cc1nc(C(C)C)ccc1C(=O)NC1CN(C(=O)CN2CCC(C)CC2)CC1F 80262,C(=O)(C(C)(C)CS(N)(=O)=O)NC1CC(C)(C)N(C(=O)CC(F)(F)F)C1 80263,Cc1ccc(O)c(C(N2CCC(C(F)C(=O)NCC=Cc3cccnc3)C2)=O)c1 80264,c1(OC)ccc(C(=O)NCC2CC(NC(C3(n4cccn4)CC3)=O)CCO2)cc1 80265,C1(COC)COCCN(C(=O)CC(C)NC(c2cc(Br)cs2)=O)C1 80266,C(=O)(C1CCc2cc(C)ccc21)NCCCOCCNC(C1(CC)CCCO1)=O 80267,C12(C(N3CC(CCCCNC(C(C)NC(CC)(C)C)=O)C3)=O)CC(CCO1)C2 80268,c1(CC(=O)NC2CCC(NC(C3CCCC3CF)=O)C2)c[nH]c2ncccc12 80269,O(NC(=O)C(CCF)NC(c1cccc(O)c1F)=O)CCCC=C 80270,c1(C(=O)NC2CCCN(C(CC3(C=C)CCC3)=O)CC2)cc(C)cc(OC)c1C 80271,N1(C(c2[nH]cc(C)c2)=O)CCC2(C1)CN(C(=O)CCCNS(C)(=O)=O)C2 80272,c1(OC)ccc(C(=O)NC(C2(O)CN(C(C3CCCSS3)=O)C2)C)cn1 80273,c1(C(N2C3C(N(C(C(CC)SC)=O)C)CC(C3)C2)=O)ccn2ncccc12 80274,Cc1nc(N2CCCCC(CNC(=O)CC(C)C)C2)c2c[nH]nc2n1 80275,CC(N=c1cc[nH]cc1S(=O)(=O)NC(c1cncn1C)CO)c1ccccn1 80276,c1(CC(=O)N(CCNC(C2(COC)CC2)=O)C2CC2)c(C)cc(Br)cc1C 80277,CCCC(C(=O)NC(C(=O)NCCNC(=O)C1CC1)C1CC1)N(C)C 80278,C(C(=O)N(C1CCCCC1N(C(=O)CN1CC=CC1)C)C)(C(C)C)N(CC)CC 80279,N1(C(c2cc(CC)nn2C)=O)CC(NC(C2CCC(CC)CC2)=O)CC12CCC2 80280,N1(C(C2C(CC)NCC2)=O)CCC(N)c2c(Br)cccc21 80281,CC(C)C(C)CC(=O)N(CCCNC(C1CC(O)(c2cccnc2)C1)=O)CCO 80282,N1(C(c2ccc(Br)c(F)c2)=O)CC2(CCC(N3CCc4ccc(Cl)cc43)CC2)C1 80283,c1(CC(CC(=O)OC)NC(C2CN(C3CCC3)C2)=O)ccc2c(c1)CCO2 80284,C1(NC(C(C)NC(N)=O)=O)CCSC12CN(C(c1cccc(C(F)F)n1)=O)C2 80285,C(c1ccc([N+](=O)[O-])s1)=CC(=O)NCCN(C)C(C1COC(=O)N1C)=O 80286,N1(C(c2cccc(N3CCCC3=O)c2)=O)CC2CCC(C1)N2C(C1CCC1F)=O 80287,CC1CCN(C(=O)CC2(NC(c3ncccn3)=O)CC2)CC1CO 80288,C1(CNC(=O)Cc2cccnc2O)CC2CC1CC2O 80289,n1(CC)ncc([N+](=O)[O-])c1C(=O)NCC(C)CNC(c1ncn(C(C)(C)C)n1)=O 80290,c1(C(=O)NCC(C2CCCC2)NC(c2cc(C3CC3)on2)=O)n[nH]c(C2CC2)n1 80291,N1(C(C=CCCC)=O)CCC(C(=O)NCCC2CCCC23CC3)C1C 80292,c1(C(=O)NC2CCCCN(C(C(CC)C#N)=O)C2)cc2cc(OC)ccc2o1 80293,n1(C(C)C(N2CC=CC(NC(=O)CCC3CC3C)C2)=O)cnc2ccccc12 80294,c1(C(N2CCCC(O)(CNC(C(C)Br)=O)C2)=O)ccc2cnccc2n1 80295,C1(C(=O)NCCCN(C(C(C)=C(C)C)=O)C2CC2)CC12CCS(=O)(=O)CC2 80296,c1(N2CCC(C)C(NC(C3CCS(=O)(=O)C3)=O)C2)ncnc2[nH]cnc12 80297,N1(C(C(c2cnn(C)c2C(F)(F)F)C)=O)CC2(CCN(C(=O)C=CS(C)=O)C2)C1 80298,c1(CC(C)OC)nc(C2CCCC2O)n(-c2ccncc2C)n1 80299,C#CC1(C(=O)NC2CCC(=O)NC2=O)CCN(C(=O)C(c2cncnc2)C)CC1 80300,C1(NC(=O)COc2ccccc2)(CO)CCCN(C(=O)C(F)C(F)(F)F)C1 80301,N1(C(Cc2cnc(C)s2)=O)CCC(CNC(c2c[nH]nc2C)=O)C(C)C1 80302,C1(NC(C2CCn3nccc3C2)=O)CCC2(CCNC2)C1 80303,c1(C(C)N(C)C(c2cn(C)cc(Br)c2=O)=O)nc2c(s1)CCCC2 80304,c1(C(=O)NCC(C)CNC(C2CC2c2ccco2)=O)coc2c1NC(=O)CCC2 80305,C(=O)(C1Cc2ccccc21)NCCOCCC(=O)NCC1N(C)CCOC1 80306,N1(CCSC2CCOC2)CCN(C(=O)NCCNC(=O)OC(C)(C)C)CC1 80307,c1(NC(C2CCCN(Cc3cccc(Cl)n3)C2)=O)ccc(O)cc1O 80308,C1(CCOC)(NC(=O)CCC2CCC2)CCN(C(=O)C2=NOC(C)C2)CC1 80309,CCCCCC(O)CC(=O)NCC12CC(CN1C(=O)CSC)C2 80310,C12(C(N3CCC(N(C(=O)C(C)N(C)C)CCC)C3)=O)CCC(O)(CC1)CC2 80311,c1(C(N2CCCC(F)(C(=O)NCCC(O)C3CC3)C2)=O)cc2occc2[nH]1 80312,CC(C)(C)C=CCNC(=O)NCCNC(=O)C(=O)NC1CC1 80313,c1(CC)cnc(O)c(C(=O)NC(C)(CNC(C2CC2(Cl)Cl)=O)C2CCC2)c1 80314,S(=O)(=O)(c1ccc(Cl)s1)N1CCN(CCN(c2ccn(CC(C)C)n2)CC)CC1 80315,C1(NC(C(CSC)O)=O)CCN(C(=O)Cc2c(F)cncc2Cl)CC(O)C1 80316,C=CCC(CC=C)C(=O)N1CCC(F)(F)C(CNC(=O)Cc2nccn2C)C1 80317,c1(C(N2C(CC(C)O)CCCC2)=O)cccc2c1COC2 80318,c1(NC(=O)NCCNC(=O)Oc2ccc(Cl)cc2Cl)cc(F)c(Br)cc1F 80319,C1(NC(C=CC=CC)=O)CCCC1(C)CNC(=O)CC(c1ccccc1F)SC 80320,CCCCS(=O)(=O)CC(=O)NC1(CC)CCN(C(=O)C(C)=C2CCCC2)CC1 80321,c1(C(=O)NCC(C2CCOC2)NC(Cc2n(C)ccn2)=O)ncccc1F 80322,c1(C(N2CCC(C)(N(C)CC)C2)=O)cnc(O)c2ccccc12 80323,c1(C2C(C(=O)NCC3N(S(CC)(=O)=O)CCC3)C2)nccc(C(=O)OC)c1F 80324,N1(C(CC(CC)(F)F)=O)CCC2CCN(C(C3C(C=C(C)C)C3(C)C)=O)C2C1 80325,C1(CNC(CC(CNC(C(C)n2cncn2)=O)C2CCC2)=O)CC2CCCC2C1 80326,CCCC(CCO)NC(C1CC1C(=O)NCc1cnc(SC)nc1)=O 80327,C(=O)(CCN(OC)C(=O)CC(C)C1CCCO1)NCc1cccc(OC)n1 80328,C1(OC)(CNC(C2CSCN2C(c2ccc(CO)o2)=O)=O)CCOC1 80329,C1(NC(=O)NC)CCN(N2CCC(Nc3nccs3)CC2)C1 80330,C1(F)(CNC(Cc2nc(CC)sc2)=O)CC(N=c2[nH]nc(C3CC3)s2)C1 80331,C=CCC(CC)C(=O)N(CC(C)NC(C1(C)COC1)=O)C 80332,N1(C(C2CC(n3cc(CCCC=C)nn3)C2)=O)CCc2ccc(Br)cc2C1C 80333,N1(C(c2c(CC)nc(C)o2)=O)CC(C(=O)N(CCCO)C2CC2)C(C)(C)C1 80334,c1(OCC(=O)OCC(c2cc(C)oc2C)=O)ccc(S(C)(=O)=O)cc1 80335,C1(NC(C(=O)NCC)=O)CCCC(CNC(=O)C(C2CCCCCC2)O)C1 80336,c1(C(=O)NC)ccc(C(N2CCCC2CNC(c2cc(O)n(C)n2)=O)=O)cn1 80337,C1(C(N2CCCC(NC(C(F)=C(C)C)=O)C2)=O)OCCOC1(C)C 80338,C1(NC(C(=O)NC(C)C)=O)CCCC12CCN(C(=O)Cc1cc[nH]c(=N)c1)C2 80339,C1(CCC)(NC(C2CCCN2C=O)=O)CCN(C(c2[nH]cnc2C)=O)CC1 80340,N#Cc1ccc(CNC(=O)NC2(C3CCC4(CC4)CO3)C(=O)C2CC)cc1 80341,n1(C(C)C(=O)NCC(C)N(C)C(c2c(F)ccnc2F)=O)cc2ccccc2n1 80342,c1(OCCN2CCCC(C(=O)NC3CC(C)(NC(C)=O)C3)C2)c(C)cc(C)cc1C 80343,C1(CNC(CC(C)OC)=O)(CO)CCN(C(c2ncoc2-c2cnn(C)c2)=O)C1 80344,C(CC(=O)Nn1cnn(C(=O)NCC=C)c1=O)N(C(=O)C(C)CCCC)CC#C 80345,Cc1ncc(C(N2CC(C)CNC(C)C2)=O)c(Cl)c1Cl 80346,CC(C)(N=[N+]=[N-])C(=O)NCC(C)(O)CNC(=O)CP(C)(C)=O 80347,CC1(C(=O)NC2C3CN(C(=O)CC4CC4(Cl)Cl)CC23)CC2(C1)CC(F)(F)C2 80348,c1(C(c2nnnn2C(C)(C)C)NC(c2ncn(C)n2)C)ccc(C#N)s1 80349,c1(OC)cccc(N(C)C(C2(CNC(C3CC(=C4CCC4)C3)=O)CCCO2)=O)c1 80350,C1(C(N2CCN(C(CSC(C)C)=O)CC2)=O)CCc2n[nH]cc2C1 80351,c1(C(N2CC3CC3(C(N3CCC(CO)C(F)C3)=O)C2)=O)cc2cccnc2s1 80352,C1(C(=O)NCCCCC)CN(C(C2CC2(C)C(F)F)=O)CC1C(C)C 80353,C1(CC(=O)NC(c2c(C)nns2)C)CN(C(c2c(C)oc(C)c2C)=O)CC12CC2 80354,n1(CCC(=O)NCC2(O)CCN(C(c3cccc(Cl)c3)=O)C2)cc([N+](=O)[O-])cn1 80355,CC1=NNC(=O)C1CC(N1C(C(=O)NCc2nnc(C)o2)CCC1C1CC1)=O 80356,Cc1ccc(C(=O)N(C(C)CCNC(C2(CCF)CCOCC2)=O)C)c(O)c1 80357,C(=O)(CCCCCN=[N+]=[N-])NCC1CCC(C)(C)C1 80358,c1(C(=O)NC2CC(CNC(CN(C)CC)=O)OCC2)sc(Cl)c(Cl)c1OC 80359,C1(NC(CC=CCC)=O)CN(C(c2cc(OC)c(O)c(N)c2)=O)CC2(CC2)C1 80360,c1(OC)cccc(C2(C(=O)NCC(CC(C)C)NC(c3cnco3)=O)CC2)n1 80361,N1(C(C(N2CC(Cc3c(C)noc3C)C2)=O)=O)CCOC(C)(C)C1 80362,c1ccc2nc(C(=O)O)c(-c3cnoc3)cc2c1.c12ccc(nc1)CC21CCC1 80363,c1(C(=O)NC(C)CNC(C2C(C)(C)C2(F)F)=O)ncn2cc(Br)sc12 80364,C1(C(N2C(CCCNC(c3cn(CC=C)nc3)=O)CCC2)=O)COCCC1(F)F 80365,CCC(CC)CCCC(=O)N1CC(C(N2CC3CC=CCC3C2)=O)(CC)C1 80366,C12(C(=O)NCc3cc(C)on3)CCCC1CCN2C(c1cn(C)cc1C)=O 80367,c1(C(C(=O)NCC2COC2)N(C(C#C)C)C)ccc(OC)c(C2CC2)c1 80368,CCC(C)(O)CCNC(=O)C(C1CCN(C(c2ncc(F)cn2)=O)C1)F 80369,N1(C(c2c(Cl)cn(C)n2)=O)CCC(c2cn(CCCO)nn2)C12CC2 80370,N1(C(c2[nH]cc(OC)c(=O)c2)=O)CCC2C1CCCN2C(c1cn[nH]c1)=O 80371,C1(C(=O)NC(C2CCOC2)(C)C)CC2CN(C(=O)C=Cc3ccncc3)CC2C1 80372,C1(C(=O)NCCNC(=O)CCOCCc2ccccc2)CCC(F)CC1.O=C1CO1 80373,C(C)(CO)(CS(C)(=O)=O)OC(=O)NCC(OCOC)C 80374,N1(C(c2scc(C)n2)=O)CCC(O)(CC(=O)Nc2cnc(Br)c(F)c2)CC1 80375,c1(COC(C(C)SC)=O)cc2c(s1)CCOC21CCN(C(=O)OC(C)(C)C)CC1 80376,c1(C(=O)NCC(CNC(c2c(C)c(N)ccc2)=O)O)ccccc1S(C)=O 80377,C1(C(C)C)OCCC1C(=O)NCC(C)(C)CN(C(=O)CC1CN(C)C1)C 80378,c1(OC)cc(C(N2CC3C(C2)N3C(C2(C)CCCC2)=O)=O)cc(C(F)(F)F)n1 80379,Cc1cc(Cl)ncc1NC(C1CCC(C)N1C(c1cccs1)=O)=O 80380,CC(C)CC(C)(O)C(=O)N1CCN(CC(=O)NCCCOCC(F)F)CC1 80381,C1(C(=O)NCC(CNC(C(C)(CO)OC)=O)(C)O)CC2(C1)CC(CO)C2 80382,C(C1c2ccccc2CCN1C(c1cnsn1)=O)NC(c1cccc(OC)n1)=O 80383,Cc1noc(C(=O)NCC2C3CN(C(=O)CCCC4CCCC4)CC23)c1C 80384,C1(NC(CCN(C(C2(C(=O)OCC)CC2)=O)C(C)C2CC2)=O)CCCCC1 80385,C1(C(N(C2CCN(C(c3c(CC)[nH]cc3)=O)CC2)C)=O)COc2ccccc2O1 80386,N1(C(c2c(OCCC)c(C)ccc2)=O)CCC2CN(C(C)C(=O)OCC)CC12 80387,N1(CCNC(c2cc(CCCCC)[nH]n2)=O)CCN(C(=O)COCCCC)CC1 80388,C(=O)(C1=NN(C)C(=O)CC1)N1CCCCCC(NC(c2nccc(CC)c2)=O)C1 80389,N1(C(c2c(C)n(C)cc2)=O)CC(CC(=O)NC(c2cnc[nH]2)C)CC1(C)C 80390,C1(NC(c2nc(Cl)cs2)=O)CN(C(C2CS(=O)(=O)C2)=O)CC2CCCC12 80391,N1(CCC)Cc2ccccc2CC1CNS(=O)(=O)CCCN1CCCC1 80392,N1(C(C(C)NC=O)=O)CCC(C)C(CNC(c2cc(O)nn2C)=O)C1 80393,Cc1nc(Cl)ccc1CC(N1CCN(C(=O)Cn2cnnc2O)CC1C)=O 80394,CC1CCCCC1C(=O)NCC(C)(C)CCNC(=O)Cn1ncnn1 80395,CS(=O)CCC(=O)N1CCCC(NC(c2cccc(OC3CCC3)c2)=O)C1 80396,CN1CC(O)(CN(C(=O)C(Cc2cc[nH]n2)NC(=O)CCC2CC2(C)C)C)C1 80397,N1(C(C2C(C)(C)C2)=O)CCCC2(CC(NC(=O)Cn3ncc4ncccc34)C2)C1 80398,C1(C(=O)OC)(C(=O)NCC2CCC2NC(=O)CC(C)C2CC2)CC2(CCC2)C1 80399,c1(NC)ncccc1C(=O)NC1CN(C(=O)CCc2cc(C)cs2)CC1C 80400,C(=O)(C(Cc1ccccc1)NC(N)=O)NCC(CC)NC(c1coc(Br)n1)=O 80401,CN=c1[nH]cc(C(=O)NC2CC(C)(NC(=O)C(C)C3CC3)C2)o1 80402,c1(C(=O)NCC2(NC(C3CCCCS3)=O)CCC2)ccnc2nccnc12 80403,Cc1nc(C=CC(N2CC(NC(c3ccc(O)cn3)=O)C(C(F)(F)F)C2)=O)cs1 80404,N1(c2n(CC3C(OC)COCC3)nnn2)CCCOC(CCc2ccccc2)C1 80405,c1(NC(C)=O)ccc(C=CC(=O)NCC(C)NC(=O)C(c2ccc(O)cc2)O)cc1 80406,CC(C)C(C(C)NC(c1cncc(C2CC2)c1)=O)NC(=O)C(F)(F)CO 80407,C=CCCCC(C(=O)N1CCSC(C)CC1)NC(=O)Cc1cccnc1O 80408,c1(N2CCC3(C(F)(F)C3)CC2)[nH]c(=NC2CCC(C3CC3)CC2)nc2sccc12 80409,c1(C(N2CC(C)C(NC(=O)C3=C(Cl)CCCC3)C2)=O)ccc2c(=O)cc[nH]c2c1 80410,Cc1csc2c(N(C)CC3CCCN3C(=O)CCCC(=O)N(C)C)ncnc12 80411,c1(C(N2CC(NC(c3cncc(C(F)(F)F)n3)=O)(CO)C2)=O)ccnc(Cl)c1F 80412,c1(C(C)C)cccc(C(=O)NC2CCC2NC(=O)CS(=O)(=O)N2CCOCC2)c1 80413,c1(C(N2CC(CC)C(NC(C)=O)C2)=O)ccc(OC)cc1OC(F)F 80414,C1(C(C)C)C(NC(C2(C)CC2C(F)(F)F)=O)CCN1C(C1C2CC3C(C2)C13)=O 80415,N1(C(c2[nH]cc(C)c2C)=O)CCC2CN(C(C3CN(C)CC(C)O3)=O)CC2C1 80416,N1(C(COC(C)=O)=O)Cc2ccccc2C1CNC(C1CCC1(F)F)=O 80417,c1(N2CCCC(NC(C(C)OC3CCCC3)=O)(CO)C2)ncnc2ccccc12 80418,C1(C(=O)OCCN(C)CC2CN(C(CNS(CC)(=O)=O)=O)C2)C2CCCCCC12 80419,c1(C(=O)NCCCN(C(c2n(CCCC)ncc2)=O)C)cc2c(ccn2C)[nH]1 80420,c1(NCC(C)C)ccc(C(=O)NC2CC(O)(CNC(C3(F)CC3(C)C)=O)C2)cc1 80421,c1(C(=O)NCCOCCNC(C(C)OCCC#C)=O)cc(F)c(F)c(C#N)c1F 80422,c1(CC)cccc(NC2CCN(C(=O)CN3CCC(C(=O)OC)C3)C2C)c1C 80423,c1(C(=O)NC2CCCN(C(C(C)c3cc[nH]n3)=O)C2)cccc(O)c1Cl 80424,O=C1NC2(C(N3CC4CN(C(C5C=CC=CC=C5)=O)CC4C3)=O)CC3CC1C2C3 80425,CC(CCC(F)(F)F)NC(=O)CC(C)NC(=O)CC1OCCCO1 80426,c1(CCNCC(CN(C)C(c2cccnc2S)=O)O)ccc(C(N)=O)cc1 80427,c1(OC)ccc(CC(=O)NCC(C)CN(C)C(C2(CC(F)F)CCC2)=O)cc1F 80428,c12cccc(c1)CNC2=O.c1(NC(=O)COCC2CCCO2)ccoc1C1CC1 80429,Cc1csc(CCNC(C2C(CNC(c3csc(=N)[nH]3)=O)C2(C)C)=O)n1 80430,c1(C(=O)NC2CN(C(=O)Cn3cncn3)CC2n2cccn2)ccc(CO)cn1 80431,N1(C(c2ccc(O)nn2)=O)CC2(C1)CN(C(c1ncoc1C(F)(F)F)=O)C2 80432,C#CC(COC)N(C)N(C)Cc1c(OC)cc(C)cc1C 80433,c1(OC)ccc(N2CCC(NC(C3CCNC(C(F)F)C3)=O)C2)cc1C 80434,c1(C(N2CC3(CN(C(c4c(CCC)cccc4)=O)C3)C2)=O)n[nH]c2c1CCSC2 80435,Nc1cccc(-c2cn(CCNC(=O)C(F)CC3CCOC3)nn2)n1 80436,C1(CC)CC(C(=O)NCC(C)=CCO)CCN1C(C1CC(C)CC(=O)N1)=O 80437,CCS(=O)(=O)c1ccc(C(C)NC(=O)Nc2c(Br)cnn2-c2ncccn2)cc1 80438,N(C)(C(=NCC(C)C)NCC1(C)CCCOC1)CC(c1nccs1)C 80439,c1(CC=C(C)C)ccc(CN2CCN(C(=O)NC3(C)COCCO3)CC2)cc1 80440,C1(CC(=O)N(CC(N)=O)C)(OC)CN(C(=O)CCCCC(C)C)C1 80441,C(CCCC(=O)N1CC(CC(C)(C)CNC(C2(Cl)CC2(C)C)=O)C1)N(C(C)=O)C 80442,c1(C(N2CC3(C(NC(C(C)n4cnnn4)=O)CC3)C2)=O)nc2n(c1Cl)CCCC2 80443,CCCCC(C(=O)NCC1(C)CCCN(C(c2ccc(F)cc2Cl)=O)C1)C(C)C 80444,Cc1nscc1CC(N1CC(O)(CN(C)C(c2ccc(C3CCOC3)s2)=O)C1)=O 80445,C(=O)(C1=CC2CCCC12)N1CCN(C(Cc2c(OC)ccc(OC)c2)=O)CC1 80446,C1(C)(NC(Cc2cccc(C)c2)=O)CCCN(C(C2(S(C)(=O)=O)CC2)=O)C1 80447,CC(C)CC(O)CC(=O)N1CC(C2(NC(c3ccncc3F)=O)CC2)C1 80448,C1(C(=O)NCC2CC(F)C2)CC2CC1CN(C(=O)CCCC1CCC1)C2 80449,N1(C(C2(CC)CCCCC2)=O)CCC2CN(C(C3CC(C)CO3)=O)CC2CC1 80450,C1(F)(C(=O)NC(C)CO)CN(C(=O)CCc2cn(C)nn2)C1 80451,c1(C(N2C(C(C)(C)NC(C(C)OCC=C)=O)CCC2)=O)cncc(C(N)=O)c1 80452,C1(F)(CNC(C2C(C)OCC2)=O)CCN(C(=O)C(C)(C)Nc2ccccc2)CC1 80453,c1(CN(C(C(C=C)O)=O)CC)ccc(CNC(=O)CCNC(=O)C(C)(C)C)cc1 80454,c1(OC)cccc(C(N2CC(CNC(c3cncc(N)c3)=O)CC2C)=O)c1 80455,C(=O)(C1(C)CCc2ccccc21)NC1CCN(C(CC=CCC)=O)CC1(C)C 80456,CC1COC2(C1)CN(C(C13CC1CCN3C(C13CCC(C1)C3)=O)=O)C2 80457,c1(CCC(=O)NCC(C2(O)CCN(C(CSCC#C)=O)C2)C)cccc(F)c1Cl 80458,C12(C(N3CCCC(NC(=O)CN4CCC(F)CC4)C3)=O)CCCC1C2(F)F 80459,c1(CNC(c2c(CC)noc2)=O)cccc(CNC(=O)COC2CC=CC2)c1 80460,c1(OC)cc(NC(C2(C)CN(Cc3c[nH]c4ncccc34)C2)=O)c([N+](=O)[O-])cn1 80461,C1(NC(Cn2nc(-c3ccccc3)n(CC)c2=O)=O)CCC(C)(C)CC1CN 80462,C(=O)(C1=NOC2COCC12)NC(CC)(CNC(c1cccn2cncc12)=O)CC 80463,c1(OCC)ncccc1C(=O)N(C)CC1CCCN(C(c2nncs2)=O)C1 80464,C12(CC)CCC(C(=O)NC3CC4(C3)CC(NC(C3CC3C)=O)C4)(CO1)C2 80465,N1(C(C(CC)=CCCC)=O)CCN(C(=O)CN2CCC(OC)C2)CC1C 80466,c1(C(=O)NC2C(NC(C(F)OC)=O)COCC2)csc2cc(C)ccc12 80467,CC1Cc2ccccc2C(Nc2cc([N+](=O)[O-])cc(Cl)c2O)C1 80468,C(=O)(C1=C(C)OCCC1)N(CCC)CCNC(c1nc(C(F)(F)F)ccc1F)=O 80469,C(=O)(CCCCN1CCCC1)NCCCCCNC(c1cc(C(=O)OC)on1)=O 80470,c1(C(N2CCC(CNC(c3cc[nH]n3)=O)C(O)C2)=O)ccc2nccn2c1 80471,CCC(CC)(CO)C(=O)N1CCS(=O)(=O)C(CCNC(C2CCN2CC)=O)C1 80472,C1(C(=O)NCC(C)(C2CCC2)NC(CSCCOC)=O)(OC)CCCOC1 80473,C(=O)(CC(CC)C(C)(C)C)N1CC(C(C)NC(c2cncc(C#C)c2)=O)C1 80474,C1(CC(=O)NCCC2CC(NC(c3cnc(CC)o3)=O)C2)CCC(=O)NC1 80475,CON(C(=O)c1cccc(-c2cnco2)c1)C1CCCOc2ccccc21 80476,C=C=CC(C)C(=O)N1CCC(CN(C)C(c2cc(CO)n(C)n2)=O)C1 80477,c1(C(C)C)cccc(F)c1C(=O)NC(C)CN(C(c1nncs1)=O)C(C)C 80478,C(C(C)(C)CC(=O)NC1CCN(C(c2ccnn2C2CC2(F)F)=O)C1)OC 80479,C1(C(N(C)CC2(CNC(C3CC4C=CC3C4)=O)CC2)=O)CC2CC1C1CC21 80480,C(=O)(C(O)CC(F)(F)F)N(C(CC)C(=O)N1CC(NC(=O)OC)C1)C 80481,n1(CC(=O)NC2CCC(NC(c3csc(C(F)(F)F)n3)=O)CC2)ccccc1=O 80482,c1(C(=O)NC2C(CNC(c3cc(C4CCC4)[nH]n3)=O)C2)ncn2cc(Cl)ccc12 80483,CCCCCS(=O)(=O)CC(=O)N1CCCC2(C1)CN(C(C1(CF)COC1)=O)C2 80484,CCC(C(=O)N=c1[nH][nH]cc1OC)c1cccnc1 80485,c1(C(=O)NCC(CC=C)NC(c2csc(C(N)=O)n2)=O)cc(C)nc(C)c1 80486,CC1(C)CC(NC(c2ccncn2)=O)CN1C(c1cn(C2CC2)nn1)=O 80487,C1(NC(C(COC)C)=O)CCN(C(=O)C2=CCOC2)CC1O 80488,c1(CN2CCCC(C)(C(=O)NC3CCNC3=O)C2)cccc2ccsc12 80489,c1(C(N2CC(C(C)NC(CC(CC)C)=O)C2)=O)cc2c(C)c(F)ccc2[nH]1 80490,C1(C(C)NC(=O)C(C2CCC2)NC(c2ccc(CO)o2)=O)CC2(CCC2)C1 80491,CC(C)(C(=O)N1CCC(NC(c2csc(C(F)F)c2)=O)C1)S(=O)(=O)C1CC1 80492,Cc1cc(C(=O)NCCC2CCN(C(c3cc(Cl)no3)=O)CC2)cc2nn[nH]c12 80493,c1(C(N2CCC(C)(NC(CCC(C)O)=O)C2)=O)cc2c(cn1)CCCC2 80494,Cc1ncnc(C(=O)NC2CCOCC2C(=O)NC2(C)CCSC2)c1C 80495,c1(C(N(CCOC)CCNC(=O)CN(C)CCO)=O)ccn(CC(F)(F)F)n1 80496,c1(OC)ccc(C(N2CC(O)(C#CBr)C2)=O)n2nccc12 80497,CC1C(NC(c2c[nH]nc2C(F)F)=O)CCCN1C(=O)C=Cc1ccc(=N)[nH]c1 80498,c1(C(N(CCCOCCNC(C(C)SC(C)C)=O)C)=O)cc(=O)cc(Cl)[nH]1 80499,n1(CC(=O)NCCN(C(=O)C(C)N(C)Cc2ccccc2)CC)ccccc1=O 80500,c1(C(N2CCC(C(C)NC(c3cc(C)nn3C)=O)C2)=O)cc2c(nn1)CCC2 80501,c1(OC)ccc2c(C(=O)NCc3cccc4c3OCC4)coc2c1 80502,C1(NC(c2cc(C)nc(O)c2)=O)CC2CC1CN(C(=O)C=Cc1ccn(C)c1)C2 80503,Cc1nc(CN2CCC2(C)C(=O)NC2CC2)co1 80504,c1(C(N2CC(NC(C(CC)(F)F)=O)C(C(F)F)C2)=O)cccc2scnc12 80505,C(CS(=O)(=O)c1ccc(F)cc1)NC(c1cnn(C)c1C)c1n(CC)nnn1 80506,c1(N2CCC(C(=O)OCC)(C(C)C)CC2)cc2c(cc1[N+](=O)[O-])CCC(=O)N2 80507,C1(NC(c2c(OC)cc(C)cn2)=O)CCN(CCc2cnn(C)c2)CC(C)(C)C1 80508,c1(NC2C(C3C(C)(C)CCC3)C2)ccc(S(=O)(=O)NC(=O)CCNC2CC2)c(Cl)c1 80509,c1(CC)cc(CNC(=O)CCC2(NC(c3[nH]ccc3CC)=O)CCC2)on1 80510,N1(C(CCC=C)=O)CCOC2(CCCN(C(=O)C(CC)N3CCCC3=O)C2)C1 80511,C1(CN(CC(c2ccccc2)=O)C)CCCN1C(=O)CNC(c1ccoc1)=O 80512,C(=O)(C(C)(C)CN(C)C)N1CCC(CCNC(Cc2c(C(=O)OC)csc2)=O)C1 80513,C1(C(N(CC(C)NC(c2ncccc2Cl)=O)CC)=O)CC(=O)NC1(C)C 80514,N1(C(c2cc(C#N)sc2)=O)CCN(C(=O)CC2C=CCCC2)CC1C(F)F 80515,C(c1ccncc1)=C(C)C(=O)NCC1CCN1C(C1CSCC(=O)N1)=O 80516,c1(C(=O)OC)c[nH]nc1C(=O)NCCCC(C)NC(C1COC(=O)N1)=O 80517,Cc1ccc(C(=O)NCC2CCC2NC(c2n[nH]cc2C)=O)c(C(C)C)n1 80518,C1(C(N(CC(CO)(CO)NC(C2=CC(C)(CC)C2)=O)C)=O)CC(=O)C12CCCC2 80519,N1(C(CSCC(=O)OCC)=O)CCOc2ncc(-c3nnc(C)o3)c(C)c21 80520,Cc1cc(C)c(CC(=O)NC2COCCN(C(c3cccc(O)n3)=O)C2)c(C)c1 80521,N1(C(CCCC#CC)=O)CC2(CCCC2NC(C2CN(C(C)C)CCO2)=O)C1 80522,c1(CC)occ(C)c1C(=O)NC1COCCC1NC(=O)CCc1cccc(O)c1 80523,CCC(CCCC(=O)N(C)CCC1CCOCC1)NC(=O)CCC(CF)CF 80524,c1(N2CCC(N(CC)CC)C2)ccc(S(=O)(=O)N2C3CCC2CC(F)C3)cc1Cl 80525,C1(CCNC(c2onc(CC)c2C)=O)CN(C(c2c(Cl)cnn2C)=O)CC(C)O1 80526,C1(NC(C2C(C=C)CC2)=O)CC2(CCCCN2C(=O)CNC(=O)CC)C1 80527,c1(C(N2C(C(N(C(C)COC)CC=C)=O)CCC2)=O)ncccc1N 80528,N1(CC(=O)NCCN(CC(C)O)C(c2scc(OC)c2)=O)CCCCC1C 80529,c1(C(=O)NCC(n2cc(COC)nn2)C)ccncc1N(C)C 80530,c1(C(N(CC(C(=O)N(c2cccc(CC)c2)C)C)C)=O)c[nH]c2nccc-2c1 80531,CC1CCC(O)(C(=O)N(CCCNC(=O)CCCc2cc[nH]n2)C)CC1 80532,c1(OC)ncc(C=CC(=O)NCCC2(NC(c3ocnc3C(F)F)=O)CC2)cn1 80533,C1(NC(Cc2cc(OC)no2)=O)CCC(C)N(CCOc2c(C)nn(C)c2C)C1 80534,C(=O)(C(CNC(c1cc(OC)n[nH]1)=O)N(C)C)NC(C#C)C1CCC1 80535,C(N=c1[nH]c(N2CC3COC(C2)C3O)nc2cc[nH]c12)c1ccnc(C)n1 80536,c1(CC)nc(C(=O)N(CC(=O)NC(C2CCCC2)CO)C2CC2)c(C)o1 80537,Cc1cn2c(n1)C(C(=O)NC(C)(CNC(c1ccc(C(F)F)o1)=O)CO)CCC2 80538,CC1CN(C(C2CC2C2CCC2)C(=O)NCc2ccccc2)CC(C)(C)O1 80539,Cc1nc(C(=O)N(C2CCN(C(C3CC(F)C(=O)N3)=O)CC2)CCO)ccc1C#N 80540,Cc1cc(C#N)cnc1C(=O)NCCC1CC(C(N2CC(S(N)(=O)=O)C2)=O)C1 80541,C1(C(=O)O)(NC(c2cnn(Cc3ccccc3)c2N)=O)CCNCC1 80542,c1(CC(=O)NC2COCCN(C(CCCC)=O)C2)ccc2ncsc2c1 80543,c1(NC(CN(C(=O)CC2(C)CCOCC2)CCC)=O)cccc2c1CCO2 80544,c1(CC(=O)NC2C(C(=O)NC(C=C)C)C2)cc(C(F)(F)F)nn1C 80545,C1(C(N(C2CCCN(C(=O)CSc3csc(=N)[nH]3)C2)CC)=O)CCCN(C)C1 80546,c1(C(=O)NCC(CNC(C=CCCC)=O)C)ccc2c(c1)N(C)C(=O)CO2 80547,c1(SNC(=O)CNc2cccc(NC(=O)C=C(Cl)Cl)c2)nccc2ccccc12 80548,c1(C(=O)NC2CCN(C(Cc3c(C)nsc3)=O)CC2)ncnc2c1CCCC2 80549,c1(CCC(=O)NC2C(NC(C=CSC)=O)CCC2)ccccc1Cl 80550,n1(CCC)cc(C(=O)NOCC(N2CCC(C(=O)OCC3CC3)C2)=O)cn1 80551,c1(C(N2CCC(C(C)NC(CCC=C=C)=O)C2)=O)c(C)nc2sccn12 80552,N1(C(C=CCCC)=O)C2CCCC1CC(NC(c1cc3cc(Cl)ccn3n1)=O)C2 80553,C1(CC)CCCCC1OCC(=O)NCC1(NC(C2CCCC2C)=O)CCCC1 80554,C1(C(N(C)CCc2ccccc2)=O)COC2CN(C(C3CCCC3)=O)CC12 80555,Cc1ccc(-n2ncc(C(=O)N(C3CCC3(C)C)C)c2C(C)C)cc1 80556,CC(C)CCCC(=O)N(C(C)C(=O)NC1CCCC(F)(F)C1)C1CC1 80557,c1(NCc2ccc(CNC(C3CC(CC)C3)=O)cc2)ncnc2c1c(Br)nn2C 80558,CCC(CCCC(=O)N(CCCC(C)O)C)NC(=O)C(C)(C)n1cnnn1 80559,C1(C(=O)NCC2(NC(C3CC4CC4C3)=O)CCCC2)CCOC2(CCOCC2)C1 80560,c1(C(=O)NCCNC(=O)CN2CC(F)CC2C2CCCCC2)cnc2cncn2c1 80561,C(CNC(=O)C=C(C)CNC(C1CCC(C)(CO)O1)=O)(C(F)(F)F)OC 80562,N1(C(C(C)N(C(C2OCCO2)=O)C2CC2)=O)CCCCCC1 80563,CC(C)(C)CC(=O)NC1CCCC1CNC(C1(C)CS(=O)(=O)C1)=O 80564,N1(CCOC)CCC(NCC2COC3(COC3)C2)C(C)C1 80565,N(C1CCCc2c(C)cccc21)C(C(=O)Nc1cc2nc(CC)oc2cc1)=O 80566,C(C(=O)NCCC(C)C(C)C)(C(C)(C)C)NC(c1cc(C)n(C)c1)=O 80567,C(=O)(CCCC(=O)N1CCCC(N(CCO)C(c2nncn2C2CC2)=O)C1)N(C)C 80568,N1(C(c2ccccc2)=O)CCC2C(CCCN2C(c2nc(C3CC3)cs2)=O)C1 80569,N1(C(c2ccc(C)cc2Cl)=O)CCC2CC(F)(F)CCC2C1 80570,c1(C(N2CC(C=C)C(NC(c3cc(Cl)cnc3C)=O)C2)=O)ccc2sccc2c1 80571,c1(C(=O)NCC2CC(F)(CNC(C3C(C)(C)CC3)=O)C2)cnnc2ccccc12 80572,C(=O)(CC(=O)N(C)C)NC(C1CC(NC(=O)CC2CSC2)C1)C 80573,c1(CC)ccc(C(=O)NCc2ncc(C(=O)NCCCCC(N)=O)cn2)cn1 80574,N1(C(CC(CC#C)c2ccccc2)=O)CCC(NC(=O)C=CCO)CC(O)C1 80575,C1(C)(CNC(Cc2nc(C(C)C)sc2)=O)CCCN(C(C2(C)COC(=O)C2)=O)C1 80576,N1(C(c2n(CCC)ncc2)=O)CC2CN(C(=O)CCn3c(C)ccc3C)CC2C1 80577,CC(CC(=O)N1CCCC(F)(CNC(c2noc(C3CC3)n2)=O)C1)P(C)(C)=O 80578,c1(OCC)cc(OC)cc(N(CC=Cc2ccccc2)CC2CCCN2CC)c1 80579,C1(C(=O)OC)CCC(C(N2CC(CO)(NC(C3CCNC3=O)=O)C2)=O)CC1 80580,CC(C)C(C(=O)N1CC(NC(c2cc3ccccn3c2)=O)CC(F)C1)C(C)C 80581,C(=O)(CCCCC(F)F)N(C1CCN(C(=O)Cc2nc[nH]n2)C1)CC 80582,N1(C(c2nc(COCC)sc2)=O)CC(CNC(=O)C=CS(C)=O)CC1(C)C 80583,C(=O)(CCNC(=O)COC1CCC1)NCC(C)N1CCC1 80584,N1(C(C(CC)F)=O)CC(N(C)C(c2ccc(C(=O)OC)c(Cl)c2)=O)C2(CC2)C1 80585,C1(NC(C2C(CC)OCC2)=O)CCCCC12CCCN(C(C1CCCC1OC)=O)C2 80586,C(=O)(C(C)(C)CNC(C)=O)NC(CC)CNC(c1nnc(CO)s1)=O 80587,c1(C(N2C(CNC(CSC(C)C)=O)CC(O)C2)=O)ccn2nccc2n1 80588,C1(NC(CSCCCC)=O)CC2CC(NC(c3cccc(CN(C)C)c3)=O)CC12 80589,C1(NC(CN2CC(C)(OC)C2)=O)CCCC12CN(C(C1CCCCS1)=O)C2 80590,CC(C)CCCCC(=O)NCc1cn(C2CN(Cc3cccc(N)c3)C2)nn1 80591,n1(CC)cc(C(=O)N(CC(C)NC(=O)C(C)=C(C)C)C)c2ccccc12 80592,N1(C(C(C)NC(=O)NC)=O)CC(NC(=O)CCN2CCOC2=O)CC(F)C1 80593,N1(C(C2CC(C(=O)OC)C2)=O)CC(=O)NCC1C(=O)NCC1CC2CCC2C1 80594,C1(C)(C(N2C(C(N(CC)CC)=O)CCC2)=O)CCCN(c2ccc(Cl)c(C)n2)C1 80595,C1(NC(CC2(C=C)CC2)=O)CCC(C)N(C(c2sccc2CC)=O)C1 80596,C1(C2(O)CN(C(=O)C#CC3CCCC3)C2)(CNC(C2C(C)OCC2)=O)CC1 80597,c1(CC(=O)NC2CC(N(C(C(C)OC3CCCCC3)=O)C)C2)nncn1C 80598,C1(C(C(=O)NC(CC)C)N(C)C(C2CCCO2)C)CCOCC1 80599,C1(CC)CC(CC(=O)N(CC)CC2CCCN2C(C2CC3CC3C2)=O)CCO1 80600,Cc1cc(C(=O)N(C2(C(N3CC(c4c[nH]nc4C)C3)=O)CC2)C)c(C)cn1 80601,Cc1cccc(-c2nc(C(C)CN(S(C)(=O)=O)C)n(C(C)C3CC3)n2)c1 80602,C1(C(=O)NCC(CCNC(CCC=C)=O)(C)C)C2CCC(O2)C1C(=O)OC 80603,CN1CC(=O)N(CC(=O)NC2CCN(C(=O)Cc3cnoc3)CC2F)C1=O 80604,Cc1nn(C)c(Cl)c1C=CC(=O)NCC(C)(C)NC(=O)CCNC(=O)C(C)(C)C 80605,CC1CCCc2cc(C(=O)NCC3(NC(c4nocc4Cl)=O)CCCC3)nn21 80606,c1(C(N2CCCC(N(C(=O)C(O)CSC)CC)C2)=O)ccc2cnccc2c1 80607,n12nc(ccc1=O)C2.CC(C)CS(=O)(=O)N1CCCC1c1nc(-c2cccs2)no1 80608,Cc1cc(C)c(C(=O)NC2CC3CN(C(c4n[nH]c(O)n4)=O)CC23)c(C)n1 80609,N1(CC(N2CC(C(C)NC(=O)C(C)CC(F)(F)F)C2)=O)C(=O)C(=O)N(C)C1=O 80610,C(=O)(C(Cc1cccc(Cl)c1)CCS(C)(=O)=O)c1c(-c2ccc(C)cc2)cccn1 80611,c1(CCC)n[nH]c(=NC(CNC(c2ccc(-c3ncc[nH]3)cc2)=O)(CC)CC)s1 80612,C1(C)(NCCN(C(C#C)C)C(=O)CC)CCCC1 80613,C1(C)(C(=O)NC(C)C(N)=O)CC12CCN(c1cncc(N(C)C)n1)CC2 80614,C(=O)(CC(C)(C)CC(F)F)NC1CN(C(C(C)SC(F)(F)F)=O)CC12CCC2 80615,C1(C(C)C)(C(N2CCCCC2Cn2cc(C(O)C(C)C)nn2)=O)CNC(=O)C1 80616,c1(C(=O)NCCC(C)NC(=O)CN(C)C(c2ccsc2)=O)coc(S(C)(=O)=O)c1 80617,c1(C(N2CCCC(NC(C(CSC)OC)=O)(CO)C2)=O)cccc2oncc12 80618,c1(CC(N2CC(C(C)NC(C(CC)SC)=O)C2)=O)coc2c(F)c(F)ccc12 80619,C1(NC(C(C)OCC(C)C)=O)CCC(CC(=O)NCCC(Cl)Cl)C1 80620,c1(C(N2CCC(NC(c3nc(C)c(C)s3)=O)C(F)C2)=O)cccc2c1OCCN2 80621,c1(C(=O)NC(C)CNC(=O)OC(C)(C)C)csc(S)n1 80622,N(C1c2ccccc2C2CCC1CC2)CC(C)(C)NC(=S)N 80623,CCC(CCCC(=O)NCc1nc(C)c(C)[nH]1)NC(C1(C2(C)CC2)CC1)=O 80624,N1(C(C2(C#C)CC2)=O)CCC(NC(=O)C(C)(F)c2ccccc2)C1 80625,c1(CC(N2CC(CC)(NC(=O)C=C(C3CC3)C3CC3)C2)=O)ccc(C)c(C)c1 80626,C1(C(N2C3CCC(NC(COCCCCC)=O)(C3)C2)=O)CCCCN(C)C1=O 80627,C(CC1=CCN(C(C2(C#N)CCOC2)=O)CC1)NC(c1c(CC=C)cccc1)=O 80628,C(=O)(CC(C)(C)Cc1cccc(O)c1)NCCCC(C)(C)NC(C1C(CC)C1)=O 80629,C1(NC(c2ccc(OC)o2)=O)CC12CC(NC(c1c(Cl)n[nH]c1C)=O)C2 80630,c1(C(N2C(CC)CN(C(C3COC(=O)N3)=O)CC2)=O)n[nH]c2c1CCSC2 80631,C1(N(C(=O)Cn2ccc(=N)[nH]2)C)CCCN(C(=O)CCc2ccsc2)CC1 80632,CS(=O)(=O)c1nc(Cl)cc(=NCC2(F)CC(NC(C3CC34CCSCC4)=O)C2)[nH]1 80633,C(CCCCC(=O)NCc1cncc(C)c1)NC(C(C)=CC1CC1)=O 80634,N1(C(C(C(C)C)NC(N)=O)=O)CCC(NC(C2CCCN(C)C2)=O)C(C)(C)C1 80635,c1(C(=O)NC(CC)CN(C)C(C2(C)CNC(=O)C2)=O)cc(F)cc(F)c1 80636,Cc1ccc2nc(C(N3CCC4CCN(C)CC34)C(=O)NC3CCC3)cn2c1 80637,c1(C(=O)NC(C(C)NC(c2cc(CC)[nH]n2)=O)C(C)C)cc2ccc(Cl)cc2o1 80638,N1(C(c2ccn(CCOC)n2)=O)CC(C)N(C(=O)CCOCC2CC2)CC1C 80639,c1(CC)oc(C)cc1C(=O)NCC1CC(NC(c2cn(C)cn2)=O)C1 80640,CCC(CC(F)(F)F)C(=O)NC1CCC(CNC(c2cc(CCO)on2)=O)CC1 80641,CN1CCN(C(=O)CCCCn2ccnn2)CC1CNC(c1cnnn1C)=O 80642,N1(C(Cn2c(C(=O)OC)cnc2)=O)CC(C)N(C(=O)C=C2CCN(C)C2)CC1C 80643,CCCC(C)C(=O)N1CCN(CC2CN(C(=O)CC(CC)OC)C2)CC1 80644,C(=O)(CC1=CCOCC1)N1CCCC(C(=O)NCC2(C(C)C)CCCC2)C1 80645,CCC(CC(=O)NC1CCCCC1C(=O)NC1CC(NC(=O)C2CC2)C1)SC 80646,c1(N(C)C(C2CCS(=O)(=O)N2)=O)ncc(C(C)(C)O)cn1.N12CCC(CC1)C2=O 80647,c1(C(=O)NCC(C)N(C(c2c(C)ccc(N)c2)=O)C)[nH]c2ccc(F)cc2c1C 80648,c1(CC)cc(C(=O)NC2(CF)CCN(C(=O)CCC3CC(OC)C3)C2)cc(C)c1 80649,CCCCCC(O)C(=O)N1CCC(N2CCN(C(=O)C(C)(C)C#N)CC2)C1 80650,C1(c2nnnn2C)(CN2CCC(CC)C2C)CCN(C(=O)OC(C)(C)C)CC1 80651,c1(C(=O)NCCC(C)N(C(c2nc(C(=O)OC)sc2)=O)C)ccnc(C2CC2)n1 80652,N1(C(C2(CCC)CCC2)=O)CCC(C)N(C(C2CC3CCC2CC3)=O)CC1 80653,c1(C(=O)NCCCN(C(C2(OC)CCSC2)=O)C2CC2)cn(C)c(C(F)F)n1 80654,c1(C(=O)NCC(CC=C)C(N2CCC3(CC2)CC3CO)=O)ccn2cncc2c1 80655,c1(NC2CCN(C(C)(C)C)CC2)ccc(S(=O)(=O)NCC2CSCCS2)cc1Br 80656,C1(CC(=O)N(C(C)CNC(=O)C(C)n2ccnn2)C)CSCCO1 80657,CCCCC(C(=O)N1CCN(C2CCC2)CC1)NC(=O)CN(C)C(C)C 80658,N1(C(c2scc(C)c2)=O)CCC(C(F)CNC(=O)C(F)(F)C2(O)CCCC2)CC1 80659,C12(NC(C(CCOC)OC)=O)CCC(CC1)N(C(c1nc(O)nc(O)c1F)=O)C2 80660,C1(C(N(CC(C)CNC(=O)CCS(N)(=O)=O)C)=O)CC12CCS(=O)(=O)CC2 80661,c1(C(N2CCN(C(C3CCC(=O)NC3)=O)CC2CO)=O)noc2ccc(Cl)cc12 80662,Cc1nc(CO)ncc1NC(C1(CCNC(C2(C)COC(=O)N2)=O)CC1)=O 80663,CC(CS(C)(=O)=O)C(=O)NCC1CN(C(c2ccncc2N)=O)CCCO1 80664,C#CCCCC(C)C(=O)N(CC(C)CNC(c1nc[nH]c1C(C)(C)C)=O)C 80665,N1(C(C(C)O)=O)CCC(CO)C(NC(=O)Cc2c(Cl)cnn2C)C1 80666,c1(C(=O)NCC2CCC(NC(C3(N(C)C)CC3)=O)C2)nnn(C)c1N 80667,Cc1ncc(CCC(=O)NC(C(=O)NC2CCNC2=O)C2(C)CC2)o1 80668,Cc1cc(F)ccc1C(O)CNCC(n1ccnn1)C1CC1 80669,C1(C(=O)NCCCCCN=[N+]=[N-])CCCCCCN1C(C1CC1C(F)F)=O 80670,N1(C(C2CC(C)N(C)CC2)=O)CCCN(C(c2sccc2C(C)(C)C)=O)CC1C 80671,c1(C(=O)NCC2(OC)CCN(C(CCSCC)=O)C2)cccn2cnnc12 80672,C(=O)(C(C)(C)CC(F)F)N1CC(C)(OCC(=O)NCc2nccc(C)c2)C1 80673,C(C)(C(=O)N1CCCC(N(C)C(c2cnc3sccn23)=O)C1)(C(C)C)OC 80674,C1(C(N2C(C)(C(=O)NC)CC2)=O)CC12CC(NC(C1COCOC1)=O)C2 80675,CC1CCN(C(=O)CCc2cnn[nH]2)C(C)C1NC(c1cncc(N=[N+]=[N-])c1)=O 80676,C1(NC(c2ccc(CC)nc2)=O)Cc2ccccc2C1NC(=O)C(C)NC=O 80677,C12(CC(=O)NC3(CN(C)C)CC3)CCC1CN(C(c1ccc(O)cn1)=O)C2 80678,c1(CC(=O)N(CC(C)NC(C(C)OCC)=O)C)c(F)cccc1Cl 80679,N1(C(Cc2c(C)noc2)=O)CCN(C(=O)C2=NOCC2)CC1CO 80680,C1(N(C(C=Cc2c(C)ccs2)=O)C)CN(C(C2CCC=CCC2)=O)CC12CC2 80681,c1(C(=O)NC(C)CN(C(=O)C(O)Cc2cn(C)cn2)C)ccc2c(c1)OCCC2 80682,CCC(C#N)C(=O)N(CCC(N1CCC(F)(C(N)=O)C1)=O)C 80683,c1(C(=O)NCC#CCNC(C(CSC)OC)=O)cccc2c1OCCO2 80684,c1(C(N2CCC(NC3N(C4CN(CC)C4)CC3)CC2)=O)ccc2n[nH]cc2c1F 80685,C1(C(=O)NCC2CN(C(c3ccnc(CC(C)C)n3)=O)C2)CC2CCC1C21CC1 80686,C(=O)(C(O)P(C)(C)=O)NCC(=O)OC(c1ccc(OC)cc1)C 80687,c1(SCCn2c(N(C(CC)CC(C)C)C)nnn2)c(OC(F)F)cccc1Cl 80688,N1(C(c2cc(CC)nc(O)c2)=O)CC(NC(=O)Cc2cnc[nH]2)C2(CCCC2)C1 80689,C(c1ncccc1C)=CC(=O)NCC(CNC(c1cccc(C)c1Br)=O)OC 80690,Cc1cc(C(N2CCC(C(C)(C)C(=O)NCCSC(F)F)C2)=O)c(C)cn1 80691,C1(C(N(C)Cc2c(C)nsc2)=O)CC12CCN(C(c1ncccc1Cl)=O)CC2 80692,CC#CCCC(=O)N1CCC(NC(c2cc(C(F)F)no2)=O)C1C1CC1 80693,C(C(N=[N+]=[N-])C(=O)NC(C)CNC(=O)C(c1ccncc1)C)OCC 80694,c1(C(COC(CC2OCC(C)OC2)=O)=O)cc(Cl)ccc1F 80695,N1(C(c2n(C)cnc2)=O)CCC2(CCN(C(=O)Nc3nc4ccccc4o3)C2)C1 80696,C(C)(C)(CCCC(=O)NCc1nc(CO)n[nH]1)NC(CSCC#C)=O 80697,c1(CNC(CCCC)(C)c2cccc(Br)c2)ccc(O)c(Br)c1 80698,c1(CCNC(=O)Nc2ccnc(N3CCOCC3)c2)ccc(F)c(F)c1 80699,Cn1cnc(C(=O)NC(C)(C)CCCNC(=O)CC2CC3CCC2C3)cc1=O 80700,C12(C)CN(CCO1)C2=O.C12(C(=O)NCc3cn(CCOCC)nn3)C=CC(CC1)C2 80701,c1(CNC(COCC(=O)NC2C(NC(C3CC(CC)C3)=O)C2)=O)ccccc1 80702,c1(C2(C(=O)NCC(CN(C)C(c3sccc3F)=O)(C)C)CC2)ccnc(Cl)c1 80703,C1(N(C(=O)C(O)C(F)(F)F)C)CC2CCC(C1)N2C(c1ccc(Cl)c(Cl)c1)=O 80704,C(=O)(C1=CCC(NC(=O)C(=O)NC(C)C)C1)NC(C(=O)OC)C 80705,C1(C#N)(CC(=O)N(CCCCCC)CCNC(C2(F)CCOC2)=O)CCOCC1 80706,C1(CNC(C(c2cn(C)nc2)(F)F)=O)CCN(C(C2CC2(F)Cl)=O)CC1O 80707,c1(CNc2ccc(OCCC(=O)OC)cc2)c(Cl)cc(Cl)c2nonc12 80708,N1(C(C(C)CNC(=O)OC)=O)CCC2CCN(C(=O)CC3CC3)CC12.C(C)(C)(C)O 80709,CC1CC(C2CN(C(C3CN(C(C4CC4Cl)=O)CCO3)=O)C2)=NO1 80710,C1(NC(c2cccc(CC)n2)=O)CCCCCC1C(=O)NOCC(C)O 80711,CC(C)CC(C(=O)NCCCN1CCC1)ONC(C1CCCCC1(C)C)=O 80712,c1(C(N(C2CCN(C(C(CC)CC)=O)C2)CC)=O)cc(OC)ncc1Cl 80713,c1(C(=O)NCC2(O)CN(C(c3c(CC)ncs3)=O)C2)cccc(Br)c1O 80714,c1(N2CCC(NC)CC2)nc(N2CCC(C)(N(C)C)CC2)nc2c1CC(C)CC2 80715,c1(C(N(C2CCN(C(C(C)SC)=O)CC2)C)=O)cc2ccsc2n1C 80716,c1(C(=O)NCCC(C)NC(COCC(C)C)=O)ccnc(C(F)(F)F)n1 80717,c1(C(=O)NC(C)C(=O)N(C)C)ccc(S(=O)(=O)NCc2c(F)cccc2F)cc1 80718,C(CC(F)F)(C(=O)NOCC1CCCC1)N(C(c1ccc(OC)nn1)=O)C 80719,c1(COC)ncc(C(=O)NCC(C(C)C)NC(C23CC(CCO2)C3)=O)c(O)n1 80720,C1(OCCC)CCCCC1C(=O)NC(C)CNC(c1c(C)noc1C1CC1)=O 80721,c1(C(N(C2CCC(NC(=O)CNS(C)(=O)=O)C2)C)=O)cn(C)c(=O)nc1O 80722,C12(C(N3C(C)CN(C(c4nccn4C)=O)CC3)=O)CCC(C)(CC1)CO2 80723,c1(CC)ccc(F)c(C(N2CCOC(CNC(=O)C(CN(C)C)CC)C2)=O)c1 80724,C1(NC(C2CCC(=C)CC2)=O)CCCCCC1C(N1CCC1CF)=O 80725,C#CCC(CC(F)F)C(=O)NC1CC=C(C(=O)NC(C)CN2CCOCC2)C1 80726,C1(C(=O)NC2(C(=O)NCC#C)CC2)CC(C)CN(C(=O)Cc2ccccc2O)C1 80727,n1(C(C)C)ncc2c(N3CC(F)C(F)C3)[nH]c(=NCC3C=CCCC3)nc12 80728,c1(C(=O)NCCC2CCN(C(C(C)N(C(C)=O)C)=O)C2)onc2c1CCCC2 80729,C1(C(=O)NCC(CNC(C(CC)SC)=O)(C)F)Cc2ccccc2N(C)C1=O 80730,N1(C(CN(C(CCSCC(C)C)=O)CC2CC2)=O)CC(C2CCCC2)C1 80731,C1(C(N(C2CC(NC(C3CC(F)(F)CS3)=O)C2)C)=O)CCc2c[nH]nc2C1 80732,Cc1ccc(CC(=O)NC(CNC(c2scnc2C(F)F)=O)CC(C)C)cc1O 80733,CC1CC(=O)NCC1C(=O)NCC1CCCN(C(=O)C(C)C2CC2)CC1 80734,c1(C(N(CCCNC(=O)CC2CCOC2)C(C)C)=O)ccc(-n2ccnc2)cc1 80735,c1(NC(C2(F)CN(C(CC(C)C)=O)C2)=O)c(F)ccc(Br)c1F 80736,C#CC(CNC(C1CN(C(=O)CC(F)(F)F)CC1C=CC)=O)CC(C)(C)C 80737,Cc1nc(NC(CCN(C(=O)C=CSc2ccccc2)C)C(C)C)cc(C#N)n1 80738,c1(CN(C(C(=O)N(C)CC2CCCNC2)=O)C)ccc2c(c1)OCO2 80739,C(CCC(C)C)(C(=O)N(C)Cc1nc(=O)o[nH]1)NC(CN(C1CC1)CC)=O 80740,c1(C(N(CC(=O)NC(c2ccccc2)C)C)=O)ccnc2[nH]cnc12 80741,CC1OCCCC1C(=O)NC12CC(C(=O)N(C)CC3CCSC3)(C1)C2 80742,N1(C(C2C(NC(=O)CC3(CO)CCC3)COCC2)=O)CCCCCCC1 80743,C(=O)(CC(C(C)C)NC(c1c(C(F)(F)F)coc1C)=O)OC 80744,c1(CNC(CCN(CC)CC)=O)cccc(CN(C)C(C2CC23CCOC3)=O)c1 80745,C(C(=O)N=c1ccc(OC(F)F)n[nH]1)=Cc1ccc(OC)c(F)c1 80746,C1(C(=O)NCC(C)N(C(CC2(OC)CCC2)=O)C)CCC(=O)CC1(C)C 80747,c1(C(=O)NCCCCCCC=C)ccc(O)c([N+](=O)[O-])c1 80748,Cc1cc(C)cc(C=CC(N2CC3CC2CN3C(C2CCC(C(C)C)O2)=O)=O)c1 80749,C1(C(=O)NCC2CC(CNC(C3CCCS3)=O)C2)CC2(CCCC2)CO1 80750,C1(C(N(CC(=O)N(CC(C)(C)C)C(C)C)C)=O)CN(C(=O)OC(C)(C)C)CCC1C 80751,Cc1cc(N2CCC(NC=Cc3ccc(Br)cc3)CC2)ccc1C(=O)O 80752,N1(C(C(C(C)C)F)=O)C(C)CC2CN(C(=O)C(C)Cn3ccnc3)CC12 80753,N1(C(CSCC)=O)CC2CC1CN(C(C1CCS(=O)(=O)CC1)=O)C2 80754,n1(CC(N2CCC(N(C(=O)CNC=O)C)C2)=O)cc(C(N)=O)c(O)nc1=O 80755,Cc1ccc(OCC(N2CCC(N(C)C(C3CC3(F)Cl)=O)CC2)=O)cc1C 80756,c1(C(=O)NCC(C2CCC2)NC(C(C)N(C(C)=O)C)=O)ccc(C(N)=O)s1 80757,C1(N(C(C2C(C(=O)OCC)C2)=O)C)CCCN(C(=O)CC2CC(OC(C)=O)C2)CC1 80758,N1(C(CC(=O)NCC#C)=O)CC=CC1(C(=O)NCc1cnn(CC)c1C)COC 80759,c1(OC)cccc2c1C(C(=O)N1CCCC1CN(C)C(C1(CCO)CC1)=O)CC2 80760,Cc1nn(C)c(C)c1CC(C)C(=O)NC1(CO)CCN(C(=O)C(C)O)CC1 80761,CC1(C)C2CCC1(C(N1CCCC(CCNC(=O)C(F)n3ccnc3)C1)=O)CC2 80762,CC(C)C(C)(C)C(=O)N1CCOC(CC(=O)N(C)CCN2CCOCC2)C1 80763,c1(NC(C(N2CC(CNC(=O)NC)C(C)CC2)=O)=O)ccc2c(c1)C(=O)NC2 80764,CCCCC(CNC(c1n[nH]cc1Br)=O)NC(c1cnccc1C(F)F)=O 80765,CC1CCCCC1(C)C(=O)CC(CO)Nc1nnn(C)c1Cc1ccccc1 80766,N1(C(c2c(OC)nc(Cl)cc2)=O)CC2CS(=O)(=O)CC2(NC(=O)C(C)C)C1 80767,C12(CNC(CCCC#CC)=O)CCCC1N(C(=O)CNC(C)=O)CCC2 80768,C1(C(=O)NC(c2cccnc2F)C)CC(NC(c2cccc(F)c2)=O)C1(C)C 80769,N1(C(=O)NCCCC)CSCC1C(=O)N(CCC(C)NC(C1CCCC1)=O)C 80770,C=CCCCCC(=O)N1CCC(N(C)C(c2nnn(C3CCCC3)c2C)=O)C1 80771,C(=O)(CCCCCCCC1CC1)NCC1(CO)CCCN(C(CC)=O)C1 80772,C1(CC=C)(NC(=O)Cc2ccnn2C)CCN(C(=O)CCc2ccoc2)C1 80773,C(c1cccs1)=C(C)C(=O)NC(C)CC1CN(C(c2cc(C(F)(F)F)no2)=O)C1 80774,Fc1ccc2scc(-c3nc(-c4ccccn4)nn3-c3ccnc(Cl)c3)c2c1 80775,S(=O)(=O)(c1cc2ccccc2s1)N1CCCC(C(=O)NCCC2CCOCC2)C1 80776,c1(C(N2CC(CC(C(N3CC4C(C(=O)NC)C4C3)=O)F)C2)=O)ccc(F)c(O)c1 80777,Cc1c(CN2CC(F)(C(N3CCN(C)C(C)C3)=O)C2)cccc1F 80778,N1(C(C(CN)c2ccccc2)=O)CCOC2CS(=O)(=O)CC12 80779,N1(C(COC(C)(C)CNC(C2CC23CC3)=O)=O)CCCOCC1 80780,Cc1cccc(C(N2CC3(CC3C(=O)N(c3nccs3)C)C2)=O)c1Br 80781,C1(NC(CN(C2CC2)CC)=O)CC(CNC(=O)C(F)n2cccn2)C1 80782,C1(CNC(CN(C(C)=O)C)=O)(CNC(C2C(C)(C)C2(C)C)=O)CCOCC1 80783,c1(C(=O)OC)ccc(C(c2ccc(C(=O)C(C)OC3CCCC3)o2)=O)cc1 80784,C1(CCNC(C(C)OCC=C)=O)CN(C(c2cncc(C)c2)=O)CCO1 80785,C1(C(=O)N(C2CC2)Cc2nc[nH]n2)CC12CCN(C(=O)C=Cc1cncs1)C2 80786,Cc1ccc(C(=O)NC2CCCC(NC(=O)CCC3CCOC3)C2)nc1O 80787,N1(C(c2ncn(CC)n2)=O)CC(N(C)C)C(CNC(C2CC3CC3C2)=O)C1 80788,C(=O)(C(CC(F)F)c1ccccc1)NC(C)CCNC(C1SCCS1)=O 80789,N1(C(C(CCSC)O)=O)CCC(C2CN(C(c3cc(N(C)C)ccn3)=O)C2)CC1 80790,CCCC(C)(CC)C(=O)NC1CC(CNC(c2cc3oc(C)cc3[nH]2)=O)C1 80791,c1(OC)cccc(C(C(=O)NCC2CC2)N(C)Cc2ccsc2)c1Br 80792,C#CC1CN(C(=O)CCSCC)CCN1C(C1CCOC(=O)N1)=O 80793,c1(C(=O)NCCCCNC(C2CN(C(N(C)C)=O)C2)=O)csc([N+](=O)[O-])c1 80794,C(=O)(C(F)CC1CN(C(=O)CNC=O)C1)N(C)CC1CCCCO1 80795,C1(c2nn[nH]n2)(CN(C=O)Cc2c(C3(C)CC3)ccs2)CC2(CCC2)C1 80796,c1(C(C)NC(C(CC)Cc2cccc(C)c2)=O)ccc2c(c1)CNC2 80797,c1(C(C(=O)O)CNC(C#CC(=O)CC)OOCC)ccc(C#N)cc1.CC 80798,Cc1cc(CC(=O)NC2CCC2CNC(=O)CC2CC2)cc(F)c1 80799,C1(C(N(CC(C)NC(c2c(CCC)nco2)=O)CC)=O)CCCCC1O 80800,C12(NC(Cc3scc(C)c3)=O)CCCC(NC(=O)CC(C)(C)O)(C1)C2 80801,c1(CC)cnc(C(=O)NC2(Cc3ccccc3Br)CC2)c(Br)c1 80802,C1(NC(C(C)CN(C)C)=O)CCCCC1CNC(=O)COc1cccc(Cl)c1 80803,c1(C(N2CC(N(C(=O)CCCC(C)(F)F)C)C(O)C2)=O)cc2c(s1)CC(C)(C)C2 80804,C=C(C)CCCC(=O)N1CC(C(C)(C)O)(CNC(C2CNC(=O)O2)=O)C1 80805,N1(C(Cc2nnc(C)s2)=O)CCSCC1CCNC(=O)C(O)CN(C)C 80806,Cc1csc2nc(CC(=O)NC3CC(NC(C4COC5CCCCC45)=O)C3)cn12 80807,C(CN=c1[nH]c(=NCc2cccnc2C)[nH]c2c1COCC2)OCC 80808,c1(C(=O)NCC#CCNC(c2ccc(C3CC3C)o2)=O)cnc(C2(CO)CC2)o1 80809,c1(C(C(=O)NCCC)N(C)Cc2c(C)noc2CC)ccc(F)c2c1CCC2 80810,C1(CNC(c2cc(C)[nH]n2)=O)CCC(C)CN1C(c1cncc(NC(C)C)c1)=O 80811,C(C(C)(C)C(=O)NCC1(F)CCN(C(=O)C(CN(C)C)c2ccccc2)C1)OC 80812,c1(C(=O)NCCNc2nccc(CC#N)n2)cccc2cccnc12 80813,c1(NC(=O)NCc2ccc(OC(C)C)cc2)nc(C)c(CNC(CC)C)s1 80814,c1(C(=O)NC(C2CCCN2C(=O)CCC2CCC2)C)ccc2ncnn2c1 80815,Cn1nc(C(F)F)cc1C(=O)NC(C)(CNC(=O)C1=CCC1)Cn1cccn1 80816,C1(C(N(CCCNC(C2CCN(C)C2=O)=O)CCC)=O)CCN(C)C1C 80817,c1(C(N2CCN(C(c3cc(OC)ncn3)=O)CC2)=O)ccc(N(C)C)cc1OC 80818,c1(C(N2CCC(NC(CSCCC)=O)C23CCC3)=O)ccc(S(C)(=O)=O)cc1N 80819,c1(-c2onc(NC(C3C(CCNC(CCC#C)=O)CCO3)=O)n2)ccccc1F 80820,C1(C(=O)NC(CC=C)CC)CN(C(c2cc(C)c(N)cn2)=O)C(C)(C)C1 80821,c1(CNc2ccc(C(N3CC(C)OC(C)C3)=O)nc2)cn2c(Br)cccc2n1 80822,CC1CC(CNC(c2[nH]ccc2C2CC2)=O)CN1C(=O)C(O)Cc1cnc[nH]1 80823,C1(OC)CCCN(C(C2CC(C)N2C(C2CC(N(C)C)C2)=O)=O)C1 80824,c1(C(N2CC(C)(CNC(c3ccc(C)o3)=O)OCC2)=O)c(N)sc2c1CCSC2 80825,c1(C(N2C(C)CC(NC(C(C)OCCC=C)=O)C2)=O)cnc2c(cnn2C)c1 80826,C(=O)(CC(C)C(F)(F)F)NCCN(C(c1ccc(F)cc1OC)=O)CC 80827,N1(C(CCc2c[nH]c(=N)[nH]2)=O)CCCC(CCNC(=O)Cc2ccoc2)C1 80828,C1(C#N)(C(=O)NC(C)CNC(=O)CC2CCCCC2)CC12CCC2 80829,N1(C(CCNC(Cc2c(C)con2)=O)=O)CCS(=O)CC1C 80830,CC1(NC(=O)CC2COCC(C)(C)O2)CCN(C(c2ns[nH]c2=O)=O)CC1 80831,C(=O)(C1=CCC(C)(C)CC1)N1CCC(C)(NC(CCc2ccc(CC)cc2)=O)C1 80832,Cc1c(C(N2CCC(CN(C)C(C3CC3F)=O)CC2)=O)sc2ccccc12 80833,Cc1ccccc1SCC(=O)NC1CC1CNC(c1cc(-c2ccco2)no1)=O 80834,C1(NC(C(CCC)F)=O)(CO)CCCN(C(C2CCCNC2=O)=O)C1 80835,c1(C(C(=O)NCC2(CCNC(C3C(C)(C(F)(F)F)C3)=O)CC2)C)cccc(O)c1 80836,N1(C(c2c(-c3c(NC(N)=O)cccc3)csc2)=O)CCC2(CCCO2)C1 80837,C1(C(C)C)N(C(=O)C(CCN(C)C)NC(=O)CC2CC3CCC2O3)CC1(C)C 80838,C(CC(C)C(=O)NCC1(NC(=O)C(N2CCCCC2=O)C)CC(F)(F)C1)OC 80839,C(=O)(CC1=CCCC1)NCCCN(C(=O)CCc1ccc(Br)nc1)C(C)C 80840,C1(C(=O)NCC(CCC=C)O)CC2CCC1N2C(=O)C(C)(C)F 80841,N1(C(C(CCN(C)C)NC(c2c[nH]c(=O)cn2)=O)=O)CC(CO)C(C)(C)C1 80842,C1(NC(C(C)(C)c2cc[nH]n2)=O)CCN(C(C2CCCO2)=O)CC1 80843,N1(C(c2ccc(N)c(F)c2)=O)CC2CCC(CNC(=O)Cn3ccnn3)C2C1 80844,C1(CNC(C2(CCCC)CCC2)=O)COCCN1C(=O)CCC1CCCCO1 80845,C1(C(=O)NCC2(O)CC(CNC(c3ncn(C)n3)=O)C2)CCCC12CCC2 80846,Cc1nc(CC(N2CC(CO)(NC(=O)Cn3cnc(C(N)=O)n3)C2)=O)n[nH]1 80847,C(CCC(C(=O)NC1(CCF)CC1)NC(=O)CC1CCC(C)CC1)OC 80848,N1(C(C2C(C(=O)OCC)CC2)=O)CC2CC1CN(C(=O)C(COC(C)C)OC)C2 80849,Cc1cc(N2CCCC(CNC(C3CCCC4(CCC4)C3)=O)C2)ncc1C#N 80850,CC(C)(C)C(O)C(=O)N1C2CCC1C(NC(c1cnc(S)nc1)=O)C2 80851,O=C1COCC2(CN(C(=O)CC3CC4(CC4)CN3C(c3cc(Cl)cs3)=O)C2)N1 80852,C1(NC(C2C(C(C)C)C2)=O)CC2(C1)CN(C(c1cnn(CC3CCOC3)c1)=O)C2 80853,n1(CC)cnc(CCNC(C2CCCC2CNC(=O)COCCCF)=O)c1 80854,C(=O)(C(O)CC(F)(F)F)NC1(CO)CCN(C(CCCc2ccc(C)s2)=O)C1 80855,C#Cc1cccc(NC(=O)COC(C2(S(C)(=O)=O)CCC2)=O)c1 80856,c1(C(C)C)cccc(C(=O)NCC2C3CN(C(=O)CN(C)C(N)=O)CC23)c1 80857,c1(NC(c2nccc(-c3ccc(C)nc3)c2)=O)cc(S(C)(=O)=O)ccc1C 80858,C1(C(=O)NC(COC)COC)COCCN1C(C1CC=CCC1C(F)(F)F)=O 80859,C1(NC(C2CC(=C)C2)=O)CC=C(C(=O)NCc2ccnc(CO)c2)C1 80860,C1(N(C(C2(C(N(C3CCCC3(F)F)C)=O)CC2)=O)CC2CC2)CN2CCC1CC2 80861,N1(C(C(CNC(C2(CCCC)CCC2)=O)CC2CC2)=O)CC(C)CC(O)C1 80862,N1(C(c2nccc(C)n2)=O)CC2(CC(NC(c3c(C)nn(C)c3F)=O)CO2)C1 80863,c1(C(=O)NC(C(C)NC(c2nc(C#C)sc2)=O)C)cnc(O)c(Cl)c1 80864,C1(C(=O)NCc2oc(C(=O)NC(COC)C)c(C)n2)CCCC(=O)N1C 80865,C(=O)(CC(C)CC(C)(C)C)NC1OCCN(C(CN2CC(C)(OC)C2)=O)C1 80866,C1(OC)CC(C(=O)N(C2CC2(C)C)C)N(C(=O)Cn2c(O)nnc2O)C1 80867,N1(C(CCC(=O)N(C)C)=O)CCCC(C)(CNC(=O)CC(O)CN(C)C)C1 80868,c1(-c2cn(C3CN(C)CC3c3ccccc3)nn2)cc2ccccc2o1 80869,N(C1CCc2cc(O)c(OC)cc21)CC(CC)OC.O(C)CC.OC 80870,c1(OC)cc(C(=O)NC(C)CCNC(=O)C(c2ccccc2)=O)c(F)c(Cl)c1 80871,c1(C(N2C(CNC(CCc3ccn(C)n3)=O)CC2)=O)nnn2c1COCC2 80872,C1(O)(CC(=O)NCCC2CCCN(C(c3scc(C)c3)=O)C2)CCCN(C)C1 80873,C=C(Cl)CC(C(=O)N1CC(F)(F)CC1C)NC(C1CCC(C(N)=O)C1)=O 80874,C1(NC(COC2(C)CN(C(=O)Cc3ccoc3)C2)=O)CC2CCC1C2 80875,C1(NC(c2cn(CCC)nn2)=O)CC2CC1N(C(=O)CCOC1CC1)C2 80876,C1(C(=O)NCC2C3N(C(C(C)NS(C)(=O)=O)=O)C(CC3)C2)CCCC2C1C2(F)F 80877,O(N1CCC(CC(=O)NCC(O)CN(C(=O)Cc2cn[nH]c2)C)CC1)CC 80878,C1(C(=O)NCC(C)CNC(=O)C=CC2CCOCC2)CCc2c[nH]nc2C1 80879,c1(C(N(CC(C)NC(c2cc(C(F)F)[nH]n2)=O)C)=O)cc(F)cc(Br)c1 80880,O=C(CC(F)(F)C(F)(F)F)NC1CC2CC1CN2C(C1(CF)CCOCC1)=O 80881,C1(CNC(c2n(C)ccn2)=O)COC(C)(C)CN1C(c1cn[nH]c1)=O 80882,C1(CNC(CC2C(C)C2)=O)CC2CCC1N(C(C1(CN(C)C)CCCC1)=O)C2 80883,N(C(=NCCC1COC(C)(C)OC1)NCC(c1cccs1)=O)CC(=O)NCC=C 80884,Cc1nc(O)ccc1C(=O)N(C1CCCN(C(=O)COCP(C)(C)=O)CC1)C 80885,Cc1ccc(CO)cc1NC(=O)CCC1CC(NC(c2cccn2C(C)C)=O)C1 80886,C(=O)(C1Cc2ccccc21)NC(CC(C)NC(c1cc(OC(C)C)ncc1)=O)C 80887,C(N=C(NC1CC1)N1CCC2=C(COC2=O)C1)C1CN(C)C(C)(C)C1 80888,CC(CCC(=O)NC1CN(C(C2CC2Br)=O)C1)N(C)C 80889,CC1(CNC(=O)CCCC#N)CCN(C(=O)COCC2CCCO2)CC1 80890,C1(C(=O)OCCOC2CCCCC2)CCCC(Sc2cn[nH]c2)C1 80891,CC(O)(CC(F)F)C(=O)NCc1ccc(C(=O)NC2CCCC2)cc1 80892,C1(NC(C2CC(OCC)C2)=O)CN(C(=O)Cc2csc(-c3ccco3)n2)CC1C 80893,c1(CNC(=O)NC(CC(=O)OC)CC(C)C)cccc2nc(CO)[nH]c12 80894,C12(NC(Cc3cc(CC)no3)=O)CCCN(C(=O)CSc3nccn3C)CC1C2 80895,c1(C(=O)NCC(C)NC(c2cccc(SCCC)c2)=O)cnn2c1CCCC2 80896,N1(C(C(=O)NCc2ccc(C)o2)C)C(C)CCCC1C 80897,C1(C(=O)OC)N(C(=O)NCC2(F)CCOC2)CC1(C)C 80898,C1(CNC(C2C(=C)C2)=O)CCCN(C(=O)CCn2ccnc2C)CC1 80899,c1(N(C)CC2CCN(CCC#C)C2)ccc2c(n1)CCC2=O 80900,C1(CC=C)(NC(=O)Cc2cnc(C)o2)CCCN(c2cc(C)nc(SC)n2)C1 80901,N1(C(C=C(C)C(C)C)=O)CC(CO)C2(C1)CN(C(C1(CF)CCOCC1)=O)C2 80902,CCC(CCCC(=O)N1CCCC1CN(C)C)NC(C1CC(O)C(F)C1)=O 80903,Cc1oc(C(C)C)cc1C(=O)NC1CCOCC1NC(=O)CCc1cc[nH]n1 80904,C1(CN(C(C(C)OCC)=O)C)COCCN1C(=O)C(O)CCc1ccccc1 80905,C(=O)(C(CC)C(=O)N1CC=C(C(=O)N2CCS(=O)C(C)C2)C1)OCC 80906,N1(C(c2nnn(CC)c2C)=O)CCC(C(F)(F)F)C(NC(=O)C(C)C2CC2)C1 80907,C1(C(N2CC(CN(C(=O)COCC3(F)CC3)C)OCC2)=O)Cc2cscc2C1 80908,c1(C(=O)OC)cc(NC(Cc2ccccc2OC(C)C)C(C)C)ccc1C 80909,N1(C(C(C(C)C)n2cncn2)=O)CCC(CO)(NC(=O)CCCCC#N)CC1 80910,C(CC(F)(F)Cn1cc(CC(O)COC)nn1)NC(c1c(CC)con1)=O 80911,N1(C(c2c(C)nn(C)c2)=O)CCN(C(c2cc(C(C)C)ccc2F)=O)C(CF)C1 80912,c1(OC)ccc(Br)c(OC)c1O.N12CCCC(C1)Cn1nnnc12.c1(C)nccs1 80913,C1(C(N2C(CC)C(NC(=O)CC(F)(F)F)CC2)=O)CCCCCC1(F)F 80914,Cc1nn(C2CCC2)cc1C(N1CC2CC1C2NC(=O)Cc1ccnn1C)=O 80915,Cc1cccc(C)c1C(N1CC(NC(c2cc3sccc3[nH]2)=O)C2(CC2)C1)=O 80916,C1(C(N2CCC(CCC)(CO)C2)=O)CC(C)CN(C(c2cccs2)=O)C1 80917,C1(C(N(C)C(C2CCC2)C2CC2)=O)COC2(C1)CN(C(=O)CC1CCC(C)(C)C1)C2 80918,C1(NC(c2cc(C)c(C(C)C)cc2)=O)CCSC12CN(C(C1CC13CC3)=O)C2 80919,c1(CC(C(N2CC(C#N)(SC)C2)=O)C)ccc(F)c(F)c1 80920,C1(C(=O)NC2C(C)C2C)CC2(CCN1C(C1CC(C)(F)C1)=O)CC2 80921,c1(OC)cnc2c(c1)C(NS(=O)(=O)CCOC1CC1(F)F)CCC2 80922,C(C(=O)NCC(O)CNC(=O)COC(C)CC)(OCC)OCC 80923,CC#CCCCC(=O)NCC12CC(COC)(CN1C(c1ccnc(OC)n1)=O)C2 80924,c1(C(N2CC3C(C(=O)Nc4c(Br)ccnc4Cl)C3C2)=O)c[nH]c2cccnc12 80925,C1(NC(c2c(CC)nns2)=O)CCC(C)N(C(C2(COC)CCC2)=O)C1 80926,CCC(CN(C)C)CC(=O)NC1C2CC1N(C(=O)CNS(C)(=O)=O)C2 80927,C1(CNC(C(C)Oc2ccccn2)=O)C2CN(CCC3CC3)CC12 80928,c1(C(=O)NC2C(NC(c3c(C)nc(Br)o3)=O)CC2)cnc2ccccn12 80929,C1(CNC(CCCC#CC)=O)C(C2CC2)CCN1C(C1CCN(C2CC2)CC1)=O 80930,C1(CC(N2CC(C(C(=O)NC(C3CCCCC3)COC)OC)C2)=O)CCCN(C)C1 80931,C1(C(=O)NCC2(C(N)=O)CN(C(C3CCC(=O)N3)=O)C2)CC2C=CC1O2 80932,C1(CCC)CCC(C(C(=O)NC(C)CC)N(c2ccncc2)CC)CC1 80933,N1(C(=O)C(Cl)=CCl)CCC2CN(C(=O)C(F)(F)c3ccsc3Cl)CC2C1 80934,N1(C(CN2C3CN(C(C(C)(C)C)=O)CC2CCC3)=O)CCC2(CC1)CNC(=O)O2 80935,C1(CC(=O)NCCOCCCNC(C2CC(CC)C2)=O)CCCC2CCCCC12 80936,C1(NC(CC2(CC)CCC2)=O)C=CC(CC(=O)NC(C(O)CO)C2CC2)C1 80937,C1(C(=O)NC(C2(O)CN(C(c3cc(N(C)C)ccn3)=O)C2)C)CC(C2CC2)=NO1 80938,C(=O)(CCCC(C)(C)C#N)N1CCCC(CN(C(C(CCC=C)(F)F)=O)C)C1 80939,C(=O)(C(C)C(F)(F)F)NCC=C1CCN(C(c2cncc(CC)c2)=O)CC1 80940,C(=O)(C1=CC(C)(CC)C1)NC(C1(O)CN(C(c2c(CCC)[nH]cc2)=O)C1)C 80941,N1(C(C(CC#C)C2CC2)=O)CCOC2(C1)CN(C(=O)C(C)(C)CO)C2 80942,CC(C)CC(C)(O)C(=O)NC(CC(=O)NC1CC(N(C)C)C1)C(F)(F)F 80943,c1(CC(CC2CC2)NC(CC2(NC(=O)OC)CC2)=O)cccc(OC)c1 80944,C(=O)(C1CCc2cccc(=O)n21)N1C(C(=O)NC)CC(OC)C1 80945,c1(C(=O)NC2CC(N)C2)cc(N2CCOCC2)nc(Cl)c1 80946,C1(NC(C23N(C(C4N(CC)CCC4)=O)CC(C2)C3)=O)CCCCCCC1O 80947,Cc1c(Br)cc(S(=O)(=O)N2CCCN(Cc3ccccc3)C(C)C2)c(C)c1C(=O)O 80948,c1(C(N(C2(CC(=O)NCC(O)CC(F)(F)F)CC2)C)=O)cccn2nccc12 80949,N1(C(CNC(=O)OC)=O)CCC(NC(c2ncc3[nH]ncc3n2)=O)C2(CCC2)C1 80950,CC(C)(CC(F)C(=O)NCc1nc(C2CC2)n[nH]1)NC(c1cccc[n+]1[O-])=O 80951,N1(C(c2ncn(C)n2)C(=O)NCSc2ccccc2)CCCC2(CO)CCCCC12 80952,Cc1nn(C)c(C(C(=O)NC2CC2)N(C)CCC2CCCCN2C)c1Br 80953,N1(C(C(C)OCCC(C)C)=O)CCC(C(C)C(=O)NCC2(C)CCCO2)CC1 80954,C12(C(=O)NCCCN(OC)C)CCCC1CCN2C(C1CCOCC1)=O 80955,N1(C(C2(CCCF)CC2)=O)CCC(O)(c2ccccn2)CC1 80956,CC1(C)CC(C(=O)NCC2(C)CC2(F)F)CN1C(c1ccc(C#N)cn1)=O 80957,N1(C(C=C(CC)CC)=O)CCC(NC(=O)CC2CC2(C)C)C12CCC2 80958,c1(OC)ncc(C=CC(N2CC(C)CCC2CNC(=O)C=C(C)C(F)F)=O)cn1 80959,C1(CC(=O)N(CCCNC(=O)C(c2ccc(C)s2)C)C)(CC)CCOCC1 80960,C#CCC(CC(F)F)C(=O)N1CC(NC(c2n[nH]c(C)n2)=O)CC1(C)CC 80961,C(=O)(C1=NNC(=O)C1)N1C(CNC(=O)CC2C=CCC2)CC1 80962,Cn1ccnc1C(F)(F)C(=O)NCC1CCN(C(=O)Cc2cnc[nH]2)C1 80963,c1(OCC)cnc(N2CC3C(CNC(=O)C(C)CCN(C)C)C3C2)nc1C 80964,C(c1cccnc1)=CC(=O)NC(C(=O)NCC(CO)C1CC1)c1ccco1 80965,Cc1ccc(C(F)(F)C(=O)N(CC2CN(CC(C)(F)F)C2)CC2CCCC2)cn1 80966,C(=O)(C(C)(C)C(C)NC(c1cn(C2CC2)cn1)=O)NCC(N1CCCC1)C 80967,c1(OC)cn(CCNC(=O)NC(CC(N)=O)C2CCOCC2)c(C)cc1=O 80968,C(=O)(CC(C(F)F)NC(=O)CCc1csnn1)N(CC)Cc1ccccn1 80969,N1(c2n(CC3CCC(C)C3)c(C(O)C3CC3)nn2)CCn2nnnc2C1 80970,C1(NC(c2cc(C)c(C)o2)=O)CC2CC(C1)N(C(=O)CCc1cn(C)nn1)C2 80971,C1(NC(Cc2c(C)cc(F)cc2)=O)C2COCC1CN(C(=O)CC1CC(F)C1)C2 80972,C1(C(=O)NC2CCCN(C(C3(C4(C)CC4)CC3)=O)C2)CCC2CC1CO2 80973,n1(CCOCCC(=O)NC(C(C)N(C)C)C)cc(C2(C)CC2)nn1 80974,CC1CN(C(=O)C(c2ccccc2)O)CC1CNC(=O)C(c1ccccc1F)O 80975,c1(C(=O)NC2CCCC(N(C(=O)CC(C)(F)F)C)C2)cc(S(C)(=O)=O)cnc1O 80976,C(=O)(CCCC(C)(C)C)NC1CCC(NC(c2cn(C)nc2Br)=O)C1 80977,c1(C(N2C(CNC(c3ccnc4cc[nH]c34)=O)CCC2)=O)cc([N+](=O)[O-])ccn1 80978,c1(C(N2CCC(NC(C3(C)CCN(C)C3)=O)C2)=O)ccnc2ccnn12 80979,C1(N(C(=O)CCc2ccon2)N(C2CCCC2)CC)CCn2ncnc2C1.CC 80980,C1(C(=O)Nc2cccc(C)c2)CC2(CCN1C(=O)CNC=O)CC2 80981,N1(C(Cc2n(C)ncc2Cl)=O)CC(CNC(C2CCCC(=O)N2)=O)C2(CCC2)C1 80982,CCCCC(C(=O)N1CC2CN(C(c3ccc(CO)cn3)=O)CC2(C)C1)C(C)C 80983,c1(OC)ccc(O)cc1C(N1CC(OC)CC1CNC(=O)CC12CCCC1C2)=O 80984,N1(C(C(C2CC2)OC)=O)CC(O)CC1CC(=O)NC(C1CCOC1)CO 80985,c1(CC)ccc(C(C)CC(=O)NC2C=CCN(C(=O)COc3ccsn3)C2)cc1 80986,C#Cc1ccc(CC(=O)NC(C)CN(C(c2ccc(C(F)F)cn2)=O)CC)cc1 80987,N1(C(C(C)SC)=O)CCN(C(C23CC(CO2)C3)=O)C2CCCCC2C1 80988,O=C(N=c1c(Cl)c[nH]cc1I)c1cc2c(s1)CCN(Cc1cnc(O)nc1O)C2 80989,c1(OC)cc(Cl)c(Br)cc1NC(c1ccc(-c2csc(C)n2)cc1)=O 80990,c1(CN(C2CCN(c3ccc(C)cc3)CC2)CCC)c(C)n[nH]c1C 80991,C1(C(=O)NCC(C)NC(C=C(C)c2ccsc2)=O)CC2(CCC(F)(F)CC2)CO1 80992,Cc1csc(=O)n1CCC(=O)NCC1(CNC(C2CS(=O)(=O)C2)=O)CCCCC1 80993,C(CCC(C)(C)N(C)C)NC(C1(CC=C)CN(C(=O)CN(C)C(C)=O)C1)=O 80994,c1(C(=O)NC(CC(C)C)(C)CNC(=O)CC2CCC2)cnc2n1CCCC2 80995,Cc1cc(C(=O)NC2CN(C(=O)CC(C)c3ccncc3)CCC2F)cc(F)c1 80996,C1(NC(c2cc(C3(C)CC3)n[nH]2)=O)CCN(C(C2CCOC2)=O)CC1CO 80997,C(=O)(C(CNC(=O)C(F)=C(C)C)(CC)CC)NCCC(CC=C)(C)C 80998,N1(C(C=CCOC)=O)CCCC(C(=O)NC(C)C(N)=O)C1 80999,c1(COC)cccc2sc(NC(C3CCC(C#N)C3)=O)nc12 81000,c1(SCC(=O)NCC2(CNC(CCCOC)=O)CCC2)cc(C)ccc1C 81001,c1(C(N(C(C)CCO)C)=O)ccc(C2COCCN2C(C2CC2C(F)F)=O)n1C 81002,c1(CCNC(=O)NC2CC(O)C2)c[nH]c2c(F)cc(Cl)cc12 81003,C12(C(N3C(C)CC(NC(CC4C(C)C4)=O)C3)=O)CCC(C)(CO1)C2 81004,C(=O)(C(C)(C)C(=O)NN1Cc2ccccc2C(=O)N1)OC 81005,C1(NC(Cc2cnc(C)[nH]2)=O)CC(C)N(C(=O)C(C2CCCO2)C2CC2)C1 81006,CCCC(C)(C)C(=O)NCC1(F)CCN(C(c2noc(C3CC3)c2C)=O)C1 81007,C12(CNC(C3C(C)(C)CO3)=O)CC1CN(C(N)=O)C2.C12CC(C1)NC2=O 81008,C1(NC(C2(c3scc(C)n3)CCC2)=O)CCC(Cc2cn(C)cc2C(F)F)CC1 81009,c1(C(=O)NC2C(NC(CC3=NNC(=O)C3)=O)C2)cc2ncc(Br)cc2o1 81010,C(c1cccc(F)c1)=CCC(=O)N(CCN(C(C1CC2(CC2)CO1)=O)CC)CC 81011,Cc1ccc(CN(C(c2ccc(C#N)s2)C(=O)NC2CCC2)C)c2ccccc12 81012,N1(C(CNC(C2C(C)=CCS2)=O)=O)CC2CCCCCC2C1 81013,Cc1ccc(CC(N2CCCC2(C)CNC(=O)COC2(C)CCC2)=O)cc1Cl 81014,c1(COC)nn(C)c(Cl)c1C(N1CCCCC(CNC(=O)C=CCO)C1)=O 81015,c1(C(N2CCCC(NC(COC(CC)(C)C)=O)C2C)=O)cnc(S(C)(=O)=O)s1 81016,c1(C(=O)NCC2CN(C(c3cnc(SC)s3)=O)CC2C)cc(C)c(F)c(C)c1 81017,CC1CN(C(=O)COC2CCCC(C)C2)CC1NC(=O)C(N1CCCCCC1)C 81018,c1(NC(C(CC=CC)NC(C2CCCN2C=O)=O)=O)cnc(C)nc1C 81019,C1(OC)(CNC(C2SCCS2)=O)CCN(C(=O)Cc2cccc(Cl)c2)C1 81020,N1(C(C(C)SCC)=O)CC(CO)C2(C1)CN(C(=O)C(c1cnn(C)c1)O)C2 81021,N1(C(Cc2c(C)cccn2)=O)CC2CCC1C(NC(c1cc(N)ccc1F)=O)C2 81022,C1(NC(C2(NC(CC3(C)CC3)=O)CCSC2)=O)CC2(CCOC2)C1 81023,Cc1noc(C)c1CSCC(=O)N(CC(C)NC(C1(O)CCOCC1)=O)C 81024,C=CCCC(C(=O)NCc1cc(C)on1)NC(=O)C(C)CC(=O)OC 81025,C(=O)(CCCC(=O)N1CC(C2CC2)(C(=O)NC2(C)CCSC2)C1)OC 81026,C12(NC3CN(CC(N)=O)C3)CC(c3nn[nH]n3)(C1)C2(F)F 81027,c1(-c2n(C)ccc2)ccc2c(n1)N(C(c1ncc(CC3CC3)cn1)=O)CCC2 81028,CC1(C)OC2(C(=O)NCCCn3cc(C4(O)CCOC4)nn3)CCC1C2 81029,C1(CC(=O)OCCC2CN(C(=O)OC(C)(C)C)C2)CCCCNCC1 81030,c1(C(=O)NCC2CC(NC(C(CC(=C)C)C)=O)C2)cc2ccc(F)cc2o1 81031,C1(NC(=O)C2=NOC3COCC23)CCC2(CCCCC2)CC1 81032,n1(CC(=O)NCC2C=CCN2C(=O)CC2C=CCC2)nc(C(F)F)c2c1CCC2 81033,c1(C(=O)NCC(CNC(c2ccc(Cl)c(Cl)c2)=O)F)cccc2ccncc12 81034,CC1CC(C(=O)NC(C2CCCC2)CNC(c2cc(O)no2)=O)CCC1C 81035,c1(C(=O)NC2(CCCNC(CC(C)CF)=O)CC2)ccc(S(N)(=O)=O)cc1 81036,C1(C(=O)NC2CCC(C)(CNC(c3nnc(C)s3)=O)CC2)CN2CCN1CC2C 81037,CCC(CC)(C(=O)NC1CCCC(CC(=O)NC(CN(C)C)C(C)C)C1)OC 81038,C=C1CC(C)(NC(=O)CC2C(NC(=O)CC3CC(C)C3)CC2O)C1 81039,C1(NC(CCC=C=C)=O)CN(C(=O)C(Cl)=CCl)CC2(CC2)C1 81040,CCC(F)(F)CC(=O)NC(C)(CNC(=O)CCNC(=O)C=CCl)C1CC1 81041,C(=O)(CCC(F)(F)C(=O)N1CC(C)(C)CC1CNC(=O)CC(C)(C)CC)OCC 81042,C12(C(=O)N)CCC(CO)(CC1)C2.C(=O)(CCNC(C1CC(CF)C1)=O)NC(CC)C 81043,c1(C(=O)NCC2(OCC)CN(C(=O)C(C3CCC(=O)N3)C)C2)ccc(=N)[nH]c1Cl 81044,c1(C(=O)NC(CC(C)NC(Cc2c(C)cccc2)=O)C)ccn(C(C)C)c(=O)c1 81045,C12(C(=O)NCC3C(CNC(C4(CC#C)CCOCC4)=O)C3)CCCC(CO1)C2 81046,C(=O)(C(C)CNC(=O)C(C1CCOCC1)=O)NCCOCCCC#C 81047,C(c1cc2ccccc2o1)=CC(N1C(C(=O)Nc2c(CC)cc(Cl)cc2)CC1)=O 81048,c1(CCC(=O)NC2CCC2NC(=O)C=CCOc2ccccc2)ccccc1F 81049,C1(C(=O)NCCN(CCC)C(C2CCNC2=O)=O)COCCC1(F)F 81050,C(=O)(C(O)C(C)C)NC1C(NC(c2ccc(CSC)o2)=O)CCC1 81051,C1(C(N(C)CCNC(=O)Cc2ccccc2O)=O)CN2CCC1(C)CC2 81052,C(CO)(CCCNC(c1occc1C1CC1)=O)NC(=O)COC(F)(F)F 81053,CC#CCC(C(=O)NCCC1(C)CCCC1)NC(c1cnn(CCO)c1)=O 81054,c1(C(=O)NCC(C2CCN(C(=O)C(N)=O)CC2)(C)O)ccc(N)cc1[N+](=O)[O-] 81055,Cc1ncn(C)c(=O)c1C(=O)NCC1(NC(=O)Cc2ccsc2Cl)CCC1 81056,C1(C(=O)NC(C)CCNC(C2(C(C)(F)F)CCC2)=O)CCOC2(CCCC2)C1 81057,C1(N(CC(N2CCN(C(=O)C3CC3)C(C3CCC3)C2)=O)C)CCC2(C1)CC2(F)F 81058,c1(C(=O)NCC2CCC(NC(C(=O)NCC)=O)C2)cc(C)ccc1N1CCCC1 81059,c1(C(C(=O)NCC(CNC(c2ccc(CC)o2)=O)(C)O)O)ccc(F)c(Cl)c1 81060,C1(CNC(=O)NC(C(=O)OCCCC)C)(CC)CCCC1 81061,Cc1cncc(CNCc2c[nH]nc2C(F)F)n1 81062,c1(N2CCC(SCC)C2)ccc(S(=O)(=O)N(C)C(c2ccc(C)c(F)c2)C)cn1 81063,CC1(CNC(C2(n3cccc3)CCCC2)=O)CCN(C(=O)CC2CNC(=O)N2)C1 81064,c1(OCC)ccc(C)cc1C(=O)NC1CCN(C(C2(C)COCCO2)=O)CC1F 81065,N1(C(C(CC)F)=O)CCC2C(CCN2C(=O)Cc2cccc(OCCOC)c2)C1 81066,c1(C(=O)NCC(CNC(=O)COc2ccccc2)OC)c(Cl)ccc2c[nH]nc12 81067,N1(C(C(c2cccc(OC)c2)OC)=O)CCC(C)(C)C(CNC(=O)C2CC2)C1 81068,C1(C(N2CC(NC(=O)C(Cc3ccccc3)OC)C(F)C2)=O)(CC)CCOCC1 81069,c1(C(N(C2CCN(C(=O)COC3(C)CCCC3)C2)C)=O)cn(C)nc1C1CC1 81070,c1(C(N(C)CC2CN(C(c3nccn3C)=O)C2)=O)cc2c(cc1O)OCCO2 81071,C#Cc1cc(NC(c2ncc(Cl)n2C)c2nnnn2CCOCC)ccc1Cl 81072,C(CO)(C(=O)N=c1ccn(CCc2c(F)cccc2Br)[nH]1)N(C)C 81073,CC1CN2CCN1C(C(=O)N(CC(=O)O)Cc1cc(F)ccc1Cl)C2 81074,CCCCC(CCCC)C(=O)Nc1ccccc1CN(C)C 81075,C1(CCNC(C(C=CC)O)=O)CC2CCC(C1)N2C(=O)CC1(OC)CCCCC1 81076,C(N=c1[nH]c2ccc(F)cc2o1)C1CCCN(C(c2ccc(OC)cn2)=O)C1 81077,N1(C(C2(NC(C3CC(C)(C)C3)=O)CC(CO)C2)=O)CCC(C#N)C1 81078,c1(OC)cc(Br)c(Cl)cc1NC(C1CCCN(Cc2cncc(C#N)c2)CC1)=O 81079,Cn1ncc2c(N(c3ccc(F)cc3)C(=O)CCOc3ccccc3)ncnc12 81080,c1(C(=O)NC(CCNC(c2c(NC)cccc2)=O)C)ccc(F)c(F)c1 81081,c1(C(N(C)CC2(CNC(c3sccc3F)=O)CC2)=O)cnc(-n2ccnc2)nc1 81082,c1(C2C(NC(C(C3CN(C(=O)C(C)(C)Cl)C3)OC)=O)C2)cnnn1C 81083,Fc1cncc(-c2nc(C3C4CC4C4CC34)n(Cc3ccsc3)n2)c1 81084,C12(NC(c3n[nH]c(C)c3C)=O)CCOCC1CN(C(C1C3(CC3)C13CC3)=O)C2 81085,c1(C(c2n(CCCC)nnn2)NC(c2noc(C)n2)C)cc(Br)nn1C(C)C 81086,CCC(CNC(=O)NCCC(C)(C)C1CC1)CC(F)(F)F 81087,c1(CCC(=O)NC2CN(C(C3(OC)CCC3)=O)CC2C)ccc2[nH]ccc2c1 81088,C1(N(C(C(CNC(C=CC)=O)CC2CC2)=O)C)CCCCCCC1 81089,C1(C(N2CCC(CC)C2CNC(=O)Cc2c[nH]nc2O)=O)CC12CCC(=O)CC2 81090,N1(C(C(C)SC(C)C)=O)CCN(C(c2ccc(Cl)s2)c2nnnn2C)CC1 81091,C(C)(C)(C(=O)N1CCC(OCCNC(c2cnc(-c3cccnc3)s2)=O)C1)OC 81092,N1(C(C(CNC(C2(CCCC)CC2)=O)O)=O)CC2CCCC1C2 81093,c1(C(=O)NC(C)C(=O)NC2CC(CF)C2)cn2ccccc2n1 81094,N1(C(c2nc(C(C)C)oc2)=O)CCN(CCN(C(=O)C(C)(C)CF)C(C)C)CC1 81095,CC(C(=O)NC1CC(C(F)(F)F)(C(F)(F)F)C1)S(=O)(=O)CCCC(F)(F)F 81096,C1(NC(=O)CC2CCCO2)CC12CCN(C(c1cc(F)c[nH]1)=O)C2 81097,c1(-c2cc(Oc3n(C)ccn3)ncc2)c[nH][nH]c1=NC(=O)c1ccsc1C#N 81098,C1(C#CC(=O)N(CC(=O)N(C)Cc2cncnc2)CC(C)C)(CC)COC1 81099,c1(C(N2C(C)(CC)CCC2)=O)cc(C(NC(CCCC#C)=O)C2CC2)n(C)c1C 81100,CC1CN(C(C23CC(CN(C(=O)CN4CCNC(=O)C4)C2)C3)=O)CCN(C)C1 81101,Cc1ccc(C(N2CCCC(N(C)C(c3ccnn3C)=O)CC2)=O)nc1F 81102,CC1C(C(=O)NC2CC(CNC(c3ccn(C)n3)=O)C2)CCN1C 81103,CC(C(=O)N1CC(O)(CNC(C2CC(F)(F)C2(C)C)=O)C1)P(C)(C)=O 81104,N1(CC(=O)NCCN(C(=O)C(O)C2CCC2)C)CCCCCC1=O 81105,c1(C(N2CC(NC(C3(CCC=C)CNC3)=O)C2)=O)ccc(OCCF)cc1 81106,C1(CC(N2C(CN(C(c3[nH]cc(C)c3)=O)C)CCC2)=O)COCC(C)(C)O1 81107,N1(C(Cn2ccc(C)n2)=O)CC2CCN(C(c3nc(Cl)oc3C)=O)CCC2C1 81108,C1(C(=O)NC(C)CCc2ccco2)CC2CC(F)(F)CC(C1)C2=O 81109,C#CCCCCN=C(NCCc1cccs1)NC1CCN(CC(F)(F)F)C1 81110,Cc1nn(CC(N2CCOCC2CC(N2C(C)CCC2C)=O)=O)c(C)c1[N+](=O)[O-] 81111,CC1CN(C(=O)CCN(C)C(C2C3CCCCC23)=O)CC1O 81112,Cc1cccc(C)c1-n1cc(C2(O)CN(C(C3(F)CCOC3C)=O)C2)nn1 81113,c1(C(=O)NC2C(CC)N(C(C3COC(C)C3)=O)CCC2)ccc(Cl)c(Cl)c1N 81114,C1(N(C2CN(CC)C2)C(=O)C(C2COC(C)C2)SSC(=N)S)CC(C)CC(C)C1 81115,c1(CC(N2CC(C)(C(=O)Nc3cnc(Br)cn3)C2)=O)ccc2c(c1)CCCO2 81116,c1(OCCC)cccc(CC(=O)NCC2CCN(C(C34CCC(C3)C4)=O)C2)c1 81117,C(C(C)CC(=O)N1CCC(N(C(c2cn(C)cc2C)=O)CC2CC2)C1)OC 81118,c1(C(N(CC)CC2CCCN2C(=O)C=CC(C)(C)C)=O)ccc(N(C)CC)cc1 81119,C1(C(=O)NCC(CNC(c2cnc(OC)nc2C)=O)O)CCC(=C(F)F)CC1 81120,N1(C(c2cc(OC)ncn2)=O)CCC2(CCC(NC(C3CCC(O)CC3)=O)C2)C1 81121,C12(C(=O)NC(C)(C)CCNC(=O)C3=NOC(C)(C)C3)CC(C)(C1)OC21CCC1 81122,N1(CC(N2CC(CC)N(C(=O)CC3CCCN3C)CC2)=O)C(=O)CC(C)(C)C1=O 81123,CC1CN(C(C2CCN(C(C3CC(O)CN3)=O)CC2)c2ccccc2)CC(C)O1 81124,N1(C(c2c(C)cno2)=O)CCCC(N(C)C(c2ccc(-c3ncc[nH]3)nc2)=O)C1 81125,c1(N2CC(C(C)NC(C3C(OCC)C3)=O)C2)cc(C)nc2cc(C)nn12 81126,c1(OC)ccc(C(=O)N(C2CCCC2)CCNC(c2ccccn2)=O)nc1Cl 81127,Cn1nnc2cc(C(=O)NCC3CC3CNC(c3conc3C(C)(C)C)=O)sc12 81128,c1(OCC)nc(Cl)ccc1C(=O)NCCC(C)(C)NC(c1cnc(C2CC2)[nH]1)=O 81129,c1(C(N2C(C(=O)NCC(F)F)CC(OC)C2)=O)cc2ccc(C)cc2s1 81130,N1(C(COC)=O)CCC2(C1)CN(C(=O)CCCC1CC1)CCO2 81131,c1(C(C)(F)F)cncc(C(=O)NC2CCCCC2NC(=O)CCC2CCCO2)c1 81132,Cn1nnc2cc(C(=O)NC3CCC34CN(C(c3cc(Cl)cs3)=O)C4)cnc12 81133,C1(N(C)C)(C(=O)NCC(O)CNC(=O)CCC2CCCO2)CCCOC1 81134,C1(C(N(C(CCO)C(C)(C)C)C)=O)N(C(=O)OC(C)(C)C)CC12CCCC2 81135,N1(C(c2ccc(CC)s2)=O)CCC2(COC(CNC(C3(C(N)=O)CCC3)=O)C2)C1 81136,C1(C(C)(C)NC(CC2CC(=C)C2)=O)CC2CCC(C1)N2C(c1c[nH]c(=N)s1)=O 81137,c1(C(N2CCC(C(C)NC(=O)C(C)=CC(C)(C)C)C2)=O)ccccc1S(C)(=O)=O 81138,C1(CCC(=O)NC(C)CN(C)C(c2nnnn2-c2ccccc2)C)CCC(=O)N1 81139,c1(C(=O)OC)cc(=NC(=O)NCCC(C(C)C)OC)[nH]n1C 81140,CCC(C)(CCC(C)C)C(=O)NC1CC(C)(NC(=O)C(C)S(=O)(=O)C(C)C)C1 81141,c1(CN(C(C(=O)NCCSC)CC2CCCCC2)C)ccc(F)cc1Cl 81142,C1(NC(C2C(=C)C2)=O)CCN(C)C12CCCN(C(=O)CNC(C1CCCC1)=O)C2 81143,C(=O)(CS(=O)(=O)C1CC1)NC12CCN(C(CCC(=O)OC(C)(C)C)=O)CC1C2 81144,C=CC1CN(C(=O)C(CC(F)F)N(C(=O)C(CCC)OCC)C)CCO1 81145,C1(COCC(=O)NC(CCN(C(C(C)C2CC2)=O)C)(C)C)CCCCO1 81146,c1(C(=O)NC2(C)CN(C(C3CC(OC)C3)=O)C2)nccn2c(C)nnc12 81147,C1(NC(CC(CC)(F)F)=O)CN(C(C2CCCN2C(=O)OC)=O)CC12CCC2 81148,c1(C(=O)NC(CC)CNC(C2CCC(F)C2)=O)ccn2ccnc2c1 81149,c1(C(C(=O)NCC=C)N(CC(C)C)Cc2ccc(C)s2)cc(Br)c(C)nc1OC 81150,Cc1nc(C(N2CC=CC2(C)C(=O)NCC2(CO)CC3CC3C2)=O)cc(O)n1 81151,N1(C(c2c(C)nn[nH]2)=O)CC(NC(C2CC(=O)N(C(C)C)C2)=O)C(CC(C)(C)C)C1 81152,c1(C(=O)NN2CC3CC3C2)cn(CCNC(=O)CSc2cn[nH]c2)cn1 81153,Cc1cc(C#N)cc(C(N2CC=CC2CNC(=O)CCc2ccccc2C)=O)n1 81154,C(=O)(C(C#N)C(C)C)NC(CCC)C(=O)NCCc1cc[nH]n1 81155,C(=O)(C(F)(F)C(F)F)NC1CCC(CNC(CC(C)(C)SC)=O)C1 81156,c1(C(=O)NCc2cnc(SC)s2)ccc2c(c1)S(=O)(=O)N(C)C2=O 81157,Cc1cc(Cl)cc(C)c1OCC(=O)N(CC(O)CNC(=O)CC1(O)CCOC1)C 81158,Cc1cc(NC(C2CN(C3CCN(C(=O)Cc4ccccc4)CC3)C2)=O)ccn1 81159,C=C(C)CC(C)C(=O)NCC(C)(CO)NC(=O)COc1ccc(Cl)c(Cl)c1 81160,C1(CNC(Cc2ccn(CC)n2)=O)CC(C)(C)CN1C(=O)Cc1ccnc(F)c1 81161,N1(C(c2c(C)nsc2)=O)CCC12CN(C(=O)C(O)C(C)(C)C)C2 81162,n1(CCOC)cc(C(=O)NCC2CC(F)(CNC(C3CCC(C)C3)=O)C2)cn1 81163,N1(c2cc(N3CCCC(c4n(C)ccn4)C3)ncn2)CC2C3CCC(CC3)C2C1 81164,C1(NC(C2(OCC)CCC2)=O)CN(C(c2cnc(C3CC3)nc2)=O)CC1C 81165,C(=O)(C1=CCC(C(F)(F)F)OC1)NC(CC)CNC(c1cnoc1C)=O 81166,C1(C(=O)NC2C3CN(C(=O)Cn4cc(Cl)cn4)CC23)CCC=CCCC1 81167,c1(C(=O)NC(C)(C)CN2CCCCC2=O)cnn2cc(F)cc(F)c12 81168,C1(NC(c2c(C(C)C)cccc2)=O)CN(C(C2(C)CC2(F)F)=O)CC1S(C)(=O)=O 81169,c1(C2C(C(N(C)CC3(O)CN(C(C(CC)F)=O)C3)=O)C2)ccc(Cl)cc1F 81170,C(CCCCC(=O)NC1(C)CCN(C(=O)C(C)Cc2cnn(C)c2)C1)OC 81171,N1(C(CS(CC)(=O)=O)=O)CCN(C(=O)CCn2cc[nH]c(=O)c2=O)CC(O)C1 81172,C12(C(N3CCC(SC)CC3)=O)CCN(C(=O)CCC=C(C)C)CCC1C2 81173,C1(NC(C(C)=CC)=O)CCCC12CN(C(c1ccc(CNC(C)=O)s1)=O)C2 81174,c1(C(=O)NC(CNC(CC(CCC)O)=O)C2CCC2)c(F)cc(F)c(O)c1F 81175,C1(NC(C(C)CF)=O)CN(C(c2cc[nH]n2)=O)C2(CCOCC2)C1 81176,c1(C(=O)NCC(C2CCOC2)NC(=O)COCCCF)c[nH]nc1C(F)F 81177,Cc1cccc(Cn2nc(-c3ccc(C(C)C)cc3)nc2-c2ccsc2CO)c1 81178,c1(C(=O)NC2C(CNC(=O)COC3CCCC3)CC2)cc(C2CCCCC2)no1 81179,O(NC(=O)C(CCOCC)NC(c1ccn2cncc2c1)=O)CCCC=C 81180,c1(C(=O)NC(CCCNC(C2(C)CCC(OC)CC2)=O)C)ccc(C#N)c(C)c1 81181,CCCCCCCCC(=O)N1CC2(CC(NC(c3cc(Br)cnc3C)=O)C2)C1 81182,C1(C(=O)NC2(C)CC(C(=O)NC3(C(COC)O)CC3)C2)CC(C)(C)CO1 81183,C=CCC(C(=O)NC(C)CCNC(=O)C=C(C)I)OC 81184,CC1(C)CC(CC(=O)NCCCCC(CO)NC(=O)CSc2nc[nH]n2)CCO1 81185,Nc1cc(C(=O)NCC2CN(C(c3cccs3)=O)CC2C(F)(F)F)ncc1Cl 81186,C=CC(C)(C)CC(=O)NCC1CN(C(=O)C(C)=C(C)CC)CCC1C 81187,C(=O)(C1=CCCC1(C)C)N1CCC(C(CNC(c2ccc(C#C)cn2)=O)F)CC1 81188,c1(C(=O)OC)ccccc1CC(C)(CO)n1cc(-c2cc[nH]c(=N)c2)nn1 81189,N1(C(C)C(=O)NC(C(=O)NCCc2cocn2)C2CCOC2)CCNC1=O 81190,N1(CC(CNC(=O)C(c2nc(N(C)C)sc2C)C)OC)CCc2ccccc21 81191,c1(C(=O)NCCC2(CNC(C3(C)CCC3)=O)CC2)cccc2sncc12 81192,C(=O)(CC(F)(F)C(C)C)NC1CC(CNC(c2c(C)noc2)=O)C1 81193,N1(C(CC2ON=C(CC)C2)=O)CCN(C(c2cnc(C(C)(C)C)o2)=O)C(CC)C1 81194,C1(C#N)(C(=O)NCC2CC(NC(C3(CN(C)C)CC3)=O)C2)CC12CCC2 81195,C1(NC(c2c(OC)n[nH]c2)=O)C2CN(C(=O)Cn3cc(C(=O)NC4CC4)nn3)CC12 81196,N(C(=NCC1CCC1)N1CCC(CN2CC2)C1)Cc1c(Br)c[nH]n1 81197,C(=O)(C1CCCn2nccc21)NCC1(OC)CN(C(C2CC=CCO2)=O)C1 81198,Cc1cc(CC(N2CCCCC2C2(C(N3CCCC3)=O)CC2)=O)c(Br)cc1F 81199,c1(C(N(c2ncc(SC)cn2)C2CCNCC2F)=O)cc([N+](=O)[O-])c(F)cc1F 81200,C#Cc1c[nH]nc1C(N1CC2CC2(NC(C2CCC(=O)N2)=O)C1)=O 81201,N1(C(c2c(C)n(C)nc2)=O)CC2CCCC2(NC(C2CC=CC(O)C2)=O)C1 81202,c1(C(N2CC(O)(C3CCCN3C(=O)C=CBr)C2)=O)cccc2ccoc12 81203,CC(CC(=O)NCCCCCNC(C1(O)COC1)=O)c1cccnc1 81204,C#CC1(O)CCCN(C(=O)C(C)(C)CNC(=O)CC2NC(=O)NC2=O)C1 81205,n1(C(C)C)cnnc1SCC(=O)NC(C)CC(C)NC(c1ccc(C(N)=O)o1)=O 81206,C1(NC(COCCOC)=O)CN(C(=O)CCN(C(=O)OC(C)(C)C)CC)CCC1F 81207,C1(OCC(N2CC(C(C(=O)NC(C3C=CCS3)CC)OC)C2)=O)CCCOC1 81208,N1(C(c2ccc(C#N)s2)=O)CC2(C1)SCCC2NC(C1CC2CCCC(C1)C2)=O 81209,C1(C(=O)Nc2nccnc2Cl)CC12CCN(C(c1ccc(CCO)cc1)=O)CC2 81210,N1(C(CCOCC)=O)CCCC2(CNC(=O)Cc3cc(F)ccc3F)CC12 81211,CC(C)C(C)(Cc1ccccc1)C(=O)N(C)CCN(C)C(c1ccc(=O)oc1)=O 81212,C(=O)(C(C)CCCC(C)=O)NC(CC#C)(C)C(=O)NCCC1(O)CCCCC1 81213,N1(CC(N2CC(F)(CNC(=O)Cc3cc(CO)on3)C2)=O)CCNC(=O)C1 81214,c1(CC)nc(=N)[nH]cc1C(=O)NC1CCC1NC(=O)CSCc1ccccc1Cl 81215,c1(COC)nc(NCCCNC(C2CCC2)=O)cc(=NC2CCC(=O)NC2)[nH]1 81216,N1(C(c2c(CNC(C3(CC)CCCC3O)=O)n[nH]c2)=O)CC(F)(F)C(F)(F)C1 81217,C1(CNC(c2scnc2C(F)F)=O)CCCCN(C(=O)CC2CCOCC2)C1 81218,C1(NC(C(C)C2CC2)=O)C2CCC1N(C(c1cccc(-c3nnco3)c1)=O)C2 81219,CC12CN(C(=O)C3=CCC3)CC1(C)CN(C(=O)CCOC(F)F)C2 81220,c1(C(N2CCCCC(NC(=O)CCc3ccc[nH]3)C2)=O)cc(I)ccc1[N+](=O)[O-] 81221,C(=O)(CS(=O)(=O)C1CC1)N1C(CNC(c2cccc3c2CCC3)=O)CCCC1 81222,Cc1nn(C)c(C(=O)O)c1S(=O)(=O)N1CCC2(CCC(O)CC2)C1 81223,C(CCF)(C(=O)N(C(C)COC)C)NC(COCCC=C)=O 81224,C12(C(=O)NCCOCCn3cc(C4(O)CCOC4)nn3)CCOCC1C2(F)F 81225,N1(C(C(C)CO)=O)CC2(C1)CN(C(c1c[nH]ccc1=O)=O)CC2CO 81226,N1(C(C2C(C)C2)=O)CCCC2(CCN(C(=O)C=CCN(CC(F)(F)F)C)CC2)C1 81227,C1(C(=O)OC)CCCC(C(=O)NCC=CCC(N2CCC(C(C)(C)SC)C2)=O)C1 81228,CCCC(CCO)N=c1[nH]c(=NCC2CC2C(=O)OCC)[nH]c2c1COCC2 81229,C1(NC(=O)Cc2ccsc2)CC(NC(c2cc(C3CCCC3)[nH]n2)=O)C12CCC2 81230,C(CC(=O)Nn1cnn(C)c1=S)Oc1ccc(C)cc1F 81231,C1(NC(CC2(C)CCN(C(=O)C(F)C3CCC3)C2)=O)C(O)C2CCOC12 81232,C1(C)(NC(c2c(CC)n(CC)nn2)=O)CCCN(C(=O)Cc2cncn2C)C1 81233,C1(C(=O)NCc2nnc(O)o2)CC2CCC(C1)N2C(=O)C(c1ccccc1)O 81234,c1(C(N2CC3ON=C(COCC)C3C2)=O)ccc2scc(C)c2c1.C1(C)C(=O)N1 81235,c1(C(=O)NC(CN(C(C=CC)=O)C)CC)cc(Br)c2[nH]nnc2c1 81236,N1(C(CC2CCC(C)CO2)=O)CCC2(CC(C(=O)NC(C3CCCC3)C)C2)C1 81237,c1(C(N2CC(NC(c3c(CC)scn3)=O)CC2(C)C)=O)cc(C)c(C)cc1N 81238,C1(N(c2nnc(C(F)F)s2)C)CCCN(C(=O)C(C)(C)CC2CCOCC2)C1 81239,N(C1CC(C)n2ncnc21)C(C=CCNC(c1cccc(C)c1O)=O)=O 81240,N(C1CC2(CCN(C(=O)CC#N)CC2)Oc2ccccc21)C(C(CCC)C)=O 81241,N1(C(=O)CC2CC2)CCCC1C1CCCN1C(C1CC1c1ccccc1)=O 81242,N1(C(C2CCCC(=O)O2)=O)CCCC2(CCCN2C(C23COC(CF)(C2)C3)=O)C1 81243,C(=O)(CC(C)C(C)(C)NC(c1nonc1N)=O)NC(C)Cn1cccn1 81244,N(C1CCSc2ccc(Cl)cc21)C(C(=O)NC1(CCC(=O)OC)CC1(F)F)=O 81245,Fc1cc(-c2ncc(CN3CCCC(CCN4CCCCC4)C3)s2)cc(Br)c1 81246,N1(C(CCOCCOC)=O)CCCN(C(c2cc(F)cc(Cl)c2N)=O)C(C)C1 81247,c1(C(N(CCNC(Cn2c(=O)ccc(C)c2)=O)C)=O)cc(F)c(Cl)cc1F 81248,C1(CNC(CN(CCC#C)C)=O)CN(C(C2CC(CCO)C2)=O)CCC12CCC2 81249,C1(CCC)(NC(C2CC(=O)N(C)C2)=O)CCN(C(c2cc(F)cc(F)c2)=O)CC1 81250,c1(OC)cc(C)c(Cl)cc1C(=O)NCC1CC(NC(=O)CN2CCC(C)C2)C1 81251,N1(C(c2cnc(C)[nH]c2=N)=O)CC2(CCN(C(=O)CSc3n[nH]c(C)n3)CC2)C1 81252,c1(NC2C(OC)CN(C)C2)nc(C)cc(=NCC2CC2c2ccc(C)cc2)[nH]1 81253,N1(C(c2nc(C(=O)OCC)sc2)=O)CCc2cc(OC(C)=O)ccc2C1C 81254,C1(C2CCC(=O)NC2)(C(=O)NC2C(NC(C(C)(C)C#N)=O)CCC2)CCC1 81255,c1(C(=O)NC2CN(C(c3c(C)cco3)=O)C(C)(C)C2)c[nH]c2ccccc2c1=N 81256,C(C(=O)N1CC(O)(CCc2cn(-c3cccnc3)nn2)C1)(C(C)C)SC 81257,c1(C2C(C(N3CC(CNC(c4c(CC)non4)=O)(OC)C3)=O)C2)ccccc1Cl 81258,c1(C(=O)NC2CN(C(c3c(CCC)nco3)=O)C2)ccncc1I 81259,[nH]1cc(C(C)(C)C)cn1.C1(NC=O)CCC(CCNC(C2(C3CC3)CCC2)=O)C1 81260,CCCCCC(C(=O)NC1CC2C(NC(C3CC(OC)C3)=O)C2C1)C(C)C 81261,S(=O)(=O)(c1ccc(C)nc1)N1CCC(C2C(c3[nH]nc(C(=O)OC)n3)C2)CC1 81262,N(C(=NCCCNc1ccccc1)NCCC1CCCC1)C1C(N(C)C)C1 81263,CCCCCCC(CC)(CC)C(=O)NCC(C(C)C)NC(C1CC12CCC2)=O 81264,C1(C(N2CCC(n3cc(-c4cscn4)nn3)C(O)C2)=O)COc2ccccc2C1 81265,Cc1oc(C(=O)NC2CC2NC(=O)CCc2ccc(C(C)C)cc2)cc1Br 81266,Nc1c(F)ccc(Cl)c1C(=O)NC(c1ccccc1)CNC(c1ccoc1)=O 81267,N1(C(C#CC(C)(C)C)=O)CCCC12CCN(C(C1(CCF)CC1)=O)CC2 81268,c1(N2CCC(C(=O)NC3CC(C(F)(F)F)C3)C2)ncc2scc(Br)c2n1 81269,N1(C(CC(C)C)=O)CCC(F)(CNC(C2(n3cnnn3)CCCCC2)=O)CC1 81270,CC1CC(C)CN(C(=O)CN2CCCCC2)C1.C(=O)(CCc1cn[nH]c1)NC(C)C 81271,c1(C(=O)OC)ccc(C(=O)NC2CN(C(=O)Cc3cc(C)no3)C2)cc1C 81272,c1(C(=O)NCC2C3CN(C(CSCC)=O)C2C3)ccc2nc(C)n(C)c(=O)c2c1 81273,Cc1c(Cl)cccc1S(=O)(=O)NC1C2CN(Cc3ccc(Br)[nH]3)CC12 81274,c1(NC(C(c2cnc(COC)s2)OC(F)F)=O)cc(Cl)ccc1OCCCF 81275,C1(NC(=O)C(c2ccc(F)cc2)CO)CN(C(c2coc(Cl)c2)=O)CC1C(F)F 81276,CC1(C)CCC(CNC(=O)CC2CCCNC2=O)N(C(=O)C=Cc2cnc[nH]2)C1 81277,c1(C(=O)NCC2CN(C(=O)C(F)Cc3ccccc3)CC2O)cc(O)ncc1F 81278,c1(CC)nnc2n1CC(Nc1cc(CC)ncn1)CC2 81279,N1(C(C(C)OCC=C)=O)CC(CO)C2(C1)CN(C(=O)CCCC1CCOCC1)C2 81280,C=CC(C)(C)CN=C(NC(CC)CC)NC1CC2(C1)CC(C(N)=O)C2 81281,C(C(C(C)C(C)C)NC(=O)C=CCCC=C(C)C)NC(C1(CCOC)CCC1)=O 81282,C#Cc1cccc(CNC2(c3nnnn3C(C)C)CN(C)CC2C)c1 81283,CCCC(C)(CC)C(=O)NCC1CN(C(c2cnn3c2N(C)CC3)=O)CCO1 81284,CC#CCCCC(=O)N1CC(NC(=NCC)NCc2noc3c2CCC3)C(C)C1 81285,C1(CNC(C(C)Cc2ccncc2)=O)CCCCN1C(=O)COC1CCCOC1 81286,O=C1CCC(C(F)C(=O)NC2CC(F)(CNC(=O)COC3CCCC3)C2)CC1 81287,N1(C(CNC(c2cccc(C)c2)=O)=O)CC2CC(NC(c3ccco3)=O)C1C2 81288,c1(C(=O)NCC2(C(=O)NC(C(=O)NC)C)CCCC2)cnc(S)nc1 81289,N1(C(COCC#C)=O)CCC2C(CCCN2C(C2Cc3nnc(C)n3C2)=O)C1 81290,C1(CNC(C(C)n2cncn2)=O)(CO)CCN(C(C2(C)C=CCCC2)=O)C1 81291,C1(NC(c2cc3ccccc3[nH]2)=O)CC2(CCCCN2C(=O)CCC2CC2)C1 81292,CCC(CNC(c1ccoc1)=O)(CC)NC(=O)CCCC1CCCC1 81293,N1(C(c2nc(CC)sc2N)=O)CCC(NC(C2C=CCS2)=O)C2(CCC2)C1 81294,c1(C(=O)NCC(CNC(C(N2CCOCC2)C)=O)C)n[nH]c2c1COCC2 81295,c1(C(=O)NCCC2OCCN(C(C(COC)(C)O)=O)C2)ccc2ncc(C)n2c1 81296,N1(C(C)=O)CCOC(C(=O)NC(C)CCNC(=O)COCc2ccc(C)cc2)C1 81297,c1(C(C)OC(=O)CC2CCCC2C(F)(F)F)cc(C(F)(F)F)ccc1F 81298,Cc1cc(F)c(C(=O)NC2(CNC(=O)C=C3CC3)CCCCC2C)cc1Br 81299,O=C1CCc2c(C(=O)NCCCCNC(c3cc4ccncc4s3)=O)cccc21 81300,C1(N(C)C(C2CC2C2(C)OCCO2)=O)CCN(C(=O)CSS(C)(=O)=O)CC1 81301,C1(C)(CCNC(Cn2c(C)ncc2)=O)CCN(C(=O)Cc2cocn2)C1 81302,CCC(C)CC(C(=O)N1CC2CC=CC1C2)NC(c1cn(C)nc1OC)=O 81303,c1(OC(C(=O)NS(CCCC)(=O)=O)C)cccc2ccccc12 81304,c1(N(C)C)ccc(C(N2CCC(C(C)(O)CNC(=O)CCC3CC3)CC2)=O)cn1 81305,C1(COC)CN(C(=O)CC2(O)CCCC2)CCN1C(=O)CC1CCC2CC2C1 81306,c1(C(N2C(CNC(C3C(C)CC(=O)CC3)=O)CC2)=O)cnc2cc(Br)ccc2c1 81307,n1(CCOCC)c(N2CC3CC3C2)nnc1COC(C)C.C1(CNC)CCC1 81308,C1(C(=O)N(C)CCc2cnc[nH]2)(NC(C(OC)OC)=O)CCC(C)(C)C1 81309,c1(OC)cscc1C(=O)NC(C)(CNC(=O)CSc1nc[nH]n1)CO 81310,c1(C(N(CC(C)(C)NC(c2c(OC)nsc2)=O)C)=O)c(C)ncc2ccccc12 81311,c1(-n2c(C3CC3Cl)nc(COC)n2)ccc(Br)c(F)c1 81312,C1(NC(=O)Cn2nnnc2C2CC2)CCC(NC(=O)C(F)C2CC2)CC1 81313,c1(OC)cc(C(=O)NCC2(OC)CN(C(=O)C(C)CC(N)=O)C2)ccc1C(F)F 81314,C1(CCNC(CCOC)=O)CC(F)(F)CN1C(=O)Cc1n[nH]c(=N)s1 81315,N1(C(C2(CN(C)C)CC2)=O)CCOC(CNC(C2(CC3CCC3)CC2)=O)C1 81316,C1(NC(C2(CC)CCC(O)CC2)=O)CCC2(CC1)CN(C(C1CCC(O)C1)=O)C2 81317,C1(C(=O)NC(CCCNC(C(C)NC(c2cccs2)=O)=O)C)CC1C1CCCC1 81318,CC1CCC(CC(=O)NC2CCN(C(c3ccc(C(N)=O)[nH]3)=O)C2C)OC1 81319,O=C(C1CCCc2ncnn21)NCC1CN(C(=O)COCC2CCC2)CCCO1 81320,N1(C(c2ccn(COC)n2)=O)CC(C)C(C)(CNC(c2cncc(SC)c2)=O)C1 81321,C(c1cncs1)=CC(=O)NC12CC(NC(c3cc(C4CCCCC4)[nH]n3)=O)(C1)C2 81322,C(=O)(C(=O)CCC(C)C)NC1(C(=O)NC2CN(CCC)C(=O)C2)CCC1 81323,C(=O)(C(F)C(C)(F)F)NC(c1occ(C(N2C(C)(C(=O)OC)C=CC2)=O)n1)C 81324,Cc1ccc(C(=O)N(C2CCCCN(C(c3cnc(S)nc3)=O)C2)C)cc1Cl 81325,C(=O)(C(F)(F)c1cnn(C)c1)NC(CN(C(CN(CCC#C)C)=O)C)CC 81326,c1(C(N2CCN(C(C(C)OCCOCC)=O)C(C)C2)=O)cc2c(cn1)COCC2 81327,C1(CNC(=O)C2=CCCC2)CN(C(c2c[nH]cc(Cl)c2=O)=O)CC(C(F)(F)F)O1 81328,c1(C(=O)NCCC2OCCN(C(C(CC)C)=O)C2)sc(Cl)c(Cl)c1OC 81329,C(C(CO)C(F)(F)F)Nc1cc(N(C)CC2CCS(=O)(=O)C2)ncn1 81330,C(=O)(C1=C(Cl)CCOC1)NC(C(C)C)CNC(=O)C(C)Sc1ccccn1 81331,CN=c1ccc(C(=O)NC(CO)C(C)NC(c2cccn2C(C)C)=O)c[nH]1 81332,C(=O)(C1=CCC(C)(C)CC1)NC1CCCC(CNC(C(C(CC)CC)C)=O)C1 81333,Cc1cc(NC(C2CCC(C3CC3)N2C(C2CC3(CCO2)CC3)=O)=O)cc(Cl)c1 81334,c1(NC(Cc2cnc(C)[nH]2)=O)ccc(Cn2cc(CC(=O)O)nn2)cc1 81335,c1(C(C(=O)OCC(c2c(C)nn(C(C)(C)C)c2)=O)C)cccc(Br)c1F 81336,C(=O)(C1CCc2nccn21)N1CC(O)(CNC(C(=C(C)C2CC2)F)=O)C1 81337,c1(OC)ccc(C(N2CCN(Cc3ccsc3)C(C)C2)=O)c(OC)c1 81338,c1(C2C3(CCC3)N2)nnnn1C1CCC1.C1(C(=O)NCC)(SC)CCC1 81339,Cc1c(C(=O)NCC2CN(C3CC3)C2)c(=O)oc2ccc(Br)cc12 81340,c1(NC(C2N(Cc3cn(CCC)nc3)CCCC2)=O)ccc2occc2c1 81341,C1(C#CC(=O)NC(Cc2cn[nH]c2)C(=O)NCCCOC(=O)NC)(CC)COC1 81342,N1(C(COCC#C)=O)CC(C(=O)NCCC2CCSC2)CCC1(C)C 81343,Cc1nc(C(N2CCC(O)(CNC(C3CCSCC3)=O)C2)=O)nn1C 81344,C1(NC(C(CC=C)(F)F)=O)CC2(CCN(C(=O)C=Cc3cccn3C)C2)C1 81345,C(CC(=O)N(C)CCN(C(=O)CC1CCCO1)C)SCC 81346,c1(C(=O)NCCC(=O)OC)ccc(NC(=O)C(C(C)C)NC=O)cc1 81347,N1(C(C=CC(=O)N(C)C)=O)CCN(C(C2CCN(S(C)(=O)=O)C2)=O)C(CO)C1 81348,N1(C(CN2C(=O)COCC2)=O)CCCC2CN(C(C3CC(OC4CC4)C3)=O)CC12 81349,c1(C2C(C(=O)NC3CCC(N(C(C(CC)C)=O)CC)CC3)C2)cc(C)cc(F)c1 81350,C1(C(C)C)COCCN(C(c2csc(C(F)(F)F)n2)C(=O)Nc2ccccc2)C1 81351,c1(OC)ccc(CCC(=O)NC(CCNC(C2(C)CCC(C)C2)=O)C(C)C)cn1 81352,C(=O)(C1=NOC(CNC(C2CCC(=O)N(C)C2)=O)C1)N1C(C(C)O)COCC1 81353,C(CCCC(=O)N(C1COCC1O)C1CC1)NC(C(C)C1CCC1)=O 81354,N1(C(C(C)c2cncs2)=O)CC(C2CN(C(=O)CCCCN(C)C)C2)C1 81355,Cc1cccn2cc(C(=O)NCC#CCNC(=O)CC3SC(=N)NC3=O)cc12 81356,N1(C(c2n(CC)cnn2)=O)CC2OCCN(C(=O)Cn3nc(O)ccc3=O)C2C1 81357,C1(CNC(c2c(C)cco2)=O)CC2(CCC2)CN1C(=O)C(C)OC(C)(C)C 81358,N1(c2nnc(C(C)(C)C)s2)CC2(C1)C(NC(c1nsnc1O)=O)CCS2(=O)=O 81359,CC1(C)CC(NC(c2cccnc2OC(F)F)=O)CN1C(c1cncc(O)c1)=O 81360,CCS(=O)CC(=O)NCc1ocnc1C(=O)N(C(C)CO)C 81361,N1(C(c2cnc(CC)o2)=O)CCC(C(N2CCCC(C#N)C2)=O)C12CCC2 81362,C1(N(C(=O)COC2CCCCC2)C)CC2CC1N(C(=O)CSc1nnnn1C)C2 81363,C1(C(=O)NC(CCC)CNC(C2(F)CCCC2)=O)CC2COCC(C1)C2 81364,c1(C(N2C(OCCCc3cn(CCCC)nn3)CCC2)=O)ccc(Cl)cc1Br 81365,N1(C(CN(C(C)C)C)=O)CC2CC(C)N(C(c3csc(C(F)(F)F)n3)=O)C2C1 81366,N1(C(C(C)(F)F)=O)CC2CCC(C1)C2C(=O)OCc1ccccc1 81367,N1(C(C2(CNC(C(CC=C)C)=O)CC(=C)C2)=O)CCN(C)C(C(C)C)C1 81368,C1(c2c(C(=O)OC)nco2)CCCN(N2CCCC2CC(F)(F)F)C1 81369,C1(CC)CCCC(c2nnnn2C2CCNC(=O)C2)(NC2CCCCCC2CO)C1 81370,Cc1nc(Cl)sc1C(C(=O)NC(C)C)N(C1CCCC1)Cc1cccs1 81371,Cc1ccc2nc(N3CCOCC3CNC(C3CN(C4CCOC4)C3)=O)sc2n1 81372,c1(NCC(C)(C(C)C)NC(C(C2CCOC2)OCC)=O)cc(=O)n(CC)c(O)n1 81373,N1(C(c2ncn(CC)c2)=O)CC(NC(c2ccsn2)=O)CC1C 81374,N1(CC(=O)N(CC(=O)OC)C(=O)Cc2cncc(C)n2)CCSc2ccccc21 81375,c1(C(=O)NC2CN(c3cc(C)ncn3)CC(C)C2)cccn2ccnc12 81376,C1(CNC(C(C)=CC=C)=O)CCCCC1C(=O)NCc1ncc(Cl)cn1 81377,C1(CNC(CC2CCC(C)O2)=O)CN(CCn2cccn2)CCCO1 81378,N1(C(C(C2CC2)OC)C(=O)NCCCF)CCOCC(C)(F)C1 81379,Cc1cccc2[nH]cc(CC(N3CC(NC(=O)CC4CC5CC5C4)C(C)C3)=O)c12 81380,Cc1c(C(=O)Nc2occ3c2CCC3)cccc1Cl.c12cn(nn1)C1CN(C1)C2 81381,C(C(=O)NCc1ccccc1)(C1=CCCCC1)N1CCCC(c2n(C)cnc2)C1 81382,N1(C(C2(CC)CCOCC2)=O)CCC(N(C(=O)C(=CC2CCCC2)C)C)C(C)C1 81383,C1(N(CC#C)C(c2ccoc2CNC(c2ccc(F)s2)=O)=O)CCC(=O)NC1 81384,Cc1c(C(=O)NCCC2CCCN(C(c3ccc(F)cn3)=O)C2)cc(O)cc1N 81385,Cc1ccc(CCNC(=O)C(=O)NCC2CCC3(CC3)CO2)cc1C 81386,C1OC2CCC1CC2.N1(C(C=C(C)C)=O)CC2(CCN2Nc2cc(Cl)ccn2)C1 81387,N1(C(c2cc(CCC)[nH]n2)=O)CC(NC(=O)C(F)=C(C)C)CC12CCCCCC2 81388,C1(C(=O)NC2C(CNC(CNC(=O)OCC=C)=O)C2)(CC)CCCNS1(=O)=O 81389,c1(C(=O)NC(CC)CN(C(=O)CC2CC3(CC3)CO2)C)cc2ncccc2[nH]1 81390,c1(C(N(C2CCN(C(c3cccc(C(N)=O)c3)=O)C2)CC)=O)cc(C#N)[nH]c1C 81391,C1(C2(NC(CCCSC(C)(C)C)=O)CC2)CCCCN1C(n1cnccc1=O)=O 81392,N1(C(C(C)OCC#C)=O)CCc2sccc2C1CNC(=O)C(C)(C)NC(C)=O 81393,c1(C(N2C(CN(C(C(C)CC3CCC3)=O)C)CCCC2)=O)ccnc(F)c1N 81394,c1(C(=O)NCC2CCCCC2)ccc(S(=O)(=O)NC2CCS(=O)(=O)C2)cc1 81395,N1(C(c2c(C)cco2)=O)CC2CCN(C(=O)Cc3ccc4c(c3)CCO4)CC2C1 81396,CCCC(C(O)C(=O)NCC1CC2CCC(C1)C2)NC(c1conc1C)=O 81397,C(=O)(C1=C(C)OCCS1)N1CCC(NC(C(CC)OC)=O)(CO)C1 81398,N1(C(c2[nH]c(=NCC)sc2)=O)CCC(C2CN(C(C3CCC=CCC3)=O)C2)CC1 81399,c1(C(N2CCC(C(F)F)(CNC(C(CC)CC)=O)C2)=O)cccc2nccn12 81400,c1(C(=O)NCC2(NC(c3n(C)c(=O)ccc3)=O)CCOC2)cnc2[nH]nnc2c1 81401,O=C(C#CC1CCOC1)NC1C2CC(NC(=O)CC3C=CCCC3)CC12 81402,C1(NC(C=C(CC)C)=O)CCCN(C(C2CCN(c3ccncc3)C2)=O)C1 81403,N1(C(c2cnn[nH]2)=O)CCC2(CCCN2c2ncnc3cc(C(=O)O)nn23)CC1 81404,C=C(C)CCC(C(=O)Nc1ccccc1C)N1CCCC(CF)C1 81405,C1(CCNC(C2N(C(CC=C)=O)CCC2)=O)CC2CCC1O2 81406,C1(C(=O)NCC(O)CCNC(c2ccc(O)nc2C)=O)(OCC)CCC12CCC2 81407,CC1C(C(N2CCCCC2)=O)CCN1C(c1ccc(O)cc1)=O 81408,C1(C#CC(=O)NC2CN(C(=O)CCC(C)N(C)C)CC2(C)C)(CC)CC1 81409,c1(C(=O)NC2(COC)CCN(C(CNC(=O)NC)=O)C2)cc(OC)ccc1C 81410,c1(CN(C(C(C)C)CO)CC(=O)Nc2ncsc2Br)ccc(Cl)c(Cl)c1 81411,N1(C(C(C)CN(C)C)=O)CCOCC(C)(CNC(=O)C=Cc2ccccc2F)C1 81412,C1(C#N)(C(N2CC(N(C)C)C(C)(C)C2)=O)CC2CCC1CC2=O 81413,N1(C(c2c(C)ccnn2)=O)C2CC=C(C(=O)NC3(CF)CCCC3)C1CC2 81414,N1(C(CC2N(CC)CCOC2)=O)C2CCC1(CNC(=O)C(C)=C(C)C)CC2 81415,CCCC(C)CC(=O)NC1CC(F)(CNC(C2CCCCN2C(C)=O)=O)C1 81416,C(=O)(C1=C(C)CC1)N(CC(=O)NCCC1(COC)CC1)C 81417,C(CCCC(=O)NCC1CC1CC(=O)NCCCCCCF)(OC)OC 81418,C1(CNC(C(CC)N(C)C)=O)CN(C(c2cc(-c3ccco3)c[nH]2)=O)C(C)(C)C1 81419,c1(C2C(C)C2)cn(CCOCCC(=O)N(C)C(C)C)nn1.C12(CC1)C(=O)NC2 81420,C1(C(=O)NC(c2cccnc2)C(=O)NCC(C)(C)C2CCC2)CN2CCN1CC2 81421,N1(C(CCC=C=C)=O)CCOCC(F)(CNC(=O)CN(C)Cc2ccccc2)C1 81422,C1(C(=O)NC2C(n3cc(CCC(C)O)nn3)COC2)CCCC(C)CC1 81423,C1(CCOC)(NC(c2n(CCC)ccc2)=O)CCN(C(c2ccsc2Cl)=O)CC1 81424,N#Cc1ccc(C(=O)NCC2CN(C(c3cnc(Cl)cc3Cl)=O)CCO2)c(O)c1 81425,CC1(C)CCCC1C(=O)NC1CCC1CNC(c1cccs1)=O 81426,N1(C(CCC2CCCN(C(=O)C#CC3CCOC3)C2)=O)CCc2cncnc2C1 81427,C1(CNC(C(CC)N(C)C)=O)CCCCN1C(=O)CCc1cccc(O)c1 81428,N1(C(C2N(C(CNC(CN(C)C)=O)=O)CC=C2)=O)CCC2(CCC2)C(O)C1 81429,C#CCC(C(=O)NCc1cc(C(=O)NC(CC)(CC)CC)ccn1)C1CC1 81430,C#CCC(CO)NC(=O)C(CO)NC(=O)C(C)OC(C)=O 81431,C#CC1(C(=O)NC(CCN(C(=O)Cc2ncc(Cl)s2)C)C(C)C)CCCC1 81432,Cc1ccc(CCCNC(c2[nH]cnc2C)c2nnnn2CC2CC2)cc1 81433,C#Cc1ccc(C(N2CCN(C(=O)C(n3nccc3C)C)C(CO)C2)=O)c(C)c1 81434,Cc1ccc(CNc2cccc(CN3C(=O)CN(CC4COC4)C3=O)c2)c(C)c1 81435,c1(C(O)CNCCn2ccc(C(F)F)n2)ccc(Br)c(Cl)n1 81436,N1(C(C2CN(C(C)=O)C2)=O)C2CCC(C(=O)Nc3ccc(N(C)C)nc3)C1CC2 81437,N1(C(CCCCC#C)=O)CC(O)(C2CCCN2C(=O)Cc2cc[nH]c2)C1 81438,C(C)(C)(CC(=O)N1CCCC1C1(C(=O)N(C)Cc2nnc(C)s2)CC1)OC 81439,C1(O)(CNC(C2N(C)CC(O)C2)=O)CCN(C(=O)C#CC2(C)CC2)CC1 81440,Cc1sc(C)c(C(=O)NCCN(C(C2CCCOC2C)=O)CC2CC2)c1C#N 81441,c1(C(=O)NC(CN(C(CC(C=C)c2ccccc2)=O)C)C)nc(Cl)c(=O)[nH]c1N 81442,CC1(C)CCC1CC(=O)NC1COCC1n1cc(C(O)C2CC2)nn1 81443,n1(CCCN(C2CC=CCC2)C)cc(C(=O)NC(C2CCCCC2)=O)cn1 81444,C(N=c1cc[nH]cc1[N+](=O)[O-])c1nc(CNC(C2CC(OCC)C2)=O)nc(O)c1 81445,C1(COC(=O)NCCC(=O)OC)CCCCN1C(c1cc(C)c(C(F)(F)F)s1)=O 81446,c1(C(N2CCC(F)(Cc3ccccc3)C2)=O)cccc(N2CCCS2(=O)=O)c1 81447,C(CCO)(C(F)(F)F)NC(CC1CCCC(NC(c2nn(CC)c(O)c2)=O)C1)=O 81448,Cc1c(F)ccc(NC(C23CC2CCN3C(C2CC(=O)NC2(C)C)=O)=O)c1F 81449,C(=O)(C(CO)C(C)(C)C)NC12CC(C(N3CC(C)(C(C)C)OCC3)=O)(C1)C2 81450,C1(C(=O)NCCCC2CCCCN2C(c2cscc2CC)=O)CCCCC12CC2 81451,CC1(NC(C23CC(C(=O)Nc4cncc(CO)c4)(C2)C3)=O)CC=CCC1 81452,C1(CNC(CC(=C)Br)=O)(NC(=O)COCCOC)CCCCC1C 81453,c1(C(=O)NC2CCC(C)(CNC(C(C)(C)SC)=O)C2)cc2c(cn1)OCCC2 81454,C(C1C(C(=O)NCCCC2CCN(C(=O)CN3CC=CC3)CC2)C1(C)C)=C(C)C 81455,CN1CCN(C(=O)CN2CC3CCC2C3)CC1CNC(C1CCC(F)C1)=O 81456,N1(C(C(C)SCC)=O)CCCCC1CCNC(=O)CNC(c1ccccc1Cl)=O 81457,C1(C(N(CCCNC(c2csc(Cl)n2)=O)C)=O)CN2CCCC1CC2 81458,C1(CCC(=O)NCCc2cnccn2)CCCN1C(c1cc(CO)on1)=O 81459,c1(C(N2CC(n3cc(C(CC(C)C)O)nn3)C2)=O)cccc(I)c1 81460,n1(CC)cc([N+](=O)[O-])c(C(=O)NC2CC(NC(C3CCN(C)C3=O)=O)C(O)C2)n1 81461,c1(CC(C)NC(c2coc(C(=O)O)c2)=O)cn(CCCCOC(C)(C)C)nn1 81462,N1(C(C(CSC)OC)=O)CC(C2(NC(=O)CN3CCN(C)CC3)CC2)C1 81463,N1(C(CNC(CN(C2CC2)CC)=O)C)CCN(C(C2(F)CCOC2C)=O)CC1 81464,N1(C(C2(CC=C)CCN(C(c3cnnn3CC)=O)C2)=O)CCN2CCC1C2 81465,N1(C(C(=O)NC)C2CCN2C(=O)OC(C)(C)C)CC(C)(C)c2cc(Cl)ccc21 81466,C(C(C)(CO)CO)N(C1CCN(C(=O)CC2CCOC2)CC1)C 81467,N1(C(c2c(C)ncc(N)c2)=O)CCN(C(c2ccsc2Br)=O)C(C)C1C 81468,CCS(=O)(=O)CC(=O)NC1CCN(C(c2cccc(C)c2O)=O)C12CC2 81469,Cc1cccc(C(N2CC(OCCC(N3CCSCC3CO)=O)C2)=O)c1C#N 81470,N1(C(C(CC=C)(F)F)=O)CCC2(CCC2NC(C2CC(CN(C)C)C2)=O)CC1 81471,Cc1nn(C)c2c(NCCCc3cnn(C)c3)nc(=NCC3CCCC3O)[nH]c12 81472,c12cccc(n1)S2.C1(N(C(C2CCC(C(N)=O)C2)=O)CC)CC2CC1CN2 81473,C1(CC)(NC(c2nccn2C)=O)CCN(C(C2(c3ccccc3)CC2(C)C)=O)CC1 81474,N1(C(C2C(C)OCCN2C(=O)CCN=[N+]=[N-])=O)CCC2(CCCCC2)C1 81475,c1(OC)c(CC(N2CC3(NC(=O)Cc4nc[nH]n4)CCC2C3)=O)cccc1Cl 81476,c1(C(=O)NCC(CNC(c2ncsc2Br)=O)OC)ccc2c[nH]nc2c1 81477,CCC(CC1CCCC1)C(=O)NC(C)CN(C)C(c1c[nH]nc1-c1ccsc1)=O 81478,CC(C)CCC(=O)C(=O)NCc1ccc(C(=O)NCC2CCCCN2C)o1 81479,c1(C(N2CCOC(C)(CCOC)C2)C(=O)NC(CC)(C)C)ccc(O)cc1OC 81480,c1(C(N2C(C)CC(NC(CSCC(=O)OC)=O)C2)=O)ccc(OC)c2ccsc12 81481,C(=O)(CCS(C)(=N)=O)N(C(C)CNC(c1csnn1)=O)C 81482,C1(C(=O)NCC2(NC(CC3CCN(C)C3)=O)CC2)CN=C2N=CNN2C1 81483,CCC(F)(F)C(C)(C)C(=O)NC1CC(CCNC(c2cn(C3CC3)nn2)=O)C1 81484,C(=O)(CC1CCc2ccc(O)cc21)NC1CC(NC(c2c(OC)nccc2)=O)C1 81485,c1(C(N(CC(C)NC(=O)C(O)C2CC2)C)=O)sc2cc(F)ccc2c1Cl 81486,CC(C)CC(CNC(=O)CCCOc1ccc(Cl)cc1)NC(C1CC1C(F)F)=O 81487,CCC(C(=O)NCC(C)(C)COC)N(C)C(c1sccc1CO)=O 81488,c1(OC)ccc(-n2cc(C(C)NC(C3CCCC3CF)=O)nn2)cc1OC 81489,c1(C(=O)NCC(O)CNC(C2(C(O)C(F)(F)F)CC2)=O)cccc(C=C(F)F)c1 81490,C1(CC)CC(C)CN(C(C(=O)NCc2nnn(C)n2)C2COC2)C1 81491,CCC(CC)(CCC(=O)NCC(O)CNC(=O)Cn1cncc1C)[N+](=O)[O-] 81492,Cc1ccc(C(CNC(c2cnc(C3CC3)[nH]2)=O)NC(=O)CNS(N)(=O)=O)cc1 81493,C1(C)(C(=O)NC2CC(CCC(=O)NCCCOC(C)C)C2)CCC(=O)N1 81494,N1(C(C(CN(C)C)NC(COCCCCC)=O)=O)CC(C)C(C)C1C 81495,C1(C(=O)NCC(C)N(CC)CC)CC2CCC(C1)N2C(c1ncccn1)=O 81496,c1(C(N2CCN(C(C(C)S(C)(=O)=O)=O)C(C3CC3)C2)=O)cnc(=NCCF)[nH]c1 81497,C12(CNC(C3CCCC3)=O)CN(C(c3cc4cccnc4s3)=O)CC1CCO2 81498,c1(C(=O)NC2CN(C(Cc3n(C)ncc3Cl)=O)C2)ccc2c(c1)CCC(=O)N2 81499,Cn1c(=O)n(C)c2c(CNS(=O)(=O)c3ccccc3C(C)(C)C)cccc12 81500,N(C1CCCc2n[nH]cc21)C(C1N(C(CC=CCCCCC)=O)CCC(C)C1)=O 81501,c1(C(=O)NC(CSCC)C(=O)N2CC(C)(C(F)(F)F)C2)ccc(C)nn1 81502,N1(C(C=C(C)C(C)(C)C)=O)CCN(C)C(C(=O)NCc2nn(C)cc2C)C1 81503,C(=O)(CCCC(C)(C)C#N)N1CCC(CNC(CC2CC(CC)C2)=O)C1 81504,C12(C(=O)NC(CCC)c3nn[nH]n3)CC(CO)(CN1C(=O)CCn1ccnc1C)C2 81505,CCS(=O)CC(=O)NCC1C=CCN1C(=O)CCC(=O)OC(C)(C)C 81506,CC(C)CC(C)(C)C(=O)N(C(CNC(c1cnc(O)n1C)=O)C1CC1)C 81507,C1(NC(CN2CCC(OC)C2)=O)CCN(C(=O)CCCC2CCCC2)CC1C 81508,C#Cc1ccc(CC(=O)NCC(C)C(F)C(=O)Nc2cccc(CCF)c2)cc1 81509,C1(C(=O)NC2CC3(CC(NC(C(CCC)CC)=O)C3)C2)CCc2ncc(C)n2C1 81510,Cc1nn(C)c(C(=O)NC(CNC(c2cnccc2C(C)(C)C)=O)C2CC2)c1Cl 81511,N(C1CC2(CN(C(=O)CC(C)(C)CN(C)C)C2)n2ccnc21)C(CSCC#C)=O 81512,n1(CC)ncc(CNC(C2C3CN(C(=O)CCCOC)CC23)=O)c1C 81513,N1(C(C(CCC)C)=O)CCN(C(=O)CCSc2nccn2C)CC(O)C1 81514,c1(CC)cc(I)c(Cl)cc1NC(=O)CN1CCN(C(=O)CSc2nc[nH]n2)CC1 81515,CC1CC(C)CN(Cc2c[nH]nc2O)C1.c12ccc(cc1)CNC2=O 81516,c1(CC(=O)NCC2(O)CCN(C(C(C)NC(=O)NC)=O)C2)ccc(S(C)=O)cc1 81517,C(C(O)CCNC(c1cnc(C2CCCO2)s1)=O)NC(CSC)=O 81518,C1(C2CCN(C(=O)CCSC(F)(F)F)CC2)(NC(c2cc(C)n(C)n2)=O)CC1 81519,N1(C(C2C(C)OCC2)=O)CC2(CC2)CC1CNC(c1ccc(C(C)(C)C)cn1)=O 81520,Cn1cc(S(N)(=O)=O)cc1C(=O)NC1CCCC1NC(C1CCCN1C1CC1)=O 81521,CC1CCN(CC(N2CCC(O)C2C(=O)NCC2CC23CC3(F)F)=O)CC1 81522,CC1CN(C(=O)Cc2csc(Br)c2)CCN1C(=O)C(F)C1CCC1 81523,C(C(=O)NCCC(CCNC(C)=O)C)(C(C)C)CCNC(=O)C=C(Cl)Cl 81524,C(C)(c1ccccc1OC(F)F)=CC(=O)NCCC1CC(NC(COC)=O)C1 81525,N1(C(CN(C(c2ccc(C#C)nc2)=O)C2CC2)=O)CC2(CCCN2C)C1 81526,CC1(C)CN(C(=O)Cc2cc(Cl)ccc2Cl)CC1NC(C1(O)CCOCC1)=O 81527,N1(C(CNC=O)=O)CCSCC1C(=O)NCc1cncs1 81528,CC1CN(C(C2CCCCC2)=O)CC2(CCN(C(c3cc(F)cc(F)c3)=O)C2)O1 81529,C(=O)(C1=CS(=O)CCC1)N(CCCCCNC(C1C(OCC)C1)=O)C 81530,c1(NC(CC(CC)NC(=O)CS(=O)(=O)CCOC)=O)cc(C)cc(C)c1C 81531,CC1(C)Cc2cc(C(=O)NCC3CCCC3NC(=O)CSC(=N)N)ccc2O1 81532,C12(NC(CCOCC)=O)COCCC1CN(C(=O)CNC(=O)CC)C2 81533,C1(NC(c2n(CCOC)nnn2)C2CC=CC2)CC2(C1)CC1CCC2C1 81534,C(C(=O)NNC(=O)Cc1ccccn1)SCc1nnc(C(N)=O)o1 81535,CCC1=NOC(C(=O)N(CCCNC(c2snc(Cl)c2Cl)=O)C(C)C)C1 81536,N1(CC)CCC(N(C(=O)C(=O)Nc2cc(C(F)(F)F)c(Cl)cn2)C)CC1C 81537,C1(CNC(CCn2c(C)cc(C)n2)=O)CCCCCN1C(C1CC2CCC2C1)=O 81538,C(C(C)(O)C(=O)NCC1CN(C(c2c(C)noc2C2CC2)=O)CCO1)OC 81539,c1(C(=O)NCC(CNC(CCCOC)=O)(C)F)nccnc1C(N)=O 81540,N1(CC(C2C(C)OC(C)C2)=O)CCOc2c(Cl)cc(Br)cc2C1 81541,CCCCCCCC(=O)N(CCN(C(=O)CCC(F)F)CC)CC 81542,N1(C(C(C(CCC)NC(=O)CCCC(C)=O)O)=O)Cc2ccc(O)cc2C1 81543,CC1Cc2ccccc2C1NC(=O)N(C1CC(c2ccccc2)C1)C 81544,c1(C(C)=O)cc(C(=O)N(CCC(C(C)C)NC(c2cnn(C)n2)=O)C)oc1C 81545,c1(C(N2C(C)(CNC(=O)C=CCF)CCC2)=O)cc2n(n1)CCCC2=O 81546,c1(NCC)cccnc1C(=O)NCC1CN(C(C2CC3C=CC2C3)=O)CC1C 81547,N1(C(Cc2nnc(C)o2)=O)CC(CNC(=O)CCC2CC2(C)C)C(C)C1 81548,CC1CN2CCN1C(C(=O)NC(C)CN(C(=O)COc1cccc(F)n1)C)C2 81549,N1(C(C(C)C)=O)CCN(C(c2cc(N3CCOCC3)nc(Cl)c2)=O)C(C(F)F)C1 81550,C1(NC(CCNC(=O)NC)=O)CCCCN(C(=O)CCCC(=O)OC)C1 81551,Cc1sc(O)nc1C(N1CC(CC(=O)NC(c2cn(C)nn2)C)CC1C)=O 81552,c1(OCCNc2nccc(C(=O)NC)c2)ccc2c(C)cc(=O)oc2c1 81553,C1(NC(=O)C2CC2)CC(O)CN(C(c2ccc(N3CCCS3(=O)=O)cc2)=O)C1 81554,O=C(C1=C(Cl)CCC1)NC(CNC(=O)CN1CCN(c2nccs2)CC1)C1CC1 81555,N1(C(C(C=C)CC)=O)CCC(C)C(CC(=O)NC2(C)CCCC2)C1 81556,C1(C(=O)NCCN(C(C2(CC(F)F)CCOCC2)=O)CC)CCC(C(N)=O)N1C 81557,c1(C(N2C(CNC(c3cc(C)cc(O)n3)=O)C(C)CC2)=O)ccn2ccnc2c1 81558,c1(C(N2CC(O)(CNC(C(CC)OC)=O)C2)=O)cc2n(n1)CCCC2=O 81559,c1(C(N2CC(C)(NC(=O)CCC3CCCC(=O)N3)C2)=O)cnc2nccnc2c1 81560,N1(C(CCC)C(=O)NCC2CCOCC2)CC(=O)N2CCCCC2C1 81561,c1(C(=O)NC2C(CNC(C3CC(=C)C3)=O)C2)cc(O)nc2ccc([N+](=O)[O-])cc12 81562,C1(C(=O)Nc2c(C)csc2)CC=CC(NC(c2cnc(=N)[nH]c2)=O)C1 81563,Cc1nc2c(N3CC4CN(C(c5cc6ccoc6s5)=O)C4C3)ncnc2[nH]1 81564,C1(CC(=O)NCCN2CCN(C(C3(n4nccn4)CC3)=O)CC2)CC(O)C12CCC2 81565,N1(C(CN(C)C)=O)CCCC2(CCCCC2NC(=O)CCNC(=O)C=CCl)C1 81566,C1(C(=O)Nc2cn(C)c(=O)n(C)c2=O)Cc2cc(S(N)(=O)=O)ccc2O1 81567,Cc1cc(C)n(CCC(=O)NCC2C=CCN2C(=O)Cc2c[nH]nc2C)n1 81568,C1(CC#C)(C(=O)N(CC(C)(C)NC(=O)Cn2cc(Br)cn2)C)CCOC1 81569,S(=O)(=O)(c1cc2c(cc1Cl)N(C(C1(CSC)CCC1)=O)CC2)NC(C)=O 81570,Cc1cc(C(N2C(CNC(C3CS(=O)C3)=O)CC3CC23)=O)nnc1O 81571,C#CCCCC(C)C(=O)N1CCCN(C(c2cc(C)cc(F)c2)=O)CC1 81572,N1(C(C=COCC)=O)CCN(C2CCN(C(c3ccnnc3O)=O)C2)CC1 81573,Cc1nnsc1C(=O)NN1CCCC1.c12cnc([nH]1)CCC1(CC1)CNC2=O 81574,c1(OC)cc(C(N2CC3(NC(=O)COc4ccccc4)CCC2C3)=O)cnc1O 81575,C(=O)(C(O)CCCNC(C1SCC=C1C)=O)N1CC(C(=O)NCC)C1 81576,N1(CC(=O)N(C2(C#C)CC2)C)CCN(C(c2ccc(Cl)o2)=O)CC1 81577,N1(C(Cn2c(=N)nc[nH]2)=O)CC(O)CC1C(=O)NCCc1ncc[nH]1 81578,N1(C(C(C=C)O)=O)CCCN(C(c2ccc(-n3cnnn3)cc2)=O)CC1CC1CC1 81579,N1(C(c2cnn(CC)n2)=O)CC(NC(=O)CCc2cccnc2)CC12CCOC2 81580,Cc1ccc(Br)c(C(N2CCCC2C(C)NC(C2CC3CC3C2)=O)=O)c1 81581,CCC1=C(C(=O)NCCCC2CCN(C(=O)C(C)CC(C)C)CC2)SCCO1 81582,CC1(C)CC(NC(=O)C(O)C(F)(F)F)CN(C(C2C3COCC23)=O)C1 81583,C(C(C)(C)C(F)(F)F)NC(C(C)(C)CNC(=O)C(C1(O)CCCC1)F)=O 81584,C1(CC=C)(NC(C2CC2CC)=O)CCN(C(=O)CCCC2CC2)C1 81585,C1(N(C(C2C(C(C)C)(CC)C2)=O)C)CCC(NC(C2(CC(C)C)CCC2)=O)CC1 81586,CC(C)CC(C(=O)NCCCCNC(N)=O)NC(c1cccn1C)=O 81587,CC(CCC(=O)NC1CC(=O)N(C2CN(C)C2)C1)CC(=O)O 81588,c1(C(=O)NC2CCCC23CN(C(c2ccnnc2)=O)C3)ccc2cnccc2n1 81589,Cc1nc(Cl)ccc1S(=O)(=O)N1CC(NC(=O)CNC(N)=O)C(F)(F)C1 81590,N1(C(C2CC2F)=O)CCC(C2CCCCN2C(C23CCC(C2)C3)=O)CC1 81591,C1(NC(C(C2CCC2)OCC)=O)CCOC(C(=O)NC(CC2CCC2)CO)C1 81592,C1(N(C(C(CSC)O)=O)CC(C)C)CCN(C(C2CCC2(F)F)=O)CC1 81593,CS(=N)(=O)C1CN(C(C2COCCN(C(=O)CC3CCCSC3)C2)=O)C1 81594,Cn1ncc2c1CC(C(N1CC(NC(c3cc(C#N)no3)=O)C(C)(C)C1)=O)CC2 81595,CC(c1ccccc1C)=CC(N1CCN(C(=O)CN2C(C)CCC2C)CC1C)=O 81596,N1(C(C(CC)CC)=O)CCC(C(N2CCOCC2CO)=O)C(C)(C)C1 81597,N1(C(C(CCCC)C)=O)CC(C2CN(C(=O)CCC3CCCC(O)C3)C2)C1 81598,C1(COC)(NC(=O)C(C)(C)C2CCCN2C(c2cc(C(N)=O)c[nH]2)=O)CCOC1 81599,C1(CC)CCN(CC2(C(=O)NC)CCCN2C(=O)CN(C)CCOCC)CC1(C)C 81600,c1(C(N2CCC3C(NC(C(C4CCC4)OC)=O)C32)=O)cc(O)ccc1C 81601,c1(C(=O)NC2C(NC(c3cnn(CCC)c3C)=O)C2)cn2c(n1)CCC(C)C2 81602,C(=O)(C(C(C)(C)C)N(C)C)NC1C(CNC(C2(CC=C)CCC2)=O)C1 81603,n1(CCOC)cc(C(=O)NC(C)C(C)(C)NC(=O)CCc2cc[nH]n2)c(C)n1 81604,C=C(C)CC(C(=O)NCC1(C)CCCO1)NC(=O)CC12CCCC1C2 81605,c1(C(=O)NC(C(C(=O)N(CC#CC)C)C)C)cncc(F)c1C 81606,CC(C)(C)C(CO)C(=O)N1CCCCC(NC(C23CC(C(F)F)(CO2)C3)=O)C1 81607,O=C(O)CCC(Cc1ccccc1)NC(c1nc2c(s1)CCC2)=O 81608,C(C)(CC(=O)NC1(C)CC(NC(=O)C(C)(F)c2ccon2)C1)SC 81609,c1(N2CCC(O)(C(C)NC(=O)CCn3cncn3)C2)ncnc2[nH]ccc12 81610,C1(NC(c2n(CC)nc(C)c2)=O)CCCCCCC1NC(=O)CCNC(=O)CO 81611,N1(C(c2ccc(OC)c(I)c2)=O)CCN(C(c2cc[nH]n2)=O)CC(O)C1 81612,N1(C(C(CCOCCO)NC(Cc2cc(C)no2)=O)=O)CCNC(=O)C1C 81613,Cc1ncc(C(=O)NCC2(C(=O)NCC3CCC(C)CO3)CCC2)n1C 81614,C(=O)(NNc1ccc([N+](=O)[O-])cc1C)c1ccc(Cn2cc(CSC)nn2)o1 81615,Cc1nc2ccccc2nc1C(=O)NCC1CCN1C(C1CCCCO1)=O 81616,c1(C(=O)NCC=C2CCN(C(C3(C=C)CCC3)=O)CC2)ccc(F)c2c1OCC2 81617,C#Cc1ccc(C(N2CCCC2C(C)NC(C2(C(C)C)CC2)=O)=O)c(C)c1 81618,c1(C(=O)NCC(CNC(C(C(C)(C)C)SC)=O)C)cc2c(cc1N)CCC2 81619,N1(c2cc(C(C)=O)ncn2)CC(C2CCCN(C(C3CSCCS3)=O)C2)C1 81620,CC12CN(C(=O)Cc3ccoc3)CC1CN(C(=O)Cc1cccc3ccoc13)C2 81621,C(C)(C)(CCC(=O)NC(Cc1cc[nH]n1)C(=O)Nc1cc(CO)ccc1C)OC 81622,C1(CNC(Cn2ncc(CC)c2)=O)CN(C(c2cc(Cl)cnn2)=O)CCC1C 81623,C1(N(C)C(C2(F)CC=CCC2)=O)CCCN(C(c2coc(C(F)F)c2)=O)CC1 81624,N1(C(CC(CC)C)=O)CC2CCN(C(=O)CCc3cccc(C)n3)CC2C1 81625,C1(CNC(c2cnc(O)nc2O)=O)CC(N=c2[nH]ncs2)C1 81626,Cc1coc(C2CC2)c1C(N1CCC(CNC(c2nc(O)c(C)s2)=O)CC1)=O 81627,c1(OC)ccc(C(=O)NCCNC(C2CN(C3CCOC3)C2)=O)cc1S(C)(=O)=O 81628,C(CC(C)C)(C(=O)N1CC(C)(NC(C2(n3cncn3)CC2)=O)C1)NC(=O)OC 81629,N1(C(C2C=CC(NC(C3CN(C)C(=O)CC3)=O)C2)=O)Cc2cccc(C#N)c2C1 81630,c1(C(N(C2CCN(C(C(C)OCCC#C)=O)C2)CCO)=O)nn(C)cc1SC 81631,C1(NC(CC(=O)NCC)=O)CCN(C(C2CC(C)(C)CO2)=O)CC1O 81632,C1CCC(F)(F)C1.CCCCCCn1nnnc1C1(N)CCOC1 81633,n1(CC)ncc(C(=O)NCCc2nc(CC(F)(F)F)cs2)n1 81634,C12(C(N3CC(CCNC(c4cnncc4C(F)(F)F)=O)C3)=O)CCC(CC1O)C2 81635,C1(C(=O)OC)CN(C(=O)C(N)CSC2CCCCC2)CC2(CCC2)O1 81636,c1(C(C)C(=O)N(CCNC(c2cc[nH]n2)=O)C2CC2)ccnn1C 81637,C(=O)(C(CC(C)C)NC(=O)C(C1(CC)CC1)N(C)C(C)C)OCC 81638,CON(CCCO)C(=O)C(c1cn(C)nn1)NC(=O)CCn1cncn1 81639,N1(C(CNS(NC)(=O)=O)=O)CCN(CCn2cc(C3CC(C)CCO3)nn2)CC1 81640,C(O)(C(F)(F)F)C1(C(=O)NC2(CN(C(=O)Cn3[nH]cnc3=N)C)CC2)CCC1 81641,CCCC(C(=O)NCCC1(NC(=O)CC(C)O)CCC1)c1ccc(Cl)cc1 81642,C(=O)(C1CCc2ccccc21)N1CCC(OC)(CNC(c2coc(CO)c2)=O)C1 81643,c1(C(=O)NC2CN(Cc3ccc(OC)cc3Cl)CC2F)cc(F)cc(C)c1O 81644,C#CC1CCCN(C(C2CCC3(CC3)N2C(C2CCC2COC)=O)=O)CC1 81645,c1(OCC)c(Cl)cc(C)nc1C(=O)NCCCN(C(=O)CCCS(N)(=O)=O)C 81646,N#Cc1cncc(CC(N2CCC2CNC(c2coc(CC3CC3)c2)=O)=O)c1 81647,C1(C(=O)NC2CC3(C2)CC3NC(=O)C(F)CC2CC2)CCn2c(O)nnc2C1 81648,N1(C(C(C)C2CC2)=O)CC(CNC(c2ccc(NS(C)(=O)=O)o2)=O)OC(C)(C)C1 81649,N1(C(CCCOCC=C)=O)CC(N(C(=O)C(CC=C)OC)C)C2(CC2)C1 81650,C12(C(N(CC(C)NC(C3(C(=O)NCC)CCC3)=O)CC)=O)CC1COC2(C)C 81651,c1(-c2cn(C3(C)CN(C(c4c(OC)ccs4)=O)C3)nn2)ccc(F)c(F)c1 81652,C1(C)(C(N2C(Cn3cc(C(CC)OC)nn3)C=CC2)=O)CS(=O)(=O)C1 81653,c1(OC)ccc(Br)c(C(=O)N(CC(c2cccc(Br)c2)O)C)c1C 81654,CC(C)(C)C(CNC(=O)CCCc1ccccn1)NC(=O)CC1CC1 81655,N1(C(CCC=C(C)C)=O)CC2(CC(C(N3CC(C(C)C)C3)=O)CO2)C1 81656,c1(NCC2CN(C(CC(CC)O)=O)C2)ncnc2ccsc12 81657,c1(CC(=O)NC2CN(C(c3nc(C)oc3C)=O)CC2C)cccc([N+](=O)[O-])c1 81658,c1(C(=O)NC2CC(NC(c3c(C)cc(C)c(Br)c3)=O)C2)cnc2c(c1)OCCN2 81659,C(=O)(Nn1cnn(CC)c1=O)C1COCCN(C(C(CC#C)O)=O)C1 81660,c1(-c2cn(C(C)CNC(c3cccc(F)c3N)=O)nn2)ccc2c(c1)CCC2 81661,c1(C(C)C)nn(C)cc1C(=O)NCC1CC(O)CN1C(=O)C(O)Cn1cncn1 81662,N1(C(Cc2n(C)cnn2)=O)CCCC(C2(NC(=O)CC(C)(O)C3CC3)CC2)C1 81663,c1(C(C)C)cnc(Cl)nc1N1CCCCC(CNC(=O)C2=CCCCO2)C1 81664,c12cnc(N)c(c1)C(=O)N2.Cc1cnn(C(C)C(=O)N2CC(c3nn[nH]n3)C2)c1 81665,CC1CC(C(=O)N2CCCCC2CCN(C)C(c2cc(F)ccc2Cl)=O)=NO1 81666,N1(C(C2CC(C)(F)C2)=O)CCC2(CCN(C(C3CC(=O)CO3)=O)C2)C1 81667,N1(C(C(COC)C)=O)CCC12CCCN(C(c1c3c(nn1C)CCCC3)=O)C2 81668,c1(C(N2CCC(CNC(c3c(CC)cno3)=O)CC2)=O)cnc(C2CC2)[nH]c1=N 81669,N1(C(c2c(C)non2)=O)CC2CCCC2C1C(=O)NC1CCOCC1F 81670,c1(CNCC(C)Cn2ccnc2)ccccc1OC(F)(F)F.CC(=O)O 81671,c1(OC)ccccc1NC(=O)C(=O)N(CCCN(C)C)C1CC1.C1(=O)C=CCN1 81672,Cn1cnc2c(N3CCC3CNC(=O)CCCC3CCCC3)nc(Cl)nc12 81673,c1(C(N2CC(C(N3CC4CC4(CO)C3)=O)C(F)C2)=O)c(O)cccc1F 81674,N1(C(CCOCCCOC)=O)C2CCC1C(NC(C1CN3CCN1CC3)=O)C2 81675,c1(C(=O)NC23C(CN(C(C4C(C(=O)OC)C4)=O)C2)CC3)cnc2c(n1)CCCC2 81676,C1(C(=O)NC(c2cn(C(C)C(=O)O)nn2)c2ncon2)CCCCCC1 81677,Nc1cccc(C(N2CC(C(C)(C)O)(CNC(=O)C(F)C3CCOC3)C2)=O)n1 81678,c1(C(N2CCCN(C(CC)=O)CCC2)=O)cc2cc(OC(C)=O)ccc2cn1 81679,CCCC(C)CN=C(NCC1CCCO1)NC1CCN(C(=O)C2CC2)CC1 81680,c1(C(=O)NCCc2c(C(=O)NCCSC)c[nH]n2)sc(F)cc1C 81681,CC(C)(C)CC(O)C(=O)NCC1COCC1NC(C1SC2C=CC1CC2)=O 81682,C1(CC)CN(C(C2(Cl)CC2C(C)=O)=O)CCC1CNC(C1CC(=O)N(OC)C1)=O 81683,N1(C(C=C(COC)C)=O)CCC2(CC1)CN(C(=O)CNS(C)(=O)=O)CC(C)O2 81684,C1(N(C(CCOCCN(C)C)=O)C)CCC(NC(=O)COCC2CCCC2)C1 81685,C12(NC(CCn3c(C)ncc3)=O)COCCC1CN(C(=O)CN(S(C)(=O)=O)C)C2 81686,Cc1cccc(CC(=O)NC(CNC(=O)Cc2c(C)noc2C)CO)c1F 81687,C1(NC(c2c(C)cc(Cl)cc2)=O)CCNCCC1(F)F 81688,C1(C(=O)NCCC23CC(CCO2)C3)C2CCC(C2)C1NC(=O)C1=CCOCC1 81689,N1(CC)CCCC(C(=O)N(CC(C)CNC(=O)CCNC(C)=O)C)C1 81690,Cc1ccc2c(CC(N3CCN(C(=O)CCn4cccn4)C4CC34)=O)c[nH]c2c1 81691,C=CCC(CC(F)F)C(=O)N(C)CC1CCCN1C(c1ccc(CC)cc1)=O 81692,C1(NC(C(c2c(CC)cccc2)(F)F)=O)CCN(C(=O)OC(C)(C)C)CC1(C)C 81693,C(C)(CNC(c1csc(=N)[nH]1)=O)(CC(C)C)NC(COCCC=C)=O 81694,C1(C(=O)NCCC2CCN(C(=O)CCC3CC3(Cl)Cl)C2)CCS(=O)CC1 81695,N1(C(C(C)=CC2CC2)=O)CC2C(CN(C(=O)CN3CCCC3C)C)C2C1 81696,c1(CC(=O)NC2(C)CCCN(C(C3(COC)CC3)=O)C2)cccc2oc(C)nc12 81697,C(=O)(CC(CC(C)C)NC(=O)C(O)CN1CCCC1)NCCCC#C 81698,C1(C(N(C(CC)CC)C)=O)CCC(CNC(=O)C(O)CSC)CC1 81699,N1(CCNC(C(CC)n2cncn2)=O)CCC(NC(=O)CC2(O)CC2)CC1 81700,c1(C(=O)NC(CC)(CC)CCNC(=O)C(C#N)CC)n[nH]c2c1COCC2 81701,c1(C(=O)NC2CC2)ccnc(OC(F)F)c1.c12ccc(o1)COCCCNC2=O 81702,N1(CC(C)C)CCN(C(=O)C(c2ccccc2)NC(=O)CC2CCOC2C)CC1 81703,c1(C(=O)NCC(=C)CCNC(=O)CCS(C)(=O)=O)cnn2c1CCCC2 81704,C(=O)(CC(CNC(C1(OC(C)C)CCOC1)=O)OC)NC(CC)C1CC1 81705,C1(NC(C(C2CCC2)N(C)CCCC(=O)NC2CC(C#N)C2)=O)CCCCC1 81706,C#CCC(C)(C(=O)NCCC(C)CCC)NC(c1cnc(O)c(F)c1)=O 81707,CC1(CNC(=O)C=CC(=O)NC2CC2)CCN(C(C2C3CCCCCC23)=O)CC1 81708,C1(CC#C)CCCN(C(=O)CC2CCN(C(c3cc[nH]c(=N)n3)=O)C2)C1 81709,C1(CNC(C2(C)C(C)C2)=O)CC2CCC1N2C(=O)C(C)(Cl)Cl 81710,c1(OC)cc(NC(c2ccc(I)cc2OC(F)(F)F)=O)c(Cl)cc1Br 81711,N1(C(c2cnc(CCOCC)s2)C(=O)NCC)Cc2c[nH]nc2CC(C)C1 81712,Cn1ncc2nc[nH]c(=NC3CN(C(=O)CC4C=CCCC4)C3)c12 81713,N12CC3C(C3C1)C2=O.C=CCS(=O)(=O)NCCN(CC)CC 81714,N1(C(CC2OCC(C)(C)C2)=O)C2CCC1C1CC1(NC(=O)CCn1ccnc1)C2 81715,CCC1=C(C(=O)NCC2CCC(C(=O)NC(C3CC4(CCC4)C3)C)C2)CCCO1 81716,CCC(F)(F)C(C)(C)C(=O)NC(C1CC(NC(c2cccnc2C(F)F)=O)C1)C 81717,c1(-n2cc(C3N(C(C(C)OC)=O)CCC3C)nn2)ccc2nc(N(C)C)oc2c1 81718,C1(NC(C(CNC(C2=CCCC2C)=O)O)=O)CCC(N=[N+]=[N-])CC1 81719,c1(CC)cc([N+](=O)[O-])ccc1N(CC(C)NC(=O)CC1=CCOCC1)CC 81720,N1(C(C2C(CCC)CN(C(=O)CN(CC(C)(C)C)C)C2)=O)CC2(CNC(=O)C2)C1 81721,c1(C(=O)NCC(C)(CNC(=O)C2=CCCC2)OC)cc([N+](=O)[O-])oc1C 81722,c1(CNC(c2ncoc2CNC(C2CCCOC2)=O)=O)ncccc1Cl 81723,c1(CC(=O)N(C2CCN(C(C3CS(=O)C3)=O)CC2)CC)cc(F)cc(F)c1 81724,c1(C(=O)NC(CC=C)CNC(=O)C(C)=CC2CC2)cccn(C(C)(C)C)c1=O 81725,C1(CNC(C2CN(C)C(=O)N2)=O)CN(C)CCN1C(=O)CSc1cn[nH]c1 81726,C1(CNC(C(C)CF)=O)CN(C(=O)C=Cc2cncn2C)CC1(F)F 81727,C1(C(N(C)CC2CCCN(C(=O)CCOCC(F)F)C2)=O)CC2CC1CC2O 81728,CCCCC(O)C(=O)NCC1(NC(c2nn(C(F)F)cc2Cl)=O)CCOC1 81729,C1(C(=O)NC(CC(C)NC(CCOCC)=O)C)C2CC1(c1ccc(Cl)cc1)CO2 81730,CC(C(=O)NCCNC(=O)C(C)Oc1cc(Cl)cc(Cl)c1)C(F)(F)C(F)F 81731,c1(NC(C2CCCN(C(C3CC(C)(C(C)(C)C)C3)=O)C2)C)ncc(Cl)cn1 81732,c1(C(N2C(C)CC(NC(C(C(=O)OCC)(C)C)=O)C2)=O)cc2ccccn2n1 81733,Cc1ccn(CC(C)(O)C(=O)NCCCNC(=O)Cn2cc(Cl)cn2)c(=O)c1 81734,c1(C(N2CC(CC)N(C(C3CCC3(F)F)=O)CC2)=O)c(F)cc(Cl)cc1F 81735,C1(NC(c2cnc(C(C)C)[nH]2)=O)CC1C1CCCN(C(=O)CC(C)(C)C#N)C1 81736,CCCCC(F)C(=O)NCC1CN(C(=O)CS(=O)(=O)NC)C(C)(C)C1 81737,CON(CCC(=O)O)C(=O)C(=O)NOC1CCC(C)(C)CN1 81738,Cc1[nH]nc(C(N2CC(NC(=O)CC3CCCCCO3)C(C)C2)=O)c1C 81739,N1(C(c2c(C)oc(C(C)C)c2)=O)CC2CCN(C(=O)CC(C)O)CC2C1 81740,C(C(=O)NC1(CC2CCC2)CC1)(C(C)(C)O)NC(C(CC=CC)C)=O 81741,N1(C(C(Cc2ccc(C)cc2)C)=O)C2CCC1C(CNC(c1csnc1Cl)=O)C2 81742,CCCC(CCNC(C1C2CC3C(C2NC(c2cnns2)=O)C13)=O)CCC 81743,C1(NC(C2C(=C)C2)=O)CCC(NC(C2CCSCC2)=O)CC1 81744,N1(C(c2cc(CC)nn2C)=O)CC(NC(c2cc(C)c(C)nn2)=O)C2CCCC12 81745,N1(C(C2CN(C)C(=O)C2)=O)CCCC2(CCN(C(c3cc(F)ccc3O)=O)C2)C1 81746,Cn1cc(CC(=O)NCC(O)CCNC(c2ccc(C(F)F)nc2)=O)c(Cl)n1 81747,C(=O)(C(C)(C(C)C)N(C)C)NCC(C)N(C(c1cnccc1OC)=O)CC 81748,c1(C(N(CC(=O)NO)CC(c2ccc(F)cc2)=O)=O)n[nH]c2c1CC1CC21 81749,C1(CNC(CC(C)OC)=O)CN(C)CCN1C(=O)Cc1cc(Cl)cc(Cl)c1 81750,c1(OC)ccc(CNSc2ncoc2C2CC2)cc1O 81751,C(=O)(C(C(C)(C)C)C1CCC1)N1CC(CN(C(=O)CC2CCCCC2O)C)C1 81752,N1(C(=O)CC23CCC(CC2)C3)CCOC(C2CN(C(c3cc(Cl)no3)=O)C2)C1 81753,N1(C(C(C2CCCC2)OC)=O)CC(NC(=O)C(=O)N(C)C)C2CCCC12 81754,C(=O)(CCCCCNC(N)=O)N1CC2C(CNC(CSCC)=O)C2C1 81755,N1(C(CC2(CNC(C(C)O)=O)CC2)=O)CCC2(CCN(C)C2)C1 81756,C=C(C)CCCC(=O)N(C1CCC(NC(c2cccnc2CC)=O)CC1)C 81757,N1(C(C)=O)CCOC(C(N2CC(NC(c3coc(C(F)F)c3)=O)CC2CO)=O)C1 81758,CC(CNC(C1C(C#N)C1(C)C)=O)CC(=O)N(C)CC1CCCC2CC12 81759,C=CCC(CC(C)C)C(=O)NC1CC(NC(=O)Cc2ccn(C)n2)C(O)C1 81760,C1(NC(c2c(CC)c[nH]c2)=O)CN(C(c2cccc(O)n2)=O)CC1n1ccnn1 81761,C12(C(=O)NC(COC)C)CCCC1CN(C(C1CNC(=O)O1)=O)C2 81762,Cc1ncc2n1CC(C(=O)NCC1(NC(C3CC3(F)F)=O)CCCCC1)CC2 81763,c1(C(=O)NC(C2CN(C(=O)Cc3nc[nH]n3)C2)C)ccc(N2CCOC2=O)cc1 81764,CC1COC2(C1)CN(C(C1CCN(C(C3C4CC5C(C4)C35)=O)CC1C)=O)C2 81765,CC(C)CC(=O)NC1COCC1CNC(=O)CCCC1CCCCC1 81766,C#Cc1cc(C(=O)NCC(CCCC)NC(=O)C=COCC)cc(N)c1 81767,N(C)(S(=O)(=O)N1CCCC1c1ccc(O)cc1)CC(CC)SC 81768,C1(C(=O)NC)CC2CCC1N2C(=O)COC(F)F.CC1CNC1=O.C(C)(C)(C)O 81769,c1(C(N(C(C(=O)N(C(C#C)C)CCCC)C)C)=O)ccc(N)cn1 81770,C1(C(=O)NCCOC2CCN(C(CC(C)(C)O)=O)CC2)CC2CCC(C1)C2 81771,C1(CC=C)(NC(=O)CC2CCC(NC(=O)CCN(C)CCO)C2)CCOCC1 81772,c1(CC(C(N2CCC(NC(CCOCCC)=O)C2)=O)O)cc(Cl)sc1Cl 81773,N1(c2nnc(C(C)(C)C)o2)CCC(CO)(CNC(C2(CO)CCCO2)=O)CC1 81774,C1(c2ncno2)CCC(F)(F)CC1.c1(C(C)N)cc(C2(O)COC2)on1 81775,C=CCC(F)(F)C(=O)NCC1(OC)CCN(C(C2(O)CCSC2)=O)CC1 81776,CC(N=c1[nH]c(=NCc2nnc(C(F)F)s2)c2ccccc2[nH]1)c1cccs1 81777,C1(F)(CNC(c2nc[nH]c2C(F)(F)F)=O)CCCN(C(=O)C2=CCOCC2)C1 81778,C1(CC(=O)NCCCN(C)C(c2csc(=N)[nH]2)=O)(C(F)(F)F)CC(=O)N(O)C1 81779,c1(N(CC(=C)C)C)cc(NCC23CC(CC2C(=O)O)C3)ncn1 81780,c1(C(N(C2CCC(NC(C3(O)CCC3)=O)C2)C)=O)cc(-c2cccnc2)nn1C 81781,C12(C(=O)NCCN(C(C3C(OCC)C3C)=O)C)C3C4C1C1C2C3C41C#N 81782,CC1CC(NC(=O)C(=O)N(CC(C2CCCCC2)O)C)CC(c2ccccc2)C1 81783,C1(CC)CN(CC=Cc2ccccc2)C(CC)CN1CC(=O)OC 81784,CC1CN2CCN1C(C(=O)NCC1(F)CCN(C(c3ccc(F)c(O)c3)=O)C1)C2 81785,c1(CC#N)ccc(OCCNC2(c3nnnn3Cc3ccco3)CCCC2)cc1 81786,N1(C(CN2CC(CC)C2)=O)C2CCC1CC(C(=O)NCc1ccc(Cl)cc1Cl)C2 81787,c1(CN2CC(C(N(CC)CC)=O)SCC2)cc(Br)cc([N+](=O)[O-])c1O 81788,CN1CCN(C(=O)Cc2csc(Cl)n2)C(CNC(=O)C(c2ccccc2)=O)C1 81789,C(=O)(C(C)(C)S(C)(=O)=O)NC1(CNC(c2ccc(OC)nc2)=O)CC1 81790,CC#CCC(C(=O)NC(c1cncs1)C)NC(C1CC(NC)C1)=O 81791,NC(=O)CC(C(=O)N1CCC(F)C(F)C1)NC(C1CCCC1C1CC1)=O 81792,C12(CNC(C(C3CC3)OC)=O)CC(NC(C3SCCS3)=O)(CCO1)C2 81793,N1(C(C(N2CCCC(Cc3scc(C)n3)C2)C)=O)CCC2(CC1)NC(=O)CO2 81794,c1(OC)cccc(OC)c1C(N1C(C)C2CC1C2NC(c1cnc(C)[nH]1)=O)=O 81795,CCC(CNC(C1CC2(C1)CC(O)C2)=O)(CC)C(=O)N(C)CCn1cncn1 81796,C(CCN=c1cc(Cl)nc(S(C)(=O)=O)[nH]1)N(C(=O)C(=O)NC1CCCC1)C 81797,Cc1ccc(Cl)c(OCCOC(=O)Cc2cncc(F)c2)c1 81798,c1(NC)ccc(C(=O)NCC(CC2CC2)C(=O)NC(C(O)CO)C2CC2)nc1 81799,C1(C(N(CCN=[N+]=[N-])C)=O)CCN(C(=O)C2CC2(F)Cl)O1 81800,CC(C)(F)CC(=O)NC1(CCNC(=O)C(O)Cc2cccc(Cl)c2)CC1 81801,Cc1nc(C)c(C(C)NC(=O)CCOCCN(C)C(c2ccc(=N)[nH]c2)=O)[nH]1 81802,Cc1ccn(CC(=O)N(CCNC(=O)CN2CCCCC2)C(C)C)n1 81803,Cc1cc(=NC(C)CC(C)NC(=O)CC2(C)CC2(F)Cl)[nH]cc1C#N 81804,C(=O)(C(C(C)C)NC(=O)CC(C)C)NCC1(NC(CC(=C)C)=O)CCOC1 81805,C#Cc1ccc(NC(c2nc(-c3ccnc(C(C)C)c3)cs2)=O)cc1 81806,C(=O)(CCCCCC(=O)OC)N(CC(C)N(C(=O)C(C)=C1CCC1)CC)CC 81807,CC1CCCCC1(C)NC(=O)C=CCN(C(=O)Cc1cnn(C)c1)C 81808,C1(NC(CC(=O)N(C)C)=O)CCN(C(=O)COCC(F)F)C(C2CC2)C1 81809,c1(NC(=O)NC2CC(CN3CCC(OC)C3)C2)ccc(Cl)cn1 81810,c1(C(c2nnnn2C2CC2)NCC2C(C(=O)OC)C2)cnc(-c2ccccc2)s1 81811,C(c1ccccn1)=C(C)C(=O)NC1CN(C(C2(c3cc(C)no3)CC2)=O)CC1F 81812,c1(C(N(CC(=O)OC)Cc2cn(CC(CC)O)nn2)=O)ccc(F)c(Cl)c1F 81813,N1(C(c2cc(C)no2)=O)CCC2CCN(C(c3ccc(C4CC4)cn3)=O)CC12 81814,CCC(C(=O)NCCN(C(=O)C(F)(F)CC(C)C)CC)C(C)(F)F 81815,C(=O)(C(C)CS(C)(=O)=O)NCC1C(NC(c2ccc(CC)cc2OC)=O)C1 81816,N1(C(CC(C)c2ccco2)=O)CCC(C)(C)C(C(=O)NC2CCCC2)C1 81817,C1(NC)CCC(C(=O)NCCNC2CCCN2S(C)(=O)=O)C1.C12CN(C1)C2=O 81818,C12(NC(c3cc(C(C)C)n(C)n3)=O)CCOCC1CN(C(C1(F)CCC1)=O)C2 81819,N1(C(c2cc(C)cc(Br)c2)C(=O)NCCOCC)CCC(C2CC2(F)F)C1 81820,C(CCCCCC(=O)NCC1CC1C1CCCC1)NC(=O)C=CCN1CCC1 81821,C1(CC(=O)NCCN(C(=O)C(C)(C2(C)CC2)OC)CC)CC=CCN1C 81822,N1(C(C2N(S(C)(=O)=O)CCC2)=O)CC(NC(=O)Cc2ccncc2Cl)CC(F)C1 81823,C12(C(N(CCC#N)CC)=O)CC(c3ccccc3)(C1)CS(=O)(=O)C2 81824,c1(C(=O)NCC2CC(NC(C3CC34CCOCC4)=O)C2)cc2ccccn2n1 81825,C(C)(C(C(C)C)NC(c1ccc(-c2cccs2)s1)=O)NC(C(C)=CC)=O 81826,c1(C(N2CC(CO)C3(CC3)C2)C(=O)NCCCOC)cccc(Br)c1F 81827,C(N=c1nc2sccc2c(NC2CS(=O)(=O)CC2C)[nH]1)c1c(C(C)C)con1 81828,C12(CN)CCC(C(=O)OC)(CC1)OC2.C1(C(CN)OCC)CCOC1 81829,C1(NC(Cc2cc(C)on2)=O)C2CC3CN(C(c4nocc4C)=O)C1C3C2 81830,C1(NC(C(C(COC)C)C)=O)CC2CC(C1)N(C(=O)CCNC(=O)C=CCl)C2 81831,N1(C(CCN(CCC)C)=O)CCCC2CN(C(C3NC(=O)C4CCC34)=O)CC12 81832,c1(NC)cncc(C(N2CCCC(C3CCCCN3C(=O)C(C)CO)C2)=O)c1 81833,CCCCC(O)C(C)C(=O)NCCCNC(=O)C(C)=CC(C)(C)C 81834,c1(NC(C23CN(C(=O)C(F)Br)CC2CCO3)=O)ccc2ccccc2c1 81835,C1(CCC)CN(C(c2cccc(Cl)c2N)=O)CCN1C(c1snnc1C1CC1)=O 81836,C12(OC(C)(C)C)CC(CN(C(=O)C(O)c3cnc[nH]3)C1)C2 81837,C(=O)(CC(C(=C)C)OCC)N(CCCC(=O)NC(C#C)(C)C)C 81838,C1(CNC(CC2(OC)CCCC2)=O)CCCN(C(=O)Cc2cnn(C(F)F)c2)C1 81839,N1(C(C2N(C(C)C)CCC2)=O)CCC(CN(C)C)(NC(=O)C(C)P(C)(C)=O)CC1 81840,N1(C(CCC(=C)Cl)=O)CCCC(C)(NC(C2CCC(OC)CC2)=O)C1 81841,C1(CC(=O)NCCC)CCC(NC(Cn2ncc(C(=O)NC)c2F)=O)CC1 81842,CCC(C)(C)CCCC(=O)N(CCNC(c1c(C)ccc(C)c1C)=O)C1CC1 81843,CC(CC(=O)N1CCC(C(N2CCC(O)CC2(C)C)=O)C1)CC(C)(C)C 81844,n1(CCN(C2CCN(CC(F)(F)F)C2=O)C2CN(C)C(=O)C2)cnc2sccc2c1=O 81845,c1(CC)cc2c(NCC3CN(C(=O)CC4CCOCC4OC)CCO3)ncnc2s1 81846,C1(CC)(NC(C2CCC(=O)C2)=O)CCN(C(=O)C(c2ccc(F)cc2)C)CC1 81847,C(CC1CC1)(C(=O)NC(C)(C)CO)NC(CCC1C(C)C1)=O 81848,N1(C(=O)NC2CC(CC(=O)OCC)C2)CC2(CCC2)OC2(CCC2)C1 81849,c1(C(=O)NC2C3CC(NC(c4c(CC)noc4)=O)CC32)cnc2[nH]ncc2c1 81850,N1(C(c2cc(N3CCCC3=O)cc(Br)c2)=O)CCC2CCN(C3CC3)C2C1 81851,N1(C(C(C)O)=O)CCC2(C1)CN(C(c1coc(Cn3cccn3)c1)=O)C2 81852,N1(C(CCCC)=O)C2CCC(C(=O)N(C)Cc3ncccn3)C1CC2 81853,Cc1nc(O)ccc1C(=O)NC1COCC1CNC(=O)CN1CCCOC1=O 81854,N1(C(CSCC=C)=O)CC2(CCN2C(c2cc(F)cc(Cl)c2)=O)C1 81855,N1(C(C(CC)NC(C)=O)=O)CC2COCCC2(NC(c2csc(Cl)c2Cl)=O)C1 81856,c1(COC)nn(C)cc1C(=O)N(CC(C)N(C(=O)C=Cc1cnn(C)c1)C)C 81857,c1(C(C)NC(c2ccc(CNC(C(C)(C)NC(C)=O)=O)s2)=O)cccc(F)c1 81858,n1(C(CC)CC)nccc1C(N1CCC1CNC(=O)C(O)CC1CCCCC1)=O 81859,N1(C(C2=C(C)CCC2)=O)CCC2(CCN(C(c3ccccc3C)=O)CC2)C(C)C1 81860,C1(CC(N2CC3C(NC(C(C)OCCCC)=O)(C3)C2)=O)OC(C)(C)OC1=O 81861,C1(NC(CCCCN(C)C)=O)CC2CC(NC(=O)CCc3cc(Cl)cs3)C1C2 81862,c1(OC)cnc(C(C(=O)NC2CCC2)N(CC(C)SC)C)cc1Br 81863,N1(C(C2(C)COC2)=O)CCC(O)(CNC(=O)C(O)Cc2c(F)cccc2Cl)CC1 81864,Cc1nncc(C(=O)NC(c2cn(CC3CC3)nn2)C2CC(F)(F)C2)c1C 81865,C1(C(N2CCC(C(N(CCN(CC)CC)C)=O)C2)=O)CC2CCCC2C1 81866,Cc1ccc(C(=O)NCCC(C)NC(c2cn(C3CC3)cn2)=O)c(F)c1Cl 81867,C1(NC(c2c(C)noc2)=O)C2CC1N(C(C13CCCCC1C3)=O)C2 81868,C1(C(=O)NCCCC(CCC)NC(C2(CO)COC2)=O)CCC2(CCC2)CO1 81869,Cc1cnsc1C(N1CC(F)(CNC(C2CC2c2ccccn2)=O)C1)=O 81870,N1(C(CC2(C=C)CCC2)=O)CC2(NC(C3CCCN3C(C)C)=O)CCCC2(F)C1 81871,O(N(CC)C(=O)CNC(C1CCOC1)=O)CC 81872,Cc1cncc(C(=O)NCCC2CSCCN2C(C2CCC(C(N)=O)N2C)=O)c1 81873,C(=O)(C(O)CCC(F)(F)F)N(CC(=O)N(CC(F)(F)F)C(C)C)CCO 81874,c1(C(N2CC3(CN(c4cc(OC)ncn4)C3)C2)=O)noc2c1CCCC2 81875,N1(CCC(=O)NCC2CN(C(CSCCN(C)C)=O)C2)CCOC1=O 81876,Cc1cc(C(N2CCC(c3cn(C4CC4)nn3)C2)=O)ncc1C(F)(F)F 81877,C1(CNC(CCC=C)(C)c2nnnn2CC)CC2(CCC2O)C1 81878,c1(CNC(C(=O)Nc2c(C)ccc(F)c2Br)=O)ccc2c(c1)CC(C)O2 81879,c1(C(N2CCN(CC(C)(C)NC(C(C)OC)=O)CC2)=O)nccc(Cl)c1C 81880,C(=O)(CC(CNC(=O)NC(CC1CC(F)(F)C1)CO)C(C)C)OC 81881,C1(C(N2C(CC)CN(C(C3CN(C(C)C4CC4)C3)=O)CC2)=O)CC2OC(=O)OC2C1 81882,CC(C)(C(=O)NC1CC1CNC(=O)CC1(CO)CC1)C(F)(F)F.C12(CC1)C(=O)N2 81883,C12(C(N(C(CSC)C)C)=O)CC1CN(C(C1(C)COC(=O)N1)=O)C2 81884,C1(C(=O)NCC(C)(O)C(=O)OC)(COC)C=CCN1C(=O)CC1CC(=O)NC1=O 81885,C(CN=C(NCC1CCCCS1)NCC1C=CCC1)SC 81886,N1(C(c2n(CC)ncc2)=O)CCC(C)(NC(=O)CC2(C)CCCCC2)C1 81887,c1(CN(C(CC)C)C)cc(OC)ncc1Cl.C12CN(C1)C2=O 81888,c1(C(N(CCCC)CC)=O)ccncc1I 81889,c1(C(=O)NCC(CC)(C)NC(=O)Cc2ccccc2Cl)cnn(C)c1C 81890,C1(OC)CCC2(C(=O)NC3CCCC(C(=O)NCCc4ncc[nH]4)C3)CC12 81891,n1(CC)nnnc1C(c1cnc(SC)s1)NC(c1ccc(C)o1)C 81892,c1(C(=O)NC(C(=O)NC(CC)C2CCC2)COC)cc(C)c(C)cn1 81893,C1(NC(C2CC23CCC3)=O)C2CC3CN(C(c4c[nH]c5ncccc45)=O)C1C3C2 81894,N1(CC)CCN(CCC(=O)N(C2CCN(C(=O)Cc3cn(C)nc3C)C2)C)CC1 81895,C1(NC(CN(C(Cc2c(C)con2)=O)C2CCC2)=O)CCOC2(CCC2)C1 81896,C(CNC(=O)CC(C)C1CCCCC1)(CCNC(=O)Cc1cc(C)[nH]n1)OC 81897,Cn1c(C(=O)N(CCC(N2CCC(c3cc[nH]n3)C2)=O)CC(C)(C)C)cnc1S 81898,C12(CSC)CC(C(=O)NCC(C3CC3)NC(=O)CC3(C)CC3(F)Cl)(CO1)C2 81899,N1(C(C(C)(C)C#N)=O)CCCC(O)(CCNC(=O)COCC2(F)CC2)C1 81900,C1(O)(CC(=O)N(C2CCC(NC(C3(C)CC(C)(C)C3)=O)CC2)C)COC(C)(C)C1 81901,C(=O)(C(C)C(=O)N(C1(C(=O)NCCc2cc(C)nn2C)CC1)C)OC 81902,C1(NC(CP(C)(C)=O)=O)CCC2(CCCN2C(=O)COC2CC2)CC1 81903,CC(=O)CCCC(C)C(=O)NCc1cccc(C(=O)NCCc2ncnn2C)n1 81904,c1(NCC2N(CC)CCCC2)ncnc(NC(c2cnn[nH]2)C)c1C 81905,c1(C(=O)NCC2CCCN(C(C3(CCO)CC3)=O)CC2)ccc2c(c1)CCC2 81906,C(=O)(C(C)C(F)(F)C(F)F)N1CCCN(C(C(c2ccc(Cl)nc2)C)=O)CC1 81907,C(=O)(C(C(C)C)NC(C1CN(c2cnccn2)C1)=O)NC1CCN(C(CC)=O)C1 81908,CCCC(O)C(=O)N1CC(C(c2cn(C3(CC)CC3)nn2)SC2COC(=O)N2)C1 81909,n1(CC(=O)NC(C2(CNC(C3C=CCC3)=O)CC2)C)ccc(Br)cc1=O 81910,N1(C(C(CC)(C)COC)=O)CC(C)(C)OC2(C1)CN(C(=O)C(C)S(N)(=O)=O)C2 81911,c1(C(=O)NCC(CN(C(C(C)=CC2CC2)=O)C)O)cc(CCCO)on1 81912,N1(C(C=CCC)=O)CCN(C(c2ccc(Cl)o2)=O)CC1C(F)F 81913,C(C(=O)NCC1(CCNC(C2CCCC23CC3)=O)CC1)(C(C)(C)C)OC 81914,C(=O)(C1=C(CC)OCCC1)NCC(C(=O)NCC(C#C)C(C)C)CC1CC1 81915,c1(C(N2CCCC(CC=C)(NC(c3cncn3C)=O)C2)=O)csc2ccncc12 81916,Cc1cc(C(=O)NC2CC(O)CN(C(=O)CCc3cc(C)[nH]n3)C2)c(O)c(C)c1 81917,CCCCC(O)CC(=O)NC(CSC)C(=O)NCCc1cn(C)nc1C 81918,c1(C(=O)OC(C)C)cccnc1NCC=CCNC(=O)C=Cc1ccccc1 81919,c1(C(=O)NCC(C)NC(=O)CSc2nc(-c3ccccc3)no2)cncc(F)c1 81920,N1(C(CN(CC#C)C(c2ccn(CCF)n2)=O)=O)CCC(C)C(C)C1 81921,C(C)(C)(CC(=O)NCC1CCC1NC(=O)Cc1ccc(O)nc1)N(C)C 81922,C1(C(=O)OCC)(NC2CCCC2NC(=O)COc2cc(C)on2)CC(F)(F)C1 81923,C1(CC#C)(C(=O)NC2CC(O)C2OC)CCN(C(=O)CC(C)(C)OC)C1 81924,C1(CCC(=O)NC2CC3(C2)CC3NC(C2CC2[N+](=O)[O-])=O)CCC(O)CC1 81925,c1(CCN(CCOC)C)cn(C(C)CNC(c2nncn2C)=O)nn1 81926,CCC(C)C(=O)C(=O)NC(Cn1cccn1)C(=O)NCC(C)(O)C(C)CC 81927,C(=O)(C(C(C)CC)OC)NC1CC(C)(C(=O)NC)C1 81928,c1(C(N(CCC(C)NC(=O)C(C)(C)n2cccn2)C)=O)nc(Cl)c(Cl)s1 81929,Cc1cccc(C(N2CCOCC2CC(=O)NCCCC(=O)N(C)C)=O)c1 81930,N1(C(C)=O)CCCCC1C1CCCN1C(c1ccc2c(c1)C(N)CCC2)=O 81931,N1(C(c2c(C)coc2)=O)CCCC1(C)C(=O)NCCN1CCCC1=O 81932,C(=O)(C(O)P(C)(C)=O)NC(C)CNC(=O)Cn1cnc(Br)c1 81933,C1(C(CO)CCN(C(CC)=O)CCO)CCN(C(=O)C(C)C)CC1 81934,C(C(C)C(F)C(=O)NOCC(=O)NC1CC2CC(=O)C1O2)NC(C)=O 81935,c1(N2CCC(C(C)(C)C)C2)ccc(S(=O)(=O)NC(C(C)(C)CO)C2CC2)cc1Br 81936,c1(CC(=O)N(CC(C)(C)NC(C(CC)Oc2ccccc2)=O)C)nn(C)cc1Cl 81937,N1(C(c2c(CC)ncnc2)=O)CCN(C(=O)C(O)(CC)c2ccccc2)C(C)C1 81938,C1(NC(c2cc(C)ncc2)=O)CC2CCC1N(C(c1ncc(C)cn1)=O)C2 81939,C(CN=c1cc[nH]cc1S(=O)(=O)N1CC=CC(OC)C1)SCC=C 81940,N1(C(c2c(C)noc2)=O)CC(C)CN(C(c2snnc2C)=O)CC1C 81941,c1(C(N2CCCC2)=O)cc(C(=O)NCCCOCCNC(C2CC2(F)F)=O)no1 81942,c1(SCC)cncc(C(=O)NCC(CNC(c2[nH]ccc2C2CC2)=O)CO)n1 81943,C(=O)(C(C)CCCC(C)C)N1CC(C(C(N2CCC(C(=O)OCC)CC2)=O)OC)C1 81944,c1(C(N(C2CN(C(C3CNC(=O)N3)=O)C2)C)=O)cccc2nc[nH]c12 81945,C(=O)(CCC(=O)N1CC2C(c3ccc(C)cc3)C2C1)OC 81946,C(=O)(C(C(C)C)(C(C)C)NC(C)=O)NCCCN(C(C(CCCC)C)=O)C 81947,N1(C(c2c(C)cncn2)=O)CC2(C1)CN(C(=O)C#CC(C)C)CC2CO 81948,c1(C(=O)NCC(C(=O)NC(CCO)C(F)(F)F)OC)ccc2[nH]ccc2c1 81949,c1(C(=O)OC)ccncc1NC(C1CCC(NC(=O)Cc2cc(C)on2)C1)=O 81950,C(=O)(C(C)(C)C(=O)NC1CCCN(C(=O)C(c2cnn(C)c2)C)C1)OC 81951,C#CCC(C)C(=O)NCC(c1ccccc1)=O.C12(CCCC1)C(=O)NCC2 81952,C1(NC(C2N(C)CCC2)=O)CN(C(c2cn(CC(F)(F)F)cn2)=O)C(C)(C)C1 81953,C1(C(=O)NCC2(C)CCCO2)CC12CCN(C(=O)C(C)(C)C(C)(F)F)CC2 81954,C1(CCC)COCCN1C(=O)C(=O)NN(C)C[Si](C)(C)C 81955,N(C)(S(N)(=O)=O)CC(=O)N(C1CCN(C(C2CC2C)=O)C1)CC 81956,c1(N2CC(NC(C(C)O)=O)(CO)C2)nc2c(cc1C#N)CCC2(C)C 81957,C1(C(=O)NC(C)C(CO)NC(c2cc(C(F)F)nn2C)=O)CCC(C)(C)C1 81958,C(=O)(C(C(F)(F)F)OC(=O)NC)NCC(CN(C(C(CC=C)C)=O)C)(C)C 81959,CC1CN(C(=O)C(F)C2CCC2)CCCN1C(=O)C1=COCCO1 81960,c1(C(=O)OC)cc(NC(=O)CC2CC(O)C23CCC3)cc(Br)c1C 81961,N1(C(CCCC#C)=O)CCn2c(C(=O)Nc3ccc(Br)cc3C#N)cnc2C1C 81962,C1(CC)CCN(C(=O)Nc2ccc(F)c(C(F)F)c2)CCO1 81963,CC1CCC=C1C(=O)NC(C)C=CC(=O)NCCc1ncc[nH]1 81964,C1(CNC(c2n(CC)ncc2Cl)=O)CCC2(CN(C(C3OCCO3)=O)C2)O1 81965,c1(OC)ccc(C(c2nnnn2C)NCCSc2ccncc2)c(Cl)c1 81966,c1(C(=O)OCC(N2C(=O)NC3(CCCC3)C2=O)C)ccc(O)c2ccccc12 81967,C(=O)(C1=CCOC1)N(CCC(C)NC(Cc1n(C(C)C)cnn1)=O)C 81968,CCCCCCCCNC(=O)NC1(C)CN(C(C2CCC(F)(F)C2)=O)C1 81969,C1(NC(CCSCCCC)=O)CC12CCC(NC(=O)C#CC1CC1)CC2 81970,N1(C(C(CC)F)=O)CC2(CC(NC(=O)CCC(C)(C)c3ccccc3)C2)C1 81971,N1(C(c2c(C)cc(O)cc2)=O)CCC(C2CC2)(NC(=O)Cc2cn3ccsc3n2)C1 81972,N1(C(c2c(C)n[nH]c2C)=O)CC(NC(=O)Cc2ccc(Br)cc2I)C2(CC2)C1 81973,c12c(C)csc1C(=O)N1CCOC(C1)CN2.c1(S)ccccc1.CCOC 81974,n1(CC)ncc2c1CC(C(=O)NC1CN(C(=O)CCc3cncs3)CC1C)CC2 81975,N1(C(C2C(=C)C2C(=O)OC)=O)CC(CNC(=O)Cc2ccc(Cl)cn2)C(F)C1 81976,C1(NC(C=C(CC)CC)=O)CC(C)(C(=O)NC(C2CC2c2ccnn2C)C)C1 81977,c1(OC)cc(Br)cc(F)c1C(=O)Nc1cnn2c1CCCC2 81978,C(=O)(C(O)CCC(C)C)NC(C(C(=O)NCc1cc(C)cc(O)c1)C)C 81979,C1(C(=O)NCC2(O)CCCC2)CC2CCC(C1)N2C(C1CC1C(F)(F)F)=O 81980,N1(C(=O)COc2cccnc2Cl)CCN(C(=O)CCn2cncn2)C(CCO)C1 81981,c1(C(=O)NC(CN(C(c2ccccc2N(C)C)=O)CC)C)ccn(C)c1C 81982,C1(C(CC)CC)CCc2nc(NC(=O)C(C)C(C)O)sc2C1.n1(CC=O)nccc1N 81983,c1(N(CC(C)C)CCC2CN(C)C2=O)nccc(O)n1 81984,C1(C(=O)NCC#CCNC(c2cncc(OCCOC)c2)=O)(CC)CCCCC1 81985,C1(C(N(C)CCC2CCC2)=O)C(O)CCN1C(c1ncn(C)n1)=O 81986,C1(NC(CNC(=O)OCC)=O)CCCN(C(C2CCCCC2)C(=O)OC(C)=O)C1 81987,C1(CC)(NC(=O)Cc2cn(C)nc2C)CCCN(C(=O)C(=O)NCC(F)(F)F)C1 81988,C1(CNC(c2cc(C)[nH]n2)=O)CC(F)CN1C(c1nc(C(F)(F)F)cs1)=O 81989,CCC(CC)C(=O)N(CC(C)(C)NC(c1cn(C(C)(C)C)nc1C)=O)C 81990,C1(NC(C2(OC)CCOC2)=O)CC2COCC(C1)N2C(c1cc(C)nc(O)n1)=O 81991,c1(NC(=O)C=CCN2CCNCC2)c(C(=O)N(CCO)CCO)cccc1Cl 81992,C1(OC)CCC2(C(N3CC(O)(C(F)C(=O)NCCn4cc(C)cn4)C3)=O)CC12 81993,N1(C(c2n(C(C)C)cnc2)=O)CCC2(CCCCC2NC(=O)C(F)CC2CC2)C1 81994,N1(C(N)=O)CCC(CO)(CNC2(c3nnnn3CCC3CC3)CC3COC2O3)C1 81995,C1(C(=O)NC(CC)CNC(=O)Cc2cc(F)ccc2Cl)CNC(=O)CC1(C)C 81996,CC1CN(C(=O)CCC2CC2)CC1CNC(c1cc(-c2cnn(C)c2)no1)=O 81997,C(=O)(CC(C)(C)CC(F)(F)F)NCCN(C(c1cc(C)sc1C)=O)CC1CC1 81998,C(=O)(C(C)CC(C)C)N1CC(C(C)NC(c2ccc(SCC)nc2)=O)C1 81999,c1(COCC)ccccc1CNC(=O)C(=O)NCc1ccc(O)cc1.C1CNC1 82000,c1(C(N2CCC3C(NC(C4N(C(C)=O)CCC4)=O)C32)=O)cc(C)cc(Cl)c1N 82001,CN1CCCC(F)(C(N2CC3(CC(CNC(=O)CCC(N)=O)C3)C2)=O)C1 82002,CC1(C(N2CCC(O)(CNC(=O)CC3COC(=O)N3)C2)=O)CCCS1(=O)=O 82003,c1(CN2C(c3n(C)ccn3)CCCC2)c(F)cc(Br)c2cccnc12 82004,C1(NC(COCCOC)=O)CCCCN(C(C2CCOC2=O)=O)CC1 82005,N1(C(C=Cc2ccc(SC)s2)=O)CCN(C(c2cc(C)c(C)cn2)=O)CC(O)C1 82006,N1(c2ncc(C)cn2)CCOC(C)(CNC(=O)COc2ccc(Cl)cc2C)C1 82007,c1(OCC)ccc(O)cc1C(=O)NC1CN(C(c2cncc(C)n2)=O)CC1C#N 82008,C(=O)(C1CCOc2ccccc21)NCC1N(C(c2cc(N)c(Cl)cc2)=O)CCC1 82009,c1(C(N2CC3C(N(C)C(=O)OC(C)(C)C)(C3)C2)=O)cc([N+](=O)[O-])ccc1O 82010,C(CCCCCNC(=O)CC1COC(=O)C1)N(C(=O)CSCc1ccccc1)C 82011,c1(OC)ccc(C(=O)N(C)CC2CCOCC2)c(C(F)F)c1 82012,c1(CCC(=O)N(CCCN(C(=O)CCc2cncn2C)C)C)cccc(C#N)c1 82013,c1(C(=O)NC(Cn2cc(C3(COC)CCC3)nn2)C)ccc(Br)cc1 82014,c1(C(N2CC3CCC(C2)N3Cc2ccc(I)o2)=O)cnc2cc(Br)ccc2c1 82015,C1(CNC(C(C)(C)C(F)F)=O)CCC2(CN(C(C3CC4(C3)CS(=O)(=O)C4)=O)C2)O1 82016,CCCCC(C(=O)N1CCCC(CN(C(c2cn(C)nc2C)=O)CC)C1)C(C)C 82017,c1(CC2(F)CN(C(Cn3cc(CC(C(C)C)O)nn3)=O)C2)ccc(F)cc1 82018,C1(O)(CNC(C2(CCC=C)CN(C(=O)CCC3CCCC3)C2)=O)CCOC1C 82019,c1(OCC(=O)NC2(C)CCN(C(C3C(C)CC3)=O)C2)ccc(Cl)c(F)c1 82020,CC1(C(=O)NCC2C=CC(NC(=O)Cc3cccc(C(N)=O)c3)C2)CCCCO1 82021,C(=O)(CC(C)(C)N(C(=O)Cc1cccnc1C)C)N(CCCC(=O)OC)C 82022,C1(N(C)C(C2CCC(c3ccccc3)C2)=O)CCN(Cc2cnccc2Cl)CC1 82023,C1(NC(c2nccc(C)n2)=O)CC2(CCN(C(C3COC(C)(C)C3)=O)C2)C1 82024,N1(C2N(C(C(C)c3cc[nH]n3)=O)CC2)CCC(C)C(C(F)(F)F)C1 82025,C1(CNC(Cc2cccc(CC)c2)=O)CCN(C(=O)C(F)(F)C(C)O)CC1(F)F 82026,N(C1CN(C(=O)CC(C)(C)OCC(C)(C)C)CCc2ccccc21)C(COC)=O 82027,N1(C(c2cnc(CC)[nH]2)=O)CC(CNC(=O)C(c2cncnc2)C)C(C)C1 82028,c1(C(C(=O)NC(CC)(C)C)N(C)Cc2cc(C)on2)ccc2c(c1Cl)OCO2 82029,c1(N(c2nc(C(C)(C)C)cs2)C(C)=O)c(NC(=O)C#CC2CC2)ccc2c1CCC2 82030,c1(OC)cccc(C=CC(=O)NCC(C)OC)c1OC(C)=O 82031,c1(C(=O)NCC2(NC(COCCC(C)C)=O)CCC2)cccn(C)c1=O 82032,C(=O)(C(C)(C)CCSC)N1CCCC(F)(CNC(CCN(C(CCC)C)C)=O)C1 82033,C1(NC(C(C)N(CC(F)(F)F)C)=O)CC(C)CN(C(c2cc(Cl)c[nH]2)=O)C1 82034,c1(C(=O)NC2C(NC(C(c3n(C)ccn3)(F)F)=O)CC2)cnc2ccccn12 82035,C1(C(=O)NCC2OCCN(C)C2)COC2(C1)CN(C(C1CN(CCF)C1)=O)C2 82036,c1(OC)ccc(C(N2CCC(NC(=O)C=Cc3ccn(C)c3)CC2C)=O)cc1F 82037,C1(CNC(C(COC(C)C)NC(C)=O)=O)COCCN(C(C2COC(=O)O2)=O)C1 82038,c1(SCC)cccc(C(=O)NC2(CNC(=O)Cc3ccccn3)COC2)c1 82039,c1(C(=O)NCC2C(NC(C=C(CC)C)=O)CC2)cnn(CCCC)c1C 82040,c1(C(N2CCCC(C)(NC(=O)C=CC3CCOCC3)C2)=O)cnc2sccc2c1 82041,C1(NC(C2(c3cc(C)no3)CC2)=O)CCC(C)N(C(=O)C(C(C)C)C2CCC2)C1 82042,CC(C(C)C(=O)N1CC(C)(F)C1)NC(c1ccc[nH]1)=O 82043,C(c1cncnc1O)=CC(=O)N(C1CCCC(NC(c2n[nH]c(C)c2Cl)=O)C1)C 82044,c1(C(=O)NCCC(C)(C)NC(C2CC2F)=O)cc(F)c(Br)cc1F 82045,N#CCCCCCC(=O)N1CCN(C(=O)CCF)C(CCO)C1 82046,CC(C)(C(=O)N1CCC(O)(CCNC(C23CC(CCO2)C3)=O)CC1)C(N)=O 82047,CCC(C)(CCC(C)C)C(=O)N1CCCC(CNC(=O)C(OC)OC)CC1 82048,N1(C(c2ccc(COC)[nH]2)=O)CCOC2(CCC(Nc3ncccn3)CC2)C1 82049,C1(NC(c2c(C)sc(O)n2)=O)CN(C(c2cc(F)cnc2O)=O)CCC1C 82050,C#Cc1cccc(NC(C)C(=O)NC(C)CNC(=O)CSCCC(F)(F)F)c1 82051,c1(CN(C(=O)CC=CCNC(C2CC2C(=O)N(C)C)=O)CC)cncn1C 82052,N1(CC(C)(C)NC(C2N(CC)CCC2)=O)CCN(C(=O)Cc2scnc2C)CC1 82053,c1(C(c2nnnn2C)NCc2c(C)noc2C)ccc(Cl)cc1F 82054,CC(F)(C(=O)N(CCNC(C1CCCOC1)=O)C1CC1)c1ccon1 82055,C(=O)(C(C(C)O)N(C)C)NCC(=C1CN(C(c2ccc(C(C)=O)s2)=O)C1)F 82056,Cc1ncnc(O)c1C(=O)N(C)CCC1CCCCN1C(=O)CC(C)C 82057,S1(=O)(=O)C2CC(C2)NC(=O)CC2CCN1C2.Cc1cc(NC)no1.C(C)(C)O 82058,C1(CC)CN(C(C2CCS(=O)(=O)C2)=O)CCN1C(=O)Cc1cn(C(C)C)nn1 82059,N1(C(C2(CC#C)CC=CCC2)=O)CCC2(CCCCN(C(=O)CNC=O)C2)C1 82060,Cn1cc(C(N2CCN(C3CCN(C(=O)C4=CCC4)C3)CC2)=O)c(C(F)(F)F)c1 82061,Cc1noc(C)c1C(C)C(=O)NCC(CNC(=O)Cc1cccnc1)CO 82062,c1(CC)nn(C)c(C(=O)N(CCNC(=O)C(CC)C(C)O)C2CC2)c1Cl 82063,C=CC(C)(C)C(=O)NCC12CC(CN1C(=O)C(C)NS(=O)(=O)CCCC)C2 82064,c1(C(=O)NCC2CN(C(C=C3CCN(C)C3)=O)C(C)(C)C2)csc(S(C)(=O)=O)c1 82065,C(=O)(CC1=CCCCC1)NC1C(C(N2CC(C(C)(C)C)OCC2)=O)OCC1 82066,C1(NC(C2(C)CC2)=O)CC2CCC1CC2NC(C1CCC(CCO)CC1)=O 82067,S(=O)(=O)(CC(=O)NCC1CN(C(=O)Cc2cc[nH]n2)C1)NC(C)(C)C 82068,C1(C)(CNC(COC2CN(C(C)=O)C2)=O)CC1(Cl)Cl 82069,N1(C(Cc2n(C)cnc2)=O)CCOCC(CNC(C2(C3CCCO3)CCC2)=O)C1 82070,Cc1noc(Cl)c1CC(=O)NCC(C)(C)CNC(c1c(C)nsc1N)=O 82071,c1(N2CC(SC)C(N(C)C)C2)ncc(C)cc1S(=O)(=O)NC1(CO)CC=CC1 82072,Cc1oc(-c2ccco2)nc1CC(=O)NCC(C)(C)NC(=O)CNC=O 82073,c1(-n2c(C(N)COc3ccccc3)nc(COC)n2)ccc(F)cc1OC 82074,c1(C(N(CCNC(c2ccnc(CO)c2)=O)CC2CC2)=O)cccc(O)n1 82075,c1(C(N2CC(C)C(NC(=O)C(c3ccc(F)cc3)(C)F)C2)=O)cccc(Cl)c1N 82076,C1(NC(CCC2(C)CN(C(COCC(=O)NC)=O)C2)=O)CCCCCC1C 82077,c1(C(N2CCC(N(C(CCC(C)C)=O)CCO)C2)=O)ccc([N+](=O)[O-])cc1 82078,N1(C(c2cc(C)[nH]c2)=O)CC2CCC(C(=O)NCC3=NOC4CCCC34)(C2)C1 82079,CCCC(C(=O)NC(C(=O)NC1CCCCC1N(C)C)C1CCCC1)OC 82080,C1(C(=O)NCCCC(C)NC(c2scc(C)c2Cl)=O)CCC(=O)C(C)C1 82081,N1(C(c2cc(Br)n3c2CCC3)=O)CCCC2C1CCCN2C(=O)CO 82082,c1(C2(C(N3CCC(C(C)O)C3)=O)CC2)ccc(Cl)c(Br)c1 82083,C1(CC#N)CCN(C(=O)NCC2(c3ccc(O)nc3)CC2)CC1 82084,c1(C(N2CCC(N(C(c3c(C)snc3)=O)C)CC2)=O)cccc2nc(CO)[nH]c12 82085,C1(OC)(CNC(C2CC(=O)N(C(C)C)C2)=O)CCN(C(C2CCSCC2)=O)C1 82086,C1(N(C(=O)CCC2CCOC2)C)CCN(C(c2ncncc2Cl)=O)CC1 82087,C=CCCCC(=O)N1CCC(CNC(=O)COC)(CC)C1.c1(O)ccsc1 82088,c1(OC2(C(N(CCCCN(C(=O)CCC3CC3)C)C)=O)CC2)cnn(C)c1 82089,Cc1cccc(CC(=O)NCCCCN(C)C(c2c(Cl)nsc2Cl)=O)c1 82090,CON(C)C(=O)CNC(c1c(CNC(=O)CC(C)=C(C)C)cnn1C)=O 82091,N1(C(CCC=C(C)C)=O)C2CCC1CC(N(C(=O)C(C)N(C)C)C)C2 82092,Fc1ccc(CNc2cc(NCC(F)F)ncn2)cc1OCC(F)F 82093,Cc1ccc(=NCCC(=O)NCCNC(c2cc3n(n2)CCN(C)C3=O)=O)[nH]c1 82094,n1(CC)ccc(C(=O)NCCCN(C(=O)C=C(C)C(F)F)C(C)C)c1C 82095,c1(C(c2n(CCCC)nnn2)NC(CC)C2CCC2)ccc(C(=O)N(C)C)cc1 82096,C(C(=O)NCC(O)CC(=O)NCC(Cl)=CCl)(C(C)(C)C)N(C)C 82097,C(=O)(CCCC(C)CC)NCC1CN(C(c2c(C)cc(CC)o2)=O)CC12CC2 82098,C(CC(C)C(=O)NCC1CN(C(C2(CO)CC(C)(C)C2)=O)C1)=CC 82099,Nc1c(F)cc(-c2ccc(-c3nccn3C3C4COCC34)c(F)c2)cc1F 82100,c1(OCC)cnc(C(N2CCC(C)C2CNC(C2CCN(CC)C2)=O)=O)cn1 82101,C1(N(C(CCCOCC)=O)C)CCN(C(=O)CCSc2ccccc2Cl)CC1C 82102,C1(C(N2CC(O)(CCNC(C3C(C)OCCC3)=O)C2)=O)CCCC2C1C2(F)F 82103,O(NC(=O)C(C1(O)CCCCC1)NC(=O)CCC(C)C)C(C=C)C 82104,c1(OC)ccc(F)c(C(=O)NCCC2CCCCN2C(C2CCC(O)C2)=O)c1Cl 82105,C1(CC(=O)NCC(C)(C)OCCNC(C(C)=C(CC)C)=O)CCCNC(=O)C1 82106,c1(CN(C(=O)NC2C(c3ccc(C)o3)C2)C)cccnc1N1CCCC1 82107,n1(CC#C)c(C)cc(C(N2CCN(C(=O)C(C)CCN(C)C)C(CC)C2)=O)c1C 82108,c1(C(N(CC(CN(C(C(CCC)F)=O)C)O)C)=O)cccc(CC)c1F 82109,C12(C(=O)NCCOCCC(=O)NCc3scc(C)n3)CCC(CC1F)C2 82110,C1(CC(N2CC(CC=C)(NC(=O)C=CCOC)C2)=O)CCOCC1(C)C 82111,N1(C(c2cc(CC)n(CCO)n2)=O)CCN(C(c2ccsc2Cl)=O)C(CC)C1 82112,Cc1cccc2c1ccn2CC(=O)N(C1CN(C(=O)C(F)C(F)(F)F)CC1O)C 82113,N1(C(=O)C=C2CCC2)CCN(C(C2C3CNC(=O)C23)=O)C(c2ccccn2)C1 82114,Cc1c(C(=O)NC2CCC2CNC(=O)CCS(C)(=O)=O)sc2cncn12 82115,c1(OC)ccnc(C(=O)NC(C)CCNC(=O)C=Cc2ccnn2C)c1N 82116,CCC(CCC(=O)NC1CCN(CCCNC(=O)Cc2cncn2C)C1)OC 82117,c1(C(=O)NCC(CNC(c2cc(C)cs2)=O)OC)cc(O)n(C)n1 82118,N1(C(c2c(COC)cccc2)=O)CCN(Cc2cc(C)sc2C)C2CC12 82119,N1(C(c2cncnc2)C(=O)Nc2cccc(Cl)c2)CC(F)(F)CC1COCCO 82120,CC1CCC(C)(C=CC(=O)NC2CC3(CCN(C(C4(C)CC4)=O)C3)C2)C1(C)C 82121,c1(C(=O)NC)cc(Cl)ccc1NCc1ccc(C(C)(C)C)cc1.C1(C)C(=O)N1 82122,c1(C(C)NC(=O)COC(c2cnc(C#N)s2)=O)cccc(OC(F)(F)F)c1 82123,c1(CN(c2c(F)cnc(OCC)n2)C2CNCC2O)ccc(F)c(Cl)c1F 82124,c1(CCC(=O)NC23CCN(C(c4ccoc4)=O)CCC2C3)cnc2ncccn12 82125,C1(CNC(c2n(C=C)ncc2)=O)CN(C(C2(C#N)CC3(CC3)C2)=O)CCN1C 82126,C(CCCCCC(=O)NCc1ccc(Cl)c(C(F)(F)F)c1)NC(N)=O 82127,c1(CNC(C(C2CCOC2)NC(C(F)=CCC)=O)=O)ncnn1C 82128,C12(NC(CC(C)C)=O)CCC(C(N3CCCC(CCO)C3)=O)(CC1)C2 82129,C(=O)(CC(O)C1CCCC1)N1C(CNC(=O)Cc2csc(Br)c2)CC1 82130,c1(N2CC(CCC=C)(C(=O)NC(c3ccc(C)cc3)C)C2)nc[nH]c2ncnc1-2 82131,N1(C(=O)NC(c2ccccc2)=O)CCN(Cc2occc2Cl)C2CC12 82132,C1(CC(=O)N(C)CC2CN(C(=O)C(F)(F)c3cscn3)C2)(OC)CCCCC1 82133,N(C(=NCCCc1ccc(Cl)c(Cl)c1)NCCCCl)Cc1c(C)cccn1 82134,N1(S(Cc2c(C)cccc2)(=O)=O)CC(=O)N(C)CC1C(=O)O 82135,CC(C)(C)CCCC(=O)NC1(C)CCN(C(C2(C)CCCO2)=O)C1 82136,N1(C(C(OC)OC)=O)CC(=O)NCC1C(=O)NCCOCCCF 82137,c1(C(N2CC3CN(C(C(CCC)O)=O)CC32)=O)ccc2cnn(C)c2c1 82138,c1(C(=O)NC2COCCC2NC(C2CCCCO2)=O)ccc2c(c1O)CCC2 82139,C1(NC(c2cnc(CC)o2)=O)CC(NC(c2nc(C)c(C)s2)=O)C12CCC2 82140,C(=O)(C1CCCc2nn[nH]c21)N(C)CC1CCN(C(CCNC(=O)NC)=O)C1 82141,N1(C(CCSC)=O)CC2C(CNC(=O)Cc3scnc3C)C2C1 82142,Cc1c(F)ccc(C(N2CCOC(CNC(C3(C)C=CCC3)=O)C2)=O)c1Cl 82143,CCC(CC)CCC(=O)NC1CCOC(C(N2CCN(CCF)CC2)=O)C1 82144,N1(C(CCCCC)=O)CCN(C(=O)CC2CCCC2C)C2(CCC2)C1 82145,c1(N(C)C)ccc(C(=O)NC2CCC2NC(c2ccncc2F)=O)cc1[N+](=O)[O-] 82146,O=C(NNc1nc[nH]n1)c1ccc2n[nH]cc2n1 82147,C1(NC(c2cnc(CC(C)C)[nH]2)=O)CCSC12CN(C(=O)CCc1nc[nH]n1)C2 82148,C1(C(N2CCCC(OC)C2)=O)COCCN(C2CCCC(C)C2)C1 82149,c1(CC)ccc(CCCC(=O)NC2CCN(C(C3CC34CCC4)=O)C2)cc1 82150,c1(N2CC3C(NC(C(CC)CCOC)=O)C3C2)c(Br)cccc1[N+](=O)[O-] 82151,c1(C(N(CC(C)(C)NC(CC2CC(OC)C2)=O)C)=O)csc(C(F)(F)F)n1 82152,n1(CCCO)nc(-c2ccc(OCc3ccccc3)cc2)nc1-c1ccon1 82153,C(N=c1[nH]c(C)ncc1F)C1C(NC(C=CCC)=O)C2(CC1)CCC2 82154,N1(C(c2[nH]c(=NC)sc2)=O)CCCC2(CCC(NC(c3ccc(C)o3)=O)C2)C1 82155,C1(C(=O)NC2CC(C(=O)NC(C(C)C)C)C2)(CF)CCOCC1 82156,Cc1cc(N)ccc1C(N1CCC(O)(CCNC(c2ccnc(CO)c2)=O)C1)=O 82157,c1(C(N2CC(C)(CCC(=O)NC(CCSC)CO)C2)=O)cc(C)c(F)cn1 82158,C1(C(N2CC(CNC(=O)Cn3cncn3)C2)=O)CC(O)CN1c1ccncn1 82159,N1(C(C2CCC(CNC(CC(C)F)=O)C2)=O)CCOC2(CCCC2)C1 82160,C1(N(C(C2CC(CC)(CC)C2)=O)C)CCCC(NC(=O)C=Cc2nccs2)C1 82161,C(=O)(CC(C)(C)CC(=O)NCC=CCNC(C1CCC1(F)F)=O)OCC 82162,c1(CC)nc(C)c(C(N2CC(NC(C34CC(C)(C3)C4)=O)CC2C)=O)o1 82163,N1(C(C2CC(NC)C2)=O)C(C(=O)NCC(=O)N(C)C2CC2)CCC1C(C)C 82164,N1(C(c2cc(OC)no2)=O)CCCCC1C1(NC(=O)CCc2cncnc2)CC1 82165,N1(C(c2ccc(OC(F)F)cc2)=O)CCOC2CCN(Cc3cccs3)CC12 82166,CC(CC(F)F)C(=O)NCC1CCCCN1C(=O)CCCNC(N)=O 82167,N1(c2nnc(C)o2)CCN(C2CCN(C(C3CCC(C)(C)C3)=O)C2)C(=O)C1 82168,c1(OC)cc(F)c(S(N)(=O)=O)cc1C(N1CCC(N2CC(F)C2)C1)=O 82169,n1(CCOC)cccc(C(N2CCOC(C3CCCCC3)C2)=O)c1=O 82170,C1(CC#C)CCN(C(C2CCC(NC(=O)CCC3CC3C)CC2)=O)CC1 82171,C1(C(=O)NC2(CF)CN(C(C3C(C)CCC3)=O)C2)COCCN1C=O 82172,N1(C(C2CCN(Cc3ccc(C#N)s3)CC2)=O)CC2CCC(C1)O2 82173,c1(NC(C2CCN(C(c3cccc(C4(C)CC4)c3)=O)C2)=O)ncc(Br)cc1C#N 82174,C12(C(=O)NC3(C)CC(NC(C(C)Cc4ccncc4)=O)C3)CCC(C1)OC2 82175,N1(C(C2(CCC=C)CN(C(C3C4C5CCC(C5)C34)=O)C2)=O)CC(O)C(C)(C)C1 82176,c1(OCC)ccc(CC(=O)NCCC2CN(C(C3CN(C)C3)=O)CC2C)nc1 82177,c1(C(=O)NCC(c2ccccc2)NC(=O)CCC2CC2)cnn2c1OCC(O)C2 82178,C1(C(=O)NCC(CNC(=O)CCc2ccc(Cl)cc2)F)NC(=O)C2CCC12 82179,N1(C(c2cnc(OCC)nc2)=O)CC2CC(NC(C3CCC4(C3)N=N4)=O)C2C1 82180,c1(C(C(=O)NCCCC(C)NC(c2ccc(CO)o2)=O)O)ccc(F)cc1 82181,c1(N2CC(O)(CCNC(C3CCC(C)C3)=O)C2)cc(F)ncn1 82182,C1(C(=O)NCCC(CCC)O)C2CCC(C2)N1C(c1coc(N(C)C)n1)=O 82183,C(=O)(CCCCC(F)F)N1C(C)CC(NC(C=Cc2ccc(C(=O)OC)cc2)=O)C1 82184,N1(C(C(C=C)(C)CC)=O)CCC(N(C(=O)CCOc2ccccc2)C)C2(CC2)C1 82185,Cn1cc(C(=O)NCC2(F)CCN(C(c3cc(N)ccn3)=O)C2)nc1O 82186,C1(OC(c2cncc(OC(C)(C)C)n2)=O)CCC=CCCC1 82187,C(c1cccc(Cl)c1)=CC(N1CC(NC(c2ccc(OCC)nc2)=O)C(O)C1)=O 82188,C1(NC(c2c(C)noc2N)=O)CN(C(C2CCCN2C)=O)C2(CCOCC2)C1 82189,N1(C(c2ccc(OC)nc2)=O)CC(NC(=O)Cn2nnc(=O)[nH]2)CC12CCOC2 82190,c1(CC(=O)NC2CCCC(CNC(C=CC=CC)=O)C2)ccc(C#N)nc1 82191,CC1CCOCC1C(=O)NCC1(C(=O)NC2CC(=O)N(O)C2)CCCCC1 82192,c1(CC(N2CC(CCCC)N(C(=O)C(C)CCC)CC2)=O)cnn2c1CCCC2 82193,O=S(=O)(c1ccc(Br)cc1NCCCCCCO)NC1(CCF)CC1.C1(C)CC1 82194,c1(C(CNC(C2CCCC2)C)O)ccc2c(c1)CCCC2 82195,C12CCCN(C1)CCN2c1ccncn1.C1=CCC(C(C2CC2)C2CC2)CC1 82196,C1(C(=O)NC2CC(NC(c3ccc(C(C)(F)F)cn3)=O)C2)C(F)(F)C12CCC2 82197,c1(C(C)=O)ccc(C(=O)NC(Cc2cc[nH]n2)C(=O)N2CC=CC2C(=O)NC)o1 82198,C1(C(=O)NCC2(COC)CN(C(c3cocn3)=O)C2)CC2(CSC2)C1 82199,c1(CCC)cccc(NC(=O)CCC2CC(NC(=O)C(C)SC)C2)c1 82200,c1(C(=O)NCc2ccc(C(C)NC(CC(C)SC)=O)cc2)ccc2nn[nH]c2n1 82201,N1(C(c2cc(C)no2)=O)CC(C)N(C(=O)CN(C(=O)C(C)C)C)C(C)C1 82202,C(N=c1cccc(S(=O)(=O)NC2CCCc3occc32)[nH]1)c1c(C#N)cccc1 82203,c1(-c2ccn(C)n2)cc(C(=O)Nc2cc(Cl)nc(Cl)c2)cc2cc[nH]c12 82204,Cc1cc(C(=O)NCc2n[nH]cc2C(=O)N(C)Cc2cnn(C)c2C)c(C)nn1 82205,N1(C(c2c(OC)ccnc2)=O)CCC2(CCCC2NC(=O)C=C2CCCCC2)C1 82206,N1(C(c2cn(CC=C)nc2)=O)CCC(C)C(NC(=O)CC(C)(O)C2CC2)C1 82207,c1(NC(C(=O)NC2C(CC)CNCC2)=O)ccc(-n2cc(Cl)cn2)c(Cl)c1 82208,c1(OC)nc(C)c(COC(=O)CCC2CC(C)(C)CO2)s1 82209,C(=O)(CCC(=O)NCC1(C(=O)NCc2ccn(C)n2)CC1)NCCC 82210,c1(OC)cc(C)c(Br)cc1NC(=O)C(c1ccccc1)OC(C)C 82211,c1(NC(C2C(C(=O)Nc3cc(C(C)(C)C)[nH]c3)C2)=O)c(O)cccc1Cl 82212,c1(C(=O)NC(C(=O)NC2(CO)CC(C)C2)c2cccs2)cc(C#N)cs1 82213,CC(CNC(C1CCCC1CNC(=O)CN1CCC(F)CC1)=O)(CO)CO 82214,c1(C(=O)NCC2C(CNC(C34CCCCC3C4)=O)C2(F)F)ccc(F)cc1F 82215,N1(C(C(CC)OCC)=O)CC2(CCN(C(C3CCC(=C4CCC4)CC3)=O)C2)C1 82216,C1(OCCNC(C2CN(C(C)=O)C2)=O)CCN(C(C2OCC2(C)C)=O)C1 82217,Cc1ccc2nc(C(N3CCN(C(=O)C#CC4CC4)C(CF)C3)=O)cn2c1 82218,C1(CNC(Cc2ccc(SCC)cc2)=O)CCCCN(C(C2OCCCO2)=O)C1 82219,CC1(C)C=C(C(=O)NCC(c2ccccc2)NC(c2cncc(Cl)c2)=O)C1 82220,C1(CNC(c2c(C)cnn2C(C)C)=O)CN(C(=O)CCCC2CC2C)CC1(F)F 82221,c1(C(=O)NCC(CNC(c2cc(C)sc2C)=O)F)ccc(N)c(C(F)(F)F)c1 82222,C1(=Cc2ncc(CCC)s2)SC(=S)N(C(C)C)C1=O 82223,C1(C)(OC)CCC(NC(C2CC(NC(=O)CC3CC(C)(C)CO3)C2)=O)CC1 82224,COn1cnc(C)c1C(N1CC(NC(C2CCC2(C)C)=O)C(O)C1)=O 82225,CC1(NC(=O)Cc2csc(S)n2)CCCN(C(C2CCCC2(F)F)=O)C1 82226,N1(C(COCC=C)=O)CC(CNC(c2cc(OCC)n[nH]2)=O)CC1C 82227,CN1CC(C)(C(=O)NCCCCC(CO)NC(c2ccc(F)cc2F)=O)CC1=O 82228,C(CNC(=O)Cc1cccs1)(CC(=O)NCCC1CC(F)C1)OC 82229,n1(C(C(=O)NC(C)CSC(F)F)C)cc(C2(N3CCC3)CCC2)nn1 82230,C1(OC)CC2CCC1CC2C(=O)NC1CN(C(=O)C(C)Cc2ccc(C)cc2)C1 82231,c1(C(CF)NC(=O)NCC2(CCOC)CC2)cccc(OC)c1 82232,c1(C(N2CC3CCN(C(C4ON=C(C)C4)=O)CC32)=O)cnc2ccc(F)cc2c1 82233,C1(CNC(C2CCC(OC)CC2)=O)CC2CN(C(C3CCN(OC)CC3)=O)CC12 82234,c1(CN(C(C(COC)O)=O)CCNC(=O)Cn2ccnc2C)ccc(F)cc1 82235,C12(CNC(C(C)NC(COC)=O)=O)CCC(CC1)N2C(=O)Cc1c[nH]nc1C 82236,c1(C(=O)NC23C(CN(C(CCC=C)=O)C2)CC3)cc(Cl)c(N)cc1F 82237,C(=O)(C(CO)C(F)(F)F)NCC(C1(O)CCCCC1)(CC)C 82238,c1(C(N2C(CC(=O)NCCCc3cc[nH]n3)COCC2)=O)occ2c1CCC2 82239,C1(CNC(CN(C)C2CC2)=O)CN(C(=O)CC2NC(=O)NC2=O)CCC1(C)C 82240,C1(C(C)NC(=O)C(C)(C)C2CCCC2)CN(C(C2COCCO2)=O)CCO1 82241,Cn1cc(C(N2CCN(C(=O)COC3(C)CCCC3)C(C3CC3)C2)=O)ccc1=O 82242,C1(C(N2CCC(=C)C2)=O)C=CCCN1C(=O)C(C)OC1CCCC1 82243,C1(CC(N2C(CCN(C)C(C3CCCS3)=O)CCCC2)=O)CCC2(CC1)CC2 82244,c1(CC)nc(N2CCC(NC(=O)CSCCN(C)C)C(F)C2)c(C)c(Cl)n1 82245,Cc1sncc1C(=O)NCC(C)C(=O)NCCNS(N)(=O)=O 82246,c1(C(=O)NC(C2CN(C(=O)COC(C)(C)C)CCO2)C)noc2cc(F)ccc12 82247,C1(C)(C(N(C2CCCN(C(C3(C#N)CCCC3)=O)CC2)C)=O)CCC(=O)NC1 82248,N1(C(C2(CC=C)CCCN2C(=O)C2=CCOCC2)=O)CCC2OCCC2C1 82249,c1(C(N2CCCC(CNC(CC(C)SC)=O)C2)=O)nn(C)c(Cl)c1Cl 82250,C(C1CCCN1C(=O)C(C)n1ccnn1)=CC(=O)NC1(C(COC)O)CC1 82251,CN=c1[nH]cc(C(N2CCC(N(CCO)C(c3cc(COC)no3)=O)C2)=O)s1 82252,C1(CC(=O)NC(CNC(CCOC(C)C)=O)CO)CCOC1(C)C 82253,C(CC(=O)N1CC(C)(NC(C2CC3(C2)CS(=O)(=O)C3)=O)C1)(C1=CCCC1)OCC 82254,C(C(C(=O)NC(c1cscn1)C)NC(=O)C(n1ccc(C)n1)C)OC 82255,C12(C(=O)OC)CCC(CC1NC(=O)C(C)CCNC(=O)CN1CCC(OC)C1)C2 82256,C1(NC(=O)C=CC(=O)NCC2(CN)CC2)CC1.C(=O)(CNC=O)N(C)C 82257,C1(CC)CN(C(=O)CC2COCCOC2)CC1C(=O)NCC1CCCS1 82258,C(N=c1nc2c(cnn2C)c(N(C)Cc2cc(C)no2)[nH]1)C1(OC)CCCSC1 82259,C1(CNC(CCC=C(C)C)=O)CN(C(=O)COC2(C)CCOCC2)CC(C)(C)O1 82260,N1(C(CCCNC(C)=O)=O)CC=CC(NC(C2C=CC2C(=O)OC(C)(C)C)=O)C1 82261,c1(CC(=O)NCC2CN(C(c3csnc3Cl)=O)CC2O)nsc2ccccc12 82262,CC(C)C(CNC(=O)COCc1cccnc1)NC(=O)C(c1cnn(C)c1)C 82263,C1(C(N(CC(C)C)CC#C)=O)CCN(C(c2ccc(C)cc2)=O)C1C(C)(C)C 82264,C12(CC)CN(C(c3ccnn3CC(F)F)=O)C(CNC(C3CC(C)=NO3)=O)(C1)C2 82265,N1(C(CS)=O)CC(NC(=O)CCNC(C)(C)C)C(C)(C)C1.Cn1cc(C(=O)C=O)cn1 82266,N1(C(c2c(SC)cnn2C)=O)CC2(CCN2C(c2ccc(Cl)c(C)c2)=O)C1 82267,c1(C(N2C(CNC(=O)CCc3ccon3)CCCC2)=O)ccc2c(c1)B(O)OC2 82268,C(=O)(CCCCCNC(c1cc(Cl)n[nH]1)=O)NCCCS(C)(=O)=O 82269,CC1C(C(N2CCC(C(CO)NC(C3CCS3(=O)=O)=O)CC2)=O)CCN1C 82270,c1(CNC(CN(CCC)C)=O)ccccc1CNC(=O)COc1cccnc1Cl 82271,S(=O)(=O)(c1ccc(Br)c(C)c1C)N(c1c(C)n(C)nc1C(=O)O)Cc1ccccc1 82272,c1(C(C)=O)cn(C)nc1C(=O)NCC(C)(C)CN(C)C(C1C=CCC1)=O 82273,C1(CCOC)(NC(c2ccc(CC(C)C)s2)=O)CCN(C(=O)C=C(C)Cl)C1 82274,CC1C(C)N(C(C2CCn3nccc3C2)=O)CCN1C(C12CC(F)(C1)C2)=O 82275,c1(N(C)C)cccc(C(=O)NC2CCN(C(=O)Cc3csc(Cl)c3)C2C2CC2)n1 82276,N1(C(CCC=C)=O)CC(N=c2[nH]c(Cl)nc(C)c2[N+](=O)[O-])C(C)(C)C1 82277,c1(C(=O)NCCC(C)(C)OC)cnc(NC(=O)OC(C)(C)C)cc1C 82278,c1(C(=O)NC(C(=O)NCCOCCC)CC(C)C)cc2cnccc2[nH]1 82279,CC1(C(=O)NCC2CCCN(C(=O)CCSCc3ccccn3)C2)CC=CCO1 82280,C1(O)(C(=O)NCC2C(C(=O)NCC3C(OCC)CC3)C2)CCSCC1 82281,c1(C(=O)NC2C=CC(CNC(=O)CN3CSCC3=O)C2)cc2cc(F)ccc2o1 82282,c1(C(N(C(CNC(C(F)OC)=O)C)C)=O)cnc2c(cnn2C)c1O 82283,c1(C(=O)NC2CN(C(C3CCC(C)(CC)O3)=O)C2)cnc(C)c(C)c1 82284,N1(C(CC(C)(C)SC)=O)CC2CCN(C(C3CC(C)=NO3)=O)CC2C1 82285,C1(CNC(c2cc(C)ns2)=O)C2CCCC1N(C(c1ccc(C)c(C)n1)=O)C2 82286,Cc1c(C(=O)NC2CN(C(=O)CO)C3(CCC3)C2)ccc(Br)c1F 82287,C(=O)(C1=CC2(CCN(C(c3cc(C)c(C)o3)=O)C2)C1)NCc1cc(C)sc1 82288,CC1(C(N2CCN(C(=O)Cc3cnc(C4CC4)[nH]3)CC2)=O)CCOCC1 82289,n1(CC(=O)NC2CCN(S(C(C)C#N)(=O)=O)CC2)ccc2ccccc2c1=O 82290,N1(C(CN2CC(CC)C2)=O)CCC2(CC1)OCCC2NC(c1cc(OC)no1)=O 82291,c1(C(=O)NCC(C)NC(=O)C(C(C)O)NC(=O)C(C)(C)C)cc(F)c(F)cc1O 82292,N1(C(C)C(N)=O)CCCC(CCNC(C2(C)CCC2)=O)C1 82293,C1(NC(C(CC)=CCCC)=O)CN(C(c2scnc2CC)=O)CC1n1cccn1 82294,C1(C(=O)NCC2CCCOC2)(CNC(=O)CCc2cnoc2)CCCCC1 82295,c1(C(C)(F)F)ccc(=NCC2CCC(F)(F)CO2)[nH]c1 82296,c1(C(=O)NC(C(C)NC(c2nc(COC)sc2)=O)C(C)C)cc(=N)[nH]c(Cl)n1 82297,C1(CNC(CS(CC)=O)=O)CCC2CN(C(c3cn4ccccc4n3)=O)CC12 82298,c1(C(N2CCCC(CN(C(C(C)C3CC3)=O)C)C2)=O)coc2c1CSC2 82299,n1(CC(=O)NCCOC(C)=O)cc(CNC(C2CCCSC2)=O)nn1 82300,C(C1CCN(C(C2CN(C)C(=O)N2)=O)CC1)=CC(=O)NC1C(OC)C(O)C1 82301,c1(NC(=O)CC2NC(=O)NC2=O)ccc(O)nc1.CC12CC(C1)C(=O)N2 82302,O=C(N=c1cc(Cl)cn[nH]1)C1CCCN1C(=O)CCc1cnccn1 82303,C(=O)(CCC(=O)N(C)C)NC(CCN(C(C1(CC=C)CC1)=O)C)C 82304,N1(C(C(=O)NCCOCCOC)=O)CC(CNC(c2scnc2Cl)=O)C2CC12 82305,C(CCC(O)C(=O)N1CC(c2nc(=O)o[nH]2)C1)NC(C1(C)CCCCC1)=O 82306,c1(C(N2C(C(=O)NCc3ccsc3)CC(OC)C2)=O)ccc(C)cc1O 82307,C1(OC)(CNC(=O)CSC2CCOC2=O)CCN(C(c2nccn2C)=O)C1 82308,c1(CC(N2CCC(N(c3cnn(-c4ccccc4)c3)C)C2)=O)ccc(F)c(F)c1 82309,C1(NC(C(=C(C)C2CC2)F)=O)CC2CC(NC(c3cnc(C)c(N)c3)=O)C1C2 82310,c1(C(=O)NC(C2CCCC2)CNC(C2C(C)C2)=O)cc(C(F)(F)F)ncc1Cl 82311,C12(CC(=O)NC3C(CNC(=O)CCN4CCOC4=O)C3)CCC(CC1)C2 82312,CCC1=NOC(C(N2CC(NC(=O)COCc3cc(C)no3)C(C)C2)=O)C1 82313,C1(C(N2CC(C)C(NC(c3ccc4c[nH]nc4n3)=O)C2)=O)CCn2nccc2C1 82314,N1(C(C(COC)OC)=O)CCN(C(c2cc(=O)n(C)cn2)=O)CC1C1CCC1 82315,c1(C(N(C)CC)=O)ccc(NC(C)(C)C(C)(F)F)cc1 82316,Cn1c(C(N2CCCN(C(=O)CN3CCCC3CO)CC2)=O)cc2c1CCOC2 82317,Cn1nnc2c1C(C(=O)NCC(C1CCC1)NC(C1(C(F)(F)F)CC1)=O)CCC2 82318,CCCC(CC(C)C)C(=O)N1CC2CC(C)N(C(=O)CCC(C)CN(C)C)C2C1 82319,C(=O)(CC(C)CC(C)(C)C)N1C(CNC(C2=C(C)OCCC2)=O)CC(C)(C)C1 82320,C1(NC(=O)CC2CCCCCC2)COCCN(C(C2CC3C(C2)C3(F)F)=O)C1 82321,c1(CC(C)C)cn(CC2CN(CCC3CCCO3)C2)nn1 82322,c1(-c2cn(CCN(C(C3CN(C)CCO3)=O)CC)nn2)cc(Cl)cc(Cl)c1 82323,O=C(C1CCc2cccc(Cl)c21)NCC1(F)CC1 82324,N1(C(c2cnc3snnc3c2)=O)CCn2nc(CO)cc2C1.C12(CCC1)CC(=O)N2 82325,c1(C(C(=O)NC(C)(C)C)N(C(CCSC)C)C)nnc2n1CCN(C)C2=O 82326,C1(CNC(C2CC(OC)C(OC)C2)=O)CCCCN(C(c2c(N)cnn2C)=O)C1 82327,N#Cc1ccc(=NC(=O)NCCN2CCc3ccccc32)[nH]c1 82328,c1(C(=O)NC(CCCC)CNC(c2cn[nH]c2)=O)ccc(C(F)(F)F)nc1OC 82329,C1(C(=O)NCCN)COCCN(c2ccc(Cl)c(N3CCCC3)n2)C1 82330,C1(CCNC(CCc2ncn(C)c2)=O)CCCN(C(c2c(Cl)cnn2C)=O)C1 82331,Cc1cc2ncc(C(N3CCC(O)(CN(C(=O)C(C)CO)C)CC3)=O)cn2n1 82332,N1(C(C2=C(C)OCC2)=O)CC2CCC(C1)N(C(c1cc3c(cc1Cl)OCO3)=O)C2 82333,C(=O)(CCCCNC(C)=O)NC1CCC(CNC(CC2(C=C)CCC2)=O)C1 82334,c1(OC)ccc(S(=O)(=O)N2CCC(O)CC2C2CC2)cc1Cc1ccc(Br)cc1 82335,c1(-n2cc(C3(C)CCCN3CC3COC(=O)O3)nn2)cc(Cl)ccc1C(F)(F)F 82336,c1(C(=O)Nc2cn(CC)nc2C(=O)NC2CC2)cccc2c1OC(F)(F)O2 82337,CC(C)CC(CNC(c1cn(C)nn1)=O)C(=O)N1OC2CCC1C2 82338,C12(NC(C(C)CO)=O)CCC(CNC(=O)C(F)(F)c3nccs3)(C1)OC2 82339,O=C(CC(C(F)(F)F)NC(=O)CCC1CCC(=O)C1)NCC1CC1(F)F 82340,C123CCCC1CCN2C(=O)c1csc(n1)N(C)C3=O.c1(NC(COC)=O)ccco1 82341,O=C(CCS(=O)(=O)N1CCOCC1)N1CCN(C(c2cc(F)c[nH]2)=O)CC1 82342,c1(OC)cc(C(=O)N(C2CCN(C(=O)CC3CCC(=O)N3)C2)CCO)ncn1 82343,c1(CC)ccc(C(=O)NCC(C)(C)CN(C)C(C2CCCCNC2=O)=O)c(C)n1 82344,N1(C(CCC(C)C)=O)CCOC2(C1)CN(C(=O)CCCCN=[N+]=[N-])C2 82345,c1(C(=O)NCC2OCCN(C(c3n(CC)nnc3)=O)C2)nc(C)ccc1C 82346,c1(C(N2CC(O)(CN(C(c3c(C)nco3)=O)C)C2)=O)ccc2c(c1)OCC(=O)N2 82347,N1(C(Cc2cccc(OCCC)c2)=O)CC(C)C(C)(CNC(C2CC2(Cl)Cl)=O)C1 82348,c1(-n2cc(CC3CCN(C(COCC)=O)C3)nn2)nnccc1C 82349,CC1(C)COCC(NC(C2CCC(C)(F)CC2)=O)CN1 82350,C=CC(C)(O)C(=O)N1CCCC(CCNC(c2cnn(CC)c2C)=O)C1 82351,c1(SC)ncc(C(=O)NC2CCN(CC3CCCCC3)C2)s1 82352,Cc1cc(Br)cc(C)c1CNC1CC(C(=O)Nc2nnco2)C1 82353,CC(C)(C#N)CC(=O)N(c1ocnc1C(=O)NOCC(=O)OC)c1ccccc1 82354,C1(N2CCC(NC(c3cnsc3)=O)C2)CCN(C(=O)COC(F)(F)F)CC1 82355,N1(C(C(C)N(C(C)=O)C)=O)CCCCC1CCNC(c1occc1C)=O 82356,C(=O)(CS(=O)(=O)CCO)N(C1CN(C(CCCn2ncc(C)c2)=O)CC1(C)C)C 82357,C1(CC(=O)N(CCC(C)NC(c2c(C)noc2)=O)C)CC(=O)NC1=O 82358,c1(C(N2CC(CCC)C(C(=O)NC(c3nc(C)cs3)C)C2)=O)ccc(F)c(C)c1 82359,c1(NC(N(C)CCN(C2CCOC(c3ccccn3)C2)C)=O)ccc(Cl)c(Cl)c1 82360,C(C(=O)NCCC(C)C)(c1cscn1)OC.C12CC1NC(=O)CS2 82361,C1(C(=O)NC2CCCCC2)CCCCC1CO.c1(C(=O)NC)sccc1C 82362,n1(CC(=O)NC(CN(C(C2(CC)CC2(F)F)=O)C)C)nc(C)n(C)c1=O 82363,N1(C(=O)CCc2cncnc2)CCC(F)(C(=O)NCC2CN(C3CC3)C2)C1 82364,C(=O)(CC(C)C(=O)NC1CCC1C(=O)NCC(=O)OC(C)C)OC 82365,c1(C(N2CCC(F)(C(=O)NC(C3CCOCC3)C#C)C2)=O)ccc(C#N)cc1 82366,C(C(F)(F)C(=O)N1CC=CC(C(=O)NCCCCc2cnc[nH]2)C1)OC 82367,c1(C(=O)NC(CN(C(=O)C2=CCCC2C)CC)C)cc(C)ccc1O 82368,CC1=CCC(C)(C(=O)NC2CN(C(=O)CCN3C(=O)CCC3=O)CC2O)CC1 82369,N1(C(c2cc(C)c(C)nc2)=O)CC(NC(=O)CNC(N)=O)C(S(C)(=O)=O)C1 82370,CC(F)(F)C(C)(C)C(=O)N1C2CCC(C(=O)NC34CCCN(CCC3)C4)C1CC2 82371,CS(=O)(=O)C1CC2CCC(C1)N2N1CC2CC1(CO)COC2 82372,Cc1ccc(F)c(C(=O)N(C)CC2CCCN(C(C3CCC(C)O3)=O)C2)c1F 82373,Cc1cc(OC(c2nnc(NC(c3ccccc3F)=O)o2)C)ccn1 82374,c1(C(=O)NC(CCNC(C=CS(CC)(=O)=O)=O)C)cc2c(s1)CCCC2 82375,Cc1c(C(N2CCC(O)(C(C)CNC(c3cncnc3)=O)C2)=O)cnn1C1CC1 82376,C1(NC(C(c2cccc(Cl)c2)CC)=O)CCC(C)N(C(c2csc(=N)[nH]2)=O)C1 82377,C1(CNC(=O)Nc2nc3ccccc3[nH]2)COC2(CCCCC2)O1 82378,C1(C(N2C(c3n(C)ncc3)CCC2)=O)C(C)(C)CCCC1(C)C 82379,C1(NC(CCOCCC)=O)CCOCC1C(=O)N(CCOC)CC 82380,n1(CC(=O)NCC(CC)NC(c2ccc(N)cc2F)=O)cc(C)c2ccccc12 82381,C1(C(=O)OC)(CO)CCOCC1.C12CCN(C1)C(=O)c1c[nH]nc1CC(=O)NC2 82382,C(=O)(C(F)(F)C(F)F)N1CC=CC(C(=O)NCC2CCCS2)C1 82383,C(c1cnc(O)nc1O)=CC(=O)NCCC(C)NC(C1SCCS1)=O 82384,N1(C(CCCC(C)=O)=O)CCCC2(NC(=O)CCC3CCC(=O)N3)CC2C1 82385,c1(C(N(C(CNC(C(C)=C(CC)C)=O)C)C)=O)cc(OC)nc2ccccc12 82386,c1(-c2nnc(N(C3CCCOC3)CC)n2C)cccc(F)c1C 82387,c1(N2CC(F)CC(C(=O)NCc3cncc(Cl)n3)C2)ncc2cc(Br)ccc2n1 82388,N1(C(c2c(C)cn(C)c2)=O)CCC(CO)(CNC(=O)CN2CCC(C)(O)C2)CC1 82389,CCCCCC(O)C(C)C(=O)NCC1(CNC(c2ccnn2CCF)=O)CC1 82390,Cc1cc(C(F)(F)C(F)(F)F)ccc1C(=O)OCc1c(C(C)C)nnn1C 82391,C1(C(=O)NCCCOCCN(C(=O)CCc2cncs2)C)CC(F)(CF)C1 82392,C1(CNC(CC(=C)C)=O)CC(NC(c2cc(CC)n(CCO)n2)=O)C(O)C1 82393,c1(NC(C23N(C(C)=O)CC(C)(C2)C3)=O)cccc2c(O)nnc(O)c12 82394,c1(C(=O)NC2(CF)CCN(C(c3ncc(CC)nc3)=O)C2)cc2ccncc2s1 82395,N1(C(CN(C)C2CC2)=O)CCOC2(C1)CN(C(C1(C)CCC1)=O)C2 82396,C1(NC(C(CC)C2CCOCC2)=O)CC2(C1)CC(NC(C1CCCC(C)O1)=O)C2 82397,C(CN=c1[nH]c(=NCc2ccc(C3CC3)o2)[nH]c2c1COCC2)(C(F)F)C1CC1 82398,CON(CCO)C(=O)C1CCCCCN1C(C1COCC1(C)C)=O 82399,C1(CNC(C(C)CF)=O)CN(C(c2cc(C(F)F)on2)=O)CCC12CCC2 82400,C1(NC(C2C(C)OCCN2C(C2CS(=O)(=O)C2)=O)=O)CC2CC1CC2(C)O 82401,CC(C)C(C(=O)NC1CCN(C(c2cc(C(N)=O)co2)=O)C1C)n1cncn1 82402,C(c1cn[nH]c1)=C(C)C(=O)NC1CCC(N(C(=O)C(F)CC2CCOC2)C)C1 82403,c1(OC)ccc(C(C)CC(=O)NCC(O)CNC(=O)C(C)O)cc1 82404,C(c1cc[nH]c1)=CC(=O)NCC=CC(=O)NCC1CC1Cl 82405,C1(NC(C(CSC)OC)=O)COCCC1NC(C1CC(C)(C)C1)=O 82406,C#Cc1ccc(Br)c(C(=O)NC2CCC(C)(C)CC2CNC(=O)C=CC)c1 82407,C1(C(=O)NC(CC(C)NC(c2cccnn2)=O)C)CN2CCN1CC2 82408,c1(C(N2C(C)(CNC(CCCC#C)=O)CCC2)=O)ccc2n[nH]cc2c1F 82409,C1(C)(CC)CCCN(C(=O)C(c2cn(C)nn2)NC(=O)CCC(C)=O)CC1 82410,C(C)(N=c1[nH]c(Cl)ncc1Sc1nnnn1CC)c1ccn(CCC)n1 82411,Cc1cc2c[nH]nc2cc1C(=O)NCC(C)CN(C(=O)C=C1CCCCC1)C 82412,C1(C(N)=O)COC2(CCN(C(=O)Cc3cc(S(N)(=O)=O)co3)CC2)C1 82413,C1(NC(=O)C=CC2CCCO2)CCCCN(C(=O)Cc2sc(O)nc2O)C1 82414,c1(NCCCCOCC)cc(C)c(S(=O)(=O)N2CCCCC(C)(C)C2)cn1 82415,C1(C(=O)Nc2cccc(NC(CCC#C)=O)c2)Cc2ccccc2CN1C 82416,C12(NC(c3cncc(-c4cc(C(=O)NC)cc(F)c4)n3)=O)CC3CC(CC1C3)C2 82417,O(C=CC(=O)NCC(C)N(C)C(c1ccn(CC)n1)=O)CC 82418,C1(NC(CCCC=C)=O)CC2CC(NC(c3cnc(N(C)C)s3)=O)CC12 82419,Cc1ccc(F)cc1C(=O)NCCC(=O)NCCOC.C(C(C)ON)O 82420,C1(F)(C(=O)NCC(C)(CO)NC(C(CSC)OC)=O)CCCCCC1 82421,C1(NC(N(C(c2cccc(F)c2)C(=O)NCC2CC2)C)=O)CCC(C(N)=O)CC1 82422,C(CCCC(=O)NC1CC(=O)N(C(C)C)C1)NC(COCCSC)=O 82423,CC(O)C(C(F)(F)F)NC(=O)CNC(=O)Nc1ccc(C(F)(F)F)cc1F 82424,C1(C(=O)NCC2CCC2NC(C2(CC3CC3)CCC2)=O)CCC2(CC1)OCCO2 82425,CC(C)CC(C(=O)N1CCCC(O)(CO)C1)NC(=O)CN(C)C(=O)C1CC1 82426,N1(C(C(F)OC)=O)CC(O)(CNC(=O)CCCC2CC2)C1 82427,c1(C(N(C2CCN(C(=O)COCC3CCCO3)C2)C)=O)cccc(N=[N+]=[N-])c1 82428,C12(NC(c3cc(C#N)sc3)=O)CCN(C(c3cc(Cl)c[nH]3)=O)CC1C2 82429,Cc1c(C(N2CCN(C)CC2CNC(=O)C(O)C(F)(F)F)=O)cccc1CO 82430,C(=O)(CC(C)C(F)(F)F)NCCC(C)NC(=O)CSCc1ncc[nH]1 82431,C1(CNC(c2n(C)ncc2)=O)CCCC(NC(c2cn(CC3CC3)nn2)=O)C1 82432,C1(NC(COC2CCN(C)CC2)=O)CN(C(C2(Cl)CC2(F)F)=O)CC1(C)C 82433,N1(C(C(C2CCC2)OCC)=O)CC(N(C)C(C2CC(OC)C2)=O)C(O)C1 82434,c1(OCC(N2CC3C(NC(COCCC)=O)C3C2)=O)cc(Cl)ccc1C(C)C 82435,n1(CCOC)cc(C(=O)N(C2CCN(C(C3(c4cc[nH]n4)CC3)=O)C2)CC)nn1 82436,CCC(C)CCC(=O)NC(CCNC(C1(F)CCCC1)=O)C(C)C 82437,N1(C(C(C(C)(C)C)O)=O)CC2CC1CN(C(c1cc(F)cnc1O)=O)C2 82438,C(=O)(C1=C(NC(C2CCN2c2ncc(CC)s2)=O)CCCC1)OCC 82439,N1(C(CCc2ncc(C)[nH]2)=O)CCCC(NC(=O)CCC2OCCO2)C1C 82440,Cc1cc(C#N)ccc1C(=O)NC(C(=O)NCc1c[nH]nc1C(C)C)C1CC1 82441,CC(C)(CCCF)C(=O)NC1CCCCC1CC(=O)NCC1(C)CC2(CCC2)C1 82442,N1(C(CS(=O)(=O)NC)=O)CCC2C(C1)NC(=O)CN2C(=O)CN(C)C(=O)OC 82443,c1(CCNC(=O)NC2COC3(CC3)C2)nc2ccccc2[nH]1 82444,C(C(C(=O)NC1(C(F)(F)F)CCC1)C(C)(C)C)NC(CCC(C)(C)N(C)C)=O 82445,c1(OC)cc(C(N2CCOCC2CNC(C2C=CC=CC=C2)=O)=O)ccc1C 82446,C1(N=[N+]=[N-])(C(=O)Nc2c(C)cccc2F)CCN(C(c2csc(C)c2C)=O)C1 82447,C(=O)(C1CCCc2nn[nH]c21)N1CCN(C2CCN(c3nc(C)on3)C2)CC1 82448,C12(CNC(C=CC(C)(C)C)=O)CC(NC(c3cc(O)nc(O)n3)=O)(CCO1)C2 82449,N1(C(c2c(C)nc(C)[nH]2)=O)CC(N(C)C(C2CCCSC2)=O)C(C)(C)C1 82450,CCC1=C(C(=O)N2CCC(n3cc(-c4cc(F)ccc4OC)nn3)C2)CCCO1 82451,N1(C(C(CCCC)C)=O)CCC2(C1)CN(C(c1ccc(CCC(N)=O)cc1)=O)C2 82452,c1(C(=O)NCC(C)NC(c2nc(C(=O)NCC=C)sc2)=O)ccc(N)cc1C 82453,C=CCC(C)C(=O)N(CCCNC(c1ccc(OC)cn1)=O)C(C)C 82454,C(=O)(C(C)N1CC(C)C1)N(CC(=O)NCC=CC)CC1CC1 82455,CC1(C)CN(C2CCN(C3CCOCC3)C2=O)CCC1NC(=O)CC(F)(F)F 82456,C1(CN(C)C(c2cc(CO)n(C)n2)=O)CCN(C(=O)COCC2CCOC2)CC1 82457,CCC(CNC(=O)CCCc1nc(C(C)C)no1)(CC)NC(c1nc(O)sc1C)=O 82458,CC#CCC(C(=O)N1CC(c2ccccc2)C1)NC(C1CC2CCC2C1)=O 82459,C1(CC(=O)NCC(C)(C2CC2)OC)CCN(C(=O)Cc2csnn2)CC1 82460,C1(C(=O)NCCC(O)CNC(=O)C(C2CC2)C2CC2)CCCS1(=O)=O 82461,CCC(CSC)N=c1[nH]c2c(c(=NC3CCC4(CCC4)C3)[nH]1)SCC2 82462,N1(C(C(C)N(CCC)C(c2cc(Cl)no2)=O)=O)CCCCCC1C 82463,N1(C(C(C)NC(CC)=O)=O)CCN(C(=O)C=CCN(C)C)C(C(C)C)C1 82464,C(=O)(CC(F)(F)CC(=O)N1CCCC1(C)CNC(C1CCC(C)CC1)=O)OC 82465,C1(CCNC(c2cn(C)nc2C2CC2)=O)CN(C(=O)C=CCO)CCS1(=O)=O 82466,c1(C(CC)(C2CC2)NCC(C)(C)NC(C)=O)nnnn1C(C)C(=O)OC 82467,Cc1cccc(C(=O)NCC2(F)CCC(NC(=O)C(c3ccccc3Cl)C)C2)n1 82468,C12(NC(=O)CCc3nnc(C4CC4)o3)CCCN(C(c3cncc(F)c3)=O)CC1C2 82469,Cc1nccc(C(=O)NC(C)CC(C)NC(=O)C(C)Sc2ccccn2)c1C 82470,C12CN(CC13CC3)C(=O)C(=O)N2.c1(COC)cccc(NC(=O)CC(C)(C)C)c1 82471,N1(C(c2cccc(CC(C)C)c2)=O)CCC(C)(C(N2CCC(CO)C2)=O)CC1 82472,N#CC1(C(N2CCC(n3[nH]c(C4CC4)nc3=O)CC2)=O)CC12CCCC2 82473,N1(C(=O)C2=CCCSC2)CCC2CCN(C(c3occc3Cl)=O)C2C1 82474,n1(CC(=O)OC)ncc2ccc(NC(c3ccoc3C(=O)OC)=O)cc12 82475,C1(C(N(C)Cc2ccon2)=O)C2CC1N(C(c1csc(F)c1)=O)C2 82476,Cc1cc(Br)c(S(=O)(=O)NCC2(CO)CC23CCOCC3)cc1Br 82477,c1(NC(CC(C)(C)NC(C(C)=CC(C)(C)C)=O)=O)cnc(F)cc1C 82478,CCCC(C(=O)NCC1(F)CCN(C(c2ccc(OC)c(C)c2)=O)C1)S(N)(=O)=O 82479,CC(CC(=O)NCCc1ncnn1C)C(C)(C)NC(=O)C=CC1CC1 82480,N1(C(c2n(CC)cc(Cl)c2)=O)CCC(CNC(=O)COCC2CCCOC2)C1(C)C 82481,C(C(C)(C)CNC(=O)C(C1CCOC1)NC(c1ccc(Cl)s1)=O)SC 82482,C1(C(=O)NCC(CNC(CCC(CC)OC)=O)(C)O)CN(C)CCN(C)C1 82483,Cc1c(C(=O)NCC(C)(C)NC(C2CCCS2)=O)ccc(F)c1F 82484,C12(C(N3CC(N(OC)C)C3)=O)CCC(CC1)N(C(=O)CC(C)C(F)F)C2 82485,C1(CNC(=O)CNC(N)=O)CCC(C(=O)NC2CC2c2ccccc2)C1 82486,c1(NC(CC)CNC(c2cc(O)n(C)n2)=O)nc2c(cc1C#N)COCC2 82487,C(N=c1[nH]c(=NCCCCN(C)C)[nH]c2c1SCC2)C1(CO)C(C=C)C1 82488,Cc1cnc(C(=O)NCC2CCN(C(=O)C=CC3CCCC3)CC2)cc1C#N 82489,c1(NC(=O)NC(CC)C(=O)N2CCC2(C)C(=O)NC)cc(CO)cc(F)c1 82490,c1(C(=O)NC2CC3CC(NC(C4(SC)CC4)=O)C2C3)cnc2[nH]c(=N)sc2c1 82491,C#Cc1nc(C(=O)NCCN(CCC)C(C2CC2(F)F)=O)cs1 82492,C1(COCP(C)(C)=O)CCCCN1N1CCCC1CC1CC(C(=O)O)C1.CC=O 82493,C1(C(N(CCCNC(c2cc(CCC)[nH]n2)=O)C)=O)COCC(C)O1 82494,C1(CC(C)NC(C2CCS2(=O)=O)=O)CCN(C(=O)CCc2cccs2)CC1 82495,Cc1ccc(F)cc1C(=O)COC(C1(C#N)CC1(C)C)=O 82496,C1(CCC)CN(C(=O)C(C)N(C)C(C)=O)CCN1C(=O)C=C(C)c1cccnc1 82497,c1(OC)ccc(C)c(C(=O)NC2CC2CNC(=O)CC2CCC(C(N)=O)CC2)c1 82498,Cc1nonc1CC(=O)N(CCCn1cc(Cc2ccccc2)nn1)CC1CC1 82499,c1(CN2CCC(C(C)C(=O)N(c3cnns3)C(C)=O)CC2)cccc(-c2cnco2)c1 82500,Cc1cc(C(=O)NCC2(O)CCN(C(c3c[nH]cc(C)c3=O)=O)CC2)ccc1Cl 82501,N(C1CCCn2nccc21)C(c1c(CNC(c2nc(C)c(C)s2)=O)ccs1)=O 82502,CC1(C)CN(C(=O)C2=COCCC2)CCN(C(=O)C2=CCCOC2)C1 82503,c1(NC2CC(F)(CNC(c3c(C)nc(C(C)C)s3)=O)C2)ncccc1[N+](=O)[O-] 82504,c1(C(N2CC(OCCNC(C=CC=CCC)=O)C2)=O)cc(C#N)c(N)cc1O 82505,S(=O)(=O)(c1ccccc1N=[N+]=[N-])NC1CN(C(C)=O)C1 82506,N1(C(COC(CC)(C)C)=O)CC2CCN(C(=O)CC3(OC)CCOCC3)C(C2)C1 82507,C(=O)(CC(C)n1cccn1)NC1CC(CNC(CSC)=O)C1 82508,c1(SC(C(=O)NC(C)CCNC(=O)C(C)C2CC2)(C)C)nc2ccccc2[nH]1 82509,c1(C(=O)NC2CCCCN(C(C(CCC)OC)=O)C2)coc(=O)c2ccccc12 82510,C(=O)(CCCCCN(C)C(C1CC1[N+](=O)[O-])=O)N1CC(CCC#C)C1 82511,N1(C(c2cnsc2)=O)CCC2(CCCN(C(C3CC34CC(O)C4)=O)C2)C1 82512,c1(C(N(C(C)CCNC(c2cc(C(C)(C)C)n[nH]2)=O)C)=O)occ2c1CCC2 82513,CC(C(C)(C)C(=O)N1CCC1C1CCCC1)NC(=O)CC1C=CCC1 82514,C1(NC(CNS(CCCC)(=O)=O)=O)CCN(C(c2ccc(O)nn2)=O)CC1CC 82515,N1(C(CCC(C)N(C2CCCC2)C)=O)CCC2CCC(C1)N2CC(n1cncn1)Br 82516,C(=O)(C1=CCC(C)(C)CC1)NC(C1CN(C(c2cnncc2O)=O)CCO1)C 82517,c1(CNc2ccc3ncn(C)c3c2)cccc2c1OCCN(C(=O)OC(C)(C)C)C2 82518,N1(C(CCC#C)=O)CCCC1(CC=C)C(N1CCC(N2CCCC2)C1)=O 82519,c1(C(=O)NCCNC(=O)NCCc2csc(C3CCCO3)n2)ccccc1 82520,CCCCCCCCC(C)C(=O)N1CCN(C(c2ccc(C)cc2)=O)CC(O)C1 82521,C(CC(F)F)(C(=O)N1CC=CCO1)NC(c1ccc(CC#N)cc1)=O 82522,C(=O)(N1OC2CCC1CC2)c1c(C)oc(CNC(c2cccc(O)c2F)=O)n1 82523,c1(CCC(=O)NCCC2CCN(c3nc(C4CC4)ns3)C2)nc(O)n[nH]1 82524,N1(C(C2(CC)CCC2)=O)CCOC(C)(CNC(C2CC2C2CCC2)=O)C1 82525,C1(N(CC#C)C(C2COC(C)C2)=O)CCN(C(C2CC(N=[N+]=[N-])C2)=O)CC1 82526,CC1(C)CC(C)(C(N2CCN(C(N)=O)CC2)=O)CN1C(c1cscc1Cl)=O 82527,C(=O)(C1SCCc2ccccc21)N1CCN(C(C=C=C(C)C)=O)C(CCO)C1 82528,C(C)(CC(C)C(F)F)NC(CCCCNC(C1(CC)CC(C)(C)C1)=O)=O 82529,c1(NC(C2N(Cc3scc(C(=O)OC)n3)CCCC2)=O)c(F)c(F)nc(F)c1F 82530,Cc1ccc2[nH]c(C(N3CCCC(N(c4ncnc(=N)[nH]4)CCO)C3)=O)cc2c1C 82531,CCCC(CC(=O)NCCC(C(C)C)N(C)C)NC(c1ocnc1C1CC1)=O 82532,N1(C(C2C(CC)N(C(=O)C(C)OCC3CC3)CC2)=O)CCC(C)CC1C 82533,N1(C(c2ccc(CC)o2)=O)C(CNC(=O)COCc2ccnn2C)CC2CC12 82534,C1(NC(C2CN(C(C)=O)C2)=O)COC2(CCN(C(c3cc(Cl)ccc3N)=O)C2)C1 82535,N1(C(CCC(=O)N(C)C)=O)CCN(C(C2CCC(C(C)(C)O)CC2)=O)CC(O)C1 82536,Cc1ccc(NC(C)(C)CCc2nc[nH]n2)c([N+](=O)[O-])c1Br 82537,Cc1ccc(C=CC(=O)N(C2CCCCC2N(C(=O)C(F)F)C)C)c(C)c1 82538,C(C(C)NC(=O)C(C)(C)n1cc(Cl)cn1)(C(C)C)NC(Cn1ccc(C)n1)=O 82539,c1(OC)nccc(C(=O)NCC(C)N(C(=O)CC(C)CF)C)c1F 82540,C1(C(N2C(CC(=O)NC)CC2)=O)CCCN1C(=O)CCc1cnn[nH]1 82541,NC(C(=O)NNC(=O)c1ncon1)c1c(F)cccc1Cl 82542,c1(-c2n(C)ncn2)ccccc1C(=O)OCCOc1ccc(F)nc1 82543,c1(C(=O)NC2CC(C(=O)O)CN(C(C(CC(N)=O)O)=O)C2)n[nH]c2c1CCSC2 82544,O=C1NCC2(CO1)CN(C(c1ccc(Br)c(Cl)c1Cl)=O)C2 82545,N1(C(CC#N)=O)CCC(C2CN(C(c3cccc4nn[nH]c34)=O)C2)C1 82546,C1(NC(CCC#C)=O)CN(C(=O)CSc2nnc(-c3ccccc3)o2)CC1C 82547,c1(CC)ccc(C(=O)N(C2CCN(C(C3CCCC(CF)C3)=O)C2)C)cn1 82548,n1(CCCC)ncc(C(=O)NCC(CC(C)C)NC(c2cnnc(Cl)c2)=O)c1C 82549,C(CO)(CCC(C)C)NC(CONC(C1(SC)CCC1)=O)=O 82550,C(=O)(C1=CC(c2ccccc2)NC(=O)N1)N(CC(=O)O)Cc1cnccn1 82551,C(c1cn(C)cn1)=CC(=O)N(C1(C(=O)NCc2nc[nH]n2)CC1)C 82552,C1(NC(C)=O)CCCN(C(C2CC(O)(CNC(c3ccn(C(C)C)n3)=O)C2)=O)C1 82553,CC1(CCC(=O)NC2CC(C)(NC(c3csc(C4CC4)n3)=O)C2)CC1(F)F 82554,Cc1cc(Cl)cc(C(N2CCC2)=O)c1O.c1(C(N2CC2C)=O)ccc(F)c(Cl)c1 82555,C1(=CC(N2CC(O)(CN(C(=O)CCCn3cncn3)C)C2)=O)CCCCCC1(F)F 82556,C1(NC(C=CCN(CC)CC)=O)CC2CN(C(=O)CS(N)(=O)=O)CCN2C1=O 82557,c1(C(=O)OC(c2ccc(Br)s2)C)ccc(C2CCCC2)c(F)c1 82558,n1(CC)cc(S(=O)(=O)N2CCCC(CCNC(=O)CC3(O)CCC3)C2)cn1 82559,N1(CC)CC(NC(=O)NCc2ncn(CC)n2)CCC1=O 82560,N1(C(C(c2c(C)cccc2Br)NC(C(COCC)C)=O)=O)CCCCCC1CC 82561,C1(CNC(C(F)=CCC)=O)C2CN(C(=O)Cc3cc(C)nn3C)CC12 82562,C12(CNC(C(C)SC)=O)CN(C(=O)Cn3ncn4cccc4c3=O)CC1CCO2 82563,c1(C(N2CC3(CC(NC(=O)Cc4c[nH]nc4O)C3)C2)=O)cnn2c1OCC(O)C2 82564,Cc1cccn2cc(C(=O)NC3CC3NC(=O)CC(C)(C(F)F)N(C)C)cc12 82565,O=C1CC2(CCN(c3ccncc3S(=O)(=O)NC3CN4CCC3CC4)C2)C(=O)N1 82566,C1(CNC(C2(OC)CCSC2)=O)CCC(CN(C)C(c2ccoc2)=O)CC1 82567,N1(C(CSCC(=O)OC)=O)CC2(NC(=O)CN3CCOCC3)CC1CO2 82568,C1(N(C(Cc2cccc(OCC)n2)=O)C)CCN(C(=O)C(C)(C)CC)CC12CC2 82569,C1(C(=O)NC(C2(C)CC2)CO)COC2(C1)CN(C(=O)C=C1CCC1)C2 82570,C(C(C)(O)C(F)(F)F)NC(C1(F)CCN(C(COCCCOC)=O)C1)=O 82571,CC1COCCC1N=c1[nH]c2c(c(=NCc3cccc4cc[nH]c34)[nH]1)CSC2 82572,C(=O)(C(C)(C)CNS(C)(=O)=O)N1C(CNC(C(C)NC(=O)C(C)(C)C)=O)CCC1 82573,C12(NC(Cc3c(C)n[nH]c3)=O)CN(C(=O)C(C)(C)CN(C)C)CC1CS(=O)(=O)C2 82574,C1(CN(C(c2ccc(C)n2C)=O)C)CN(C(=O)CC2CC=CCN2C)CC12CC2 82575,c1(SC)cc(C(=O)NCC2(CCNC(=O)CCCCn3ccnn3)CC2)c(C)o1 82576,c1(C(N(CCN(C(C)C)C(c2cnn(C3CCOC3)n2)=O)C)=O)cnnn1C 82577,C=CCC(C)(C(=O)NC1CCN(C(=O)Cn2nc(C)c(Cl)c2C)C(C)C1)N(C)C 82578,Cc1[nH]c(C)c(C(=O)NCC2CC2NC(c2csc(C(F)F)c2)=O)c1C 82579,C1(NC(c2cn(CCOC)nc2)=O)CN(C(c2c[nH]nc2C2CC2)=O)CC1C 82580,c1(CNC(C(c2ccccc2F)C)=O)cnn2c1CN(C(=O)CCS(C)=O)CC2 82581,C1(NC(c2cscn2)=O)CN(C(=O)COc2cccc(SC(F)F)c2)CC1O 82582,CC(=Cn1ccnn1)C(=O)N1CCCC(NC(c2coc3c2CSC3)=O)C1C 82583,c1(C(=O)NC2C(NC(c3c(C)nncc3)=O)COC2)cc2ccccc2[nH]1 82584,N1(CC)CCCC(NC(=O)CC2CCN2C(C2CCCN2C(=O)OC)=O)C1 82585,C(C1CN(C(=O)CC(C)=C(C)C)CC1C(=O)NCCC)=CC 82586,C1(C(N2CC=C(CNC(c3c(OC)scc3)=O)CC2)=O)CCCN(S(N)(=O)=O)C1 82587,CCCC(O)CC(=O)NC(C1(O)CCN(C(C2CSCN2C)=O)CC1)C 82588,C1(C(=O)NC(C)C(C)NC(=O)Cn2ncc(C#N)c2N)COCCN1C=O 82589,c1(C(=O)NCCC2OCCN(C(C3(C#C)CC3)=O)C2)cc(O)ncc1Br 82590,N1(C(C2N(CC#C)CCC2)=O)CC(NC(c2cc(N)cnc2C)=O)C(C)(C)C1 82591,c1(C(=O)NCCCCN(C(CC(CC)CC)=O)C)ccn2ncccc12 82592,C1(CNC(=O)C(O)C2CCCC2)CCCN1c1nnco1 82593,N1(C(C(c2c(C)cc(C)cc2C)NC(=O)NC)=O)CCCC2(CO)CCCCC12 82594,C1(SCC)CN(C(=O)C=NOC)CC1NC(=O)C=CCn1cncn1 82595,C1(N(C(C(c2scc(C)n2)C)=O)C)CCCCC1N(C)C(c1ccc(O)cn1)=O 82596,C(=O)(C1Cc2ccccc21)NC1C=CCN(C(CC2CCN(C)CC2)=O)C1 82597,Cc1nc(NCc2cncc(Br)c2)cc(=NCC(C)N2CCCCC2)[nH]1 82598,C(=O)(C1=CCCCO1)NCCCC1(NC(c2snc(C)c2Br)=O)CC1 82599,C1(NC(CCCC=C)=O)CN(C(c2ccc(F)cc2)=O)CC1C=C 82600,C1(NC(CC(C)O)=O)CCC(C(=O)Nc2cccc(CS(N)(=O)=O)c2)OC1 82601,c1(OC)cc([N+](=O)[O-])ccc1C(=O)NCC1CC(NC(c2ccccc2O)=O)C1 82602,C1(CCC(=O)N(C2CCCCC2)Cc2ccc(F)cc2)CCC(C(F)(F)F)CC1 82603,C(=O)(CCC(=O)N1CCCCC1CNC(=O)CC1(O)CCCCC1)N(CC)CC 82604,c1(C(N2CCC(NC(c3c(C)nns3)=O)CC2)=O)cc([N+](=O)[O-])c(C)s1 82605,N1(C(CCN(CC=C)C(C2CCC2OC)=O)=O)CCCC(C2CC2)CC1 82606,C1(NC(c2cn(C(C)(C)C)nc2)=O)CCC(O)CN(C(C2CCCN2C=O)=O)C1 82607,Cc1cc(Br)c(S(N)(=O)=O)cc1C(N1CCC(CO)C(C2CC2)C1)=O 82608,c1(C(N2CCC3CC23C)C(=O)NC(CC)(C)C)ccc(F)cn1 82609,C1(C(=O)NOCCN2CCCC2=O)(NC(C=CC(=O)N(C)C)=O)CC(F)C1 82610,C(C(C)(C)C(=O)NC(C)CCNC(=O)CN1C(=O)CNC1=O)SC 82611,C1(OC)CN(C(c2ccn(C)c2C)=O)CC1NC(C1CC2CC1C2)=O 82612,c1(C(N(C)C)=O)cccc(C(N2CCC(C3CC(N)CCO3)CC2)=O)n1 82613,c1(C(N(CCNC(C(CC(C)C)NC(C)=O)=O)C2CC2)=O)ccn(C)c(=O)c1O 82614,Cn1c(C(=O)NCCC2CN(C(C3CCCCC3C(F)(F)F)=O)C2)cccc1=O 82615,C1(CC(=O)NCC(C)N(C(CCOCC)=O)C)CCCN1C(C)C 82616,c1(CC(=O)NC2CN(C(c3c(C)nc(C4CC4)o3)=O)C(C)C2)nc([N+](=O)[O-])n[nH]1 82617,C(c1cncs1)=CC(=O)N(CCC(=O)NCC(C)(C)OCC)CCO 82618,CC1CN(C(=O)CC2CC2)CC1NC(C1CC1c1cccs1)=O 82619,N1(C(c2c(Br)cn(C)n2)=O)CCOC2(CCN(C(C3C4C=CSC34)=O)CC2)C1 82620,C(=O)(C#CC1(C)CC1)N(C1CCN(C(C(CC)COC)=O)C1)CCO 82621,c1(CC(N2CC(F)CC(NC(=O)C3=CCSC3)C2)=O)cncc2ccccc12 82622,Cc1cc(CC(=O)N(CCCCN(C(=O)CCOC2CCC2)C)C)cc(C)c1 82623,C1(NC(C(=O)NC(C2CCCCO2)CC)=O)CCCN(CCOC)C1 82624,C1(C)(NC(C(C=C)NC(=O)OC(C)(C)C)=O)CCCC1NC(=O)C(C)CC 82625,CC1CN(C(c2cncs2)=O)CC1CCNC(C1CCCN1C)=O 82626,n1(CCC(=O)NCCc2ccc(CNC(C(C)=CC)=O)cc2)ccc(O)nc1=O 82627,C(C(C)(C)C1=CCCC1)NC(C=C(CNC(C1(NC(C)=O)CCCCC1)=O)C)=O 82628,C(=O)(CP(=O)(C(C)C)C(C)C)N1C2C(NC(c3c(C)cnn3C)=O)CC(C2)C1 82629,c1(N2CCC(CC(C)NC(c3cscn3)=O)CC2)ccn2nccc2n1 82630,C12(C(=O)NCc3cccnc3C(F)(F)F)CC1CN(Cc1nc(C)sc1)C2 82631,n1(C(C)C)ncc2c(N3CCC(NC(c4csc(S)n4)=O)C3(C)C)nc(Cl)nc12 82632,c1(SC)cc(C(=O)NC2CN(C(c3cc(C(C)C)oc3C)=O)C2)c(C)o1 82633,N1(C(C(c2ccccc2)NC(CCCCC=CC)=O)=O)CCOC(C)(C)CC1 82634,N1(C(C(C)Cc2ccc(Cl)cc2)=O)CC(NC(C23CC4CC2C3C4)=O)CC(C)C1 82635,CC(CC(N)=O)N=c1[nH]c(C(F)(F)F)c(-c2ccccc2)s1 82636,N1(C(CC(=O)NC)=O)CCOC2(CCN(C(=O)CCc3cccnc3Cl)CC2)C1 82637,N1(Cc2c(C)ccnc2)CCC(NC(C2(F)CCC2)=O)CC(C)(C)C1 82638,N1(C(C=Cc2n(C)ccc2)=O)CCCC(O)(CNC(c2scnc2C2CC2)=O)C1 82639,C1(CNC(=O)CCSc2ccccc2)CCC12CN(C(=O)C1=COCC1)C2 82640,N1(C(C=C(C)C(=O)O)=O)CCC2CN(C(C3CCC3)=O)CCC12 82641,N1(C(C2CCC(C(C)C)CC2)=O)CCN(C(C2CC3(C2)CC32CC2)=O)C(C)C1 82642,n1(CCC)ncc(Br)c1C(=O)NCCN(C(=O)C(C)N1CC(C)C1)C 82643,N1(C(C2C(CC)C2)=O)CCOC2(CCN(C(C3CCC4(CC3)CC4(F)F)=O)CC2)C1 82644,c1(NC(C(C)C)=O)cccc(NC(=O)N(CCCCCCO)C)c1 82645,Cc1ccc(C(N2CCC2CNC(c2cccc(CCC#N)c2)=O)=O)cc1 82646,n1(C(C)CC(=O)NCC2CC2NC(C2CCC2)=O)cnc2ccccc12 82647,c1(C(=O)NC2CC(F)(CNC(C3CC(OC)(OC)C3)=O)C2)nc[nH]c2nccc1-2 82648,C1(O)(CNC(c2ccc(OCC(F)(F)F)nc2)=O)CCN(C(=O)C2CC2)CC1 82649,N1(C(c2n(CC)ncn2)=O)CCCOC(CNC(C2(OC)CCS(=O)(=O)C2)=O)C1 82650,C(C(C)C(=O)OC)N(CCC(C)C)C(=O)C=CC=C(Cl)Cl 82651,N1(C(c2c(C)nn[nH]2)=O)CC2C=CC1C(C(=O)NC(c1ncc(F)cn1)C)C2 82652,CC(O)C(C(N)=O)NC(=O)NC1CC2CC2N1C(C1CCCCC1)=O 82653,C(=O)(C(O)CC[S+](C)C)N(C)C(C(C)CN(C(=O)C=CCCc1ccccc1)C)=O 82654,C(=O)(C(C)(C)C)NC(C)C(=O)NCC1C=CCN1C(c1ncoc1C1CC1)=O 82655,C(=O)(C(Cc1ccco1)C(=O)NC1CC(CC(=O)NC2CCOC2)C1)OC 82656,N1(C(C(C)=CC2CC2)=O)CCC(C)(C)C(NC(=O)CCC2CCCN2C)C1 82657,CC(Cc1ccccc1)C(c1nnnn1C)Nc1cn(CCOCCO)cn1 82658,c1(NCCC(C(C)C)OCC)ncccc1S(=O)(=O)N(C)CCSC 82659,C1(NC(c2n(CC)ncc2)=O)CCC2CN(c3ncc(C)c(C)n3)CCC2C1 82660,c1(OC)cn(CC(=O)NC2CC2NC(=O)CCCC(N)=O)c(C)cc1=O 82661,C1(OC)CC(C(=O)N(C)Cc2cnc(C)s2)N(C(=O)CCn2ccnn2)C1 82662,C(=O)(C1=CCC(F)(F)CC1)NCC(CC)NC(c1cccc(O)n1)=O 82663,N1(C(C(Cc2c(C)cccc2)C)=O)CC2CCN(C(C3CCC3)=O)C2C1 82664,N1(C(=O)C(C2CC(F)(F)C2)O)CCOCC(CNC(C2(CO)CC2)=O)C1 82665,N1(C(CC(COC)C)=O)CC2CCCC(NC(c3coc(C4CCC4)n3)=O)C2C1 82666,N(S(=O)(=O)N1CCCC1C)(C1CCCCC1)Cc1c(CC)cccc1 82667,c1(C(=O)NCC(CC)NC(c2cnc(O)nc2O)=O)ncc(Cl)cc1Cl 82668,c1(C(=O)OC)nccc2cc(NC(=O)C(=O)NCc3ccc(SC)cc3)ccc12 82669,C(=O)(CS(=O)(=O)NC)N1CC(O)(C(C(=O)N(CCOC)CC)F)C1 82670,N1(C(C(c2cccs2)NC(CCCNC(C)=O)=O)=O)CCn2ncc(C)c2C1 82671,CC(C(C)(O)C(=O)NCC(C1CC1)N(C)C(c1cnns1)=O)c1ccccc1 82672,CCC(C)C(CC(=O)NCCc1cccc(C)n1)NC(=O)C1=C(C)CCOC1 82673,Cc1cc(C)c(C(=O)NCC2CCCN2C(C2CC(C(C)C)C2)=O)o1 82674,C1(C)(C(=O)NCC(C)(O)C2(C)CC2)CC(O)CN1C(C1C2CCC(F)(F)C12)=O 82675,Cc1cccc2cccc(NC(C3(O)CCN(C(C4(C)CC4)=O)C3)=O)c12 82676,CC(C)C(C)C(C)CC(=O)NCCCN(C)C(c1ccc(CCN(C)C)cc1)=O 82677,C1(NC(Cc2c(C(C)C)con2)=O)CCCN(C(=O)COCC2CCCCO2)C1 82678,C1(CNC(C(C)SC(F)(F)F)=O)CN(C(=O)CC2CSC2)CCC1(F)F 82679,S(=O)(=O)(c1c[nH]c2ccccc12)N1C(C(=O)Nc2cccc(CO)c2)CCC1 82680,C12(NC(C(Br)=C(C)C)=O)CCCC1CN(C(c1[nH]c(C)nc1C)=O)C2 82681,c1(OC)ccc(Cc2noc(-c3c[nH]nc3-c3cnn(C)c3)n2)cc1 82682,Cc1n[nH]c2ncnc(NC(C3CCCN3C(c3cncc(Cl)c3)=O)=O)c12 82683,S(=O)(=O)(c1ccc2oc(O)nc2c1)N1CC(NC(c2ccn(C)c2)=O)C1 82684,CN1CCCC(CNC(C23CC(CN2C(=O)C=Cc2cncn2C)C3)=O)C1 82685,C(=O)(C(F)C(C)(F)F)NCC1(C(=O)NCC2CC(C)C2)CC=CC1 82686,C1(C(N(CCN(C(C2CCCN(C)C2)=O)C)C)=O)CN=C2N=CNN2C1 82687,C1(C(=O)NCC2(NC(C3CC4(C3)CC4F)=O)CCOC2)(CC)CCC(F)(F)CC1 82688,C(=O)(C1CCCc2sccc21)N1CC(OCCNC(=O)CN2CCOCC2)C1 82689,N1(C(C(C)=C2CCC2)=O)CCN(C(=O)CCC(C)C)C(C2CCC2)C1 82690,c1(C(N2CCC(CNC(=O)C(O)C3CCCC3)C(O)C2)=O)nccc2cc[nH]c12 82691,C=CCC(CC)C(=O)N1CC2CC(NC(=O)C=Cc3ccnn3C)C1C2 82692,C1(C(=O)NCCN(C)C(c2cn(C3CC3)cn2)=O)CC1C1CC(F)(F)C1 82693,c1(OC)cc(C(=O)NC(C2CCCN(C(c3cnnn3C)=O)C2)C)n(C)n1 82694,c1(C(N2CCC(N(C(=O)CC3COC4CC3C4)CCC)C2)=O)occ2c1CCC2 82695,c1(OCC)nc(C)ccc1C(=O)NCC1(OC)CN(C(C2(C)CC=CC2)=O)C1 82696,C(c1cccc(Cl)c1)=CC(=O)NC1CCCC1NC(C1CCCC12CC2)=O 82697,N1(C(C(n2cc(C)nc2)(C)C)=O)CC(C(=O)NCC2CCC=CCC2)CCC1C 82698,Cc1cc(NC(C2CC3CC3N2C(=O)CCc2ccc(F)nc2)=O)c(F)cc1Br 82699,CC(CS(C)(=O)=O)C(=O)N1CCN(C(c2cnc(-c3ncccn3)s2)=O)CC1 82700,Cc1cc(CC(N2CCC(=CCNC(=O)C(C)(C)C(C)O)CC2)=O)ccc1F 82701,C1(NC(c2cc(CC)sc2)=O)CC(NC(C2(C#N)CCCCC2)=O)C12CCC2 82702,N1(C(c2c(-c3cn(C)nc3)c[nH]c2)=O)CC2CN(C(=O)CNC=O)CC2C1CO 82703,C1(OC)CN(C(c2cnc(Cl)[nH]2)=O)CC1NC(=O)C(F)(F)c1ccncc1 82704,c1(CCC(=O)NC(C)CC2CCCCN2C)c(CCCCF)[nH]c2ccccc12 82705,O=C(C1=CCC(NC(c2ccncc2F)=O)CO1)N1CC(O)CO1 82706,CC#CCCC(=O)NC(CNC(=O)CCCNC(c1ccco1)=O)CC(C)C 82707,C1(O)(CN(C)C(C2(C)CSC2)=O)CCN(C(=O)CCC2CCCCN2C)C1 82708,n1(CC(=O)N(CCC(=O)NCC2CCOC2C)CC=C)c(C)ccc1C 82709,c1(C(N(CCNC(CC2(COC)CC2)=O)CC2CC2)=O)nc[nH]c1C(C)(C)C 82710,c1(NC(CN2CCC(=O)CC2c2ccccc2)=O)cc(Cl)c(Cl)c(Cl)c1 82711,c1(C(=O)NC(C)CC(=O)NCC2CCC3(CC3)C2)cnc(CO)nc1 82712,CN1CCN(C(=O)C#CC2CCC2)C(C(=O)NCC(O)CCC2CC2)C1 82713,n1(CCC)ncc(C(=O)NCC(O)CNC(=O)C=Cc2cc(C)no2)c1C1CC1 82714,C(C(=O)NCC1CCCO1)(C(C)CC)NC(C(C=C)C)=O 82715,c1(C(=O)NC(C)C(N)=O)ccc(-c2cccnc2F)nn1 82716,N1(C(c2c(=O)ccn(C)c2)=O)CCC2(CCN(C(c3ccc(C(F)F)s3)=O)C2)C1 82717,CC(C)C(O)CC(=O)N1CC=C(C(=O)N2CCC(c3cnn[nH]3)C2)C1 82718,c1(N2CCC(C)C2)nc(N2CCC(CC#N)C2)nc2c1ncn2C 82719,CC1(C)C2CN(C(C3CC34CC(NC(c3csnc3Cl)=O)C4)=O)CC12 82720,C1(NC(C2=C(C)CC2)=O)C2CC3CN(C(c4cc(C)nc(C)c4)=O)C1C3C2 82721,N1(C(C2=C(C)CCC2)=O)CCCC2(CCN(C(=O)CC(O)CC(C)(C)C)C2)C1 82722,C#Cc1ccc(CC(=O)NCC2(O)CN(C(c3cncc(Br)c3C)=O)C2)cc1 82723,c1(C(c2n(C(CC)(C)C)nnn2)NC2CCCSC2)c(I)cnn1C 82724,N1(C(CC2N(C(C(CC#C)C3CC3)=O)CC2)=O)Cc2ccccc2C1 82725,CC(CCC(=O)N(C)CC1C2CN(C(=O)C=C3CCC3)CC12)N(C)C 82726,C1(N(C2CCCCC2O)C(C2C(c3ccc(OC)cc3)C2)=O)CCNCCC1C 82727,c1(COC)cccc(C(=O)N(CCCNC(C2(C)COCCO2)=O)C(C)C)c1C 82728,N1(C(c2c(Cl)cn(CC)n2)=O)CC2CCCN(C(C3CCCS(=O)(=O)C3)=O)C2C1 82729,C(CC(C)(C)C)(C(=O)N1CCC(CCC(=O)N2CC(n3ccnn3)C2)C1)OC 82730,c1(CC)cccc(C(=O)NC(COC)C(=O)NCC2(C)CC(C)=NO2)c1 82731,N1(C(c2cc(C)no2)C(=O)Nc2ccccc2Cl)CCC2(CCCOC2)CC1 82732,C1(O)(CNC(C(C(C)C)N2CCCC2=O)=O)CCCN(C(c2csc(=N)[nH]2)=O)C1 82733,C1(NC(C(C(CC)C)O)=O)CN(C(c2ncc[nH]c2=O)=O)CCC1(C)C 82734,C1(CN2C(=O)CN(CCC(COC)C)C2=O)COc2ccccc2C1 82735,N1(C(C(CCOC)C)=O)CCN(C(c2sccc2Cl)=O)CC(C)(F)C1 82736,Cc1nn(C)c(C)c1CN(CCO)C(C1(C)CC1(F)F)=O 82737,C1(C(=O)NCC(COC)(O)CO)C2CC3C(C2NC(C2CCCC(=O)CC2)=O)C13 82738,N(C1CCCn2nccc21)c1c(C)c(NCc2nnc3n2CCC3)ncn1 82739,c1(NC(c2cn[nH]c2)C)nccc(=NCc2cccc(Br)c2F)[nH]1 82740,c1(OC)c(C(N2CC(C)(NC(C3CC(C(C)C)=NO3)=O)C2)=O)[nH]c2ccccc12 82741,CN1CC(C)(C(=O)NC2CC(CO)N(C(c3cc4[nH]ccc4s3)=O)C2)CCC1=O 82742,CC1(C(=O)NC(c2ccnn2C2CN(CCCCCC(C)(C)C)C2)=O)CC2(CC2)C1 82743,C1(NC(C2CC(OC)C2)=O)CCC(C)N(C(c2cnc(C)c(N)c2)=O)C1 82744,C#CCC(O)C(=O)NCC1CC(F)(CNC(=O)C=CC(C)C)C1 82745,C1(NC(C(CC)(C)C)=O)CCCN(C(=O)Cn2ccc(Br)cc2=O)CC1F 82746,c1(C(=O)NC2(CCCNC(c3cnc(C)s3)=O)CC2)ccc[n+]([O-])c1 82747,c1(CC(=O)NC2C(C(=O)NC(c3nn[nH]n3)CC)COC2)ccc(C)nc1 82748,C1(C(C)C)C(=O)N1.N1(C2CC(n3cc(-c4c(C)ocn4)nn3)C2)CCS(=O)CC1 82749,C1(NC(C(C2CCCCC2)OC)=O)CN(C(C2C3CC4C(C3)C24)=O)CC1OC 82750,C#CCCCC(C)C(=O)N1CCCCC1C(N1CCCC(CCCO)C1)=O 82751,c1(C(N)=O)c[nH]c(C(N2CC(O)(CNC(=O)CCC3CCC3)C2)=O)c1 82752,c1(CC(=O)NCCC2CCN(C(C34CC(C3)S(=O)(=O)C4)=O)C2)cccc(O)c1F 82753,C1(NC(COCCOCC)=O)CC2CN(C(C3C(c4ccccc4)C3C)=O)CC12 82754,c1(C(=O)NCCCCNC(Cn2c(C)nc(C)n2)=O)cc(C)c(O)c(N)c1 82755,N1(C(C2(N(C(c3n(CCC)ccc3)=O)C3CC3)CCC2)=O)CCCN(CC)C(=O)C1 82756,n1(CCOC)cc(C(=O)NC2CCC(N(C)C(c3cnns3)=O)C2)c(=O)cc1C 82757,Cc1c(C(N2CC(N(C)C(c3[nH]nnc3C3CC3)=O)C(O)C2)=O)ccc(F)c1F 82758,N1(C(C2CC(N(C)C)C2)=O)CC=C(CNC(=O)CCC2NC(=O)NC2=O)CC1 82759,C(CCN=C(N)NC1CCCSC1)=C(C)C.C(C)=O 82760,C(CCCCCCCCCCn1cc(CO)nn1)NC(c1scc2c1CCCC2)=O 82761,N1(C(C(C)=CC2CC2)=O)CC2CCCC(N(C)C(c3ccc(Cl)cn3)=O)C2C1 82762,C(C)(C)(CCC(=O)N1CCCC(C(N2CCSC(C)(C)C2)=O)CC1)N(C)C 82763,CCC(COC)C(=O)N1CC(CNC(=O)C(C)NS(=O)(=O)Cc2ccccc2)C1 82764,C1(NC(C2CCCO2)=O)COC2(C1)CN(C(C1CCCCC1)=O)C2 82765,CCCCC(O)C(C)C(=O)NCCC1CSCCN1C(=O)CC(C)(C)C 82766,C(=O)(CC(C)(O)C(F)(F)F)N1CC2C(CNC(C(C)(C)N(C)C)=O)C2C1 82767,N1(C(c2cnc(CC)s2)=O)CCC2(CCC2NC(c2ccc(Br)o2)=O)CC1 82768,C1(C(=O)NCC(CC)(C)Cl)CCC(C)N1C(c1cnn(C)c1)=O 82769,c1(C(=O)NCCOc2cccc(C(=O)OC)c2C)cc2ccc(Cl)cc2cn1 82770,Cc1ccc(OCC(N2CCCC(Nc3ccccc3)C2)=O)c(C)c1 82771,CCC(CC(F)(F)F)C(=O)NCC(CC)NC(c1ccccc1CCN(C)C)=O 82772,CC(C)C(C(=O)N1CCC(NC(C2(F)CCCC2)=O)C1)c1ccccc1 82773,Cc1cc(NC(C2C3CC3CN2C(=O)CCCCC#N)=O)ccc1Cl 82774,C1(CC(N2CCC(CC(C)NC(=O)C(CO)N(C)C)CC2)=O)CCCCCCC1 82775,S=C(Sc1ccc(CN2CCCCO2)cc1)c1ccccc1 82776,N1(C(c2cc(OC)cc(Cl)c2)=O)CCC2CC2(NC(c2csc(S)n2)=O)CC1 82777,N1(C(C2C(C)OCCO2)=O)CC2(CC(CC(=O)NC3CNC(=O)C3)C2)C1 82778,C1(NC(C=CCN(CC)CC)=O)CCCC1NC(C1CCOC1C(C)C)=O 82779,C1(C(=O)NC(C)Cc2cccs2)(CC)CCN(C(=O)CC2CCCSC2)C1 82780,C1(c2cn(Cc3cnoc3)nn2)(NC(C2CC=CCO2)=O)CCCOC1 82781,c1(CC)nc(C(=O)NCC2(COC)CCCN2C(c2scnc2Cl)=O)c(C)o1 82782,C1(CCn2cc(CN)nn2)C2CN(C(c3ccc(N(C)C)nc3)=O)CC12 82783,N1(C(CC2(C)CC2(F)F)=O)CCC2(CC1)CCN(C(c1ccnn1CC#N)=O)C2 82784,C1(C(=O)NC(C2(O)CN(C(c3ncc(Cl)nc3Cl)=O)C2)C)CC12CCSCC2 82785,C(CC(=O)N(C(C)CNC(c1nnn(C)c1C(F)F)=O)C)(C1=CCCC1)OCC 82786,C1(CNC(C2CC(C)OC2C)=O)CCN(C(C2CCOC2C)=O)C12CC2 82787,c1(C(=O)NCC2CC(NC(C3CCC(C)(C)O3)=O)C2)ccc2c(c1)NCCC2 82788,c1(COC(C)=O)cc(F)c(S(=O)(=O)N2CCCCC2c2nccn2C)c(F)c1Cl 82789,n1(C(COC)CO)cnc2c(N3CCC(Cc4ccccc4)CC3C)ncnc12 82790,c1(CC)cc(C(=O)N(CC(C)NC(=O)CCC(F)F)C)nn1C 82791,c1(C(N(C(c2ccncc2)CC)CC)=O)cc(Cl)c(Br)c(Cl)c1 82792,N1(C(c2c(C)scn2)=O)CC(F)CC1CNC(=O)Cc1csc(NC=O)n1 82793,c1(C(=O)NC2CCN(C(c3nc(C)c(C)s3)=O)C2)cc2c(C)cccn2n1 82794,C1(CNC(CCSCC)=O)(NC(=O)C=Cc2cccnc2C)CC2CCC1CC2 82795,C12(C(N(CC(C)(C)NC(=O)C=Cc3ccccn3)C)=O)CC1COC2(C)C 82796,N1(C(c2c(C#C)c[nH]n2)=O)CC2CCCC(NC(c3ccc(C)nc3C)=O)C2C1 82797,c1(C(=O)OC)ccc(NC2COC(CO)C2)c(C)c1 82798,Cc1c(C(=O)NC2CCC(CCNC(c3nnc(C(C)(C)C)s3)=O)C2)cnn1C 82799,Cn1ncc(C(=O)NCCCN(C(=O)CC2CC(=O)C2)C2CC2)n1 82800,CCCCC(CNC(=O)C(CC(C)C)NC(=O)CCCNC(=O)OC)CC 82801,N1(C(c2cc(OC)cc(Cl)c2)=O)CCCC(C2CCN(Cc3cnsn3)C2)C1 82802,C1(C#CC(=O)NCC2(C(C)(C)O)CN(C(=O)Cc3ccc(Cl)cc3)C2)(CC)CC1 82803,c1(CC(N2CC(CCCNC(C(C)C(F)F)=O)OCC2)=O)ccc2c(c1)OCO2 82804,c1(C(C)NC(c2scc(C(C)=O)c2)=O)ccc(CNC(c2ccsc2)=O)cc1 82805,N1(C(CC2C(C)(C)CC2)=O)CCCC2CN(C(=O)C=Cc3cccs3)CC12 82806,C1(NC(CCCC=C)c2nnnn2C2CC(F)(F)C2)CCC(=O)N(C2CC2)C1 82807,c1(OC)cnccc1C(c1nnnn1C1(C)CC1)NCc1cc(Cl)no1 82808,c1(OC)cc(C#N)ccc1OCC(N1CCCCC(NC(=O)C(O)C(F)F)C1)=O 82809,c1(C(N(CCN(C(c2ccc(C3CC3C)o2)=O)CC)CC)=O)cc(C#N)on1 82810,N1(C(C(C(C)O)(F)F)=O)CCC(C2(NC(=O)CC(O)CC(C)(C)C)CCC2)CC1 82811,N1(C(CC(C)OC)=O)C2CCC1CC(NC(c1coc(C(F)F)n1)=O)C2 82812,CC1SCCCC1C(N1CCC(CC(=O)NC2(N3CCCC3)CC2)C1)=O 82813,c1(CC)nc(NCCCS(N)(=O)=O)cc(N2CCC(C)(C(N)=O)C2)n1 82814,C1(C(C)(C)C)CCN(C(C2CC(O)(CNC(C3CCS3(=O)=O)=O)C2)=O)C1 82815,c1(C(=O)NC2C(NC(C(C)CF)=O)CCCC2)ncc(C2CC2)cc1F 82816,CC1(C)COCCC1C(=O)NCCCC1CCCN1C(c1ccc(CO)cc1)=O 82817,c1(SC(C)C(=O)NC2COCC2NC(=O)CC(F)F)ccccc1 82818,C1(C(N2C(C)(C(=O)NCC3(O)CCN(C)C3)CCC2)=O)CCC(C)(C)OC1 82819,C1(NC(CSCC=C)=O)CN(C(=O)C(C)(C)N(C)C)CC1C(F)(F)F 82820,N1(C(c2c(CC)[nH]c(=N)s2)=O)CC2CCN(C(C3OCC4CCCC3C4)=O)C2C1 82821,CC1=NS(=O)(=O)NC(C)=C1CC(=O)NCC(O)CCNC(C1CNC(=O)N1)=O 82822,c1(OC)ccc(SC)cc1OCCNC(C)CCC=C(C)C 82823,CN1CCC(c2nnnn2C(C)(C)C)(NCCC2OCCCC2(C)C)CC1 82824,C1(CNC(c2cc(C)cc(F)c2)=O)CN(C(c2cnc(C)o2)=O)CC2(CCC2)O1 82825,CC1(C)CCC(C)(Cc2cn(CCNC(c3c(F)cc(F)cc3F)=O)nn2)CC1 82826,CC1CC(=O)NCCN1C(=O)CC(C)C(C)(C)NC(=O)C#CC1CCCC1 82827,C(=O)(C(F)C(C)C(F)(F)F)N1CC(CNC(CC(CC)c2ccc(C)cc2)=O)C1 82828,C(CC(=O)N1CCOCC(O)C1)(C(C)CC)N(C(CC=CC=C)=O)C1CC1 82829,c1(OC)cc(F)c(C(=O)NCC(CNC(=O)C(C)(C)OC)C(F)(F)F)c(F)c1 82830,O=C(CN=C(NC1CCC1)N1CCC(OC)C1)N.c1(CC)cc(F)c(F)c(F)c1 82831,c1(C(C)(C)C)nc(CC2CCCN2C(=O)CSc2nc[nH]n2)n(-c2nc[nH]n2)n1 82832,c1(CC(=O)NCCCN(C)C(c2nc(Cl)sc2Cl)=O)cccc(C2CC2)c1 82833,C(CCCCCNC(=O)CC(C)c1cnn(C)c1)N(C)C(c1cncn1C)=O 82834,c1(N2CCC(C(C)NC(=O)CCN3CCC(F)C3)C2)nc(C2CC2)nc(=N)[nH]1 82835,Cc1[nH]c2ccc(C(=O)NC3CC(NC(C4(O)CC(C)(C)C4)=O)C3)cc2c1C 82836,C1(NC(C(CCSC)OC)=O)CN(C(c2ccc(N)cn2)=O)C2(CCC2)C1 82837,C=C(Cl)CC(C(=O)N1CC2C=CC2C1)NC(=O)COC1(C)CCC1 82838,N12CC(O)C(O)C(O)C1C2=O.c1(CN(C)C)ccccc1C(c1ccccc1)=O 82839,CCS(=O)(=O)C1(CNc2cc(NCC3(C)CCCCC3O)nc(C)n2)CC1 82840,C(=O)(C(C(=O)N1CC(F)(C(N2CCC(F)(C(N)=O)C2)=O)C1)OC)OCC 82841,Cc1ccc(OC(C)C(=O)NC(c2ccccc2)CN(C(=O)CC(C)C)CCl)cc1 82842,C(c1ccc([N+](=O)[O-])s1)=CC(N1CCC(CN(C)C(C2(C)C=CCCC2)=O)C1)=O 82843,c1(C(=O)NCC(C)CN(C(=O)C=CS(C)=O)C)ccnc(C(C)(C)C)c1 82844,c1(C(=O)NCC2C(C)CCN2C(c2ccns2)=O)ccc2c(c1)CCC2 82845,N1(C(C)=O)CCC(N=c2[nH]c3c(c(=NCC4CCC(C5CC5)O4)[nH]2)SCC3)C1 82846,Cc1nnn(CC(=O)N(CCC(C)NC(=O)CC(C)c2ccncc2)C)n1 82847,C(CCCC(CO)NC(=O)C(F)=C(C)C)NC(C=C(C)c1ccsc1)=O 82848,C(=O)(CS(=O)(=O)C1CC1)N(CCOC)CCNC(c1cc(OC)nn1C)=O 82849,C1(CC(C)N(C)C(=O)NCC2CC(NCS(C)(=O)=O)C2)CCOC1 82850,C1(C(=O)NCCN(C(=O)CCc2ccncc2)CCCN(C)C)CCOCC1 82851,CC(CCNCCCCCC1OCCO1)CC(C)(C)C 82852,Cn1ncc(C(=O)NCc2nocc2C(N2CC(SC(F)F)C2)=O)c1N 82853,Cc1cnc(Cl)c(C(=O)N(C)CC2CN(C(C3(C)CCCC3)=O)CCO2)c1 82854,N1(C(C(CC)(C)OC)=O)CCCCC(CNC(=O)CC2CCCC2)CC1 82855,C1(C(=O)NCC2C(NC(C3CC4(CCOC4)C3)=O)CC2)CN2CCC1CC2 82856,C1(C2CC2)(C(=O)Nc2c(C)noc2CC2CC2)CN(C(C2CC23CC3)=O)C1 82857,c1(CC(N2CCCCC2Cn2cc(CCCO)nn2)=O)cccnc1Cl 82858,N1(C(CSC(C)(C)C)=O)CCC(NC(C2(F)CC3(CCC3)C2)=O)C(C)(C)C1 82859,c1(C(=O)NCCCCC(C)NC(C(C)n2ccnc2)=O)ncc(F)cc1F 82860,CC(C)CCC(C)NC(=O)C(C)(C1CCC1)NC(=O)CCN=[N+]=[N-] 82861,c1(C(=O)NCC2C(NC(C3(C)CC3(F)F)=O)CC2)cnc(Cl)c(N)c1 82862,N1(CCc2scc(C)n2)CCOCC1c1cccs1 82863,Cc1nn(C)c2c(NCC3COCC3O)nc(=NCCCC3CCCCC3)[nH]c12 82864,CC1CN(c2cc(CNC3CCNCC3C)ccn2)CCO1 82865,c1(C(=O)NCC(CNC(CCOCC#C)=O)(C)O)cc(C)n(CCO)n1 82866,C12(NC(C3C(=C)CC3)=O)CCC(C1)N(C(c1ccnc(-c3ccco3)c1)=O)C2 82867,N1(C(C(COC(C)=O)C)=O)CCC2(CC1)CN(C(c1cnn3c1CCC3)=O)C2 82868,Cc1nc(CCCNC(=O)C(C2CC2)NC(=O)CC2CCCSC2)n[nH]1 82869,N1(C(C(CSC)C)=O)CCN(C(C2CCCN(C(=O)CCC(F)F)C2)=O)CC1 82870,C1(NC(C2N(C(CC)=O)CCCC2)=O)CN(C(=O)CC2CN(C)C2)CCC1C 82871,c1(CC)ccoc1C(=O)NCCCC(c1ccccc1)NC(c1cnc(C)s1)=O 82872,CCCC(CNC(c1n[nH]c2c1COC2)=O)C(=O)NC1(CC)CC1 82873,C1(NC(c2ccnnc2O)=O)C=CCN(C(c2ccc(CF)cc2)=O)C1 82874,C1(C#N)(CNC(CCC2CCCN(C(C(CO)OC)=O)C2)=O)CCOCC1 82875,C(=O)(CCCCCCCCCO)N1C2C(NC(CCOCC)=O)CC(C2)C1 82876,N1(C(C(C)SC)=O)CCCCC1C(=O)NCC1CC1(C)C 82877,C#Cc1ccc(C(=O)NC2CC23CC(NC(=O)C(O)CC2CCCCC2)C3)nc1 82878,S(=O)(=O)(c1cccnc1)NC(CCSC)C(N1CCOC(C)C1COC)=O 82879,CN1CC(NC(C2CN(C(=O)Cc3ccccn3)CCO2)=O)CC1CO 82880,C1(NC(C(C2CCC(C)CC2)CC)=O)CCCN(C(=O)CN2CCCCC2)CC1 82881,N1(C(COCC)=O)C2CCC1CN(C(=O)C(C)Cc1cnc[nH]1)C2 82882,CC1=NNC(=O)C1CC(=O)NC(CO)C(C)NC(=O)CCCn1c(C)csc1=O 82883,C12(C(CNC(C3CCCC3C)=O)NC(CC=C(C)C)=O)CCC(CC1)C2 82884,C1(=CC(=O)NC2CCCC(Nc3ccnc(C4CCC4)n3)C2)CN2CCC1CC2 82885,C(CC(=O)Nc1cc(O)cc(F)c1)(C(F)F)NC(c1n(CC)nc(C)c1)=O 82886,C1(NC(c2ccc(OCC)cc2)=O)CCC12CCN(C(c1snnc1C)=O)CC2 82887,C=CC(C)(CC)C(=O)N1CCN(c2ccnc(CSC(F)(F)F)n2)C(C)C1 82888,c1(CNC(=O)CC(O)C2CC2)ccc(-c2cn(-c3ncc(Br)s3)nn2)cc1 82889,C(=O)(C1CCCc2ccccc21)NC(C)CNC(=O)C(C1CCC(=O)N1)C 82890,c1(C(C)NC(CCn2cc(COC)nn2)=O)cccc(C(C)(C)C)c1 82891,C(=O)(CC(C(F)(F)F)NC(c1ccc2c[nH]nc2c1)=O)NCCC 82892,C1(NC(C(C)(C2CC2)OC)=O)CCN(C(=O)CN2CCOCC2)CC1C 82893,C12(CNC(C3(CC#C)CCOC3)=O)CC(CO1)N(C(c1cc3n(n1)CCC3)=O)C2 82894,C=C1CC(C(=O)NC(C2CCCCC2)CF)(CNC(=O)CN2CCCC2SC)C1 82895,C1(C(N2C(C)(CNC(=O)COc3ccc(F)nc3)CCC2)=O)CCCCNC1=O 82896,c1(OC)ccc(C(=O)NC2CC(F)(CNC(C3(C4CC4)CC3)=O)C2)s1 82897,C1(C)(C(N2CC(CCCCC)C2)=O)CCN(C(=O)C(C)(CC)OC)C1 82898,O(N=C1CCCCCC1)CC(=O)NCC(CNC(C(C)OCCC=C)=O)F 82899,N1(C(C2(CC)CC2(F)F)=O)CCN(C(c2cc(-c3ccccn3)no2)=O)CC1 82900,N1(C(c2ccc(C(C)=O)c(F)c2)=O)CCN(C(=O)Cn2cnnc2O)C(C)C1C 82901,C(=O)(CCCS(C)(=O)=O)NC(C1CCCN(C(c2cccc(C)c2N)=O)C1)C 82902,CC(C)S(=O)(=O)CC(=O)NC1(CNC(=O)C(=O)Nc2ncc[nH]2)CCCCC1C 82903,N1(C(C2(COC)CCOCC2)=O)CCCC(CNC(c2cc(OC)cs2)=O)CC1 82904,Cc1onc(CO)c1C(=O)N(CC(C)NC(c1ccc(C(C)(C)C)nc1)=O)C 82905,C1(CCOC)CN(C(c2csc(-c3ccncc3)n2)=O)CCN1C(=O)C(N)=O 82906,N1(C(C2C(OC)(OC)CC2)=O)CCC(F)(CNC(c2cnn(C(F)F)c2)=O)C1 82907,c1(C(=O)NCCCCCNC(c2ccc[n+]([O-])c2)=O)ncc(F)cc1F 82908,Cc1nccc(C(N2CCCCC2CCC(=O)N(C2CCOC2)C)=O)n1 82909,C(C)(C(=O)NC1CC(F)(CNC(C2(N(C)C)CCCOC2)=O)C1)(C(C)C)OC 82910,C1(C(=O)NC2C(C)CN(c3nnc(C#N)s3)CC2)CN2CCN1C(C)C2 82911,C1(C(=O)NCCN(CC(F)F)C)CC2CCC1N2C(=O)CC1CCCO1 82912,c1(C(=O)NCCNC(C(COC(C)(C)C)N(C)C)=O)cc(Br)ccc1O 82913,C(c1cn(C)cn1)=CC(=O)NC(CCOC)CNC(C1CCCN1C1CC1)=O 82914,CC1CN(C(=O)CC2CCN(C)CC2)CCC1N(C(=O)Cc1ccnn1C)C 82915,C1(COC(CCC(=C)C)=O)CCCN(C(c2cc(NC(C)=O)cnc2C)=O)CC1 82916,N1(C(CNS(NC)(=O)=O)=O)CCN(C(=O)CCc2ccsc2)CC(CO)C1 82917,S(=O)(=O)(c1cc(C(F)(F)F)ccc1NCCF)NC(c1cc2ccccc2o1)C 82918,c1(CNC(CCC2(C)CCN(C(C3C(C)(C)C3)=O)C2)=O)ccnc(C#N)c1 82919,C(CCC(C)CO)NC(CC1(OCC)CCC1)=O 82920,C=C1CC(C(=O)Nc2cc(C(=O)OC)no2)N(C(=O)Cc2ccc(Br)cc2)C1 82921,Cc1nnc2n1CC(C(N1CCOCC(NC(=O)Cc3ccoc3)C1)=O)CC2 82922,Cc1cc(NC(=O)CCF)ccc1NC(c1cnn(C2CC2)c1C1CC1)=O 82923,C(=O)(C1COc2ccc(Cl)cc21)N1CC(NC(C(C)(C)C2CC2)=O)C(C(F)F)C1 82924,C1(CC(=O)N(CC(c2nn[nH]n2)C)C2CC2)CCCN1C(=O)CCc1ccoc1 82925,n1(CC)nccc1C=CC(=O)N(C(C)CN(C)C(c1snnc1C)=O)C 82926,c1(C(N(CC(C2CC(F)(F)C2)O)C)=O)ccc(N)c(Cl)c1 82927,c1(C(=O)NC2CC2C(=O)Nc2ncc(F)cc2Br)cc(Cl)c(Cl)cc1F 82928,C(=O)(CC(F)(F)C(F)F)N1C(CC(=O)NC(c2ccc(Cl)nc2)C2CC2)CCC1 82929,N1(C(c2ccc(OCCN(C)C)cc2)=O)CCN(C(=O)C=C2CCC2)C(CF)C1 82930,Cc1nc(-c2cccs2)sc1C(N1CCCC1C(C)(C)NC(=O)COCCF)=O 82931,CC(C)C(O)C(=O)N1CCC(C(C)(C)NC(=O)CCCn2cnc(C#N)n2)C1 82932,c1(CN2CC3C(C(N4CCC(C)CC4)=O)(C3)C2)cc(F)ccc1F 82933,c1(NC(=O)COC(F)F)nccc2ccncc12.C12CN(CC1C1CC1)C2=O 82934,c1(C(N(C)CC2C(C)OCC2)=O)c(CNC(C2SCCS2)=O)nnn1C 82935,C1(CCNC(c2ncc(C)nc2)=O)CN(C2CCc3ccccc32)C1 82936,C1(NC(C2(C3N(C(C(CSC)C)=O)CCC3)CC2)=O)CCC(F)(F)CC1 82937,c1(CC)ccc(CNC(=O)CC(C)NC(C2CCOC2C(C)C)=O)cc1 82938,CC1(C(N2CCCCC2C(=O)NCCN2CCC(CO)C2)=O)CCCCC1 82939,CC1CC=C(C(=O)NCc2cc(C(=O)NCC(C)C(C)(F)F)n[nH]2)CC1 82940,c1(-n2cc(CNC(Cc3c(C)nsc3)=O)nn2)ccc(F)cc1C(F)(F)F 82941,C1(NC(CCC(=O)OCC)=O)CCCC12CCN(C(C1CCC1(C)C)=O)CC2 82942,Nc1cc([N+](=O)[O-])ccc1C(N1CCCCC(NC(c2c[nH]c(Br)c2)=O)C1)=O 82943,c1(C(=O)NC2CCC(N(C(c3c(CC)nc[nH]3)=O)C)C2)ccnc(OC(C)C)c1 82944,c1(CN2C(C=C)(c3ccccc3)COCC2)nc2c(F)cccc2n1C 82945,C1(CC)CN(C(c2ccnc(F)c2F)=O)CCN1C(=O)Cc1ccccc1OC 82946,c1(N2CC(C)C(NC(=O)CC3CC(F)C3)CC2)ccc(Br)cc1[N+](=O)[O-] 82947,N1(C(c2ncc(-c3ccncc3-n3cccn3)s2)CC)CC2CC(OC)C(C2)C1 82948,N1(C(c2nn(C)c(=O)cc2)=O)C2CCC1CN(C(c1ncc(Cl)c(N)c1Cl)=O)C2 82949,N1(C(C2(COCC)CC2)=O)CCCC(CCNC(C2CCCC(O)C2)=O)CC1 82950,c1(CC(=O)NCC(C2CCOC2)NC(CC2(OC)CCCC2)=O)ccncc1F 82951,CC1CN(C(C2CC(C)(F)C2)=O)CC2(CCN(C(c3ccoc3)=O)C2)O1 82952,c1(CN(C(C(=O)NC(CC)C(=O)N(C)C)=O)C)ccc(C(N)=O)cc1F 82953,C1(NC(Cc2n(C)nnc2)=O)C2CC(O)C1N(C(c1ccc(C(F)(F)F)s1)=O)C2 82954,Cc1cc(=NC(C)C2CCCCO2)[nH]c(=NCc2ncoc2C(F)F)[nH]1 82955,CCCC(CC)CCC(=O)NC1CCC(NC(c2sccc2OC)=O)CC1 82956,N1(C(C(C)OCC2CC2)=O)CCC(NC(=O)CCC2CCOCC2)C(CO)C1 82957,CC1(C)CC(CNC(C2CC23CC(O)C3)=O)CN1C(=O)CCC1CCC1 82958,c1(C(=O)NC2(CN(C(=O)CCC(N)=O)C)CC2)cnc(O)c2cccnc12 82959,Cc1cc(C)c(CC(N2CCOC(CCNC(C3CCC3)=O)C2)=O)c(C)c1 82960,C1(CC(=O)N(C)Cc2[nH]nnc2C)(OC)CN(C(c2cnn(C)c2)=O)C1 82961,CC1CCCC(n2cc(C3CCOCC3)nn2)C1.N12CC=CC1NC2=O 82962,c1(CN(C(Cc2c(C)occ2)=O)CCNC(C23CC(F)(C2)C3)=O)cccc(Cl)c1 82963,C1(NCc2cncc(C)c2)CCN(C(=O)COCC2CCC2)CC1(C)C 82964,C1(C(=O)NCCc2ccc(C)cn2)(OC)CCN(C(c2ncon2)C)CC1 82965,C(=O)(C(C(C)=Cc1ccc(Br)s1)N1CCC(OCCCNC)CC1)NCC=C 82966,CCC(CC(=O)NCC(O)CN(C)C(c1ncoc1-c1cnn(C)c1)=O)C(C)C 82967,c1(CC(=O)OC)ccccc1C(=O)NCC1C2CC2CN1C(C1C=CCC1)=O 82968,c1(CC(=O)NC2(CC#C)CC2)ccc(OCC#N)cc1.c12cc(co1)C(=O)NC2 82969,N(C(=NCCN(CC(F)(F)F)C(C)C)NCCN1CCCC1)C1CCC(C)CC1 82970,C1(CNC(CCN(C(=O)CCOC2COC2)C)=O)(CO)CCCO1 82971,C1(SC)CCCC1C(=O)NC1CC(CCNC(=O)CCOC2CCCC2)C1 82972,C1(C)(NC(C2CN(CC)C(=O)C2)=O)CCN(C(C2CC(CC(C)(C)C)C2)=O)CC1 82973,N1(C2CCN(CC)C2=O)CC(NC(c2ccn(-c3ccncc3)n2)=O)C(C)(C)C1 82974,c1(C(=O)NCC2C=CC(NC(c3cc(CCC)on3)=O)C2)ccc(C(N)=O)cn1 82975,C12(C(=O)NC3C(NC(=O)Cn4cnc(Br)n4)C3)CC(C1)C(C(F)(F)F)O2 82976,C=CC(O)C(=O)N(CCNC(=O)CN1CCC(C)C1)CC 82977,c1(N2CCN(CC)C(C)(C)C2)nc(N(CC(F)(F)Br)C)c2ncn(CC)c2n1 82978,c1(C(=O)NCC2(C)CCCN2C(c2ncccc2Br)=O)n[nH]c2c1COC2 82979,C1(NC(c2ccc(F)cc2Cl)=O)COCC1C1CC1 82980,C1(NC(c2c(CC)nco2)=O)CCC2CCN(C(C3(C)CC(C)C3)=O)C1C2 82981,c1(COC)nccc(=NCCN(C(=O)CC2Cc3ccccc3O2)C(C)C)[nH]1 82982,c1(CNC(C=CC(C)NC(C2(O)CCSCC2)=O)=O)c(F)cccc1F 82983,C(=O)(C1=Cc2ccccc2C1)N1C2CC(C(N3CCCC(OC4CC4)C3)=O)(OCC2)C1 82984,N1(C(C(C2CCC2)OCC)=O)CC2(CCCCN2C(c2ccnc(S)c2)=O)C1 82985,CC(C)(C)CC(F)C(=O)NC1CCN(C(c2cc3cnccc3[nH]2)=O)CC1O 82986,CCCC(C(=O)N1CCC(C)N(C(c2cc(C)c(F)cc2F)=O)CC1)S(N)(=O)=O 82987,N1(C(C)=O)CCN(Cc2ccc(CNC(=O)C(F)OC(F)(F)F)cc2)CC1 82988,Cc1coc(C(=O)NC(C)CC(C)NC(=O)C(C)NC(c2cccs2)=O)c1 82989,Cc1cc(=NC(=O)NC(CO)C(O)c2ccccn2)[nH]n1C(C)C 82990,Nc1sc2ccccc2c1C(N1C2CCCC1CN(C(=O)COCCCF)C2)=O 82991,CCC(CC(C)C)C(=O)NC1CC(F)(CNC(c2cc3ccccc3o2)=O)C1 82992,CCC(CC)(C(=O)N1CCC(NC(=O)CCC(C)(C)F)C(C)C1)OC 82993,c1(OC)cc(C)cnc1C(=O)N(C)CC1C2CN(C(C3CC3C)=O)CC12 82994,c1(NC)cnc(C(=O)N(C)CCN(C)C(c2ncoc2C2CCC2)=O)cn1 82995,CCCC(O)CC(=O)N1CCOCC1CNC(c1sc(C)nc1CC(C)C)=O 82996,C1(C(=O)NC(C(=O)NC2CN(C(C)C)C(=O)C2)C2CC2)CN(C)CCN1C 82997,CC1CN(C(=O)C2=CCC(NC(=O)CCC(F)(F)F)C2)C(C)C1C 82998,Cc1cccc(C(=O)NCC2CC(CC(N3CCCC3(C)C(=O)N(C)C)=O)C2)n1 82999,Cc1nc(-c2ccccc2)ncc1C(N1CC(O)(CN(C(=O)C(C)C#N)C)C1)=O 83000,c1(OC)ccc2[nH]nc(C(=O)NC3(CNC(c4cncs4)=O)CC(OC)C3)c2c1 83001,C(=O)(C(F)C(=O)NCC(CC)NC(=O)CCCc1cc(C)no1)OCC 83002,CCC(C(=O)NC1CC(F)(CNC(=O)C(C)CC2CC2)C1)OC 83003,C(CCCc1ccco1)(c1nnnn1CCOc1cccs1)NCC1C(C)C1C 83004,CCS(=O)(=O)C=CC(=O)NCC1CC2CCC(C1)N2C(=O)CCC=C(C)C 83005,C12(C(N3CC(CNC(Cc4c(C)n[nH]c4)=O)C(C)C3)=O)CCC(CC1)CC2 83006,c1(C(=O)NCCN(C(=O)C(C)(C)n2cnc(C)c2)CCOC)ccc(C)n1C 83007,C1(CN(C(c2[nH]cc(C(=O)OC)c2)=O)C)CCCCN1C(C1CC1C)=O 83008,C1(NC(=O)C=Cc2cnccn2)CS(=O)(=O)CC1NC(c1cc(Cl)ccn1)=O 83009,C1(CCNC(CN2C(C)CC2)=O)CSCCN1C(=O)CSCC(N)=O 83010,C1(C(=O)NCC2C(C(N3CCC(C(C)C#N)CC3)=O)C2)CC12CCOCC2 83011,Cn1cnc2nc(=NCc3nncs3)[nH]c(NCC3C4CCCCCC34)c12 83012,C=C(Cl)C(C)(C)C(=O)N1CC(NC(=O)Cc2cc(OC)ccc2Cl)C2(CC2)C1 83013,CC(C)CC(C(=O)N1CCCC(C)(NC(c2cn3ccnc3cn2)=O)C1)C(C)C 83014,C12(C(=O)Nc3cccc(-n4ccnc4O)c3)CCCC1C2(F)F 83015,C(=O)(N=c1[nH]onc1C(C)(C)C)N(c1ccc(C(=O)OCC)cc1)C.C1CN1 83016,C(CCCCCNC(c1ccc[n+]([O-])c1)=O)NC(c1ccsc1)=O 83017,C1(N(C(C(C)N=[N+]=[N-])=O)C)CCCN(C(=O)C(c2cncnc2)C)CC1 83018,C12(NC(c3c(Cl)ccc(C#C)c3)=O)COCCC1CN(C(=O)CC(C)(C)C)C2 83019,C(CCCCC(=O)N1CC2(CC(NC(=O)C(n3cc(C)cn3)C)C2)C1)SC 83020,C1(CC)CN(C)CCN1C(C1CCN1C(=O)CNc1ccccn1)=O 83021,C1(OC)CC(NC(C2(CCF)CCC2)=O)CN(C(=O)Cn2cccc2)C1 83022,c1(OC)cc(OCCCNC(=O)CCn2cnnn2)ccc1C(=O)NCC1CC1 83023,C(CC1CC1)(C(=O)NC(CC1CCCC1)C(=O)N1CCC(N2CCC2)C1)OC 83024,Cc1cc(C(N2CC3CCC3(CCNC(c3cnc(N)cn3)=O)C2)=O)cc(C)c1 83025,C1(C(=O)OCC)CN(C(c2ccc(N(C)C)cc2)=O)CCC1N 83026,CC(CC(=O)c1ccc(F)cc1)C(=O)OC(C)(C)C(=O)N(C1CCCCC1)C 83027,c1(C(=O)NC2CN(C(c3cc(C)no3)=O)CC2F)c[nH]c2cnccc12 83028,c1(NC2CC3CN(C(c4cc5sccc5[nH]4)=O)CC32)nc2ccccc2s1 83029,C1(NC(c2c(C)cc(SC)s2)=O)CN(C(c2n[nH]c(C)n2)=O)CC(C)(C)C1 83030,c1(OCC)cc(C(=O)NCC(CNC(=O)CSc2ccncc2)CO)cc(F)c1 83031,c1(OC)c(Br)cccc1S(=O)(=O)N1CCC(NS(C)(=O)=O)C1 83032,C12(C(=O)NCCN(C(C34CCCC3C4(F)F)=O)CC)CCCC1CC(=O)C2 83033,C1(C)(CC)CC(NC(c2cc(F)ccc2F)COC)CCO1 83034,n1(C(C)C)ncc(Cl)c1C(N1CCCC1(C)c1cn(-c2ccc(N)cc2)nn1)=O 83035,Cc1ccc(C(=O)NC2CCC(C)N(C(C3CC4(C3)CC(O)C4)=O)C2)cc1C#N 83036,C1(C(N2CCC(CCNC(C3C(C)(C)CC3)=O)CC2)=O)OCCOC12CCC2 83037,N1(C(c2c(C)c[nH]n2)=O)CCC2(CCC2)C(NC(=O)CSCCN(C)C)C1 83038,c1(C(=O)NCC2(C)CCC(NC(c3cc[n+]([O-])cc3)=O)C2)cnc2n1CCC2 83039,c12nc(C)c(s1)CC(=O)NC2.C(C(CO)NC(C1CC1CC)=O)CC(=C)Cl 83040,CC1C(=O)N(C)CCN1C(=O)C(C)(c1ccccc1)NC(=O)CCCN(C)C 83041,Cc1cc(N2CCCCC2CCNC(=O)Cn2nccn2)cc(C#N)c1[N+](=O)[O-] 83042,CCCC(C(=O)NCc1ccccc1)N1CCCC1CC1CCCCC1 83043,c1(-c2cc(OC)cc(F)c2)cc(-c2nccn2C(C2CCC2)C)cc(Cl)c1OC 83044,c1(NC(=O)CC23COC(C2)C3)ccc2cccnc2c1Br 83045,C1(NC(C2C(NC(C(CO)OC)=O)CCO2)=O)C=C(C)CCC1 83046,N1(C(CCC=C(C)C)=O)CCN(C(c2cccnc2C(N)=O)=O)CC1C(F)F 83047,c1(C(N(CCC(=O)NC(C2CCCC2)C)CCO)=O)cccnn1 83048,CC#CC1CCN(C(c2cc(CNC(C3CC3C(C)C)=O)nn2C)=O)C1 83049,Cc1cc(O)ncc1NC(C1(C)CC(O)CN1C(=O)C(C)C)=O 83050,c1(OC)ccc(C(=O)NC(C2CCCN2CCc2ccccc2)C)cc1 83051,C1(CNC(=O)CCc2nc[nH]n2)CCCCC1NC(=O)CCc1cn[nH]c1 83052,N1(C(C(=O)NCc2nnn(C)n2)c2cncs2)CCCc2occc2C1 83053,N1(C(=O)CC2CC2)CCCCC1C1CCCN1C(=O)Cc1ccccc1 83054,C1(CCNC(C(C(C)C)OC)=O)CCCN(C(c2c(C)noc2N)=O)CC1 83055,CN1C2CCCC1CN(C(=O)C1=NOC(CNC(=O)C3=CCCCCC3)C1)C2 83056,N1(CCC(=O)OCC)CC2(CNC(=O)C2)C1.C1C(CN=[N+]=[N-])S1 83057,C1(F)(C(=O)NCCOCCC(=O)NCc2nc(C)[nH]n2)CCCCCC1 83058,C(=O)(CC(C)(C)COC)NCC1N(C(c2cc(C(C)=O)oc2)=O)CC(N(C)C)C1 83059,C(=O)(C(C)CC(F)F)N1CC(C(C(N2CC(O)C(O)C2)=O)OC)C1 83060,Cc1ccc(C(N2CC3CCC2C3NC(c2ncsc2C)=O)=O)cc1OC(F)F 83061,N#Cc1ccc(S(=O)(=O)N2CCCC3CC2C32CC2)cc1NCCCF 83062,c1(C(N(CCN(C(C2CC(C)(C)O2)=O)CC)CC)=O)cc2cccnc2s1 83063,N1(C(=O)OC)CC(OC)CC1C(N1CC(C)(NC(c2ccc(C)cc2)=O)C1)=O 83064,C1(C(=O)NC(C2CCN(C(c3c(F)cncc3Cl)=O)C2)(C)C)COCCC1(F)F 83065,N1(C(C2C(C)C2C)=O)CCCCC2(CCN(C(C3CC(=O)NC(=O)N3)=O)C2)C1 83066,N1(C(c2c(CC)nn[nH]2)=O)CCOC(C(=O)NCc2nc(C)cs2)CC1 83067,C(CC(CC)C(=O)NC(CN(C(=O)CN(S(C)(=O)=O)C)CC)CC)=CC 83068,C1(NC(C2C(OC)CCC2)=O)CC2CCC(C1C)N2C(c1cc(C)ncn1)=O 83069,C1(NC(CC=C)=O)CC2(C1)CC2NC(=O)C(c1ccc(Cl)s1)C 83070,C1(C(=O)NCCCCC2C(C)C2)CN(C(=O)CC2CCCC(=O)C2)CC(C)(C)C1 83071,N1(C(c2cnc(C(C)(C)C)s2)=O)CCC(NC(c2nsnc2O)=O)C(F)C1 83072,N#Cc1cccc(I)c1NC(C1CCCCC1NC(c1ccc(CO)cc1)=O)=O 83073,c1(C(=O)NC(CCOc2ccc(C)cc2)(C)C)ncnc2cccnc12 83074,c1(CNC(=NC)NCC2(c3ccc(OC)cc3)CC2)ccc(I)cc1 83075,c1(C(=O)NCC(C)CN(C(=O)CN2CCSCC2)C)conc1C1CCCO1 83076,c1(OCC=C)c(OC)cc(-c2nn[nH]n2)cc1NC(c1cccc(C)c1CC)=O 83077,Cc1c(F)ccc(C(=O)NCC(CNC(=O)CC2OCCC2(C)C)CO)c1C#N 83078,Nc1ccc(C(=O)N(CCC(=O)NCC2CC2Cl)C2CC2)nc1 83079,C1(C(=O)NC(C)Cc2nc3ccccc3s2)CC(c2ccc(F)cc2)=NO1 83080,Cc1ccnc(C(=O)NC2CC(=O)N(C3CN(C(c4ccco4)=O)C3)C2)n1 83081,C1(CCCCNC(CN(C)CC)=O)CCN(C(C23CCCC2C3)=O)CC1 83082,N1(C(C2CC(C)C2)=O)CCOCC2(COCCN2C(=O)C2=CCCC(C)(C)C2)C1 83083,C(=O)(C(C)(C1CCC1)NC(c1c(SC)con1)=O)OC 83084,CC1C(C)N(C(c2coc(O)n2)=O)CCN1C(c1cc(F)ccc1O)=O 83085,c1(C(=O)NCCC2N(C(c3c(=N)[nH][nH]c3)=O)CCC2)cc(O)nc2ncccc12 83086,c1(CC)ccc(CN2CCN(C(c3cc(COC)nn3C)=O)C3CC23)c(O)c1 83087,C1(CNC(C)Cc2ccc(N(C)C)cc2)COCCC1c1ccccc1 83088,c1(CC(=O)N(CC(=O)NC(c2ccccc2)C#N)C)cc(O)nc2ccccc12 83089,C(=O)(C(F)(F)C(O)CC)NCC(CC)NC(=O)Cc1sc(C)nc1C 83090,C12(CNC(Cc3c(OC)cccc3Cl)=O)CCCC1CN(C(c1nc[nH]n1)=O)C2 83091,N1(C(C=CCN(CC)CC)=O)CC2CC(C1)CN(C(C1CCCCN1C)=O)C2 83092,Cc1cc(N)c(C(=O)NC(CO)C(C)NC(C2C3CC4C(C3)C24)=O)c(F)c1 83093,C(=O)(C1CCCc2cncn21)NC(C(C)C)CCNC(c1c(O)cccc1Cl)=O 83094,c1(NS(CC(=C)C)(=O)=O)sc(CCO)cc1C#N 83095,c1(C(=O)NCC(CC=C)NC(C2CS(=O)(=O)C2)=O)cnc2c(F)cc(C)cc2c1 83096,CCCC(C(=O)N1CC(N2CC(F)C2)C1)NC(=O)C(C)c1cccs1 83097,C1(CCC(=O)NC2C(NC(CNC(=O)OCC)=O)CCC2)NC(=O)NC1=O 83098,C1(F)(CNC(C(C)(C)OCC)c2nnnn2Cc2ccccc2)COCCOC1 83099,C#Cc1cc(C(=O)NCC(C)CNC(c2ccc(Cl)nc2O)=O)ccc1C 83100,CC(=O)CCCC(C)C(=O)N1CCSCC1C(N1CC(C)(C)C1)=O 83101,C1(C(=O)NC2C(NC(c3cccc(OC)n3)=O)CCC2)CC12CCC(F)(F)CC2 83102,C1(NC(C2CCCOC2)=O)CCCN(C(=O)C(O)C2CCC2)CC1 83103,c1(C(=O)NCCC(C)N(C(=O)C=CC2CCCC2)C)cccc(N)c1 83104,Cc1cc(C#N)ccc1C(=O)NC1CC2(C1)CC2C(=O)NC12CCC(C1)OC2C 83105,C1(C(N2CC(C(=O)OC)OCC2)=O)COC2(C1)CN(C(=O)CNC(=O)OC)C2 83106,C(=O)(C(C)CC(C)(F)F)NC1CC2(CN(C(c3cc(C)c(Br)o3)=O)C2)C1 83107,C1(O)(CC)CCN(C(c2nc[nH]c2C(F)(F)F)=O)CC1 83108,C(=O)(C1CC(=O)c2ccccc21)NCCC1CCN(C(c2c(C)scc2)=O)CC1 83109,N1(C(CC(C)F)=O)CC2(CCOCC2)CC1CNC(=O)Cc1nccn1C 83110,C1(OC)(CNC(=O)CC2C(NC(=O)CN3CC(C)(C)C3)CC2O)CCOC1 83111,N1(C(C(CCCNC(c2cc(CC)on2)=O)(C)C)=O)CCC2CCC(O)C1C2 83112,CC1(CN=c2[nH]nco2)CCN(C(=O)C=CC(N)=O)C1 83113,C1(C(N2C(C)(C(=O)NCCNC(=O)NC)CCC2)=O)CC2(CCC2=O)C1 83114,N1(C(C(C)CC2CCC2)=O)CC2(C1)CN(C(=O)CC1(C)CC1(F)Cl)C2 83115,C(CCCCC(=O)NCC1CN(C(c2ocnc2C(C)C)=O)CCO1)OCC 83116,C12(C(=O)NC(CC)C(=O)OC)CC(CN(C(C3CC(=O)C3)=O)C1)C2 83117,c1(CC(N2C(CCC(=O)NCc3cc(F)ccn3)CCC2)=O)ccc(Cl)cc1Cl 83118,N1(C(C(C)c2ncco2)=O)CCN(C(c2cnnn2C)=O)CC1C 83119,N1(C(C2CC(SC)C2)=O)CC(C)CC1C(=O)NCc1nonc1C 83120,C1(F)(CNC(=O)COCC2CCC2)CC(CNC(c2cnn(C(F)F)c2)=O)C1 83121,C1(C2N(C(Cn3ncc(CC)c3)=O)CCC2)CCN(C(C2CC2C(F)F)=O)CC1 83122,C1(CC)(CC)CC(NC(=O)CC(C)c2cccnc2)CN1C(=O)CCN1CCC1 83123,c1(C(=O)NCC(c2ccc(F)cc2)O)ccc(-c2ccnnc2)c2cc[nH]c12 83124,C1(NC(C2CN(c3nncs3)C2)=O)CCN(C(=O)Cc2csc(Cl)n2)C1 83125,C(=O)(C#CC1CCCCO1)NCC1N(C(C(CC)CCOC)=O)CCC1 83126,c1(SCc2cccc(NC(c3ccc(F)cc3)=O)n2)c(F)cncc1Cl 83127,N1(C(C2(CC)CC2)=O)CCC2(CCOC2)C(CNC(c2ccnnc2S)=O)C1 83128,c1(OC)cc(C(N2CCCC2CCNC(=O)CC2COCC(C)O2)=O)n(C)n1 83129,c1(C(N2CCC(CC)(NC(=O)CC34CC(C3)C4)CC2)=O)noc2c1CCCC2 83130,C=CCC(CC)C(=O)NCC(CC)NC(=O)C(=O)NCCOCCCC 83131,O=C(C1=COCCO1)NCC12CC(C1)C(NC(c1ncccc1F)=O)CO2 83132,C12CC(O)CN1C(=O)COCCCNC2=O.CC(CCO)N1CCCC1 83133,Cc1cc(Cl)ccc1C(=O)NCC1CCC(C)N(C(=O)CSC(F)F)C1 83134,c1(OC)cncc(C=CC(=O)NC(C)CCNC(c2c(C(F)F)n[nH]c2C)=O)c1 83135,C12(NC(CCCSCC)=O)CCCC1N(C(c1ccc(OC3CC3)cc1)=O)CC2 83136,C12(CNC(c3c(CC)noc3C)=O)CCCC1CN(C(C1CC3(CC3)C1)=O)C2 83137,N1(C(C=C(CC)C)=O)CCN(C(c2cc(F)cc(Cl)c2)=O)CC1C1CC1 83138,CC1(C)OCCOC1CC(=O)NC(C)(CNC(=O)C=CC=C(Cl)Cl)CO 83139,C1(CC(=O)NCC(C2CCCCC2)NC(c2c(C)coc2)=O)CCC(=O)N1C 83140,c1(C(C(N2CC(CNC(C=NOC)=O)(OC)C2)=O)O)ccc(Cl)c(Cl)c1 83141,C(C(C)C(C)C(=O)N(CCCCCNC(c1ccoc1)=O)C)OC 83142,C1(C(N2C(CNC(c3c(C)nn[nH]3)=O)CC2)=O)CC(C)CC(C)(C)C1 83143,c1(OCCOC)cccc(CC(=O)NC2CC(C)N(C(C34CC3C4)=O)C2)c1.C(C)(=O)O 83144,N1(C(c2c(CC)noc2C)=O)CCCC2(CCN(C(=O)C(CC)CO)C2)C1 83145,c1(C(N(C2CCCN(C(=O)C(C(C)C)C(C)C)C2)CC)=O)cc2n(n1)CCCN2 83146,N1(C(c2cncc(C)n2)=O)CC(NC(c2ccn(CCF)n2)=O)CC12CCOC2 83147,c1(NC(C(=O)NCC2(SC)CCCOC2)=O)ccc2n[nH]cc2c1 83148,C(CC(F)F)(C(=O)NCc1ccc(C)nc1O)N(C(C(CC=C)C)=O)C 83149,C(=O)(C(C(C)OC(C)(C)C)C)N(C)C(=O)O.C1(CCOC(C)(C)C)(CNC(C)C)CC1 83150,c1(OC)cc(C)ccc1C(=O)NCC1CCCN(C(=O)C(C)(Cl)Cl)CC1 83151,C(C(C)C(=O)NC1(C)CC(NC(=O)CSCc2ncc[nH]2)C1)OC 83152,C1(CNC(CSCCN(C)C)=O)C2CCCC1N(C(c1cnc(C(C)O)s1)=O)C2 83153,C1(CCNC(CC2CC(NC(C=C(CC)CC)=O)C2)=O)CCC(C)C1 83154,Cc1c(Cl)ccnc1C(=O)NCC(C)(CC(C)C)NC(c1n[nH]c2c1CCC2)=O 83155,C1(NC(c2ccc(OC)s2)=O)CC2CCC1N2C(c1ccc(C#N)n1C)=O 83156,c1(C(=O)NCC2N(C(C3N(C=O)CCC3)=O)CC(O)C2)ccc(Cl)c(Cl)c1 83157,CC1=C(C(=O)N2CC(CNC(=O)CCc3cn(C)cn3)CC2C)C(=O)OC1(C)C 83158,C(=O)(CCCCCF)NC1CC(OCC(=O)NC2CC(C)(C)C2)C1 83159,c1(NC(C2OCCN(C(c3cccc(OC)n3)=O)C2)=O)cnc2ccc(F)cn12 83160,N1(CC=C(C)CSc2ccccc2)CCCC(O)C1C(C)C 83161,C1(NC(c2c(C)ncs2)=O)CCC2(CC1)CC2NC(c1snc2ccccc12)=O 83162,C1(CNC(C=CC)=O)CN(C(c2cncc(C(F)(F)F)n2)=O)CCO1 83163,C(c1ccc(F)cc1)=C(C(=O)NCC1(C)N(C(C2C(CC)C2)=O)CCC1)C#N 83164,c1(CCC(=O)NCC(CN(C(=O)C(O)CF)C)O)cc2ccccc2o1 83165,C1(C(=O)Nc2c(C)ncnc2)CC(F)CN(S(=O)(=O)C(F)(F)F)C1 83166,c1(SC)ccc(C(=O)NC(C2CCCC2)CNC(=O)C(C)OC2CC2)s1 83167,c1(C(C(=O)NC2CCCC(NC(=O)Cc3ccoc3)C2)O)cccc2c1OCC2 83168,c1(-c2scc(C(N3CCCC3c3cccs3)=O)n2)ccccc1F 83169,C=C(C)CC(C(=O)NCCCCOC(=O)NC)NC(=O)CCOC 83170,Cc1ccc(C(=O)C(=O)NCCCCC(C)NC(c2cnc(Cl)cn2)=O)cc1 83171,C(=O)(C(C)CCCCCCC)N1CCN(C(C2CC(C#C)(O)C2)=O)C(C)C1 83172,N1(C(CCc2cccc(C)c2)=O)CCN(C(C2CC2F)=O)CC1C 83173,N1(C(C(C2CC2)NC(C(F)=CCC)=O)=O)CCC2(COC(=O)N2)C1 83174,N1(C(C2CCC(C)CC2)C(=O)NCCOCC)CCCC(C)(OC)CC1 83175,N1(C(c2ccc(C(C)=O)[nH]2)=O)CC=CC1(C)C(=O)NCc1nccc(C)n1 83176,c1(OC)cc(C(N2CCOC(CC(=O)NC3CSC3)C2)=O)cc(OC)c1O 83177,CS(=O)c1ccccc1C(N1CCCC(NC(=O)C(=O)NCC(F)F)CC1)=O 83178,N1(CCCC)CCCCC1C(N1CC2(CNC2)C1)=O 83179,c1(C(=O)NC2CCN(C(=O)Cc3c(O)ncnc3O)CC2)cccc2ccsc12 83180,C#Cc1ccc(C(=O)NC2CC(O)CN(C(=O)CCc3nc(C)no3)C2)c(F)c1 83181,N1(C(CC(C=C)CCC)=O)CC=C(CC(=O)N2CC(C)CCC2CC)CC1 83182,N1(C(c2ccc(CNC(Cc3cn(C)nn3)=O)o2)=O)CCCC1(C)C1CCC1 83183,c1(C2(C(=O)NCC(CN(C(c3cc(C)sn3)=O)C)C)CC2)cncc(Br)c1 83184,N1(C(Cc2ccc(OCC)cc2)=O)CCC2(CC1)CC2CNC(=O)C(O)CC 83185,N1(C(Cc2nc(NC=O)sc2)=O)CCOCC(F)(CNC(C23CC(F)(C2)C3)=O)C1 83186,C1(SCC(=O)NC2(C)CC(NC(C(C)N(C(C)=O)C)=O)C2)Cc2ccccc2O1 83187,Cc1nc2c(F)cccc2cc1C(N1CC2CC1C2NC(c1cnsn1)=O)=O 83188,Cc1nc(C(=O)NC(CNC(=O)CN2CCC(C)CC2)C(C)C)cc(O)n1 83189,CN1CC(NC(=O)CC(N)c2nccs2)C(O)C1 83190,C1(NC(C23C(CN(C(CCCC#C)=O)C2)C3)=O)CCn2ccnc2C1 83191,n1(CC(=O)NC(C(CO)NC(CNC(CC)=O)=O)C)cnc2c1CCCC2 83192,c1(CC(N2CCC(n3cc(CCC)nn3)C2)=O)ccc(Cl)cc1Cl 83193,N1(C(c2cccc(CC)c2C)C(=O)NCCCCCC)CCn2c(C)nnc2C1 83194,C1(C)(CNC(c2c(CC)nn[nH]2)=O)CCCC1NC(=O)C(C)n1ccnc1 83195,C1(N(C(C2CS(=O)(=O)C2)=O)CC)CCN(C(c2oc(CSC)cc2C)=O)CC1 83196,CCC(C)C(C(=O)N1CC(N(C)C(c2cnc(N3CCOCC3)s2)=O)C1)OC 83197,N(C1CCc2c(Br)ccc(Cl)c21)C(C1C2(C(=O)O)CC(C)(C2)O1)=O 83198,C1(C(=O)NC2(CC=C)CCN(C(=O)Cc3cnns3)C2)CCC=CCCC1 83199,C1(C(=O)NCC#CC(=O)NC(C=C)(C)CC)CC2(CCC2)CO1 83200,c1(C(=O)NC(C2(CNC(C)=O)CC2)C)ccc(C#N)c(F)c1Br 83201,C1(NC(c2c(NC)snc2C)=O)CCC2CCN(C(c3cc(C(N)=O)c[nH]3)=O)C12 83202,C1(C(N2C(CNC(C(N3CC(C)C3)C)=O)CC(F)C2)=O)NC(=O)OC1(C)C 83203,c1(C(=O)NC2C(C)CN(C(=O)C(C)(C)C3CCOC3)C2)cn2ccsc2n1 83204,C1(C(N2C(C)CC(CNC(c3c(CC)csc3)=O)C2)=O)CC2CCC(C1)C2=O 83205,N1(CC=CCOC2C(n3c(C)nnn3)CCC2)CCOC(C)C1 83206,O=C(N=S1(=O)c2ccccc2Nc2ccccc21)C1COCCC1(F)F 83207,C12COCCC1C(=O)N2.c1(NC(=O)CN2CC(COC(F)F)C2)cccc(O)n1 83208,C=CC1CN(c2cc(C)nc(N3CCCC(CCO)CC3)n2)CCO1 83209,N1(C(CC)=O)CC2CCN(Cc3cn(-c4coc5ccccc45)nn3)C2C1 83210,C(=O)(C1=C(c2cnn(CC)c2)N(CCOC)C(=O)NC1c1cccn1C)OCC 83211,N1(C(CCOCCN(C(=O)CCC2CCC(=O)C2)C)=O)CC(C)(C)C1 83212,CC(CC(=O)NCCN(C(=O)Cc1nnc(O)s1)C)P(C)(C)=O 83213,c1(CNC23CCC(NC(C4CN(C)C4)=O)(CC2)C3)c(F)ccc(Cl)c1F 83214,CCCCCCCCCC(=O)NCCN(CCC)C(c1cc(C)cc(C)c1N)=O 83215,C(=O)(C(O)CCCC)N(CC(=O)NCC1CC(CC)C1)C(C)C 83216,C1(C(=O)NCCSCc2ccccc2)CCCN(CCC2CCCCO2)C1 83217,N1(C(CSCC=C)=O)CC2OCCN(C(c3ccc4n[nH]cc4c3C)=O)C2C1 83218,N1(c2c(C#N)c(Cl)ns2)CCCC(C2CCN(C(C3CCCC3O)=O)CC2)C1 83219,C(C(O)C(=O)N1CCCC1CCCNC(=O)CCc1ncc(C)[nH]1)SC 83220,C(CCC(O)C(=O)NCP(C)(C)=O)NC(c1cccc(OC)c1)=O 83221,C(=O)(CCCC(N)=O)NCC1C(C)CCN1C(=O)CCc1cnn(C)n1 83222,N1(C(Cc2cn(CC)nc2)=O)CCC(C)C(N(C(=O)CCCC(C)=O)C)C1 83223,C1(C=C)(C(=O)NC2C(C#C)CCC2)CCN(C(=O)CC2COCCO2)CC1 83224,CC1(C)CCC(CN2CCN(Cc3ccc(Cl)cc3)C(=O)C2)c2ccccc21 83225,C1(NC(C(CC#C)C2CC2)=O)CCN(C(=O)C=Cc2cnccn2)CC1(C)C 83226,c1(C(=O)OC)ccc(F)c(NC(C2CC(F)CN2C(=O)CN2CCCCC2)=O)c1 83227,N1(C(C2(C)N(C(c3cc(C(C)C)no3)=O)CCC2)=O)CC(O)CC(O)C1 83228,c1(C(=O)OCC)nc(Cl)c(Cl)nc1NCC1(C)CCN1Cc1c(F)cccc1Br 83229,c1(N(CCN(C(C)=O)C)C)nnc(-c2cncc(Cl)c2)n1CCN(C1CCC1)C 83230,C1(NC(COCCC)=O)(COC)CCN(C(C2CCN(OC)CC2)=O)CC1 83231,C1(NC(C(=O)NCC)=O)CC2(C1)CC2NC(=O)CC1(C(F)(F)F)CC1 83232,N1(C(c2cc(C)cc(Cl)c2O)=O)CCC2(CC1)CCN(C(=O)OC(C)(C)C)CC2 83233,n1(CC(=O)NC2C(CNC(C(F)OC)=O)CCC2)nc(O)ccc1=O 83234,c1(C(=O)NC(CC(C)C)CNC(=O)CC#N)cccc2cccnc12 83235,CC1(C)CCc2c(C(=O)NC3(CCCNC(C4COCCO4)=O)CC3)csc2C1 83236,c1(CC(C)C(=O)N(CCCN(C)C)CCNC(C2C(C)C2C)=O)ccccc1F 83237,Cc1cc(C(N2CC(NC(c3cnc(Cl)cc3I)=O)C(C#N)C2)=O)cc(C)c1F 83238,Cc1cc(C)c(C(=O)N(CC(C)NC(c2ccnc(CC(C)C)n2)=O)C)cc1N 83239,C1(CCC(=O)NCC(C=C)O)CCN(C(=O)Cc2cccs2)C1 83240,CCCC(CCCNC(C1(C)CCC(=O)NC1)=O)NC(c1cncc(C)c1)=O 83241,c1(OC)c(Cl)ccc(C(=O)NCC2(O)CN(C(=O)C(C)(C)SC)C2)c1N 83242,C(=O)(C(C)(C)C(C)NC(=O)CN1CC2CCC1C2)NC(CC)C(F)(F)F 83243,c1(OC)ccc2c(c1)C(C(=O)N(CCCNC(=O)C1=CS(=O)CCC1)C)CCC2 83244,c1(NC(C2(CNC(c3c(CC)c[nH]n3)=O)CC2)=O)ncc(F)cn1 83245,N1(C(CCN(C)CC)=O)CCN(CC(=O)NCc2ncc[nH]c2=O)CC1 83246,C1(CC(=O)NCCCN(C(=O)C#CC2CC2)C2CC2)CCC(F)(F)CC1 83247,c1(CC(=O)NCC2N(C(C3C(C(N)=O)C3)=O)CCC2)c(Cl)cccc1Cl 83248,Cc1cccn2cc(CC(N3CCN(CCNC(=O)C(C)C)CC3)=O)nc12 83249,N1(C(CC(C)F)=O)CC2CCC(CNC(=O)C(C3CC3)C3CC3)C2C1 83250,C(CN=C(NCC1(OCC(F)(F)F)CCSC1)NCC(F)F)SC 83251,c1(C(=O)NCCCC(C)NC(C2CCC(CC)O2)=O)snc(C)c1N 83252,CC1CCC(C(N2CC(N(C)C)C2)=O)CN1C(=O)CC1CCCC(=O)C1 83253,c1(C(N2C(CNC(c3cc(CC(C)C)on3)=O)CCC2)=O)cc2n(n1)CC(F)C2 83254,CCCC(C)(C)CC(=O)N1CCC(C(C)(COC)NC(=O)C(O)C(C)(C)C)C1 83255,c1(C(=O)NC2CCC(CNC(C3(CC)COC3)=O)CC2)ccc2nnn(C)c2c1 83256,C(=O)(C1=CC2(CCN(C(=O)CCCCSC)C2)C1)N(C(CC)(C)C)CC(C)C 83257,N1(C(C2C3C(C)(C)C2(C)CC3)=O)CCCC12CCS(=O)(=O)CC2 83258,C12CCC(CC1)CNC2=O.c1(C(N2CC(C(C)NC(CC)=O)C2)=O)ccccn1 83259,N1(C(C(C=C=C)C)=O)CC2(CC(C(=O)NCc3cc(OC)ccn3)CO2)C1 83260,n1(CCC(=O)NC2C=CCN(c3c(C)cnc(C)n3)C2)cc([N+](=O)[O-])nc1C 83261,CCC(C)CCCC(=O)N(CCNC(c1ccc(C#N)cn1)=O)C(C)C 83262,c1(NC(C)CCC(=O)OC(C)(C)C)ccc(NS(C)(=O)=O)cc1F 83263,c1(C(C(N2CC(NC(C3CCOCC3)=O)C3(C2)CC3)=O)O)cc(F)c(F)c(F)c1 83264,N1(C(C(CNC(C2CCCCCCC2)=O)O)=O)CCC(CO)C(c2ccccc2)C1 83265,C(CCCCC(=O)N1CCOC(CCCNC(=O)C(C)C)C1)NC(C)=O 83266,C1(C(C)(C)C)(CNC(=O)Cc2ccns2)CCN(C(C2COCCO2)=O)C1 83267,C1(C(=O)NCCC(=C)CNC(c2cc(C)n(C)n2)=O)CCOC(C)(C)C1 83268,C12CCCC1NC2.c1(CN(C(CN(CCC)C)=O)C)csnc1C 83269,c1(N(C(C2CCCNC2)C)Cc2ccc(Br)c(F)c2)ncnc2cc(I)sc12 83270,C1(F)(C(N2CC(NC(COCCCC)=O)C(C(F)(F)F)C2)=O)CCS(=O)(=O)C1 83271,C(=O)(CC(CC1CC1)NC(=O)CC(C1CC1)C1CC1)NC(C#C)C(C)C 83272,c1(C(N2CCCCC2CCN(C)C)C(=O)NC(CC)C)nccnc1OC 83273,N1(C(C)=O)CCN(C(=O)CCC(=O)c2ccc(F)cc2)CC1.C(C(=O)C1(Cl)CC1)NC 83274,C1(C)(C(=O)NCC2(Cn3cc(-c4ccc(C(C)=O)cc4)nn3)CC2)CCC(=O)N1 83275,C1(CC=C)(NC(=O)C=Cc2ccncc2C)CCCN(C(C2(C)CC2Br)=O)C1 83276,C1(O)(C(C)NC(=O)CCOc2cccnc2)CCN(C(=O)C=CC2CC2)CC1 83277,c1(NC(C2N(C(C(CSC)OC)=O)CCC2)=O)cnc(Cl)nc1 83278,Cc1nnc(CCC(=O)NC23CC(NC(=O)CCN4CCC(O)CC4)(C2)C3)n1C 83279,C1(NC(C(CNC(=O)Cc2cccs2)Cc2cccc(F)c2)=O)CCS(=O)(=O)C1 83280,C1(NC(C=CC(C)C)=O)C(CNC(C2(S(C)(=O)=O)CCCC2)=O)CCC12CCC2 83281,C=CC(C)(CC)C(=O)NC1CCC(CN(C(=O)C(c2ccc(Cl)cc2)=O)C)CC1 83282,Cc1c(CNC(=O)C(C[Si](C)(C)C)NC(=O)OC(C)(C)C)cnc(Cl)c1Br 83283,N1(C(C=CCCC)=O)CCC(CNC(=O)C(C)Oc2cccc(CO)c2)C12CC2 83284,CC1CCCC1(C)C(=O)NC1CCC(N(C(=O)CCCN(C)C(C)C)C)CC1 83285,c1(OC)cccc(Cl)c1C(=O)NC(C)CC(C)NC(c1cnoc1C1CC1)=O 83286,C1(C(N2C(C)CN(C(c3ccncc3F)=O)CC2)=O)CCC2C(C1)C2(F)F 83287,c1(C(CC)C(=O)N(CCNC(=O)C=CC(C)C)C(C)C)ccc(OC)cc1 83288,c1(C(=O)NC2CC(n3cc(-c4cnccn4)nn3)C2)ccc2c(c1)CCO2 83289,C(CCCCC(=O)NCc1cn(C(C)C)nn1)N(C(c1c(C)cn(C)n1)=O)C 83290,N1(C(c2cc(COC)[nH]n2)=O)CCOCC(C(N2CCSC(C(C)C)C2)=O)C1 83291,C(CC(C)C)(C(=O)NCC(c1ccccc1)NC(c1ccn(CC#N)n1)=O)OC 83292,C(=O)(C(CNC(c1cnn(C(C)C)c1)=O)CC1CCCC1)NCC(CC)(C)O 83293,c1(C(=O)NCC2(F)CC(CNC(CC3(C#N)CC3)=O)C2)ccncc1Br 83294,CCC(O)CC(=O)NCC1(NC(=O)Cc2cncc(C)c2)CCOC1 83295,C1(C(N(C(C(=O)OC)C)C)=O)(NC(C2CC2(F)F)=O)CCN(C)C1 83296,c1(C(=O)NC2C(NC(CCc3c(C)cccc3)=O)CCCC2)ncc(F)cc1F 83297,C1(C(=O)OCC)CCCN(C(C2(C)CCN(Cc3ncc(N(C)C)cn3)C2)=O)C1 83298,c1(C(c2n(CC)nnn2)NCCOC2CCOC2)ccc(Br)cc1Cl 83299,c1(CCNC(CN(C(C)C)C)=O)ocnc1CN(C1CCCC1)C(=O)CC1CC1C 83300,N(C(=NCCN1CCCC1)NCC1CCOC1)CC(C)(C)CSc1ccccc1 83301,N(C(=NCCCCN1CCCC(C)C1)NC(C)C)CC(c1ccc(F)cc1)OC 83302,c1(C(=O)NC2CN(C(CN3CCC(C)CC3)=O)CC2(C)C)ccnc2ncnn12 83303,Cc1nc[nH]c1CC(O)C(=O)N(C)CC1(CNC(c2cn(C3CC3)cn2)=O)CC1 83304,N1(C(C(n2c(C)ncc2)C)=O)CC2(CC(CC(N3CC(O)CC3C)=O)C2)C1 83305,N1(c2n(CC=C)c(C(C)(C)O)nn2)CC(NC(=O)OC(C)(C)C)C2(CCC2)C1 83306,C12(C(N3CC(C)C(NC(C4(C#N)CC4(C)C)=O)C3)=O)CCCCC1OCC2 83307,C1(N(C(CCCN(C(c2c(CC)n[nH]c2)=O)C)=O)CC)CCCC(O)C1 83308,N1(C(c2ccc(CSC)cc2)=O)CCCC(CCNC(=O)C=CSC)CC1 83309,C1(C(=O)NC(C#CC#C)(C)C)CN(C(C2(C(C)C)COC2)=O)CC(C)(C)C1 83310,C(N1CCN(C(C)=O)C(C)(C)C1)N1CCCC(SC)C1 83311,Cc1c(NC(C23CC(C(=O)NC4CCCN(CC5CC5)C4)(C2)C3)=O)cnn1C 83312,C(=O)(CCCc1ccsc1)NCCN(CCC)C(c1csc(C(C)OC)n1)=O 83313,N(C(=NCCc1ncccc1C)NCc1ccc(Cl)cc1Cl)C1C(SC)C1 83314,Cc1cc2ncc(C(N3CC(NC(C4CCC(C)(F)CC4)=O)C4CC34)=O)cn2n1 83315,c1(C(N2CC(NC(C(C)OCC=C)=O)C(C)C2)=O)cccc2c1OC(C)(C)C2 83316,Cc1cc(CC(=O)NCC2CCCCN2C(=O)CCc2cccnc2)ccc1Cl 83317,CP(C)(=O)c1ccc(C(N2CCCC2CNC(=O)CSc2n[nH]c(O)n2)=O)nc1 83318,N1(C(c2cc(C)ns2)=O)CC2CCC(NC(=O)C(C)S(C)(=O)=O)(C2)C1 83319,N1(C(CCC(=O)N(C)C)=O)CCCC2(NC(c3nncn3C)=O)CC2C1 83320,c1(NCC(O)CCCc2ccccc2)ccc2nc(Cl)ccc2c1 83321,c1(C(=O)NCCCCCCNC(C(N)=O)=O)cccc2c1OCC(=O)N2 83322,c1(C(=O)NCc2cn(CCNC(c3ccn(C)n3)=O)nn2)[nH]cnc1C#N 83323,C1(C(=O)NCC(CNC(c2cccc(F)c2)=O)O)CC2(C1)CC2(F)F 83324,c1(SC)nc2ncnc(NC(CN(C(=O)C(N3CCCCCC3)C)CC)CO)c2s1 83325,c1(C(N2CC(CNC(c3cc(C)[nH]c3C)=O)C3(C2)CC3)=O)ccnc2c1CCO2 83326,c1(C(=O)NC(C2CCN(C(c3cccc(C(=O)NC)c3)=O)C2)C)cc(Cl)nnc1O 83327,C=C=C(C)CC(=O)N(C1CCN(C(=O)CN(C)C(=O)OC)C1)CC 83328,C1(C)(CNC(C2CC(CC)(CC)C2)=O)CCC(NC(=O)C=Cc2cnccn2)C1 83329,CC(C)(CNC(=O)CCCn1ccnc1)CC(=O)NC(C1CCOC1)(C)C 83330,c1(C(N2CCC3CCC(C2)S3)C(=O)NC2CCCC2)csc2ccccc2c1=O 83331,c1(C(C(=O)NC)N(C)CC2CCCS2)cc(Br)c(F)cc1F 83332,C=CC1(O)CCN(C(=O)CNC(=O)CNC(c2nn(C)cc2C)=O)C1 83333,c1(C(N2C(CCC)COCC2)C(=O)NCCC)ccc(C)c(C#N)c1 83334,N1(C(=O)Cc2ccsc2)CCC2C1CCN2C(c1cc(F)ccc1Br)=O 83335,Cn1cc(C(N2CC=CC2(C)C(N2CCCCC2CC(N)=O)=O)=O)ncc1=O 83336,c1(NC(C)=O)ccc(F)c(F)c1.c12ncccc1C(=O)CNC(=O)C(C)O2 83337,c1(C(=O)Nc2scc(-c3ccc(OC)cc3OC)c2)cc(Cl)c(Cl)cc1Cl 83338,N1(C(C2C(C)CC2)=O)CC2CC(C1)C2NC(=O)CCC(C)(C)C 83339,c1(C(=O)NCC2N(C)CCN(C(C3CCCCS3)=O)C2)cc2c(nn1)CCOC2 83340,C(CN=c1[nH]c(C2CC2)nc(=N)[nH]1)(C(C)C)NC(C(C)OCC(C)C)=O 83341,c1(C(N2CCCC(CNC(c3c(C(C)=O)ccs3)=O)C2)=O)ccc(C)c(O)n1 83342,C1(NC(C=CC(C)NC(C2CS(=O)(=O)C2)=O)=O)CCCC(O)CC1 83343,Cc1ccc(CN(C(=O)CCOCCCNC(=O)Cc2conc2C)C)cn1 83344,c1(C(=O)OCC)ccc(NC(=O)N(C2CC3(C2)CC3F)CCN(C)C)cc1 83345,C=CCC(CNC(=O)CC1CCCCCC1)C(=O)NC(C)COCC 83346,c1(C(=O)NCc2cccc(C#C)c2)cc(F)c(F)cc1F 83347,c1(OC)ncc(C2C(=O)O2)cn1.C1(C(C)NC(=O)OCC(F)(F)F)CCCCC1 83348,C1(OC)(CNC(=O)CN=[N+]=[N-])CN(C(=O)CCSC)C1 83349,c1(C(N2CC(C3(NC(=O)Cc4cccs4)CC3)C2)=O)cc2c(=O)[nH]ccn2c1 83350,C1(NC(C(C)NC(=O)NCC)=O)CC(NC(=O)CCc2ccc(F)nc2)C(O)C1 83351,C(CCN=C(NCCN1CCOCC1)NCC1(O)CCC(C)(C)CC1)SC 83352,C1(C(=O)NC(CNC(=O)C(C2CC2)C2CC2)C2CCC2)CC12CCCC2 83353,Cc1ccc(CNC2CCN(C(c3ccc(C4CC4)cn3)=O)CC2C)c(O)n1 83354,c1(CN2CCN(C(c3cccnc3C)C(=O)NC)CC2)cnc2ccsc2c1 83355,c1(CC)cc(NC2CCCC(NC(c3coc(CC4CC4)n3)=O)C2)ncn1 83356,N1(C(C2(CC)CCN(C(=O)CC(F)(F)C(F)F)C2)=O)CCC2(CCCO2)C1 83357,N1(C(c2cc(C)oc2C)=O)CCC2(COC(CNC(C3(C)CCC(C)C3)=O)C2)C1 83358,c1(C(N(CCN(C(CC(=O)OC)=O)C)C)=O)cccc2c3c([nH]c12)CCCC3 83359,c1(C(N2CCC(NC(C(=Cc3ccccn3)C)=O)C2)=O)ccc2c(c1)C(=O)NC2 83360,c1(C(N(CC(C)NC(=O)CC2CCCN(C)C2)C)=O)cccc2c1CCCCC2 83361,C12(CNC(C=C(C)C(C)(C)C)=O)CCC1CN(C(c1cc(O)ccc1Cl)=O)C2 83362,C#Cc1ccc(C(=O)NCCC(C)N(C)C(c2cc3scnc3[nH]2)=O)c(C)c1 83363,c1(COC)cc[nH]c1C(=O)NCCC1CCN(C(=O)CC2CC2F)C1 83364,C1(CN(C(CC2C(C)C2)=O)C)COCCN1C(c1ccc(N(C)C)cn1)=O 83365,C(C)(C(F)(F)C(F)(F)F)=CC(N1C2(CN(C(C3CCC(=C)CC3)=O)C2)CC1)=O 83366,C1(NC(CSCC#C)=O)CCCC(NC(C2(c3cccnc3Cl)CC2)=O)CC1 83367,C1(C(C(=O)NC2C(NC(Cc3cc(C)[nH]n3)=O)C2)C)CCCCCC1 83368,c1(N(C(c2n(CC=C)nnn2)(CCC)C2CCC2)CC)nc2c(n1C)CCCC2 83369,c1(C(=O)OC)cnc(N2CCN(C(C3CC3C)=O)C(C)C2)nc1C 83370,C1(C(F)F)(OC)CC(C(=O)NCCN(C(=O)CCCNS(C)(=O)=O)C2CC2)C1 83371,C(=O)(CCCC(F)(F)CO)NC(CNC(c1n(CC)ccn1)=O)(CC)CC 83372,Cn1cc(CCC(=O)NCC2CCC(NC(=O)CC3CCCOC3)C2)cn1 83373,c1(C(=O)NCC2N(C(C3N(C(N)=O)CCC3)=O)CCC2)ncc(C#N)cc1Cl 83374,c1(CC)c(C(=O)NCC2CCN(C(=O)CCCCN(C)C)C2)cnn1C 83375,C(CCC(C)C(=O)NCC(C)(C)CCNC(c1sccc1OC)=O)OC 83376,N1(C(c2nc(COC)sc2)=O)CCC2(CCCC2NC(c2[nH]c(C)nc2C)=O)C1 83377,C#CCCCCC(=O)NC(C)(CNC(c1cn(C2CCOC2)cn1)=O)C1CCC1 83378,C1(C(N2CC(CC(CNC(CC(=O)OC)=O)(C)C)C2)=O)CCCC12CCOCC2 83379,C1(NC(CC2N(CC)CCC2)=O)CN(C(c2cc[nH]c2)=O)CC1C(F)(F)F 83380,C(CC1CC1)(C(=O)N1CCCC1C(C)CC)NC(C(C)=C(CC)C)=O 83381,C1(C(=O)NCC2=C(C)CCC2)CC2CCC(C1)N2C(c1c[nH][nH]c1=N)=O 83382,Cc1oc(C(=O)NC2CCN(C(=O)CCc3cccc(O)c3)C2C)cc1Br 83383,C1(CC)CC(O)CN1C(=O)CC1CC(NC(=O)CC2OCCC2C)C1 83384,C(=O)(C(C)C(=O)NCC1(CC(=O)NC(c2cncs2)C)CC1)OC 83385,N1(C(CSC)=O)CC2(COC(CNC(=O)COC3CCOC3)C2)C1 83386,C1(C(F)(F)F)(NC(CC(C)(C)CNC(=O)CC2CC23CC3)=O)CCCCC1 83387,c1(OC)cc(C(N2CC(F)CC2CN(C(=O)Cc2cnn(C)c2)C)=O)n(C)n1 83388,c1(C(N2CC=C(CNC(=O)Cc3ccc(CO)cc3)CC2)=O)cc(Cl)ncc1F 83389,c1(C(C)(C)C)ccccc1C1CC1C(=O)NCCC(F)Cn1cc(C2CC2)nn1 83390,C(=O)(CCC(=O)OC)N(C(C)C(=O)NC(COC)CO)CCC 83391,c1(C(=O)NC2CN(C(CC(CC)SC)=O)CC(O)C2)cncc2sccc12 83392,c1(NC(c2n(C(C(=O)OC)C)nnn2)(C2CC=CC2)C)cc(C)cc(Br)c1 83393,c1(C(=O)NCC(c2ccccc2)NC(C(C)SCC)=O)cccc(F)c1C 83394,CC(C)CC(C(=O)N1CCCC1CCNC(=O)CC1CCC(=O)NC1=O)N(C)C 83395,C1(CNC(C(CCC)(C)CCC)=O)CC2(CCOCC2)CN1C(c1cscn1)=O 83396,N1(C(C2(C)CN(C(c3cccc(COC(C)C)c3)=O)C2)=O)CCC(O)C(F)(F)C1 83397,N1(C(C=C(C)C)=O)CC2CC(NC(c3cc(C)on3)=O)C2C1 83398,C12(C(N(CCCNC(=O)CN(C3CCC3)C)C)=O)CCC(C1)c1ccccc12 83399,N1(C(c2cc(C)nnc2)=O)CCC(NC(C2CCCS(=O)(=O)C2)=O)C2(CCC2)C1 83400,c1(NCC)ccc(C(N2CCC(N(C(=O)C(F)(F)CO)CCCC)CC2)=O)c(Cl)c1 83401,N1(C(CCS(C)(=O)=O)=O)CCC(NC(=O)CC2CCCCC(=O)N2)C(F)(F)CC1 83402,C1(C(C)(C)C#N)CCN(C(c2cc(Cc3cccs3)ccn2)=O)CC1 83403,Cn1c(C(=O)NCC2COC(CNC(=O)CCCCCF)C2)cc2occc12 83404,CN=c1[nH]c(=NCC2CCC2(F)F)[nH]c(=NCCS(=O)(=O)N(C)C)[nH]1 83405,c1(CC)nn(C)cc1C(C)NC(=O)Nc1cccc(OC2CC2)c1 83406,c1(C2C(CN(C)C(C3(CC4CCC4)CC3)=O)C2)c(F)cccc1F 83407,C1(NC(C2CCC(CNC(c3ccc(O)cc3)=O)C2)=O)CC1C1CCC1 83408,C1(O)(CN(C)C(C2CCC(F)(F)C2)=O)CCCN(C(c2ccc(C3CC3)o2)=O)C1 83409,C1(NC(C(CC)c2ccccc2)=O)CC(F)(F)CC1NC(c1ccc(Cl)cc1)=O 83410,c1(CN(C2CCC23CCNCC3)C(C2CCCCO2)=O)cccc([N+](=O)[O-])c1F 83411,C1(CC(N2CCC(C(C)(C)NC(CCCCC#C)=O)C2)=O)CCCC2(CCC2)O1 83412,C(=O)(CC(C(=O)NCC1CC(NC(c2coc(Cl)c2)=O)C1)N(C)C)OC 83413,S(=O)(=O)(c1ccc(Br)cn1)N1C(C(=O)Nc2ccccc2I)CC(F)(F)C1 83414,C1(C(=O)NC(CC)C(=O)N(C)CC2COC(=O)N2)CCCCC(=O)C1 83415,CCCC(CCCNC(=O)CC(C)Cc1cccc(F)c1)NC(C1OCCO1)=O 83416,C#CCCCC(C)C(=O)NC1CC12CCN(C(c1ccccc1C(C)=O)=O)CC2 83417,CC1(C)CC(C)(C(=O)NCCCC(F)(F)F)CN1C(C1CC1C(N)=O)=O 83418,Cc1ccc2c(C(=O)NC3C4CCC(C4)C3C(=O)O)n[nH]c2c1 83419,C1(NC(c2c(C)csc2)=O)CCCCC12CCN(C(=O)C(C)(C)C(F)(F)F)C2 83420,C1(C2CCN(C(C3CCCC3C)=O)C2)(NC(C2CC(C)=C(C)CC2)=O)CC1 83421,C1(CNC(C)(C)C)C2CCC(C2)N1C(=O)NCCc1c(C(=O)OC)cccc1 83422,C1(CC(=O)NCC(CNC(c2c(C(C)(C)C)c[nH]c2)=O)O)CCS(=O)(=O)C1 83423,C1(NC(c2c(OC)n(C)nc2)=O)COC2C(NC(=O)C(C)C(=O)C3CC3)COC12 83424,CCC(CN(C)C)CC(=O)NCC1CCN(C(c2cc(COC)[nH]n2)=O)CC1O 83425,c1(CC(=O)NCc2scc(CNC(C=COCC)=O)n2)cc(O)nc(O)n1 83426,N1(C(CC(C=C)(C)O)=O)CCN(C(=O)C(C2CCOCC2)O)C2(CCC2)C1 83427,CC(C(=O)NC(C)Cn1cc(-c2cc[nH]c(=N)c2)nn1)C(F)(F)C(F)F 83428,c1(OC)ncc(C(=O)NCC2CC(NC(C3(OC)CC3)=O)CC2O)cc1Br 83429,c1(C(=O)NC(C2NCC2)=O)cc(C(F)F)cs1.C(CCC)=CC 83430,CCCCC(C(=O)NC)NC(C12CC(CO)(CN1C(C1(CC)CCCO1)=O)C2)=O 83431,Cc1c[nH]nc1C(=O)NC(CNC(C1(C)CC1(Cl)Cl)=O)CO 83432,Cc1ccc(CCNC(C2COCCN2)=O)cn1 83433,c1(OC)ccc(C(=O)NC(C2CN(C(c3ccc(C(C)C)s3)=O)C2)C)c(Cl)c1 83434,C1(CC(=O)N(CCCCNC(=O)CCN2CCCC2)C)CCC2CC12 83435,Cc1[nH]nc2c1CCN(c1ncnc(NC(c3ccncc3)C)c1C)C2 83436,c1(CC)cc(CC(C2C(C(=O)NCc3cccc(OC)c3)C2)=O)c(NC(C)=O)[nH]1.C(C)O 83437,c1(C(=O)NCCC(C)NC(CCCOCCOCC)=O)cccc(F)c1F 83438,c1(N(C(=O)C(C)C)CCNC(c2ccc(N(CC)CC)cc2)=O)ccc(C#N)cc1 83439,C(C)(CC(C)NC(=O)C=CC(=O)NC1CC1)NC(C1(C(C)C)CC1)=O 83440,c1(C(=O)OC)cnc(OC)c(C(N2CCC(NC(c3ccccc3)=O)C2C)=O)c1 83441,c1(C(N2CC(O)CC(NC(CCc3scc(C)n3)=O)C2)=O)cc(N)c(Cl)c(O)c1 83442,c1(OCC)ncc(C(=O)N(CC(C)NC(=O)C(O)CF)C)s1 83443,CC1(C(=O)NCC2(F)CC(CNC(=O)C3CC3)C2)CC(C(F)(F)F)=NO1 83444,C(C(C)C(=O)NNC(=O)C(C(C)C)c1nc[nH]n1)OC 83445,N1(C(C(=O)Nc2cccc(C(=O)OCC)c2)C2CC2Cl)CCn2ncnc2C1 83446,C[S+](C)CCC(O)C(=O)N1CC2CCC2(CNC(c2cccc3nc[nH]c23)=O)C1 83447,C1(C(N(C2CC3CCC2O3)C)=O)C(O)CCN1C(=O)C(=C1CCCCC1)F 83448,C(c1ccccn1)=C(C)C(=O)NC(C(F)(F)F)c1ccc[nH]1 83449,c1(C(C)C)nocc1C(=O)NCC(C)(CO)NC(=O)COC1CCOC1 83450,Cc1ccc(C(=O)C(=O)N(C)CCOCCNC(=O)CCc2ncc(C)[nH]2)cc1 83451,C(CC(C)(C)CC(=O)NCC1CC(NC(c2nc(C)n(C3CC3)c2C)=O)C1)OC 83452,CC(O)C(C(=O)NCC(O)CN(C)C(c1coc(Cl)c1)=O)N(C)C 83453,C1(NC(C23N(C(c4ccc(Cl)cn4)=O)CC(C2)C3)=O)CCCCCC1F 83454,c1(C(=O)NCC2(F)CCC(NC(CCOC)=O)C2)nn(C)cc1S(C)(=O)=O 83455,C1(NC(c2cc(OC)ns2)=O)CN(C(=O)CCCn2ccnc2)C2CCCC12 83456,C#CC1(C(=O)NC2CC(OC)C2(C)C)CCN(C(C2COCC2C(N)=O)=O)CC1 83457,C12(NC(CCCCC)=O)CCCCCC1N(C(=O)CC(C)(C)CC(=O)OC)CC2 83458,C(=O)(C(C)(CC)OC(=O)C(CCSC)NC(=O)OC(C)(C)C)OC 83459,CC1(C)CC(C(N2CCn3ccnc32)=O)CN(C(=O)C=Cc2cscn2)C1 83460,Cc1cc(C(=O)NCC(O)CNC(C2CC(C)(F)C2)=O)c(C)o1 83461,N1(C(CC(CN(C)C)OC)=O)CCC(O)C(C)(O)C1.C1(C(=O)N)(C)CCCC1 83462,c1(N2CCC(CNC(c3n(C)nc(C4CC4)c3)=O)C23CC3)ncnc2c1CCC2 83463,CCCCC(C(=O)NCCCCC(=O)NC(c1cncn1C)CO)N(C)C 83464,n1(CC(=O)NC(CNC(CC)=O)(CC)CC)ccc2ccc(Br)cc12 83465,CN1C(C(=O)OCc2ccc(O)cc2F)CCS1(=O)=O.C12(CC1)C(=O)N2 83466,N1(C(c2n(CC)ncc2Br)=O)CC(NC(=O)C(C)CF)C(S(C)(=O)=O)C1 83467,c1(C(=O)NC2CCN(C(Cc3c(C)n[nH]c3)=O)CC2F)cn2ncccc2n1 83468,c1(OC)ccc(CC(=O)N(C(C)CNC(C2CCCOC2C)=O)C)nc1 83469,N1(C(c2cncn(C)c2=O)=O)CC2CN(C(=O)CSCC(N)=O)CCC12 83470,c1(C(=O)NCC(c2ccc(C)cc2)NC(C2CCC3CC23)=O)ccc(C)c(C)n1 83471,Cc1ccc2nc(C(=O)NC3CCCC(NC(=O)CC(C)N(C)C)C3)cn2c1 83472,N1(CCC(=O)NC(CNC(C(C)N(CC)CC)=O)C)CCCS1(=O)=O 83473,C12(C(=O)NCCCCNC(C3(c4ccno4)CCC3)=O)CCC(CC1)O2 83474,C(=O)(C1=C2CCN=C2NC=C1)N1CCC2(OCC(NC(c3c(C)nco3)=O)C2)C1 83475,CN1CCC(=CC(=O)NCC2CCC2NC(=O)CNC(=O)CC2CCCC2)CC1 83476,N1(C(COCC)=O)CC(F)(F)CC1C(=O)NCC1(O)CCCOC1 83477,c1(OC)ccc(C(=O)N(CC(C)(C)NC(=O)C(C)Cn2ccc(C)n2)C)c(F)n1 83478,Cc1oc(Cl)nc1C(=O)NC(C1CCN(C(=O)Cc2cnns2)C1)C 83479,C#Cc1ccnc(C(=O)N(C)CC2CN(C(C34CCCC3C4(F)F)=O)CCO2)c1 83480,C=CCC(Cc1ccccc1)C(=O)NCCCCN(CCCN)C 83481,C1(C(=O)NC(c2occ(C(N(CC(=C)C)CC)=O)n2)C)C2CC3C(C2)C13 83482,N1(C(C(C)(F)F)=O)CC2(CCN(C(C3CCCC4(CC4)C3)=O)CC2)C1 83483,c1(C(=O)NC2CN(C(c3c(C)sc(Cl)n3)=O)C(C)CC2)cc[nH]c(=N)c1[N+](=O)[O-] 83484,C1(NC(Cc2cc(C)no2)=O)CCCC12CCN(C(=O)C(O)c1ccsc1)CC2 83485,C#Cc1ccc(C(N2CCCC(C)(NC(=O)Cc3nnc(O)s3)C2)=O)cn1 83486,c1(NCC(=O)NCC(C)(CO)NC(=O)CC2NC(=O)NC2=O)ccc(F)cc1F 83487,C1(C(=O)NC(C(=O)NC(c2ccncc2F)C)C2CC2)CCCC(O)C1 83488,N1(C(c2[nH]ccc(=N)n2)=O)CCC2CCN(C(c3cc(C(F)F)no3)=O)CC2C1 83489,N1(C(C(C)OCCC)=O)CC=CC1C(=O)NCc1cc(C(=O)OC)on1 83490,c1(C(N2CCOCC2CC(c2ccccc2)O)C(=O)NCC=C)cnc(C)n1C 83491,Cn1nc(C(N2CC(c3ccccc3C(F)(F)F)(O)C2)=O)cc1C1CC1 83492,C1(CNC(c2scc(OC)c2)=O)CC(NC(=O)CCCC#N)C12CCC2 83493,N1(C(CS(=O)(=O)N(C)C)=O)CC2(CCCC2NC(C2CC3CC3C2)=O)C1 83494,c1(OC)ccc2c(c1)OCCC2NC(=O)NC1CCN(c2ccc(C)cc2)CC1 83495,c1(C(=O)NCCC(C)N(C)C(C2CC2c2ccc(Cl)cc2)=O)nc(Cl)ccc1N 83496,C(=O)(CS(=O)(=O)CC)NCC1N(C(C2CN(S(CC)(=O)=O)C2)=O)CC1 83497,N1(C(COC2(C)CCC2)=O)CCOC(CCNC(c2cc(F)c[nH]2)=O)C1 83498,c1(NC(C2N(C(C3CCC(CC)CC3)=O)CC(O)C2)=O)cnc(Cl)nc1C 83499,c1(C(N2CC(CC(C)NC(c3cscn3)=O)C2)=O)nc2c(cc1Cl)OCCO2 83500,C12(C(N3CC(F)(CNC(C4C(C)C4C)=O)C3)=O)C3CCC(CC13)C2(F)F 83501,N1(C(C(C)SC)=O)CCC(NC(c2ccn(-c3ccncc3)n2)=O)C(O)C1 83502,c1(C(N2CCC(NC(c3cccnc3)=O)C(O)C2)=O)ccn2c1CCCC2 83503,C(CS(=O)(=O)NC1(C(F)F)CCC1)(C1CCOC1)OC 83504,c1(C(=O)NCC(C)N(C(=O)Cc2nc[nH]n2)C)ccc2nnn(C)c2c1 83505,N#CC1CN(C(C2(O)CCN(C(c3cccc(C(N)=O)c3)=O)C2)=O)CCO1 83506,N1(C(c2scc(C(=O)OC)c2)=O)CCN(C(=O)C(=O)N(C)C)CC1C(F)F 83507,c1(CC(=O)NCC(C2CC2C2CC2)NC(COCC#C)=O)cccc(Cl)c1 83508,c1(OC)nccc(C(N2CCC(NC(=O)C(C)=C(C)C)C(CO)C2)=O)c1F 83509,C(C(CNC(=O)CCCCC1CC1)S(C)(=O)=O)NC(c1cc(C)no1)=O 83510,c1(OC)ccnc(C(=O)NC(C)CCN(C(=O)C(F)(F)C2(O)CCC2)C)c1F 83511,C1(NC(=O)Cc2cn[nH]c2)CCCC1Cn1cc(-c2nc(C3CC3)cs2)nn1 83512,C(CNC(=O)C(C)n1ccnc1)(CC(=O)NCC(C)C(C)O)OC 83513,c1(C(N(CCN(C(C2C(CC)CCC2)=O)C)C(C)C)=O)cc(=O)n2nccc2[nH]1 83514,CC(C)(CNC(=O)CCOCC(F)F)CC(=O)NCC1(CC2CC2)CC1 83515,CC1(C(=O)NOCC2CCCO2)CCN(C(C2CC23CC3)=O)CC1 83516,C(=O)(CCS(C)(=O)=O)NC12CC(NC(CCc3c(OCC)cccc3)=O)(C1)C2 83517,C(C1COCc2ccccc21)NC(c1ccc(OCC(C)C)cc1)=O 83518,CC(C)CS(=O)(=O)CC(=O)NCC1CC2(CO1)CN(C(=O)C(C)S(C)(=O)=O)C2 83519,N1(C(CCSCC)=O)CCN(C(=O)CCc2ccc(OC)cc2)C(CC)C1 83520,C1(NC(C2(C(N(C(C)C)C)=O)CC2)=O)CCCC1NC(=O)C1=CCC1 83521,c1(C(C)=O)cccc(OC(C)C(=O)NC2(CNC(c3c(C)coc3C)=O)CC2)c1 83522,CC1(C)C(C)(C)C1(F)C(=O)NC1CN(C(c2c[nH]ccc2=N)=O)C2CC12 83523,C1(C(N2CC(O)(CNC(c3cn(C4CC4)cn3)=O)C2)=O)(COC)CC1(F)F 83524,C1(O)(CN(C)C(c2c[nH]c(=N)o2)=O)CN(C(=O)COCCCF)C1 83525,C1(NC(c2cn(CC)nc2C(C)C)=O)CCCCN(C(C2CC23CCCC3)=O)C1 83526,C=C1CC2(C1)CC(C(=O)NC1CC3CC1N(C(C1CC(C)(C)C1)=O)C3)C2 83527,C1(N(C(Cc2c(C)con2)=O)CCF)CCCN(C(C2OCC2(C)C)=O)C1 83528,c1(CC(=O)NCC(C(C)C)NC(=O)C(C)CO)cnc2n1CCCC2C 83529,C1(NC(C(COC)O)=O)CN(C(c2ccnnc2S)=O)CC1c1ccccc1 83530,C1(SCC(=O)NC(C)CCNC(=O)CSC(F)(F)F)CCOC1=O 83531,c1(NC(N2CC(F)CC2C(=O)O)=O)cnncc1Br 83532,C1(NC(c2ccc(SC)s2)=O)CCCCN(C(C2CC3(CCO3)C2)=O)C1 83533,C1(C(=O)N(S(=O)(=O)CCCl)C(C)(C)C)CC(F)CN(C(C2C(C)CCO2)=O)C1 83534,c1(C(=O)NCC2OCCCN(C(C3N(C)CSC3)=O)C2)cccc([N+](=O)[O-])c1 83535,C1(NC(CCCn2cc(C(C)(C)F)nn2)=O)CNCCNC1=O 83536,c1(CC(=O)NC(CNC(=O)COCC2CC2)C2CCC2)ccsc1Br 83537,C(=O)(C(C)(F)C(C)(C)F)N(C)CCN(C)C(C1(F)CCCOC1)=O 83538,CC(C)CC(C(=O)NC(C)C(C)C(=O)N1C(CO)CC1CO)N(C)C 83539,N1(C(COCC=C)=O)CCC(C2CCN(C(c3cc(CSCC)on3)=O)CC2)C1 83540,CC1CNc2ccc(C(=O)NCCCOCCNC(C3CCCCO3)=O)cc21 83541,c1(CCC(N2CCC(Cn3cc(CC(C(C)C)O)nn3)C2)=O)ccc(F)cc1F 83542,C(=O)(C(F)C(C)CNC(=O)CCN1CCCC1=O)NCC(CC)CC 83543,C1(CCC#C)CCCN1C(C1CCC(CNC(=O)Cc2cc(C)[nH]n2)C1)=O 83544,c1(OC)cccc2c(C(=O)NC3CN(C(c4n[nH]cc4OC)=O)C3)c(C)[nH]c12 83545,CC1CC(CNC(c2cncn2C)=O)CN1C(c1cc(C2CCC2)nn1C)=O 83546,c1(C(=O)NC2CCC(NC(CC(CCC)(C)C)=O)C2)ncc(F)c2ccccc12 83547,CC1(CCC2CC2)CN(C)C1.c1(C(C2CC2)Sc2ccccc2)c[nH]cn1 83548,Cc1cc(Br)cc(C)c1CN1CCN(C(=O)C(C)Cn2cccn2)C(CC#N)C1 83549,N1(c2ncn(C)c(=O)c2Br)CCCC(C2CC2NC(C2(F)CC2)=O)C1 83550,N1(C(C(CNC(c2c(CC)ncnc2)=O)O)=O)CCN2CCCCC1C2 83551,c1(C(N(C2CC(NC(C3(CC#C)CCCC3)=O)C2)C)=O)ccccc1C1CCC1 83552,C1(C(N(C(CCC)C)CC)=O)CN(C(c2cnn(CCF)c2)=O)CC12CCC2 83553,c1(OC)ccc(CC(=O)NC(C)C(CO)NC(C)C)cc1[N+](=O)[O-] 83554,C1(C(N(C)CC2N(C(c3ccc(CC)cn3)=O)CCOC2)=O)CC(C)(C)CCO1 83555,C#CCCCC(C)C(=O)NC1(CNC(c2nocc2Cl)=O)CCCCCC1 83556,N1(C(C(C(=O)OCC)C2CC2)=O)CCOC2(C1)CN(C(C1(C)CCCC1)=O)C2 83557,C#CC1CCC(CN2CC(C)CC(C(=O)NCc3c(C)cccc3F)C2)CC1 83558,C1(NC(=O)CC2C3COCC23)CCC12CCCCC2 83559,N1(CCCNC(=O)CC2COC(=O)C2)CCN(C(=O)C=C(C2CC2)C2CC2)CC1 83560,CC1(CNC(C2(F)CN(C(=O)Cc3cscn3)C2)=O)NC(=O)NC1=O 83561,c1(C(=O)NCC(=O)NCC(=O)NC(c2nncs2)C)cccnc1S 83562,N1(C(c2ncc(CC)cn2)=O)CCC(CO)(CNC(c2cnsn2)=O)CC1 83563,c1(C(=O)NC2C(CNC(=O)CC3C=CCCC3)COC2)cc2scc(Cl)c2[nH]1 83564,C#Cc1cccc(CC(=O)NCc2nc(CC)ns2)c1 83565,C1(CCCCNC(CCOCC)=O)CCN(C(=O)C(O)CC2CCOCC2)CC1 83566,C#CCC(CC(F)F)C(=O)N(C1CCC(NC(=O)C2=C(Cl)CCC2)CC1)C 83567,c1(CCC)cc(C(=O)NCCN(C(=O)CCCn2cccn2)CCOC)nn1C 83568,Cc1c(CCC(=O)NC(C)CC2CN(C(=O)C(CCO)N(C)C)C2)cnn1C 83569,c1(C(=O)NC2CN(C(CCCCC#C)=O)CC(O)C2)cncc2n[nH]cc12 83570,C1(C(=O)NC(c2ccc(F)cc2F)(C)C)C2CCC(C2)C1N 83571,c1(CC(=O)N(CC(C)(C)NC(C(C)O)=O)C)cnnn1C 83572,c1(NC2CCN(CCOC)C2)cc(Br)ccc1S(=O)(=O)NCc1ccc(Cl)nc1 83573,CCC(CC(=O)N(C)CCOCCNC(c1ccc(COC)s1)=O)OC 83574,C1(C(=O)NC2C=CCC(C(N(CC)Cc3ccsc3)=O)C2)CN(C)CC(C)O1 83575,c1(C(N2CCC(C)(NC(=O)Cc3ccns3)CC2)=O)ccc2sccc2c1 83576,c1(C(=O)NCCN(CCC)C(C2(C)CCCCO2)=O)cc(CC)nn1CC 83577,CC1CCCCN1CC(N1CCC(N(C)C(c2ccc(N3CCC3)nc2)=O)C1)=O 83578,Cn1cccc(C(=O)NC(C)(C)C=CC(N2CCC3C(C(N)=O)C3C2)=O)c1=O 83579,C(C(CC1CC1)C(=O)NCC1C2CCCCC12)NC(c1ccc(CC)o1)=O 83580,c1(C(=O)NC2C(CNC(c3c(=N)cc[nH]c3)=O)C2)cccn2nccc12 83581,CC1CCN(Cc2ccc(Cl)cc2Cl)CC1NC(c1cnn(C(C)(C)C)c1)=O 83582,CCCC(CNC(C1CCCCCN1C)=O)C(=O)NC1CCCCC1CCO 83583,N=c1[nH]cc2c(c1C(N1CC3(CCN3C(C3C=CCC3)=O)C1)=O)CCC2 83584,N1(C(CCCC(C)O)=O)CCCC12CCN(C(c1cc(Cl)c(Cl)[nH]1)=O)C2 83585,C1(C(=O)NC2(C)C(C)CCC2)C2CCC(C2)N1C(c1ccc(F)s1)=O 83586,C12(C(=O)NC3CCCN(C(C(F)OC(C)=O)=O)C3)CCCCC(OC(C)C)(C1)C2 83587,CCCCCC(C)(C)C(=O)NCC(O)CNC(c1nnn(CC)c1C)=O 83588,c1(C(=O)NC2C3CN(C(c4cc(C)c(C)nn4)=O)CC32)cccc2nsnc12 83589,N1(CCC)CCCC2(CCCN2C(c2cccc3c2CCNC3)=O)C1=O 83590,c1(NC(C2N(C(C(C)C)=O)CC(F)(F)C2)=O)ccc2c(c1)C(=O)N(C)C2 83591,C=CCCCC(=O)NC1(c2ccccc2)CCN(C(=O)C(C)NC(=O)C2CC2)C1 83592,C12(COC)CCOC1CN(C(=O)C(=O)Nc1ccc(C(C)C)cc1Cl)C2 83593,c12ccc-1cc2.c1(CN(C(=O)CN2CCOC2=O)C)cc(-c2ccccc2)no1 83594,N1(C(C(CC=CC)CC)=O)CCc2cc(CNC(c3nnsc3C)=O)ccc2C1 83595,c1(C(N(C)CC)=O)cc(NC(c2ccc(-c3cccnc3)cc2)=O)cn1C 83596,c1(CC(N2CC(F)(C(=O)NCC3COCC(C)O3)C2)=O)cccc2ccoc12 83597,N1(C(CNS(N)(=O)=O)=O)CCOCC(CNC(c2ccc(-c3ccco3)o2)=O)C1 83598,C(=O)(CCCCC(C)(C)C)N(c1ccc(C2CC2)nc1C)CC.c1(=O)c(=O)n1CC 83599,CN1C(=O)C(NC(c2cccc(C#N)c2Cl)=O)c2cc(Br)ccc21 83600,N1(CC(=O)NC(C2(O)CCN(C(C3(C=C)CC3)=O)C2)C)OC(C)(C)CC1=O 83601,C(=O)(CC(C)C(=O)NCC=CCNC(=O)C=Cc1ccc(OC(F)F)cc1)OC 83602,N1(C(C(C)C(F)F)=O)CCN(C(C2(C#N)CCSCC2)=O)CC1CF 83603,N1(C(C2C3CN(C(C4N(C)CC(O)CC4)=O)CC32)=O)CCC12CCOCC2 83604,N1(C(N2CCN(c3ccc(-c4ccc(CN)cc4)cc3)CC2)=O)CCC12CCOC2 83605,C=C1CC(C(=O)NN2CCOCC2)N(CCC23CC(c4ccccc4)(C2)C3)C1 83606,CC(C)S(=O)(=O)C(C)C(=O)NCC(C)(C)NC(=O)Cn1cc([N+](=O)[O-])ccc1=O 83607,c1(NCCCSCC)oc(C)nc1C(=O)NC1CCCCC1 83608,C#CC1CN(C(C2(NC(C3CC3(F)Cl)=O)CCSC2)=O)CCO1 83609,C1(C)(C(N(C)OC2CCCC2)=O)CCCN1C(C1COC(=O)N1)=O 83610,C1(C(N(C2CCN(C(C3(CO)CC3(F)F)=O)C2)C)=O)CC2(CCC2)C1 83611,c1(N2C(CCNC(Cc3cncc(C)c3)=O)CCC2)ccc2c(n1)CCC2=O 83612,C1(CNC(C(CCC)F)=O)N(C(=O)CN2CC(C)(OC)C2)CCCC1(C)C 83613,N1(C(C)=O)CC2(C1)CN(C(=O)C(CC(F)F)N(C(=O)C=CC(C)(C)C)C)C2 83614,C1(C(=O)NCC2N(C(c3c(C)ccc(N)c3)=O)CC2)CCCN1S(=N)(=O)N(C)C 83615,N1(C(C2CCC(O)C2)=O)CCC(F)(C(=O)N(C2CC2)CC2CCOC2)C1 83616,CC(C)C(F)C(=O)NC1(CNC(c2cscc2C#N)=O)CCOC1 83617,C(c1ccc(S(N)(=O)=O)cc1)=CC(=O)NC(CCNC(C(CC(C)C)C)=O)C 83618,CC1C(=O)NC(=O)CN1C(=O)C(CN=[N+]=[N-])NC(c1ccc(C(N)=O)o1)=O 83619,N1(C(CC2C(NC(C3C=CCC3)=O)CCCC2)=O)CCCC12CCOC2 83620,c1(C(=O)NCC2CC(NC(CC(COC)(C)O)=O)C2)ccc(P(C)(C)=O)s1 83621,Cc1nnc(CNC(C2CCC(NC(C3CCCCC3)=O)C2)=O)o1 83622,C(=O)(C1=CCCOCC1)NC(C(C(=O)NC1(CC)CCOCC1)C)C 83623,C(=O)(C(CO)C(F)(F)F)NC1CN(C(c2cccc(C(C)(C)C)c2)=O)CC1SC 83624,CC1OCCC1CC(=O)NCc1cn(C2CN(C(=O)CNC(=O)C3CC3)C2)nn1 83625,c1(OC)ccc(CC(=O)NC2CCC2NC(c2sc(N)nc2C)=O)cc1F 83626,C1(C)(C(=O)NCC(CNC(c2nn(CC)nc2C)=O)C)COCC1(F)F 83627,C=CCC(CNC(=O)C(C)(C)COC)C(=O)Nc1cncc(C(N)=O)c1 83628,CCCC(CCC)C(=O)NCC(c1ccccc1CC)NC(c1c[nH]nc1C)=O 83629,Cc1cnc(CC(=O)N(C(CNC(=O)CCCN2CCCCC2)C2CC2)C)s1 83630,N1(C(CCOCC(C)C)=O)CC(NC(C2C3CCCCCC23)=O)CC(F)C1 83631,CC(C)CCCCN(C(=O)C(n1cc(-c2cnc(C3CC3)s2)nn1)C)C 83632,C1(C(=O)NCC(CC)(CC)NC(=O)Cc2ccc(C)c(O)c2)CC12CCSCC2 83633,C(=O)(C(CCOCCO)NCCCCC)NCCNC(=O)C(C)n1ccnc1 83634,N12CC3(CC(F)(C1)C3)OC1CCN(CC1O)C2=O.C(C(F)(F)F)OC(C)(C)C 83635,Nc1c(C(=O)NC2C3CN(C(C4CC5CC5C4)=O)CC23)ccc(F)c1Cl 83636,C1(CCNC(=O)C(=O)NCC2CCCC(C(=O)OC)N2)CCc2ccccc2N1 83637,c1(C(=O)NC2C(NC(=O)Cc3cncn3C3CC3)C2)cc2ccccn2n1 83638,N1(C(C=Cc2ccc(C)o2)=O)CC(NC(C2CN(c3nnnn3C)C2)=O)CC(C)C1 83639,Cc1ccccc1OCC(=O)NC1CC(NC(=O)OCC(C)CO)C1 83640,C1(C)(CNC(COC(CC)C)=O)CCCN(C(c2cc(C(C)(C)C)n[nH]2)=O)C1 83641,N1(C(C(C(C)(C)C)n2ccnn2)=O)CCCC(C2(NC(=O)CC3CC3)CC2)C1 83642,O=C(CCCCn1ccnn1)NC(C1(CC(N2CC3(CCC3)C2)=O)CCCCC1)=O 83643,N1(C(N)=O)CCCC(N=c2[nH]c(=NCCc3cnc[nH]3)c3cccc(F)c3[nH]2)C1 83644,C(=O)(C(=O)N=S(C)(C)=O)N1CCC(C)(NC(C2C(=C)CC2)=O)C1 83645,C1(CNC(C2(CC(C)C)COC2)=O)CN(C(=O)CC2CC(O)C2(C)C)CC1C 83646,C(=O)(C#CC1CCCCO1)N1CC(CC(C)NC(C(C)NC(C)=O)=O)C1 83647,CC(C)CC(CC(=O)N1CCCC[Si](C)(C)C1)NC(=O)CCCNC(N)=O 83648,N1(C(CSCCOC)=O)CC2(CNC(=O)C=CC=C(Cl)Cl)CC(F)(C1)C2 83649,CCC(C)C(C(=O)NC1CCN(C(=O)C(F)C(C)(C)O)C(C)C1)OC 83650,c1(CCC)nnc(N2CC(O)(C(C)NC(=O)C(C)SCC3CCCO3)C2)s1 83651,c1(C(C)NC(C2CCN(C(=O)CCCC3CC3C)C2)=O)nn(C)cc1O 83652,C1(NC(C(c2ccc(Cl)s2)C)=O)CN(C(c2cncc(O)c2)=O)CCC1CO 83653,C1(NC(CC(C)(C)C)=O)(CO)CCCN(C(=O)C(F)CC2CCCCC2)C1 83654,c1(OCC)cc(C(=O)NC2CC(NC(=O)CCCOC)C2)ccc1C 83655,C1(CC(=O)NCC2CN(C(=O)Nc3ccc(Cl)cc3)C3CC23)CN2CCC1CC2 83656,C12(NC(CN(C)C(=O)OC(C)(C)C)=O)CCC(NC(C3(Br)CCC3)=O)(CC1)CC2 83657,N1(C(C(N2CCC(C)C2)=O)=O)CCCC(C)(NC(c2cncc(N)c2)=O)C1 83658,c1(C(N(C2(CC(=O)NCc3ccon3)CC2)C)=O)cnnn1C 83659,c1(CC(=O)NC2(C(N3CCC3C3CCCCC3)=O)CCOCC2)ccc(F)nc1 83660,CCCCCC(C)CC(=O)NC(CCN(C(=O)CCS(C)(=O)=O)C)C(C)C 83661,C1(CNC(CCC(N)=O)=O)(NC(C2CC(=O)N(CCF)C2)=O)CC2CCC1CC2 83662,c1(-c2cc(C(CC)C)no2)nc(-c2ccnc(Cl)c2)nn1C1CCCCC1 83663,CC1CN(C(C2C3CCC2(c2ccco2)C3)=O)CC1CNC(=O)CN(C)C 83664,C1(C2CN(C(=O)COc3cccc(Cl)c3Cl)C2)(NC(c2nc(C)nn2C)=O)CC1 83665,C1(C(=O)NC(C(C)C)c2nc[nH]n2)(CC)CCCN1C(c1ccncn1)=O 83666,c1(OC)cc(CNC(c2oc(CNC(c3c(C)nsc3N)=O)nc2C)=O)ncn1 83667,CC1CC(C(=O)NC(C)(C)CN(C(=O)COc2ccc(CO)cc2)C)C(=O)O1 83668,C#CC(CNC(=O)CCCC(C)NC(c1ncc[nH]1)=O)CC(C)(C)C 83669,CCC(Cc1cn(CC2CCCN2C(c2nscc2C)=O)nn1)C(=O)NC 83670,C(=O)(C#CC1CCC1)N(C1CCN(C(CC(C)(O)c2ccccc2)=O)C1)C1CC1 83671,C(=O)(C1=NNC(C(F)(F)F)C1)N(CC(C)NC(CCC(=O)c1ccc(C)s1)=O)C 83672,N1(C(CCC(C)OC)=O)C2CCC1CC(N(C(=O)CCc1cc(C)no1)C)C2 83673,Cc1noc(N)c1C(=O)NCc1cc(C(=O)NC(C)Cc2ccccn2)n(C)n1 83674,C1(NC(C(CCCNC(C)=O)C)=O)CCSC12CN(c1cc(C)nc(C)n1)C2 83675,c1(C(N2CCC(C)(CNC(c3ccccc3)=O)C2)=O)cc(=O)c2ccccc2o1 83676,C1(OC)CN(C(c2ccc(C(C)C)cc2)=O)CC1NC(c1scnc1C)=O 83677,c1(OCC)ccc(C)nc1C(=O)NC(C)CN(C)C(c1[nH]ccc1CN(C)C)=O 83678,N#CC1CN(C(=O)CC2CCN2C(=O)C2=CCOCC2)CCO1 83679,C(=O)(C1=CC2CCCCCCC12)NCCC(C)NC(=O)C(c1cccc(F)c1)C 83680,N1(C(C(C2CCCCC2)C)=O)C2CCC1C(F)C(NC(c1cc(Cl)n[nH]1)=O)C2 83681,C(C(=O)C(N)C(C)(C)C)NC(c1ccc(N(C)C)cc1)C 83682,N1(C(C(C=CC)O)=O)CCC(C=CC(=O)NC2(COC)CC=CCC2)CC1 83683,c1(C(c2nnnn2C)NC)cc(F)c(F)cc1NC(c1c(F)cccc1Br)C 83684,c1(CNC(c2n(C)cnc2Br)c2nnnn2CC(F)F)cccn2ccnc12 83685,c1(C(=O)NC2(CNC(C(c3ccccc3)OC)=O)CCOC2)cccc(C)c1Cl 83686,Cc1occc1C1CC1C(=O)NCC1C=CCN1C(c1c[nH]c(=N)s1)=O 83687,Cc1nc(C)c(C(N2CC3(COC(CNC(C4CN(C)C4)=O)C3)C2)=O)c(C)n1 83688,CC1CN(C(=O)CS(N)(=O)=O)CC1(C)CNC(c1sc2nc1-2)=O.C(F)(F)F.CCC 83689,C=CC1OCCC1C(N1CCC2C(NC(=O)CCn3cccnc3=O)C12)=O 83690,N1(C(c2c(C#C)c[nH]n2)=O)C2CCC1CN(C(c1ncn3c1CCC3)=O)C2 83691,C1(C(=O)NCC2CC(C(C)C)C2)(NC(=O)C(C)c2cc[nH]n2)CCN(C)C1 83692,C(=O)(C1CCOc2ccccc21)NC(CNc1c(C#N)nccn1)C1CC1 83693,c1(C(=O)NC2(C)CN(C(C3CCCN(C)C3)=O)C2)cnn2ccn(C)c12 83694,c1(OC)cc(C)cc(C(=O)NC2(CN(C)C(C34CC3CNC4=O)=O)CC2)c1N 83695,N1(C(CC2(OC)CCC2)=O)CC(C)CN(C(c2cncc(C)c2Cl)=O)CC1C 83696,C(=O)(C(F)(F)CC(C)C)NC1CCN(C(c2n(CC)cnn2)=O)CC1C 83697,N1(C(CO[Si](C)(C)C)=O)CC2(CCCC2CC(=O)Nc2cc3cc[nH]c3cn2)C1 83698,C1(C2CCC2)(CNC(C(C2CCC2)OCC)=O)CCN(C(c2cnsn2)=O)CC1 83699,c1(C(N2CC(NC(c3n(C)cc(Cl)c3)=O)C(F)C2)=O)ccc2sncc2c1 83700,C(CC(CC)C(=O)N1CC(O)(C(C)(C)CNC(=O)COC(F)F)C1)=CC 83701,C1(NC(c2ccc(CNC(=O)C(F)F)nc2)=O)CC2(C1)CC(O)C2 83702,N1(C(c2c(OC)nc(C)s2)=O)CCN2C(=O)N(C)C(=O)C2C1 83703,C=CC(C)(CCOC)C(=O)NCC1(C(=O)NCC(C)(C)C#N)CC1 83704,Cc1cc(C)c(C#N)c(NC(C)CN(C)C(c2c[nH]cc(C)c2=O)=O)n1 83705,S(=O)(=O)(c1cccc(=NCC2CCOC(C)(C)C2)[nH]1)NCC1CCCN(C)C1=O 83706,C1(CNC(C(C)C2(O)CCC2)=O)CC(C(=O)N2CCOCC2C(N)=O)=NO1 83707,N1(C(=O)NCC(c2ccncn2)(C)C)CCOC2c3ccccc3OCC12 83708,N1(C(C(COC)C)=O)CC(NC(c2cn3ncccc3n2)=O)CCC(O)C1 83709,c1(OC)nc(C(=O)NCCCC(C)(C)NC(=O)C(C)N2CC(C)C2)sc1C 83710,C(C1CCCO1)=CC(=O)NCC1CCN1C(=O)CC1(C2CC2)CCC1 83711,C12(NC(CC3(COC)CCOCC3)=O)CCN(C(=O)CSC(C)(C)C)CC1C2 83712,Cc1cc([N+](=O)[O-])cn(CC(=O)N(C)Cc2ccc(C(F)(F)F)cc2F)c1=O 83713,c1(C(N2C(CC(=O)NC)CC2)=O)ccc(C(=O)NC(C2CCCOC2)C)cc1 83714,N#Cc1cccnc1NC1CC(C(=O)NC2CCCC2)C1.C1(N)CCC(CN)CC1 83715,c1(C(=O)NC2CCC(C)(CNC(CC=C=C)=O)C2)ccc2cc(F)ccc2n1 83716,c1(OC)cccc(C(=O)NCC2CCN(C(=O)CCC3CCC3)CC2)c1 83717,C(=O)(C1CCCc2nncn21)N(CCC)CCNC(=O)Cc1ccnc(O)c1 83718,c1(OC)cc(Cl)c(C)cc1C(N1CCCC(NC(c2c(Cl)ccnc2C)=O)C1)=O 83719,c1(CCC)cc(C(=O)NC2CC3(C2)CC3NC(=O)C(O)C2CC2)nn1C 83720,N1(C(C(C)(C)C)=O)CC2CCCC2(Nc2cc3nncn3cn2)C1 83721,C1(NC(c2scc(COC)c2)=O)CC2CCC1(Cn1cc(-c3cc[nH]n3)nn1)C2 83722,C12(NC(c3[nH]cc(C#N)c3)=O)CC3CCC(C1C2)N3C(=O)CN1C(=O)CCC1=O 83723,N1(C(C(=O)NCC(=C)C)C)CCCC(C(C)NC(=O)C=C(C)C2CC2)C1 83724,C1(CCC(=O)NC(CC#C)CO)CCCCN1C(=O)Cc1csnn1 83725,CC1(C)OC(=O)CC1C(N1CC(NC(=O)CCSc2ccccc2)C2CC2C1)=O 83726,c1(COC)c(C(=O)N(C)C(c2cn(CC(O)CC)nn2)C)oc2ccccc12 83727,CCC(C)(C(=O)NC1CCCCC1NC(c1cnc(C(C)(C)C)s1)=O)OC 83728,c1(C(=O)NCC2C(NC(C3C(CC)C3)=O)CCC2)cccn2c(O)nnc12 83729,CC(C(=O)NCCN(C(=O)CCC(F)(F)F)C1CCCCCC1)C(C)(C)C 83730,C1(COC)(CNC(=O)C(F)(F)COC)CCCN1C(C1CCSC1)=O 83731,C(C(=O)NNC(=O)C(N)CC(F)F)N1CC(=O)N(Cc2cnn(C)c2C)C1=O 83732,CC(Cl)(Cl)C(=O)NCC(CO)NC(=O)CCC1CCC1 83733,c1(OC)nc(C(=O)NC2CC3CCC2CC3OC)cc2ccc(Br)cc12 83734,N(C1CC(C)n2ncnc21)C(C(=O)Nc1ccc(OC)c(-n2nnnc2C)c1)=O 83735,Cn1ncc(C#N)c1C(=O)NC1CC(O)CN(C(C2CCC(OC(F)F)CC2)=O)C1 83736,c1(C(=O)NCC(C)(CO)NC(c2n[nH]c(C)c2Br)=O)nccc(Cl)c1F 83737,N1(C(c2cc(CNC(C3(OC)CCCC3)=O)[nH]n2)=O)CC(C(N)=O)OC(C)C1 83738,c1(OC)cccc(CNC(C2(NC(=O)CCC(C)C)CC2(C)C)=O)c1 83739,N#CC1(CC(N2CCCC(O)(CNC(=O)CC3CCC4CC34)C2)=O)CCOCC1 83740,N1(C(CCc2ccn(C)c2)=O)CCC2(NC(=O)C3=NOCC3)CCCCC12 83741,c1(NC(=O)NS(c2c(C)onc2O)(=O)=O)noc2c1CC(C)(C)CC2 83742,c1(C(=O)NCC(C)(C)NC(c2ncnc(C)c2C)=O)ccc2cccnc2c1N 83743,c1(C(=O)NC(C(=O)NCc2c(C)cccn2)CCC2CC2)cc2ccccn2n1 83744,c1(CC)cccnc1C(=O)NC(c1ccnn1C)C(N1CCC(NC(C)=O)C1)=O 83745,N#CC1CCC(NC(=O)C(=O)Nc2ccnn2C2CCOC2)C1 83746,C(C(=O)N1CCC(CO)C(NC(=O)CC2(CS(C)(=O)=O)CC2)C1)(C(C)(C)C)OC 83747,C(=O)(CC(C)(C)c1ccccc1)NCC(CNC(C(CC)n1nccc1C)=O)C 83748,N1(C(C2CCC(OC)CC2)=O)C(C)C2CC1C2NC(=O)CCCCn1ccnn1 83749,C1(COC)CN(C(c2ccc(Cl)cn2)=O)CCN1C(=O)CC1CCCCN1C 83750,C1(NC(C(COCC)C)=O)CCCCC1CNC(=O)CC1CS(=O)(=O)C1 83751,CC1CC(n2nnnc2N2CC(O)CC(O)C2)CC(C)(C)C1.c1(C)ccccc1 83752,c1(-n2cc(CC(CO)N(C(CC3(CC(=O)O)CC3)=O)CCO)nn2)ccc(Br)nc1 83753,Nc1c(-c2nc(CC(N3CCCC3)=O)no2)sc2nccnc12 83754,C(=O)(C1=NNC(=O)CC1)N1CC(C)C(CCNC(=O)CC2CCN(C)C2=O)C1 83755,C1(CC#C)(C(=O)NCCCC(C)O)CCN(C(=O)COC2CCCCC2)C1 83756,N1(C(c2c(C)cc(Cl)cc2)=O)CCN(C(=O)C=CC2CC2)C2CCC12 83757,c1(C(N(CCC(C)NC(c2cnn(C(F)F)c2)=O)C)=O)ncnc2c1CCCC2 83758,N1(C(C(C)OC)=O)CCCC2C1CCN2C(c1cc(Br)c(C)cc1F)=O 83759,c1(OC)nc(Br)ccc1C(N1CC(NC(=O)CNc2ccccc2Br)C1)=O 83760,C(Cc1ccccc1)(C(=O)N(C(C)CO)CC)NC(N(CC)CC)=O 83761,N1(C(C(C)N(CC)CC)=O)CC2CCN(C(C3CN(C)CCN(C)C3)=O)CC12 83762,c1(C(N2CCC(C=C)C2)C(=O)NCc2ccccc2Br)cc(S(N)(=O)=O)co1 83763,CC1C(C)CCCN1C(=O)C(=O)Nc1nnc(C(C)(C)C)s1 83764,C1(C(=O)Nc2cnc(OC)nc2)(NC(=O)CCc2cn(C)nn2)CCC(C)(C)C1 83765,C1(OC)(OC)CCOCC1NC1C=CC(CSC)C1 83766,C1(C(=O)NC(c2cn(C(c3ccccn3)OC)nn2)(C)C)COCC1C1CC1 83767,c1(N(CC(Cc2ccccc2)N2CCCC2)C)cc(NC2CC2)ncn1 83768,N1(C(C2OCCC(C)C2)=O)CC(NC(c2c[nH]nc2F)=O)CC2(CCOCC2)C1 83769,C1(C(=O)NC(CNC(C2(CC=C)CC=CC2)=O)CO)CCc2nncn2CC1 83770,c1(C(N2CCN(Cc3cccc(OC)n3)C3C2C3)=O)cc([N+](=O)[O-])ccc1C 83771,CCC(CCC(=O)Nc1cnc(F)cc1C)NC(=O)C(C)COC(C)=O 83772,C1(CC(=O)NC23CC(NC(CC=C)=O)(C2)C3)CCC2(CCC2)O1 83773,C1(NC(C(C)c2cccs2)=O)CC2CCCC(C1)N2C(c1nccs1)=O 83774,N1(CC(=O)NCCC2CN(C(c3c(COC)cc[nH]3)=O)C2)CCCCCC1 83775,N1(C(C(C)=C2CCCC2)=O)CCCC2(CCC(NC(c3n[nH]cc3Cl)=O)C2)C1 83776,C1(CC(N2CCC(=CCC)C2)=O)CCCN(C(=O)C(C)OCCCC)CC1 83777,n1(C(C)C)nccc1-c1nnc(NC(=O)CCC2CCCC2)s1 83778,c1(CNC(C(C)=CC=C)=O)cc(C(=O)Nc2ccsc2C)on1 83779,C1(CC(=O)N(CC(C)NC(C(C)=C(CC)C)=O)C)CCc2ccccc2C1=O 83780,C1(C)(C(=O)NC2CC(C)(NC(c3cc(C)sc3)=O)C2)Cc2ccccc2NC1=O 83781,C#Cc1ccnc(C(=O)N(CC(=O)N(C)Cc2c(C)cnn2C)C)c1 83782,c1(C(N2C(CNC(Cc3cccc(OCC)c3)=O)C=CC2)=O)cnc(C)[nH]c1=N 83783,CCC(C)(O)C(=O)NC(CO)C(C)NC(c1cncc(NS(C)(=O)=O)c1)=O 83784,C1(CNC(CC(C)C2CCCO2)=O)CCCN(C(c2c(C3CC3)cnn2C)=O)C1 83785,C(C(F)(F)C(=O)NC(C)C(c1ccccc1)NC(C1CN(S(C)(=O)=O)C1)=O)OC 83786,C1(C(=O)NCC(CC)NC(c2ccc(O)cc2C)=O)CCN2CCOCC12 83787,C12(NC(C(C(C)C)C)=O)CCCC1N(C(=O)CCCC(=O)c1ccccc1)CC2 83788,Cc1cc(NC(C2CN(C(c3ccc(C)c(F)c3)=O)CCN2)=O)c(O)c(C)c1 83789,N1(C(C(C)NC(C)=O)=O)CC2CC(C)N(C(c3cnn(C(F)F)c3)=O)C2C1 83790,N1(C(C2CN(C(=O)OC(C)(C)C)C3CCN2C3)=O)CCC(O)C2(CCOCC2)C1 83791,N1(C(CSC)=O)C(C(=O)NCC(C)S(C)(=O)=O)CCC12CC2 83792,c1(COC)ccccc1CC(=O)NCC1CCC1NC(c1ccc(OC)o1)=O 83793,C1(C(=O)NCc2c(CC)nccn2)CN(C(C2(CC3CC3)CCC2)=O)CC12CC2 83794,C1(NC(CCC=CC)=O)C2CC1CN(C(c1cc(N3CCCC3)nc(Cl)c1)=O)C2 83795,n1(CC=C)cc(C(=O)NCCC(=O)NC(C(C)(C)O)C2CC2)nn1 83796,Cc1cccc(-c2noc(C(N3CCN(C(=O)OC(C)(C)C)CC3=O)C)n2)c1C 83797,N1(C(c2n(C)c(S)nc2)=O)CCC2(CCC(NC(=O)CC3(C)CCC3)C2)CC1 83798,Cc1nc(N)cnc1C(=O)N(C)CCOCCNC(=O)Cc1cnnn1C 83799,c1(C2C(C(=O)NC3C=CC(CNC(C(CC)=CC)=O)C3)C2)cccc(Cl)c1 83800,C1(C(=O)NC2(CNC(CN(C3CCC3)C)=O)CCC2)COCC(=O)N1C(F)F 83801,CC(C)S(=O)(=O)C1CCN(C(c2cc3cc(Br)cc([N+](=O)[O-])c3o2)=O)CC1 83802,Cc1ncc(C(=O)NC2CC2CNC(c2cccc(C(C)(F)F)c2)=O)c(C)n1 83803,C1(CNC(c2ncncc2Cl)=O)CN(C(=O)C(F)(F)CC2CCCO2)CCC1(F)F 83804,Cc1cc(I)ccc1NC(=O)NCC1CCOC(C)(C)C1 83805,C(C(=O)N1CCC(CNC(C2(C(=O)N(C)C)CC2)=O)C1)(C(C)C)SC 83806,c1(OCC(N2CCC(C(=O)NC(c3ccccc3O)C)C2)=O)ccc(Cl)cc1 83807,C(C(C(=O)NCC(C)CN1CCCC1)C(C)C)NC(CC(C)C)=O 83808,C1(NC(CCCN(C)C)=O)COCCC1C(=O)NCC(CO)C1CCC1 83809,n1(CC)c(NC(=O)NC2CC3OC(C)(C)OC3C2)nc2c1CCCC2 83810,CC1CN(C(c2ccon2)=O)CC1CCNC(C12CSCC1C2)=O 83811,C(C(O)C(F)(F)F)N(C(=O)C(C)CN(C)Cc1ccccc1)CC(=O)OC 83812,c1(OC)cc(NC(C2CCCCN2C(=O)CCC2CC(F)(F)C2)C)ncn1 83813,c1(C(N2CCC(C)(CNC(C(CCSC)NC(N)=O)=O)C2)=O)cccc(F)c1F 83814,N1(C(CSCC#C)=O)CCN(C(c2ccccc2C)=O)C(CF)C1 83815,C(=O)(C#CC1(C(F)(F)F)CC1)N1CC(C(C)NC(c2c(CC)noc2)=O)OCC1 83816,Cc1ccc(F)c(C(=O)NCC2CCC(C(=O)NCC(C)(C)O)C2)c1 83817,C1(NC(c2coc(Cl)n2)=O)CC2CCC1(CNC(C1CC1CF)=O)C2 83818,N1(C(c2ocnc2C)=O)CCC(F)(F)C(CC2CCOC2)C1.CC(C)(C)O 83819,CC(C)C(C)CC(=O)N1CC2CC(C1)C2NC(=O)CC1COCCN1C 83820,N1(C(=O)C=CCOc2ccccc2)CC2CC(C1)N2C(=O)Cn1cccc1 83821,C1(CNC(C(CC)F)=O)CCN(C(=O)Cc2ccc(C3CCC3)cc2)CC1(F)F 83822,c1(C(=O)NCC(C)CN(C(=O)C(C)(C)C(C)(F)F)C)c[nH]c2ccccc12 83823,c1(C(=O)NCc2cc(C(N3CC4CC(C3)O4)=O)ccn2)cccn2nccc12 83824,C1(C(=O)NC(C)CCNC(=O)CCCNC(N)=O)CC(=O)N(c2cnn(C)c2)C1 83825,Cc1ncnc(N2CCCC(NC(c3cc(=O)n(C)cn3)=O)C2C)c1F 83826,C(CC(C(=O)NC(C1CCOC1)CO)NC(c1sc(C)cc1C)=O)OC 83827,C(=O)(C1CSc2ccccc21)NC1CC(NC(C=C(CC)CC)=O)C1 83828,C(=O)(C(N=[N+]=[N-])C(C)C)NCC1(C(=O)NCc2ncc(C)nc2)CC1 83829,C1(NC(=O)OC(C)(C)C)CCC(C(=O)NC2CCN(C3CCCC3)C2)CC1 83830,CCC(CC)C(C)C(=O)N1CCCC(CCNC(=O)C(C)C2CCCO2)CC1 83831,Cc1csc2cc(CNCC3CN(C(=O)OC(C)(C)C)CCN3C)[nH]c12 83832,C1(COC)(NC(=O)C=CS(C)(=O)=O)CCN(C(=O)C=Cc2cscn2)CC1 83833,CC(C)C(O)CNC(=O)CCOCCNC(=O)CCc1nccs1 83834,Cc1cc(C(F)F)n(CC(=O)NCC(O)CNC(=O)C(c2cn(C)nc2C)O)n1 83835,c1(-c2ncc(NC3CC(c4ccccn4)C3)s2)ccc2c(c1)OCCO2 83836,Cc1noc(C(C)(C)NC(C2CC(N(C(=O)CCn3cnnn3)C)C2)=O)n1 83837,C(=O)(C#CC1CCOC1)NC1CCC(C)(CNC(CCS(=O)(=O)N(C)C)=O)CC1 83838,C#CC1(C(N2CC(C)(CSC)C2)=O)CN(C(=O)CN2C(=O)CNC2=O)C1 83839,C1(NC(c2c(OC)n[nH]c2)=O)CCN(C(=O)CC(C)F)CCC1(F)F 83840,C(CC(=O)N1CCCCC1C(C)(C)O)(C(C)C)NC(c1cc(C)on1)=O 83841,C1(C(C)C)C(O)C(=O)N1C1CC1.N1(C(CC)=O)CC(C)(CF)C1.CO 83842,C1(NC(C2CC(=O)NC(=O)C2)=O)CN(C(=O)CCCN2CCCC2)C2CCCC12 83843,C(=O)(C(C)CC(C)(F)F)NCCN(CCC)C(c1cc(C)c(C#N)cn1)=O 83844,CC(c1ccccc1)=CC(=O)NC(CC(=O)NCCC1NC(=O)NC1=O)C(F)F 83845,C1(C(N2C(CN(C(=O)C(C)(C)n3cccn3)CC)CCC2)=O)CCS(=O)(=O)N1C 83846,N1(C(C(=O)NC(C)C)c2ncco2)Cc2cccc(F)c2C1 83847,CC(C)CN=c1[nH]c(N2CCN3C(=O)CCC3C2)nc2c1CCCCC2 83848,C1(CNC(=O)Nc2nc(C3CC3)nc(=N)[nH]2)(Cc2ccccc2)CC2CCC1C2 83849,N1(C(C2(C(C)C)CCC2)=O)CCCN(C(=O)C=CBr)CC1CO 83850,CCC(C)C(C)C(=O)NC1(C)CCN(C(=O)C(C2CC2)N(C)C)C1 83851,N1(C(Cc2ccc(SC)cc2)=O)CCC(NC(=O)CCCCCF)CC1C 83852,C12(CCCC1)C(=O)N2C1CCC1.c1(C(=O)O)cn(CC(C)C)nn1 83853,C1(NC(CCc2c[nH]c(=N)[nH]2)=O)CC2CC1CC2NC(=O)CN1CC=CC1 83854,c1(CC)onc(C)c1CN(C1CCCN(C(=O)C(C)N2CCC2)C1)CCO 83855,C1(C(=O)NCC(C)(C)OCCNC(C2(COC)COC2)=O)CCC(=O)N1C 83856,S(=O)(=O)(c1ccc(F)c(-c2ccc3c(c2)OCO3)c1)C(N1CCCCC1)=O 83857,C(CC(=O)N(C)CC1(C)CCCC1)(C(C)(C)C)NC(Cc1c(C#C)cccc1)=O 83858,C1(C(N2CCC(CC)C2CNC(=O)Cc2cn[nH]c2)=O)CN2CCCC1C2 83859,C1(C(=O)Nc2c(F)ccc(SC)c2)COC2(CCN(C(N3CCCC3)=O)CC2)C1 83860,C1(NC(=O)Cn2cc(CO)nn2)CCCCN(C(c2ccc(F)nc2)=O)C1 83861,C(CCCCC(=O)NC1(CCCNC(=O)C(c2ccccc2)O)CC1)SC 83862,c1(C(=O)NCCC2CN(C(C3CC(C(C)C)C3)=O)C2)ccc(S(=O)(=O)CF)cc1 83863,C1(C(N(CCCNC(C(C)Cc2cnco2)=O)C)=O)CCC(O)CC1 83864,N1(C(C2CCCCN2C(C2CS(=O)C2)=O)=O)CCC(C2=NOCC2)C1 83865,Cn1cccc1C(=O)N(C1CCN(C(C2CCC2)=O)C1)CC1CC1 83866,C1(COC)CCCCC1C(=O)N(CCCCO)C.C12CC1C(=O)NCC2 83867,C1(C(=O)NCCC2(C)CCN(C(CC3C(C)CC3)=O)CC2)CCc2c[nH]nc2C1 83868,C(CCC(O)C(=O)NCCC(C)N1CCCC1)NC(CC(C=C)C)=O 83869,C(CC(C(=O)NOC(C)C)NC(c1cnc(C)o1)=O)=CC 83870,Cc1ccsc1CN(C)C(C1CC(NC(=O)COc2cccnc2)C1)=O 83871,N1(C(C2C(C(=O)Nc3cccc(OC)c3Br)C2)=O)CCC2(C1)CC2(F)F 83872,C1(COC)(NC(=O)CC2CNC(=O)C2)CCCN(C(C2(C(=O)OC)CC2)=O)C1 83873,Cc1nc(C)n(CC(N2CC(NC(=O)CC3CCC3(C)C)C(C(F)F)C2)=O)n1 83874,c1(OC)ncc(C(N2CCCC(CNC(=O)C(C)(F)F)CC2)=O)cc1C(F)(F)F 83875,N1(C(C(c2ccc(Cl)cc2)N(C)C)=O)CC2CCC(CNC(=O)C=CCO)(C2)C1 83876,Cc1cc2cc(C(=O)NC3CC(NC(=O)C=CC4C(C)C4(Cl)Cl)C3)oc2cc1C 83877,N1(C(CN=S(C)(C)=O)=O)CC2CC(C1)N(C(=O)Cc1cnc(O)nc1O)C2 83878,C(C)(CCC(=O)Nc1cnccc1CO)NC(c1c(CCC)[nH]cc1)=O 83879,C#CC1CN(C(=O)CCC2CCN(C(c3snnc3CC)=O)C2)CCN1C 83880,c1(SC(c2ccc(F)cc2)c2n(C)ccn2)ccc(-c2cn[nH]c2)cc1 83881,Cc1nn(CC(=O)NC(CNC(=O)CCc2cn(C)nc2C)C(C)C)c(C)c1C 83882,C(CCC(=O)NCC(C)(F)CNC(=O)C(C)N1CCCC1)SC 83883,CCCCC(O)CC(=O)NC(CC(F)F)C(=O)N(C1CCCCC1O)C 83884,C1(CC(=O)NC(C)Cc2cnc[nH]2)CCCN(C(=O)CC2CSC2)CC1 83885,CC1(C)CC(CC(=O)NCc2cccnc2)CN1C(=O)Cn1cnnc1O 83886,c1(C(c2n(CC(=C)C)nnn2)NCC2CCC2)ccc(OC(C)C)cc1F 83887,C12(C(=O)NCC3C(CNC(C4(C)COC4)=O)C3)CCC(C(F)F)(CC1)C2 83888,CN1CCN(C(=O)CC2C=CCC2)CC1CNC(c1ncccc1Br)=O 83889,N1(C(C(C)=C2CC2)=O)CCC2CCN(C(C3(C#N)CCC3)=O)CC2C1 83890,C1(C(NOC)=O)CCN(C(c2cnc(-c3ccccc3F)s2)=O)CC1 83891,c1cc(=NC2CC3CCCC(C3)C2)[nH]c(N2CCOC(C3CC3)C2)n1 83892,c1(OC)ccc(F)cc1CCC(=O)NC1(CCNC(=O)CCSC)CC1 83893,N1(C(c2c(C)snc2)=O)CCC2(CCCN2c2ncnn3cccc23)CC1 83894,C12(CNC(C=CCCC)=O)CCCC1CCN2C(=O)CCOc1ccccc1 83895,C1(NC(C=CC=CCC)=O)CCN(C(=O)CC(C)=C(C)C)C1 83896,c1(C(=O)NC2CC2CNC(c2ccnn2C2CCC2)=O)coc2ccccc12 83897,CCCCCC(C)(CC)C(=O)NCC1(F)CCN(C(c2ccc(C)cc2)=O)C1 83898,c1(-c2onc(C3CCN(C(=O)OC)CC3)n2)ccc(N(C)C)c(F)c1 83899,c1(C(=O)NCCNC(C(c2ccc(C#N)cc2)C)=O)cc(F)ccc1F 83900,CCCC(C(=O)NCC1CC2CCC1N(C(=O)CCCF)C2)S(N)(=O)=O 83901,CCC(C)C(C(C(=O)NCCSC)N1CC(O)C(C)(C)C1)OC 83902,C=CC(C)(CCOC)C(=O)N(C)CCN(C(=O)C(c1ccc(C)cc1)C1CC1)C 83903,C1(C(=O)NC(C(C)C)C(=O)N(C)CCc2cc[nH]n2)CC2CC(=O)C1O2 83904,c1(NCC(=C)CC)nc2ccccc2nc1NCCc1nncn1C1CC1 83905,C1(C(=O)NCC2CC3(CC3)CN2C(c2ccc(F)cn2)=O)CCN2CCCC2C1 83906,N1(C(CCCOCCC)=O)CC(NC(C2CCCNC2=O)=O)CC(F)C1 83907,C1(NC(CC(C)c2cnn(C)c2)=O)CN(c2ncc(I)cn2)CC2(CC2)C1 83908,c1(C2(C(=O)NCCN(C)C(C34CCCC(CO3)C4)=O)CCCC2)ccc(F)cc1F 83909,N1(C(CC(C#CC)c2ccc(O)cc2)=O)CCCC2(CCCN2C(=O)CNC=O)C1 83910,C1(O)(CNC(C2C=CCN(C(C3C(C)(C)C3)=O)C2)=O)CCCCCC1 83911,Cc1cc(Cl)ccc1OCC(N1CCCOC(CNC(=O)C(C)(C)C(C)O)C1)=O 83912,C#CC(C1CCc2ccccc21)NC(=O)Nc1ccnc(C(F)(F)F)n1 83913,c1(CN(C(CN(C(=O)C2=CCCC2)CC#C)=O)C)ccc(C)nc1 83914,C1(NC(CC(C)OC)=O)CN(C(=O)CCCOCCc2ccccc2)CC1C 83915,N1(C(C2(COC)CC2)=O)CC(NC(=O)CC23COC(C(=O)OC)(C2)C3)C2(CC2)C1 83916,c1(N2CC3C(C)(C)C(C3)C2)nc2ccccc2nc1NCC1CCCS1 83917,C=Cc1ccc(C(N2CC3CCC3(NC(=O)CC3CCN(C)C3=O)C2)=O)cc1 83918,N1(C(C(C)(C)n2cccn2)=O)C2CCC(C2)C1CNC(c1cc(C2CC2)cs1)=O 83919,C1(OCC)CC(C(N2CC(CCCCc3cc(N)ccc3C)C2)=O)C12CCC2 83920,C(CC(F)F)(C(=O)NC1CCC(O)CC1)NC(=O)CC1(O)CCC1 83921,c1(C(C)C)nn(C)c(Cl)c1C(N1CCN(C(C2CC2C(F)F)=O)C(C2CC2)C1)=O 83922,c1(CC)nnc(O)c(C(=O)NC2CCCN(C(=O)C(C)(CC)OC)C2)c1CC 83923,C1(CC(=O)NC2CC(NC(=O)CC3CCNC3=O)C2)CCCC1(F)F 83924,C1(C)(C(N2CC(C(C)NC(c3coc(CO)c3)=O)C2)=O)CC2CCC1C2 83925,c1(C(N(C(CNc2nccc(CC(=O)OC)n2)C)C)=O)coc2ccc(C)cc12 83926,c1(C(=O)NCCN(C(c2cc(Cl)c[nH]2)=O)C2CC2)cc(-c2ccccc2)on1 83927,C(=O)(C(C)C(C)NC(c1ncoc1C1CC1)=O)N(CC=C)CCOC 83928,C1(CNC(C(CC2CC2)OC)=O)CN(C(c2cnnn2C(C)C)=O)CC1O 83929,Cc1cc(C(=O)NCC(CC2CC2)C(=O)NC2CC2C(C)(C)C)ccc1F 83930,C1(CNC(CNC(=O)OC)=O)CC2CCC1N(C(=O)C(C)Cc1cccnc1)C2 83931,n1(CC(=O)NCC2(OC)CN(C(c3cocn3)=O)C2)cc([N+](=O)[O-])nc1C 83932,C1(C(N2CC(C)(CNC(C(C)C)=O)OCC2)=O)CCc2ncccc2C1 83933,C12(C(=O)NCC#CCNC(c3n(C)ncc3C(F)F)=O)CCCCC1NC(=O)C2 83934,CCC(O)C(C)(C)C(=O)N(CCCN(C)C)CCNC(=O)C(C1(CC)CCCC1)C 83935,C(=O)(CC(C(F)(F)F)NC(C1(C)CCCO1)=O)N1CC2(CC(N(C)C)C2)C1 83936,n1(CC)ncnc1C(=O)NCC1(COC)CN(C(=O)C(F)=C2CCCC2)C1 83937,CCC(CC(F)(F)F)C(=O)N(C)CC1(NC(=O)COCc2nc[nH]n2)CC1 83938,c1(C(=O)NC2CCN(CCNC(C(C3CC3)OC)=O)CC2)c(C)nn(C)c1N 83939,c1(C(N2CCC2c2ccccc2)=O)cc2cccc(-c3ccc(CO)o3)c2[nH]1 83940,N1(C(c2ccc(C#C)c(C)c2)=O)CCC2CCC(C1)N2C(=O)Cn1ccnc1C 83941,N=c1nc(O)c(CC(=O)NC2CN(C(c3ccc(OCCO)cc3)=O)C2)c[nH]1 83942,c1(CCSC)cc2ccccc2[nH]1.C12CCCCC1NC(=O)CCn1cc2nn1 83943,N(C(=NCCOC(=O)OC)NCc1ccccc1)CC(c1n(C)ncc1)O 83944,c1(C(=O)NC(C)(C(N2CC(O)C(F)C2)=O)C2CCC2)ccc(N)cn1 83945,C(=O)(C(O)CN1CCCC1)OC(C)C(=O)NC1CCCCC1 83946,c1(CN(C(CC)C#N)C(=O)Nc2cc(C)c(C)s2)cc(F)c(C(F)(F)F)cc1Br 83947,c1(C(C)C)cccc(C(N2CCOCC2CNC(C2CC3CC3C2)=O)=O)n1 83948,C(=O)(C#CC1CCOC1)NC(CC#C)C(=O)N(C1(c2cc[nH]n2)CC1)C 83949,C1(NC(=O)NCC(=O)NC(CN(C(C2CC2F)=O)CC)C)CCCCC1 83950,CC1C(C(=O)N(C)CCC2CC2)CCN1C(=O)Cc1ccccn1 83951,Cc1cc(=NCC23CC(NC(c4ncc(Cl)cc4Cl)=O)(C2)C(C)O3)c(C#N)c[nH]1 83952,N1(C(c2c(OC)nc(Cl)cc2)=O)CCCc2nc(Br)ccc21 83953,C1(CNC(=O)CSc2ccccc2O)CC12CCN(C(=O)C(O)C(F)(F)F)CC2 83954,C(=O)(C1=CC=CN2CCS(=O)(=O)N=C12)NC1CN(C(c2c(C=C)cnn2C)=O)C1 83955,N1(C(c2nn(C)cc2Br)C(=O)NC(CC)(C)C)CC(S(C)(=O)=O)CCC1C 83956,c1(C(=O)NC2CCCC(NC(CCc3cc(C)sc3C)=O)C2)ccnc(C)c1N 83957,[N-]=[N+]=Nc1cccc(C(=O)NCC2CCCC2NC(=O)CCc2cc(Cl)cs2)c1 83958,c1(C(=O)NCC2N(C(CCN(S(C)(=O)=O)C)=O)CC(O)C2)cc2ccccc2s1 83959,c1(COC)ccc(C(N2CCCC2CC(=O)NCC(C)OC)=O)o1 83960,CC(C)CC(C)CC(=O)N1CCN(CCOc2cc(O)ccc2OC(F)F)CC1 83961,C1(NC(CN(C(C(CCCOC)C)=O)C)=O)CC1C1CCCCC1 83962,C(N=c1cc(Cl)nc(C2CC2)[nH]1)C1OCCN(C(C2CCC(C)(C)OC2)=O)C1 83963,N1(C(c2n(CCOC)ncc2)=O)CCC(CNC(c2ncc(Cl)n2C)=O)C(C)C1 83964,C1(SC)CN(C(c2c(Cl)noc2C)=O)CC1NC(=O)C(c1ccccc1)F 83965,C1(NC(c2n(CCCCCC)nnn2)(C)C2CC2)Cc2cc(OC)ccc2C1 83966,Cc1ccccc1C=CC(N1CCC(C)(CNC(C2C3CCCCC23)=O)C1)=O 83967,c1(CNC(C2CCN(C(C=CC(=O)OCC)=O)CC2)=O)cc(F)c(F)cc1F 83968,c1(OC)cccc(C(=O)NCCCCNC(C2CCN(C)C(=O)C2)=O)c1N 83969,C(CCCN=c1[nH]c(Cl)nc2c1SCC2)NC(C(CCCC)O)=O 83970,Cn1nc(C(=O)NC2CC2NC(c2ncsc2C(F)(F)F)=O)ccc1=O 83971,Cc1cc(C)c(C(N2CC=CC(NC(=O)CCCc3csc(C)n3)C2)=O)c(N)c1 83972,N1(C(C#CCNC(=O)CSc2nc[nH]n2)=O)CCn2ncnc2C1 83973,c1(CCC(=O)NCC(C)NC(CCC=CC)=O)cccc(C#N)c1 83974,n1(C(C)C)cncc1C(=O)OCC1CC=CCO1 83975,c1(NC(=O)NC2CC(NC(C3CC(C(F)F)C3)=O)C2)ccccc1Br 83976,N1(C(c2cc(C)[nH]n2)=O)CC2CC(C1)N(C(C1CCC(C)(C)O1)=O)C2 83977,CCCCCC(C(=O)N(CCC)CCNC(c1cc2scc(C)c2[nH]1)=O)C(C)C 83978,N1(C(C2CC(C)=C(C)CC2)=O)CC(CNC(=O)C=CC2CCCC2)CC12CCC2 83979,C#CCC(C)(C(=O)NC(C(O)CO)C1CC1)NC(=O)C(C)C1(O)CCC1 83980,N1(C(c2ccc(COC)o2)=O)CC(CNC(=O)Cn2nnc(=N)[nH]2)CCC1C 83981,c1(C(=O)NC(CC(C)NC(c2ccc(CC)cn2)=O)C)nc(OC)ccc1C 83982,Cc1cc(NCCC2CCC(NC(C3(C)CCCOC3)=O)C2)ccc1[N+](=O)[O-] 83983,c1(C(N2CCC(SC(F)(F)F)CC2)C(=O)NCCCCCC)cc(C)nnc1C 83984,Cc1ccc(C2CC2C(=O)NCC2(NC(=O)CC(C)C(C)C)CCC2)c(Cl)n1 83985,Cc1c(C(=O)NC(c2ccccc2)C(=O)NCC2CCCOC2)cccc1C#N 83986,N1(C(c2c(F)ccc(C)c2)=O)CCCN(C(c2cc(Cl)cs2)=O)CC1C 83987,Cc1cnc2c(C(N3CC(NC(=O)Cn4cnc(=N)[nH]4)CC(F)C3)=O)cccn12 83988,C1(CNC(CC2(N(C(C(COC)(C)O)=O)C)CC2)=O)CC(C(N)=O)=NO1 83989,N1(C(CNC(CC)=O)=O)C2CCC(C2)C1CNC(c1c(F)cccc1F)=O 83990,c1(C(=O)NC2CC(NC(c3cc(Cl)c(Cl)cn3)=O)C2)cnc2cc(Cl)ccn12 83991,C12(C(N3CCCC(CC=C)(NC(=O)C=CC(C)C)C3)=O)CCC(C#N)(CC1)CC2 83992,CC(CC(=O)NC1CSC1)N(C(=O)Cc1ccn(C)n1)C 83993,c1(CC)ccc(Br)cc1C(N1CCCCC1C1CCN(C(=O)COC)C1)=O 83994,C(CCCCCCC(=O)NC1CC2CN(C(c3occc3Cl)=O)CC2C1)SC 83995,O=C(N1CC(n2cc(C3(O)CCCC3)nn2)CO1)C1CCCCN1C1CCCC1 83996,C(=O)(C(CCC)C(C)C)NCCC1CCCN(C(C(CCC)F)=O)CC1 83997,C(=O)(CC(C)(C)OCc1ccccc1)N1CC(N(C(=O)CN2CCSCC2)C)C1 83998,C1(C(=O)NOCC(C)C)(CCOCC)CCN(C(c2cnn(C)c2)=O)CC1 83999,C(=O)(C(C)(C)C(C)(F)F)NC(C)CN.C(=O)(C(CC(N)=O)N(C)C(C)=O)OC(C)(C)C 84000,C(=O)(CCCCC(F)F)NC1(CNC(c2cnn(C)c(=O)c2)=O)CCCC1 84001,c1(C(N(CCNC(C2CC(CC(C)(C)C)C2)=O)CC)=O)ccc(Br)nc1N 84002,C1(C(N2CC(OC)CC(NC(CCC#C)=O)C2)=O)CC(C(C)(C)C)=NO1 84003,c1(C(=O)NCC(CC=C)NC(=O)C(O)CN(C)C)ccc(Cl)cc1C 84004,c1(C2(C(N(CCC)CCOC)=O)CC2)ccc(OC(F)F)cc1 84005,N1(C(CCCN(C)C)=O)CCN(C(c2cccc(-n3ccnc3)c2)=O)CC1CO 84006,CC(C(=O)NC1C2CC1CN(C(c1ccnn1C1CCOCC1)=O)C2)C(C)(C)C 84007,CC1(C)CCN(C(=O)C=C2CCCCC2)CC1NC(=O)CC1CCCOC1 84008,C=CCC(C)(C)CC(=O)N1C(C)C2CC1C2NC(c1cnc(O)n1C)=O 84009,C1(CC(C)NC(=O)C(C)Sc2nncn2C)CCN(C(=O)C=CC(C)(C)C)CC1 84010,CN1CCN(CCC(=O)NC(C)(C)CN2CCN(C(C3CCOC3)=O)CC2)CC1 84011,c1(C(=O)NCC2C(C)CN(C(c3cccc(Cl)c3)=O)C2)cc2cnn(C)c2s1 84012,CC(CC(=O)NC1CCCC(NC(c2ccn(C)c(=O)c2)=O)C1)CC(F)(F)F 84013,N1(C(CC(C(C)C)O)=O)CCC2(CCCCN(C(c3cn(C)c(=O)cn3)=O)C2)C1 84014,C(C)(CNC(=O)C(C)C(C)(F)F)(CC(C)C)NC(CCOC(C(C)C)=O)=O 84015,c1(C(N2C(CC(=O)NCCC(=C)C)CCCC2)=O)n[nH]cc1[N+](=O)[O-] 84016,c1(CN2CC(C(=O)Nc3ccc(CC)nc3)OCC2)ccc(I)c(O)c1 84017,C=CCC(CC(=O)NC(C)C(CC)CC)NC(=O)Cc1ccc(C)s1 84018,c1(C(C(=O)NCCOC)N(CC(C(=O)OCC)(F)F)C2CC2)sc(C)c(C)c1C 84019,C(=O)(C1CCCc2nncn21)C1(C)C(CNC(C(CCC(C)C)NC(C)=O)=O)C1C 84020,C1(NC(c2cc(C)sc2)=O)CN(C(C2CCCSC2)=O)CCC12CCOCC2 84021,C1(C(N2C3(CNC(CCOC)=O)CC(C2)C3)=O)CC1C1CCCCC1 84022,c1(CC(N2CCC(C)(CNC(c3c(C)ncnc3)=O)C2)=O)ccc2nn[nH]c2c1 84023,CC1(C)CCCCC1=CC(N1CC(CNC(C2C3CCCOC23)=O)C(O)C1)=O 84024,N1(C(CC)CC)CC(C(N2CC(O)(CNc3ncc(C(F)F)cn3)C2)=O)CC1=O 84025,C1(O)(C(=O)NC2CC(CCNC(c3cc(OC)n[nH]3)=O)C2)CC2(CCOCC2)C1 84026,C1(C(=O)NC(C2CCOCC2)C#C)CCN(C(c2ccsn2)=O)CC1O 84027,Cc1noc2cc(C(N3CC(CCNC(=O)CN(C)CCO)C(C)C3)=O)ccc12 84028,CCCC(CC(C)C)C(=O)N1CCOCC(NC(c2occc2COCC)=O)C1 84029,c1(C(=O)NCC2(F)CCN(C(c3cn(CC=C)nc3)=O)C2)c(C)cc(C)oc1=O 84030,CC1CCN(C(C2CC(=O)N(C)C2)=O)CCN1C(=O)CCN1CCCCC1=O 84031,N1(C(C2N(CC)C(=O)CC2)=O)CCCC2(CCN(C(c3nccnc3C)=O)C2)C1 84032,C(CC(C(C)C)NC(c1nccnc1C(N)=O)=O)NC(C(C)=C(C)C)=O 84033,CC(C)CC(CNC(=O)CC1(C)CC1)NC(c1ccc(C2CC2)o1)=O 84034,c1(OCC)ccc(-c2nc(COC)nn2-c2ccnn2C)cc1OC 84035,C(C)(CO)(C(=O)N1CCOC(Cn2cc(C)cn2)C1)NC(CNC(=O)OC)=O 84036,CC(C)(C)[Si](C)(C)OCC1CCCN(CC(=O)Nc2cnc(C#N)nc2)C1 84037,N1(C(CCCOCCOC(CC)(C)C)C)CCCCCC1 84038,c1(NC2CCN(C(CC)C)CC2)[nH]c(=NCC(CC)C(C)(F)F)nc2sccc12 84039,c1(NC(N2CC(C(C(=O)OCC)C)C2)=O)cc(COC)no1 84040,C(=O)(C(C)C(C)(C)C)NC(C1CCCN(C(COc2c(C)cccc2)=O)C1)C 84041,N1(C(C(C)OC)=O)CC2CCC(C1)C2C(N1CCCC1c1ccccc1)=O 84042,c1(C(N(CC(CNC(C(c2cccc(C)c2)=O)=O)O)C)=O)cc2sccc2n1C 84043,Cc1cc(C(=O)NCC2C3CCC(C3)N2C(=O)CCc2cnn(C)c2)c(C)cn1 84044,C(=O)(C(C)(C)CC(F)F)NC1(CF)CCN(C(c2cnn(C)c2C(C)(F)F)=O)C1 84045,C(C(N=c1nc[nH]n2cccc12)C1CC1)NC(c1cnc(C)[nH]1)=O 84046,C#CCCN=C(NCCOC1CCS(=O)(=O)C1)NCc1cnn(C)n1 84047,C1(CNC(Cn2ccc(C)n2)=O)CC2CN(C(=O)C(c3ccc(F)cc3)F)CC12 84048,N1(C(COCC=C)=O)Cc2n[nH]cc2C1C(=O)N(C1CCCCCC1)C 84049,C(c1ccccn1)=CC(=O)NC(C)C(C)NC(=O)Cc1cccc(F)c1 84050,c1(C(=O)NCc2c(C(=O)NCC(CCC)O)n[nH]c2)c[nH]ccc1=O 84051,c1(CCC(N2CCC(n3cc(C(COC)OC)nn3)C2)=O)cccc(N(C)C)c1 84052,c1(CN2CCC(O)(Cc3cccc(F)c3)CC2)noc2c1COCC2 84053,CCC(C)CCCC(=O)NC(C1CCCN1C(=O)CSCc1ncc[nH]1)(C)C 84054,N1(C(C2C(=C)C2C(=O)OC)=O)CCN(C(C23CCOC(C)(C2)C3)=O)C(C)C1 84055,c1(C(=O)NCC(CN(C(c2cc(C)no2)=O)C)O)ccc(N)c(C)c1C 84056,O=C(C1=CCCOCC1)NCC1(O)CN(C(=O)C=Cc2ccc(Cl)s2)C1 84057,c1(NC(CC2(C=C)CN(C(=O)C(C)CSC)C2)=O)ccc(F)c(CC)c1 84058,N1(C(c2n[nH]c(C)c2[N+](=O)[O-])=O)CCc2ccc(N=[N+]=[N-])cc2C1 84059,N1(C(c2c(CC)nn[nH]2)=O)CCC(CF)(NC(=O)CCCN(C)C)C1 84060,CC1CN(C(C2(C#N)CCCC2)=O)CCC1N(C(=O)C1=NOCC1)C 84061,N1(C(CCCC)=O)CCN(C(=O)C(c2ccc(Cl)c(F)c2)OC)CC1CF 84062,c1(OC)ccc(C(C)=CC(=O)NC2(CO)CCCN(C(C3(O)CC3)=O)C2)cc1 84063,C(C)(c1ccc(F)cc1)=CC(=O)NCC1N(C)CCN(C(C(C(CC)O)C)=O)C1 84064,c1(C(=O)NCC2C(NC(C(c3ccccc3F)OC)=O)C2)cc(C#N)[nH]c1C 84065,N1(C(CCOCCC)=O)CC(NC(=O)Cc2cc(F)c(N)cc2F)CC2(CC2)C1 84066,C1(CCNC(C(CC)C)=O)CN(C(c2cc(Br)cn2C(C)C)=O)CCO1 84067,CC(O)C(C(=O)N1CCC(CCNC(=O)C(c2ccccc2F)O)CC1)N(C)C 84068,C1(C)(CNC(C(F)OC)=O)CN(C(c2cnn3c2CCC3)=O)CCO1 84069,N1(C(c2nc(C)oc2C)=O)CC(C)(C)CC1CNC(=O)C=CC1CCCN1C 84070,CC(CC(=O)NCCC(O)(CC)CC)C(C)(C)NC(=O)C(CO)C(C)(C)C 84071,c1(OC)cc(C(N2CC(C)(NC(c3cnn[nH]3)=O)C2)=O)c(F)cn1 84072,C(CNC(=O)C(c1ccccc1F)F)(C(C)(C)C)NC(C(C)CN(C)C)=O 84073,N1(Cc2ccc(OCC)cc2)CCOCC(C(=O)Nc2nccnc2C(N)=O)C1 84074,N1(C(CC(CC)CC)=O)CCC(C2CC2)(CNC(=O)C(c2cn(C)nc2C)O)C1 84075,C1(NC(Cc2cc(C)c(CO)cc2)=O)CCCC12CCN(C(=O)C(N)=O)C2 84076,Cc1nn2ccccc2c1C(=O)NCC1(CCNC(C2(C)CC=CCC2)=O)CC1 84077,N1(C(C(CC)=CC)=O)CCC2(CCC2NC(=O)COC(C)(C)CC)CC1 84078,N1(C(C=C(CC)C)=O)CCC2(CC1)CCN(C(=O)C(C)(C)CF)CC2C 84079,c1(C(=O)NC(C2N(C(COCC#C)=O)CCC2)(C)C)ccc2c(c1)CCNC2=O 84080,CC1CC(NC(=O)Cn2ccc(O)nc2=O)CN(C(=O)CNS(=O)(=O)N(C)C)C1 84081,C1(NC(CC=CC=C)=O)C2CCCN(C(C3CC4OC3C3CC43)=O)C2C1(C)C 84082,C1(NC(c2ccc(OC)c(OC)c2)=O)C2CCCC(F)(F)C12 84083,n1(CCCC(=O)NCC(CNC(CC2(C)CC2(Cl)Cl)=O)CO)ccccc1=O 84084,c1(C(N2CCCC(NC(c3c(C)ncn3O)=O)C2)=O)cc([N+](=O)[O-])n[nH]1 84085,C1(C(=O)Nc2ccc(C(C)(C)C#N)cc2)CC2C(C1)C2(F)F 84086,c1(NC(C(CC)F)=O)cccc(NC(=O)CC(C)CNS(=O)(=O)CCCOC)c1 84087,c1(C(=O)NC2CN(C(C3CCCC(OC)C3)=O)C2)ccc2c(c1)NCCO2 84088,N1(C(C(C(=O)OC)(C)F)=O)CCC2(CCN(C(c3ccc4nccn4n3)=O)C2)C1 84089,c1(C(=O)NC(CC)CN(C(C2CCC(CCO)CC2)=O)CC)cnc(O)c(F)c1 84090,Cc1cc(O)ccc1NC(c1c[nH]nc1CCNC(=O)C(C)(C)N=[N+]=[N-])=O 84091,C1(NC(C2(C)ON=C(C)C2)=O)CC2(CCN(C(c3sc(C)nc3C)=O)C2)C1 84092,N1(C(c2ncn(CC)c2)=O)CCCCC(CNC(C2CCC(C)(F)CC2)=O)CC1 84093,C1(C(N(CCC#C)CC)=O)CCCC(NC(c2ccnc(O)c2)=O)CC1 84094,C12(CCCCC1)C(=O)N2C1CC1.C1(O)(CC#C)CC(C(=O)NCC2(C)CC2(C)C)C1 84095,CCC(CC)C(C)C(=O)NCCC(=O)N(C1CCC1)CCN(C)C 84096,C1(N(C(CN(C)Cc2ccccc2)=O)C(N)=O)CCCN(C(=O)C(N)=O)C1 84097,C12(NC(C3CC(C(=O)OC)C3)=O)CCCC1(F)CN(C(c1coc(C)n1)=O)C2 84098,Cc1cc(C(N2CCC(OCC(=O)NC(C)(C)C3CC3)C2)=O)nnc1O 84099,C1(N(C(Cc2cc(C)no2)=O)C)CCCN(C(=O)C2=CCCS2)C1 84100,C=CC1(CC(=O)NC)CN(C(C2CCN(CC3(CC4CC4)CCOC3)C2)=O)C1 84101,N1(C(C=CSC)=O)CCn2nc(C)c(CNC(=O)C(C)C(C)(C)C)c2C1 84102,c1(-c2c(C(N3CC(CNC(=O)CC4COC(=O)C4)C3)=O)cno2)ccccc1F 84103,c1(N(CCCN(C(C(C)OCCCC)=O)C)C)nc(Cl)nc2cc(C)sc12 84104,C12(C(=O)NC(CN(C(C)C)C)C)CC1CN(C(=O)Cn1c(O)nnc1O)C2 84105,Cn1cc(C(=O)NC2CCCC(C(N3CCC(F)(CF)C3)=O)C2)n(C)c1=O 84106,c1(CC(N2C(C)(CNC(C=CCCC)=O)CCC2)=O)cccc(F)c1O 84107,C1(NC(=O)CSc2nnc(S)s2)(CO)CCCN(C(c2ccncn2)=O)C1 84108,N1(C(C(C)(C)c2ccno2)=O)CC(NC(c2cc3occc3s2)=O)CC2(CC2)C1 84109,c1(C(=O)NCC2CCCN(C(c3ccc(C(C)=O)nn3)=O)C2)cc(F)ccc1Br 84110,Cc1cc(CCC(N2CCC(c3ccc(F)cc3)C(N)C2)=O)nc(C)n1 84111,C1(NC(=O)NCC(C2CCOCC2)OC)CC(C)(C)C12CC2 84112,c1(CC)ccc(C(=O)NC(C2CN(C(C3CCCC(F)C3)=O)C2)C)nc1 84113,N1(C(CC2CCN(C)C2)=O)CCC2(CCN(C(C3CC4CC4C3)=O)CC2)C1 84114,c1(-c2nc(C)[nH]n2)ccc(C)c(NC(=O)Cn2cnnc2CCO)c1 84115,n1(CC(=O)NC(CN(C(C(COCC)C)=O)CC)C)nc(C)n(C)c1=O 84116,N1(C(c2c(C)cc(F)s2)=O)CCC2(C1)CN(C(=O)C(C(C)O)N(C)C)C2 84117,C1(CCNC(CN(C)C2CC2)=O)COCCN1C(c1ccc(C(C)(F)F)cn1)=O 84118,C(N=c1[nH]c(N(C)Cc2cc(Br)ccc2F)nc(=N)[nH]1)C1C(C)CCC1 84119,N1(CC)CCC(NC(C2CCCN(C(=O)CCOCC(C)(C)C)C2)=O)CC1C 84120,C1(CC)CCN(C(=O)NCc2cnn(CC)c2OC)C1CC 84121,N1(C(c2c(Cl)ccc(C)c2)=O)CC2CC(C1)N(C(C1CC1F)=O)C2 84122,N1(C(c2ccc(C)o2)=O)CCC2(CC1)CC2(C)C(=O)Nc1cccnc1 84123,Cc1nc2ccc(C(N3CC4CN(Cc5nccnc5Cl)C4C3)=O)cc2o1 84124,c1(OC)ccc(OC)c(CC(=O)NCC2CCN(C(c3oncc3C)=O)CC2)c1 84125,c1(C(N2CC3CCC(C2)N3C(=O)Cc2ccnc(O)c2)=O)cccc2nsnc12 84126,c1(C(N2CCCC(CNC(c3nc(C(C)OC)oc3)=O)C2)=O)ccc(Cl)cc1N 84127,CCCC(C(=O)OC)C(=O)N(CCCNC(=O)C(C(C)C)n1ccnc1)C(C)C 84128,CCCCC(O)CCC(=O)N1CCC(C2CCCN2C(=O)C=CC2CCOC2)C1 84129,C1(C(=O)NCC(c2cccc(C)c2)NC(=O)C(Cl)=CCl)CCn2cncc2C1 84130,C1(C(=O)NC(C#CC#C)(C)C)CC(C)CCN1C(C1CC1Cl)=O 84131,Cc1nc(C)c(C(=O)NC(C)CCCNC(=O)C(c2cccnc2)C)[nH]1 84132,c1(CCC(=O)N(C)CC2CCC(CNC(=O)C(F)F)CC2)ccc(CO)cc1 84133,C(=O)(C(C)CC(N)=O)NCC(CCCC)NC(=O)C(C)Cc1ccccc1C 84134,c1(C(N(CCN(C(c2c[nH]c(=NC)o2)=O)C)C)=O)c(OC)cnnc1OC 84135,CC(CC(=O)NCc1ccc(Cl)cc1N)CC(=O)c1ccc(Br)cc1 84136,N1(C(c2cc(C(F)(F)F)no2)=O)CCC2(CCCN2C(=O)C2=CCCO2)C1 84137,CC1C(NC(c2nnc(O)nc2O)=O)C(C)CCN1C(=O)C=CC1CCCC1 84138,c1(OC)ccc(NC(C2(C)CCN2Cc2sc(Br)nc2Br)=O)cc1Br 84139,c1(C(N2C(C)(COC)CC(NC(=O)C(OC)OC)C2)=O)n[nH]c2cc(Cl)ccc12 84140,CC1CC(NC(=O)CN2CCSCC2)CN1C(=O)CCC(=O)OC(C)(C)C 84141,Cn1cc2c(n1)CCC(C(=O)NCCC1(NC(c3ccc(Cl)c(O)c3)=O)CC1)C2 84142,C=C(CCN(CC#N)Cc1ccccc1CS(C)(=O)=O)C(=O)OC 84143,C1(C(N2CCCC2CNC(=O)CCCOC2CCOCC2)=O)(OCC)CCCC1 84144,N1(C(c2nn(C)c(Cl)c2)=O)CCC(c2ccccc2)(NC(=O)C2=CCCS2)CC1 84145,C(=O)(CCCCC(=O)NC)N(CCCNC(C(CCC)=CCC)=O)CC 84146,N1(C(CC=CC=C)=O)CCOC(C(C)NC(=O)CN2C(=O)CCC2=O)C1 84147,C1(C(N2CC3CC3(CO)C2)=O)(NC(CN(CCOC)C)=O)CCN(C)C1 84148,c1(C(N(CCN(C)C)CC2C3COCC23)=O)sccc1F 84149,c1(C(N2CC3C(N(C(C4CCC(OC)C4)=O)C)C3C2)=O)c(F)ccc(F)c1O 84150,c1(C2(C(N(CCC(C)NC(=O)CC3(CO)CC3)C)=O)CC2)ccc(F)c(F)c1 84151,Cc1cccc(C(c2ccccc2)NC(=O)C(F)(F)c2ccncc2)c1 84152,c1(C(=O)OC)c(CCC(=O)N(CCCCNC(=O)C(C)C2CCC2)C)c[nH]c1C 84153,C(=O)(C(C)(C)CCC)N1CCN(CC(C)NC(C2CC(C#C)(O)C2)=O)CC1 84154,CN1CCCC(CCC(=O)NCC2(NC(c3cn[nH]c3)=O)CCCC2)C1 84155,C12(CCN(C)C1)C(=O)N2.C1(CNC(C2CC(C)(CC)C2)=O)CC(=O)N(C)C1 84156,N1(c2oc3cccc(C)c3n2)CCCC(C2CCN(C(C3(F)CC3)=O)CC2)C1 84157,CCC(C)(C#N)C(=O)NCCC(C)(C)NC(=O)CN1CCCC(C(F)(F)F)C1=O 84158,c1(C(N2C3CC(CNC(CC(C)(C)C4CC4)=O)C(C3)C2)=O)cc2c[nH]cnc-2n1 84159,C(=O)(CC1CCCc2oc(C)nc21)NCC1(OC)CN(C(COCC=C)=O)C1 84160,C1(C(=O)NCC(C)NC(C(=O)NCC)=O)CC(C2CC2)C1 84161,C1(N(C(CC2(OC)CCCC2)=O)C)CCN(C(=O)CC2=CCCCC2)CC12CC2 84162,c1(CNC(C(C2CCN(C(CC(C)(C)OC)=O)C2)F)=O)cc(F)ccc1C 84163,c1(NC23C(CN(C(C4CCC(C)CC4)=O)C2)CCC3)nc(Cl)nc2cnn(C)c12 84164,CCCCCCC(CC)C(=O)N1CC2(C1)CN(C(=O)CC(=O)N(C)C)C2 84165,C(=O)(CCCS(C)(=O)=O)NC(CNC(C=CC(c1ccc(C)cc1)=O)=O)(C)C 84166,C1(NC(C(C(C)C)OCC(C)C)=O)CCCCCN(C(c2nnc(C)s2)=O)C1 84167,c1(C(=O)NCC2(COC)CN(C(CSCCC)=O)C2)cn(C)nc1CC 84168,Cc1ccc(C(=O)NC(CCN(C(=O)CC2(CO)CC2)C)C(C)(C)C)c(C)n1 84169,c1(-c2c(C)onc2)ccc2c(C(N3CCNC(=O)C3C)=O)cnn2c1 84170,C1(CCNC(=O)Cc2ccsc2)COCCN1C(C1CCOC1=O)=O 84171,N1(C(=O)Cc2ccc(SCCN3CCOCC3)cc2)CCC(O)(c2ncc[nH]2)CC1 84172,C1(C)(CNC(CC(C=C)C)=O)CN(C(C2CC(S(C)(=O)=O)C2)=O)CCO1 84173,c1(C(=O)NCC2C(NC(CNC=O)=O)C3(CC2)CCC3)cccc2[nH]nc(O)c12 84174,C1(OC)CN(C)C(C)(C(N2CC(CO)(NC(=O)CC(C)(F)F)C2)=O)C1 84175,C1(CC(=O)N(CC(CC)NC(=O)CCn2ccnn2)CC)CCCOCC1 84176,Cc1cc(O)c(C(=O)NC2(CO)CCCN(C(c3c[nH]c(Br)c3)=O)C2)nn1 84177,c1(OC)ccc(C(N)CNC(c2ccnc(-n3ccnc3C)c2)=O)cc1OC 84178,C#Cc1cccc(OCC(=O)NCC2CCN(C(=O)CCC(=O)OC)C2)c1 84179,N1(C(CSC(C)C)=O)CCC2(CNC(c3ccnc(F)c3F)=O)CCCCC12 84180,C(CCN=c1ccn2c(Br)cnc2[nH]1)N(C(C(C=CCCC)O)=O)c1ccccc1 84181,C1(NC(c2ccc(CC)s2)=O)CCC(F)(CNC(c2cccn2C2CC2)=O)C1 84182,C12(C(N3CC(C#N)(COC)C3)=O)CCC(CN(C(C3C=CCC3)=O)C1)C2 84183,CC(O)(CCc1ccccc1)C(=O)NC1CCN(C(c2ccnc(Cl)c2O)=O)C1 84184,c1(C(N(C2CCCN(C(c3cc(CO)[nH]n3)=O)C2)CC)=O)nccc2[nH]ccc12 84185,C1(C(=O)NCCC=C=C)CCC(O)CN1C(c1c[nH]nc1C)=O 84186,c1(OC)ccc2c(C(=O)NC3CCCN(C(=O)CC4OCCCO4)C3)c[nH]c2c1 84187,C1(C(N(CCN(C(C(CCCC)CC)=O)C)C)=O)CCC(F)(F)CC1(C)C 84188,c1(C(N2CC(C)C(NC(=O)CC3CC=CCC3)C2)=O)cc(F)cc2cnccc12 84189,c1(OC)cc(C(=O)NC2COCCN(C(=O)CC3CSC3)C2)cc([N+](=O)[O-])c1C 84190,C1(CNC(c2cc(OC)n[nH]2)=O)CC(C)CCN1C(=O)CCCc1ccncc1 84191,N1(C(c2n(CC)ncc2Cl)=O)CC(CNC(=O)C(C)C2CC2)CC(C)(C)C1 84192,C12(NC(c3ccc(Br)c(F)c3)=O)CCCCC1CN(C(C1(CO)CC1)=O)C2 84193,C=CCCC(C(=O)OCC1CN(C(C)C)C1)NC(C1CC12CCOCC2)=O 84194,CCCCC(CC)NC(C1CSCCN1C(c1cc(CO)c(C)o1)=O)=O 84195,N1(C(C(C)(C)NC(C2(CC(=O)OC)CC2)=O)=O)CC(S(C)(=N)=O)C1 84196,N1(C(C(C)N(C)C)=O)CCC(C(=O)NC(CC2CC2)C2CC2)C(C)(C)C1 84197,C1(C(=O)OC)(CO)CCCN(CC2(C3(c4ccccc4)NC(=O)NC3=O)CC2)C1 84198,c1(C(=O)NCC2C(NC(=O)COCC(F)(F)F)CC2)n[nH]c(C2CC2)c1Br 84199,c1(C(=O)NC2C(NC(CSCCC(C)C)=O)CC2)n[nH]cc1-c1ccncc1 84200,N1(C(=O)C2CC2)CCN2CCN(C(=O)COC3CCCC(=O)N3)CC2C1 84201,N1(C(c2ccc(P(C)(C)=O)cc2)=O)CCC2CN(C(=O)COC(F)F)CCC2C1 84202,N1(C(C2C(NC(C3C(C(=O)OC)C=C3)=O)CCO2)=O)CCN(C)CC1C 84203,N(C(=NCCCC(=O)N1CCCC1)NCC12CCCC1CCO2)CC(C)C 84204,c1(C(=O)NC(CNC(c2ccc(=N)[nH]c2)=O)C2CC2)ccc2cnnn2c1 84205,C(=O)(CC(C)NC(=O)CC1CC=CCC1)NCCOCCOCC 84206,Cc1nn(Cc2nc(-c3cccc(COC(C)(C)C)n3)nn2C)c2ncccc12 84207,N1(c2nc(CCn3cc(C(C)N(C(N)=O)C4CC4)nn3)on2)CCCCCC1 84208,c1(CC(C(=O)NC2CC(CC(=O)O)C2)N(C)CC)ccc(C)cc1 84209,Cc1cc(NC(C2(NC(=O)CN(C)C)CCCCC2)=O)ccc1O 84210,C1(CC)(CC)CN(C(C23CCC(C2)C3OC)=O)CC(C)O1 84211,C(C(=O)N1CC(NC(c2cc(O)n(C)n2)=O)CC1(C)C)(C(C)(C)C)NC(C)=O 84212,C(C)(C)(CCCC(=O)N1CCOCC1)NC(CC1CCN(C)CC1)=O 84213,N1(C(CC2C(C)CCC2)=O)CCC(CCNC(C2(n3cc(Cl)cn3)CC2)=O)CC1 84214,CCC(CC)CCC(=O)NCCN(CCCCCC)C(c1ccc(F)cc1OC)=O 84215,Cc1ccc(C(=O)NC2CCC(NCc3cc(C(=O)O)ccc3F)C2)cc1Cl 84216,N1(C(CN2CCN(C)CC2)=O)CCC2(CC1)CC(C(=O)NC1CCOCC1)CO2 84217,N1(C(c2c(C)c[nH]c2)=O)CCc2cc(C(=O)NCC(N)=O)cnc2C1 84218,C1(CC)(CC)CC(NC(c2cc(O)nc(C)n2)=O)CN1C(=O)C(C)N1CCCC1 84219,N1(C(C#CC2(C)COC2)=O)CCC2CCN(C(c3ncc(F)cn3)=O)C2C1 84220,N1(c2snc(COC)n2)CCC2C(CCCN2C(=O)C(c2ccccc2)OC)C1 84221,c1(N2C3C(O)CC(C3)C2)nc2ccccc2nc1NCc1ccc(CO)c(Cl)c1 84222,CC(CC(=O)N1CCCN(CCNC(C23CSC(C2)C3)=O)CC1)CC(C)(C)C 84223,C=CC(C)(C)CC(=O)NCCCN(C(C1CC(O)CN1c1ccncn1)=O)CC 84224,C(=O)(CCCN(C)N=O)NCC1CC(C)CN(C(=O)CC2(C)CCC2)C1 84225,c1(C(N2C3CN(C(c4c(OC)cccn4)=O)C(C3)C2)=O)oc2ccccc2c1C 84226,C1(C(N(C2(C(=O)NCc3nccc(C)c3)CC2)C)=O)C2CCC(C2)C1C 84227,C(C)(CNC(C1(c2ccn(C)n2)CC1)=O)(C(C)C)NC(c1c(CC)ccs1)=O 84228,N1(C(C2(C#C)CCCCC2)=O)CCC2CC2(C(=O)NC(CO)C(C)CC)CC1 84229,CC1=CCC=CC1C(N1CC2C(NC(=O)CC(C)O)C2C1)=O 84230,S(=O)(=O)(C1(CNC(N2CCC(Cc3cccc(Cl)c3)C2)=O)CC1)N(C)C 84231,N1(C(C(C)C2CCCO2)=O)CCC(COC2CN(C(=O)Cc3ccon3)C2)CC1 84232,C1(NS(C)(=O)=O)CC2CCC(C1)N2C(C1CCN(Cc2ccccc2)CC1)=O 84233,N1(c2nc(OC)c(F)c(C)n2)CCCC2(CCN(C(=O)C(C)(C)SC)C2)C1 84234,C1(NS(CC)(=O)=O)CCCN(C(=O)Cc2cnccc2C)C1 84235,N1(C(C(CC)OCC)=O)CCN(C(c2cnc(O)nc2O)=O)CCC1C 84236,C(=O)(C(C)(C)C(N)=O)N1CC(C2N(C(C(C)OCCC(C)C)=O)CCC2)(O)C1 84237,N1(C(C(C)NC(=O)NC)=O)CCC(F)(CNC(=O)C(F)CC(C)C)CC1 84238,n1(C(C)(C)C)cnc(C(N(C2CCC(NC(=O)C(=O)N(C)C)C2)CCF)=O)c1 84239,C=CCC(CC(C)C)C(=O)N1CCOC2(C1)CN(C(=O)COCCN(C)C)C2 84240,c1(NC(C)=O)ccc(C(N2CCCC(N(C)C(c3cccn3C)=O)C2)=O)cc1F 84241,N1(C(C2OCCC(NC(C34CCCC3C4)=O)C2)=O)CCc2ccccc2C1 84242,CN1CC(C(=O)NCCCN(C(C2CCCS2)=O)CC2CCCC2)CC1=O 84243,c1(C(=O)NCC2N(C(C3(COC)COC3)=O)CC2)cc(F)cc2nc[nH]c12 84244,c1(C(N2C(CNC(CCC=CCC=C)=O)COCC2)=O)cc(F)cc(C)c1N 84245,Cc1cc(C(C)NC(C2CCN(C(c3ccnnc3)=O)C2)=O)on1 84246,CCCC(CC1CCCC1)C(=O)N1CCCC(N(c2ccncn2)C)C1 84247,C(=O)(CCC(C)(C)[N+](=O)[O-])N(C(C)C(=O)NCCc1ccns1)C1CC1 84248,C(=O)(CCCCC(=O)NCC(C)N(C(=O)C(O)C1=CCCCC1)C)OC 84249,CN1CCC(=CC(N2CC3C(CNC(=O)CCC4(C)CC4)C3C2)=O)CC1 84250,Cc1csc2c(NC3CN(C(C4CCN4C(C)(C)C)=O)CC34CCC4)ncnc12 84251,c1(OCC)ccc(C(C(=O)NCCOCC2(C)CC2)N(CC(C)OC)C)nc1 84252,C(CC(O)C(=O)NCCC(C(=O)NCC(O)C(C)C)OC)SC 84253,c1(CCC(=O)NC(C2(O)CN(C(C3(CC=C)CC3)=O)C2)C)ccc(Cl)cc1 84254,C(=O)(CC(C)C(C)(C)NC(=O)C1=CCCOC1)Nc1ccc(CC)cc1C 84255,C(CN=C(NCCF)N1CCC(O)(c2ccc(F)cc2)C1)=CCC 84256,N1(C(c2cc(-c3ccco3)[nH]n2)=O)CC2CCC(C1)N2C(C1(CC(F)(F)F)CC1)=O 84257,c1(C(N2CCCC2c2cccc(Cl)c2)=O)cc(Cl)c(F)cc1[N+](=O)[O-] 84258,c1(C(=O)NC(C2(O)CCN(C(c3c(C)ncnc3)=O)C2)C)cnn2c1OCCC2 84259,N1(C(C2CCCC(CC)C2)=O)CC2=C(C1)CN(C(c1cc(F)cc(Cl)c1)=O)C2 84260,c1(OC(C(=O)NCCN(C(=O)C(O)C(C)C)CCC)C)cccc(C(C)=O)c1 84261,CC(C(F)(F)C(F)F)NC(=O)C(C1CCCN(C(=O)OC(C)(C)C)C1)(C)C 84262,C(=O)(C(Cc1ccco1)NC(=O)CCC1CCCOC1)N(CC=C)C 84263,N1(C(CN(C(COC)=O)C)=O)CCN(C(=O)CCCCCSC)CC1CCO 84264,c1(CC)cc(C(=O)N(C2CCN(C(=O)CCc3cnc(C)o3)CC2)C)c(C)o1 84265,c1(CN2CC(n3ncc(NC(c4ccnc(O)c4)=O)c3)C2)cccc2c1CCC2 84266,C(CC(CNC(C1(C)CC(F)C1)=O)NC(=O)COCCF)OC 84267,c1(CC(N2CC3CC(CNC(C4(C)CC4)=O)C3C2)=O)ccc2ncsc2c1 84268,N1(C(CC2N(CC)CCOC2)=O)CCC2OCCN(C(=O)CCOC)C2C1 84269,C1(CC(N2CC(CCNC(C3CC3[N+](=O)[O-])=O)C2)=O)CSCCO1 84270,C123CCCC(CN1C(=O)C(=O)N2)C3.C(c1cn(C2CC2)nn1)=CC 84271,C1(C(=O)NC2CN(C(c3cc(SC)oc3C)=O)CC2C)(OC)CCOCC1 84272,S(=O)(=O)(c1cccc(C(F)(F)F)c1)N1C(C2CCN(C(C(=C)F)=O)CC2)CCC1 84273,c1(CC)ccc(OCCNC(c2cnc(-c3ccccc3O)s2)=O)cc1 84274,c1(C(=O)NCC(CNC(C(C)OCC=C)=O)CO)cc(F)ccc1NS(C)(=O)=O 84275,C1(CNC(N(C2CCCN(C)C2)C)=O)CCCN2CCCCC12 84276,CC(C)CCCCC(=O)NC1(C)CC(NC(c2cnn(-c3ccccn3)c2)=O)C1 84277,c1(CC)c(C(=O)N(C(C)C(=O)NCCC(C(=O)OC)OC)CC)nnn1C 84278,C(=O)(CC(CC(C)C)NC(C1CCOC1)=O)N1CC(c2onc(C)n2)C1 84279,C12CCCCC1N2.N1(C(=O)OCCOC)CCCC(N2CCCCC2)C1 84280,N1(C(CN2CCN(C(C(C)n3ccnn3)=O)CC2)=O)CC2CCCCC2C1C 84281,C(C)(CNC(c1c[nH]nc1C(F)F)=O)(C(C)C)NC(C(CO)OC)=O 84282,C1(N(C)C)CCC(C(=O)NC2C3CC2N(C(C2(C)CC=CC2)=O)C3)CC1 84283,c1(C(N2C3CCC2COC3)C(=O)NC)cnc2ccc(F)cc2c1 84284,N(C(=NCCF)N(C)Cc1ncn(-c2cc(Cl)ccc2Cl)n1)C1CC(C)OCC1 84285,C1(C(=O)NC(C)CNC(=O)C(C)SCc2ccccn2)CCCCC1(F)F 84286,c1(OC)c(C(=O)NC2CCC(CNC(C3(C)CCOC(C)C3)=O)C2)c(C)nn1C 84287,C1(O)(CC)CCCN(C(C2CC3C=CC2O3)=O)C1 84288,CCC(CNC(=O)Cn1cnc(C#N)n1)(CC)C(=O)N1CCCc2nccn21 84289,N1(C(c2c[nH]c(=NC)s2)=O)CCC2(CC1)CC2C(N1CCOC(C(C)(C)C)C1)=O 84290,c1(C(=O)NC2(CNC(=O)C(O)C3CCC3)CCOC2)cc2ccccc2cn1 84291,Cc1c(C(N2CCC(C(C)NC(c3cnc(N(C)C)nc3)=O)CC2)=O)nnn1C 84292,C1(COC)(NC(C2(n3cccn3)CC2)=O)CCN(C(=O)CCn2cncn2)C1 84293,C1(CC(=O)NC2(C)CN(C(c3cc(C)oc3)=O)C2)CCC(=O)NC1 84294,C(=O)(C(C)(C)C(N)=O)N1CCN(CC(C)NC(c2cnc(O)c(F)c2)=O)CC1 84295,N1(CC(=O)NC(C)C)CC2C3CCC(C2C1)N(C(=O)Cn1cc(C(C)O)nn1)C3 84296,CC(=O)CC(C)(C)C(=O)NCC1CC(C(=O)NCC(C)CC2CCC2)C1 84297,C1(C(N(CCCC=C)CC)=O)CCC(C2CC2)N1C(=O)C=Cc1cc[nH]n1 84298,c1(C(=O)NC2C(CNC(=O)CN3CCCC3)CCC2)ccncc1F 84299,c1(C(=O)NC2(COC)CCN(C(=O)CC3CCOCC3)C2)cnc2n1CCCC2 84300,C(CO)(CCCCNC(=O)CC(C)c1cccnc1)NC(c1nc(CC)sc1)=O 84301,c1(C(N2CC=CC(NC(CC3COCC(C)O3)=O)C2)=O)cccc(F)c1F 84302,C(CCCCNC(=O)CCCF)NC(C(C)c1cccs1)=O 84303,C1(C(=O)NCC2(CCC)CC2)CCCCN(C(=O)C(C)(CO)OC)C1 84304,C(=O)(C1=CCOCC1)NC(C1(O)CCN(C(=O)CC2SC(=N)NC2=O)C1)C 84305,n1(C2(C(N3CC(N4CCOC4=O)C3)=O)CC2)cc(-c2cccs2)nn1 84306,c1(CNC(CNC(=O)NC)=O)ocnc1C(=O)NCCC1CCN(C)C1 84307,Cc1ccc(C(N2CCCOC(CNC(=O)C(=O)N(C)C)C2)=O)c2c1CCC2 84308,N1(C(C(N2CCC(c3ccc(N(C)C)cc3)CC2)C)=O)CCN(C)CC1 84309,c12ccc(cc1C)o2.C(=O)(C=CSC)NCC1C(NC(CCOC(C)=O)=O)CC1 84310,C(=O)(C(C(C)(C)C)C1CCCCC1)N(C)CCNC(c1cn(C)[nH]c1=N)=O 84311,CC1CN(C(C2CC(c3ccccc3)C2)=O)CCN1C(c1ccc(O)nc1Cl)=O 84312,CCCC(C)C(=O)NC1CCCN(C(C2(C#N)CCC2)=O)C1 84313,Cc1cc(F)c(CN2CCCC2CNC(c2csc3c2CCCC3)=O)cc1Br 84314,CCC(CNC(=O)C(c1cncnc1)C)(CC)C(=O)NCC(O)C1(Cl)CC1 84315,Cc1scc(C(=O)NC(C2(O)CCN(C(=O)CC3CCOCC3)C2)C)c1C 84316,CC1(C)COC(CCC(=O)NCCN(C(=O)CCOCC(F)F)C2CC2)C1 84317,c1(OC)cc(F)cc2[nH]c(C(=O)NCCCNC(C3(C(F)F)CCCC3)=O)cc12 84318,Cc1cc2[nH]c(C(=O)NCC3(F)CCN(C(C4(CC5CCC5)CC4)=O)C3)cc2o1 84319,C(CC(C(=O)N(C)Cc1nnnn1C)NC(C1CC(OC)C1)=O)OC 84320,C12(NC(=O)Cc3ccc(F)cc3Cl)CCCC1N(Cc1cccc(Cl)c1Cl)CC2 84321,N#Cc1ccc(CC(=O)NCCOC2CCN(c3ncc(Br)cn3)C2)cc1 84322,CC(O)C(C)(C)CNC(c1ccc(CNC(C2(F)CC2)=O)nc1)=O 84323,Cc1cc(NC(=O)NCC(c2ccccc2)(C)C)cc2n[nH]cc12 84324,C1(CC(=O)NCC(C)N(C)C)CCCCN1C(C1CCCCO1)=O 84325,C1(NC(C=C(CC)CC)=O)C2CC3CN(C(c4ccc(F)c(Br)c4)=O)C1C3C2 84326,c1(C(=O)NC(C2CCCCC2)CNC(C2CCC(O)C2)=O)cn2ncccc2n1 84327,C(C(c1nnnn1CCSC)NCC1(OC)CCC1)(C(C)C)OC 84328,C1(C)(C(N(C(c2ccccc2)CC)CC)=O)CN(CC(C)C)CCO1 84329,c1(C(CC)C(=O)N(C)CCN(C)C(C2CNC(=O)C2)=O)cccc(Cl)c1 84330,c1(C(=O)NC(C(C)C)C2CC2)cc(CNC(C2C3CCCCC23)=O)nn1C 84331,CCC(CC1CCCC1)C(=O)NCC(C)NC(C1CC(C)(F)C1)=O 84332,C(=O)(C1=CC(C)(C)C1)NCC(c1ccc(F)cc1F)NC(C(CC=C)OC)=O 84333,c1(C(N2CC(CNC(C(C=C)OC)=O)C(OCC)C2)=O)cccc2ccoc12 84334,C1(C(=O)NCc2ncccc2C)(CC)CCCN(C(c2cnn(C3CC3)c2)=O)C1 84335,N1(C(c2scc(C(=O)OC)n2)C(=O)NC2CC2)CCC(F)(F)C(C)C1 84336,c1(CNCC2(C)CCC(C)C2)nc(O)c2cnn(-c3ccccc3)c2n1 84337,N1(C(C(=O)NCC)=O)CCC(NC(c2ncncc2Br)=O)C(C)C1 84338,CN1CCC(NC(C2C=CCN2C(C2CC3CCC3C2)=O)=O)CC1=O 84339,C1(CNC(c2cc(OC)ncn2)=O)CC2(CC(NC(=O)C(F)(F)CC3CC3)C2)C1 84340,C1(NC(CC(C(=O)O)NC)=O)CCC2(C1)CN(C(c1cc3cn[nH]c3cn1)=O)C2 84341,N1(C(C=CC2N(C)CCC2)=O)CC2CCC2(CNC(c2cnnn2C)=O)C1 84342,N1(C(=O)CC2CC2)CCC2(CCCN(C(c3cccnn3)=O)C2)C1 84343,CC1CCC(C)(CNC(c2c(CNC(=O)C(O)C3CC3)nnn2C)=O)CC1 84344,C1(C(NOCC#C)=O)C2CN(C(=O)C(CO)OC)CC12 84345,N1(C(Cc2ccc(OCC)cc2)=O)CCN(C(=O)CNC2CCSC2)CC1CO 84346,c1(C(=O)NC(C(C)C)CNC(c2cc(F)c[nH]2)=O)cccc(OCCF)c1 84347,C(=O)(CCCCCNC(=O)CC1CCOC1(C)C)NC(CC(=O)OC)(C)C 84348,C1(C(N2CCC(O)(C(C)NC(C(CC)SC)=O)CC2)=O)CCc2cnc(C)n2C1 84349,C(=O)(CC(CC)C(F)F)N(C1CC(C(N2C(CCC)C=CC2)=O)C1)CC 84350,C(=O)(CCCCC(C)(C)C)N1C2CC(C(=O)NC(c3ccn(C)n3)C)(OC2)C1 84351,C(=O)(CCCCCCBr)N1CCC(C(C(=O)N(CC(=O)NC)C)C)CC1 84352,C(CC(C)CCNC(c1cnn(CCC)c1C(F)(F)F)=O)NC(CC=CC=C)=O 84353,C=CCC(C)(C(=O)NC1CN(C(=O)CC2CCN(C)C2=O)CC1C)N(C)C 84354,c1(C(N2C(C(N3C(C)CCCC3)=O)C3CCC2C3)=O)ccc(S(N)(=O)=O)cc1 84355,c1(C(N2CC(OCCNC(C(Br)=C(C)C)=O)C2)=O)nc(C)oc1C 84356,C1(NC(=O)Cc2ccc(Cl)s2)CCCC(C(N2CCC(Br)C2)=O)C1 84357,c1(OC)cccc(CSCC(N2CC(NC(C3CCN(C)C3=O)=O)CC2C)=O)c1 84358,c1(C(N2C(CO)CC(NC(C(C=C)O)=O)C2)=O)ccc2c(c1C)CCC2 84359,c1(C(N2CC3C(C(=O)Nc4onc(C)c4C#N)(C3)C2)=O)cccc([N+](=O)[O-])c1I 84360,Cc1cc(C)nc(CCNC(=O)NCC2CN(C)CC2c2ccccc2)n1 84361,c1(C(=O)NCC(Cn2cc(-c3n(CC)ncc3)nn2)OC)ccc(F)cn1 84362,C1(CNC(C(CC)(C)C#N)=O)CC12CCN(C(c1cnccc1C(F)F)=O)CC2 84363,Cc1cc(Cl)cc(C(N2CCCC(CO)(NC(=O)C=CC3CCC3)C2)=O)c1C 84364,CC(C)C(CNC(c1nnnn1C(C)(C)C)c1ccnn1CC1CC1)C(C)C 84365,C1(C(C)(C)NC(C(N2CCC(OCC)CC2)=O)=O)CCc2ccccc2O1 84366,N1(C(C(C=C)OC)=O)CCC(C(N2CC3(C2)CN(C)C3)=O)C1(C)C 84367,N1(C(CC=CC)=O)CCCC1CN(C)C(c1cscc1SC)=O 84368,Cc1ncc(C#N)cc1NC(=O)C(CCC1CCC1)NC(=O)CC1CCOC1 84369,CC1C(=O)CCC1C(=O)NCC1(c2ccccc2)COCCO1 84370,C12(C(=O)NCCCC)C(NC(=O)CC3(O)CCOC3)C3CC1C2C3 84371,N1(CCC(=O)NC2CC(C)(NC(C(CSC)C)=O)C2)C(=O)CCC1=O 84372,N1(C(=O)Cn2cncn2)CCN(C(c2n[nH]cc2[N+](=O)[O-])=O)CC1C1CC1 84373,c1(C(=O)NCCC2(CNC(COC(C)=O)=O)CC2)ccc2nnn(O)c2c1 84374,CS(=O)(=O)CC(=O)NCC(O)CNC(=O)COc1cn[nH]c1 84375,CCC(O)C(F)(F)C(=O)NC1CCN(C(c2cscc2C(F)F)=O)C1 84376,c1(C(=O)NCC(CNC(c2ccc(C3C(C)C3)o2)=O)F)cc(Cl)nnc1O 84377,c1(C(=O)NC2C(NC(=O)Cc3cc[nH]c3)CCCC2)cnc(O)c2ccccc12 84378,C(=O)(C1=CC2CCCCCC12)NCC1(O)CC2N(C(C3CN(C)C3)=O)C(CC2)C1 84379,c1(COC)nc(NCC2(CN(C)C)CCOC2)cc(=NC2CC3(COCCO3)C2)[nH]1 84380,C12CCC(=O)N(C1)C2.C1(COC(C(N)=O)=O)CCCN1C(c1ccccc1)=O 84381,c1(C(CC)NC(N2CCCC2c2ccc(C)s2)=O)c(OC)cccc1F 84382,Cc1ccc(-c2c[nH]cc2C(=O)NCC2CC2NC(C2CC(N(C)C)C2)=O)s1 84383,C1(C(N(C)CC2CCCN2C(=O)CC(O)c2ccccc2)=O)CC2OC1C1CC21 84384,C1(C(=O)NCCN(C(c2ccc(F)cc2O)=O)CC)COC2(CCC2)C1 84385,c1(NC)cnncc1C(=O)N(CC(=O)NCC(C)(C)C1(O)CCC1)C1CC1 84386,c1(C(C)NC(C2(NC(=O)C=Cc3ccc[nH]3)CC2(C)C)=O)cc(F)cc(F)c1 84387,CCC(C)CC(C(=O)N1CCC12CC(O)C2)NC(C1CCC(O)CN1C)=O 84388,CN1CCC(NC(=O)CCN(C(c2ncc(F)cc2F)=O)C2CC2)C(C#N)C1 84389,c1(CC)nc(C(C(=O)NC(c2ccccc2)C)N(c2ccccc2)CC)n[nH]1 84390,c1(CCOC(C(Cc2cn(C)nc2)OC2CCS(=O)(=O)C2)=O)ccccc1Br 84391,N1(c2c(OC)cncn2)CCCC(C)(CNC(=O)CC2CCC(O)C2)C1 84392,c1(C(N(C2CCN(C(C3C(CC)OCCC3)=O)CC2)C)=O)cc2occc2s1 84393,Cc1cc(C(=O)NC2CN(C(c3csc(C)c3)=O)CCC2CO)nc(C)c1 84394,CCCCCS(=O)(=O)CC(=O)N1CC2CCN(C(=O)Cc3ccccc3)CC2C1 84395,Cc1cc(=NCCCCNC(=O)C(c2ccccc2C)(F)F)[nH]c(Cl)n1 84396,c1(CN(c2nc(C)cc(C)n2)C)ccc2c(cnn2C)c1.C12CN(C1)C2=O 84397,N1(C(C(C)n2cccn2)=O)CCOC2(CCCCC2NC(C2CCCN2)=O)C1 84398,c1(C2(N(C)C)CC2)cccc(NC(=O)C(=O)NC2(F)CCNC2)c1 84399,C1(NC(Cc2cc(C)on2)=O)C2CCC1N(C(=O)COCc1nccn1C)C2 84400,c1(C(=O)NC2CCC(NC(C(C)CS(C)(=O)=O)=O)CC2)cccc2oc(O)nc12 84401,C(=O)(C(C(C)(C)C)OC)N1CC(NC(CC(CC)SC)=O)(CO)C1 84402,C(=O)(C#CC1(C)COC1)N1C(C)CCC(C(=O)N(C)CCC2CN(C)C2)C1 84403,CC(CC(=O)NCC1CC1C(=O)NC(C)(C)C(C)(C)C)CC(C)(C)C 84404,c1(CC)cccc(CC(N2CC(NC(C3(CO)CC3(F)F)=O)CC2CO)=O)c1 84405,N1(Cc2cccc(C)c2)CC(C)C(O)C(C)C1.c12nnc(s1)C2 84406,Cn1cnc(C=CC(=O)NC2CCCC2C(=O)NC2(C(N)=O)CCC2)c1 84407,C(=O)(CCC(=O)NN(C)C)NC(CSCC)C(=O)N(C)CCn1ccnc1C 84408,C(C1=NOC2CN(C(c3cscc3Cl)=O)CC12)NC(=O)Cc1cnn(C(F)F)c1 84409,C1(C(N(CC(CNC(c2c(SC)ccs2)=O)(C)C)C)=O)CC2CCC1O2 84410,c1(CC(N2CC(CNC(CCCOC(C)=O)=O)C2)=O)ccc2c[nH]nc2c1 84411,C(C)(CO)(C(=O)N1CCC(OC2CC2)CC1)NC(C1C(C)C1C)=O 84412,C(=O)(C(C)(C)C(C)C)NC(CC)CN(C(=O)CSc1nc[nH]n1)C 84413,CCC(F)(F)CC(=O)NCC1CC(C)CCN1C(=O)CC(c1ccc(F)cc1)C 84414,N1(C(C=CC=CC)=O)CCCC2C1CCCCN2C(c1cncn(C)c1=O)=O 84415,c1(CC)ccc(C(=O)NCC2(NC(c3cc(F)cnc3O)=O)CCCC2)cc1F 84416,c1(C(N2CCC(N(C(c3c(O)ncc(CC)c3)=O)C)C2)=O)nc[nH]c2ncnc1-2 84417,N1(CC(N2CCC(C(C(=O)NC(COC)(C)COC)F)C2)=O)CCC(=O)CC1 84418,c1(C(=O)NC2CCN(Cc3c(OC)cccc3F)CC2O)nc(C)c(C)nc1C 84419,CC1CCC(C(=O)NCC2(NCCC34CCCC3C4)CCCC2)CC1 84420,CCC(CC)(CN=c1[nH]nc(C(C)C)o1)NC(c1nocc1C)=O 84421,CCC(CNC(C1C2CN(C(=O)C#CC(C)C)CC12)=O)CC(C)C 84422,N1(C(CCOC2CN(C(COCCOC)=O)C2)=O)CC(O)C(O)C12CCC2 84423,Cc1ccc2c(c1)CC(C(=O)NC(CNC(c1ccc(C(F)F)cc1)=O)CO)S2 84424,CCCCC(F)C(=O)NC1(C(=O)N(C)CC2(O)CCC2)CCN(C)C1 84425,N1(C(C(C)NC(C)=O)=O)CCC2(NC(=O)CCc3cn[nH]c3)CCCCCC12 84426,N1(C(C2C(OC)(OC)CC2)=O)CCC2CCC(NC(=O)CC3(CO)CCC3)C1C2 84427,N1(C(c2c(Cl)cn(CCC)n2)=O)CCN(C(c2ccccc2)=O)CC(CO)C1 84428,CC1CN(C(=O)C(=O)NCC2CC2)CCCN1C(c1ccc2scnc2c1)=O 84429,c1(SCCc2ccc(C(F)(F)F)cc2)ccc2c(c1)OCCO2 84430,Cc1ncn(C)c1C(N1CCC(C)C1CNC(c1c[nH]c(C(F)(F)F)c1)=O)=O 84431,N1(C(c2c(C)cnn2C)=O)CCC2CCC(C1)N2C(=O)CCC1CC(F)(F)C1 84432,Cc1cc(C(=O)Nc2ccc(-c3nnc(CCN)o3)cc2)c(C)o1 84433,C(=O)(C(CCOC)NC(C1CCC2CC12)=O)NCC#CC 84434,c1(OC)cccc(CN2CCC(C(=O)N(CC(C)O)CCOC)CC2)c1.S(C)(=O)(=O)N 84435,C1(O)(C(N2C(C)CC(NC(=O)Cn3cc[n+](C)c3)CC2)=O)CCCC(C)(C)C1 84436,C(=O)(CC(C(C)C)NC(c1cnc(Cl)n1C)=O)NCC(C(=O)OC)(F)F 84437,CC1(C)OCCC1C(=O)NCC1CCN(C(c2cnc(S)[nH]2)=O)C1 84438,N1(C(CC(=C)Br)=O)CCN(C(=O)Cc2ccc(F)cc2)C2CCCCC12 84439,c1(SCC)cccc(C(=O)NC2CC(NC(c3sccc3OC)=O)C2)c1 84440,C1(C(=O)NCCC2OCC(C)(C)C2)CC12CCN(C(=O)Cn1ccnc1O)CC2 84441,C(c1c(F)cccc1F)=CC(=O)N(C)CC1(O)CCN(C(COCC#C)=O)C1 84442,C(=O)(C(C)(C(F)F)c1ccccc1)NCCOCCNC(C(CC=C)C)=O 84443,N1(C(C=C(COC)C)=O)C2CC1CN(C(C1(F)CCN(C)CC1)=O)C2 84444,C(=O)(C#CC1CCOC1)N(CC(CN(C(c1c(F)ccc(C(C)C)c1)=O)C)O)C 84445,c1(C(N2C(CN(C)C(c3cnc(N)cn3)=O)CCC2)=O)cnc2c[nH]nc2c1 84446,CCC(C)(CO)C(=O)NC(c1ccccc1SC)CNC(c1ncn(C)n1)=O 84447,Cc1cc(NC(C2CCCCCCC2)=O)ccc1NC(c1ccncc1O)=O 84448,c1(CC(=O)NCC(n2cc(Br)cn2)C)cc(C(C)OC(C)(C)C)on1 84449,C12(CNC(C(C=C)(C)C)=O)CCCC1CCN2C(=O)CC1(O)CCC1 84450,c1(CNC(C(CCC)C)C)cc(C#N)ccn1 84451,C1(NC(CC=C)=O)CCN(C(c2ccc(-c3cc[nH]n3)cc2)=O)CCC1(F)F 84452,C(=O)(C(F)(CNC(C1CCCCO1)=O)C(C)C)NCc1n(CCC)ccn1 84453,N1(C(c2c(CCC)occ2)=O)CCCC(CCNC(c2snc(Cl)c2Cl)=O)C1 84454,N1(C(c2ccc(CC)o2)=O)CC(OC)CC1(C)CNC(c1cn(C)cn1)=O 84455,c1(C(c2nnc(N3CCCC(C(C4CC5(CC5)C4)C)C3)n2C)(C)O)ccc(F)cc1 84456,CCCC(F)C(=O)NCC1(CC(F)F)CCC1.C(=O)(C=CCN(CC)CC)N 84457,c1(OC)ccc(F)cc1C(=O)NCC(C)CNC(c1c(C(F)F)cccc1N)=O 84458,N1(CC(N2CC(C)(NC(c3c(C)n(C4CC4)nc3)=O)C2)=O)CCC(=O)NC1=O 84459,C1(C(=O)NCc2c(CC)c[nH]n2)CCCN1NC(=O)C=CC(=O)OC 84460,c1(N(C)C)ccc(N(C)C(c2ccccc2OC2CCCCC2)=O)cc1 84461,C(=O)(C(F)(F)C(F)F)NCC1N(C(C2(C(F)(F)F)CCCCC2)=O)CCCCC1 84462,C=CC(F)(F)C(=O)NC(CN(C)C(c1cnn(C2CCCCC2)c1)=O)CC 84463,C12(CNC(C3CCCCCC3)=O)CCCN(C(c3cc4sccc4[nH]3)=O)C1C2 84464,c1(C(N)=O)nc(Br)cnc1NC(C1CCCN(C(C2(Br)CC2)=O)C1)=O 84465,C1(NC(CN(CCC)C)=O)CC(C(=O)Nc2cc(C)ccc2CO)C12CCC2 84466,C1(CNC(c2cc(CC)no2)=O)(NC(c2csc(C(F)(F)F)c2)=O)CCCCC1 84467,c1(C(=O)NC2C(CNC(CCN(CC)CC)=O)C2)sc(-c2ccc(C)o2)nc1C 84468,N1(C(C2C(C)(C)C2C#N)=O)CC2(C=C(C(=O)NC3CN4CCC3CC4)CO2)C1 84469,Cc1ncc(NC(N2CCC(Cc3ccccc3)C2)=O)cc1CC(C)C 84470,C1(CC(N2C3C(CNC(c4cnc5sccn45)=O)C(C3)C2)=O)CC(O)C12CCC2 84471,C12(C(=O)Nc3c(C(N4CCOCC4)COC)cccc3C)CCCCC1OCC2 84472,n12nnnc1C1(CCC1SCCCOC)NC2(CN(C)C)C.C1(COCC)CC1.C 84473,Cc1nnc2cc(NC3CCCC34CN(C(=O)C(C)(C)OC(C)C)C4)ncn12 84474,CC1(O)CCN(CC(=O)NC2CCCCC2CNC(=O)CNC=O)C1 84475,Cc1cccc(C(N2CC(C(=O)NC(C)(C)CCCF)CCC2C)=O)c1C 84476,c1(OC)c(C(=O)NCC(F)CNC(c2c[nH]nc2[N+](=O)[O-])=O)cccc1F 84477,N1(C(CCN(CCC)C)=O)CC(NC(c2nnc(O)cc2C)=O)C(C)(C)C1 84478,C1(C(N2C(C(C)(C)NC(CC3N(C)CC=CC3)=O)CCC2)=O)C2CC3C(C2=O)C13 84479,C1(C(=O)NC(c2ncnn2C)CC)CC12CCN(C(C1(C)CC1)=O)C2 84480,CC1CN(C(c2ccccc2O)=O)CC1CNC(c1nnn(C)n1)=O 84481,N1(C(c2cc(C)ncc2)C(=O)NC2COC2)CC(C(N)=O)OC(C)C1 84482,C=C(Cl)CC(C(=O)NCC(C)C(C)C)NC(c1ccc(=O)n(C)c1)=O 84483,C(=O)(C(O)CC(F)(F)F)NCC(CCOC)NC(c1c(F)ccc(F)c1Cl)=O 84484,c1(CCC=CC(=O)NCC(C)N(C(=O)CN(S(C)(=O)=O)C)C)ccccc1 84485,Cc1ncccc1C(N1CCCCC1C(=O)NCC(O)CC1CCCC1)=O 84486,C1(CC(=O)NC(C2N(C(C=CC(C)C)=O)CCC2)(C)C)CCC(=O)NC1 84487,C1(C#N)(CC(=O)NCC2C(NC(CC3(C)CCC3)=O)CCC2)CCOCC1 84488,C1(NC(c2c(CC)ccs2)=O)CCCN(C(c2cnc(O)c(C)c2)=O)C1C 84489,c1(CC(N2CCC(NC(C(C)OCC3CC3)=O)C2)=O)csc(Br)c1 84490,C1(NC(c2cccc3nc[nH]c23)=O)CCCCC1N=c1nc(C2CC2)[nH]s1 84491,c1(C(N2CC(CNC(C3(COCC)CC3)=O)(OC)C2)=O)cn(C)c(O)n1 84492,N(C1CCCc2occc21)C(c1cnc(O)cc1C)c1n(CC)nnn1 84493,c1(C(=O)NCC2C(NC(c3ccc(Cl)c(F)c3)=O)C2)cccc2[nH]ncc12 84494,c1(C(N2CCCC(NC(c3csc(Cl)n3)=O)C2)=O)ccc([N+](=O)[O-])cc1F 84495,c1(C(=O)NCC2(C)CCN(C(CC(CC)C3CC3)=O)C2)ccc2c(c1)COC2=O 84496,CC(C)CCC(C(=O)NC1CNC(=O)C1)NC(=O)Cc1cc[nH]n1 84497,CC1CCC(c2cn(CCCCC(=O)NCCC3COCCO3)nn2)CC1 84498,N1(C(CCC=CCC=C)=O)CCC2CC(C1)CN(C(=O)C(C)(C)C(N)=O)C2 84499,c1(OC)cc(NC(=O)CC(CC2CC2)NC(=O)Cc2ccns2)cc(O)c1 84500,c1(C(=O)NC(CC=C)CNC(=O)C(C2CCC2)C2CCC2)cc2n(n1)CCO2 84501,N1(C(C2N(C(C)=O)CCCC2)=O)C(C)CC2CN(C(=O)CCc3cnn[nH]3)CC12 84502,C1(F)(CNC(COCc2n(C)ncc2)=O)CCC(NC(=O)CC2CCCOC2)C1 84503,C(CC1CCC1)(C(=O)N1CC(O)(CN(C)C(c2cnns2)=O)C1)OC 84504,c1(C(=O)NCCCCN(C(C(C=C)(F)F)=O)C)cnc(C(F)(F)F)c(OC)c1 84505,C1(NC(c2cc[nH]n2)=O)CCOCC1NC(C1(C2CCCO2)CCCC1)=O 84506,N1(C(C2(NC(C3CC=CCO3)=O)C(C)(C)C2)=O)CC2CCC=CC12 84507,N1(C(C=Cc2cnc(C(C)(C)C)s2)=O)CC2CC(NC(C3(Br)CC3)=O)C(C2)C1 84508,C1(c2onc(C)n2)COCCN1C(c1cc(Br)no1)C(=O)NCCC#N 84509,CC1CC(C(=O)NCCC2(C(=O)NC3(C)CCCC3C)CCC2)CC(=O)N1 84510,c1(CNC(c2ncn(CC)n2)=O)cccc(NC(=O)Cc2csc(Cl)c2)c1 84511,N1(C(CCc2onc(C(C)(C)C)n2)=O)CCN(CCNC(C23CCC2C3)=O)CC1 84512,c1(C(C(=O)NCC)N(CC(C)(C)C)CCC)cccc(S(N)(=O)=O)c1 84513,CCCC(C(O)C(=O)NC12CC(C1)C2)NC(=O)C(CC)(CO)OC 84514,C1(CSc2ccco2)CC2CC(C1)N(C(=O)C=CSNC(=O)Cc1csnn1)C2 84515,C1(NC(C(CC)=CC)=O)CCC(n2cc(C3(O)CCOCC3)nn2)CC1 84516,C1(C)(CC(=O)OC)CCN(C(c2ccn(C)c2)C(=O)NC2COC2)C1 84517,C(c1cccc(F)c1Cl)=CC(=O)NC(CNC(c1c[nH]nc1C(F)F)=O)C1CC1 84518,c1(C(=O)NC2(CO)CCCN(C(CCC(=O)NC)=O)C2)ccc2c(n1)CCC2=O 84519,Cc1cocc1C(=O)NCCCCC1(NC(C2CCCCC2)=O)CC1 84520,c1(CC)cnc(C(=O)NCC(CC)NC(C2CCN(c3ccncc3)C2)=O)cn1 84521,c1(C(COC)=O)cccc(S(=O)(=O)Nc2cc3ccccc3n2C)c1 84522,C1(S(C)(=O)=O)(C(=O)NC2C(C)CN(C(c3c[nH]ccc3=N)=O)CC2)CC(O)C1 84523,Cc1ccnc(C)c1CNC(=O)C1=CCC(NC(C2(C3CC3)CC2)=O)C1 84524,c1(C(=O)NCC(=C)CCNC(=O)Cc2nc(C)sc2C)c(F)cc(C)cc1F 84525,c1(C(=O)NCC2CCN(C(C3CC=C(C)CC3)=O)CC2)cc(F)ccc1F 84526,CC1(C)C2CCC1(COC(C1CC3CCCN(C1)C3)=O)CC2 84527,c1(C(N2CCC(CCO)CC2)=O)ccc(C2=CCOCC2)c2cc[nH]c12 84528,CC1(C)CCN(C(=O)CCNC(N)=O)CC1CNC(=O)COCC1CCCO1 84529,N1(C(CC2CC(=C)C2)=O)CCOC(CCNC(C2CC2c2ccnn2C)=O)C1 84530,S(=O)(=O)(c1cnoc1C)N1CC(NC(CCc2c(OC)nccc2)=O)C(F)(F)C1 84531,C1(C2CCN(C(=O)C=C(C)C(F)F)CC2)(NC(C2CN(CC)C(=O)C2)=O)CC1 84532,N1(C(CNC(CCN(CC(COC)C)C)=O)=O)CCCCC1 84533,c1(NC(CCCN(CCC)CCC)=O)cc(C(=O)OC)cc(CC)c1 84534,C1(C(=O)NCCN(C(=O)C(C(C)(C)C)n2ccnn2)CC)CCc2nncn2C1 84535,CC(C)(C)CCCCCC(=O)NC1CC(NC(=O)C2=NNC(=O)CC2)C1 84536,C1(NC(C(CC#C)(C)C)=O)CC2CCCC(C1)N2C(=O)C(C)SC 84537,N1(C(C(CC=C)(C)O)=O)CC(C(=O)NC2CCC(C3CC3)C2)CCC1(C)C 84538,C#Cc1cc(F)ccc1C(=O)NCCN(C)CC 84539,c1(C(C(=O)NC(CCCNC(C2=C(C)OCC2)=O)C)=O)cc(S(N)(=O)=O)cn1C 84540,C1(NC(c2ccc(C#N)[nH]2)=O)CN(C(=O)CCc2cccc(O)n2)CC1C1CC1 84541,CCC(C)(C#N)C(=O)NCCN(CC(C)O)C(=O)Cn1nc(C)cc1C(F)F 84542,c1(C(=O)NC(C(CO)NC(CCCC(CC)C)=O)C)cc2ccoc2cc1F 84543,N1(C(C2CC=C(C)CC2)=O)CCCC(C(N2CCOCC2C)=O)CC1 84544,C1(C(=O)NCCCN(C(C2=CCN(C)C2)=O)C)CCn2cnnc2C1 84545,C(C)(CCN=c1ncc(C(F)F)c[nH]1)NC(c1ccnc(OC)n1)=O 84546,c1(C(=O)NC(C2CCN(C(CCN(CCC)C)=O)C2)C)c(C(C)C)n[nH]c1C 84547,c1(C(N(CC(C)NC(=O)C=Cc2ccccc2Cl)C)=O)cccn(C)c1=O 84548,c1(OC)ncc(NC(C2CC(C)N2C(=O)CC23CCCC2C3)=O)cn1 84549,CC12CN3CN=C(NCC(F)F)N(C)C1(C3)C2.C1(COCC(F)(F)F)CCOC1 84550,c1(C(N(C(CCCN(CC)CC)C)C)=O)nc2c(s1)CCC2 84551,N1(C(c2c(CCC)cccc2)=O)CCC2(CCC(NC(=O)C(C)N3CCC3)C2)C1 84552,C(=O)(CC(C)CNC(c1ccc(OC)cc1)=O)N(CCCC#C)C 84553,C1(CC(N2CC(C(C)NC(c3ccc(CCC)[nH]3)=O)C2)=O)CCCOCC1 84554,c1(C(=O)NCC(CCC)OC)cccc(Cl)c1C(F)(F)F 84555,CC1CCN(C(C2CC2F)=O)CC1CNC(c1cnn(CC2CC2)c1)=O 84556,C1(CC#C)(C(=O)OC)CCN(C(CC(C2CCCC2OC)C)=O)CC1 84557,Cn1ncc(C(=O)NC2(CCC(=O)NOCC3CCCCC3)CCC2)cc1=O 84558,N1(C(c2[nH]nc(C(=O)OC)n2)C(=O)OC)CCCC2(C1)NC(=O)N(C)C2=O 84559,CC(C)CC(=O)NCC=CCC(=O)N(C(C)(CO)C1CCCC1)C1CC1 84560,c1(-c2nc(-c3ncc(OC)c(Cl)c3)nn2CCOC(C)C)ccc(S(C)(=O)=O)s1 84561,c1(CCC(C)=O)ccc2oc(C(=O)OCCCS(=O)(=O)N3CCOCC3)c(C)c2c1 84562,N1(C(c2ccnc(OC)n2)=O)CCN(C(c2cn(C)nc2Cl)=O)C(C2CCC2)C1 84563,N1(CC(=O)NCC(CC)N(C(=O)Cc2nc(C)sc2C)C)CCC(C)CC1 84564,c1(C(C)C)c(C(=O)NC(C)(CNC(=O)CCC#N)C2CC2)cnc2ncnn12 84565,C(C(CC(F)(F)F)NC(c1nnc(O)cc1O)=O)NC(CC1CCCC(C)O1)=O 84566,S(=O)(=O)(c1csc(C(=O)NCC2COCCN2C(=O)C2CC2)c1)NC 84567,N1(C(c2cc(C3(C)CC3)on2)=O)CCOCC(C(N2CCC(CC(N)=O)C2)=O)C1 84568,c1(C(=O)NCC(CNC(COC2(C)CCC2)=O)CO)ccc([N+](=O)[O-])s1 84569,N1(C(CCC#C)=O)CCCC(O)(CCNC(C23CC(CN2C2CC2)C3)=O)C1 84570,c1(C(=O)NC23CC(NC(c4cc(C5CC5)on4)=O)(C2)C3)ccc2nccnc2c1 84571,C12(C(N(C3(CCO)CC3)C)=O)CCCC1CCN2C(=O)Cc1cccnc1 84572,c1(C(N2CCN(C(CSC)=O)CC3C2CCC3)=O)cc(OC)cc2c1CCCC2 84573,c1(N(C)CCO)ccc(CN2CCC(CNC(c3ccnnc3O)=O)CC2)cc1 84574,c1(C(=O)NCC(C)(O)C(F)F)[nH]nc2ncccc12 84575,Cc1noc2cc(N3CCC4(CN(C(=O)C(C)C)CC4O)CC3)nc(Cl)c12 84576,C(=O)(C1=CNC2=NCCC2=C1)C(C1CCN(C(C)=O)C1)=O.C(C(C(C)(C)C)N)N 84577,S(=O)(=O)(CCCCCl)NCCCO.c1(NC(=O)NCCCO)ccc(N)cn1 84578,C1(C(N(CCCNC(C2C(C)C2C)=O)C)=O)CC12CC(F)(F)C2 84579,C(CC(=O)NOCCN(C)C)OCCNC(CCCO)=O.C=CCCSCC 84580,CCC(C)CCCC(=O)NCC(C)(C)CC(=O)NC(C)(CO)C1CCCC1 84581,C1(C(=O)NCC2(CNC(C(CC#C)C)=O)CCCCC2)COc2ccccc2C1 84582,C1(C(=O)NCC2OCCN(C(Cn3ccc(C)n3)=O)C2)CCC=CCCC1 84583,N1(C(C2C(=C)C2)=O)CCN(C(c2ccc(-n3cncn3)c(N)c2)=O)CC(C)(F)C1 84584,C1(NC(C2C(NC(C(C)N(C)C)=O)C=CCC2)=O)CCCC2(CC1)CC2 84585,c1(C(N2CC(NC(C34CCC(CC3)OC4)=O)CC(O)C2)=O)ccc2nncn2c1 84586,CCCCCC(O)C(C)C(=O)N1CCC=C(CNC(=O)CC2CCCCO2)C1 84587,c1(C(N2CC(C)C(Nc3ccc(OC(F)F)cc3F)C2)=O)ccc([N+](=O)[O-])cn1 84588,C1(NC(C(C)OCCC=C)=O)CCCC1NC(c1cc(CC(C)C)on1)=O 84589,C1(N2CCC(COC)C2)C(C)OCC12CCN(C(c1cc(Br)ccc1Br)=O)CC2 84590,C(=O)(C(C(C)CC1CC1)N1CC(C(=O)O)CC(C(=O)O)C1)NCCSC 84591,N1(C(C(CCC)NC(N)=O)=O)CC(C(N2CCC(O)C(CO)C2)=O)CC(C)(C)C1 84592,N1(C(C(C)OCC)=O)CCN(C(c2cccc(OCC(F)(F)F)n2)=O)CC1C 84593,C(=O)(C1SCCc2sccc21)NC1CC(C)(NC(=O)C(O)CC(F)F)C1 84594,C(=O)(CC(CC)C(C)(C)C)NCC(CCCC)NC(=O)C1=CCCC1 84595,CN1CCC(N2CC(C(=O)NCCC3(C(=O)NCC4(C)CC4)CC3)C2)CC1 84596,C(=O)(C(C)(C)C(C)C)NCC1CC(NC(c2c(C(=O)OC)c(C)[nH]n2)=O)C1 84597,CC1CCN(C(=O)C(=O)NCC(c2ccccc2)CC2CC2)C1.C1(=O)COC(=O)CN1 84598,CCC(C(=O)NCC1(CNC(=O)CCCN2CCCCC2)CC1)C(C)C 84599,c1(C(=O)NCC(CC=C)NC(=O)CN2CC3CC3C2)cnn(CCO)c1C 84600,C1(CNC(COCC=C)=O)CN(C(C23CC(C(F)F)(CO2)C3)=O)CCO1 84601,C(=O)(C1=C(Cl)CCOC1)N1CCC(O)(C(C)NC(CCC=CCC=C)=O)C1 84602,c1(C(=O)OCC)ccc(S(=O)(=O)NCC(O)C(N)=O)c(Br)c1 84603,N1(C(C2(CC)CCC2)=O)CC(N(C)C(c2cc(OC)cnn2)=O)C2(CC2)C1 84604,C1(NC(c2cc(C)no2)=O)COCCC1NC(=O)CCc1cc(Br)cs1 84605,Cc1onc(Cl)c1C(=O)NCCC(C)NC(c1c(C(F)(F)F)n[nH]c1C)=O 84606,N1(C(CC#N)=O)CC2(CCC(C(N3CC(S(N)(=O)=O)C3)=O)O2)C1 84607,C(c1ccc(Cl)cc1Cl)=CC(=O)NCCCCCCNC(C(CC)(C)CO)=O 84608,N1(C(CCSCCCC)=O)CCC2CN(C(=O)C(C3CCC3)N(C)C)CC12 84609,N1(C(c2cc(CCCCC)[nH]n2)=O)CCCC2(CCN(C(C)C(=O)NC)C2)C1 84610,C1(CNC(=O)C=CCF)CCCN(C(=O)CNS(=O)(=O)C2CC2)CC1 84611,c1(N2CCN(C(C=C(C)C(=O)O)=O)C(C(F)(F)F)C2)ncnc2[nH]c(C)nc12 84612,N1(C(C2OCOC(C)C2C)=O)Cc2ccc(CNC(=O)CCC3CC3)cc2C1 84613,c1(NC(C2C(NC(CC=C)=O)CCCC2)=O)ccc(C)c(CC)c1 84614,c1(OC)ccc(NC(c2nc(-c3c(CO)cccc3F)sc2C)=O)cc1OC 84615,c1(NCC(C2CCCC2)NC(c2ccc(OC)nc2)=O)c([N+](=O)[O-])cnn1C 84616,Cc1ccc(C(=O)NCC(C)NC(c2c(C)noc2N)=O)cc1[N+](=O)[O-] 84617,Cc1cc(Br)cc(S(=O)(=O)N2CC3(CCC(NC(c4nccs4)=O)C3)C2)c1 84618,N1(C(c2c(C)ncnc2C)=O)CCN(C(c2cc3ccccc3s2)=O)CC(O)C1 84619,C1(C)(CNC(COC(CC)C)=O)CCCN(c2nnc(C(=O)OC)s2)C1 84620,C(=O)(C1=CC2(CN(C(=O)C(C)(C)CC(F)F)C2)OC1)N(C(CC)COC)C 84621,C1(NC(C=C(COC)C)=O)CC12CCN(C(=O)C(C)C(=O)OC(C)(C)C)CC2 84622,Cc1ccc(C23CC2CN(C(=O)NCCc2noc(C)n2)C3)cc1 84623,Cc1cncnc1C(=O)NC1(CNC(=O)COc2cccc(F)n2)CC(F)(F)C1 84624,C1(C(N(CCCCNC(C(CC=C)(C)CC)=O)C)=O)CCC2(CC1)CC2(F)F 84625,Cc1cccc(F)c1C(=O)NC1C2CC1CN(C(C1COCC(C)O1)=O)C2 84626,c1(C(=O)NCC2C(CC(=O)NC(c3ccns3)C)C2)cc(Cl)cn1C 84627,N1(CC)CC(NC(=O)C(CN(C)C)NC(c2cccs2)=O)CC1=O 84628,c1(C(N2C(C)CC(NC(C=CCN(C)CC)=O)C2)=O)ncc([N+](=O)[O-])cc1C 84629,CC1=C(C(=O)N(CC(O)CNC(=O)Cc2c[nH]nc2O)C)SCCO1 84630,NS(=O)(=O)c1cccc(C(=O)NCCNC(=O)CCSCc2ccccc2)c1 84631,Cc1cc(F)sc1C(=O)NC1(CNC(c2cc(C(F)(F)F)[nH]c2C)=O)CCCC1 84632,C(=O)(CC1C(=O)Nc2cc(Cl)ccc21)NCC1(OC(C)=O)CCOC1.C1C(=O)N1 84633,C=CCC(CC=C)C(=O)NC1CN(C(=O)Cn2cnc(=N)[nH]2)C2CCCC12 84634,CC(C)C1=NOC(C(=O)N(CC(=O)NCC2CCC(=O)O2)C)C1 84635,CN=c1[nH]cc(C(=O)NCC2CCC(C(=O)NC(C(C)C)C3CC3)C2)o1 84636,c1(COC(C)C(=O)N(C)CCN(C(=O)CCN2CCCC2)C)ccccc1 84637,c1(CN2C(CC(=O)N(CCO)CC)CCC2)ccc(C#N)s1 84638,c1(C(C)=O)ccc(N2CCCC2C2(NC(=O)C(C)SC(F)(F)F)CC2)nc1 84639,c1(COCC(=O)NCCN(C)C(C2CN(C3CCCCC3)C2)=O)ccncc1 84640,c1(COC)cc(C(=O)NCC2C(C)CCN2C(c2ccc[nH]2)=O)c(C)o1 84641,C1(CC)CCN(C(=O)C(CC)N(C)C)C1CNC(c1ncncc1Cl)=O 84642,C1(CNC(c2scnc2Cl)=O)C(C2CC2)CCN1C(c1cccc(CO)n1)=O 84643,C12(C(=O)NCCCCCNC(C3CC34CCOC4)=O)CCN(CC1)CC2 84644,N1(C(COC(C)C)=O)Cc2nccnc2CC1C(N1CCC(O)C(F)(F)C1)=O 84645,CC1(CNC(c2cc(F)c[nH]2)=O)CCN(C(=O)C=CCN2CCCCC2)CC1 84646,C1(C(C)NC(c2c(CC)cns2)=O)CCCN(C(c2n[nH]cc2Cl)=O)C1 84647,Cn1ncc2c1CCN(S(=O)(=O)c1c[nH]c(C(=O)O)c1)C2C(=O)OC(C)(C)C 84648,C=CC(C)CC(=O)NC1COCC1NC(=O)C(C)=C1CC1 84649,N1(C(C(CSC)C)=O)CC2(CCC(CNC(=O)CNC(=O)CCC(C)C)O2)C1 84650,N1(C(c2nc(C(C)C)oc2)=O)CC(O)CC1(C)C(=O)NOCCOCCOC 84651,C#CCC(C)(C)C(=O)NCC1CCN(C(=O)CSCc2cscn2)C1 84652,C1(C(=O)NC2CCN(C(Cn3nc(C)c(Br)c3)=O)C2)CCC2C(C1)C2(F)F 84653,CCC(C)CCCCC(=O)N1CC(NC(=O)C=Cc2cnccn2)C2(CCC2)C1 84654,C(=O)(C1c2ccccc2CN1C(c1cnc(C)c(C)c1)=O)NCC(=O)NC 84655,c1(C(=O)Nc2cccc(CNC(C=CCN(C)CC)=O)c2)nnc2ccccn12 84656,C(=O)(CCCCC(F)(F)F)NC1CCCC(NC(COC(CC)C)=O)C1 84657,C1(C(=O)NCC(O)CNC(c2cccnc2O)=O)(OC)CCCC(C)(C)CC1 84658,C(C1c2ccccc2CN1C(C1C2COCC12)=O)NC(C(NOC)=O)=O 84659,N1(C(Cc2c(C)ccs2)=O)CC2CC(NC(C3CCC(C)(C)O3)=O)CC1C2 84660,N1(C(c2ccc(F)cc2Cl)=O)CCC(N=c2[nH]nc(CO)s2)(CO)CC1 84661,Cc1cc(C(=O)N(C(C)(C)CC(=O)NC2CCCC2(C)O)C)nc(O)c1 84662,C1(C(=O)NCC2(C(C)NC(Cc3c(C)ocn3)=O)CC2)CC2C=CC1CC2 84663,C1(COC)CN(C(C2CC3CCC(C2)O3)=O)CCN1C(=O)CNC(=O)OC 84664,N1(C(c2c(OC)c(C)ccc2)=O)Cc2ccnn2CC(NC(=O)CC(F)F)C1 84665,c1(C(N(C2CCN(C(=O)CSCc3nnc[nH]3)C2)CC)=O)cccc2sncc12 84666,c1(C(CNC(=NCC2CCC(SC)C2)NC2CCC2)N(C)C)ccc(F)cc1C 84667,N1(C(CN2CCC(C)C2)=O)CC2CCCC2C1C(N1CC2CC(C1)C2(C)C)=O 84668,C=CCC(C)(C)C(=O)N1C2CCC(C2)C1C(=O)NC1COCC1C=C 84669,c1(OC(C(=O)NC2CC(CNC(c3c(C)cns3)=O)C2)C)ccc(Cl)cc1 84670,C1(O)(CNC(C(Cc2ccccc2)OC)=O)CCN(C(=O)CCC(C)(C)C)CC1 84671,C1(C(=O)NCCCOCCCNC(c2cnc(C(C)(C)C)s2)=O)CN2CCC1C2 84672,N1(C(C=CC(C)C)=O)CCC2CCN(C(c3ccc(F)c(C(F)F)n3)=O)CC2C1 84673,c1(C(=O)NCC(CN(C(=O)C=C(C2CC2)C2CC2)C)O)c(Cl)cccc1Cl 84674,N1(C(C2CN(C(C3C(COC)CC3)=O)CC2C(C)C)=O)CCC(C2CC2)C1 84675,C(CC(C)(C)C(=O)NCC(CO)NC(C1(F)CCN(C(C)(C)C)C1)=O)OC 84676,c1(C(N(CCCCNC(CC(CC)OC)=O)C)=O)cc2cccc(Cl)c2[nH]1 84677,c1(C(=O)NCc2ccc(C(C)NC(COCC)=O)cc2)nnn2c1CCCCC2 84678,C(=O)(C(C)C1=CCCC1)NCc1ccc(C(C)NC(c2c(C)[nH]cc2)=O)cc1 84679,N1(C(C2CC(NC(CCCOCCC)=O)C2(C)C)=O)CC2(C1)CC(C)(C)C2 84680,C(=O)(CCN=[N+]=[N-])N(CCC(=O)NC(c1nc(=O)o[nH]1)C)CC1CC1 84681,CC(N=c1[nH]c2c(c(=NCc3ccn(C)n3)[nH]1)CCCC2)c1ccc(O)nc1 84682,C1(N(C(=O)C(F)C2CCCC2)C(=O)CC2CCC2)CCC2CCC12 84683,Cc1cc(C(N2CC(NC(c3cc(C4CCC4)nn3C)=O)C2)=O)ncc1C(N)=O 84684,C1(C(N(CC#CC)C)=O)CC2(CC2)CN1C(C1CC12CCC2)=O 84685,c1(C(=O)Nc2c(C)cc(NC(C3CCCOC3)=O)cc2)ccnc2c1cnn2C 84686,C1(C(N(CCCNC(c2ccnn2C)=O)CC)=O)CCCOCC1 84687,C(C(C(=O)NCCc1cn(C)cn1)NC(=O)Cn1cccn1)OC 84688,C1(C(=O)NC2(CN(C(=O)Cc3ccc(F)cc3)C)CC2)Cc2cc(Cl)ccc2O1 84689,S(=O)(=O)(c1cc(Br)c(C)cc1F)N1CCCC(CN(CCC)C)C1 84690,Cc1ccc2c(C(=O)NCCC(C)NC(=O)C(C)C(C)(C)C)coc2c1 84691,N1(C(C(CCOC)C)=O)CC2(CCCC2NC(=O)CC2(OC)CCOCC2)C1 84692,N1(C(c2c(C)nc(Br)s2)=O)CCC2C(CCN2C(c2cc(Cl)cc(Cl)c2Cl)=O)C1 84693,CCCC(CCC)C(=O)NC1CN(C(=O)Cc2cc[nH]n2)C1 84694,C1(N(C(c2cnc(CCCC)[nH]2)=O)C)CCCCN(C(c2cc(C#N)no2)=O)C1 84695,C(C(C(C)(C)C)NC(C1(C)CC1(Cl)Cl)=O)NC(C(C)c1cncs1)=O 84696,C1(NC(C=CCOC)=O)C2CC1CN(C(c1ncoc1C)=O)C2 84697,N1(C(CSC2C(=O)OCC2)=O)CCC2(CC1)CCN(C(C1CC1F)=O)CC2 84698,C1(NC(CCOCC)=O)CC(C)(NC(c2cnc[nH]2)=O)C1 84699,C1(NC(CN(c2ncccn2)C)=O)CCCCN(C(=O)CCOCC2CCCO2)C1 84700,N1(C(C(CC)(C)C)=O)CCC(O)(CCNC(c2cc(C)c(C)nn2)=O)CC1 84701,C1(CC(C(=O)NC2CC2)N(CC)Cc2ccc(O)cc2)CCOC(C)(C)C1 84702,C12(CNC(c3c(OC)nn(C)c3)=O)CC(C1)C(NC(=O)C1=CCOCC1)CO2 84703,c1(OC)cc(=NC(=O)C(CCC(C)C)NC(c2ccsn2)=O)[nH]n1C 84704,N1(C(c2n(C)c(S)nn2)=O)CC(CNC(=O)COCC2(F)CC2)CC12CCC2 84705,Cc1cccnc1CC(=O)N(C1CCN(C(=O)Cc2ccc(Cl)cc2)CC1)C 84706,c1(C(=O)NCC(CC)NC(=O)CCCCCSC)c(C)cccc1O 84707,C1(C(=O)NCCN2CC(Cn3ccnc3)C2)COC(C2CC2)C1 84708,C1(CCC)CN(C(=O)C(C2(O)CN(C(=O)Cn3cnnn3)C2)F)CCO1 84709,C(C(C)CC(=O)N(C(C)C(C)(C)O)C)NC(c1c(C)nco1)=O 84710,C1(C(N2CC(CNC(=O)C(F)(F)CC3CCCO3)C2)=O)CCc2[nH]nc(O)c2C1 84711,Cc1nc(CC(=O)NC(c2cccnc2)C(=O)NCCCC(=O)N(C)C)cs1 84712,CC1CC(C)N(C(c2coc(CO)c2)=O)CCN1C(=O)CC1CN(C)C1 84713,C(=O)(C(O)CC(F)(F)F)N(C1CCN(C(c2ccc(O)nc2Cl)=O)C1)CC1CC1 84714,Cc1nc(CC(F)(F)F)sc1CC(=O)NCCN(C(=O)C(O)CF)C(C)C 84715,C1(C)(CNC(c2cn(C)nc2C(F)F)c2n(C(C)C)nnn2)CC2CC2C1 84716,C12(NC(C(C)=C3CC3)=O)CCCC1N(C(c1cnn3c1OCC3)=O)CCC2 84717,C12(NC(CCC)=O)CC1CN(C(c1cnn(Cc3ccccc3)c1F)=O)C2 84718,C1(NC(CC2C(OC)CC2)=O)CCC(NC(=O)CC=Cc2ccccc2)CC1 84719,C1(CC(F)F)(C(=O)O)CCN(C(=O)C=Cc2cccnc2)C1 84720,CC(C)CN(CC(O)C1CC1)C(C)C 84721,C1(CNC(C(C)OCCN(C)C)=O)CN(C(C2C3CC4C(C3=O)C24)=O)CC12CC2 84722,N1(C(C(C)Cn2ccnc2)=O)Cc2cccn2CC(C(N2CCOCC2)=O)C1 84723,CC1CC(CNC(=O)CCOCC(F)F)CN1C(=O)CCN1CCCC1=O 84724,C1(C(=O)NC2C(NC(=O)CCc3ccc(F)cc3F)CC2)Cc2ccccc2C1 84725,C12(NC(c3cn(CC(N)=O)nn3)=O)CCCC1(F)CN(C(C1CCC1)=O)C2 84726,CC1CC2(CC(C(=O)NOCC(=O)NCC(O)C3CC3)C2)C1 84727,n1(CC(=O)N(C(CNC(COCCSC)=O)C)C)ccc(=O)c([N+](=O)[O-])c1 84728,C1(NC(CC(C)(C)C#N)=O)CCCCCN(C(=O)C2=CCCC2(C)C)C1 84729,N1(C(C(CC)OCC)=O)CCN(C(=O)C=Cc2c(C)coc2C)C(CC)C1 84730,c1(NC(C(c2csc(Cl)c2)N(CC(C2CCCC2)OC)C)=O)ccc(F)cc1 84731,c1(OCC)oc(C)nc1C(=O)NC1CC(N(C(=O)CC(O)c2ccccc2)C)C1 84732,C(C(F)(F)C(=O)NC1CCOCC1C(=O)NCCC(C)(O)C1CC1)OC 84733,C12CCCCCN1C2=O.C1(C(C(=O)NCCOCCOCCO)=O)CC(F)(F)C1.CO 84734,c1(NC)ccc([N+](=O)[O-])cc1C(=O)NCCC1CN(C(=O)CC2(C)CC2(F)F)C1 84735,Cc1nn(CC(=O)NCCN(CCOCCO)C(C2(O)CC(F)(F)C2)=O)c(=O)o1 84736,C1(NC(c2cccc(C)c2)=O)CC2CCC(C1)N2C(C1(CF)CC2(CCC2)C1)=O 84737,c1(CN2C3CN(C(C4N(C)CCC4)=O)C(C3)C2)ccc(F)c([N+](=O)[O-])c1 84738,C1(C)(C(N(CCCCCNC(C(CC)N(CC)CC)=O)C)=O)CCCNC1=O 84739,C1(C(N(C2CCCN(C(C(c3ccn(C)n3)C)=O)C2)CC)=O)CCCC(C)(C)C1 84740,c1(C(N2CC3C(C(=O)NCCCC(=O)OC)(CC3)C2)=O)c(F)cc(Br)cc1Br 84741,c1(CCC(=O)NCC(CNC(C2(CC#C)CCOCC2)=O)O)c(F)cccc1F 84742,C(CC(=O)NC1CCC(c2nncn2C)CC1)(C(F)(F)F)OCC 84743,C1(NC(c2ccn(CC(C)C)n2)=O)(CO)CCCN(c2ccc(C#N)nc2)C1 84744,Cc1ccc(C(c2nnnn2C)NC(c2cccc(F)c2C)C)cc1Cl 84745,CC1(C)CCCC(CC(=O)NCC2(C)CCCC2NC(=O)Cn2cccn2)C1 84746,N1(CC(=O)NCCCC(C)SC)CCNC(=O)C1.C12(CC1)C(=O)N2 84747,C(=O)(CCCC(F)(F)F)N1CC(C)C(C)(C(=O)NC2CCn3ccnc3C2)C1 84748,C1(C(N(C(CNC(=O)C(C)NS(C)(=O)=O)C2CC2)C)=O)CCCN1C1CC1 84749,c1(C(=O)NC(c2ccc(F)cc2)CC)cc(C)c2sccc2c1 84750,C1(NC(C2C(=C)C2)=O)CC(C)CN(C(c2ccc(-n3cccc3)cc2C)=O)C1 84751,N1(C(c2nc(OCC)oc2)=O)CCC(NC(C2CC(=O)N2)=O)C(C)(C)C1 84752,C1(NC(c2ccnc(OC)n2)=O)CC2CC1CC2C(=O)N(C)Cc1ccoc1C 84753,c1(C(N2CCC(n3cncn3)C2)C(=O)NCC(=C)C)cc(F)ccc1Br 84754,C(Cn1cncn1)(C(=O)NC1C2CCCC12)NC(C1CC(=C)C1)=O 84755,c1(OC)cc(C)cc(C)c1S(=O)(=O)N1CCCCCC1c1ccc(C(F)(F)F)cc1 84756,N1(C(c2c(CC)onc2C)=O)CCC(NC(=O)C=CC2CCCC2)C(C)C1 84757,c1(C(=O)NCC2C3CN(C(Cc4c(C)n(C)nc4)=O)C2C3)n[nH]c2c1CCCC2 84758,C=CCC(C)(O)C(=O)NC1C2CC3C1C3C2C(N1CCN(C)C(CC)C1)=O 84759,C1(C2N(C(C3(CCC=C)CC3)=O)CCC2)CCN(C(=O)CC(C)CC)CC1 84760,C=CC1OCCCC1C(=O)N(C)CCOCCN(C)C(c1ccc(F)cc1N)=O 84761,C1(C(=O)NCCCCCN(C)C)CCN(C(C2(C)C=CCCC2)=O)CCO1 84762,C1(NC(C2(Br)CC2)=O)C2CN(C(C3(n4cccn4)CCOCC3)=O)CC12 84763,C(=O)(C1=NOC2(CCOC2)C1)N1CCCN(C(C2N(N=O)CCCC2)=O)CCC1 84764,CCCC(C(=O)NCC(C)(C)C(=O)NCC1OCCC1C)N(C)C 84765,C(CN=C(NCC1CC2(C1)CC21CCC1)N1CCC(C(F)F)CC1)OCC 84766,c1(N(C(=O)C(C)OC2CCCC2)CCN(CC)CC)ncc([N+](=O)[O-])c(C)n1 84767,C#Cc1cc(F)cnc1NC(C1CN(C(c2cncc(F)c2)=O)CCC1O)=O 84768,N1(C(c2c(OC)nsc2OC)=O)CCC(C)C(NC(C2SCCCS2)=O)C1 84769,C1(CNC(C(COC)C)=O)CN(C(=O)C(c2ccc(C)s2)C)CCC12CCC2 84770,c1(C(=O)NCCC(C)N(C(=O)CC2(C)CCCCC2)C)cc(Br)cn1C 84771,CCC(C)CC(=O)NCC1(NC(=O)CSCC(N2CCOCC2)=O)CCCC1 84772,C1(F)(C(N(CCCCC=C)C)=O)CCN(C(C2SCC=C2C)=O)CC1 84773,Cc1cc(C(=O)Nc2ccnn2-c2ccccc2Cl)c(C)[nH]1 84774,C(=O)(C1=NOC2(CCOC2)C1)N1CCOCC(F)(CNC(C2CC=CC2)=O)C1 84775,C1(NC(CN(C2CCCC2)C)=O)CCN(C(=O)CSc2nncs2)CC1 84776,C1(C2CCN(C)CC2)(C(=O)NC2CCCC(CNC(COC(CC)C)=O)C2)CC1 84777,N1(C(c2ccc(N)c(F)c2)=O)CC2(CCCC2NC(C2CCCC3(CC3)C2)=O)C1 84778,Cc1c(NCCCCCN(C)C)ncnc1NCC#CCN1CCCC1 84779,N1(C(c2ccc(NC=O)cc2)=O)CC2CC1CN2C(c1cnc(C2CC2)o1)=O 84780,c1(C(N2CC(CC(=O)N(C)Cc3ccccc3Cl)OCC2)=O)cnc(O)cc1O 84781,c1(C(N2CCCC(N(C(=O)C(F)C3CC3)CCF)C2)=O)cc(Cl)cc(Cl)c1 84782,c1(CC(=O)N(C)CC2(O)CN(C(c3cc(Cl)c[nH]3)=O)C2)c(F)cccc1F 84783,C1(C(=O)NC(C(C)NC(c2cc(C(F)(F)F)cs2)=O)(C)C)CCCN(CCF)C1 84784,C1(CC)C(NC(C2CC2c2cccs2)=O)CCN1C(=O)CCOc1cccnc1 84785,CC1CN(C(c2ccoc2)=O)CC2(CCN(C(c3cccc(N)c3O)=O)CC2)O1 84786,C1(NC(CCOCCN(C)C)=O)CC(O)CN(C(c2ccc(O)nc2Cl)=O)C1 84787,C(=O)(C(O)CC[S+](C)C)N(C)CC1N(C(CC(C)(C)SC)=O)CCOC1 84788,c1(CN2CCC(CN(CCOC)C)C2)nc(N(C)C)[nH]c(=N)n1 84789,Cc1cc(C(=O)N(C)CC2(NC(C3CCC(C#N)C3)=O)CC2)c2c(C)noc2n1 84790,CN1C2CCC1CC(C(N1CC3(CCC3NC(c3cccn(C)c3=O)=O)C1)=O)C2 84791,CC1CN2CCN1CC2C(=O)N(C)CC1CCN(C(c2cnc(S)nc2)=O)C1 84792,S(=O)(=O)(c1cn(C)nc1C)Nc1ccc(-c2c(C)ccc(Cl)c2)nc1 84793,C(=O)(C(C)(C)C1CCCN1Cc1ccncc1)N(C1CC(=O)C1C(F)(F)F)C 84794,CC(CN(C)C)CCC(=O)NC1C=CC(NC(=O)COCC2CCOCC2)C1 84795,c1(C(N2CCN(CC)CC2C)C(=O)NC2CCOC2)nc(Cl)cc(C)c1Br 84796,c1(C(=O)NCCCNC(c2cccc(C3CC3(F)F)c2)=O)cc(Cl)cc(Cl)c1F 84797,C(=O)(CC1OCCc2ccccc21)NC(CNC(C1(OC(C)C)CCC1)=O)(C)C 84798,C(CCC(C)C)(C(=O)Nc1cnc(C)c(Cl)c1)NC(CN(C(=O)OC)C)=O 84799,c1(SC)cc(C(=O)NC2CC2NC(=O)Cc2cncn2C)ccn1 84800,CCC(C)CCCCC(=O)NS(=O)(=O)c1ccc(C#N)o1 84801,c1(N2C(CN(C)C(c3ccnc(F)c3Cl)=O)COCC2)ccc2nccnc2n1 84802,c1(C(=O)NCCC(C)NC(c2cnn(C)c2Br)=O)ccc(C(=O)CF)cc1 84803,C1(C(N2C(CNC(c3n(C=C)ncc3)=O)CCCC2)=O)CCc2nnc(O)n2C1 84804,CC1(CCNC(C2(n3cncn3)CC2)=O)CCN(C(C2CCCC(=O)O2)=O)C1 84805,c1(NCCNC(C2CCCN(C(CSCC#C)=O)C2)=O)cnc(CC)nc1C 84806,C1(C(N(CC#C)CCO)=O)N(C(=O)C(C)CSC)CCC1(C)C 84807,Cc1ccc(F)cc1C(N1CCC(CNCC(c2ccccc2)C)C1)=O 84808,C(=O)(C1=NOC(C)(C)C1)NC1CCCC(NC(c2c(C)ncc(C)c2)=O)CC1 84809,C1(NC(C(C)(C)NC(Cc2cn(C)nc2)=O)=O)CC12CC(O)C2 84810,C(=O)(CCCC(=O)N(c1ncnc(C)c1Br)C1CCNCC1F)OC 84811,C#CCC(C)(C)C(=O)NC(C1CCCN(C(c2cn(CC)nn2)=O)C1)C 84812,N1(C(c2ccc(CSCCC)o2)=O)CCCC(C)C1CNC(c1cncs1)=O 84813,NS(=O)(=O)c1ccc(SCC(N2CC(C3=NOC(C)(c4nn[nH]n4)C3)C2)=O)cc1 84814,N1(C(CCN(CCC)C)=O)CC(c2ccccc2)(NC(c2occc2Cl)=O)C1 84815,C1(NC(c2ccns2)=O)CCN(C(=O)CCOc2ccccc2Cl)CC12CCC2 84816,c1(NC(C2C3(CCN(Cc4cc(C)c(Cl)nc4)C3)C2)=O)c(Br)cc(F)c(F)c1F 84817,c1(CN(C)C(C2(CNC(C34CCC(C3)C4)=O)CC2)=O)ccn(C)c1 84818,c1(C(N2CC(C)(CC(=O)Nc3ccc(Cl)cc3)C2)=O)cc2cc(Br)ccc2s1 84819,C(=O)(CCCCC(=O)NC1CN(C(C2(O)CCOC2)=O)CC2(CC2)C1)NC 84820,C1(NC(=O)CCCn2cncn2)CCOC1(C)C.c12nocc1C(=O)NC2C 84821,C(C(C)(C(=O)NCC(CO)NC(C1(CCc2ccccc2)CC1)=O)OC)OC 84822,n1(CCCC)nc(C)c(C(=O)NC23CC2CN(C(=O)CN2CCCC2C)C3)c1Cl 84823,N1(CC2CCN(C(Cn3c(C)cc(C(F)F)n3)=O)C2)CCC(O)C(C)C1 84824,Cc1cc(C(=O)NC2(C)CC(NC(C3CC(=O)NC(C)C3)=O)C2)cc(C)n1 84825,COn1cnc(C)c1C(N1CC(NC(c2c[nH]nc2C(C)(C)C)=O)C(F)C1)=O 84826,N1(C(C2CC(OC)C2)=O)CCC2(CC2)CC1C(=O)NC(CCO)C1CCC1 84827,CC1OCCC1(F)C(=O)NCCC1CCCN(Cc2ncc(Cl)s2)C1 84828,C1(CNC(c2ccc(CC)[nH]2)=O)CN(C(=O)CSc2cn[nH]c2)CCC12CCC2 84829,c1(NC(C2NCCN(C(c3c(C)ncnc3)=O)C2)=O)ncnc2[nH]c(Br)nc12 84830,N1(C(C=CC)=O)CC(NC(=O)C(Cc2ccccc2)CC(C)C)CC2(CCC2)C1 84831,CC1CCOC1CCNC(=O)C(C1(C)CC1)NC(=O)Cc1ccon1 84832,C1(C(=O)NCc2cccnc2Br)CC12CCN(C(c1cn[nH]c1)=O)C2 84833,c1(C(N2CC(C)(NC(C(C)C)=O)C2)=O)ccc(NC2CC2c2ccc(Cl)s2)cc1 84834,C1(C(=O)NCCC2(C)CCCO2)CCN(C(=O)CC2CCCC3CC23)CCO1 84835,C1(NC(CC(C)C)=O)CC2CC(NC(C3CNC(=O)N3)=O)CC12 84836,S(=O)(=O)(c1cccc(=NCC(C)C(C)C)[nH]1)N1CCC(C(C)CCCCO)CC1 84837,N1(CC)CCC(CNC(c2conc2NC(=O)CC2CC3CC3C2)=O)C1 84838,c1(C2(C(=O)NCC(C)(O)CNC(c3ccncn3)=O)CC2)cccnc1Cl 84839,C1(CNC(=O)C(N2CCCC2c2ccc(Cl)cc2)=O)CCCS(=O)(=O)C1 84840,C1(=CCNC(C=CCCC(C)C)=O)CCN(C(c2c(C(C)C)cnn2C)=O)CC1 84841,C(=O)(C(F)CC(CC)CC)NCC(=C)CCNC(C1(C(=O)NC)CCOCC1)=O 84842,CCCCC(CC)C(=O)N(CC(=O)N(C)Cc1ncn(C)n1)CC1CC1 84843,N1(C(c2cnn(C(C)(C)C)c2)C(=O)NC(C)C)Cc2ccccc2C(C)(C)C1 84844,CC1CSCC1(c1nnnn1C(C)(C)C)NCCOc1ncc(Cl)cn1 84845,c1(C(C(=O)NCC#CCNC(C2OCCN(C)C2)=O)=O)ccc(F)cc1F 84846,C1(C(N2CCC(Cc3onc(C)n3)CC2)=O)CCOC2(CCC2)C1 84847,Cc1cc(C)c(N(C(c2cccnn2)C2CNC2=O)CC2CCCO2)c(C)c1 84848,C(=O)(NNc1ccc(Br)c(F)c1F)NCCC1(C(=O)OCC)CCOCC1 84849,C1(C(=O)NCCOCCOCC)CCOCC1NC(=O)C=NOC 84850,CC1CN2CCN1C(C(=O)NC1C=CCN(C(c3cnc4[nH]ccc4n3)=O)C1)C2 84851,C1(c2cn(Cc3c(C)nc(CC)o3)nn2)CN(C(c2ccnn2C)=O)CC1(C)C 84852,C(C(C)(O)CC(=O)NC(C)CN(C(=O)C(c1ccc(Cl)cc1)(C)C)C)OC 84853,N1(CC(CC)CC(C)(C)C)CC(C(=O)OC)C2(CN(C(=O)OC(C)(C)C)C2)C1 84854,N1(CC(=O)N(C)CC2C(NC(C3N(C)CC3)=O)CCC2)C(=O)CCCC1=O 84855,C1(NC(CCC)=O)CC(C)(C(=O)NCC(CO)C2CC2)C1 84856,n1(CC(=O)NCC(CNC(C23CCCC(CO2)C3)=O)CO)cnc2ccccc12 84857,C1(C(N2CC(CNC(C(CC)n3ccnc3)=O)OCC2)=O)CC(C)(C)C(C)(C)C1 84858,C1(CNC(=O)C(c2cccnc2)C2CCCCC2)CCCC1C(=O)O 84859,FC1CC2CC1CC2NCc1cccc(C2CC2)c1 84860,N1(C(=O)CC2CCCC2(F)F)CC2CCCC(C1)N2C(c1cncc(Cl)c1)=O 84861,c1(C(=O)NC(C)CCNC(c2cc(Br)co2)=O)n[nH]cc1[N+](=O)[O-] 84862,c1(C(=O)OC)sc(-c2ccc(C(=O)NC(C)CN(C(=O)C(N)=O)C)cc2)nc1C 84863,Cn1cc(C(=O)NCC23CC2CN(C(c2ccc(O)nc2Cl)=O)C3)ccc1=O 84864,C#CCCCCCC(=O)N1CC2CCC1CN2C(=O)CCCC 84865,N1(CCC(=O)NC2CC3CN(C(C(C=CC)O)=O)C2C3)CCc2ccccc2C1 84866,c1(C2OCCN(CC(=O)Nc3nnc(CN(C)C)s3)C2)ccc(F)c(F)c1 84867,N1(C(c2n(CC)cc(Cl)c2)=O)CCCC(N(CC(N2CCC(C)CC2)=O)C)CC1 84868,c1(C(=O)NCCNC(CC2C(C)C2)=O)cccc2c1NC(=O)CC2 84869,c1(CCC)cc(=NCC2CN(C(c3ncsc3C(C)C)=O)C2)[nH]c(Cl)n1 84870,N1(C(c2c(C)cno2)=O)CCC2(CCCN2C(c2ccc(C(C)C)c(Cl)c2)=O)C1 84871,C1(F)(CNC(=O)Cc2ccc(Br)cn2)COCCN(C(c2ccon2)=O)C1 84872,C1(SCC)CC(C(=O)NCC(C)(C)CCNC(c2nc(O)sc2C)=O)CCO1 84873,c1(C(N2CCN(C(C(C)=C3CC3)=O)CC2C2CC2)=O)cc2cc(Br)ccc2[nH]1 84874,N1(C2CCN(C(CSCC(N)=O)=O)CC2)CCN(C(=O)CO)CC1=O 84875,CC(=O)CCCC(=O)N1CCC(C)C1CNC(=O)C(O)C1CCC1 84876,C1(NC(CN(C)C(=O)C2CC2)=O)CS(=O)(=O)CC1NC(=O)Cc1c(Cl)cnn1C 84877,c1(CNCC2N(C(c3c(OC)cncc3)=O)CCOC2)cc(F)ccc1Br 84878,N1(CC#C)CCN(C(CC2CCOC2)C(=O)NCc2nnn(C)n2)CC1 84879,CS(=O)(=O)C1CC(C(=O)NCC2CCN(C(=O)CC3C=CCC3)C2)C1 84880,C1(CNC(c2c(CC)non2)=O)CCN(C(c2cc(OC)cc(C)c2)=O)CC1C 84881,C(=O)(C1CC(=O)c2c(F)cccc21)NCC(CNC(c1c(C)cccc1Cl)=O)C 84882,c1(NC)c(OC(C)=O)cccc1OC.n1(CCOC)nnnc1C(C(C)C1CC1)OC 84883,C1(NC(CC2C(C)(C)C(O)C2)=O)CC(N=c2ccn3nccc3[nH]2)C1(C)C 84884,N1(C(C2N(C)CCOC2)=O)CC2(C)CN(C(C3CC(F)(CO)C3)=O)CC2(C)C1 84885,N1(CC)CC2CN(C(=O)C(O)CNC(C3(NC(N)=O)CCCCC3)=O)CC2C1 84886,c1(C(N2CC(OC)C(NC(C3(C)CC=CCO3)=O)C2)=O)cc(Cl)cc2c1CCC2 84887,C(=O)(C=CS(F)(F)(F)(F)F)NC1CC2CN(C(CN3C(=O)CC(=O)N3)=O)C(C1)C2 84888,c1(C(=O)NC2C(C)CN(C(=O)C(Cl)=CCl)C2)ccc(O)c(CO)c1 84889,C1(NC(c2c(CC)n(C)nn2)=O)CC(CNC(=O)CCc2cnn[nH]2)C12CCC2 84890,C(=O)(C(CNC(=O)C1=CCCC1C)C(C)C)NC(COC)(C)C(N)=O 84891,CN1CCn2ncc(C(=O)NC3(C)CCCN(C(=O)COCC(C)(C)C)C3)c21 84892,N1(C(c2ccc(N)cc2F)=O)CCC2(NC(=O)CC3=CCCC3)CCCCCC12 84893,C1(C(=O)NC2C=CCN(C(Cc3scc(C)c3)=O)C2)CCc2cnnn2C1 84894,Cc1ccc(C(N2CCC(NC(=O)CC3CCC(C)(C)C3)CC2)=O)c(O)c1 84895,CC1CC=C(C(=O)NC2(C(=O)NCC3(CO)CCC3)CSC2)CC1 84896,c1(NC(=O)NC2(C(=O)NC3CC3N)CC2)ccccc1.O=C(CC1CSC1)N 84897,CN1CCCC(CCC(=O)NC2CC(NC(C3(CS(C)(=O)=O)COC3)=O)C2)C1 84898,c1(C(=O)NC2CC(NC(c3cc(C)c(Br)s3)=O)C2)cccc(Br)c1O 84899,N1(C(C(Cc2c(C)nc[nH]2)O)=O)CCC(NC(=O)CCCCCN(C)C)C12CC2 84900,O=C(C1=CSCCO1)NCC(c1ccccc1F)NC(C1CC1F)=O 84901,N1(C(c2c(C(C)C)cco2)=O)CC(NC(c2ccc(Cl)s2)=O)C2(CCOCC2)C1 84902,N1(C(C(C2CCCNC2)C)=O)CCCC(CC2(C(F)(F)F)N=N2)C1 84903,c1(CC)ncccc1NC(=O)CC1CCCN1C(c1cncc(Br)c1)=O 84904,c1(C(=O)NCC2CCN(C(CC(n3ccc(C)n3)C)=O)C2)cccnc1C 84905,CC1=C(C(=O)NC2CC(N(C)C(c3ccnc(OCCO)c3)=O)C2)SCCO1 84906,C1(CNC(C(C(C)C)C)=O)CN(C)CCN1C(c1ccc(C(N)=O)o1)=O 84907,c1(C(c2nnnn2C2CC2)NCc2c(OCC)cccc2)cc(Cl)ccc1[N+](=O)[O-] 84908,C(CC(=O)N(C1CC2CC2C1)C)(C(C)CC)NC(c1cn(CC=C)nn1)=O 84909,c1(N(C)C)cccc(C2CCN(C(C3CCC4CC34)C(=O)NC3CC3)C2)c1 84910,c1(C(=O)NC2CCN(CCNC(CC(C=C)C)=O)CC2)c(F)ccc2n[nH]cc12 84911,C1(C(C)C)CN(C(C2CC(=O)C2C)=O)CCN1C(C1CS(=O)(=O)C1)=O 84912,C(=O)(C(C)(C)C(=O)N1CCC(C(C)NC(=O)C(C)=CC2CC2)CC1)OCC 84913,c1(C(N(CC=CC(N2C(C(C)O)COCC2)=O)C)=O)coc2ccccc12 84914,c1(C(=O)NCC(CC=C)NC(=O)C(C)(F)CCCC)cnc2c(ccn2C)c1 84915,N1(CCC(N2CCC(NC(C3CCC(C#C)CC3)=O)C2)=O)Cc2ccccc2C1 84916,c1(C(N(C(C)CNC(c2cnn(C)c2Cl)=O)CC)=O)ccc(NC(C)=O)c(F)c1 84917,N1(C(c2c(F)ccc(CC)c2)=O)CCC2(CCC2NC(=O)C2=CCCC2C)CC1 84918,C=CC1(C(=O)NCCCCCN(C(=O)Cc2csc(NC=O)n2)C)CCC1 84919,C1(N(C(=O)C=Cc2cc[nH]n2)C)CCCC(NC(=O)C=Cc2ncc[nH]2)C1 84920,C1(C)(C(=O)NC2CCC(C(=O)NC(CCC)c3ccco3)C2)CCC(=O)N1 84921,C1(C(=O)OCC)CC2CC2N1C(C1(F)CC1(Cl)Cl)=O 84922,c1(CNC(C(C)N(C(C2C(CC)C2)=O)C)=O)ccnn1C 84923,c1(C(=O)NC2CC(NC(c3ncnc4sccc34)=O)C2)ccc2cc[nH]c2c1 84924,c1(C(C(=O)NCCC)N(CC)Cc2ccc(OC)cc2)ccc2c(c1)CC(C)O2 84925,c1(C(N(CCC)CCNC(C23CCC(F)C2CC3)=O)=O)nc(O)nc(O)c1F 84926,C1(C)(NC(C2C(C)OCC2)=O)CCCN(C(c2c[nH]cc2Br)=O)C1 84927,C(N=c1[nH]c2c(c(=NC3CCOC(C)(C)C3)[nH]1)CCC2)c1ccc(C)c(N)c1 84928,Cc1ccc(C)c(C(N2CC(CN3CCN(C(C4CC4C#N)=O)CC3)C2)=O)c1C 84929,N1(C(C2CCC(=O)NC2)=O)CCN(C(=O)Cc2cc(Cl)ccc2Cl)C(CCO)C1 84930,Cc1cc(C(=O)NC2COCC2NC(=O)C#CC(C)C)c(C)cc1Br 84931,C1(NC(C2CCN(CC3CC3)CC2)=O)CN(C(C2(O)CCOC2)=O)CC12CCC2 84932,c1(C(=O)NCC(N(C(c2cc(C)ncn2)=O)C)C2CC2)ccc(Cl)cc1O 84933,c1(C(=O)OC)cncc(OCCNc2ccsc2Cl)c1 84934,CC1CC(NC(c2cnc(Cl)n2C)=O)CCN1C(c1cc(F)cc(Cl)c1)=O 84935,C1(CNC(c2ccc(CSC)o2)=O)CCCCC1NC(=O)CCc1n[nH]c(=N)s1 84936,C1(NC(=O)C2=CCC2)COC2(CCCN(C(c3sccc3C(F)F)=O)C2)C1 84937,c1(C(N2C(C(C)NC(C(CCSC)N(C)C)=O)CCC2)=O)cnc2sccc2c1 84938,C12(CNC(c3ccccc3F)=O)CC(C1)C(NC(C1CC13CCC3)=O)CO2 84939,C1(C(N2CCC(N(C(C3C(=C)C3)=O)CC)C2)=O)CC2(C1)CS(=O)(=O)C2 84940,CCC(C)C(C(=O)NC1CCN(C2CC2)CC1)N(C(=O)CC(C)C)C 84941,C1(NC(CCC=CC)=O)CN(C(C2(F)CCCC2)=O)CCC1CO 84942,N1(C(c2ccn(C)c2-c2ccccc2)=O)CC(S(N)(=O)=O)C1 84943,N1(C(C2CC(NC(c3ncc(C)[n+]([O-])c3)=O)C2)=O)CC2CC3CC2C1C3 84944,C1(CNC(Cc2n(C(C)C)cnn2)=O)CN(CC(F)(F)C(F)F)CCC1(F)F 84945,Cc1cn2c(n1)CC(C(=O)NC1CCN(C(=O)CNS(C)(=O)=O)CC1CO)CC2 84946,c1(OC)cc(OC2CC2)ccc1C(=O)NC1CC(CNC(=O)CC2CCCO2)C1 84947,C1(CNC(CCC#N)=O)CCCN(C(C2CCC(C(N3CCCCC3)=O)C2)=O)C1 84948,N(C1COc2ccccc21)C(=O)CCn1cc(Cn2cccc2)nn1 84949,c1(CC(N2CCC(=CC=C)CC2)=O)ccc(-c2ccccc2)c(F)c1 84950,CCCC(C(=O)N(C)CC1CC(O)C1)NC(c1cn(C)cc1C)=O 84951,c1(CN=C(NC2C(C)(C)C(O)C2)NCc2ccco2)cc(Cl)cc(Cl)c1 84952,n1(CCC)cccc1C(=O)N(CCO)Cc1ccn(CC)n1 84953,C=CCC(C)(CC)C(=O)N1CCC(N2CCN(C)CC2)C(C)C1 84954,C1(N(C(C)C)C(c2c(CCN3CCCCC3)cccc2)(C)C)CC12CCNCC2 84955,C1(S(C)(=O)=O)(C(=O)NC(CNC(C(CC)(C)OC)=O)C)CCOCC1 84956,c1(C(=O)NCCC(C)NC(=O)C(C)(F)F)cc(Br)cc2ccccc12 84957,N1(C(c2cncc(C)c2)=O)CCN(C(C2(F)CCS(=O)(=O)C2)=O)CC1CC1CC1 84958,N1(C(c2cnn(-c3ccccc3)c2F)=O)CCCN(C(C2(F)CCOC2)=O)CC1 84959,C(=O)(C1=CCCC1C)NCCN(CCC)C(C1CC1c1cnc[nH]1)=O 84960,C1(OCCC(N2CC(CC(C)NC(C=C(CC)CC)=O)C2)=O)CCOCC1 84961,c1(C(=O)NCCC(C)NC(c2c(SCC)cccc2)=O)ccc2oncc2c1 84962,N1(C(C2CN(C(=O)NC)C2)=O)CC(C)(C)OC2(C1)CN(C(=O)Cc1cnoc1)C2 84963,C=CCCCCC(C(=O)NCCC)N(C1CCN(S(C)(=O)=O)CC1)C 84964,c1(CC(=O)NCC(C2CC2)NC(C(C)(O)C2CC2)=O)ccc2c(c1)OCCCO2 84965,C1(CCOC)(NC(=O)Cc2nc(C)cs2)CCN(C(C2CC2OC)=O)C1 84966,C1(c2nc(C)on2)CCCCCN1C(=O)CN1CCCNS1(=O)=O 84967,NC(=O)CCCC(=O)NC12CC(CNC(=O)CC3CC(O)C34CCC4)(C1)C2 84968,CCC(CNC(=O)C=NOC)(CC)NC(c1cnc(-c2ccccc2F)s1)=O 84969,c1(N(CCC(N)=O)C)nc(=NCCCCCO)[nH]c2c1SCC2 84970,C(C(CC(F)(F)F)NC(C1CC1(Cl)Cl)=O)NC(c1cncc(C2CC2)c1)=O 84971,C(C)(CC(=O)NOCCCO)N(C(C1C(C(C)=O)C1)=O)C 84972,c1(C(N2C3C(CNC(c4cc(OC)no4)=O)C(C3)C2)=O)cc2n(n1)C(C)CCC2 84973,C(=O)(C#CC1CCOCC1)N1C(C(N2CC(C=C)C2)=O)CN(C)CC1 84974,C1(OC)CN(C(=O)C=CC(C)C)C(C)(CNC(c2ccc(O)c(F)c2)=O)C1 84975,C(=O)(C1=CCN(C(=O)CC23CCCC2C3)CC1)NCCN(C(CC)C)C 84976,c1(OC)cnc(F)c(C(=O)NC2CCC(N(C)C(c3cccc[n+]3[O-])=O)CC2)c1 84977,N1(C(C=CCCC)=O)CCOC2(CCN(c3nc(O)c4ccccc4n3)C2)C1 84978,N1(C(C2C(C)=C2)=O)CCC(C2CCN(C(c3cccnc3N)=O)CC2)CC1 84979,c1(C(=O)NC2C(C)N(C(c3ccns3)=O)CC2)cc2c(F)ccc(Cl)c2[nH]1 84980,C1(NC(c2cnc(C)nc2)=O)C(C)(C)C(NC(=O)CC2CC2C2CC2)C1(C)C 84981,c1(C(N(C)CCOCCNC(C2(CO)CCCC2)=O)=O)c(Cl)cccc1[N+](=O)[O-] 84982,c1(C(N2CC(CCO)(NC(C=CC)=O)C2)=O)ccc([N+](=O)[O-])c(C)n1 84983,c1(C(=O)NCC2CC(CNC(c3c(Cl)nc(OC)s3)=O)OC2)cnc(O)cc1C 84984,N1(CC(c2ccc(C(N3CCOCC3)=O)[nH]2)=O)CCSC2CCC12 84985,CCCCC(C(=O)NCc1[nH]nnc1C)NC(=O)C=Cc1ccc(C)cc1 84986,C(CC(C)(C)C(=O)N1CCN(C(=O)CCCc2ccc(OC)cc2)C(C)C1)OC 84987,c1(C(C)(C)C)cnc(CNc2nccn2CC(F)(F)F)o1 84988,C1(C(=O)NC2CCC(NC(c3cccc(Cl)c3Cl)=O)C2)CCC2CC1CO2 84989,N1(C(CNC(c2[nH]cc(C(C)=O)c2)=O)C)CCC(C(=O)NC(C)(C)C)CC1 84990,CC1(C)C(C(=O)NCC(C)(C2CC2)NC(c2cc(F)cc(F)c2)=O)CCS1(=O)=O 84991,C1(C(N(CC(C2CC2)OC)C)=O)CNC(=O)CN1C(=O)Cc1cc(C)ccc1C 84992,Cc1cc(CN(C(N2CCCCC2c2ccc(C(F)(F)F)cn2)=O)C(C)C)cc(C)c1 84993,Cc1c(NC(=O)Cc2ccc(-c3cnn(CC#N)c3)c(F)c2)cccc1[N+](=O)[O-] 84994,C1(NC(Cc2c(C)non2)=O)CCCC2CN(C(c3cn(C)nn3)=O)CC12 84995,C1(C(=O)NC(C2CN(C(=O)CCCC3(C)N=N3)C2)C)CCc2cnn(C)c2C1 84996,Cc1cc([N+](=O)[O-])cc(C(=O)NC2CCN(C(=O)C#CC3CCCC3)C2)c1Cl 84997,C#Cc1ccc(F)c(C(N2CC(C)C(NC(=O)C=C3CCSCC3)C(C)C2)=O)c1 84998,c1(OC)cccc(CC(=O)N(C2CC(O)C2)CC2CCNC2)c1Cl 84999,C1(CC(=O)N(C(C)CC(=O)NC2CC2)C)CCCC(=O)N1.C12(CC1)C(=O)N2 85000,n1(CC)cc(C(=O)C(=O)NCC(C)(C)OCCNC(C2(C)CCCS2)=O)cn1 85001,C1(C(N2C(C(C)(C)NC(C=CC(C)C)=O)CCC2)=O)CCC(=O)NC1 85002,C1(C#N)(C(N2CC(C(C)NC(c3c(CC)con3)=O)OCC2)=O)CCCCC1 85003,c1(C(=O)OC)nn(C)nc1C(N1CC(CNC(C2(C)CCOC2)=O)(OC)C1)=O 85004,CCC(CC(=O)NCC1(C(=O)Nc2cccc(O)c2)CC=CC1)SC 85005,N1(C(C2(C)COC2)=O)CCOCC(F)(CNC(c2cn(C3CCC3O)nn2)=O)C1 85006,C1(CC)CC(N=c2[nH]c(=NC(C)c3ccccn3)[nH]c3c2CCCC3)CCO1 85007,C(CSC)(C(=O)N(C)CC1(O)CN(C(=O)C(C2CC(F)(F)C2)O)C1)OC 85008,N1(C(c2ccn(CCOC)n2)=O)CCSCC1CCNC(=O)C(C)CC1CCC1 85009,C(=O)(CC1=NNC(=O)C1)NCC1(CNC(C2OCC(C)C2)=O)CCOCC1 85010,N1(C(CCNC(C)=O)=O)C(C(=O)NCc2ccco2)C2CC(O)C1C2 85011,C(CCC)(CCCNC(=O)CCc1ncc[nH]1)NC(C(CC=C)NC(C)=O)=O 85012,c1(C(=O)NC(CC)CN(C(=O)CCC(C)C)C)cccc(F)c1C#N 85013,N1(c2snc(C)c2C#N)CCC2(NC(=O)CCCN3CCCC3)CCCCCC12 85014,c1(CN2C(CC(N3C(C(=O)OC)CSC3)=O)CCC2)c(C)[nH]c2ccccc12 85015,N1(Cc2cc(OC)ncc2Br)CC2CCN(C(c3nc(C)cs3)=O)C2C1 85016,CCC(CC(=O)N1CCCC1C1(NC(=O)CCCn2ccnc2)CC1)CC(C)C 85017,n1(CC(=O)NCC2(C(=O)NC3C(CNC(N)=O)CC3)CC2)cnc(C(N)=O)n1 85018,c1(C(=O)NCC(C)NC(c2oc(Br)nc2C(F)F)=O)cn2ccccc2n1 85019,N1(C(C(C)OCCCC)=O)CCC2(C1)CN(C(C1(C)CCN(C)CC1)=O)CCO2 85020,N1(C(C(CC)COC)=O)CCC(NC(c2cccc(-n3cncn3)n2)=O)C12CC2 85021,C1(C(C)C)COCCN(C(C2CCN(C(=O)C(C)(C)C3CC3)CC2C)=O)C1 85022,C1(NC(C(CC)c2ccccc2)=O)CCC(NC(=O)C(C)(C2CC2)OC)CC1 85023,c1(CC)nc(C(=O)NCC2C(CNC(=O)CC(C)N(C)C)C2(F)F)cs1 85024,C1(SC)CCN(C(C2C3CCCC23)C(=O)Nc2cccc(Cl)c2C)C2(CC2)C1 85025,C1(CC(=O)N(C(C(N2CCC(COC)C2)=O)C2(C)CC2)C2CC2)CCN(C)CC1 85026,N1(C(CN(C(CCc2c(C)noc2)=O)C2CC2)=O)CCCC1(C)CC(C)C 85027,c1(C(N(CCNC(c2c[nH]nc2Br)=O)CC)=O)nccc(OC)c1N 85028,N1(C(CCOCC)=O)CCC(C2CCN(C(c3ccnc(C4CC4)c3)=O)CC2)C1 85029,c1(C(=O)NCC(C)N(C(c2cn(CCC=C)nn2)=O)C)c(C)nn2c1NCCC2 85030,C(=O)(C(C)C(O)CC(C)C)N(C1CC(C#N)C1)CC(=O)NC(C=C)CO 85031,C(=O)(C(CNC(C1CCCC1O)=O)C(C)(C)C)NCCSC 85032,C1(CC(=O)NC2CCC(NC(C3(C)CCCOC3)=O)CC2)CCC(=O)NC1=O 85033,N1(C(c2c(C)c(O)ccc2)=O)CC(CNC(C2(C)CCN(C)C2)=O)CC(C)(C)C1 85034,c1(-c2nc(C(=O)NCC(CN(C(CCCC)=O)C)C)c(C)o2)ccc(Cl)c(Cl)c1 85035,C=CCC(CO)NC(=O)C(C)CNC(=O)CCC1CC1C 85036,N1(C(c2c(CC)scc2)=O)CC(C)(C)OCC1CNC(=O)C(c1ccc(C)o1)C 85037,C=CC(CCC)CC(=O)NC(CNC(C1(c2cccs2)CCCCC1)=O)C1CC1 85038,c1(N(CC(C2CCC2)OC)C)nc(N2CCCOCC2)c2c(n1)c(C)nn2C 85039,C1(C(=O)NCC(C)(C)NC(=O)CC2(C)CCCO2)CCC12CCC2 85040,N1(C(C2N(C)CSC2)=O)CC2(CNC(=O)C(F)C3CCC3)CC1CO2 85041,N1(C(c2cnc(CC)s2)=O)CCCC(C(C)NC(=O)C=CCN2CCOCC2)C1 85042,C1(CC(=O)NCc2nc(CNC(C3CCCN(C)C3)=O)sc2)CCCS(=O)(=O)C1 85043,N1(C(c2csc(C)c2N)=O)CCC(NC(C2CCC(C(N)=O)N2C)=O)CC(O)C1 85044,C1(C(=O)NC2CC(NC(c3c[nH]nc3CN(C)C)=O)C2)COCCN1C1CCCC1 85045,c1(C(N(C)CCNC(c2cnc(C3CCOC3)s2)=O)=O)csc2nnsc12 85046,CCC(C(=O)NCC1(C(=O)N(C2(C)CC2)C2CC2)CC1)n1ccnc1 85047,Cc1sc(N)c(C(=O)NCC2CCCC2NC(c2cnn(C)c2C(F)F)=O)c1C 85048,N1(C(c2cccc(CC)c2F)=O)CC2(CCCN(C(c3cccc(C)c3)=O)C2)C1 85049,N1(C(C(C2CCOCC2)OCC)=O)CCN(C(c2ccoc2)=O)C2COCC12 85050,N1(C(CC)=O)CCCC(C2(NC(=O)CCCCCF)CC2)C1 85051,Cc1n[nH]cc1CNC(=O)C=CCC1(NC(=O)CCn2ccnc2)CCC1 85052,C12(CNC(CC=CCC)=O)CC1CN(C(C13CC(c4ccccc4)C1C3)=O)C2 85053,c1(OC)ccccc1CN(C(c1csc(-c2cccs2)c1)C(=O)NCC(C)C)C 85054,N1(C(C(=O)N(C(C2CCCC2)C)C)=O)CCC(c2cccs2)CC1 85055,c1(C(N2C(CNC(C(C)CN(C)C)=O)CC3(CC3)C2)=O)cc2cc(N)ccc2[nH]1 85056,c1(C(N2CC(NC(C(C)O)=O)C(CO)CC2)=O)ccc2occc2c1 85057,Nc1ccc(Cl)c(C(=O)NCC2CC(NC(=O)C3=CCCOC3)C23CCC3)c1 85058,N1(C(c2scc(-c3n(CC(C)C)ncc3)c2)=O)CCCC(O)C1 85059,CC1(C)NC(=O)N(CCC(=O)NC2CCN(C(C3C=CCC3)=O)C2)C1=O 85060,S1(=O)(=O)c2cc(ccc2OC)N1.C1(CC#C)CN(C(=O)OC)CCO1 85061,c1(-c2nc(C)sc2)cccc(C(N2CC3(NC(C4COC4)=O)CC2C3)=O)c1 85062,N1(C(c2cc(C)sc2)=O)C2CCC1(CNC(C1CCCC3(CC3)C1)=O)CC2 85063,C1(C(N2C(CC(=O)NC)CC2)=O)CN(C(c2cc(O)ccc2C)=O)C(C)(C)C1 85064,C(N=c1cc(C)nc(N2CC(C3CC3)OC(C)C2)[nH]1)C1(CCOCC)CCC1 85065,c1(CN(C(CNC=O)=O)CCNC(=O)C(F)(F)c2nccs2)ccc(F)cc1F 85066,N1(C(C2(C(=O)NC)CC2)=O)CCN(C(c2nn(C)cc2C)=O)C2CCCCC2C1 85067,CCN=C1NCCN1.C1(CC2(C)CCC2)CCCCN1S(C)(=O)=O.C1(=O)CN1C 85068,C1(NC(CC(C)CF)=O)CCC2(CCN(C(c3cc[nH]c4nccc3-4)=O)CC2)C1 85069,C1(N(C(CSCC#C)=O)C)CN(C(c2c[nH]nc2C)=O)CC1F 85070,c1(NC(CC)(CCCl)c2nnnn2C(C)C)cc(Br)ccc1OC 85071,C1(CC)C(=O)NCCN1C(C1CCCN1C(=O)CCCc1cnn[nH]1)=O 85072,CCCC(C)C(=O)NC1CCCC1CNC(c1sc(=N)[nH]c1C1CC1)=O 85073,c1(NC(C2C3CN(Cc4n(C(C)C)ncc4)C2C3)=O)ncnc2c(F)cccc12 85074,C1(NC(c2c(Br)cn(C)n2)=O)CN(C(c2ocnc2C2CC2)=O)CCC1F 85075,C1(CNC(C(C)(C)c2cnsc2)=O)COCCN1C(=O)C=Cc1cccs1 85076,S(=O)(=O)(c1cccc2c1OCCO2)Nc1ccc2c(c1)N(C)CC2 85077,C=CC1OCCCC1CNCC1CN(C(=O)OC(C)(C)C)CCC1C 85078,C(C(C(=O)NCC1(O)CC(N(C)C)C1)NC(=O)C(O)C1CCCC1)OC(C)C 85079,C(C(C)C(=O)NC1CNC1=O)OCC.C(CCSCC)NC(C)=O 85080,Cn1ncc(C(N2CC=C(CNC(C3CC34CCOCC4)=O)CC2)=O)c1C#N 85081,C1(CCCNC(C2CCCN(C(C)(C)C)C2C)C)CCC(F)(F)CC1 85082,N1(C(=O)OCC)CC2CCC1(C(=O)N(C(C)CC1CC1)C)CC2 85083,Cc1c(O)nnc(N2CCN(c3ncc(Br)cn3)CC2)c1C 85084,N1(C(CN(C(=O)NCCCC)C)=O)CCN(Cc2c(CC=C)nn(C)c2)C2CC12 85085,c1(CC(N2CC=CC(NC(c3cc(C(C)C)sn3)=O)C2)=O)ccc(F)cc1F 85086,C1(C(N(CC#C)CC)=O)CC2CC1CN(C(C1CCC(=O)CC1)=O)C2 85087,c1(CC(N2CCC(CN(C(C(C)(C)OC(C)=O)=O)C)C2)=O)cc2ccccc2o1 85088,N1(C(C(C)=C2CCCC2)=O)CCCCC12CC(NC(=O)C(C)CC1CCC1)C2 85089,N1(C(COCCCC)=O)CC2CN(C(=O)C(c3ccccc3F)(C)F)CC2(C)C1 85090,c1(N2CCC(CCOC)(NC(=O)C(C)SC)CC2)ccc([N+](=O)[O-])cc1C#N 85091,N1(C(CC2(C=C)CCC2)=O)CCC2(NC(c3ccnc(C)c3)=O)CCCC12 85092,C1(NC(C(CSC)OC)=O)CC2(C1)CC2C(=O)NCC1COCCN1C 85093,C(=O)(C#CC1CCCCC1)NC1C(NC(=O)Cn2cnnn2)CCCC1 85094,N1(C(C(CNC(c2c(C)nsc2C)=O)OC)=O)CCCC(C2(C)CC2)C1 85095,c1(OC)ccc(C(CNCC23COC(CO)(C2)C3)OC(=O)OC(C)(C)C)cc1 85096,c1(OC)ncc(Br)c(N2CC3CC(NC(=O)CCCN4C(=O)CCC4=O)C3C2)n1 85097,Cc1ccnn1CC(=O)NCC(O)C(=O)NC(c1cn[nH]c1)C 85098,N1(C(CC(C(C)C)O)=O)CCN(C(c2ccn(C(C)(C)C)n2)=O)C(C)C1C 85099,CCC(C#N)C(=O)NCC(C)=CC(=O)NCC1CCN(CC)CC1 85100,c1(C(N2CC(C(C)NC(c3nsnc3O)=O)C2)=O)ccc(-c2cccs2)nc1O 85101,C1(CC(N2CCCC(NC(c3n[nH]cc3F)=O)C2)=O)NC(=O)CNC1=O 85102,C1(C(=O)NCCn2ncc(CC)c2)CN(C)CCN1C(C1CCCC(=O)N1)=O 85103,C1(CNC(CC=CC=C)=O)CCC2CN(C(c3ncc(C=O)s3)=O)CCC2C1 85104,C1(NC(C2C(CC)CCC2)=O)CCC(NC(c2cc(OC)c(Cl)s2)=O)CC1 85105,S(=O)(=O)(c1cccc(F)c1)NCCNC(c1cn(CCOC)nc1)=O 85106,N1(C(=O)CCCCCn2cc(C3CCCOC3)nn2)CCCC2(CCNC2)C1 85107,N1(C(c2cccc(OC)c2OC)=O)CCCCC12CN(C(c1ccoc1C)=O)C2 85108,C1(CNC(COC)=O)CN(C(C2COCCN2C)=O)CC(C)(C)C1 85109,Cn1ccc(C(=O)NC2CC(CNC(C3(N(C)C)CCC3)=O)C23CCC3)cc1=O 85110,N1(C(C)C(=O)NCC(F)(F)F)CCC2(CN(C(=O)C(C)(C)C3CCCO3)C2)C1 85111,C1(O)(CCNC(C(C)OCC#C)=O)CN(C(=O)Cn2nccn2)C1 85112,CCC(CC(=O)NC1(CC(=O)NCC2CC[Si](C)(C)C2)CC1)C(C)C 85113,Cc1cccc(Br)c1C(C(=O)NC1CC1(C)C)NC(C1CCC2(CC2)C1)=O 85114,Cc1ccc(C)n1CC(=O)NC1C=CC(C(=O)NCC2CCC(C)C2)C1 85115,c1(OC)cc(O)c(C(=O)NC(C)(CNC(=O)CC(F)F)CO)cc1Br 85116,C1(CC(=O)NC2CC3CCC(C2)N3C(C2CC=CCO2)=O)CCCC2(CCC2)O1 85117,c1(C(=O)NC2CCC(NC(CC=C=C)=O)C2)csc(C)c1CC 85118,CC(C)(C#N)CCCC(=O)NC1CCCC1NC(C12CCC(CC1)C2)=O 85119,C(=O)(C1COc2ccccc21)NC1CCN(C(c2n[nH]c(C)c2C)=O)CC1C 85120,C(=O)(CC1OC(=O)c2ccccc21)NC(CN(C(C=CCCC)=O)C)C 85121,C1(NC(C2(F)CCN(C(C(C)C3CCCO3)=O)CC2)=O)CC2CC1CC21CC1 85122,c1(C(=O)NC(CNC(C(CC)=CC)=O)CC)nccc(C)c1N 85123,N1(C(c2nn(C)c(OC(F)F)c2)=O)CC(NC(=O)CCCn2ccnc2)CC(O)C1 85124,C(C(=O)NCC1COC(CNc2ccc(C(=O)O)nc2)C1)(C(C)C)N(CC)CC 85125,c1(C(N2C(C)CC(NC(=O)C(C)(Cl)Cl)CC2)=O)ccc2n[nH]cc2n1 85126,O=C(CC(F)(F)F)N1CCC(N2CCN(C(c3c[nH]c(=O)cn3)=O)CC2)C1 85127,C(=O)(C1=NOC2(CCOC2)C1)NCC1(OC)CN(C(=O)C(F)n2cccn2)C1 85128,N1(C(C2C(C(C)=O)C2(C)C)=O)CCC(O)C(N(C(=O)CC2CCCN(C)C2)C)C1 85129,C1(NC(CSCCOC)=O)CN(C(=O)C=CSC)C(C)(COC)C1 85130,N1(C(C2C(C)OCC2)=O)CCC(C(C)(C)C)(CNC(=O)COC(F)(F)F)C1 85131,N1(C(c2ncccc2Cl)=O)CCC2(CCCC2Nc2nccc(CO)n2)CC1 85132,c1(C(=O)NC(CNC(C2(C(=O)OCC)CC2)=O)C)ccc(N)cc1C 85133,C1(CNC(C(C)(C)CO)=O)COCC2(CCN(C(=O)CC3=CCCCC3)C2)O1 85134,CC1CN(C(C2CCC(n3cc(-c4c[nH]nc4F)nn3)C2)=O)CC1CO 85135,C1(C)(CC)C=C(C(=O)NC2CC(NC(=O)C(C#N)Oc3ccccc3)C2)C1 85136,N1(C(c2occ(C)c2)=O)CC(C)CN(C(=O)OC(C)(C)C)c2ccccc21 85137,N1(C(Cn2cc(C(C)O)nn2)=O)CC2(C1)SCCC2NC(=O)C1=CCCCO1 85138,N1(C(c2ncnc(C)c2C)=O)CC(O)(C2(CNC(=O)CC(O)C(C)C)CC2)C1 85139,C1(NC(CC(=O)OC)=O)CC2CCC(C1)N2Cc1ccnc(Cl)c1F 85140,C12(NC(COCCCCC)=O)CC(C(=O)NCC3(F)CC3)(C1)C2 85141,C1(O)(CN(C(c2ncn(CC)c2)=O)C)CCN(C(c2ccoc2Cl)=O)C1 85142,C=C(C)CC(C(=O)NC1CCN(C(=O)CC2(COC)CC2)C(C)C1)OC 85143,C12(CNC(CNc3[nH]c(=N)sc3)=O)CNCCN1CCOC2 85144,C(=O)(CS(=O)(=O)CCO)NCC(CCNC(c1cc(CC)ncc1)=O)O 85145,N1(C(CN(CC)CC)=O)CCC2CCN(C(c3cc(F)c(C)cc3CN)=O)CC12 85146,C1(OC)(OC)CC2(CN(C(C(=O)NC3COC3)C(C)c3ccccc3)C2CO)C1 85147,N1(C(C2CC(OC)(OC)C2)=O)CCCCC1CCC(=O)NCC(C)CC1CC1 85148,Cn1ccn2ncc(C(=O)NCC3CC3CNC(=O)CC3CC4CCC3C4)c12 85149,N1(C(C2CCC(=O)N2)=O)CCC(CNC(c2cnc3n2CCC3)=O)C(F)(F)CC1 85150,C=C(C)CCCC(=O)NCC(CC(=O)N1CCCC1(CO)CO)OC 85151,N1(C(c2c(CC)scn2)=O)CCC2(CCCN(C(c3ncccn3)=O)C2)C1 85152,c1(NC(=O)C=CC(F)(F)F)cncc(CO)c1.C12CCC(C1)NC2=O 85153,c1(-n2cc(-c3ncn(C)c3)nn2)cccc(C(=O)NC2C(O)CC2O)c1 85154,C1(C(=O)NC2CC(C)(NC(C(CCSC)NC(C)=O)=O)C2)CCC(=O)N(C)C1 85155,CC1CCCC(NC(=O)OC(C)(C)C)C1.c12csc(n1)OC(=O)C1CC21 85156,C(c1ccncc1)=C(C)C(=O)NCC1CCCCC1NC(C1CCC2CC12)=O 85157,N1(C(CC2N(C(C=CC(=O)OCCCC)=O)CCOC2)=O)CCCC(O)(CC)C1 85158,n1(CC(N2C(CN(C(CC3CC(C)C3)=O)C)CCCC2)=O)nc2c(n1)CCCC2 85159,C1(NC(CC2C(C(=O)OCC)C2)=O)CCCC1NC(c1c[nH]nc1OC)=O 85160,c1(OC)ccc(-c2cn(C3CC(NC(C4(C5(C)CC5)CC4)=O)C3)nn2)c(F)c1 85161,C1(C(=O)NCC2(CNC(C(C(C)C)C3CCC3)=O)CCC2)Cc2nccn2C1 85162,c1(C(=O)NCCC(C)N(C(CC(CC)C)=O)C)cc[nH]c(=N)c1Cl 85163,c1(OC)nc(C)cc(=NCC2CCN(C(=O)CC(C(C)C)OCC)CC2C)[nH]1 85164,N1(C(c2c(C(C)C)ncnc2)=O)CCC(NC(=O)C(O)C(C)(C)C)C12CCCC2 85165,c1(OC)ccc(F)cc1CCC(N1CC(NC(=O)Cc2cncn2C)C(C)C1)=O 85166,C1(C2CC2)(C(=O)NCC(C)(C)OCCNC(C2C3CCCOC23)=O)CC=CC1 85167,C12(CCC(=O)N(CCC(C)NC(C3(CF)CC3)=O)C)CCC(CC1)C2 85168,C1(C(F)F)(CNC(C(C)OCCCC)=O)CCN(C(c2cncc(OC)n2)=O)C1 85169,N1(C(C2CCN(C)S2(=O)=O)=O)CC2(CCN(C(=O)C=CC3CCOC3)CC2)C1 85170,C(=O)(C(C)CC(F)(F)F)NC1CCCCN(C(C2CC(OC)C(OC)C2)=O)C1 85171,CCCC(CNC(C1CC1OC(C)=O)=O)C(=O)NCC(C)(CC)CO 85172,N1(C(C(=C(C)C2CC2)F)=O)CC(CCNC(C2(C)CCN(C)CC2)=O)OC(C)C1 85173,N1(C(CCNC(=O)OC)=O)CCC(C(=O)Nc2cc(Cl)ncn2)C(O)C1 85174,C1(NC(c2c(C)nn(CC)c2C)=O)CC2CC(C1)CN(C(=O)C(F)C(C)(C)O)C2 85175,C1(C(=O)NC2C=CC(C(=O)NC)C2)(CNC(CCCSCC)=O)CC2(CC2)C1 85176,C(=O)(C(Cl)=CCl)NC(C1CCOC1)CNC(CC1CN(C)C1)=O 85177,C1(NC(c2nc(CC)oc2)=O)CC(CNC(c2ncc(F)cn2)=O)C1(C)C 85178,C=C(C)CC(C(=O)NC1CN(C(=O)CSC)CC1CC)NC(C)=O 85179,Cc1ncc(C#N)cc1-n1ccnc1-c1nncc(CCCO)c1C 85180,C1(NC(c2ccc(C(C)O)cc2)=O)CN(C(c2ccc(C#N)nc2)=O)CC1C#N 85181,C1(NC(C(c2cc(C)sc2)(F)F)=O)CCN(C(=O)C(C)C#N)C(C)C1 85182,Cc1nc(C(=O)NCC(c2ccccc2)NC(C2(C)CCCO2)=O)cn1C(F)F 85183,c1(OC)c(C(=O)NC2CC(CNC(=O)CN3CC(C)C3)CC2O)ccnc1F 85184,C(=O)(C1=Cc2ccccc2C1)NC(C(=O)NC(C1CSC1)C)c1ccoc1 85185,C(=O)(C1=NNC(=O)C1)N1CCC(CC2C=NN(C)C2=O)C1.c12cn(nn1)CC2 85186,CCC(C(=O)NCC1(COC)CN(C(=O)CCCNC(=O)C(C)(C)C)C1)N(C)C 85187,Oc1cc(NC(C2CC2NC(CC2CCCC2)CO)=O)cc(F)c1 85188,N1(C(C(CC)(C)c2ccc(CC)cc2)=O)CCCN(C(=O)C(C)CC(C)C)CC1 85189,N1(C(C(C2CC2)OC)=O)CC2CCC1C(CNC(=O)CC1CCCC(C)C1)C2 85190,CC(C(=O)N(CCC(=O)NCCC1CC(=O)N(C)C1)CCCO)C(F)F 85191,N1(C(CC(C(C)OC)NC(C23CCC(CC2F)C3)=O)=O)CCC2(CC1)CSC2 85192,CC1CCn2cc(C(=O)NC3CC4CCC(C3)N4c3nccnc3F)nc2C1 85193,CC1CN(C(=O)C(Cn2cncn2)NC(=O)C(C)NC(N)=O)C(C)C1C 85194,C(C1CCN(C(=O)CC2CCCC23CC3)CC1)=CC(=O)NC1CCCC(CC)C1 85195,Cc1cc(C(N2CCCC(NC(=O)CCS(C)=O)C2)=O)ncc1Cl 85196,N1(C(C(CC)Oc2ccccc2C)=O)CCC2(CCC2NC(=O)CC#N)CC1 85197,Cc1cc(C2CC2)ccc1CNC1CN(C)CC1(C)C 85198,CCC(F)(F)CC(=O)N1CCC(C)(C)C1CC(=O)NCCN1CCOCC1 85199,C1(NC(C=C(CCC)C)=O)CC2(CCN(C(c3cncc(OC)n3)=O)C2)C1 85200,C#Cc1cccc(NC(C)C(N2CC(NC(C)=O)CC(c3cnn(C)c3)C2)=O)c1 85201,c1(C(=O)OC)cnc(Cl)cc1NCC1CC(C)CN1CCO 85202,c1(CC)noc(C(=O)NCC2(C(N3CCOC(CC(=O)OC(C)C)C3)=O)CC2)c1C 85203,c1(CCC(=O)NC(C(C)NC(CNC(CC)=O)=O)C)ccc(OCC(C)C)cc1 85204,N1(CCn2cc(COC)nn2)CCN(C(C2CN(C)C2)=O)CC1 85205,c1(C(N2CCC(CNC(C(N(C)C)C3CC3)=O)C2)=O)ccc(CO)cc1F 85206,C1(C(N2CC(c3nc(C)on3)C2)=O)CC(C)CN1C(=O)Cc1cnc(C)s1 85207,CC1OCCOC1CC1CCN(C(=O)Nc2cnn(N3CCOCC3=O)c2)CC1 85208,Cc1cc(C(=O)NC2CCN(C(=O)Cc3nc(Cl)cs3)C2)cc(F)c1 85209,C(=O)(C(CO)N(C)C)NCCC1CN(C(C(C)OC2CCOC2)=O)C1 85210,N1(C(CN2CCCC(CC)C2)=O)CC2C3CCC(C2C1)N(C(=O)NC1CC1Cl)C3 85211,C(=O)(C(C)(F)C(=O)N1CC(NC(c2sccc2-n2ccnn2)=O)C(O)C1)OCC 85212,N1(C(C(C2CCCC2)NC(C)=O)=O)CC2CC(N(C)C(C3(F)CCCCC3)=O)C1C2 85213,N1(C(CCCN(C(C)=O)C)=O)CC(CC(=O)OC(C)(C)C)CC12CCC2 85214,c1(OC)ccc(NC(=O)C(C(C)C)OC(c2cc(Cl)cs2)=O)cc1 85215,C123CCN(C1C2)C3=O.C(C)(C(=O)N(CCCNCO)C)OCCOCC.C(C)(=O)O 85216,C1(C)(C(=O)NCC(COC)O)CCN(C(c2cccnc2O)=O)C1 85217,C1(C)(CNC(CSCCOC)=O)CN(C(c2c[nH]c(=NC)o2)=O)C(C)(C)C1 85218,c1(CC)nccnc1C(=O)NC1(C(=O)NC2CCOCC2C)CCOCC1 85219,Cc1cncc(C(=O)NC(C)C(C)NC(c2scc(C)c2Br)=O)c1 85220,CC1CCC(C)(CNC2(c3nnnn3Cc3nnn(C)n3)COCCC2C)CC1 85221,Cc1ccc2oc(C(N3CCN(C(C4CC=CCO4)=O)C4CCCC34)=O)cc2c1 85222,CC1CCN(C(=O)Cc2ccc(Br)cc2)C(CNC(C2CC=CCC2)=O)C1 85223,S(=O)(=O)(CCC(=O)NCCNC(c1ccc(Cl)s1)=O)NCCNC(C)=O 85224,C(CCC(C)C(=O)N(CC(C)NC(=O)Cn1cnccc1=O)C)OC 85225,CC(CNC(=O)CCn1cncn1)CNC(C1CC(N2CCCC2)C1)=O 85226,Nc1cc(F)c(C(=O)NC(CNC(c2cnc(O)o2)=O)C2CCC2)cc1Cl 85227,c1(C(N2CC(NC(C=C(COC)C)=O)C(C3CC3)C2)=O)cc2c(cc1O)OCO2 85228,N1(C(CC(c2ccc(F)cc2)C)=O)C2CCC1(CNC(C1CCC(=O)N1)=O)CC2 85229,CC(C(=O)N=c1cc2ccccn2[nH]1)NC(c1ccc(=N)[nH]n1)=O 85230,C12(NC(=O)C=Cc3cnc[nH]3)COCCC1CN(C(=O)CC13CC(C1)C3)C2 85231,N1(C(CCC=C)=O)CCC(C)N(C(=O)CC2CCOC(C)(C)C2)CC1 85232,C1(NC(=O)CCN2CCCC2)CCN(C(=O)C2=NOCC2)CCC1CO 85233,c1(OC)ncc(C)c(C(=O)NC(C)CNC(c2nc(C3CC3)cs2)=O)c1Cl 85234,c1(OCC(=O)NC2CCCN(C(CN)=O)C2)cc(Cl)ccc1Cl 85235,C#CCC(C)C(=O)N1CCCC1C(C)NC(c1ccc(-c2cscn2)nc1)=O 85236,c1(NC(=O)NC(CCCCC)c2ccccc2)cc(F)ccc1NC(C)=O 85237,CCC(C)C(C)C(=O)NCc1ccccc1CNC(=O)Cn1cnnc1O 85238,N1(C(=O)CC2CSC2)CCN(C(c2cnccn2)=O)C(CC(F)F)C1 85239,c1(CNC(CC2N(C(C3C(CC)C3)=O)CC2)=O)nc(C)ns1 85240,C1(NC(CCc2cncc(C)c2)=O)CN(C(=O)C(C)c2cccs2)CC(F)(F)C1 85241,c1(C(N)=O)cc(C(=O)NC2(CNC(=O)C(c3ccc(F)cc3)F)CC2)cc(F)c1 85242,CC1CC(NC(C23CC(CF)(CO2)C3)=O)CCN1C(c1cncc(Cl)c1)=O 85243,C(=O)(C(C)(F)C(=O)OC)N(CC(CNC(c1c(CC)ccs1)=O)C)C 85244,C(=O)(CC1=NNC(=O)C1)N(C1CCN(C(c2c(C)nsc2C)=O)CC1C)C 85245,c1(C(=O)OC)sc(C(=O)N(C2CN(C(C3CCC4CC34)=O)C2)C)cc1C 85246,C(=O)(C1Cc2ccccc21)NCC1(O)CCN(C(C2C(C)OCC2)=O)CC1 85247,c1(C(C)C)cc(C(=O)NC2CN(C(=O)CC3CCCCO3)CC2O)c(C(C)C)[nH]1 85248,C1(C(N(C(CC)CC)CC(C)C)=O)COCCN(C(c2ccc(O)nc2C)=O)C1 85249,CC(C#N)CCC(=O)NCC1CCC(NC(=O)Cc2cccc(Cl)c2Cl)CC1 85250,N1(CC)CCOC(C(N2CC(O)CC2C(=O)NCCc2nccs2)=O)C1 85251,C1(CC(=O)N(C(C)CC(=O)NCCCCOC(C)C)C)CCCNC1=O 85252,n1(CCC(COC)O)cnc2c(N(CCF)Cc3cccc(Cl)c3Cl)ncnc12 85253,CC1(C)NC(=O)CCC1NC(=O)CC(C(F)(F)F)NC(c1ccncc1N)=O 85254,N1(C(c2cc(F)ccc2F)=O)CCC2CCCC(C1)N2c1ncc(F)cn1 85255,C1(C)(C(=O)NC(C(C)NC(C2CCN(C)CC2)=O)C)Cc2ccccc2C1 85256,N1(S(CC(C)C)(=O)=O)CC2(CC(CC(=O)NC(c3ccccc3Cl)C)C2)C1 85257,C1(C#N)(C(=O)NCCC(C)NC(c2n[nH]cc2C2CC2)=O)CC2(CCC2)C1 85258,c1(C(=O)NCC2CN(C(Cn3c(=O)ccc(C)n3)=O)C2)nc2ccccn2c1F 85259,CC(C)C(C(=O)NC(C)C(=O)NO)C(C)NC(=O)CCc1nc(=N)[nH][nH]1 85260,C(C(C(=O)NC1CC1)N1CCC(O)(C(N)=O)C1)(C1CCCC1)OCC 85261,c1(C(=O)NC2(CC(=O)COC)CC2)cccnc1.C1(COC)(CN)CC1C=O 85262,CCCCCC(C)CC(=O)N(CC(CC)NC(c1ncc2[nH]ncc2n1)=O)C 85263,c1(OC)c(Cl)ccc(C(N2CC(NC(=O)CS(C)(=O)=O)CC3(CC3)C2)=O)c1N 85264,CC1(C(N2CCC(CCCO)CC2)=O)CCCN1C(c1cc(=O)cco1)=O 85265,C(=O)(C(F)(F)C(O)C(C)C)N1CC2C(Nc3cc(OCC)nc(C)n3)C2C1 85266,C1(CNC(C(C)=CC)=O)CC2(CO1)CN(C(c1ccc(OC)c(Cl)c1OC)=O)C2 85267,c1(C(=O)Nc2ccc(NC(C(CC)OC)=O)cc2C)cc(C)cc(Br)c1F 85268,c1(C(=O)NCC(C(C)C)NC(CC(CC)C2CCC2)=O)ccc2ncncc2c1 85269,c1(CC)nc2n(n1)CCCC2NC(=O)C(n1cc(C(C)C(OC)OC)nn1)C 85270,C1(C(N2CCC(C)(CNC(c3n(C)ncc3)=O)C2)=O)CCC(S(N)(=O)=O)CC1 85271,CCC(C)(C)C(C)CC(=O)NC1CCN(C(c2ccc(F)c(Cl)c2)=O)CC(O)C1 85272,C1(O)(CC)CCC(NC(=O)C(C)CN(C)C(c2nonc2C)=O)CC1 85273,C1(NC(c2c(COC)nn[nH]2)=O)CC2CN(C(C3CCSCC3)=O)CC2C1 85274,C(CC(C)N=c1[nH]c2c(c(=NCCN3CCCCC3=O)[nH]1)CCCC2)OC 85275,N1(C(C(CC)=CCCC)=O)CC2CC(C)N(C(=O)CC=Cc3ccccc3)C2C1 85276,c1(OC)cccc(C(N2CCN(C(=O)C(C)C(C)(F)F)CC2CC(F)F)=O)c1C 85277,C1(C(=O)NC(C2CCCC2)CNC(c2nc(Cl)cs2)=O)CCNC1=O 85278,C1(NC(c2c(C(C)C)n[nH]c2)=O)CC2CC1N(C(=O)CC(C)F)C2 85279,C(C(C)(C)C(=O)NCC(C)CN(C)C(C1CCCC(=O)C1)=O)NC(C)=O 85280,C(C(N=c1nc(CC)[nH]s1)C(C)C)CNC(C(C)(C)NC(=O)NCC=C)=O 85281,c1(C(=O)OC)ccc(CC(=O)NCC(F)CNC(c2nn(C)cc2Cl)=O)c(Cl)c1 85282,C1(NC(C(c2c(C)cccc2)C)=O)CC2CC1CN(C(c1ccsc1)=O)C2 85283,c1(C(N2CCC(CCNC(c3cc(CC)sn3)=O)CC2)=O)cn2ccsc2n1 85284,C1(NC(c2ccc(C)n2C)=O)CCCCN(C(=O)Cc2nnn(C(C)(C)C)n2)C1 85285,C(=O)(C1=CC(O)C(NC(=O)CCc2cncnc2)C1)N(C)CCO 85286,C1(=CC(N2CC(O)(CNC(c3n(CC)ccn3)=O)C2)=O)C2CC3CC(C2)CC1C3 85287,c1(C(=O)NC(CC)CN(C)C(C2(F)CC2C)=O)ccc(Br)c(N)c1 85288,C1(C(N(CCC)CCNC(=O)C(C)OC2CCOC2)=O)CC2CC1CC2O 85289,N1(C(C2CC(C)=C(C)CC2)=O)CCC=C(C(=O)N2CCOCC(C)(O)C2)C1 85290,N1(C(CCCSC)=O)CCC2(CCCCC2NC(=O)CCCCCO)C1 85291,CC(C)CC(C(=O)N1CC(S(C)=O)C1)ONC(C1(C#N)CCCCC1)=O 85292,N1(c2snc(COC)n2)CCCCC(CNC(=O)CCN2CCOCC2)C1 85293,N1(C(C2(CC(C)C)CC2)=O)CCC2C(CCCN2C(c2cnn(CCF)c2)=O)C1 85294,C1(CNC(C=CCCC=C(C)C)=O)CN(C(C2CC3C=CC2C3)=O)CC12CCC2 85295,C(c1ccc[nH]1)=CC(=O)NC(CNC(CCC)=O)CC 85296,c1(Cc2nc(-c3c(C)n(-c4ccccc4F)nc3)on2)ccc(C(C)C)c(Cl)c1 85297,N1(C(CC2C(C)(C)C2)=O)CCC(CN2CCC(C(F)(F)F)(C(F)(F)F)C2)C(O)C1 85298,N1(C(CCC(=O)OC)=O)CCN(C(c2cnnc(O)c2)=O)C2CC12 85299,O=C(C1=CCCSC1)NC1(C(N2CCN(CCO)CC2)=O)CCSC1 85300,c1(NC(C)CCOC)ccc(S(=O)(=O)NCC(c2ccco2)O)cc1Br 85301,CC(CC(=O)N1CCC(CN(C(=O)C=Cc2ncc[nH]2)C)C1)P(C)(C)=O 85302,c1(OC)c(C(N2CC3CC2CCC3NC(c2ocnc2C)=O)=O)cc(Cl)cc1C 85303,N1(C(C2CC(SC)C2)=O)CCn2c(CNC(=O)C(C)=C3CC3)nnc2C1 85304,c1(C(N2CCC(C(C)NC(C=CCOC)=O)C2)=O)ccc([N+](=O)[O-])cc1 85305,c1(N2CC=CC(NC(C(C)CC(C)(C)C)=O)C2)ncc([N+](=O)[O-])cc1F 85306,C1(CNC(C(Cn2ccc(C)n2)C)=O)CC2(CCOCC2)CN1C(=O)C=C(Cl)Cl 85307,c1(C(C)C)c(N(CCO)C=O)cncc1F.C1(C)(NC(C)(C)C)CCS(=O)(=O)C1 85308,C1(CC(=O)NCC(N(C)C)C2CC2)CCN(C(C2(Cl)CC2(F)F)=O)C1 85309,C(=O)(C1CCCc2nc[nH]c21)NCCCN(C(C1CC(C)C1)=O)CCO 85310,c1(C(C)OC(C2(C)CCC2)=O)nc2ccccc2n1Cc1ccccc1CON 85311,c1(CC)noc(C)c1C(=O)NCC(CC(=O)N1CCC(O)(CN(C)C)C1)OC 85312,C(=O)(C(Cc1cnc[nH]1)NC(=O)C(C1CCCCC1)=O)NCC(C)CC1CC1 85313,C1(NC(CC(OCC)OCC)=O)CC12CCN(C(c1sc(C)cc1C)=O)C2 85314,c1(C(N2CC(C)(CC(=O)NCc3ccc(C)cc3F)C2)=O)cn2nc(C)sc2n1 85315,CCC(C)C(C(=O)N1CC(C)(C)CC1CC(=O)NC1CC(CCF)C1)N(C)C 85316,C1(NC(C(CC)CC(F)F)=O)CN(C(=O)Cn2nccn2)C2CCCCC12 85317,Cc1c(C(N2CCC(N(C(=O)CC3CC=CC3)C)C2)=O)cc(N)cc1O 85318,C1(CC=C)(NC(=O)CSC(C)(C)C)CCCN(C(c2cc(Br)c[nH]2)=O)C1 85319,c1(C(N2C(C3CCCN(C(=O)Cc4cn[nH]c4)C3)CCC2)=O)cc(O)cc(Cl)c1 85320,C1(NC(c2cnc[nH]2)=O)CN(C(=O)Cc2cnccc2Cl)CC12CCC2 85321,C1(NC(C(C)(C)C(F)(F)F)=O)CN(C(C2CCC(C)(C)O2)=O)CC12CCOCC2 85322,Cc1cncc(CC(=O)NCC=CC(=O)NC(C)Cn2cncn2)c1 85323,C(=O)(C(F)CC(C)C)NCC(C)(C(C)C)NC(C1CCN(C(C)=O)CC1)=O 85324,N1CCCCCC1NC(=O)N.C1(N(c2ccc(CC)o2)C)CCN(C2CC2)CC1 85325,C(C)(C)(CC(=O)N1CCCCC1C(C)NC(=O)C=Cc1scnc1C)OC 85326,C1(C2CCCN(C(C3C4CCCOC34)=O)C2)(NC(c2cn(C(C)C)nn2)=O)CC1 85327,c1(C(N2CC3CN(C(Cc4nnc(C)o4)=O)CC32)=O)cc2cc[nH]c2cc1Cl 85328,CC(C)(O)C(C)(C)NC(C1CCC(NC(=O)CCc2ccncn2)CC1)=O 85329,C(CCC(=O)NCCCC1CCCN1C(=O)C(CC)OCC)N(CCC)CC 85330,c1(NCC=CCNC(C(c2cccc(Cl)c2)CC)=O)cc(C)ccc1[N+](=O)[O-] 85331,c1(N2CC(C)(C)OC(CNC(=O)C=Cc3cn[nH]c3)C2)ncc([N+](=O)[O-])c(=N)[nH]1 85332,c1(CNC(C(C2CN(C(C(n3c(C)ccn3)C)=O)C2)O)=O)ccc(O)nn1 85333,C1(COC)(NC(=O)Cc2nnc(S)n2C)CCN(C(c2c(O)noc2C)=O)CC1 85334,Cn1nnnc1SCCC(=O)NCC1CC(F)(CNC(=O)Cc2cnoc2)C1 85335,C1(C(N2CCC(CC=C)(NC(c3cc(C)sc3C)=O)C2)=O)CN2CCC1CC2 85336,c1(N2CCC(CC=C)C2)nc(=NCCC(C)(C)OC)[nH]c2c1SCC2 85337,C1(C(=O)NCC(COC)(C)CO)CCCN(C(C2CC3CCCC3C2)=O)CC1 85338,C=CCC(C)(CC)C(=O)N1CCN(C(c2cc(C(F)(F)F)cs2)=O)C(C2CC2)C1 85339,Cc1ccc([N+](=O)[O-])c(C(=O)NC2CC2NC(=O)COc2ccsc2Cl)c1 85340,N1(C(c2cc(CCC)on2)=O)CCC(NC(=O)CC2CC2(C)C)C(O)C1 85341,Cc1ncc2cc(C(N3CC4C(NC(=O)C(F)(F)C5CC5)C4C3)=O)ccn12 85342,CN1CC(C(=O)NCC(N)=O)C1.C12(CC1)CC(=O)NC2 85343,c1(C(=O)NC23C(CN(C(CC4ON=C(C)C4)=O)C2)CC3)csc2c1CCC(C)C2 85344,N1(C(C(=O)NC2CC(NC(c3cc(C)no3)=O)C2)C)CCCCCC1 85345,C12(C(=O)NCc3c(C)nn(C)c3)CCCC1CN(C(C1CCCCS1)=O)C2 85346,O=Cc1ccnc(NC(=O)N(C2CCS(=O)(=O)C2)C2CC2)c1 85347,CCC(C(=O)NCC(C)CC(=O)N1CCC1C)C(C)(C)CC 85348,c1(CNCC)cncc(COC(=O)CC2CCCN(C(=O)OC(C)(C)C)C2)n1 85349,c1(C(N(CC(CC)NC(C2(C)CCC(C)CC2)=O)C)=O)cc2cc(C)ccc2o1 85350,CCCCCCC(F)C(=O)N(C1CCN(C(c2cccc(Cl)c2N)=O)C1)C 85351,C1(C(N(C2CCN(C(=O)Cn3cc(Cl)c(C)n3)CC2)CC)=O)CC(C2CC2)C1 85352,O=C(C1=C(Cl)CCC1)NCCC1CCN(C(=O)COc2ccccc2)CC1 85353,CN1CCN(C(c2ncc(F)cc2N)=O)C(CNC(=O)CCCNC(N)=O)C1 85354,C(=O)(C(C(=O)NC1CCCC(CNC(=O)CSC(C)(C)C)C1)C1CC1)OCC 85355,C=CC(CC)CC(=O)N1CCCC(NC(=O)CCNC(=O)C=CCl)C1 85356,C1(C(C)C)CN(C(c2cncc(F)c2)=O)CCC1NC(=O)C=CC1CC1 85357,c1(C(=O)NC(CC)CN(C(=O)C(C)C2CC2)C)cccc(CCO)c1 85358,C1(NC(c2nc(C(C)NC(COCCC(C)C)=O)oc2)=O)CC2CC1CC21CC1 85359,CCCC(CCCNC(C1OCCC1(C)C)=O)NC(=O)CNC(=O)C1CC1 85360,CC1CN(C(C2(O)CC(F)(F)C2)=O)CC1NC(C1(F)CC1)=O 85361,CCC(CCC(=O)NC(C)CC1CCN(C(c2cccc(SC)c2)=O)CC1)OC 85362,C12(C(N(OC)C(C)C)=O)CCC(CC1)N(C(=O)Cc1ccoc1C)C2 85363,CON=C(C(=O)NCCC(C)N(C)C(c1coc(S(N)(=O)=O)c1)=O)c1ccco1 85364,C1(NC(CSC)=O)CC2CCC1N2C(=O)Cc1cccc(Cl)c1 85365,C1(C(=O)NC(C)CCNC(=O)C=C2CC2)CC2(CCCCO2)C1 85366,C(=O)(CC(C(F)F)NC(C1C2CCC(C2)C1C)=O)NCCc1ccc(C)s1 85367,c1(C(N(CC(CC)NC(=O)Cn2ncccc2=O)C)=O)cc(C)c(C(N)=O)cn1 85368,c12nc(no1)COC2.c1(C(=O)OC(=O)C(c2ccccc2)O)csc(C2CC2)c1 85369,N1(C(CN(S(C)(=O)=O)C)=O)CC2CCC1(CNC(=O)CC(CN(C)C)C(F)F)CC2 85370,N1(C(C2N(C(C=C(CCC)CCC)=O)CCC2)=O)CC(O)C(O)C1C(=O)OC 85371,O=C(C1CCCc2scnc21)N1CCCCC2(CCN(C(=O)COCCCF)C2)C1 85372,c1(C(=O)NC(C(C(C)C)NC(c2cnc(S)[nH]2)=O)C)ccccc1N=S(C)(C)=O 85373,C1(C(=O)NC(Cc2ccco2)C(=O)N2CCC(CCO)C2)CC2(CCC2)C1 85374,c1(C(N2CC(NC(=O)CCC(=O)N3CCOCC3)C2)=O)ccc2c(c1)CC2 85375,c1(C(N2CCC(NC(CCc3cc(C)[nH]n3)=O)C2C(C)C)=O)c(O)cccc1F 85376,c1(CNC(N(C(C)C)CCO)=O)nocc1CS(C)(=O)=O 85377,N1(C(C(C)(N(C(=O)CC2C=CCCC2)C)C2CC2)=O)CCCCCCCC1 85378,c1(C(C(=O)NCC(CNC(C2(CC(C)C)CCC2)=O)C)(C)C)cc(Cl)cc(Cl)c1 85379,c1(CC)ccccc1C(=O)NC1CC(C)N(C(=O)CC2CN(C)C2)C1 85380,O=C1CCC(C(=O)NC(CNC(c2cccn3ccnc23)=O)CO)=NN1 85381,c1(C(=O)NCC2(OC)CN(C(=O)CSCCC#N)C2)ccccc1SC(F)(F)F 85382,C(CCC)(C(=O)N1CCC(C(=O)NCCOCCOC)C1)=CC 85383,C1(CNC(C2CC(OCC)C2)=O)CCCCC1C(N1CC(O)C1)=O.C=O.C1CC1 85384,CC(C(=O)N1CCC(NC(c2csc(-c3ncc[nH]3)n2)=O)C1)C(F)(F)F 85385,C(=O)(CCCCC(=O)OC)N1CCC(N(C(CC(CCC)O)=O)CC)CC1 85386,c1(C(=O)NCCNC(C2C(C)OC(=O)N2)=O)nnc2ccccc2n1 85387,C(C)(C(=O)N(CCCNC(c1nc(Cl)c(Cl)s1)=O)C)(C(C)C)OC 85388,C1(NC(N(C(CC)C(C)O)C)=O)CCOC(CNC)C1 85389,c1(C(N2CCC(C(C)(C)NC(c3cn(C)nc3O)=O)C2)=O)c[nH]c2cccnc12 85390,c1(C(=O)NC2C(NC(CCc3ccc(C)cc3)=O)C2)ccc(S(N)(=O)=O)o1 85391,c1(C(=O)NCC2CCN(C(c3c(C)nncc3)=O)C2)cnc2ccccn12 85392,CC(=O)CCN=C(NCC1CC2(C1)CC(C)(C)C2)NCC1CCC2CC1C2(C)C 85393,c1(N(C2CCN(C(C3(C)C=CCC3)=O)CC2)C)ncc2ncnc-2[nH]1 85394,c1(C(=O)NCCC2CSCCN2C(C2CC23CC3)=O)nc(O)[nH]c(=O)n1 85395,C(=O)(CCC(=O)NCC1CC(O)CN1C(=O)CCc1cnc(C)s1)NCCC 85396,c1(OCCCC)ccc(C(=O)NCC2CCN(C(C3CCCOC3)=O)C2)c(Cl)c1 85397,CC(CC(C)(F)F)C(=O)NCCCCNC(=O)CCC(=O)c1ccccn1 85398,c1(OC)ccc(CC(=O)NCCC(C)NC(=O)C(C)(CO)OC)c(OC)c1 85399,CN1CCCC2CN(C(c3ccnc(C(F)(F)F)c3)C(=O)NC3CCC3)CCC12 85400,C1(CNC(C2C(C)(C)C2)=O)CCCCN1C(=O)Cc1cnsc1 85401,N1(C(c2c(OC(F)F)cc(C)s2)=O)CC2CCC(C1)N2C(=O)CCc1cnn[nH]1 85402,CC1=C(C(=O)N2CC(O)(CCNC(C3CC4CCC(C3)C4)=O)C2)SCCO1 85403,C(=O)(C1=CCC2CCC1N2C(c1cccs1)=O)Nc1c(C)n(C2CC2)nc1 85404,C1(C(=O)NCC(CCOC)NC(COCCCC)=O)CC2CCC(C1)O2 85405,c1(N(CCCCNC(C(CC)NC(c2cc(C)on2)=O)=O)C)ccc(F)cc1 85406,Cc1cc([N+](=O)[O-])cnc1C(=O)NCCN(C(c1cc(CO)c(C)o1)=O)C(C)C 85407,N1(C(C2CC(NC(Cc3n(C)cnc3)=O)C2)=O)CCC2(CCCOC2)C1 85408,C1(C2CCN(C(C3CC3C)=O)CC2)(NC(c2cc(C)cc(Br)c2N)=O)CC1 85409,N1(C(CCN(C(c2n(C=C)nnc2)=O)C)=O)CCN(C)C(C)C1C 85410,CC1CC(NC(c2cc(C(N)=O)co2)=O)CN1C(c1snc(O)c1Cl)=O 85411,c1(NC)ccnc(C(=O)N(CCC(=O)NCc2cc(C)on2)C)c1 85412,CCC(CC(F)(F)F)C(=O)NCC(C)(CC)NC(C1CC2C=CC1C2)=O 85413,Cc1ccc2c(c1)CC(C13CC(C(=O)OCC(C)(C)C)C(C1)CO3)S2 85414,c1(CC(=O)N(C(C)CN(C)C(=O)C2CC2)C)ccc(NC(=O)NC2CC2)cc1 85415,C(=O)(C(CC1CCC1)NC(=O)CSCCOC)NCC(C)OCC#C 85416,CCC(F)(F)C(=O)N1CCC(N(C(=O)CN2CC=CC2)CCOC)CC1 85417,c1(C(=O)NC2CC(C)(CNC(CCCOCC)=O)C2)ccc2[nH]cc(C#N)c2c1 85418,CCC(C)C(C)(O)CNC(=O)C(C1(O)CCC1)NC(=O)CCCn1cccc1 85419,c1(N2CCN(C(C)C(N)=O)CC2)nccc(=NCCc2cccc(Cl)c2)[nH]1 85420,c1(-c2cc(OCC)cc(F)c2)cc(C(=O)NCCS(=O)(=O)NC)c2cn[nH]c2c1 85421,c1(C(N2CC3C(NC(=O)Cc4cc[nH]n4)(C3)C2)=O)ccc(O)cc1O 85422,C1(CC(N2CC(C)(NC(C3C(C)OCCO3)=O)C2)=O)COC2(CCC2)CO1 85423,CC1=C(C(=O)NCc2cc(C(=O)N(C34CC(C3)C4)C)on2)CCO1 85424,C1(C(=O)NC2C3CN(C(C(CCC)C#N)=O)C2C3)CCc2nnnn2C1 85425,c1(C(N(CCOCCNC(C2(NC(C)=O)CC2)=O)C)=O)cc(C)nc(C)c1 85426,C(CC(C)(C)C(=O)N1CCC(C)C(CNC(=O)CC2CSC2)C1)OC 85427,c1(OC)cccc(C(C)CC(=O)NC(C)CCNC(=O)CCc2ccon2)c1 85428,S(=O)(=O)(c1cccc(=NCc2cc(C(N)=O)no2)[nH]1)NCc1c(COC)cccc1 85429,CC1(C)CC(C(=O)NCCN2CCC3CC23)CN1C(=O)C(F)C(F)(F)F 85430,C#CCCC(C(=O)NCC(=O)NCCOC)NC(=O)C(C)N(C)C 85431,c1(C(=O)NCC(=O)NC(C)C(=O)NCC(F)F)cn(C2CC2)cn1 85432,C1(CC(=O)NC2CCN(C(c3ccc(CCC=C)cc3)=O)C2)CC(F)(F)C1(F)F 85433,C1(CCC)CN(C(C2(Cl)CC2(C)C)=O)CCN1C(=O)C=CBr 85434,N1(C(CN(C(=O)C(=O)Nc2ccccc2)C2CC2)=O)CC2CCC(CO)(C2)C1 85435,N1(C(c2c(CNC(C(C)(C)n3cnnn3)=O)cco2)=O)CC2C=CC2C1 85436,C(=O)(C(C)S(=O)(=O)C1CCOCC1)NC1CCC(NC(C(C)NC(C)=O)=O)CC1 85437,c1(C(C2CCC2)NC(=O)NC(C)CC2CCC2)ccc(F)cc1F 85438,N1(C(COC)=O)CCCC(NC(=O)CC2CC2)CC1 85439,c1(NC(C2=C(C)OCC2)=O)ccc(C2=CCN(C(C3CCC(C)O3)=O)CC2)cc1 85440,C(=O)(C(CCOC)NC(=O)C=CC(=O)NC1CC1)N(CCCCC)C(C)C 85441,N1(CC(=O)N(CCCCN(C(=O)CCc2csnn2)C)C)CCC(F)(F)C1 85442,CC1CCCN(C(c2cccnc2)=O)C1CNC(C12CC3CC1C2C3)=O 85443,CC1OC2(CNC(C3CCCCCCC3)=O)CC1(NC(=O)C=Cc1cocn1)C2 85444,CCC(O)CN(C(=O)C(F)OC(F)(F)F)CC1CC1 85445,c1(CC)[nH]c(=N)sc1C(N1CC(NC(=O)Cc2ccnc(F)c2)C(C)C1)=O 85446,Cc1cc(C(=O)NC(C2CCCCN2C(=O)CCSc2nnnn2C)C)ccn1 85447,C(CC(C)C(=O)N1CCCC(C(=O)NCCN2CCOCC2=O)C1)=CC 85448,Cc1nc(-c2ccccc2)c(CN2CC(F)CC2C(N2CCCCC2)=O)s1 85449,Cc1ccc(C(=O)NC(CNC(=O)C(Cc2ccccc2)C2CC2)CO)c(Cl)c1 85450,C1(C)(CNC(c2ccn(C)n2)=O)CN(C(=O)CCOC2CC2)CCO1 85451,c1(NC(C2CC(OC)CN2C(=O)Cc2ccc(O)cn2)=O)ccc(O)cc1Br 85452,N12CC=C(CCNC1=O)CC2.C1(SC(C)(C)C)CCOC12CCCC2 85453,C#CC1(NC(C2(NC(=O)CN(C)C(C)=O)CCCC2)=O)CCCCCC1 85454,c1(C(=O)NC2CCN(C(CCC)=O)CC2C)c(Cl)nc2cc(Cl)ccn12 85455,c1(C(C)NC(C(C)SC(F)(F)F)=O)ccc(CNC(C2(C)CCOC2)=O)cc1 85456,c1(-n2c(CN3CCCC3=O)nc(CCCCC)n2)ccc2nccnc2c1 85457,CC1(C)CC(NC(=O)C(CN=[N+]=[N-])NC(c2nc[nH]n2)=O)C(=O)O1 85458,Cn1ncnc1COCC(=O)NC1CCC1CNC(=O)CC1(C)CCOC1 85459,c1(CC(=O)N(C2CCN(C(c3coc(O)n3)=O)C2)C)cn(CCO)nn1 85460,C(=O)(CCCCCF)NCC1C(NC(c2c(CC)ncs2)=O)C1 85461,C1(CNC(C=C(C)C2CC2)=O)CC12CCN(C(=O)C=CCN1CCOCC1)CC2 85462,C(=O)(C1(C)OCCc2ccccc21)N1CC(C(C)NC(=O)C(C(C)(C)C)SC)C1 85463,Cn1nnc2c1CCN(C(=O)C(C1(C)CC1)NC(C1CCCOC1)=O)C2 85464,C1(C)(C(C)C)C(=O)N1.n1(CCC)c2nnc1SC2.c1(CO)ccc(Cl)cc1.SC 85465,n1(CC)ccc(CC(=O)NC2CCN(C(=O)C(C)(C)c3cscc3Cl)C2)n1 85466,CC1CC(N(C(=O)C(C2CC2)N(C)C(c2ccoc2Cl)=O)C)CC(C)C1 85467,N1(C(C(C)S(N)(=O)=O)=O)CCN(C(C2Cc3ccccc3C2)=O)C2CCCC12 85468,Cc1c(C(=O)N(CCCCN(C(=O)CC2(C)CCCCC2)C)C)cnn1CCO 85469,C1(NC(N)=O)CCN(C(=O)C(N)Cc2ccoc2)C1 85470,C(=O)(CCCC(CC)CC)N1CC(CC(=O)NCCC(CCC)C2CC2)C(C)C1 85471,C1(C(=O)NCC(C)(C)C2CCC2)CSCCN1C(=O)C=CCO 85472,N1(C(C=CC=CC)=O)CCC(C)C(CNC(c2cc(C3CCOCC3)[nH]n2)=O)C1 85473,c1(CCCNC(=O)NCCNc2cc(C)ncn2)ccc(F)c(F)c1 85474,N1(C(C(C#C)(C)C)=O)CCCN(C(C2CCC(=O)N(C(C)C)C2)=O)CC1 85475,c1(C(N2CC(CN(C)C(c3ncc[nH]3)=O)C2)=O)cn(C)c2ccccc12 85476,C(=O)(CN=S(C)(C)=O)NCC(CNC(C(C(C)O)N(C)C)=O)CO 85477,C(=O)(C(CC(C)C)C(C)C)N1CC(C(C(=O)N(CCCCCC=C)C)O)C1 85478,N1(C(C(=O)NCCOC)CCC2CC=CCC2)CC2CC1CN2C1CC1 85479,C12(C(=O)NC3CCN(C(C4CCSCC4)=O)C3)CC(CO)(C1)OC21COC1 85480,N1(C(CCCC#CC)=O)CC2(CNC(C3CCCSC3)=O)CC1CCO2 85481,c1(CC(C)NC(=O)C(N2CCCC2)=O)ccncc1Cl 85482,Cc1nc(C(=O)NCC(C)(C2CC2)NC(c2ccn(-c3ccncc3)n2)=O)co1 85483,CC1(C)CCCCC1=CC(N1CC2CC1C2CNC(c1ccc(Cl)o1)=O)=O 85484,CC(CC(=O)NC1CCC(CNC(C2CCOCC2)=O)C1)C(C)(C)C 85485,c1(-c2cn(CC(C3CC3)NC(CCCC(C)C)=O)nn2)ccc2cnccc2c1 85486,c1(CNC(c2nccn2-c2ccccc2)C)ccc(C(=O)O)o1 85487,c1(C(=O)NCCCNC(C2CC(CC)C2)=O)cc([N+](=O)[O-])cnc1N 85488,Cn1nc(Cl)c(NC(N2CCC(CSc3ccccc3)CC2)=O)c1C(F)(F)F 85489,CC1CC(NC(=O)CN2CCN(C)CC2)CN(C(c2ccc(Cl)nc2N)=O)C1 85490,CC1(C)CC(NC(C2CC(C)N2C(C2(Cl)CC2)=O)=O)C1 85491,C(c1scnc1C)=CC(N1C(C(CNC(Cc2c(C)nc[nH]2)=O)(C)C)CCC1)=O 85492,C1(CC)C(NC(c2ncncc2N)=O)CCCN1C(=O)CN(C)C(=O)C1CC1 85493,N1(C(C(COC)NC(C)=O)=O)C2CCC1C(NC(c1ncoc1C1CCC1)=O)C2 85494,C(C(CC1CC1)C(=O)NCc1cccnc1F)NC(c1nc(CC)oc1)=O 85495,Cc1nc(C(=O)NC(C)CN(C)C(c2ccc3snnc3c2)=O)ccc1[N+](=O)[O-] 85496,N1(C(=O)NC(C)Cc2ccccc2OC(F)(F)F)CC2(CO)CCCC1C2 85497,N1(C(C(C)Oc2cccnc2)=O)CC(C(=O)NCC(=O)C2CC2)CC2OCCC12 85498,C=CCC(C)C(=O)NCC(C(C)C)NC(c1cc(C(C)=O)c(C)o1)=O 85499,S(=O)(=O)(c1ccc(C(=O)NCC(CO)NC(c2ccc3cnnn3c2)=O)o1)NC 85500,Cc1scc(CCC(O)CN(C)C)c1C.c1(C(=O)O)ccccc1 85501,c1(C(N(C2CCN(C(C(CC)F)=O)C2)C)=O)cc(C(F)F)ccn1 85502,C(C(=O)NNc1ncnc2c1CCC2)c1c(C)cc(C2CC2)cc1 85503,CC1(CNC(c2ncn(C(F)F)n2)=O)CC(NC(c2cc(C3CCCC3)no2)=O)C1 85504,c1(CC)c(OC)cc(C(=O)NCC2CCN(C(=O)C=CC(F)(F)F)C2)cc1OC 85505,CC(C)CC(=O)NCCC(C)N(C(=O)C(n1cc(Br)cn1)C)C 85506,c1(C(N2CCCCC(NC(C(C)CC3CC3)=O)C2)=O)cc(C#N)c(O)nc1N 85507,c1(OC)ccc(N(C(=O)CONC(=O)Cc2cn[nH]c2)C)cc1 85508,c1(C(=O)NCC(C)N(C)C(c2cn(C3CCCCC3)nn2)=O)cccn(C)c1=O 85509,C1(CNC(c2c(OC)n[nH]c2)=O)CN(C(c2ccccc2C)=O)C2(CCC2)C1 85510,C1(NC(C(c2scc(C)n2)C)=O)CN(C(=O)CC2CC2(Cl)Cl)C2CCCCC12 85511,C1(C(=O)OC)CN(C(c2sc(C)cc2Cl)=O)CC1(C)C 85512,c1(N2CC3CC(NC(C(CC)C)=O)CC3C2)ncc(C(=O)OC)cc1[N+](=O)[O-] 85513,CC1CC(C(=O)NCC(C2CCCN2C(=O)Cn2nccn2)(C)C)CCS1(=O)=O 85514,c1(C(N2CCC(C(=O)OCC)(CC)CC2)=O)[nH]c2nccc-2cc1Cl 85515,N(C1CCCc2c[nH]nc21)C(C1CC(NC(c2c(CC)cns2)=O)C(O)C1)=O 85516,N1(C(CCn2cc(CCC(C)=O)nn2)=O)CC2CCC(C1)O2 85517,N1(c2nccc(SC)n2)CCC(NC(=O)Cc2cn[nH]c2)C1(C)C 85518,c1(NC(C(C)N(C(=O)C(c2ccccc2)C)CC)=O)cccc(OC)c1C 85519,c1(C(C(=O)NCCN(CCOC)C(c2cscc2Cl)=O)C)ccccc1Cl 85520,c1(CC)cc(N2CCCC(NC(c3cccc(-c4ncon4)c3)=O)C2)ncn1 85521,c1(C(=O)NCC(CO)NC(c2c(C)nc(CC)s2)=O)nc(C)n(C)c1C 85522,N1(CC=C)CCN(C(=O)CC2(CN(C(=O)Cc3ccc(O)cc3)C)CC2)CC1 85523,C(CCCC(=O)N1CCCC(N(CC(C)C)C)C1)NC.C1CS1 85524,c1(CNC(C2CCC(NCc3cc(F)nc(F)c3)CC2)=O)ccc2c(c1)OCO2 85525,Cc1cccn2nc(C(=O)NCC(C)N(C(=O)CCC3CC3(Cl)Cl)C)cc12 85526,C(=O)(NN1CCCC1C(=O)NC1CCCC1CCOC)C1C(CC)N(C)CC1 85527,c1(C(C)(C)OC)nc(=NCC2(c3ccc(C)cc3)CC2)s[nH]1 85528,c1(C(N2CCCC(C3(C)N=N3)C2)=O)cc2cc(C#N)ncc2[nH]1 85529,Cc1cnc(C(=O)NC(CNC(c2cnc(C3CC3)nc2C)=O)CO)c(Br)c1 85530,c1(C(=O)NCC2C(CNC(C3CCC(C)(O)CC3)=O)C2)cc2n(n1)CC(F)C2 85531,C(=O)(CS(=O)C(F)(F)F)NCCN(C(c1c(C)ccs1)=O)CCOCCO 85532,c1(-c2c(-c3cn(CCC=C)nn3)cccc2)ccc(F)cc1F 85533,N1(C(C2(C)CCN(C)C2)=O)CC(C2CCCN(C(=O)C(C)(C)CS(N)(=O)=O)C2)C1 85534,Cc1cc(C(=O)NC2CN(Cc3n[nH]c4ccc(C)cc34)C2)c2n[nH]cc2c1 85535,Cc1n[nH]c(C)c1CC(C)C(=O)NCC(O)CN(C(=O)CSCC(N)=O)C 85536,C1(C(=O)NC(c2cncnc2)C)C2CC(O)C(C2)N1C(c1cc2n(n1)CCO2)=O 85537,C(=O)(C(CC(C)(C)C)OC)NCC1OCC(C(=O)NCCOCCC#C)C1 85538,c1(OC)cc(OC)cc(C(N2CC(CN(C)C(C3CCCC3(C)C)=O)C2)=O)c1 85539,N1(C(CC(CC)(C)C)=O)CCCC2(CCN(C(=O)Cn3cc(CO)nn3)CC2)C1 85540,C1(C(N2CCC2CC2CC2)=O)C(C2CC2)CCN1C(C1CCCCCC1)=O 85541,Cc1ncc(CNC2CCCC2NC(=O)CC2CN(C3CCCCC3)C2)[nH]1.C=O 85542,c1(C(N2C(CNC(c3ccoc3Cl)=O)C=CC2)=O)cc(O)c2ccoc2c1 85543,C1(C(C)OC)CCN(C(c2ccc(CNC(=O)CCOC3CCCC3)o2)=O)CC1 85544,c1(C(=O)NC23CCCC2CN(C(c2cc(O)cs2)=O)C3)cnc(O)c2ccsc12 85545,CC(C)(C)CCC(F)C(=O)N1CC(CNC(=O)C=C2CCOCC2)C2(CCC2)C1 85546,C(=O)(C(C)(C)CN(C(=O)CC(C)COC)C)NCc1cc(CC)no1 85547,C(C(O)C(F)(F)F)NC(CC1N(C(C2C(C)(C)C2)=O)CC1)=O 85548,c1(NC(N(CCO)Cc2scc(C)n2)=O)ccc(I)cc1Cl 85549,c1(CC)ccc(NC(=O)CN2CC(c3ccc(F)cc3)C(N)C2)cc1 85550,c1(NC(CNC(CNC(COCC=C)=O)CC=C)=O)ncc(N)cc1C 85551,c1(N2CCC(CC)(CC)CC2)nc(NCC2(C)CCCCO2)c2ncsc2n1 85552,C(=O)(C(C(C)(C)C)NC(c1cc(OC)ccc1N)=O)NCC(CC)OCC 85553,CC1(C)CN(C(=O)COC2CCCOC2)CC1C(=O)NCCn1cccnc1=O 85554,c1(C(=O)OCC(N)=O)ccn2[nH]c(=NC(=O)C3CC3Cl)nc2c1 85555,Cc1c(Br)ccc(NC(C2CC2C(=O)NCc2ccc(Br)cc2Cl)=O)c1F 85556,C=CC(CC(=O)NC12CC(C1)N(C(c1cncc(NC)c1)=O)C2)c1ccccc1 85557,c1(OC)c(F)cc(C(=O)NCC=CCNC(=O)C(C2CC2)C2CC2)cc1Br 85558,C1(CNC(C=Cc2ccc(C)nc2)=O)CN(C(c2ns[nH]c2=O)=O)CC(C)(C)C1 85559,c1(C(=O)NCCNC(C(CCSC)NS(CC)(=O)=O)=O)cc2scc(Cl)c2[nH]1 85560,CC(CC(=O)NCC12CCCC(CN1C(C1CCC1)=O)C2)CC(F)(F)F 85561,CC(C)C(C(=O)NC1CN(C(=O)C=CCO)CC1F)N1CCN(C)CC1 85562,C(CCCCCN=c1[nH]c2ccc(F)cc2o1)NC(C(CC)SC)=O 85563,C=CCC(CNC(c1c[nH]c(C(N)=O)c1)=O)NC(c1occc1C1CC1)=O 85564,c1(NC2CC(CNC(C(C)n3cccn3)=O)C2)nc2ccc(O)cc2s1 85565,CCC(CC(=O)N1CC(C(=O)NCc2ncnn2CC)C2(CCC2)C1)C(C)(C)C 85566,N1(C(C(CCC)OCC)=O)CCC(C)(C)CC1C(=O)NCc1cc(C)nc(C)c1 85567,Cc1c(S(=O)(=O)N2CCCC(C)CC2)sc2cc(F)ccc12 85568,c1(C(N(C2CN(C(CC(C)C3CC3)=O)CC2O)C)=O)cc2c(cnn2C)nc1O 85569,N1(C(C(=O)N(C)C)=O)CCN(C(C2CCC3CC23)=O)C2(CC2)C1 85570,CC1=C(C)CC(C)(C(=O)NC(C)CNC(c2sc(C(F)(F)F)nc2C)=O)CC1 85571,c1(C(N2CCC(NC(c3n(CC)nnc3)=O)(CO)C2)=O)c(OC)ccnc1O 85572,Cc1cn2cc(C(=O)NCC(CC(C)C)NC(=O)C(C)n3cnnn3)sc2n1 85573,Cc1cc(C)c2nc(N(C3CCN(C(C4(O)CCSC4)=O)C3)C)sc2c1 85574,c1(C(=O)NCC(CC)NC(CCCCCC)=O)c(N)sc2c1CCC2 85575,Cc1cc(Cl)nc(N)c1C(N1CCCC(O)(CNC(=O)CC2CCCC2O)C1)=O 85576,c1(CC)ccccc1OCC(=O)N(CC(C)(C)CNC(=O)C=C1CC1)C 85577,c1(C(=O)NCC2(NC(CCc3cnc(C)o3)=O)CC2)ncn2cc(Cl)ccc12 85578,c1(NCc2cc(C)ncn2)nc(N2CC3CC3(CO)C2)nc2sccc12 85579,C1(C)(NC(c2ncn(C)c2)=O)CCN(C(c2nnc(C(C)(C)C)s2)=O)C1 85580,N1(C(C2N(C)CC(O)C2)=O)C2CC=C(C(=O)NCc3n[nH]c4c3CCC4)C1CC2 85581,c1(C(C)=O)ccc(CC(=O)NC2CC(F)(CN(C(=O)CN3CCCCC3)CC)C2)s1 85582,Cn1ncc(Br)c1C(C(=O)NC1(C)CC1)N1CCC1c1cccc(Cl)c1 85583,N1(C(CC(C)C)=O)CCCC(CN(C(=O)Cc2ccccc2F)C)C1 85584,N1(Cc2c(CC)noc2CC)CCC(NC(=O)CC2CCCC2(F)F)C(C)C1 85585,C#Cc1ccc(NC(N2CC(C)(c3ccccc3)C2)=O)cc1Cl 85586,C1(CNC(c2c(C)nc(O)[nH]2)=O)CCC12CCN(C(=O)Cc1csc(Cl)c1)CC2 85587,C1(N(CCCc2nccc(C)c2)CC(=O)OC(C)(C)C)CCC2(CC1)CNC2 85588,Cc1cc(C(=O)NC2CCC(NC(c3ccc(O)nc3C)=O)C2)cnc1C 85589,C=C(C)CN=C(NCc1ccc(Cl)cc1Br)N(C)CCOc1ccc(SC)cc1 85590,C1(C(=O)NC(CC)CNC(=O)C(C)C)CC(c2cnn(C)c2)=NO1 85591,C#CC1(O)CCN(C(C2(OC)CCN(C(=O)CCC3CC3C)C2)=O)C1 85592,Cc1ccc(O)c(NC(C2(CNC(C3CC3C(=O)N(C)C)=O)CC=CC2)=O)c1 85593,Cc1ccc(C(=O)NC23CCC2CN(C(c2cc(C4CC4)on2)=O)C3)nc1C 85594,N1(C(C2CC(OC)C2)=O)CCCC(C)C1CNC(c1cnn(C)c1Cl)=O 85595,Cn1ccc2[nH]c(N(CCO)CC3CN(C(=O)NCCCCl)C3)cc12 85596,N1(C(c2c(OC)n[nH]c2)=O)CCC2(CC1)CC2CNC(C1CC(F)C(=O)N1)=O 85597,c1(C(N2C(C(C)NC(CCCCC)=O)CCCC2)=O)cccc2c1oc(=O)n2C 85598,NCC(C(F)(F)C(F)(F)F)NC1CCCCC1c1ccccc1 85599,S(=O)(=O)(c1c[nH]ccc1=NCCn1cnc(C)c1C)NC(C=C)(C)CC 85600,c1(OCCNC(N(CC(C)C)CCC)=O)cc(O)ncc1Br 85601,C1(CCNC(C(=O)Nc2cccc(N3CCN(C)C3=O)c2)=O)CCC(F)(F)CC1 85602,C(CC(C)(C)NC(C1(SC)CN(C(=O)C(CO)OC)C1)=O)OC 85603,c1(C(=O)NCC2(F)CC(CNC(C3C(C)C3)=O)C2)ccc2nc(=N)[nH]n2c1 85604,C=CCCCC(C)(C)C(=O)NC1CCCC(NC(c2ccccc2CC)=O)CC1 85605,C1(NC(c2cc(C)nc(C)n2)=O)C(C)CCN(C(=O)CC(F)(F)C(F)F)C1C 85606,Cc1cn2cc(C(N3CCC(CF)(NC(C4COCCO4)=O)C3)=O)ccc2n1 85607,N1(C(C(C2CCOC2)OC)=O)CCN(CCNC(c2cnc(C)s2)=O)CC1 85608,c1(OCC)ncc(C(=O)NCC2CCCN(C(C3(C)CCCO3)=O)C2)cc1Cl 85609,C=CCCCCCCCCC(=O)NC1CCSC12CN(C(=O)Cc1ccoc1)C2 85610,c1(C(=O)NC2CC(CCNC(COC)=O)C2)cc(C2CC2)nc2onc(C)c12 85611,CC(F)CC(=O)NC(C1CCCCC1)CNC(=O)Cc1cnnn1C 85612,Cn1nccc1C=CC(=O)NCC1CC2CC2N1C(=O)CSc1n[nH]c(=N)s1 85613,N1(C(CCCC#C)=O)CC2(C1)CN(C(c1sccc1Br)=O)CC2C(=O)O 85614,N1(C(C2(NC(C(CC=C)C)=O)CC(O)C2)=O)CC2CN(C)CC2C1 85615,N1(CCC=C=CC)C(=O)CN(CC2CCC(C)(C)O2)C1=O 85616,C1(C(=O)NC2CCCC(NC(=O)CCCC3CC3)CC2)CCn2ncnc2C1 85617,C(=O)(C(C(F)(F)F)C(F)(F)F)N1CCC2(C(CNC(CC(CC)CC)=O)C2)CC1 85618,C1(CNC(C2(CC=C)CC=CC2)=O)CCCN(C(=O)CC2C(C)C2(F)F)CC1 85619,C12(NC(C(C)CF)=O)CCCC1N(C(c1ccnc(S)c1)=O)CC2 85620,c1(C(N(C(CNC(C2CN(C(C)=O)C2)=O)C2CC2)C)=O)cc([N+](=O)[O-])cnc1O 85621,C(C(CNC(=O)C(=O)NCC(F)F)S(C)(=O)=O)NC(C1(CO)CC(C)(C)C1)=O 85622,N1(C(C=CCC2(NC(c3c(C)con3)=O)CCC2)=O)CCCC(CN(C)C)C1 85623,C(CC(C)C(=O)N(C1CCCN(C(c2ccccc2NCCO)=O)C1)C)OC 85624,N1(C(C2C(CC)C2)=O)CC(CNC(c2cnnn2CC)=O)(COC)C1 85625,C1(OC)CC2CC(NC(=O)CC3CCCN3C(=O)CC(=O)NC3CC3)CC12 85626,CCCC(C)(CCC)C(=O)N1CC2CCN(C(c3[nH]nnc3C)=O)C2C1 85627,c1(C(=O)NCC2C(NC(COC(CC)(C)C)=O)C2)ccc(OC)c(F)c1 85628,N1(C(c2c(C)ccs2)=O)CC2(CC2)CC1CNC(C1CC2CC1CO2)=O 85629,c1(C(=O)NCC2CC(NC(c3c[nH]c(=NC)o3)=O)C2)cc(NC(C)=O)cnc1C 85630,N1(C(CC(=O)OCC)=O)CC(F)CC1CN(C)C(c1ccccc1)=O 85631,c1(CN(C)C)ccc(C(=O)NC(c2ccccc2)CNC(C2(Br)CC2)=O)cn1 85632,c1(OC)cc(C)ccc1NC(C12CC(CO1)N(C(c1ccnc(O)c1)=O)C2)=O 85633,N1(C(C(CC)F)=O)CCC2(CNC(=O)CN3CCCCC3=O)CCCCC12 85634,C(=O)(CC(C)(C)C)NC(COC)C(=O)NCCC1CCCC1 85635,C(Cc1ccccc1)(C(=O)NC(C)(C)CNC(C1CC(CCF)C1)=O)NC(C)=O 85636,N1(C(c2c(C(C)(C)C)ncs2)=O)CC2CC(NC(=O)CCCCCF)CC1C2 85637,C#CCC(C(=O)N(CCCC(F)(F)F)C)NC(C1CCC(OC)CC1)=O 85638,C(C(C(=O)N(C1CCC(C)(C)CC1)C)C(C)C)NC(c1c(C#C)c[nH]n1)=O 85639,c1(C(c2nnnn2CCN2CCOCC2)NCc2cn(C)nn2)cccc(CO)n1 85640,N1(C(C(CCC)O)=O)CCCC(C)(NC(c2occc2Cl)=O)C1 85641,C1(C(=O)NCCCC2N(C(=O)C=CBr)CCC2)(CF)CCC(F)(F)CC1 85642,O=C1CS(=O)(=O)CC(C(=O)NCC2CN(C(c3ocnc3C3CC3)=O)CC2O)N1 85643,c1(C(=O)NCC(CNC(c2cc(F)n(C)n2)=O)OC)cc(F)c2ncccc2c1 85644,Cc1ccc(=O)n(CC(N2CCC23CN(C(C2CC24CCOC4)=O)C3)=O)n1 85645,c1(C(C(=O)NC2(c3cn(C(C(=O)NC(C)C)C)nn3)CCC2)O)ccccc1Cl 85646,N1(C(CNS(CC)(=O)=O)=O)CC2CS(=O)(=O)CC2(NC(C2CCC2OC)=O)C1 85647,c1(-n2ccc(CNC(Cc3c(C)cccc3)CO)n2)ccc(F)cc1F 85648,c1(CC)cc(C(=O)NC2CC2NC(=O)Cc2coc(C)n2)oc1CC 85649,Cc1cccc(CNCC2(C)CCN(C(c3nc(-c4nc[nH]n4)sc3C)=O)C2)c1 85650,c1(OC)ccc(C(=O)NCC2CCN(C(=O)C=CCF)C2(C)C)c(F)c1Cl 85651,C1(C(=O)NCC2C(C)(C)C2)CC2(CCN(C(=O)COCCCF)C2)C1 85652,N1(C(C2C(C)OC(=O)N2)=O)CC2CC1CN2C(=O)CC1CC2CC2C1 85653,c1(OC)cc(Cl)c(C)cc1NC(=O)C(N1CCC1CNC(=O)OC(C)(C)C)=O 85654,N1(C(c2cc(C)ns2)=O)CCC(C(=O)N(C)CCO)CC1C 85655,c1(C(N2CC3(CN(C(C=CC(=O)OCC)=O)C3)C2)=O)cc(C)c(Br)cc1C 85656,N1(C(c2cc(OC)n[nH]2)=O)C2CCC1(CNC(=O)C(C)CC1CCCO1)CC2 85657,c1(C(=O)NCC(N(C)C)C2CC2)cc(O)nc2c(Br)cccc12 85658,C1(C(F)(F)F)(COC)CN(C(C)C(=O)Nc2cc(Cl)cc(Cl)c2)CCO1 85659,C1(C)(CC)C=C(C(=O)NC(C2CCCN2C(C2CC=CCC2)=O)(C)C)C1 85660,c1(C(=O)NCC(CNC(C2CCC(C)O2)=O)(C)C)ncccc1N 85661,Cc1cc(C)c(C(=O)NCC2CCN(C(=O)C(C)N(C)Cc3ccccc3)C2)[nH]1 85662,c1(C(C(=O)NCCCOC)N(C)Cc2ccccc2)cc(C2CC2)n[nH]1 85663,Cc1sc(C(=O)NCC2(F)CCC(CNC(=O)C=CC3CC3)C2)cc1Br 85664,C(CN=C(NCC1(C(F)(F)F)CC1)NC(c1ccc(Cl)nc1)C)SC 85665,CC(CCCCNC(c1ccncc1Br)=O)NC(=O)CC1(C2CC2)CC1 85666,N1(C(c2cncc(C#C)c2)=O)CC2CC(O)C1C2NC(=O)CC1C(C)(C)C1(C)C 85667,Cc1ccc(OCC(O)CNCCCC2CC2C)c(C)c1Br 85668,c1(NC(C2CC(=C)CN2C(C2(C)CC2)=O)=O)cccc(Br)c1OC 85669,C1(NC(c2cnc3ccsc3c2)=O)CC2CCC1N(C(=O)C=CC1CCOC1)C2 85670,c1(C(=O)NCC2CCCN(C(C(CC=C)(C)C)=O)CC2)c(Cl)nc2ccccn12 85671,c1(C(=O)NC(CCO)C2CCC2)cc(F)c(Cl)c([N+](=O)[O-])c1 85672,CC1(CNC(=O)CCOCCCNC(c2c[nH]nc2[N+](=O)[O-])=O)CCCCC1O 85673,n1(CC(N2CC3CC(NC(C(C)OCC#C)=O)C3C2)=O)cc(C#N)c(O)nc1=O 85674,N1(C(c2cc(-c3cccs3)[nH]n2)C(=O)NC2(C)CC2)CC(CO)C(CCO)C1 85675,N1(C(c2c(C)oc(C(C)(C)C)c2)=O)CCC2C(C1)CN2C(=O)C(=O)C(C)(C)C 85676,C1(C(=O)NC2C=CCN(C(=O)CCC3CCCO3)C2)CC2CCCC(C1)C2 85677,n1(CC(=O)NC2CCCN(C(c3csc(C)c3N)=O)C2)cccc([N+](=O)[O-])c1=O 85678,C1(C(=O)NC(C(=O)OCC)C2CC2)CCC(C)(C)N(C(c2cccc(CC)n2)=O)C1 85679,C(=O)(C(C)(CC)CO)NCC1(Cc2cn(CCCC(=O)OCC)nn2)CC1 85680,N1(C(C(=O)NC2CC2)=O)CCCCC1C(=O)NCC1(c2cccc(F)c2)CCC1 85681,c1(NC2CC(NC(C3(F)CCCC3)=O)C2)nccc(Oc2ccccc2)n1 85682,CN1CCCC2C1CC(C(=O)NC1CC3CC1CC3N)N2 85683,C1(C(N(CC=C)C)=O)CC(NC(=O)OCc2ccccc2)C2CC12.OC 85684,N1(C(C2(OC)CCCC2)=O)CCCN(C(C2CCCC(C)(C)C2)=O)CC1 85685,c1(C(N2CCN(C(C(C=C)(C)O)=O)CC2CCO)=O)n[nH]c2ccc(C)cc12 85686,N1(C(=O)C=CC2CCCC2)CCN(C(c2ccc(CF)cc2)=O)C(CCO)C1 85687,N1(C(CC(CNC(C(CC)(C)OC)=O)O)=O)CCC2(CCC2)C1 85688,Cc1cc(=NC2COCC2F)[nH]c(=NCc2ccc(N(S(C)(=O)=O)CCO)cc2)[nH]1 85689,c1(N(CCCC)C)ccc(C(=O)NCCCOc2cccnc2C)c(F)c1 85690,C1(CCNC(c2cc(COC)sc2)=O)CCCCN1C(C1COC(=O)N1)=O 85691,CCC(C)C(O)C(=O)NCC1CC(O)(CNC(c2ccn(C(C)(C)C)n2)=O)C1 85692,c12ccc(C)c(c1)C(=O)NCc1cn-2nn1.Cc1cc(C)n(CC(C)N(C)C)n1 85693,C12CCN(C(=O)CNC1=O)O2.C1(C(C)C)CCN1C(N)=O 85694,C(c1cnc(C(C)(C)C)s1)=CC(=O)NCC(CC)NC(C1(CC(C)C)CCC1)=O 85695,CCC(Cc1ccc(N)cc1)C(=O)NCCNC(=O)CCc1nnc(C(C)C)o1 85696,c1(-c2c(CC)n[nH]c2)nc(C2CCN(C(C)=O)C2)nn1CC1CCCCC1 85697,c1(C(CCCC)C2CC2)cccc(Cl)c1.C1(C2CNC(=O)N2)CCCCC1 85698,C1(NC(=O)CC2OCCO2)CC2(CCOC2)C1 85699,c1(C(N2CCCC3(COC3)C2)=O)ccc2nc(-c3ccccc3)[nH]c2c1 85700,C1(C(=O)NC(c2ccc(F)cc2)CNC(C(CO)N(C)C)=O)CSCC(=O)N1 85701,c1(C(C)=O)ccc(Cl)cc1NC(C1CC2(C1)CN(C(c1ccon1)=O)C2)=O 85702,CC1=NOC(C)(C(N2CC(C)(NC(c3cc(C)c(-c4ccccc4)s3)=O)C2)=O)C1 85703,c1(CN2CCC(c3n(C)cnc3)C2)cnc2ncccn12 85704,C1(CC)CN(C(c2cnc(C3CC3)[nH]2)=O)CCN1C(c1cccc(C(F)F)c1)=O 85705,C1(NC(COC2CCN(C(c3n(C)nnc3)=O)C2)=O)CCCCCCC1 85706,C(CCN(C)C(C1(C)CC=CC1)=O)(C(C)(C)C)NC(C(c1ccccc1Cl)C)=O 85707,C1(NC(c2ccc(OC)cc2F)=O)CCCCN(C(=O)C(=O)NC2CC2)CC1 85708,C1(C(=O)NCCCN(C(=O)CCc2cccn2C)CC)CCNC1=O 85709,C1(C(N2C(CNC(Cc3cn(CC)nn3)=O)C(C)CC2)=O)CCn2cncc2C1 85710,c1(NC(=O)NC2(C3CCC3)CCC2)ncc(C(F)F)cc1Cl 85711,N1(C(C(C(C)C)SC)=O)CCC2(CC1)CCN(C(C1CCC3CCCCN13)=O)C2 85712,Cc1nc(N2CCC(C3CC3)C2CNC(C2(CF)CCC2)=O)c2scc(C)c2n1 85713,C1(NC(CC23CCC(OC)(CC2)C3)=O)CC2CC1C(O)C2O 85714,c1(C(N2CCCC(C(=O)OC)C2)=O)nc2ccc(-c3ccnnc3)cc2o1 85715,N1(C(C(C)CO)=O)CCCC(C(=O)NCCn2cccnc2=O)CC1 85716,C(=O)(C(C)(O)C(C)C)N(C)CC1N(C(c2cc(CCOC)on2)=O)CCCC1 85717,C1(=CC(=O)NC(C2CCCC2)CNC(C(CCSC)O)=O)CCCCC1(C)C 85718,c1(C(NNC(C(C)NC(=O)N(C(C)(C)C)CCO)=O)=O)ccc2c(c1)oc(=O)n2C 85719,Cc1cc(CC(N2CCN(C(=O)C3=CCCCC3)C(C)C2)=O)cc(C)c1 85720,c1(CC(=O)NC(C2CC=CCC2)C(=O)N(CCCOC)CCO)ccnc(O)c1 85721,c1(CC(=O)N(C2CCN(C(CN3CC(CC)C3)=O)C2)C)c(C)noc1Cl 85722,C1(NC(C2N(C(C)C)CCC2)=O)COC2(C1)CN(C(c1cncs1)=O)C2 85723,C(=O)(C1CCOc2ccc(Br)cc21)N1C(c2cn(C)nc2)C(=O)NCC1 85724,C1(C)(CC)CC(NC(c2ccc(CO)cn2)=O)CN1C(=O)C(C)C 85725,c1(C(=O)NCCN(C(C(c2scc(C)n2)C)=O)CC(C)O)csc(C#N)c1 85726,C12CN(CCO1)C2=O.C1(CN(C)C)CCC(NCc2cccnc2)CO1 85727,C(=O)(CC(C)CC(C)C)NC1CC(N(C(CNC(=O)NC)=O)C)C1 85728,CC(C)C(C(C1CCCCC1)NC(=O)C(N)=O)NC(c1nc(Cl)cs1)=O 85729,C1(C(=O)N(CC(F)(F)Cl)C)(CC)CCN(C(c2cc(Cl)ns2)=O)C1 85730,C1(NC(=O)Cc2n[nH]c3c2CCCC3)CCC2(CCNC2)CC1 85731,C1(C)(C(N2CC(CNC(c3c(CC)c(C)sc3)=O)C2)=O)CC(=O)N(C)C1 85732,N(C1CCc2c(Cl)ccc(Br)c21)S(c1c(C)cccc1Cl)(=O)=O 85733,C(=O)(CCC(C)CN(C)C)NCCN(C(=O)CC(C)F)CC.C#CC1COC1 85734,C12(C(=O)NC3(C)CN(C(c4ccn(C)c(=O)c4)=O)C3)CC(C)(C1)OC21COC1 85735,C1(CNC(CN(C(COC)=O)C)=O)C(C)CCCN1C(c1scnc1Cl)=O 85736,c1(C(=O)NCCCCCNC(=O)C=Cc2ccccc2)c[nH]c2c(F)cccc12 85737,C1(C(=O)NC(CC)(CNC(c2cnccc2OC)=O)CC)CC2(CCCC2)CO1 85738,c1(C(c2n(CCC)nnn2)NCC2(SC)CC2)ccc(SC)cc1 85739,Cc1ncc(CNC(C2CCN(C(C3(O)CCOC3)=O)C2)=O)o1 85740,CCC(CCC(=O)N(C1(C(N2CCOC(C)C2CO)=O)CC1)C)OC 85741,C1(CN(CC(C)(C)C)C)CCN(C(C2CC=CCC2)=O)CC1 85742,CC1CC(NC2=NCCNC(=O)NN2)CCN1C.C(=O)(C1CC1)NC1CC1 85743,c1(C(=O)NCCC(C)N(C)C(C2CCCN2C2CCCC2)=O)ccncc1N 85744,c1(NC(C(C)(C)NC(c2cn(CC)nc2)=O)=O)cn(C)nc1C 85745,Cc1nocc1CNC(C1(NC(=O)CCc2ccccc2)CC1C)=O 85746,c1(C(=O)NC(CCOC)CNC(C2CC3(CCCO3)C2)=O)[nH]nc2cnccc12 85747,C(C)(CCCC(C)C)OCC(=C)C(=O)NC1(CCC#N)CCOC1 85748,CN=c1ccc(C(=O)NC2(C(N3CCC3C(N)=O)=O)CCCC2C)c[nH]1 85749,C1(OC)CN(C(=O)Cc2n[nH]c(C)n2)CC1NC(=O)CCOC1CCCC1 85750,c1(CCNC(C(c2ccco2)NC(COC(CC)C)=O)=O)c[nH]nc1O 85751,c1(-n2c(C3CCC(OC)C3)nc(-c3ccoc3C)n2)cc(F)cc(F)c1 85752,C1(C(N2CC3C(CNC(=O)C4=CCCCO4)(C3)C2)=O)CCC2(CCC2)CC1 85753,C=CC(C)(CC)C(=O)NC1C2CC1N(C(c1ccsc1OC)=O)C2 85754,C(=O)(C1(C)CCn2ccnc21)N1CCC(O)(CN(C)C(C2CCCC(F)C2)=O)C1 85755,Cc1cc(=NC2C(C)C2C)[nH]c(N2CCOC(c3cc[nH]n3)C2)n1 85756,c1(C(N2C(C)CC(CNC(=O)C(C)(C)CC3CCOC3)C2)=O)cnc(O)c(F)c1 85757,C1(C)(CNC(CC(=O)OCC)=O)CCN(C(=O)C(C(C)O)N(C)C)C1 85758,c1(C(=O)NCCOC2CN(C(C(CN(C)CC)F)=O)C2)cccc(COC)c1 85759,C(=O)(CC(=O)N1CC(NC(C2CC(OC)C2)=O)C1)OCC 85760,c1(C(=O)OC)cc(C(N2CCC(CNC(=O)COc3ccsn3)C2)=O)cc(F)c1 85761,C1(NC(CCC#CC)=O)CN(C(c2cccc3ccoc23)=O)C2(CCCC2)C1 85762,CCCC(C)CC(=O)N1CCCC1CN(C(=O)C(C1CCOCC1)=O)C 85763,C12(C(=O)NC3C(NC(c4ccc(CC)[nH]4)=O)COCC3)CCC(C)(CC1)CO2 85764,n1(CC(=O)NCC(CNC(=O)C#CC2CCCO2)O)sc(=O)c2ccccc12 85765,Cc1cc(C(=O)NCC2CC2CNC(c2ccccc2F)=O)cc(C)n1 85766,C(C#Cc1cccnc1)NC(c1cccc(CNc2ccccc2)c1)=O 85767,Cc1ncc(CCC(N2CCN(C(=O)CCNS(C)(=O)=O)C3CC23)=O)c(O)n1 85768,C=C(C)CC(C)C(=O)NCCOC1CN(C(C2COC(=O)N2)=O)C1 85769,CC1(C)CC(C)(CNC(=O)Cc2ccon2)CN1C(=O)CC1CCC(=O)O1 85770,O=C(CC1COCCO1)NOC1CCOC1.C(C=O)O 85771,c1(C(=O)NC(C(C)NC(C#CC(C)C)=O)CO)cccc(S(=O)(=O)NC2CC2)c1 85772,c1(C(=O)OCCSC2CCCCO2)cc2c(=O)cc[nH]c2s1 85773,CC1(C)CC(CO)CN1C(=O)CN(C1CC(C#N)C1)C(=O)CC1CNC(=O)O1 85774,CC(C)(C#N)CC(=O)NC(C)(C)CCNC(c1cc(F)cc(Br)c1)=O 85775,C1(C(C)NC(=O)C=Cc2nccs2)CN(C(=O)C=C2CCOCC2)CCO1 85776,C(CC1CC1)(C(=O)NCCC1(C)CCCO1)NC(C(C)=CC(C)(C)C)=O 85777,c1(C(=O)NC2C(F)CCN(C(C(C)c3cccs3)=O)C2)cc2ccc(F)cc2[nH]1 85778,C1(CNC(CC(C)F)=O)CCN(C(C2CC2c2ccncc2F)=O)CC1(F)F 85779,C(=O)(CCCC(N)=O)NCCC(C)NC(=O)COCc1nccn1C 85780,N1(C(CC=CC=C)=O)CC2C3CCC(C2C1)N(C(=O)CCc1ccnn1C)C3 85781,c1(OC)nn(C)cc1C(=O)NC(C1(O)CN(C(=O)CSCC(C)C)C1)C 85782,O=C(C1=CCC(NC(=O)CCc2ncccn2)C1)NC1(C(N)=O)CC(CO)C1 85783,Cc1c(NC(=O)C(=O)NCCN(CCO)Cc2ccccc2)cnn1CCC(C)C 85784,C=CCC(CNC(=O)CSCc1cscn1)NC(C1C(C)C1(F)F)=O 85785,c1(OC)cc(N)c(C(=O)NCCC2(OC)CN(C(=O)C3=CCCCO3)C2)cc1F 85786,N1(C(CCN(CCCCC)C)=O)CCN(C(C2(C)CC=CCC2)=O)CC1C 85787,C12(C(=O)NC(c3ncc(-c4ccc(C)cc4)[nH]3)C3CC3)C3CC(CC13)C2(F)F 85788,C(CC(C(C)C)NC(C1(NC(=O)CC2CCCC2O)CC(O)C1)=O)OC 85789,N1(C(c2c(C)n(C)nc2)=O)CC2CN(C(c3cc4c(s3)CCOC4)=O)CC2(C)C1 85790,c1(C(=O)NCC(CC)NC(c2ccc3snnc3c2)=O)cccn2cc(C)nc12 85791,N1(CC2OCC(=O)C2)CCn2c(Cc3ccccc3)nnc2C1 85792,N1(C(=O)NCC2N(c3n(CC)ncc3)CCC2)Cc2nc(C)nc(O)c2C1 85793,C(CC(C(=O)N1CCCC1)NC(=O)CCC1CC1(F)F)SC 85794,c1(C(=O)NCCN(C(=O)CCc2ccsc2Cl)C)nnn(C2CC2)c1C(F)F 85795,c1(OCCSCC(=O)NCC(C)NC(CC(=O)OCC)=O)ccccc1COC 85796,C(=O)(C(C)(C)CS(N)(=O)=O)N1CCC(C)C(CNC(c2ccc(Cl)cc2)=O)C1 85797,CC1CN(C)CC(C(=O)NCC2(NC(c3cc(=O)cc(Cl)[nH]3)=O)CCC2)O1 85798,c1(CNC2CCCCN2C(C2(OC)CCC(C)(C)C2)=O)cc(F)cc([N+](=O)[O-])c1 85799,Cn1ncc2c(O)nc(=NCCCNC(c3csc(CO)n3)=O)[nH]c12 85800,c1(CC)cscc1C(N1CC(C(=O)NCCNC(C23CC(CO2)C3)=O)C1)=O 85801,C(N=c1[nH]nc(C)o1)C1CCCC(NC(CCc2cc(OC)no2)=O)C1 85802,N1(C(c2c(CCC)occ2)=O)CCN(C(=O)C(O)Cc2[nH]cnc2C)CCC1C 85803,CC(CC(=O)N1CCCCC(NC(=O)C(C2CCCC2)C2CCCC2)C1)C(F)F 85804,C1(C(=O)NC2C(NC(c3cc(C)sc3)=O)CCC2)OCCOC1(C)C 85805,N1(C(c2cnc(CC)nc2C)=O)CC2CN(C(C3CC3C3CC3)=O)CCC12 85806,c1(N(CC)CC)cc(CNC2(C(F)(F)F)CCOCC2)ncn1.C1CN(C(C)=O)C1 85807,CC1(NC(=O)CCOCC(F)F)CCN(C(=O)CCc2ccco2)CC1 85808,C(CCCCC(=O)NCC(C)N(C)C(c1cc(Br)nn1C)=O)SC 85809,c1(CC)ccccc1C(=O)N(C1CCN(c2nnnn2Cc2ccccc2)C1)C 85810,Cc1ncc2c(n1)CN(C(=O)OC(C)(C)C)C2C(=O)NCc1cnnn1C 85811,C(=O)(CC1=CCCC1)N1C(C(=O)NC2CC3CCC2O3)C=CC1 85812,c1(CC)nc(C)ncc1C(=O)NC1CCN(C(=O)CCn2ccc(C)n2)C1 85813,c1(NC(CC)=O)ccccc1C(=O)NC1CC1NCCSC(C)(C)C 85814,C1(C)(CNC(C(C)SC)=O)CC(F)(F)CN1C(c1cccc(OC(C)(C)C)c1)=O 85815,CN1CCC(C)(C(N2CCOC(CNC(=O)CN3CCCOC3=O)C2)=O)C1 85816,N1(CCC(=O)N(C)CC2CCN(C(c3sncc3Br)=O)C2)C(=O)CCC1=O 85817,N1(C(C(C(=C)C)(C)O)=O)CCCC2(CCCN2C(=O)CCSC)C1 85818,CC(C(C)C(=O)NOCCCO)NC(c1cnn2cccc2c1)=O 85819,C#CCCCCC(=O)N1CC(C=C)(CC(=O)NC(CO)C(C)(C)CO)C1 85820,C=CC1CCN(C(=O)C(C2CCCCC2)NC(C2CCCN2C=O)=O)C1 85821,N1(C(C2(C(C)C)COC2)=O)CC(CNc2nccc(OCC(F)(F)F)n2)C(O)C1 85822,N1(CC(=O)NCC(c2ccncc2)C)CCC(NC(=O)NC2CCCCC2)C1 85823,CN1CC(C)(C(N2CC(C)(CCC(N3CC(=O)NC(CO)C3)=O)C2)=O)CC1=O 85824,C1(C(=O)NC2CC(F)(CNC(C(C)SC(C)C)=O)C2)CCC12CCC2 85825,N1(C(c2cnc(OC)s2)=O)CC2CCCC2(NC(=O)CCOCC2CCCO2)C1 85826,CC1CN=C2NC(C(=O)N(C(C)CCNC(c3sccc3C3CC3)=O)C)=NN2C1 85827,C(=O)(C1=C(F)CN(C(c2csnc2Cl)=O)CC1)N(C(CC)CC)C1CC1 85828,C(C)(C)(CCCN=c1ccnc(SC)[nH]1)NC(CC)=O 85829,O=C1CCC(C2(C(=O)OC3(C4CC4)CC3)CC2)CC1 85830,Cc1nc(O)nc(O)c1NC(C1(F)CCN(S(=O)(=O)CC(C)C)CC1)=O 85831,C(=O)(C#CC(C)(C)C)N1CCC(N(C(COC)=O)CC2CC2)C1 85832,c1(C(N2CCCC(C)(CNS(=O)(=O)C(F)(F)F)C2)=O)ccc2ccoc2c1 85833,C1(C(=O)NC(CNC(C(COC)(C)C)=O)C)CCc2ccccc2O1 85834,C1(C(=O)NC2CC(C)(NC(c3cnn(C)c3Br)=O)C2)CCCCS1(=O)=O 85835,C1(CC)CN(C(C2CC2C(C)O)=O)CCC1NC(=O)C(F)OC(F)(F)F 85836,c1(C(=O)NC(C=CC(=O)NCC(=O)OCC=C)(C)C)cccc(F)c1 85837,CC1N(C(=O)C(C2CC2)NC(C2CC2C2(C)COC2)=O)CCCC12CCC2 85838,N1(C(c2c(C(=O)OC)cncc2)=O)CC(C2CCCN(C(=O)CC(C)C)C2)C1 85839,c1(C(N(CCNC(Cc2nc(C(C)C)sc2)=O)C2CC2)=O)ccc(C2CCC2)nc1 85840,C1(C(=O)Nc2c(F)cc(Cl)cc2Br)CC2(CCN(CC3CC4C=CC3C4)CC2)C1 85841,c1(C(=O)OC)cnc(C)cc1N1CC(C)(NC(c2cnn(C3CC3(F)F)c2)=O)C1 85842,C1(NC(c2c(C)nc(CC(C)C)o2)=O)CC2CC(C1)N(C(C1(C3CC3)CC1)=O)C2 85843,CC1CN(C(C2CC(F)(CO)C2)=O)CCC1NC(=O)CCN(S(C)(=O)=O)C 85844,c1(C(N2CC(NC(C(C(=C)Cl)(C)C)=O)C(F)C2)=O)nc2ncc(CCO)cn2n1 85845,C1(NC(C(C)(C)F)=O)CCN(C(=O)C(C)(C)C2CCCO2)CC1O 85846,c1(CCNC(=O)Nc2cccc(OCCF)c2)c[nH]c2ncc(F)cc12 85847,C12(C(N(CCOCCOC)C)=O)CCC(CC1)N(C(c1cn(C3CC3)nn1)=O)C2 85848,C1(C(=O)O)CC2(C1)CC(C)N(C(=O)C(O)CN1CCCCC1)C2 85849,c1(C(N2CC(C)(NC(c3c(CC)onc3)=O)C2)=O)ccnc(Cl)c1O 85850,c1(C(=O)NCC2(NC(C(COC)C)=O)CCC2)cc(F)c2nc(C)cn2c1 85851,CCCC(C(=O)OC)C(=O)NCC1CCC(C(=O)NCc2nc(C)ccc2O)C1 85852,C1(C)(c2cccc(C)c2)NC(=O)C2=C1N(C)C(=O)N(C)C2c1cc(Br)ccn1.CC=O 85853,Cc1ccnc(C)c1C(=O)NCCC1CC(NC(C2CC23CCOC3)=O)C1 85854,N1(C(C2C(C)C2)=O)CCCC2CN(C(c3n[nH]c4c3CCCCC4)=O)CCC12 85855,N1(C(CSC)=O)CCN(C(=O)C(F)C(C)(C)O)C(CS(C)(=O)=O)C1 85856,c1(C(N)=O)ccc(-c2cn(-c3ccc(C(=O)NC4CC4C(F)F)nc3)nn2)cc1 85857,C12(CNC(C(CCSC)O)=O)CC(C(N)=O)(C1)C1(CN(C(=O)C=CC(C)=O)C1)O2 85858,N1(C(Cc2c(C)ncs2)=O)CCC(C)(C)CC1C(N1CC2C(C1)C2(C)C)=O 85859,CCCCC(C)CCC(=O)N1C(C(=O)NCc2ncccn2)CCC1C 85860,C12(C(N3CCC(CCNC(C4CN5CCC4CC5)=O)CC3)=O)CCC(CC1)CO2 85861,N1(C(Cn2cc(-c3occ(C(=O)O)n3)nn2)=O)CCC(O)C(F)(F)C1 85862,CCC(C)CCCCC(=O)N1CC(OCCNC(c2c(F)cc(O)cc2F)=O)C1 85863,C1(C)(CNC(C23CC(C(=O)OC)(C2)C3)=O)CN(C(=O)Cc2ccc(O)nc2)CCO1 85864,C1(C(=O)NCCCOC=C)CC(NC(=O)CCC(=O)N(C)C)C1(C)C 85865,c1(C(C)NC(=O)NC(c2nc(C)sc2C)C)ccc(C)c(Br)c1 85866,N1(C(c2n(C=C)nnc2)=O)CCCN(C(C2CC2CC)=O)CC1 85867,C(C)(c1ccc(OC)cc1)=CC(=O)NCC(C)(CC)NC(C1C(=C)CC1)=O 85868,C1(O)(CNC(COCCCCC)=O)CCCN(C(=O)C(F)C(C)C)CC1 85869,C1(C(N(CC(C)NC(CSCC)=O)C)=O)CCC(=O)O1 85870,CC1(C(=O)NCC2Cc3ccccc3C2)CC12CCN(Cc1ccns1)CC2 85871,c1(C(N(C2CCOC2)CCCNC(C2(CC(=O)OCC)CC2)=O)=O)ccccc1 85872,c1(OC)ccc(C)cc1C=CC(N1CCCCC1CNC(c1n[nH]cc1C)=O)=O 85873,N1(C(CCCc2c(OCCC)nc(Cl)cc2)=O)CC2(CCOC2)c2ncccc21 85874,c1(C(N2CCC(CF)C2)=O)coc2c1CN(C(=O)C=CC1CCCC1)C2 85875,C1(NC(C2CN(C(N)=O)C2)=O)CN(C(=O)CCC(=O)c2cccc(F)c2)CC1O 85876,N1(CC(=O)NC(C(=O)N(CC(CCC)O)C)CC2CCC2)CCC(=O)CC1 85877,C1(C(=O)NCCN(C(C(Cc2ccc(OC)cc2)O)=O)C)CCN(C)S1(=O)=O 85878,C1(C(=O)NCCC(C)CCNC(=O)COC2(C)CCC2)(OC)CCC12CCC2 85879,N1(C(c2cc(CCC)oc2C)=O)CCC(C)C(N(C(=O)C(C)OCC(C)C)C)C1 85880,c1(NC(C2N(C(CCOCC#C)=O)CCCC2)=O)ccc2oc(C(N)=O)cc2c1 85881,c1(NCCCC(CC)O)nccc(=NCCOc2cccc(F)c2)[nH]1 85882,C12(C(=O)NC3CN(C(C4C(Cl)(C(=O)OC)C4)=O)C3)CC(CN1OC(C)=O)C2 85883,O(N(C)C(=O)CC(C)(C)N(C(=O)C(C)(O)CC(C)C)C)CC(=O)OC 85884,Cc1ccsc1CC(=O)NC1(CNC(=O)C(C)CN(C)C)CCOC1 85885,C1(N(C(CC(C)C2CCCCC2)=O)CCNC(C2CCSC2)=O)CCCCCC1 85886,C1(c2scc(C)n2)CN(C(=O)Cn2cc(CN(C)C)nn2)CCO1 85887,N1(C(C(CC)=CC)=O)CC(CNC(=O)CC2(O)CCCC2)CCC1C 85888,CC1(O)CCN(C(=O)CC(O)CNC(=O)C2=C(Cl)CCCC2)CC1O 85889,N1(C(c2nc(-c3ccccc3)ncc2Cl)=O)CCSCc2ccccc21 85890,C(C)(C)(CCCNC(C1NC(=O)CC1C)=O)NC(COCc1nnc(C)s1)=O 85891,C1(C)(CC)CCN(c2nccc(C(C)(F)F)n2)C1 85892,CCCCC(F)(F)C(=O)NC(CC1CCCC1)C(=O)NOCC(=O)OCC 85893,C1(S(C)(=O)=O)(C(=O)NCCC(C)(C)NC(c2n(CC)ncc2)=O)CCOCC1 85894,c1(OC)c(C)cc(C(=O)NC2CCC(CNC(c3cccc(C)n3)=O)C2)cc1C 85895,C(=O)(N=c1ccn(CCN2CCCC2)[nH]1)N(C)CCc1ccccc1Cl 85896,C1(N(C(c2c(CNC(Cc3cc(C)[nH]n3)=O)noc2)=O)C)CCCC1(C)O 85897,c1(OC)ccc(C=CC(=O)NC2CCCC2NC(c2cccn2C)=O)c(C)c1 85898,C(=O)(CCCSC)OC(=O)C(C#N)C1CC1.N(CCN)(CC)CC 85899,C1(C(=O)NC(C2CCCC2)CNC(c2cccnc2F)=O)CC2C=CC1CC2 85900,O(P(C)(=O)CNC(CCN(C)C)C(=O)NCCC1C(=O)N1)CC 85901,c1(C(N2C3(CNC(C4(O)CCC(CC)C4)=O)CC(C2)C3)=O)c(C)[nH]c(C)c1C 85902,O=C(C(O)CC(F)F)N1CCN(CC2CCCO2)CC1 85903,C1(OC)(CNC(=O)CCSc2ccccn2)CN(C(C2CC2(C)C(F)F)=O)C1 85904,N1(C(C(C)=NOCC#N)=O)CCOCC(CNC(=O)CSC(F)F)C1 85905,C1(NC(C2CN(C(C)C)C2)=O)CN(C(C2CC3(CSC3)C2)=O)CC1N=[N+]=[N-] 85906,Cc1nc(C)c(C(N2CCOC(CNC(C3CC3(C)C)=O)C2)=O)o1 85907,N1(C(CCC(=O)OC)=O)CC(C)CN(C(=O)C=Cc2ccccc2C)CC1C 85908,CCC(C)C(C(=O)N(C1CCCC1C#N)C)NC(=O)CSC(F)F 85909,C(=O)(C(C)(CC)OC)NCC(CC=C)NC(c1ccoc1Br)=O 85910,c1(CC)cccc(CC)c1CC(N1CCC1CNC(c1nc(C)c(C)[nH]1)=O)=O 85911,Cc1cnc(C(=O)NCC2CN(C(c3ccc(CO)cc3F)=O)C2)cc1C 85912,CC(C)CC(C(=O)N(C1CCN(C)C1)C)ONC(=O)C1(C(N)=O)CC1 85913,c1(C(N2CCC(N(C(C(C)OCCCCCC)=O)CC)C2)=O)cc[nH]c(=NC)c1 85914,C1(OC)CC(CNC(C2CCCC3CC23)=O)N(C(c2cc[n+]([O-])cc2)=O)C1 85915,C(=O)(CCCC(C)C)NC1CN(C(CS(CC)=O)=O)CC1CC1CC1 85916,C1(CC(=O)NCc2ccccc2CNC(c2ccncc2O)=O)CCC1C1CC1 85917,Cc1c2cccc1C(=O)N2.C1(O)(C(C(=O)NC(CNC(C)C)(C)C)F)CCCC1 85918,CC(CCC(C)(C)C)C(=O)N1CC2COCCC2(NC(=O)CCc2cc[nH]n2)C1 85919,N1(C(=O)Cc2cc(Cl)cs2)CCC2(C1)CN(C(c1cncn1C1CC1)=O)CCO2 85920,C(=O)(C1CSc2ccccc21)N(CCCN(C)C(c1n[nH]cc1Br)=O)C 85921,C(CC(C(=O)NCCCCC1CC1C)N(C)C)NC(CC1C(CC)C1)=O 85922,N1(C(C(c2cncnc2)C)=O)CCCC(C2CC2NC(=O)Cc2csc(Cl)c2)C1 85923,c1(C(N2CCC(CN(C(C3CC(OC)C3)=O)C)C2)=O)nc2c(cc1Cl)OCCO2 85924,N1(C(C)=O)CCCC1CNC(C1CC(NC(=O)CCC=CC(C)C)C1)=O 85925,N1(C(c2c(C3(C)CC3)cccc2)=O)CC2(C1)CN(C(=O)C(O)C1CCC1)C2 85926,c1(CN2CCCC(C(=O)NCc3nnc(C)o3)C2)ccc(F)c(Br)c1F 85927,N1(C(C=CCN(CC(F)(F)F)C)=O)CCC2CN(C(C3CCCO3)=O)CC2C1 85928,C1(NC(C2(OCC)CCOC2)=O)CC2(C1)CC2NC(c1ccc(Cl)cn1)=O 85929,c1(CCC=C)ccc(C(=O)NC23CC2CN(C(=O)CN(CC(C)(C)C)C)C3)cc1 85930,CC(N=c1nc(C(F)(F)F)[nH]s1)C1CCN(C(=O)CCc2ccc(F)cc2)C1 85931,c1(C(N(CCCNC(c2c(F)ccc(C)n2)=O)C)=O)cn(C)c2ccc(F)cc12 85932,c1(OCC)cc(C(=O)NC2(C3CCCN3C(=O)C(F)OC)CC2)ccn1 85933,C(=O)(CC(C)CC(C)(C)C)NCc1cc(C(=O)NCC(C(C)O)(C)C)n(C)n1 85934,CC1(C)C(C(=O)NCC2CN(C(c3cc(C(N)=O)cs3)=O)CC2O)C1C#N 85935,CC1(C)CN(C(c2ccnnc2O)=O)CCC1C(N1C(CO)CC1CO)=O 85936,N1(C(C2CC3CCC(C2)N3)=O)Cc2cccc3c2C(CCC3)C1 85937,c1(C(=O)NC(CNC(c2c(CC)[nH]nc2Cl)=O)(C)C(C)C)sc2cncn2c1C 85938,C1(NC(CSCCCC)=O)CC(C)N(C(c2cnc(C(F)(F)F)nc2)=O)C1 85939,CC(C)CC(C)CC(=O)N(CC(C)(C)CNC(=O)C=C(Cl)Cl)C 85940,N1(C(C(=O)N(CC)CC)=O)CCN(C(=O)Cc2cc(C)ccc2OC)CC1CF 85941,c1(C(=O)NC(CC)CNC(=O)C(C)(O)COC)cc2c(n1C)CCOC2 85942,N1(C(CCC)C)CC(C(=O)OCC2(CO)CCCC2)CC1=O 85943,Cc1cc(C(=O)NC2(C(N3CCCC3)=O)CSC2)[nH]c1C 85944,c1(CNc2cn(C(C)C)nc2Br)cnc2c(cnn2C)c1 85945,c1(OCCOCC)ccc(C(C)OC)cc1.C1C(=O)O1 85946,O=C(C1CCOc2ccccc21)N1CCC(c2nn[nH]n2)(C(F)(F)F)C1 85947,c1(C(N2CC(CCNC(c3ccc(C)cn3)=O)C2)=O)cc(=O)n2nccc2[nH]1 85948,CC1CN(C(=O)Cn2cc(Cl)cn2)CC(C)C1Nc1cc(C(N)=O)ncn1 85949,C1(NC(c2cc(C3CCCC3)on2)=O)CC1C1CCCNC1 85950,C1(NC2CCC(C(=O)NCC)CC2)CCCN(Cc2cccnc2NS(C)(=O)=O)C1 85951,Cc1cccc(SCC(=O)NC2CCN(C(=O)CC(C)n3ccnc3)C2)c1 85952,C=CC(C)C(C)C(=O)N(C)CCN(C(=O)CCc1ccc(Br)s1)C 85953,CC(C)CC(C)(O)CNC(C1CC(NC(=O)Cc2cncs2)CCO1)=O 85954,c1(SC)cccc(C(N2CCCCC2CN(C(=O)C(Cl)=CCl)C)=O)n1 85955,C1(NC(c2nc(C)[nH]n2)=O)CN(C(c2c[nH]nc2C)=O)CCC1CO 85956,C12(C(N3C(CN=[N+]=[N-])CC3)=O)CCC(CC1NC(C1CCS1(=O)=O)=O)C2 85957,c1(C(N(C)CC2N(C(C(COC)(C)OC)=O)CCC2)=O)cc(C)cc2ccoc12 85958,c1(C(N(CC(=O)NCC)CC(=O)NCC)=O)cc2nc(F)ccc2o1 85959,C#CC1(NC(C2COCCN2C(c2c[nH][nH]c2=N)=O)=O)CC2CCCC12 85960,Cn1nnc2c1CCC(C(=O)NCC1CCCN(C(c3ccc[nH]3)=O)C1)C2 85961,c1(C(N(C2CN(C(COCC(C)C)=O)CC2F)C)=O)cc2c(nc1O)CCOC2 85962,c1(C(N2CCC(N(C(Cn3c(CCC)ncc3)=O)CC)C2)=O)cnn(CC)c1C 85963,C(=O)(C(CC(C)C)ONC(c1cnn(C(F)F)c1)=O)NC(C(=O)OC)(C)CO 85964,CCCCCCn1nnnc1C(c1cnn(CCCSC)c1)NCCOCCOC 85965,C(=O)(CCCCCC(C)O)N1CC(N(C(c2c(C)[nH][nH]c2=N)=O)C)C1 85966,C1(O)(CCN(C)C(C2(N(C)C)CC2)=O)CCN(C(C2CCCC(N(C)C)C2)=O)CC1 85967,C1(O)(C(=O)NC(C2CCCN(C(=O)OC(C)(C)C)C2)C)CN2CCC1CC2 85968,C1(C(=O)NCc2c(C)ocn2)CN(C(=O)C(C)(C)CN(C)C)CC12CC2 85969,C1(C(=O)NC(C2CC(NC(CCc3c(C)noc3)=O)C2)C)CCN(C)CC1 85970,c1(C2(C(N(CC(C)NC(c3cc(Cl)n(C)n3)=O)C)=O)CCC2)ccc(F)c(Cl)c1 85971,C(=O)(CCC(=O)N(C1CCCN(C(=O)CSCC(F)(F)F)C1)CCF)NCC 85972,n1(C(C(=O)OCC)C)cc(CNC(=O)NCCOCCN(C)C(C)C)nn1 85973,c1(NC(=O)CSCC(=O)N(C2CCCNC2)CC2CCCCC2)ccc(F)cc1 85974,C1(C(N2CCC(NC(c3cncn3C)=O)C2)=O)(OC)CCOC1 85975,c1(C(=O)NCC2C(NC(C(CCC)(C)O)=O)C2)ccc(Br)c2ccccc12 85976,C1(CCNC(C(CC)C)=O)CCN(C(C2(F)CC2(Cl)Cl)=O)CC1(F)F 85977,c1(OC)c(C(N2CC(CCNC(C3(C)CC3)=O)OC(C)C2)=O)occc1=O 85978,c1(N2CCCC(NC(C3CC(O)C3)=O)C2)ncnc2c(F)cccc12 85979,Cc1ncc(C(=O)NCC2(O)CCN(C(=O)CC3CNC(=O)C3)C2)n1C(F)F 85980,N1(C(C2(OC)CCC2)=O)CCN(C(=O)C(C)O)C(CC(F)(F)F)C1 85981,N1(C(c2c(C)snn2)=O)CCC2(CC1)CC2NC(=O)CC(C)n1cccn1 85982,N1(C(COCC(C)(C)C)=O)CCC(NC(C2CCC3CC3CC2)=O)C(F)C1 85983,C=CCC(CC)C(=O)NCC(CNC(=O)Cn1nccc1C)C(F)(F)F 85984,O=C(C1=CC2(CCOCC2)C1)NC1(C2CN(C(C3CC4CC4C3)=O)C2)CC1 85985,c1(C(=O)NC2CCC(NC(CCCCCSC)=O)C2)onc2c1CCCC2 85986,C1(NC(=O)CCCF)CC2CCC1CN2C(=O)Cn1cnnc1 85987,c1(CC(=O)NC2CCN(C(c3cn(C)nc3)=O)CC2O)c[nH]c2cccc(Cl)c12 85988,C(=O)(C1Cc2ccc(F)cc21)NCC(CN(C(Cn1c(C)ncc1)=O)C)O 85989,c1(OCC(=O)NCC#CCNC(C2OCC(C)C2)=O)ccccc1C(C)(C)C 85990,C1(C(N2C(C3(NC(C45CC(OC)C4C5)=O)CC3)CCC2)=O)CCS(=O)CC1 85991,C12(CCNC(C=CSC)=O)CCC(C1)N(C(c1ccco1)=O)C2 85992,CC1(C)CCCCCC1NC(C1(F)CCN(C(=O)Cc2cccnc2)C1)=O 85993,Cc1ccc2c(c1)CCN2C(=O)CC(C(C)C)NC(=O)Cn1ncnn1 85994,c1(C(=O)NCCC2CCC(NC(C3CSC3)=O)C2)ccc(F)cc1OC(F)F 85995,C1(C(=O)NC2CCC(N(C(c3cccc(C)c3)=O)C)CC2)CC2(CCO1)CC2 85996,N1(C(CC(C)C(C)(C)C)=O)CCCC2(CCCN2C(c2cc(C3CC3)ns2)=O)C1 85997,c1(NCC2(NC(C(C(COC)C)C)=O)CCOC2)c(F)cc(C#N)cc1[N+](=O)[O-] 85998,C1(NC(c2ccc(CC)o2)=O)CCCCN(C(=O)CCCCCc2cnc[nH]2)C1 85999,C1(N(C(C(C(C)C)C)=O)C)CC2CCC(C1)N2C(c1cccn2cnnc12)=O 86000,CCCCCCCC(C)N(C(C(C(=O)N)(C)C)=O)CCOC.OCC 86001,C1(NC(=O)CCc2nc(-c3nc[nH]n3)no2)C2CC1CN(C(C1CC1CF)=O)C2 86002,N1(C(C=CC)=O)CC2CN(C(C34CC(c5ccccc5)C3C4)=O)CC2C(F)(F)C1 86003,C1(C(=O)NC(C)CC2(O)CCC2)CC(C)CN(C(c2cccnc2)=O)C1 86004,c1(C(=O)NC2C(CNC(C(N3CCCCCC3)C)=O)C2)ccc2oc(S)nc2c1 86005,C1(C(=O)NC2CCC(C(N3CCC(c4cc[nH]n4)CC3)=O)C2)C2CC3C(C2)C13 86006,C1(O)(CC(=O)N(CCC(=O)NCCCn2ccnn2)CC=C)CCOCC1 86007,c1(C(=O)NC2CC(NC(c3cccc(C)c3)=O)C2)coc2c1N(C)C(=O)CCC2 86008,C(C)(C)(CC(C)NC(=O)CC1CCC(NC(=O)C(F)CC2CCOC2)C1)OC 86009,C1(CC(=O)NC(C#C)C(C)OC)CCC(NC(=O)C=C2CCC2)CC1 86010,CC(CC(C)(C)O)NC(=O)C(Cc1cn[nH]c1)NC(=O)CCc1cn[nH]c1 86011,S(=O)(=O)(c1ccc(C(C)C)cc1)NC1CN(C(CC(C)C)=O)CC1C#N 86012,C1(CC)CN(C(C2C3CC4C(C3NC(C3CCCN3C(N)=O)=O)C24)=O)CCCO1 86013,C(=O)(C#CC(C)(C)O)N1C(C(=O)NCCOC)CCC1C(C)C 86014,CC1C(NC(=O)CC(F)(F)Br)CCN1C(c1cnn(C)c1)=O 86015,c1(C(N2CC(CCCCNC(=O)C=C3CCC3)C2)=O)coc2c1CS(=O)(=O)C2 86016,C(CCCC(=O)NOCC1CCCO1)NC(C(CO)OC)=O 86017,N1(C(=O)NC)CCCC1C(=O)N(CCCN(C(=O)C(C)OCC(F)(F)F)C)C 86018,c1(C(=O)NC2CCCCN(C(c3cncc(OC)c3)=O)C2)onc2c1CCCC2 86019,c1(C(=O)NC(CC=C)CNC(=O)CC2CC2)c[nH]c2ccccc12 86020,N1(C(C(C2CN(C(c3csc(Cl)n3)=O)C2)OC)=O)CCC(N(C)C)CC1 86021,Cc1cccc(C)c1NC(=O)C1=CCN(C(C2COCC2C(N)=O)=O)C1 86022,CC(C)(CC(=O)N1CCCCC1CF)NC(=O)CSc1nc[nH]n1 86023,c1(C(N2C(CNC(c3c(C)ocn3)=O)CC(C)(C)C2)=O)cc(P(C)(C)=O)cs1 86024,CC1(CNC(=O)CC2(C)CC2(F)Cl)CCN(C(c2cnoc2-c2cccs2)=O)C1 86025,C1(C)(C(N(CCN(C)N(C)C)C)=O)CN(C=O)CCO1.C(C)(C)(C)OC(C)(C)C 86026,C(=O)(C1CCCc2nc(C)[nH]c21)N1CCCC(N2CCN(C(CCC)=O)CC2)C1 86027,c1(OC)cc(C(=O)NCC(C2CC2)NC(c2ccc(C)cc2)=O)c(N)cc1F 86028,N1(Cc2ccc(C(=O)OC)[nH]2)CCn2ncc(C3=CCSCC3)c2C1 86029,c1(C(N2CC3(CCCCN3C(=O)Cc3cnns3)C2)=O)ccc2ncccc2n1 86030,N1(C(c2c(=N)cc[nH]c2)=O)CCN(C(C2CC2=C2CCOCC2)=O)C2CC12 86031,N1(C(CC(C)OC)=O)CCOCC(C)(CNC(c2c(C)nsc2C)=O)C1 86032,CC1CC(NC(=O)CC(=O)NC2CC2)CN(C(c2cc(CCO)on2)=O)C1 86033,c1(C(N2CC(N(C(=O)COC(C)(C)C)C)C2)=O)cccc(CC2CC2)c1 86034,C1(CNC(N(CCC#CCC)C)=O)CCC(F)CC1 86035,C(=O)(C(O)C(C)c1ccccc1F)NCCN(C(=O)Cc1ccn(C)n1)CCC 86036,CC1(C)CN(C(=O)NC2CCN(c3ccc(C(F)(F)F)cc3)C2)C1(C)C 86037,Cc1cc(CC(=O)NC2CCCN(C(=O)Cc3cc[nH]c(=N)c3)CC2)cc(C)c1 86038,c1(NC(N(C(C2CCCC2)C)CCO)=O)ccc2nc(O)[nH]c2n1 86039,C1(CNC(c2c(C)cn(C(C)C)c2)=O)C(C)CCCN1C(c1ncccc1F)=O 86040,C(=O)(C1CCc2c[nH]nc21)N(C1CCCN(C(CC)C(=O)NCC)CC1)C 86041,N1(C(c2nc(C)on2)C)CCC2(CCCN(C(=O)CCc3ccncc3)C2)C1 86042,CCC(CC(C)C)C(=O)NCc1nocc1C(=O)N1CC(C)(O)CO1 86043,CCCC(C(=O)NCCC1CCN(C(c2ccnn2C(C)C)=O)C1)OCC 86044,C(=O)(C1=C(F)CN(C(C2(Cl)CC2(F)F)=O)CC1)NC(CCCC)COC 86045,C1(C(N2CC(CC(C#C)C)C2)=O)CC(C)N1C(=O)C(C1CC1)C1CC1 86046,C(=O)(C(CO)C(C)(C)C)NCC1N(C(c2cc(C)cc(C)c2)=O)CCC1 86047,N1(C(=O)Nc2c(F)ccc(C)c2)CCN(C(=O)C2=CCCCCC2)C(C)C1C 86048,N1(C(C2CC(C)(NC(c3cc(C(C)=O)[nH]n3)=O)C2)=O)CCC(O)(C(C)C)C1 86049,CC(C(C)(C)NC(=O)CC1(O)CCOC1)NC(=O)CC1CC1 86050,c1(C(=O)NC(C)CCCNC(c2[nH]cnc2C#N)=O)cnn2c1OCC(C)C2 86051,C1(NC(C)=O)CCN(C(=NCCCN2CCCC2)NCCC2=CCCCC2)C1 86052,c1(C(C)=O)cc(C(=O)NCC2CC2CNC(=O)CC2CCCC23CC3)n(C)c1 86053,C1(CCCC(=O)N(C)CCNC(c2cc(-c3ccoc3)[nH]n2)=O)CCCC(=O)N1 86054,C1(CNC(COC)=O)(NC(C2CCN(CC(C)C)CC2)=O)CCOCC1 86055,C(=O)(C(C)C(C)(F)F)NCC1(F)CC(CNC(C(C)C2CCC2)=O)C1 86056,C1(c2cn(Cc3c(C)c[nH]n3)nn2)CN(C(=O)C(=O)Cc2ccc(Br)s2)CCO1 86057,N1(C(C=CC)=O)C2CCC1CC(F)(CNC(C1(c3ccncc3)CC1)=O)C2 86058,c1(C(=O)NCC(CO)NC(C(COC)N(C)C)=O)ccc(=N)[nH]c1 86059,c1(C(=O)NCCC2(O)CCN(C(c3c(C)cccc3)=O)C2)ccc(S(C)(=O)=O)[nH]1 86060,C1(NC(c2n(CC)ccc2)=O)CC2C1CCN2C(c1cc2cscc2s1)=O 86061,c1(C(=O)NC(CCCC)CNC(=O)C(C2CCC2)OCC)occc1S(C)(=O)=O 86062,C(=O)(CCC(=O)NC1C=CC(CC(N2CCC(OCCO)C2)=O)C1)NCC 86063,c1(OC)cc(OC(F)F)nc(C(=O)OCC(N2CCCC(O)(C(F)(F)F)C2)=O)c1 86064,Cc1cc(C(=O)NC(CC(F)F)C(=O)NC(c2cncnc2)C)cc(C#N)c1 86065,CC(C)C(F)(CNC(C1(C)CCCCO1)=O)C(=O)NCC(C)(CO)CO 86066,N1(C(CC(C)SC)=O)CCC(CNC(=O)CCN2CCCCCC2)C(O)C1 86067,c1(C(C)C)ncc(Br)c(N2CC(C(C)NC(=O)CC3(C)CC3)C2)n1 86068,C(=O)(C1=NOC2(CCC2)C1)N1C(C(=O)NC2C(C)CC=CC2)C(C2CC2)CC1 86069,n1(CCC(=O)NCC2CN(C(C(COC)C)=O)CC2C)nc2ccccn2c1=O 86070,C(=O)(CCCCC(F)(F)F)N1CC(NC(C2CCN(C)C(=O)C2)=O)CC(F)(F)C1 86071,c1(C(N2C(C)(CNC(=O)CN3C(=O)CCC3=O)CCC2)=O)cnc2cccnn12 86072,C1(CNC(CCC2C(C)=NOC2=O)=O)(NC(=O)C#CC2CC2)CCC(F)(F)CC1 86073,c1(C(C)=O)ccc(C(=O)NCC(C)(C)NC(C2CCOC2C)=O)nn1 86074,C1(C(=O)NCc2c(CC)nns2)CCCCCC1NC(C1(C)CCC(=O)N1)=O 86075,C1(N(C)C(c2cnnn2C)=O)CCC(NC(=O)CCOCC2CCC2)CC1 86076,C=C(F)C1(CC(N2CCC(C(=O)Nc3ccccn3)CC2)=O)CCC1 86077,C1(c2nc(CNC(C3C(CC)C3)=O)[nH]n2)CCN(C(c2cc(=O)n(C)o2)=O)CC1 86078,c1(CC(=O)NC(C2CCN(C(c3cc(F)n(C)n3)=O)C2)C)nc(F)c(F)cc1F 86079,CCC1C(=O)N(CC)CCNCC(=O)N1.c1(SCC(C)(C)C)nc(C)cs1 86080,C(CC(=O)NCCn1cc(CC2(C(=O)O)CCCO2)nn1)(C1=CCCC1)OCC 86081,c1(C(=O)Nc2scc(CC(=O)Nc3cc(Cl)ncn3)n2)cccc(F)c1O 86082,n1(CCC)cc(NC(=O)CNC(=O)C(O)CN(C)C)cn1 86083,CC1(C)CC2C(CN1Cc1cc3cccc(Br)c3s1)C2(F)F 86084,C1(C(=O)NC2(CCNC(C3CC(C)OC3)=O)CC2)CC(=O)NC(=O)C1 86085,C1(C(=O)NC2CCC(NC(c3cc[nH]c3C3CC3)=O)C2)CC2(CCOC2)C1 86086,C1(C2CC2)(CNC(c2scc(C)c2Cl)=O)CCN(C(=O)C(C)(C)COC(C)C)C1 86087,c1(NC(CC(=O)N(CC#C)CC2CC2)=O)cc(C)nc2c(C)cccc12 86088,C=C=CCCC(=O)N1CCCCC1CNC(C12CCC1C2)=O 86089,N1(C(C2C(OCC)C2C)=O)CCCC(NC(c2conc2C2CCCC2)=O)C1 86090,c1(C(=O)NC2CCCN(C(=O)CC3CCCCO3)CC2)cncc2ccsc12 86091,N1(C(CCC(C)SC)=O)CC2(CCC2)CC1CNC(c1cc(C)ns1)=O 86092,C(=O)(C(CNC(=O)Cn1cnnc1C)CC(C)C)NCC(C(F)(F)F)OC 86093,C1(N=[N+]=[N-])(C(=O)NCC2CN(C(CSC(C)(C)C)=O)CC2O)CCOCC1 86094,N1(C(c2c(CC)nccc2)=O)CCN(C(C2CC3(CCO2)CC3)=O)C(C(C)C)C1 86095,c1(C(N(CCCNC(C(c2cccnc2)C)=O)C2CC2)=O)nocc1Br 86096,CCCCCC(C(=O)NCC1CC1NC(C1CCCN1C(=O)CC)=O)C(C)C 86097,C(=O)(C1CCCc2cncn21)N(C(C)CCNC(=O)C(CC1CC1)CC1CC1)C 86098,CCCCCCC(CC)N=c1cccc(S(=O)(=O)NCC2CN3CCC2CC3)[nH]1 86099,C=CCCC(F)(F)C(=O)NCC1CN(C(c2ncoc2C2CC2)=O)CC12CCC2 86100,c1(C(=O)NCC2(F)CN(C(Cc3scc(C)c3)=O)C2)cnn(C(C)C)c1F 86101,Cc1ccc(CC(N2CCOC(CNC(C3(C#N)CCCC3)=O)C2)=O)c(Cl)c1 86102,C(=O)(C1=CC2C=CC(C1)C2)NC(CC)(CNC(c1[nH]ccc1C)=O)CC 86103,C(CC(O)CC(=O)NCCC1CCCN(C(C)=O)C1)SC 86104,n1(CC)nncc1C(=O)NCCC1(OC)CN(C(=O)C(C)COC)C1 86105,c1(OC)cnc(C(=O)NC2C3CC(NC(C4CC(CC5CC5)C4)=O)CC23)cn1 86106,c1(C(=O)NCC(C2CCCC2)NC(CSCCCC)=O)cc2c[nH]nc2s1 86107,C(c1ccccc1)=C(C)C(N1CC(F)CC1C(=O)NCC(c1ccsc1)O)=O 86108,Cc1cc(C(N2CSCC2C(=O)NCC2CC2Cl)=O)cc(C)c1 86109,C(=O)(NNc1cc(F)cc(Cl)c1)c1cc(C(=O)O)c2c(c1)scc2 86110,c1(OCC#C)ccc(C(=O)NCC2CN(C(=O)C(c3ccc(F)cc3)F)C2)cc1 86111,N1(C(C2(C#N)CCOCC2)=O)CCN(C(=O)CC2CCCC(=O)N2)C2(CC2)C1 86112,c1(OC)cc(C(=O)NCC2CN(C(c3cccnn3)=O)CC2N(C)C)nn1C 86113,CC1=C(C)CC(C)(NC(=O)CC(C)(C)N(C(=O)CNC(=O)CN(C)C)C)CC1 86114,c1(CC)ccc(C(C)NC2C3CN(C(=O)CCC(=O)N(C)C)CC23)cc1 86115,CC1CCC(C(=O)NC2CC(=C3CC3)C2)N(C(C2CCCO2)=O)C1 86116,c1(OC(=O)CN(C(c2cn[nH]c2)=O)C(c2ccccc2)=O)ccc(I)nc1 86117,Cc1ccc2c(C(=O)N(C)CCn3cc(C4COC(C)(C)O4)nn3)ccnc2c1 86118,c1(N(CCN(C(C2(CCOC)CC2)=O)C)C)nc(Cl)sc1C 86119,C#Cc1cccc(C(=O)NC2(CNC(c3c[nH]nc3Br)=O)CC2)c1 86120,C1(C)(NC(c2cn(CCNC(C3(CC)CCCC3O)=O)nn2)=O)CCCC1(C)C 86121,Cc1sccc1C(=O)NCc1cc(C(=O)NCC(C)C(C)O)n[nH]1 86122,C1(NC(C2(CCC=C)CC2)=O)CN(C(c2snnc2C2CCC2)=O)CCC1CO 86123,c1(C(=O)NC2CC3CN(CC4CCc5ncnn54)CC23)cc[nH]c2nccc1-2 86124,Cc1c(C(=O)NC(c2cn(Cc3ccc(Br)s3)nn2)(C)C)ncn1C 86125,c1(CNC(C(C#C)(C)C)=O)ccc2c(c1)CCN(C(=O)C(C#N)C(C)C)C2 86126,C#CCC(CC(=O)Nc1cccc(OC)c1)NC(=O)CCC(C)(C)OC 86127,C(=O)(C(C)C(O)C(C)C)N1CCC(C(=O)NCc2snc(C)n2)C1 86128,c1(C(=O)NCC2CN(C(C3(Br)CC3)=O)CCO2)nc2ccccn2n1 86129,Cc1ccc(C(=O)NCC=C2CCN(C(=O)Cn3nnc(=N)[nH]3)CC2)cc1CO 86130,N1(CC)CCCC(NC(C2CCCN2C(=O)C(C)NC(N)=O)=O)C1 86131,CCCCC(CNC(C1(F)CCCC1)=O)NC(c1ccc(C(F)(F)F)cn1)=O 86132,c1(OC)cc(N(CC(C)NC(C2CC3C(C2)C3(C)C)=O)C)c([N+](=O)[O-])cc1OC 86133,N1(c2snc(CC)n2)CC(C)(C)CC1CNC(=O)CC(C)C1CCCCC1 86134,c1(C(N2C(CNC(C(=O)NCC)=O)CC(CCOC)C2)=O)ccc(=O)n(CC)n1 86135,c1(C(=O)NCC(CNC(c2cn(CC)nn2)=O)CO)c[nH]c2c(C)cccc12 86136,Cc1cc(S(=O)(=O)O)ccc1NC(C1CCC(C)N1C(=O)CCCCCCBr)=O 86137,N1(C(C2N(CC)CCC2)=O)CC(C2CC2C(=O)NCC(C)(F)C(C)(C)F)C1 86138,N1(C(CCCCC=CC)=O)CCC(C2CCN(C(=O)COCC(F)F)C2)C1 86139,c1(COC)n[nH]c(=NC(=O)N2CCOC(Cc3ccccc3)C2)s1 86140,c1(C(=O)NCC(C)(C2CC2)NC(=O)CSc2nnc(S)s2)cc(C(N)=O)ccn1 86141,C(=O)(C1=CCOCC1)N1CCC(CCNC(c2cccc(F)c2F)=O)C1 86142,C1(C(NOC(C)(C)CO)=O)CC2CN(C(C3(N4CCCC4)CC3)=O)CC2C1 86143,N1(C(C2CCCN(C(C(C)S(C)(=O)=O)=O)CC2)=O)CC2CC(C)(C)C2C1 86144,c1(CN(C(Cc2ccc(C)o2)=O)CCNC(C2COCCO2)=O)ccc(Cl)nc1 86145,c1(C(=O)NCC(C(C)C)(C)NC(=O)C=CC2CCC2)c(F)cccc1Br 86146,CC#CCC(C(=O)NCC(O)CC1CCC1)NC(=O)CCc1ncnn1C 86147,C(C1CSc2ccccc21)N(C(=O)N=c1nc(C(F)(F)F)[nH]s1)CC 86148,C(CCCCCC(=O)NC(C(F)(F)F)C1CC1)n1cc(COCC(C)O)nn1 86149,CCC(CC(=O)NC(C)C(C)C(=O)NCCc1cc(C)on1)C(F)F 86150,C1(O)(CN(C(=O)C(=O)NCC2CC2)C)CCN(C(=O)C(C2CCCCCC2)O)C1 86151,CCCC(C(=O)NC(C1(C)CCN(C(c2ccnc(OCCO)c2)=O)C1)C)OC 86152,Cc1ccc(C(C)C)c(C(N2CC3CC2CC3NC(=O)C#CC(C)C)=O)c1 86153,C1(NC(=O)CCCn2cc(C3(O)CC3)nn2)CCCC(CO)CC1 86154,c1(C(N2C3C(NC(c4ncncc4Cl)=O)CC(C3)C2)=O)cnc2cc[nH]c2c1 86155,C1(NC(C2(COC)CN(C(c3nnccc3C)=O)C2)=O)CN2CCC1(F)CC2 86156,N1(C(CC=CCC)=O)CCN(C(=O)CCC(=O)N(CCC)CCC)C2(CC2)C1 86157,C1(CNC(C(C)(C)NC(=O)NCC)=O)COCCN1C(c1cnc(OCC)s1)=O 86158,CC1CN(C(C2COCC(=O)N2C)=O)c2ccc(C(F)(F)F)cc2O1 86159,C(=O)(C#CC1CCCCC1)N1CC(C(=O)NCC2(CCOC)CC2)OC(C)C1 86160,CC1CC(CNC(C2(C)C=CCCC2)=O)CCN1C(c1cc2scnc2[nH]1)=O 86161,C(=O)(CCC(C)C)OC.C1(N2CC(C3C4CCC3(c3ccn(C)n3)C4)C2)CCCN(C)C1 86162,C(=O)(CC(O)CC(C)(C)C)N1CCCC(C(=O)NC2(C3CCCC3)CC2)(CC)C1 86163,c1(CC(C(=O)N(CC(CNC(COC(C)=O)=O)O)C)C)c(C)noc1C 86164,CCN=C(NC1CC12CC2)NC1CC(C(F)(F)F)C1 86165,Cc1cc2ccc(C(=O)NCC(C3CC3)NC(=O)CN3CCCC3C)cn2c1 86166,CC(C)(C)CCCCCC(=O)N1CCN(C(=O)C#CC2CCC2)CC1C(F)F 86167,O=C(C(O)C(F)(F)c1ccccc1)NCC1(C2CCCCN2)CC1 86168,C(c1cncnc1O)=CC(=O)N(CCCCNC(CC1C(C)OCC1)=O)C 86169,O=C(C#CC1CCCOC1)NCC1(C(N)=O)CN(C(=O)CN2CCCCC2=O)C1 86170,Cc1cc(Cl)cc2cc(C(N3CCC(C)C3CNC(C3(CO)CC3)=O)=O)[nH]c12 86171,C1(C(=O)NCCCCOCC)(CO)CCN(C(C2CCC(O)CC2)=O)C1 86172,c1(OCC=C)cccnc1C(=O)NCCC1CCC(NC(c2cc(C)co2)=O)C1 86173,C(CN=c1[nH]c2ccc(S(=O)(=O)NC(C)CC#N)cc2s1)c1nccc(OC)n1 86174,c1(C(N(C(C)CNC(=O)Cc2cccc(OC)c2)CC)=O)cc2sccc2[nH]1 86175,Cc1nc(NCC2CCCCN(C(c3cc(CF)on3)=O)C2)ccc1[N+](=O)[O-] 86176,C=C(C)CC(C(=O)OC)NC(C1CC=CC(n2cc(C(CCC)OC)nn2)C1)=O 86177,C1(CC)CN(C(=O)C=C(C)C)CCC1NC(C1CC(F)(F)C1(C)C)=O 86178,CC1CC(=O)NCC1C(N1CCCN(C(=O)CCC23CCC(CC2)C3)CC1)=O 86179,N1(C(C(=O)NCSc2cccc(F)c2)C2C(C)C2)CCC(C(N)=O)CC1 86180,C1(NC(=O)Cc2ccc(Cl)nc2)CN(C(C2(F)CCC2)=O)CC2(CC2)C1 86181,CC1CN(C(=O)CC2(N(C(=O)C(n3cc(Cl)cn3)C)C)CC2)CC1N(C)C 86182,C1(NC(CC(C)OC)=O)C2CC1N(C(=O)CCc1cncn1C)C2C 86183,C1(OC)CC(CNC(=O)CCCc2ccc(Cl)cc2)N(C(C2CC(C#N)C2)=O)C1 86184,C1(NC(CC(CC=C)NC(c2cncc(C)c2)=O)=O)COC2(CCCC2)C1 86185,N1(c2cccc(S(=O)(=O)NCCC(=O)NC(C)C)n2)CCCC2(CCN(C)C2)C1 86186,C1(N(C)C(c2n[nH]cc2Cl)=O)CCCN(C(C2CC23CC3)=O)CC1 86187,C1(CNC(c2ccc(N(CC)CC)nc2)=O)CN(C(C2CC2C)=O)C(C)(C)C1 86188,C1(NC(c2ccc(COC)[nH]2)=O)CC2CC(C1)N(C(=O)CC1NC(=O)NC1=O)C2 86189,c1(NS(C)(=O)=O)ccccc1NC(=O)C(N1CCCCC1CO)=O 86190,c1(CC(C)OCCNC(CCOCCCOC)=O)ccccc1 86191,N1(C(CC2(CSC)CC2)=O)CCCN(C(=O)Cc2ccnn2C)CC1C 86192,N1(C(CCCC2(NC(=O)C=C(C3CC3)C3CC3)CCC2)=O)CCOCC(C2CC2)C1 86193,c1(C(C)(C)C)noc(CCC(=O)NCC2(NC(c3cc(C(F)F)no3)=O)CC2)n1 86194,C12(C(N(CCOCC)CC)=O)CC(CN(C(C3CCSC(C)C3)=O)C1)C2 86195,N1(C(c2c(C)cc(=O)n(C)n2)=O)CCC2CN(C(c3cnc[nH]3)=O)CC2C1 86196,C(=O)(CCCNC(=O)CSC1CC1)NC(C1CCC1)C 86197,c1(C(=O)NCCNC(c2c(C)nccc2Cl)=O)ccc([N+](=O)[O-])c(S(N)(=O)=O)c1 86198,N(C(=NC(C)CN(C)C)N(C)Cc1ccccc1)C(COC)C 86199,Cc1ccc(Cl)c(C(=O)NC(CNC(C2(C(F)F)CC2)=O)CC(C)C)c1N 86200,c1(C(N(C)CC2N(C(CCC=C(C)C)=O)CCC2)=O)ccc2c(c1)ncn2C 86201,C(C)(N=c1[nH]c2c(c(=NCCN(C(=O)N(C)C)CO)[nH]1)COC2)c1cc(C)c(F)cc1 86202,C1(NC(C2(C(=O)OCC)CCC2)=O)CC2CCC(C1)N2C(=O)C(C)CC(F)(F)F 86203,N1(C(C=CCCC)=O)CCCC(CC(=O)Nc2cnn(CCC)c2)CC1 86204,C1(C2CCC2)(C(N(CC)CC2CCN(C(=O)OC(C)(C)C)C2)=O)OCCO1 86205,CC1CN(C(=O)CC2CCOC2)CCC1N(C(=O)C1CC1)CCOc1ncccn1 86206,C1(C(=O)NCC(C)N(C(c2[nH]cc(C)c2)=O)C)CCCCN1C(C1CCCC1)=O 86207,c1(C(N(C(C)CC(=O)NOCC(=O)N(C)C)C)=O)cc2cc[nH]c2cn1 86208,C1(NC(C(CC)(C)F)=O)COC2(C1)CN(C(=O)C(C)(C)C(=O)OC(C)(C)C)C2 86209,C1(C(=O)NCc2ncc(C(N3CC(OC)(CO)C3)=O)cn2)CCOCC1(C)C 86210,N1(C(c2ncc(OC)cn2)=O)CCC2(C1)CN(C(c1cc(Cl)c(Cl)s1)=O)C2 86211,c1(OC)ccc(F)c(NC(=O)C(C)(CSC)NC(=O)CC(C)C)n1 86212,C1(CC(=O)NCC2CC(NC(=O)Cn3cnnc3)C2)CC2(CCC2)CCO1 86213,Cc1cc(C(N2CC(O)(C(C)NC(=O)CC(c3ccccc3)N(C)C)C2)=O)co1 86214,N1(C(C2(C)CC2)=O)CC2(CCN(C(C3(c4cccnc4)CCCCC3)=O)CC2)C1 86215,c1(OC)ccc(CNc2cccnc2C(N2CCc3sccc3C2)=O)c(F)c1F 86216,C1(CCNC(c2n(C=C)nnc2)=O)CCCN(C(=O)C(F)CC2CCOC2)CC1 86217,C1(CNC(c2nc(C)[nH]n2)=O)(NC(c2cnc(C(F)F)nc2)=O)CCCCC1C 86218,CC1(C)C(CC(=O)NC2(C)CCN(C(c3ccccn3)=O)C2)C1(C)C 86219,N1(C(CC(CC)SC)=O)C2CC=C(C(=O)NCC3C(C)C3(F)F)C1CC2 86220,N1(C(C(C(C)C)CO)=O)CC2(CCC2)CC1CNC(c1ccc(C(N)=O)cc1)=O 86221,c1(CN(C)C(C2COCC2(C)C)=O)cncc(O)c1 86222,C12(CNC(C3(CCCC)CC3)=O)CCC1CN(C(=O)C=Cc1ccc(C)s1)C2 86223,N(C(=NCC1C(C)C1C)NCC1(OC)CCC1)CC(C1CC1)OC 86224,C1(F)(C(=O)NCc2occ(C(=O)NC(CCC=C)C)n2)CCCCC1 86225,c1(NC(C2CCC(NCc3nc(COCC)on3)C2)=O)cccc(C#N)c1 86226,CC(CC(=O)NCC1(F)CN(C(C2(F)CCOC2)=O)C1)c1ccncc1 86227,CCCCCCCCCC(=O)N1CC(C)(NC(=O)C(c2ccccn2)O)C1 86228,N1(CC)CCN(CC2(C(=O)Nc3ccc(-c4nn[nH]n4)cc3)CC(F)(F)C2)CC1 86229,C12CCCCC1C(=O)N1CC(C1)C(=O)N2C.C(CCN=[N+]=[N-])NC(=O)CSC1CC1 86230,C1(CNC(c2cnnc(O)c2)=O)CCN(C(c2ccccn2)=O)CC1O 86231,Cc1ccc(CC(=O)N(CCNC(=O)C(C)(C)c2cscn2)C(C2CC2)CO)cn1 86232,C(=O)(C(C)C(CC)CC)N(C1CCN(C(c2c(CC)n[nH]c2)=O)C1)CC 86233,N1(C(c2c(C)nc(C)s2)=O)CC(NC(=O)COCC(F)F)C(C2CC2)C1 86234,c1(N(CCNC(=O)C(C)CC2CCC2)CC)ccc(F)cc1C#N 86235,C1(NC(c2nc(C(C)C)sc2)=O)CCCC1(C)NC(=O)C(C)C1CC1 86236,c1(C(=O)NCC2CC(O)(CNC(C3(COC)C=CCC3)=O)C2)ccc(C)nc1C 86237,Cc1[nH]c(=N)nc(O)c1CCC(=O)NCC1CN(C(=O)CCC2CCCCO2)C1 86238,c1(NC(C2C(C(=O)Nc3ccc(N(CCO)CC)cc3)C2)=O)c(Cl)nc(C)nc1Cl 86239,C1(OC2CC(Cn3cc(-c4ccn(C)n4)nn3)C2)CCN(C(N)=O)CC1 86240,n1(C(C)C)cnc(C(=O)NC(C)(C)CN(C(=O)Cc2cncs2)C)c1 86241,N1(C(c2n(C3(C)CC3)ncc2)=O)CCCC(N(CCO)C(C2CCC(=O)O2)=O)C1 86242,N1(C(C2C(C)C2C)=O)CCN(C(=O)C(Cl)=CCl)CCC1C 86243,C1(NC(c2cc(C)n(C)n2)=O)CN(C(=O)C(Cl)=CCl)C2(CCCCC2)C1 86244,N1(C(C(CSC)C)=O)CCN(C(C2CN(C3CCCCC3)C2)=O)CC1C 86245,C(C(C)(C)CC(=O)N1CCCC(CC(N)=O)C1)NC(C=CC)=O 86246,C(CCCC#N)(c1nnnn1C1CC1)NC(c1ccc(N2CCCCC2)cc1)C 86247,c1(CC(=O)NCC(CC)NC(=O)C(C2CC2)C2CC2)ccccc1CO 86248,N1(C(Cc2c(COC)cccc2)=O)CCN(C(=O)C2=NOCC2)C2CC12 86249,C12(C(=O)NCC(C)(O)CCO)CCC1CN(C(=O)CCOCC(F)F)C2 86250,CCCC(CNC(C1CSCCN1C(c1cocn1)=O)=O)CCO 86251,c1(C(N2C(CN(C(CC(C)SC)=O)C3CC3)CCC2)=O)sc2nccnc2c1N 86252,C=CCC(CNC(c1nc[nH]n1)=O)C(=O)NCCOC1CC1(F)F 86253,N1(C(C(CC)N(C)C)=O)CC(NC(c2ccnc(OC)c2)=O)C2CCCCC12 86254,N1(C(c2c(C)cco2)=O)CCC(N=[N+]=[N-])(C(=O)N(C)CC2CC2(C)C)C1 86255,c1(NC(C(C2CCC2)NC(c2cc(COC)[nH]n2)=O)=O)cncc(SC)c1 86256,C12(C(=O)Nc3cccc(C)c3)CCCC1CCN2C(=O)C(C)Oc1ccccn1 86257,CCN=C(NCCCC(C)(F)F)NCCC1CCCC1(C)C 86258,Cc1ccc(C(=O)NC(CC(=O)NCc2c(F)cncc2F)C(C)C)c(C)n1 86259,C1(CNC(=O)C#CC2CCC2)CCC2(CO1)CC(NC(=O)COc1ccon1)C2 86260,N1(C(c2cnc(C(C)C)nc2)C(=O)Nc2c(C)cccc2)CC2CC3CC2C1C3 86261,c1(C(N2C(C)CC2C(=O)NC2(CO)CCC2)=O)cc[nH]c(=N)n1 86262,c1(OC)ccc(C(N)=O)cc1C(=O)NCC(C)(C)NC(=O)C=CCO 86263,Cc1cc(C(=O)NC(C2CCCCC2)CNC(C2CC(=O)N2)=O)ccc1[N+](=O)[O-] 86264,c1(OC)ccc(C=CC(=O)NC(C)CC2CN(C(=O)C(C)C(C)(C)C)C2)cc1F 86265,c1(C(N2CCCCC(NC(C3C(C)C3)=O)C2)=O)cccnc1S(=O)(=O)C(F)(F)F 86266,c1(CC)ncccc1C(=O)N(C1CCC(NC(c2cccnc2)=O)C1)C 86267,c1(SC)ncc(C(=O)NC2CC(NC(C3(n4ccnn4)CC3)=O)C2)c(O)n1 86268,c1(C(=O)NC(C(=O)NC2CC(C(C)C)OC2)CC2CC2)ccn2ccccc12 86269,c1(C(N(C(CNC(c2c(C)ccc(Br)c2)=O)C)C)=O)coc2c(C)cccc12 86270,C=C(C)CC(C(=O)N(C1CCCN(C)C1)C)NC(c1cc(OC)ccn1)=O 86271,CC1CC(NC(c2cccc(=O)o2)=O)CN1C(=O)Cc1ccccc1Br 86272,N1(C(=O)COCCOCCO)CC(NC(c2c(N)cccc2F)=O)CC(O)C1 86273,Cc1ccc2sc(N3CC(CC(C)NC(=O)C(C)(O)C4CC4)C3)nc2c1 86274,c1(C(N2CC3C(CNC(CC(C)(C)C4CC4)=O)(C3)C2)=O)cc(O)ccc1Cl 86275,S(=O)(=O)(c1cnc(NCC23CCCC2OCC3)c(Cl)c1)NCCCN(CC)CC 86276,c1(C(=O)NC2CCN(C(CCC(=O)NCC)=O)CC2F)cccn2c(C)nnc12 86277,c1(OC)c[nH]ccc1=NC(=O)CC1CC(OC(C2CN(C(C)=O)CCO2)=O)C1 86278,CC(F)(F)CCNC(=O)CC1CCN(C(=O)CSCC(N2CCCC2)=O)C1 86279,CC1(NC(c2coc(Br)n2)=O)CCN(C(=O)CCCn2ccccc2=O)C1 86280,N1(C(CCC(=O)OCC)=O)CCC(CO)C(NC(=O)CCCn2ccnn2)C1 86281,N1(C(C(CC)O)=O)CC2CC3CC2C1C3NC(=O)CCc1cscn1 86282,N1(C(C=C(C)Cl)=O)CC(NC(=O)C(c2ccnn2C)O)C(O)C1 86283,N(C(=NCCC1CS(=O)(=O)C1)NCc1cccs1)Cc1onc(C(N(C)C)=O)n1 86284,c1(CC(=O)N(CCC(C)NC(c2c(OCC)cccn2)=O)C)cc(C)cc(C)c1 86285,N1(C(CCCC)=O)CC2CC(NC(c3ccc(CCF)cc3)=O)C1C2 86286,C1(C(=O)O)CCCC(CNC(c2occc2-c2ccccc2)=O)C1 86287,c1(C(=O)NC2C(CNC(c3cccc(C(=O)NC)c3)=O)C2)ccc(Cl)c(N)c1Cl 86288,N(C(=NCCF)NC1C(C)(C)C1(C)C)CC(c1ccc(Cl)cc1)OC 86289,c1(CC)ncncc1C(=O)NCCC(C)NC(=O)CCS(C)=O 86290,CC(C)(CCCNC(=O)CC(F)(F)F)C(=O)NCC1CCC(F)C1 86291,c1(OC)cc(C(=O)NC(C)(C)CCCNC(C23CCN(CC2)CC3)=O)cc(F)c1 86292,c1(N2CCC(CSC)C2)nccc(=NC(C)COC2CCCC2)[nH]1 86293,N1(C(=O)NCC2(C)COC2)CCC(O)(C(F)(F)C(N)=O)C1 86294,CN(Cc1cc(-c2cccc(Br)c2)no1)N1CC(Cn2cc(Br)cn2)C1 86295,N1(C(C2C(COC)CC2)=O)CC2CC2(NC(C2CC(C(C)C)C2)=O)C1 86296,c1(C(N2C(C)C(=O)NCC2)C(=O)NCc2ccco2)cc2ccccn2n1 86297,N(C(=NCCCC(C)(F)F)NC(C)C1CC1)C(c1cccnc1)C 86298,C1(CNC(CC(=O)OC)=O)CN(C(=O)CCn2cccnc2=O)CCC1C 86299,c1(OC)cc(Cc2nc(C(N)C(C)(C)C)n(-c3c(F)cccc3Cl)n2)ccc1C 86300,C(N=c1ccn(CCC#N)[nH]1)(c1ccn(CCC)n1)c1nnnn1C1CCOC1 86301,FC1(F)CCC2C(CCCN2C2CC(=O)N(c3ccccc3)C2)C1 86302,c1(-n2cc(CC(CC(=O)OCC)N)nn2)cccc2ccsc12 86303,C(=O)(C1=COc2ccccc2O1)N(C1C2CN(C(C3CCC3)=O)CC12)C 86304,N1(C(c2c(CC)nn[nH]2)=O)CCC(C(C)C(=O)NC2(C(N)=O)CCOC2)CC1 86305,c1(C(N2CC(C(C)NC(C3(CC=C)CC3)=O)OCC2)=O)cc2c(cn1)OCCO2 86306,C=C(Br)CCC(=O)NC1CCC(CNC(c2ccc(C(F)F)nc2)=O)C1 86307,Cc1c(O)c(=O)ccn1CC(N1CC2CC(NC(=O)C(F)C3CC3)C1C2)=O 86308,c1(C(=O)NCCC2CC(NC(C3C(C(C)=O)C3)=O)C2)c(C(N)=O)cnn1C 86309,Cn1cc(-n2cc(C3CC(NC(c4cc[nH]n4)=O)C3)nn2)cn1.C1(CO)CCC1 86310,C(CC(C(C)(C)C)NC(=O)C(C)OC1CCOC1)N(C(c1c(C)noc1N)=O)C 86311,CC(C)(CC(=O)N1CC(NC(C2CCCCN2N=O)=O)CC(F)C1)CC(F)F 86312,C1(NC(C(C)O)=O)CC2(C1)CC(NC(c1c[nH]cc(F)c1=O)=O)C2 86313,c1(C(N(C(C)CNC(C2CCCN2c2ncccn2)=O)C)=O)ccnnc1S 86314,C1(NC(C(CCC)F)=O)Cc2ccccc2C1NC(=O)CC1C=CCC1 86315,CC(Cc1ccccn1)N=c1[nH]c(=NCCN2CCC(O)C2)c2sccc2[nH]1 86316,N1(C(c2cnc(OCC)nc2)C(=O)NC(C)(C)C)CCN(C)C(CC)C1 86317,c1(C(N(C)CC2N(C(C(C(C)C)SC)=O)CCOC2)=O)ncnc2c1ccn2C 86318,c1(C(=O)NC2C(NC(Cn3ncn(C)c3=O)=O)CCC2)c(N)ccc(F)c1F 86319,C(C(C(=O)N1CCC1CNC(c1ccc2c[nH]nc2c1)=O)C(F)(F)F)OC 86320,c1(C(N(C2C(C)CCN(C(=O)CC3(C)CC3)C2)C)=O)ccc(Cl)c2ccccc12 86321,C1(NCCC(C)(C)OC)CCC2CN(C(=O)CCC=C(C)C)CC2C1 86322,C#CC1CN(C(=O)CCc2nncn2C)CCN1C(=O)COCCN(C)C 86323,N12CC(C(C)(C)C1)CNc1cnn(c1)CC2=O.C1(C(=O)OCC)CCCC(C)C1 86324,C1(C(=O)NC2(C)CN(C(C3(CC=C)CCOC3)=O)C2)CC2CCC(C1)C2 86325,N1(C(c2cnc(C)o2)=O)CC=CCC1C(=O)NC(C)C1CC1 86326,c1(CC(=O)N(C)CC2CCCN2C(=O)CN2CCOC2=O)c(F)cccc1Cl 86327,c1(OC)ccc(C(=O)NCCC2CCN(C(C3(C(C)C)CC3)=O)CC2)nc1 86328,C(=O)(C1=CCCOCC1)N1CCC(CC#C)(C(=O)NCc2ncc(CO)o2)C1 86329,C1(CNC(C(N2CCCCC2)C)=O)N(C(=O)CSc2nncn2C)CCC1(C)C 86330,C(=O)(C1=NNC(=O)CC1)NC(CC)(CNC(=O)Cc1ccccc1SC)CC 86331,N1(C(c2cc(CN(C)C)on2)=O)CCC2CN(C(=O)Cn3ccnn3)CCC2C1 86332,N1(C(c2c(CC)n(CC)nn2)=O)CC(O)(C2(CNC(C3CC(C)CO3)=O)CC2)C1 86333,c1(CC(N2C(CN(C(COCCOC)=O)C3CC3)COCC2)=O)cc(C)ccc1O 86334,CC(C)C(C(C1CCCCC1)NC(=O)COCCF)NC(c1ocnc1C1CC1)=O 86335,C1(C(=O)NCC2CC(CNC(C(C)OCC#C)=O)C2)CCc2nnnn2C1 86336,c1(C(N(C2CCN(C(=O)C(C#N)CC)C2)CC#C)=O)cn(C)nc1CC 86337,C1(C)(C(N2CCC(N(C)C)CC2)=O)CCCN(Cc2scnc2Cl)C1 86338,C1(NC(CN(c2ccccc2)CC)=O)CCC2CNCCC2C1 86339,Cc1cccc(C)c1C(C)OCc1cc(Br)sn1 86340,N1(C(CN(C)CC)=O)CCC2CCCC(C1)N2C(c1cc2c(nn1)CCCO2)=O 86341,c1(C(=O)NC23CCN(C(CC4(C)CCCC4)=O)CC2C3)cc(F)c(F)cc1F 86342,N1(C(C(COC)OC)=O)CC(C(=O)N(CCCO)C(C)C)C(C)C1 86343,C1(C(=O)NCC2C(CNC(Cc3ccn(CC)n3)=O)C2)C(C)(C)C1(C)C 86344,N1(C(CSCCC(C)C)=O)CC=C(C(C)(C)C(=O)NCCc2ncc[nH]2)C1 86345,c1(C(=O)OC)cc2n(n1)CCCC2NCc1ncoc1C(C)C 86346,c1(C(=O)NCC2(NC(C3CCS(=O)CC3)=O)CCC2)ccc(F)cc1[N+](=O)[O-] 86347,C12(CNC(C(CCC)C#N)=O)CN(C(c3c[nH]nc3C(F)F)=O)CC1CCO2 86348,Cc1nc2cncc(C(N3CCC4CN(C(c5cnsc5C)=O)CC4C3)=O)c2[nH]1 86349,CC(C)CCCCNC(c1ccn(CCNC(C2CC3(CC3)C2)=O)c1)=O 86350,C1(NC(CC2(OC)CCCC2)=O)COCCC1NC(C1CCC(C(C)C)CC1)=O 86351,c1(C(=O)NC(CC(C)NC(C2C(C)C2)=O)C)n[nH]c2c1CC(C)CC2 86352,C(CNC(=O)CCC1CC1C)(C(C)(C)C)NC(c1cc(CCCCC)[nH]n1)=O 86353,c1(-c2n(C)nc(CO)n2)cc2c(s1)C(C)(C)CCC2 86354,C=CC(C)CC(=O)NC1CC(CNC(c2ccccc2OC(F)(F)F)=O)C1 86355,c12cc(ccc1F)C(=O)N2.C(CCCCNC(=N)N)OC 86356,Cc1cc(C(=O)NC2CCN(CC34CC(c5ccccc5)C3C4)CC2)ncc1N 86357,N1(CNC(=O)C(=O)Nc2cccc(OC3CCCCC3)c2)CC(COC)CC1=O 86358,N1(C(c2c(C)n[nH]c2C)=O)CCC2(CCNC2)C1 86359,c1(C(=O)NC(CC=C)CNC(=O)CC(C)(C)C#N)cc2c(C)cc(OC)cc2o1 86360,c1(C(=O)NC(CC)(C)CNC(=O)C#CC(=O)N(C)C)n[nH]c2ccc(O)cc12 86361,N1(C(C(COC)OC)=O)CCOCC(NC(=O)CCCCCO)C1 86362,C1(O)(CC(=O)NCCCCNC(CSc2nc(C)[nH]n2)=O)CCCOC1 86363,Cc1ccc2c(C(=O)NCCCNC(=O)C(F)=CCCF)cnn2c1C 86364,CC1CC(C(N2CCOC(CCF)C2)=O)N(C(=O)CCC2(C#N)CCC2)C1 86365,C=CC1(CC(=O)NCC(C)OC(F)F)CN(C(c2c[nH]ccc2=O)=O)C1 86366,c1(N2CCCCC(NC(CC(=C)C)=O)C2)nccc(S(C)(=O)=O)n1 86367,c1(C(=O)OC)cccc2c(C(=O)NCC3CCCCC3C)cccc12 86368,N12CCCC(C1)N(C(C1COC(=O)N1)=O)C(CSc1ccccc1)C2=O.CO.OC 86369,C1(CNC(CC=C)=O)CCN(C(=O)CCc2nc3ccccc3o2)C12CCC2 86370,C(=O)(CC(C)(C)C=C)N(C(CC(=O)N1CCC(OCC=C)C1)CC)C 86371,N1(C(C(C(=O)OCC)(C)C)=O)CCc2sc(CNC(=O)CS(N)(=O)=O)nc2C1 86372,N1(C(=O)OC(C)(C)C)CC2(CCCN(Cc3ccc(F)c(O)c3)C2)C1 86373,C1(CCC(=O)N(CC)Cc2cnn(C)c2)CCCCN1C(C1C=CCCC1)=O 86374,c1(C(=O)OCC)nn(C)[nH]c1=NC(=O)c1noc(C)c1I 86375,N1(Cc2c(C(=O)OCC)ccs2)C(C(=O)Nc2cnnc(OC)c2)CC2CC12 86376,CC1(C)NC(=O)CCC1NC(=O)NCC1CCN(CC2CC(F)(F)CS2(=O)=O)C1 86377,C1(NC(=O)C=CC2CCC2)CCC12CN(C(C1CCN(C3CC3)C1=O)=O)C2 86378,C=CC(O)C(=O)NCC1CCC(NC(=O)CN(C(=O)COC)C)C1 86379,O=C(CCC(CF)CF)NCC(c1ccc(F)cc1)NC(=O)CCc1ccc[nH]1 86380,N1(C(CCCC#CC)=O)C(C(=O)N(CC(C)C#N)C2CC2)C2CC(O)C1C2 86381,c1(C(=O)Nc2c(NCCC)ccc(C(=O)O)c2)cccc(S(N)(=O)=O)c1 86382,C1(C(N(CCN(C(c2cc(C(C)(C)C)on2)=O)CC)CC)=O)CCc2nnnn2C1 86383,CC1CN(C(=O)Cc2n[nH]cc2Br)CC1CNC(=O)CCc1cncn1C 86384,c1(C(N2C(C)C(C)N(C(C3CC(=O)CCO3)=O)CC2)=O)cn2cc(Cl)cnc2n1 86385,c1(C(=O)NCC2CC(OC)CN2C(=O)CNC(=O)C2CC2)cc(C)n(C)c1C 86386,c1(CC)nc2c(C(=O)OCC#Cc3ccc(Cl)cc3)ccnc2[nH]1 86387,C(=O)(CCCC(=O)OC(C)(C)C)NC(CNC(C1CN(C(C)C)C1)=O)(C)CO 86388,C1(CNC(C2(C(=O)OCC)CCCC2)c2nnnn2C2CC2)CCOC(C)(C)C1 86389,CCC(F)(F)CC(=O)NC1CCCC(NC(c2ncccc2NC(C)=O)=O)CC1 86390,c1(C(N2C3CCC(NC(C=CC=CCC)=O)C(C3)C2)=O)cnn2ccc(O)nc12 86391,c1(NC(C2CC3CC3N2C(=O)CC2CCCCO2)=O)ncc(Br)nc1Br 86392,Cc1cc(=NCCN2CCC(N(C)C)C2)[nH]c(NC2CCC3(C(C)C)CC23)n1 86393,c1(SCC)cc(C(F)(F)F)ncc1C(=O)NC1CC1c1ccsc1 86394,c1(OCCN)ccc(=NC(=O)N2CCS(=O)(=O)C(CO)C2)[nH]n1 86395,C1(CC(=O)NC(C2CCCN2C(c2c[nH]nc2C(F)F)=O)(C)C)CCC2CC2C1 86396,C1(NC(c2cc[nH]n2)=O)CCCC(NC(C23CSC(C2)C3)=O)C1 86397,N1(C(CC2COCC(C)(C)O2)=O)CCc2ccccc2C(NC(C2COC2)=O)C1 86398,c1(NC(=O)NC2CC(c3ccc(Cl)cc3)C2)ccc2nc(O)sc2c1 86399,CC1NC(=O)C(C)N(CC(c2nccn2-c2ccccc2)=O)C1C 86400,c1(NC(=O)NCC2CCCN(CC(F)(F)F)C2)snc(-c2ccccc2)c1C#N 86401,N1(C(CN(C(C(C)C)=O)C)=O)CCCCC(C(=O)NOCC=CCl)C1 86402,C#Cc1ccc(C(=O)NCC(C)(C)CNC(c2c[nH]cc2C2CC2)=O)nc1 86403,N1(C(C(C)NC(C)=O)=O)CCCC(CCNC(c2conc2C(C)(C)C)=O)CC1 86404,Cn1cc2ncc(C(N3CCN(C(=O)CC4CCCO4)CC3)=O)cc2n1 86405,C1(c2n(C)cnc2)CN(C(C2(C)CNC(=O)C2)=O)CC1NC(=O)C=CC(F)(F)F 86406,c1(C(N2CCC(OC)C2)C(=O)NCCSC2CCOCC2)ncc(C)cc1C 86407,Cc1noc(C(=O)NC(Cc2ccccc2)C(=O)O)n1 86408,CN1CC2CCC(C1)N2C(C1CCN1C(c1cc(-c2ccncc2)no1)=O)=O 86409,C(C(C)(CC)C(=O)N(C)CC1CCN(C)C1)NC(CC1(CSC)CC1)=O 86410,C12(NC(C3C=CCC3)=O)CC3CCC(C1C2)N3C(=O)Cn1ncc2ncccc12 86411,C(CCCCC(=O)N1CC(N2CCN(C(=O)COC3CCOC3)CC2)C1)OCC 86412,C(=O)(C1CCCc2scnc21)NCC(C)(C)Nc1nc(Cl)nc2c1CCC2 86413,N1(c2nnc(CCC)s2)CCN(C(c2ccc(CCC)[nH]2)=O)CC(C)(F)C1 86414,CCCC(C(O)C(=O)N1CC(N2C(=O)CCC2=O)C1)NC(C12CCCC1CCC2)=O 86415,N1(C(c2cc(CC)no2)=O)CCOC(CCNC(C2CCCN(C(N)=O)C2)=O)C1 86416,C1(CC(=O)NCC)CN(C(=O)Cn2ccc(C)c2)CCO1 86417,Cc1cc(CNC(C2CC(C)CN(C(c3c[nH][nH]c3=N)=O)C2)=O)cc(F)c1 86418,N1(CC)C(C)CN(Cc2c(OC)nsc2OC(C)C)CC1C 86419,CCCC(CNC(c1cc[nH]n1)=O)C(=O)N1CCCC1C1(CC)CC1 86420,N1(C(C2C(CCC)CN(C(C3COC(=O)N3)=O)C2)=O)CCn2nccc2C1 86421,c1(C(N2C(CNC(=O)CCC(C)C)CC(OC)C2)=O)nccc2c(F)cccc12 86422,C1(C2CCCCC2)(C(=O)NCC(CNC(c2ncn(C)n2)=O)OC)CCCCC1 86423,c1(CN2CCC(C)C(C)(C)C2)ccc2cc(F)cc(Br)c2n1 86424,C1(C(N2C(C3(N4CCN(C)CC4)CC3)COCC2)=O)CC2CCCC2C1 86425,N1(C(c2ccc(F)c(Br)c2F)=O)CCOC2CCNCC12 86426,Cc1nn(C)c(=O)c(C(N2CC(F)(CNC(=O)C(n3cc(Cl)cn3)C)C2)=O)c1C 86427,Cc1c(C(=O)NC(CNC(c2ccsn2)=O)CO)cnc2ncnn12 86428,C1(NC(C=CC(=O)N(C)C)=O)C=CC(C(=O)NCC(F)Br)C1 86429,c1(SC)cnn(C)c1C(=O)N(CCCNC(=O)C(c1ccc(C)s1)C)C 86430,c1(C(N2CC3CC2CN3Cc2cscc2Br)=O)cc2n(n1)CCC2 86431,C12(CNC(C3(SCC)CC3)=O)CCC1CN(C(=O)Cc1ncsc1Cl)C2 86432,CC(C)(CO)C(=O)NC1CC1NC(c1ncoc1C(C)(C)C)=O 86433,C=C(Cl)CC(C(=O)NC1CCC(=O)NC1)NC(=O)C(F)CCC 86434,Cc1c(C(=O)NC(C)C(CO)NC(C2(C)CC(C)C2)=O)cnn1C(C)C 86435,C1(NC(c2c(C)n(CC(F)F)nc2)=O)CC2(CCN(c3ccnc(C#N)n3)C2)C1 86436,Cc1nc(NCCc2nnc3n2CCS3)cc(=NC(C)c2cc[nH]n2)[nH]1 86437,Cc1cccc(C(O)C(N2CC(C)(NC(c3cncc(N(C)C)c3)=O)C2)=O)c1 86438,N1(C(C(C(C)(C)C)O)=O)CCN(C(=O)CC2=NNC(=O)C2)C2COCC12 86439,c1(COC(=O)CC2CC2(Cl)Cl)c2c(coc1=O)CCCC2 86440,N1(C(C2N(CC)CCC2)=O)C2CCC1CC(C(=O)NCC(F)C1CCC1)C2 86441,c1(C(=O)NCC(CNC(c2cncc(C)n2)=O)OC)c[nH]nc1[N+](=O)[O-] 86442,C12(C(N(C(C)C)C)=O)CC1CN(C(=O)CN1CCN(S(C)(=O)=O)CC1)C2 86443,Cc1nncn1NC(=O)C1CC(NC(c2csc(CO)n2)=O)CCO1 86444,CC1CCN(C(c2c(F)cccc2Cl)=O)CCC1N1CCCC1C(N)=O 86445,c1(C(=O)OCC)cc(C(=O)NCc2cc(C)c(C)o2)c(C)cc1NC 86446,C1(C(N(CC(C)NC(c2ccncn2)=O)C)=O)C(C)CCN1C(=O)OC(C)(C)C 86447,C(=O)(CCCC(C)=O)N1CCC(CC(=O)NC(c2ccncc2)CC)C1 86448,N1(C(c2cc(CC)c(F)cc2)C(=O)NC(C)C)C2C=CCC1CCC2 86449,c1(C(N(C2CN(C(C3CC34CC(O)C4)=O)C2)C)=O)ccnc(F)c1 86450,c1(C(N2CCC(CCC(=O)N(C(C#C)C)CCCC)C2)=O)cc(C#C)ccn1 86451,c1(NC(c2nnc(O)o2)C)[nH]c(=NCc2ccc(=N)[nH]c2)nc2scnc12 86452,CCCC(C(O)C(=O)NC1CCN(CCOC)C1)NC(=O)CC(C)(C)COC 86453,CN1CCC(C(=O)NC2CCN(C(c3cccc(NS(C)(=O)=O)c3)=O)C2)C1=O 86454,c1(C(N(C)CCOCCNC(=O)Cn2cnnc2O)=O)cn2ccsc2n1 86455,O=C1CS(=O)(=O)CC(C(=O)NC2CC(CCNC(C3CC(F)(F)C3)=O)C2)N1 86456,c1(CC2(C(N(CC(C)NC(c3cnn(C)c3)=O)C)=O)CCCC2)ccc(Cl)nc1 86457,N1(C(C(CCC)OCC)=O)CC2(C(=O)NCC(CO)C3CCC3)CC1CO2 86458,Cc1cnc(C)c(NC(C2C=CCN2C(c2cccc(Cl)c2F)=O)=O)n1 86459,c1(C(=O)NCCOCCCC#C)ccnc(CNC(C2(C)CC3CC3C2)=O)c1 86460,N1(C(C2(CC=C)CC2)=O)CC(C(=O)NCCF)C(C)C1 86461,C(=O)(C1=CCCN(Cc2ccc(C)cn2)C1)NCc1ccc(OC)cc1 86462,c1(NC(c2c(CNC(CSCCC#N)=O)noc2)=O)cccc(F)c1 86463,C1(NC(c2c(C)cn(C)n2)=O)C(C)CCN(C(c2cnc3scc(C)n23)=O)C1C 86464,c1(C(N2C(CNC(c3nc(C4CC4)cs3)=O)CC(O)C2)=O)cc(F)ccc1Cl 86465,C(C(C(=O)N1CCCC1CNC(c1cc(C)ns1)=O)C(C)(C)C)OCC=C 86466,C(=O)(C1=C(Cl)CCCC1)NCC(C(C(=O)NCC(=C)Cl)F)C 86467,N1(C(C)C)CCCCC1C(=O)NC1(C)CN(C(C2(S(C)(=O)=O)CC2)=O)C1 86468,CC(CN(C)C)CCC(=O)NCc1ccc(C(=O)NCC2C3CCCC23)s1 86469,N1(C(CCC)=O)CCCC(C(N2CC(O)(CNC(=O)CCC(N)=O)C2)=O)C1 86470,C(=O)(C1CCCc2scnc21)NCC(CC)NC(C1CCc2nncn2C1)=O 86471,c1(CC(=O)N(c2nccc(C#N)n2)C2(C(C)(C)C)CCC2)ccc(C#N)c(F)c1F 86472,C1(NC(CSCCCC)=O)CCCN(C(=O)CCc2ccoc2)C1C 86473,N1(C(C(C(C)(C)C)=O)=O)CCC(C(N2CC3C=CCC(C3)C2)=O)C(C)(C)C1 86474,Cc1noc(C)c1-c1cn(C2CCCC2NC(c2ccn(CC(C)C)n2)=O)nn1 86475,N1(CCNC(C2(CCNC(C3(CC)CCC3)=O)CC2)=O)CCNC(=O)C1 86476,c1(-n2cc(CC(C(=O)NCCN(C(=O)OC)C)O)nn2)cccc(C(=O)O)c1 86477,CC1(CCCCNC(N2CCCC2c2ccc(Cl)nc2)=O)NC(=O)NC1=O 86478,Cc1c(C(=O)NCCCCCN(C)C(c2cncc(C(C)C)c2)=O)ncn1C 86479,c1(C(=O)NCCNC(C2CCCOC2)=O)ccc2c(Br)cccc2c1 86480,C1(C(=O)NC2(C(=O)NC3CN(CCC)C(=O)C3)CC(F)(F)C2)CCCC1C1CC1 86481,c1(C(=O)NC2C(NC(C3C(C(C)C)C3)=O)CCC2)nc(-c2ccccc2)sc1N 86482,CCC(CNC(C1CN(C(N)=O)C1)=O)(CC)NC(C1CCNC1=O)=O 86483,C1(CNC(C2(COCC)CC2)=O)CC(C)(C)CN1C(c1ccc(SC)cc1)=O 86484,c1(C(=O)NCCC2C(C)CN(C(=O)C(O)C3CCC3)C2)cc2ncccc2[nH]1 86485,c1(N2CCCC(Cn3ccnc3)C2)nc(Cc2ccsc2)cn2ccnc12 86486,c1(C(N2CCOC(CC)C2)C(=O)NCCC)cnc2cnccn12 86487,c1(C(=O)NC(C)CNC(c2ccncc2N)=O)cc2nccc(C(F)(F)F)n2n1 86488,C1(NC(C(C)OCC=C)=O)CCS(=O)(=O)C12CN(C(=O)CSCC#N)C2 86489,N1(CC(=O)NC(C(C)C)CCNC(C2CCO2)=O)CCc2ccccc2C1=O 86490,C(=O)(CCS(=O)(=O)CC(C)C)N1CC(NC(C2=C(C)S(=O)(=O)CC2)=O)C(C)C1 86491,Cc1cc(C(N2CCOCC(NC(c3ncc(Cl)s3)=O)C2)=O)c(N)c(Cl)c1 86492,N1(C(C2CCC(C)O2)=O)CCC(F)(C(N2CC(Cc3ccco3)C2)=O)C1 86493,C1(C(C)NC(C2(C(F)F)CC(=C)C2)=O)CCN(C(C2(C)CCCOC2)=O)CC1 86494,C(=O)(C1=CC(O)CCC1)NCC1CC(OC)CN1C(c1ccc(F)cc1)=O 86495,n1(CC)nc(C)c(C(=O)NCC2CN(C(c3cc(F)n[nH]3)=O)CCC2C)c1Cl 86496,c1(C(N(C)Cc2ccc(Br)nc2)=O)cc2c(C(F)(F)F)cc(N)cc2s1 86497,c1(C(C(=O)NCC(=C)C)N(CCC(=O)OCC)C)cn2c(Br)cnc2s1 86498,N1(C(C(COCC)n2cc(-c3ccc(C)c(F)c3)nn2)=O)CCC(C23CC(C2)C3)C1 86499,CC1Cc2cccc(C(=O)NC3CC(NC(c4ccc5ncccc5c4)=O)C3)c2O1 86500,C1(C(C(=O)NCCCOC)N(CC(CC)(C)OC)C)CCC(C)(C)C1 86501,c1(N(CC(=O)NCC(N2CCC2C(N(C2CCCN2C)C)=O)=O)C)ccncc1 86502,N1(C(c2cc(NC(C)=O)ncc2)=O)CCN(C(C2(C)CCCCC2)=O)CC1C#N 86503,c1(-c2cn(CC3CC(NC(CC4(C)CCCS4)=O)C3)nn2)ccc(C#N)c(F)c1 86504,C1(N(C(=O)CC2CN(C(C)=O)CCO2)CC)CCN(C(c2cnc(Cl)[nH]2)=O)CC1 86505,C1(C(N2CC(O)(C(C)NC(c3c(OC)c[nH]n3)=O)C2)=O)C2CCCCC12 86506,c1(C(=O)NC(C2CCN(C(C=C(C)C(C)(C)C)=O)CC2)(C)C)c(F)ccnc1Cl 86507,CC1(C)CC(CNC(c2cnc(C(N)=O)s2)=O)CN1C(c1cccc(F)c1)=O 86508,C(=O)(C(O)CC(C)(C)C)N1CCC(O)(C(C)CNC(C23CCC(CC2)OC3)=O)C1 86509,c1(C(=O)NCCCN(C(=O)CCCC(=O)NC)CC)ccc2cccc(F)c2n1 86510,c1(CC)ccc(C(=O)NCC2(NC(=O)Cc3c(C)nn(C)c3C)CCC2)cc1N 86511,N1(C(CSCCC(C)C)=O)CCC2CC1CN2C(=O)C(c1cncc(F)c1)C 86512,N1(C(C2(NC(=O)Cc3ccccc3O)C(C)(C)C2)=O)CC2(C)COCC2(C)C1 86513,C1(OC)CC(NC(C2CCCS2)=O)CN(C(c2cnn(C3CCC3)c2)=O)C1 86514,c1(C(=O)NC(CN(C(=O)C(C)Cc2ccco2)CC)C)ccsc1OC 86515,C1(C(C)C)CN(C(c2cc(N(C)C)ccc2F)=O)CCC1NC(C1CC=CC1)=O 86516,C(=O)(C(C)(O)C(C)(C)C)NC(CNC(C1CC2(CC(=C)C2)C1)=O)C1CC1 86517,Cc1cc(C(=O)N(CCCNC(C2(C)CC(=O)N(C)C2)=O)C)cc(C(F)F)c1 86518,CC1(C)CCN(C(C2C3CCCOC23)=O)CC1NC(c1cccc(Cl)c1)=O 86519,c1(C(N2CCC(C(CNC(CC(C)OC)=O)F)CC2)=O)cc(N)c(F)cn1 86520,Cc1cc(C(N2CC3(CCN(C(=O)C4=CCCC4)C3)C2)=O)c2cc(F)ccc2n1 86521,N1(C(CCCCCC#C)=O)CCc2[nH]nc(CNC(=O)C(C(C)C)N(C)C)c2C1 86522,N1(C(CCc2cnc(C)o2)=O)CC2CC1C2NC(=O)CCSc1nccn1C 86523,c1(C(=O)NC(C2N(C(Cc3cnc(C)s3)=O)CCC2)C)ccc(CO)cc1 86524,N1(C(CCCNC(CC2(NC(C)=O)CC2)=O)=O)CC(C)C(C)C1C 86525,N1(C(C(CC=C)C)=O)CCC2(CCCC(C(=O)OCC)O2)CC1 86526,C1(NC(C(C(C)C)O)=O)CC2CCC(C1C)N2C(=O)Cc1c[nH]c2cccnc12 86527,C1(NC(c2c(=N)[nH][nH]c2)=O)CCCC2CN(C(C3CCCCCC3(F)F)=O)CC12 86528,c1(C(C)C(=O)NCCN(C(C2CC(C)(C)O2)=O)C2CC2)ccc(F)cc1F 86529,C1(C(=O)NCC2CC(C(=O)NC3CCS(=O)(=O)C3)C2)(CC)CNC(=O)C1 86530,C(CC(C)(C)C)(c1n(CCOCC)nnn1)NC(C)CSC 86531,C1(CC=C)(NC(=O)C(O)C=CC)CCN(C(c2cccc(=O)o2)=O)C1 86532,Cc1cc(C)c(C(=O)NCCC2CCN(C(=O)C3=COCCO3)C2)c(=O)o1 86533,C1(C(N2CC(=O)N3CC(C3)C2=O)C2CC2)CCOC1C.CC1CC1.N1CCC1 86534,Cn1cnc2cc(C(N3CCC(C)(C)C(c4cn(CC(N)=O)nn4)C3)=O)cnc12 86535,N1(C(CC(CC)OC)=O)CCC(CNC(c2ccc(Cl)c(Cl)c2)=O)C(C)C1 86536,N1(C(Cc2c(C)nc(S)s2)=O)CCCN(C(C2(C(F)F)CCCO2)=O)CC1 86537,c1(C(N2CCC(N(C(C(C)C(C)(C)C)=O)CC3CC3)C2)=O)cccc2occc12 86538,C1(C(C)NC(C(C2CCC2)OC)=O)CCN(C(C2(CO)CCCC2)=O)C1 86539,CN1CCC(NC(=O)CCN(C(=O)Cn2c(O)nnc2O)CCO)C(C)(C)C1 86540,c1(C(=O)NCCC(=C)CNC(=O)CCc2cnco2)ccc(Cl)cc1 86541,c1(C(=O)OCCCC#C)nn(CC)c2c1COCC2 86542,N1(C(C(CCC)C)=O)CC2CCC(C1)C2CCNC(c1ccccc1CC#N)=O 86543,C1(C(=O)Nc2cn(COC)nc2)CCCC12CCN(Cc1cnc(Cl)cc1F)C2 86544,N#Cc1ccc(C(=O)NCC2CC(NC(c3c[nH]c(Br)c3)=O)C23CCC3)c(O)c1 86545,C1(CC(N2CCC(CN(C(=O)CSCc3ccccc3)C)C2)=O)NC(=O)NC1=O 86546,C(=O)(C(C(=O)N1CCC(C(=O)NCCCCF)(C(C)C)C1)OC)OC 86547,CCC1=NOC(C(=O)NCC(O)CNC(=O)C(C)(C)NS(C)(=O)=O)C1 86548,CC(C)(C(=O)N1CCC(NC(C2CCOC2C(F)(F)F)=O)C1)c1ccsc1 86549,Cc1cc(=NCCNC(N2CCn3cc(C)nc3C2)=O)[nH]cn1 86550,C1(C(N(C)Cc2cccc(C)n2)=O)CCCCCCN1C(C1CC1C(N)=O)=O 86551,N(C(=NCC1CCCO1)NC1CC(=O)N(c2ccccc2Cl)C1)CC(C)(F)F 86552,C(C(C(=O)NC(C)COC(F)(F)F)NC(=O)CCc1nc(C)no1)SCC 86553,c1(CC)cccc(C(=O)N(CCCCCCNC(C23CCC2C3)=O)C)c1 86554,c1(C(=O)NC2(C)CCN(C(C3N=C(C)SC3)=O)C2)cc2cccc(C)n2n1 86555,c1(C(N2CC(C(=O)OC)OCC23CC3)=O)[nH]nc2c1COC2(C)C 86556,C1(NC(C2CCN(C)CC2)=O)CCc2nc(NC(=O)Cc3ccccc3)sc2C1 86557,c1(C(=O)NCCN(C(c2n(CC(C)C)ncc2)=O)C)ccn2cnnc2c1 86558,c1(CN2C(C(=O)Nc3c(C=C)cccc3)CC(O)C2)c[nH]c2c(C)cccc12 86559,n1(CC)nc(C)cc1C(N1CCCC1C(C)NC(=O)C(COC)OC)=O 86560,C1(NC(=O)OCC)CCN(C(c2ccc(F)s2)=O)CC1 86561,N1(c2cc(CC)nc(Cl)n2)CC(F)(F)CC1(C)CNC(=O)C=Cc1ccc(Cl)s1 86562,Cc1nc(Cl)nc(N2CC(CO)(NC(=O)CC3CCC(=O)N3C)C2)c1F 86563,c1(CC)n[nH]cc1C(=O)N(CCCNC(=O)CC1CCC(O)C1)C 86564,N1(CC#C)CCC(C(N2CC(O)(C(C)NC(c3ncoc3C3CC3)=O)C2)=O)CC1 86565,CN(C1CCSc2ccc(Br)cc21)C(N1CCC(CO)CC1)=O 86566,C1(CC(=O)N(CCC#C)CCO)CCCN(C(=O)CCc2ccoc2)C1 86567,C1(C(=O)NC(C)C(C)(C)NC(=O)CSCC(F)(F)F)COC2(CCC2)CO1 86568,C(CSC)(C(=O)N1CC(CC(C)NC(=O)COC2CCOC2)C1)OC 86569,c1(C(=O)NC(CNC(C2(CSC)CC2)=O)CO)ccc(=O)n(C)c1 86570,c1(CC)ccc(C(=O)NCCCNC(c2cc(=O)c(C)c[nH]2)=O)c(N)c1 86571,c1(C(=O)NC2CC(O)(CNC(CCN(C)CC)=O)C2)cc(OC)cc(C(C)=O)c1 86572,CCC(C)(C(=O)NCC1CC(NC(=O)C(c2cccnc2F)(C)C)CC1O)OC 86573,n1(CCC(C)C)cc(NC(=O)NCC(N2CCCC2)c2cccs2)cn1 86574,C1(C(N2CC(F)(CNC(CS(=O)(=O)NC)=O)C2)=O)CC2(CCC2)CO1 86575,CCCC(CCC)=CC(N1CC(NC(=O)C(CC2CC2)OC)C(F)C1)=O 86576,c1(C(N2CC3C(CCNC(CCOCC#C)=O)(CC3)C2)=O)nc[nH]c2ncnc1-2 86577,C1(NC(c2ccc(-c3nc[nH]n3)cc2)=O)C2CCC1N(C(=O)CC1=CCCC1)C2 86578,C#CC1(C)CCCN(C(=O)C(O)CCCNC(=O)C(C)(O)C=C)C1 86579,c1(C(=O)NCC(C)(C(C)C)NC(c2ccn(CCC)n2)=O)ccnc(F)c1N 86580,c1(C(N(CCCN(C(CSCC#C)=O)C)C)=O)ccc(C(C)=O)[nH]1 86581,c1(CNC(C2CCC3(CCC3)C2)=O)c[nH]c2ncccc12.C123CC1CN(C2)C3=O 86582,C1(C)(CNC(=O)NC(C2CC3CCC2C3)C)CCN(C)CC1 86583,C1(NC(C(C)=C(CC)C)=O)CN(C(=O)COCC2CCC2)CCC1CO 86584,Cc1nc(=N)[nH]c(C)c1C(N1CCC(NC(c2cc(Cl)on2)=O)C(C)C1)=O 86585,c1(C(N2CCC(NC(c3c(C)c(N)cnc3)=O)(CO)C2)=O)cnc2[nH]cncc1-2 86586,N1(C(CSC)=O)CCCC(N2CCN(C(=O)CC3CCCC34CC4)CC2)C1 86587,C(=O)(CCCC(N)=O)NCC(C)CNC(=O)Cc1ccn(C)n1 86588,N1(CCNC(=O)OC(C)(C)C)CCC(Cc2cncnc2)CC1 86589,C(=O)(C1COc2ccc(Cl)cc21)NC(CC=C)CNC(c1ccsc1OC)=O 86590,N1(CC2CCCN(c3n(CCOC)nnn3)C2)CCc2cc(C)cc(C)c2C1 86591,c1(NC(c2c(F)ccc3c2OCO3)C)ccc2nc(N(C)C)[nH]c2c1 86592,C1(CC)CN(C(C2CC(F)C(=O)N2)=O)CCN1C(=O)Cc1cc(C)ccc1F 86593,O(NC(=O)C(C)(CSC)NC(=O)C(CC)N(C)C)CCCC#C 86594,c1(CC(=O)NCCN(CC(C)O)C(C2CC2F)=O)cccc(C(C)(C)C)c1 86595,Cn1nc2c(c1C(=O)Nc1cnccc1Cl)CN(C(C1CCCCO1)=O)CC2 86596,CC(C)C1=NOC(C(=O)NCC=C2CCN(C(C3CC(C4CC4)C3)=O)CC2)C1 86597,c1(NC(C2C(NC(C(C)(C)OC)=O)C2)=O)cc(F)cnc1Br 86598,CCC(C)(C)C(=O)NCC1(F)CC(NC(c2ccc(C(F)(F)CF)cc2)=O)C1 86599,C1(NC(C(c2ccc(C)cc2)=O)=O)CN(C(=O)CC23CCCC2C3)CC1(C)C 86600,c1(C(=O)OC)c(C)[nH]c(C(=O)NC2CC2CNC(c2cc(C(N)=O)c[nH]2)=O)c1C 86601,C(=O)(C(C)CC(F)(F)F)NCC1COCCN(C(Cc2ccc(C)cc2)=O)C1 86602,N1(C(C2CC(OC)C(OC)C2)=O)CCOC2(C1)CN(C(=O)C=Cc1cscn1)C2 86603,Cc1c(CC(=O)NC(C)(CNC(c2cnn(CCO)c2N)=O)C(C)C)cnn1C 86604,c1(Nc2cccc(OCC(=O)NC(C)CCF)c2)ccc(S(N)(=O)=O)cc1 86605,C1(C)(CNC(CN(S(CC)(=O)=O)C)=O)CC(NC(=O)CC(C)NC(N)=O)C1 86606,c1(C(=O)NC(CC)CN(C(=O)Cc2ccns2)CC)occ2c1CCCC2 86607,c1(NC(C2CCN(C(CN(C(CCC)=O)C)=O)C2)=O)cc(Cl)c(OC)c(Cl)c1 86608,C1(C(N(CCCNC(c2cnc3[nH]ccc3n2)=O)C)=O)CCCCC1P(C)(C)=O 86609,CC1=CCSC1C(=O)NCC(C)CNC(=O)C=CCOC(C)(C)C 86610,N1(C(c2c(C#N)ccs2)=O)CCCCCCC1C(=O)NC1CCC2CC12 86611,N1(C(=O)C=CSC2CC2)CCC2(NC(C3CC(N4CCCC4)C3)=O)CC2C1 86612,c1(OC)ccc(CC(=O)NC2CCC(NC(C3CC(F)C3)=O)C2)c2ccccc12 86613,Cc1cccc(C(F)(F)C(=O)N(C)CCN(C(c2ccc(Br)cc2)=O)C2CC2)c1 86614,C1(n2c(C(C3CC(C)C3)(C)NCc3cnns3)nnn2)CCCCCC1 86615,c1(C(N(CC(CC)NC(C2C(C)(C)C2(F)F)=O)C)=O)ccc2ccnn2c1 86616,N1(C(C=CS(C)(=O)=O)=O)CCC2(CC1)CN(C(=O)COc1cc(F)cc(F)c1)C2 86617,C(C)(C)(CC(=O)NCC1CCN1C(c1cccc(OCC2CC2)c1)=O)N(C)C.OC 86618,C=Cn1nccc1C(=O)NC1CCN(C(=O)C(C)Cc2cnn(C)c2)C1C 86619,N1(C(c2cc(C)on2)=O)C2CCCC1CC(NCc1ncc(Br)cc1[N+](=O)[O-])C2 86620,N1(C(c2n(CCCC)ncc2)=O)CCC2CN(C(c3ncoc3C3CC3)=O)C2C1 86621,C1(C)(C(N2CC(F)(C(=O)NCC3(CC=C)CCCC3)C2)=O)CC(C)=NO1 86622,C(=O)(C(CCOC)NCC1CCC(CNC(=O)Nc2ccc(OC)cc2)CC1)OC 86623,N1(C(C(CC)F)=O)CCC(O)(CNC(=O)CC(c2ccc(C)cc2)C)CC1 86624,C(=O)(C(C(F)(F)F)C(F)(F)F)NC1C(C)N(C(C2CN3CCCC3CO2)=O)CC1 86625,C1(C(=O)NCC2CCCN(CC(F)F)C2)CC2(CCCCCCC2)N1 86626,C1(C)(NC(C(C)Cc2ccccc2)=O)CCC(NC(=O)COCC2(F)CC2)CC1 86627,C1(CNC2CC(C(=O)Nc3ccc(SC)cc3)C2)CCC(F)(F)CC1 86628,c1(-c2cnc(NC(c3nn(C(CC)CC)c(C)c3)=O)s2)cccc(C#N)c1 86629,C1(CNC(C=CC)=O)CC(F)(F)CN1C(=O)C(O)Cc1[nH]cnc1C 86630,c1(C(N(CCOCCC(N2CCC(C(N(C)C)=O)C2)=O)C)=O)cc[nH]c(=N)n1 86631,Cc1nn(CC(=O)NCC(O)CCNC(C2CN(C3CCCCC3)C2)=O)c(=O)n1C 86632,c1(C(N2CC(C(=O)NCC(=O)OCC)OCC2)=O)c[nH]c2cc(F)ccc12 86633,c1(NC(CCC2(NC(CCC)=O)CCC2)=O)c(C)ccn(C)c1=O 86634,N1(C(C(C)c2cccs2)=O)CC(C2CCCN(C(C3(C4CCC4)CCC3)=O)C2)C1 86635,c1(CN(C(c2c(C)cc[nH]c2=N)=O)C)c(Cl)cc(Cl)cc1Cl 86636,CON(C(=O)c1c[nH]nc1CNC(=O)C(C1CCCCC1)C)C1CCCC1 86637,C(=O)(CS(=O)(=O)C1CCCC1)N1CC(CN(C(CCC=CC)=O)C)OCC1 86638,CC(C)(CNS(C)(=O)=O)C(=O)N(C1CCCCCC1)CCNC(=O)CNC(N)=O 86639,C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CC)(CNC(c1cnco1)=O)CC 86640,C(=O)(CC(=O)NC1CC1)NC(C1CCCN1C(c1csc(-c2ncc[nH]2)n1)=O)C 86641,CC(C)C(O)C(F)(F)C(=O)N1CC2CCN(C(=O)CCCC(C)(C)C)CC2C1 86642,C1(C(=O)NC2(CF)CN(C(C(CC#C)C3CC3)=O)C2)CC2(C1)CC2(F)F 86643,C1(C(=O)NC(C)(C)CCNC(=O)Cc2cncnc2)CCCC(N(C)C)C1 86644,CCC(CC(=O)NCC1(O)CCN(C(c2ncoc2Br)=O)C1)C1CCC1 86645,c1(CC)cc(C(=O)NCCC2CC(NC(=O)CC3CCN(C)CC3)C2)oc1CC 86646,C(=O)(C(CC)CC(F)(F)F)NCC1CN(C(CCCC)=O)CC(C)(C)C1 86647,c1(C(=O)NCCC2N(C(C(C=C)OC)=O)CCOC2)cc(C)c2occc2c1 86648,CCC(C(=O)N(C)CCn1cc(C2CCCCO2)nn1)N(C)C 86649,c1(C(=O)NCC2CCS2(=O)=O)ccc2c(c1)NC(=O)CCN2 86650,Cc1ccnc(C(C)(C)C(=O)NC2CCC2NC(C2COCC2(C)C)=O)c1 86651,c1(CNC(=O)C(F)(F)F)cc(F)c(Nc2cc(-c3ccncc3)ccn2)c(F)c1 86652,C1(NC(CCC(=O)NCC)=O)CN(C(c2ccc(N)c(F)c2)=O)CCC1(C)C 86653,c1(CCC(N2CC(CC=C)(NC(=O)C=C(C)CCC)C2)=O)cncc(OC)c1 86654,C1(NC(C2CN(C)C(=O)C2)=O)CCS(=O)(=O)C12CN(C(C1(CO)CCCC1)=O)C2 86655,C1(NC(C2C(OC)C2)=O)CCCCC1C(=O)NCc1ccccc1OC(F)(F)F 86656,c1(C(N2CC(NC(CC(C)(C)O)=O)C3(C2)CC3)=O)cc2ccc(F)cc2[nH]1 86657,C=CCC(C)(C)CC(=O)N1CCC(C)CC1CNC(=O)CC1(N(C)C)CCC1 86658,c1(C(N2CCCC2CNC(C2CC(F)(CF)C2)=O)=O)ccc2c[nH]nc2n1 86659,c1(C(N2C(CNC(CS(CC)(=O)=O)=O)CC2)=O)cc(Cl)c(C)cc1[N+](=O)[O-] 86660,c1(C(=O)NCCCC(=O)NCCC2CC=CCC2)cc(O)ncc1F 86661,CC(C)CC(C)C(=O)NCC(C)(F)CNC(C1(CO)CCC1)=O 86662,Cc1cnc(C(=O)NC(C)(C)CN(C)C(c2ccc(C(C)(F)F)nc2)=O)cc1C 86663,N1(C(C(Cn2cncn2)NC(c2cc(C)[nH]c2)=O)=O)CCCC(C)(F)C1 86664,c1(COC)cccnc1C(c1nnnn1C)NCC(C)C(C)(C)C 86665,C1(CNC(C(C(=C)C)(C)C)=O)CN(C(=O)CC2(O)COC(C)(C)C2)CCC12CCC2 86666,C1(c2nnnn2C2CC2)(NCc2ccncn2)CC2COC1C2 86667,C1(CNC(c2[nH]cc(C)c2)=O)(NC(=O)CCN(CC(F)(F)F)C)CCCCC1C 86668,C(=O)(C1CCCc2ncnn21)NCCCN(C)C(c1cc(Br)ccc1F)=O 86669,c1(OC)ncc(C(=O)NC2CC(F)(CNC(=O)CCCN(C)C(C)=O)C2)c(C)n1 86670,N(C(=NCC1CC1)NCC1(C)CCCC1)CC(C)(C)OC 86671,n1(C(C)C)nnc(=NC(=O)Cc2cc(Br)cc(C#N)c2)[nH]1 86672,c1(OCC(N2CC(NC(CC=CC=C)=O)C(F)C2)=O)ccc(C)cc1C 86673,c1(Cc2cn(C3CCN(C(C=COCC)=O)C3)nn2)c(Cl)cc(Br)cc1Cl 86674,c1(C(=O)NC2C=CCN(c3nnc(C4CC4)s3)C2)ccc2c(c1)CCCC2 86675,N1(C(C(c2c(C)cccn2)(F)F)=O)CCOC(C)(CNC(c2ccc(Cl)o2)=O)C1 86676,c1(CC)ncsc1C(=O)NC1(CNC(=O)C(F)CC2CC2)CC1 86677,C12=NC=CC(=NC(C)c3ccccc3CN1)N2.c1(CC(=O)OC)csc(CC)n1 86678,C1(NC(CC(C)(C)O)=O)CC2CC(C1)N(C(c1cnncc1C(F)(F)F)=O)C2 86679,CCCC(C(=O)NCC1CCN(C(C2CC2COC)=O)C12CC2)S(N)(=O)=O 86680,c1(C(=O)NCC(O)Cc2ccccc2Br)coc2c(Cl)cc(Br)cc12 86681,CC(CNC(=O)CN(C(c1cc(C#N)cs1)=O)C1CC1)CC(C)O 86682,C1(NC(=O)Cc2cccnc2O)CN(C(c2ccoc2)=O)CC2CCCC12 86683,c1(-c2cnc(OCC)nc2)nc(C(=O)Nc2ccc(C(=O)NC)cn2)ccc1F 86684,c1(C(N2C(C(=O)NCc3cocn3)CC(=C)C2)=O)c(O)ccc2ccccc12 86685,C1(CNC(C2(CC#C)CCOC2)=O)(NC(=O)C(O)P(C)(C)=O)CC2CCC1CC2 86686,C1(NC(CC2CC(NC(CCCC=C)=O)C2)=O)COCCN(C)C1 86687,c1(NC(=O)NCCc2nc(CC)sc2)ccccc1NCCO 86688,c1(C(=O)NCCN(CCC)C(C2CC2(C)Br)=O)cn[nH]c1 86689,c1(CCC(=O)NCCN(C(C2(C)CCC(=O)C2)=O)CC)ccc2ccccc2c1 86690,C1(CNC(C=C(C)C(C)(C)C)=O)CC2CN(C(C3CC3C(=O)NCCO)=O)CC12 86691,c1(N2CCCC(CO)CC2)ncnc2ccc(O)cc12 86692,CN1CCc2[nH]nc(C(=O)Nc3ccc(CN=[N+]=[N-])nc3)c2C1 86693,c1(C(N2CCC(NC(C(C(C)C)SC)=O)C23CC3)=O)ccc2c(C)noc2c1 86694,CCC(CCC(=O)N(c1ccccc1)CC)NC(C1CCCS1)=O 86695,N(C1COc2ccc(Cl)cc21)C(C(Cc1ccccc1Br)NC(C)=O)=O 86696,c1(NC(C(=Cc2cocn2)C)=O)cnc(OC2CCOC2)c(C)c1 86697,c1(C(=O)NCC2(C)CN(C(c3ccc(F)nc3)=O)C2)cnc(O)c(Br)c1 86698,S(=O)(=O)(c1ccc(N2CCOC3(CC3)C2)c(C#N)c1)NC1C(OC)CN(C)C1 86699,c1(OC)ccc(C)cc1C(=O)N(C1(CC(=O)N(CC(O)C2CC2)C)CC1)C 86700,C12(C(=O)NC(CC)CO)CC1CN(C(=O)C(C)NC(=O)Cc1ccccc1)C2 86701,c1(C(N2CC3CCC2CC3)C(=O)NC(CC)C)ccc2cccc(Br)c2n1 86702,N1(C(C(c2cnccn2)C)=O)CCC(CNC(=O)C(C2CC2)C2CC2)C12CC2 86703,Cc1ncnc(C(=O)N(C)CC=CC(=O)NCCCc2nc[nH]n2)c1C 86704,C(CCC(=O)N(C1CCCCC1)CCNC(=O)C=CC1(C)COC1)N(C(C)=O)C 86705,N12CC(F)(F)CC1CONC(=O)c1cn2ccscn1.C1(C=O)(CO)CCCC1 86706,C(=O)(CCC(=O)NC1(C(N2CCC(OCCSC)C2)=O)CCC1)OCC.OCC 86707,C(C)(C)(CCCC(=O)NCc1cn[nH]c1)NC(c1n(CC#C)ccc1)=O 86708,C=C(Cl)CCC(=O)N(CCCNC(=O)CNC(c1cccnc1)C1CCCC1)CC 86709,c1(C(CC)NC(=O)C(N2C(C)CC2(C)C)CC)ccc(OCCOC)c(OC)c1 86710,c1(C(N(CCCCCNC(=O)C#CC2CCCO2)C)=O)ccc2nnc(S)n2c1 86711,c1(C(=O)NC(CNC(c2cocn2)=O)C2CCC2)cc(Cl)nnc1O 86712,c1(CN(C)C(=O)NCC2CC2c2cn[nH]c2)cccc(O)n1 86713,c1(CN2CCN(CC)C2)nc(C2=NOC(C)C2)n(-c2ccc(C)c([N+](=O)[O-])c2)n1 86714,c1(NC(C2(C(=O)OC)CC2)=O)cn(C)c(NC(c2cocn2)=O)n1 86715,CC1=C(C(=O)NCCOC2CCN(C(c3oc(C)nc3C)=O)C2)CC1 86716,N1(C(c2[nH]cc(C)c2)=O)CC(CC(=O)N(C2CCOC(C)C2)C)CC1(C)C 86717,c1(N2CCCC(CO)CC2)nc2ccc(Cl)cc2c(=NCCN2CCC(O)C2)[nH]1 86718,C1(NC(C(CSC)(C)C)=O)CN(C(=O)CN(C(=O)COC(F)F)C)CC1O 86719,c1(OC)cc(C(N2CCN(c3ccc(C(F)(F)F)nc3)CC2)=O)ccc1N 86720,c1(C(N(C)CC2CN(C(C3CCOC3)=O)C2)=O)csnc1Cl 86721,n1(CC)nnc2cc(C(N3CC4CCCC4(NC(c4cnn[nH]4)=O)C3)=O)ccc12 86722,CCCCC(O)CC(=O)N1C2CCC1(CNC(=O)CN(c1ccncc1)C)CC2 86723,CC(CCCc1cn(CC(c2ccn(C)n2)O)nn1)C(=O)N(CC(F)(F)F)CCO 86724,C(=O)(C1=C(C)Oc2ccccc2C1)N1CCC(C(C)NC(CC(=O)OCC)=O)C1 86725,N1(C(C(CCC2CC2)NC(C(C)SC(C)C)=O)=O)CC2(CCNC(=O)O2)C1 86726,N1(C(CCCC#C)=O)CCCC(C2CCN(C(c3cscc3Cl)=O)C2)C1 86727,C1(C)(CC(=O)NCCC(=O)NC(c2ccn(C)n2)C)OCCO1 86728,N1(C(c2c(CC)occ2)=O)CCC(C(=O)NCC(=O)N(C)C)C12CCC2 86729,N1(C(C23CC(C2)C3)=O)CCC12CCN(Cc1cccc(F)c1O)CC2 86730,N1(C(c2c(CCC)n(C)nc2)=O)CCCN(C(=O)CC=C(Cl)Cl)CC1C(C)C 86731,c1(OC)ccc(Cn2nc(C3CCOC3)nc2-c2nc(C)sc2Br)cc1 86732,C1(C(=O)NC2(C3N(C(C=CC(C)=O)=O)CCC3)CC2)C(C=C(C)C)C1(C)C 86733,S(=O)(=O)(c1cc(Cl)c(Br)cc1F)N1CC(C(=O)Nc2cncnc2O)SCC1 86734,c1(CSCC(=O)N(C)CC2CC2c2ccccc2)ncccc1Br 86735,c1(C(=O)NCC(C)NC(C(c2c(C)ccc(F)c2)O)=O)ccnc2c1ccn2C 86736,C(=O)(C(CC1CC1)NC(C1CCNC1=O)=O)NCC(c1cccs1)C 86737,c1(-n2c(-c3cnc4cccnc4c3)nc(C(CC)C)n2)cccc2ccccc12 86738,N1(C(C(C)(C)OC(C)=O)=O)CCC(C(F)F)(CNC(C2CCC3CCC23)=O)C1 86739,c1(NC(=O)NC)cccc(C(N2CC3CC3(CNC(=O)CN(C)CCO)C2)=O)c1 86740,c1(CC(=O)NCc2ccc(CNC(=O)CC3(O)CCC3)cc2)cc(Cl)cc(Cl)c1 86741,c1(-c2cn(CCN3C(N4C(=O)OCC4)COCC3)nn2)ccc(F)c(Br)c1 86742,N1(C(Cc2c(C)cco2)=O)CC2CC(C1)C2NC(=O)CNS(=O)(=O)N(C)C 86743,CC1(NC(=O)CCC2CC2)CCCCC1C(=O)NC1COCC1C(F)F 86744,C1(NC(=O)CCF)COCC1NC(c1cn(-c2ccccc2)nn1)=O 86745,Cc1c(C(N2CC(C)N(C(=O)OC(C)(C)C)CC2C)=O)cc(F)cc1[N+](=O)[O-] 86746,CCCCCCCS(=O)(=O)Cc1ccc(C(C)(C)O)cn1 86747,N1(c2cn(C)nc2)CCN(C(=O)Nc2ccc(N3CCC3=O)cc2)CC1 86748,n1(CCC)ccc(=NC(=O)C2CCC(C(C)C)N2C(C2CC2C#N)=O)[nH]1 86749,C1(C(N2C(CNC(CC3(S(N)(=O)=O)CC3)=O)CCC2)=O)COc2ccccc2O1 86750,c1(OC)cc(O)ncc1C(=O)NC(CNC(C1(C#N)CCC1)=O)CC(C)C 86751,C(=O)(CC(O)C(C)CC)NCC(CC(=O)N(CC(C(=O)NC)C)C)O 86752,C(C(CNC(c1ccns1)=O)S(C)(=O)=O)NC(C1N(C(C(CC)C)=O)CSC1)=O 86753,CCC(C(=O)NC1CN(C(C2(c3cccc(Cl)n3)CC2)=O)CC1O)C(C)(F)F 86754,C1(NC(c2c(C)csc2Cl)=O)CCN(C(=O)COC2CC(F)(F)C2)CCC1CO 86755,N1(C(C2C=CCCC2)=O)CCC2(CC1)CCN(C(C1CCC(F)(F)CO1)=O)C2 86756,c1(C(=O)NC(CNC(C2CN(C)C(=O)CC2)=O)(C)CO)csc(=NC2CC2)[nH]1 86757,CS(=O)(=O)c1ccc(F)cc1C(=O)NC1CC(F)CN(C(C2CCC(=O)N2)=O)C1 86758,C1(CN(C)C(c2cnn(C3CCC3)c2)=O)CN(C(C2CC(F)C(=O)N2)=O)CCO1 86759,c1(NC)ccc(C(=O)NC(C(=O)NCc2cccc(Cl)n2)C(C)C)nc1 86760,CC1OC2(CO)CC1(C(=O)NCCN(C(c1cc(N)nc(Br)c1)=O)C1CC1)C2 86761,C1(NC(C(CCSC)O)=O)CCN(C(c2ccc(Cl)s2)=O)C12CC2 86762,C=CCC(C)(C(=O)NC1(CNC(=O)C(C)CC)CCC1)N(C)C 86763,C(=O)(C1Cc2ccccc21)NC1CN(C(C=C(C)C)=O)CC12CCC2 86764,c1(C(=O)NC2C(NC(c3c(C)noc3C3CC3)=O)CC2)onc2ccccc12 86765,C1(C(=O)NC(c2ncccn2)CC)CN(C(C2(C)CNC(=O)N2)=O)CCO1 86766,c1(C(N2CCC(NC(CC(=O)N(C)C)=O)CC2)=O)noc2c1CCCC2 86767,CC1(C)CCC(C(=O)NC2(C)CN(C(=O)CC3(C(F)(F)F)CNC(=O)C3)C2)O1 86768,S(=O)(=O)(C(Cl)(Cl)Cl)NCC(N1C(C(=O)Nc2scc(C)n2)CCC1)=O 86769,N1(C(CCOC2CN(C(C(CSC)OC)=O)C2)=O)CCC(C)(F)C1 86770,N1(C(COc2cc(C)on2)=O)CCN(C(c2nc3c(s2)COCC3)=O)C(C)C1C 86771,C1(CNC(C(CSC)(C)C)=O)CC(C)CN(C(=O)CC2CC(F)C2)C1 86772,C(CC(=O)NOC(C)C)(C(F)(F)F)NC(CCNC(=O)NCC)=O 86773,C(=O)(C1=CCCC1(C)C)N1C(CN(C(c2c(CC)cc(OC)cc2)=O)C)CCC1 86774,C1(C(N2CCC(C(C)CO)CC2)=O)(CC)CCCOC1 86775,C1(O)(CC(=O)NCC(CCOC)NC(CSCCOC)=O)CCCCC1 86776,Cc1nnc(NC2CCCN(C(c3nc(C)n4ccccc34)=O)C2)c(C#N)c1C 86777,O(NC(=O)C(C)(C)CCCNC(=O)CCC(C)OCC)CCC 86778,c1(C(=O)OC)ccc(I)cc1NC(C1CCN1Cc1ncco1)=O 86779,C12(C)CN(C1)O2.C1(C(=O)NC(C)=O)(NC(=O)COC(C)(C)C)CC1 86780,C1(F)(C(=O)NC2CC(NC(c3cc(C(=O)OC)[nH]c3)=O)C2)CCS(=O)(=O)C1 86781,c1(OC)ccnc(C(=O)NCC(C)NC(=O)CC(C)n2ccnc2SC)c1F 86782,C1(CC(=O)NC(C(=O)NCC(N2CCCCC2)C)CO)CCC(C)(C)C1 86783,Cc1ccc(NC(N2CCOCC(C(=O)OC(C)C)C2)=O)c(C)c1 86784,N1(C(C=CC)=O)CCOC(CN(C)NC(C2CC2C(N)=O)=O)C1 86785,C1(NC(c2c(C)noc2)=O)CC12CCN(c1cc(=O)n(-c3ccccc3)[nH]1)CC2 86786,C1(NC(C2(CC=C)CCCC2)=O)CN(C(C2CC2(C)C(F)(F)F)=O)CC(C)(C)C1 86787,N1(C(C2(COC)CC2)=O)CCC(CNC(=O)C(C(C)C)NC(C)=O)C1(C)C 86788,c1(OC)ccc2nc(N3CC(C)CC(C)C3)[nH]c(=NCc3cc(OC)ns3)c2c1 86789,c1(C(C(=O)NCC2C(NC(CC(C)SC)=O)C2)N(C)C)c(F)cccc1F 86790,C1(NC(C=CCC)=O)CN(C(c2ccc(-n3ccnc3)cc2)=O)CCC1C 86791,C1(C(N2CC=CC(NC(c3cc(Cl)c(Cl)s3)=O)C2)=O)(OC)CCCCC1 86792,c1(COC(c2n(CCC)nc(C)c2)=O)c(Cl)cccc1Br 86793,c1(C(N(CC(C)NC(=O)Cn2cc(C#N)cn2)C)=O)ncccc1OC(F)F 86794,c1(SC)ccc(C)c(C(N2CCCC3(NC(c4ccns4)=O)CC23)=O)c1 86795,CS(=O)(=O)c1ccc(CN2CCC(O)(C(=O)Nc3ncc(I)nc3Cl)C2)cc1 86796,c1(C(N2CC(CC=C)(NC(c3cnn(C)n3)=O)C2)=O)ccc2ncn(C)c2n1 86797,C(C)(CCC(=O)NOC(c1ccncc1)C)NC(C1CC(SC)C1)=O 86798,C1(NC(C2(CC=C)CC2)=O)CC2CC1CC2C(=O)NC(CO)C1CC1 86799,C1(CN(C)CC2CCN(C(c3ccccc3)=O)C2)CCS(=O)(=O)N1 86800,C1(NC(C2CCO2)=O)CCC2(CC1)CN(C(c1ccc(C3CC3)cn1)=O)C2 86801,C1(NC(c2cc(C=C)cc(F)c2)=O)CC(C2CCN(C(=O)CC3=CCCC3)C2)C1 86802,C=CCC(CNC(=O)Cc1ccn(C)c1)C(=O)N(c1ccc(C)cc1C)C 86803,C(=O)(C#CC1CCCOC1)N1CCN(C(c2c(COC)scc2)=O)C(COC)C1 86804,N1(C(C(CC=CC)CC)=O)CCC2(CC(NC(c3cc(C)c(Cl)cc3C)=O)C2)C1 86805,c1(C(=O)NC(C2CCCC2)C)c(CNC(=O)CC(C)(C)N(C)C)cnn1C 86806,CS(=O)(=O)CCC(=O)N1CCN(C(=O)COC(F)F)C(C(C2CCC2)OC)C1 86807,N1(C(c2ccc(C)cc2O)=O)CC2CCC(C1CO)N2C(=O)Cc1cccnc1 86808,C12(C(=O)NC(C)CCNC(=O)C(C)C3CCOC3)CC=CC(C1)OC2 86809,Cc1ccc(C(N2CC(N(C)C(C3CCOCC3)=O)C(F)C2)=O)c(N)c1C 86810,C1(C(=O)NC(C)C(N)=O)CC(F)(F)CN1Cc1cccc(-n2cncn2)c1 86811,c1(NC(C(c2ccnn2CCSC)N(C(C#C)(C)C)C)=O)cccc(Cl)c1 86812,N1(C(C2C(C)C2C)=O)CCC(CCCNC(C2(C)CCCOC2)=O)CC1 86813,c1(C(N(CCNC(c2ccccc2)=O)CC)=O)ccc2nnn(C)c2c1 86814,C1(CNC(c2c(C)[nH]nc2Br)=O)COCCN(C(C2CN(C)CCO2)=O)C1 86815,c1(C(N(C2CCN(C)CC2)CC(C)C)=O)cc(C2CC2)n(C(C)(C)C)n1 86816,c1(C(=O)NC(c2cn(C(C)C)nc2)C)cccc2c1CCO2 86817,C1(C(=O)NCCCOCCNC(C2C=CC=CC=C2)=O)CCC2(CCOC2)O1 86818,C(=O)(C(CCC(N)=O)NC(=O)Nc1ccc(Cl)cc1)NCCCC(=O)N(C)C 86819,N1(C(C2C(C(N)=O)COC2)=O)CCC(C2CN(C(C3CCCCO3)=O)C2)CC1 86820,C1(NCc2ccc(C(=O)OCC)[nH]2)CCN(C(C2CC2OC(C)=O)=O)CC1 86821,C1(NC(C2(CC)CCCC2)=O)CCN(C(c2ccnn2CC(F)F)=O)CC1CO 86822,Cc1cnccc1C(=O)NCC1C2CN(C(c3cc[nH]c3C)=O)CC12 86823,C1(C(=O)NC(CCC)C2CCC2)CCC(O)CN1C(C1CC2C=CC1O2)=O 86824,C(CCC(O)CO)N(C(CC1(C)N(C(C=CC=CCC)=O)CC1)=O)C(C)C 86825,N#Cc1cccc(F)c1NC(C1CC(F)CN1C(c1ncccc1Cl)=O)=O 86826,C1(NC(C2(CNC(CCc3cc(C)on3)=O)CCC2)=O)CCCC1C1CC1 86827,N1(C(=O)OC(C)(C)C)CC(C(N2CCC3(CCC3O)C2)=O)C(C2CCCC2)C1 86828,C(=O)(C(CC(C)(C)C)OC)NC(C(=O)NCC(COC)(C)O)(C)CO 86829,C1(C(=O)NCCCN(C(=O)CC2CCCC(=O)N2)C)Cc2c[nH]cc2S1(=O)=O 86830,N1(C(CSC2CC(C)C2)=O)CCC(OC(F)F)C1 86831,C1(C(=O)NCCCN(CCCNC(C2(C(C)C)CC2)=O)C)CCCC1(C)C 86832,C1(CNC(C=CS(C)=O)=O)CC(C)(C)CN1C(=O)Cc1nc(=N)[nH][nH]1 86833,C1(NC(c2c(N)c(Cl)ncc2)=O)CC12CCC(NC(C1CC1F)=O)CC2 86834,c1(OC)cc(Br)c(F)cc1NC(=O)CC1CCCN1C(c1ccc(C)cc1I)=O 86835,CCS(=O)CC(=O)N1CCC(C(=O)NC(C)C(C)(C)C#N)(CF)C1 86836,N1(C(c2cnn(C)c2C#N)=O)CCCC2(CCCN2C(C2CCC2(C)C)=O)C1 86837,Cc1ccc(NC(=O)C(C)(C2CC2)N(C(=O)C(O)C(F)(F)F)C)cc1Cl 86838,c1(C(=O)NCC(CN(C)C(C2CC2(C)Br)=O)O)ccc(N)cn1 86839,C1(C(=O)NCC2(C#C)CC2)CC(C)(NC(C2CC(O)(C(F)(F)F)C2)=O)C1 86840,c1(CNC2CC(CC(=O)NC(C=C)CO)C2)csc(Br)n1 86841,CN1N=C(CC(=O)N2CC(=O)NCC2C(N2CC3C(C(N)=O)C3C2)=O)CC1=O 86842,Cc1cc(C)c(NC(=O)Nc2cc(C)[nH]n2)c(C)c1.C12CC3CC1CN3C2=O 86843,C#CC1(CO)COCCN1C(C1CCCN(Cc2nccn2CCOC)C1)=O 86844,c1(N2CCC(NC(C(CCCC)(C)F)=O)C(F)C2)nc(Cl)nc2c1ncn2CC 86845,C1(C(=O)NCCCN(CCCC)C)CCCN1CCC(C)C 86846,C(=O)(C(F)C(C)(F)F)N1CCC(CC(=O)N(C2CCS(=O)(=O)C2)C)CC1 86847,N1(C(CC2(OC)CN(C(=O)CC3CCCSC3)C2)=O)CCC12CN(C)C2 86848,N1(C(C(C=C)OC)=O)CCC(C(=O)NC2CC3(CC3)C2)C12CCC2 86849,Cc1cc(C(=O)NCC(C)(O)CNC(=O)CCSCC(C)C)nn1C(C)C 86850,C(=O)(CCC(C)(C)C)NCCCCN(C(=O)CC(O)c1cnc(Cl)s1)C 86851,C1(C(NOCCCN(C)C)=O)CCOCCN1C(C1CC(=O)NC1(C)C)=O 86852,N1(C(c2ncccc2F)=O)CCC2CC2(C(=O)NCCCn2ccnn2)CC1 86853,c1(OCCC(N2CCC(CC=C)(NC(=O)C(C)CSC)C2)=O)cc(F)ccc1F 86854,c1(-c2cccc(CO)c2)c[nH]c2ccc(Oc3ccccn3)cc12 86855,c1(OC)cnccc1C(=O)NC1CC(CNC(=O)CC2CCC23CCC3)C1 86856,C(CC(C(=O)NC1C2CCCCC12)NC(C1CCC1C)=O)=CC 86857,CC(C(=O)NC(C1CCCN1C(c1csc([N+](=O)[O-])c1)=O)(C)C)P(C)(C)=O 86858,C(C(C)(C)C(=O)NCC(C(=O)N(C)C(C1CCCC1)C)N(C)C)OC(C)C 86859,C(N=c1[nH]c2ccccc2s1)C1CCC(NC(c2cncc3[nH]ccc23)=O)C1 86860,c1(C(=O)NC2C(CNC(C(C)OCCCCCC)=O)CC2)ccn2cccc2c1 86861,C1(CNC(c2cnn(C)c2C(N)=O)=O)CCC2(CN(C(=O)OC(C)(C)C)C2)O1 86862,N1(C(C(C=CC)O)=O)CC2CCN(C(c3nn(C)c(Cl)c3Cl)=O)C2C1 86863,c1(C(N(C2CCC(NC(C3CC4(C3)CC4F)=O)CC2)C)=O)cc(N)c(Cl)c(O)c1 86864,c1(C(N2C(CN(C(c3cccc(C#C)c3)=O)C)CCC2)=O)ccc2c(c1)OCC2 86865,Cc1cc2[nH]c(C(=O)NC34CCN(C(c5cnn(CCO)c5)=O)CC3C4)cc2s1 86866,N1(C(C=C(CC)CC)=O)CCCC(O)(CNC(=O)CC2CCCN(C)C2)CC1 86867,N1(C(c2nc(CNC(C(C)C3CCCC3)=O)oc2)=O)CCC2(CCCO2)C1 86868,c1(CCC(=O)Nc2cc(OC)c(F)cc2)ccc2[nH]ccc2c1 86869,c1(C(=O)NC2CN(C(C(C=C)(F)F)=O)CC2C(F)F)ccc(Cl)c(C)c1N 86870,N1(C(C=C)=O)CCc2c(NC(C3(C)CCCOC3)=O)cccc21 86871,CC1CCC(C(=O)NC2(CO)CC(F)(F)C2)N(C(c2cn(C)cn2)=O)C1 86872,C1(CNC(=O)COC2COC2)CCCC12CCN(C(C1CCCC3CC13)=O)CC2 86873,Cc1cc(C(N2CCOC(CNC(=O)Cc3conc3C)C2)=O)ccc1Cl 86874,Cc1cc(C(=O)NC2CC3(C2)CN(C(C2CCCC2C2CC2)=O)C3)c(F)cc1F 86875,N1(C(Cn2c(C)cnc2)=O)CC2CCC1CN2C(C1CCOC(=O)CC1)=O 86876,C(CCCCCN=c1[nH]nco1)N(C(c1nc(CCC)sc1)=O)C 86877,CC1CCn2c(C(=O)N(c3cc(C4(C(F)(F)F)CC4)nc(Cl)n3)C(C)C)cnc2C1 86878,c1(OC)cc(C=CC(N2CCN(C(=O)C(C#N)C(C)C)C(CF)C2)=O)ccc1O 86879,CCCC(C(=O)N1CCC12CN(C(=O)C(C)Cc1ccnn1C)C2)S(N)(=O)=O 86880,c1(C(N2CC3C(NC(C4(C)SCCCS4)=O)C3C2)=O)cnn2ccccc12 86881,N1(C(c2c(C)ncc(Br)c2)=O)CCN(Cc2ccc(C3CC3)s2)CC1C#N 86882,c1(NC(C(c2cnc(CC)[nH]2)N2CCCC2C(=O)N(C)C)=O)ccc(F)cc1C 86883,C(=O)(C1(CC)CCCc2ccccc21)N(CCNC(C(CCC)C)=O)C 86884,C1(C(=O)NCCC(C)SC)N(C(c2cc(C)cc(O)n2)=O)CCCC1(C)C 86885,C(=O)(C(CNC(c1nccnc1OC)=O)CC(C)C)NCCCCC(=O)NC 86886,c1(C(N2CC(OCCC(=O)NC3CC(C)(C)OC3)C2)=O)cc(F)ccc1Cl 86887,CN1CC2CN(C(C3OCCC3C(C34CCC(C3)C4)=O)=O)CC2(C)C1 86888,CCCC(C)(C)CC(=O)NC1(C2CN(C(c3nc[nH]c3C(F)(F)F)=O)C2)CC1 86889,C(CNC(C1CCCCC1n1cccc1)=O)(CC)(CC)NC(COC)=O 86890,C1(C(N(CC(C)N(C(C=COCC)=O)C)C)=O)CC(=O)N(C(C)(C)C)C1 86891,c1(OC)ccc(C(N2CCC2CNC(=O)COC2CC=CCC2)=O)cc1C 86892,C1(C(=O)OC)CCN(C(=O)C2CCCN2C(=O)Cn2nnc(C)n2)O1 86893,c1(C(=O)NCC(CN(C(c2cc(CC)sn2)=O)C)C)ccc(C)nc1 86894,c1(N2CC3CCCC(NC(Cn4c(C)nnn4)=O)C3C2)ncc([N+](=O)[O-])cc1C#N 86895,C1(CNC(CONC(c2ccc(CC)s2)=O)=O)(CO)CCCCC1 86896,C(=O)(C(C)(C)C(=O)NC)N(CC(CN(C(C(CC)n1ccnc1)=O)C)O)C 86897,C(C(C)C(=O)NC1CC(C(C)NC(C2CC2C(=O)OC)=O)C1)OC 86898,N1(C(=O)CC2CCOC2)CC2(C1)CN(C(C1SCCCS1)=O)C2 86899,C1(CC(=O)NC(CNC(C(COC)(C)OC)=O)(C)C)CCCS(=O)(=O)C1 86900,N1(CCOCC=C)C(=O)CN(Cc2cnn(C)n2)C1=O 86901,C1(NC(c2ccc(CSCCC)o2)=O)C2CC1N(C(C1(CN(C)C)CC1)=O)C2C 86902,c1(C(=O)NCC2OCCN(C(C(CC)=CCCC)=O)C2)ccc2c(c1)ncn2C 86903,C1(O)(CNC(C(C(C)(C)C)SC)=O)CC2CCC(C1)N2C(=O)CN1CCCC1=O 86904,N1(C(Cc2c(F)ccc(C)c2)=O)CC2(CCN(C(=O)CCCCN(C)C)CC2)C1 86905,C(=O)(CC(C(C)OC)NC(C1(CO)COC1)=O)NCCCOC 86906,Cc1ccc(C(C)C(N2CCN(Cc3nccs3)CC2)=O)cc1 86907,CC1CN(C(C2CC3C=CC2C3)C(=O)Nc2ccc3c(c2)CCC3)c2cccnc21 86908,C=CCC(CC(=O)N(C)CC1CC(O)C1)NC(C1CC2(C1)CC2(F)F)=O 86909,c1(C(=O)NC(C2CCOC2)CNC(CCOCC)=O)c(O)cc(F)cc1F 86910,Cc1cc(F)c(C(=O)NC2CCCC2NC(=O)Cc2ccsn2)cc1F 86911,N1(C(Cc2cnc(C)[nH]2)=O)CCC(N(CCO)C(c2nccn2C)=O)CC1 86912,C1(C(=O)NCc2ccccn2)CSCCN1C(=O)CC1CC2C=CC1C2 86913,CC1(C)CCCC(C(=O)NC2CC3(C2)CC3NC(c2csc(C3CC3)n2)=O)CC1 86914,Cc1cc(Cl)c(C(=O)NC2C3CC2N(C(c2ocnc2C(F)(F)F)=O)C3)s1 86915,Cc1cccc(C(F)C(=O)NCCCCCNC(C2CS(=O)C2)=O)c1 86916,N1(C(C(C)(C)C2CCC2)=O)CC(CNC(=O)CCc2cc[nH]n2)C2(CCC2)C1 86917,c1(CC)noc(C(=O)NCC(C(C)C)NC(=O)CC2CCCOC2)n1 86918,C12(CNC(C(C)S(C)(=O)=O)=O)CCCCC1N(C(c1ccncc1)=O)CCC2 86919,CC1(C)CC(C)(C(=O)NC2CCSCC2)CN1C(=O)CC1CC(F)(F)C1 86920,c1(C(=O)NCC(c2ccc(O)cc2)O)n[nH]c2c1CN(C(=O)Cc1ccco1)C2 86921,N1(C(Cc2n(C)ncc2Cl)=O)CCCC2CN(C(c3csc(O)n3)=O)CC12 86922,CS(=O)CCCCNC(C1C=CCN(C(=O)C=CCF)C1)=O 86923,N1(C(C(C)n2cccc2)=O)CC2(CCC2)CC1C(=O)NC1C2CCCOC12 86924,N1(C(CCC2N(C(C(CSC)OC)=O)CCCC2)=O)CC(=O)NC(C)C1 86925,C1(CNC(C(c2ccc(Cl)cc2)CC)=O)C2CN(C(=O)CSC(C)C)CC12 86926,c1(CCC(=O)N(C2CC2)Cc2cccnc2S)ccc(S(=O)(=O)NC2CC2)cc1 86927,CC1CCN(C(C2CCCS2)=O)CCN1C(c1cc(Cl)ccc1F)=O 86928,C1(NC(C2C(NC(CN=[N+]=[N-])=O)CCO2)=O)CC2CC1CC2CO 86929,C1(C(=O)NCCC2(O)CCN(C(C3CCC=CO3)=O)CC2)CCC2C(C1)C2(F)F 86930,Cc1cc(C)n2nc(C)c(C(N3CCC(C)(NC(=O)C(C)S(N)(=O)=O)C3)=O)c2n1 86931,c1(C(C)NC(c2c(O)ncc(C(C)C)c2)=O)ccc2ccccc2c1 86932,C(C(C)(COC)CC)NC(C1(C)CN(C(c2nc(COC)oc2)=O)C1)=O 86933,c1(N(C)C(C2CCC2)=O)nc2ccccc2n1CCC#N 86934,N1(C(C2OCCC(C)C2)=O)CCC2(CCC2CNC(=O)CN2CCCCC2)CC1 86935,Cc1cc(F)cc2c1N(C(C1Cc3cc(F)ccc3C(=O)O1)=O)CC2 86936,N1(C(CCC(C)(C)C)=O)CC(NC(=O)CN=c2cc[nH]cc2)CC2(CCC2)C1 86937,N1(C(CN2CCN(C(C3CCCN(CC)C3)=O)CC2)=O)CC2C(C1)C2(C)C 86938,C(=O)(C1=Cc2ccccc2C1)NCC(CC(=O)N(CC(F)F)C)C1CCC1 86939,C1(CCNC(=O)Cc2csnn2)COCCN1C(=O)CC1(CC2CC2)CCC1 86940,c1(C(=O)NCC2C(NC(COCc3cccc(OC)c3)=O)C2)cc(N)cnc1Cl 86941,CCCC(C(=O)N1CC2CC(NC(C3CC4(C3)CC4(F)F)=O)C2C1)C(C)C 86942,C(CC1CCC1)(C(=O)N(C)CCC1CCCC1)NC(C(C)OCCCC)=O 86943,c1(C(=O)NC2CC(F)(CNC(C3CCC(C)C3)=O)C2)ccc2n[nH]cc2c1 86944,N1(C(C=CC(C)(C)SC)=O)CCCCC1CC(=O)NCCc1cc[nH]n1 86945,CC#CC1CCN(C(=O)C(F)CC2CN(C(c3cnn(CC)c3)=O)C2)CC1 86946,C1(C(N2C3(CN(C(c4cn(C5CCC5)nn4)=O)C3)CC2)=O)CC2CCCCN2C1 86947,N1(C(CN(C2CCCC2)C)=O)CC2C(CNC(C3CCC(C)(C)C3)=O)C2C1 86948,C1(NC(C2CC(Cl)(Cl)C2)=O)CCC2(CCCN(C(c3ccncc3)=O)C2)C1 86949,c1(NC(C(CCSC)NC(c2sccc2Cl)=O)=O)cc(C)cnc1C 86950,N(C1c2ccccc2CC1NC(=O)C(C)C(O)CC)C(c1cn(CCC)nc1)=O 86951,C1(C(=O)NC2(C=C)CCC2)CCC=CC1NC(c1ccc(C)cc1)=O 86952,c1(C(N2CCCC(NC(C3C4COCC34)=O)C2)=O)ccc(C(F)(F)F)cc1Br 86953,N1(C(CC(C)C)C(=O)Nc2ccc(Cl)cc2F)CCS(=O)(=O)CC(C)C1 86954,N1(C(C(CC2(OC)CCC2)N)=O)CCN(C2CC2)C(C)C1 86955,CC(O)CCCC(=O)N(C(C)CCNC(C1(S(C)(=O)=O)CCC1)=O)C 86956,C1(C(=O)NC(C(C(=O)Nc2c(CCC)cccc2)C)C)CC(=O)OC1(C)C 86957,c1(C(=O)NCC(CNC(CN(C(=O)OCC)C)=O)(C)F)ncncc1C 86958,C(=O)(C(CO)C(C)(C)C)N1CCC(O)(C(C)NC(=O)Cn2cccn2)C1 86959,C(=O)(C1=NOC(C)(C)C1)NC1CN(Cc2nc(C)sc2C)C(C)CC1 86960,CC(CC(F)F)C(=O)N1CCCCC(N(C(=O)COCC2CC2)C)C1 86961,CC(C)S(=O)(=O)CC(=O)NC(C)C(CO)NC(c1ccccc1Br)=O 86962,c1(C(N2CCCCC2Cc2cn(CCCCF)nn2)=O)[nH]nc([N+](=O)[O-])c1Br 86963,c1(CC)ccccc1CC(=O)NC(CN(C(=O)C(CC)NC(C)=O)CC)CC 86964,C1(N(C)CC)CCN(C(C2CCOCC2NC(C2CCN(C)C2)=O)=O)CC1 86965,Cc1ccn(C(C)CC(=O)NCC2C=CCN2C(=O)CCc2nc(=N)[nH][nH]2)n1 86966,CS(=O)(=O)C1CCCC1C(=O)NC1(c2nn[nH]n2)CN(C(=O)NC(C)(C)C)C1 86967,C1(C(=O)NCC2CN(C(c3c(SC)ccs3)=O)CC2O)CC2(CCC2)CCO1 86968,c1(C(=O)OCC)sc(NC(=O)C(=O)NCC(C)OC(F)F)cc1C1CC1 86969,C1(C(=O)NC(CCSC)C(N)=O)CC12CCN(C(=O)Cc1ccccc1Cl)CC2 86970,C1(CC(N2CCN(C)C(CNC(C3CCC=CO3)=O)C2)=O)Cc2ccccc2O1 86971,CC(C)C(C(=O)N1CCC(c2cccc(F)c2)(NC(c2cocn2)=O)C1)NC=O 86972,C(=O)(N=c1[nH][nH]c2c1CN(S(=O)(=O)CCCl)C2)c1cc(C)c(Cl)nc1 86973,C12(CC)CN(C(=O)CCCSC)C(CNC(c3sc(C)c(C)c3C)=O)(C1)C2 86974,C1(C)(C(N(C(CC)CSC)C)=O)CC(NC(=O)CN(C)C(=O)OC)C1 86975,c1(C(=O)NCC(c2cnn(C)c2)NC(C)=O)ccc([N+](=O)[O-])c(OC)c1 86976,c1(C(=O)NC2CC(C)(CNC(C3(C)ON=C(C)C3)=O)C2)cc(C)c(C)cn1 86977,N(C(=NCCN1CCSCC1)NC1CCS(=O)(=O)C1)C1C(C)C1C.N1CCOCC1 86978,c1(COC)cc(C(=O)NC(CC(=O)NC2CC(C(F)(F)F)C2)C2CC2)no1 86979,N1(C(C2(OC)CCSC2)=O)CC2CCC(C1)C(NC(=O)C1=COCCC1)C2 86980,C1(c2cn(CC(=O)OC)nn2)CCCCC1OCC(=O)NCCN1CCCOCC1 86981,N1(C(c2c(C)[nH]c(C#N)c2)=O)CCN(C(=O)C(C)(C)C2CCC2)CCC1C 86982,N1(C(C23N(C(c4cc(C)n(C)c4C)=O)CC(C)(C2)C3)=O)CCC(C)C(C)(C)C1 86983,N1(C(C(C=C)(C)C)=O)CCC(C)N(C(c2ccc(C(F)(F)F)s2)=O)CC1 86984,c1(C(=O)NC2CC(C)(NC(c3c(NC)cnnc3)=O)C2)cc2c([nH]1)CCCC2 86985,N1(C(c2c(CC)ccs2)=O)CC=CC1(C)C(=O)NC(C)CCN(C)C 86986,C(=O)(C1=CCCC1)NCCC(C)N(C(=O)CCC1CCCO1)C 86987,c1(C(=O)NCCCC(C)NC(C2CC2C)=O)ccc2c(=O)n(C)c(O)nc2c1 86988,CC1CCC(NC(=O)CCN2CCN(C)CC2)CN1C(C1SCCS1)=O 86989,c1(NC(=O)NC2CC(F)C(C(=O)O)C2)ccccc1OCc1cccnc1 86990,C(CC(O)C(=O)NC1COCCC1C(=O)NC(CO)CCO)N(C)C 86991,c1(CN(C(=O)Nc2c(C)n[nH]c2)Cc2c[nH]nc2C2CCOC2)cc(F)cc(F)c1 86992,N1(C(Cn2nc(C)n(C)c2=O)=O)CCC2CN(C(=O)C(C)n3cncn3)CC2C1 86993,C(C)(C(C(=O)NCCC(C)N(C(=O)CSc1cn[nH]c1)C)N(C)C)OC 86994,c1(NC(C2C(NC(c3ccc(CO)o3)=O)CCC2)=O)ccc2c(c1)CCC2 86995,c1(C(=O)NCC(C)(C)OCCNC(C2CCN(C)C2)=O)cccc(C#N)c1 86996,N1(C(C(=C)F)=O)CC2CCN(C(=O)Cc3ccc(O)c(O)c3)CC2C1 86997,CC1=NNC(=O)C1CCC(=O)NCC(C1CCC1)NC(C1(n2cccn2)CC1)=O 86998,N1(C(C(C)N(C(C2ON=C(C)C2)=O)C2CC2)=O)CC(S(C)=O)C1 86999,C1(C(=O)NC(C2CN(C(=O)CC3CCCC3C)CCO2)C)(OCC)CCOCC1 87000,C1(C(=O)Nc2c(C(=O)OC)scn2)CCN(C(c2cc(F)nc(F)c2)=O)CC1O 87001,N1(C(C2(N(C)C)CC2)=O)CCC(F)(C(=O)NCCC2COC(C)(C)C2)CC1 87002,N1(C(CC(C)=C(C)C)=O)CCN(C(c2cnn(C)c2)=O)CC(O)C1 87003,C1(C(=O)NCCC2(C(N(CC(F)F)CCOC)=O)CC2)OC2CCC1C2 87004,C(=O)(CCCCOC)N1C(C(C(=O)NCc2cn(CC=C)nn2)C)CCC1 87005,C1(NC(=O)Cn2ccnn2)CN(C(=O)C=Cc2ccncc2)C2(CCOC2)C1 87006,C(=O)(C1=COCCO1)N(CCN(C(=O)C(N1C(C)CCC1C)C)C(C)C)C 87007,c1(CC(C)(C)NC(=O)NCC(C(=O)O)C2C(OC)C2)ncccc1C 87008,C1(OCC)(NC(=O)NCC2COC3CC2C3)CCCCC1 87009,N1(C(C(CCC)OC)=O)CC(CNC(=O)CCn2cncn2)C2(CCOCC2)C1 87010,N1(C(CCN(C)CC)=O)CC2(CC(NC(=O)C(C)C3CC3)c3nccn32)C1 87011,C(=O)(CC(C1CCCC1)NC(=O)CC(C)c1cnn(C)c1)OC 87012,CON(C)C(=O)C1(NC(=O)C(O)C2CCCC2)CCC1 87013,C12(NC(C(C(C)OC)NC(=O)Cc3cccnc3)=O)CCCN(CC1)C2 87014,C(=O)(C1Cc2c(Cl)cccc21)N1C(CNC(C2(C)CCC(=O)CC2)=O)CC1 87015,C1(Cc2cn(CCOCC)nn2)COCCN1C(c1cc(-c2ccco2)[nH]n1)=O 87016,c1(C(C)S(=O)(=O)NCC2(O)CCNC2)cccc(Br)c1 87017,N1(C(=O)Cn2cc(C(c3ccc(F)cc3)O)nn2)CCCC(O)C1.CO 87018,Cc1cc(=NCc2ccc(C(C)(C)C)o2)[nH]cc1S(=O)(=O)NC(c1ccco1)C 87019,c1(CC)cn2c(n1)CC(c1nc(CC3CCCCC3)nn1C1CSC1)CC2 87020,c1(NC(C2(C)CN(C(c3cc(F)c(F)cc3I)=O)C2)=O)ncc(Cl)cc1[N+](=O)[O-] 87021,c1(CC)sc(C(N2CCC2CNC(=O)CC(C)(C)F)=O)cc1Br 87022,c1(N2CCN(OCC)CC2)nc(=NC2CCC(N(C)C)C2)[nH]c2c1ncn2CC 87023,Cc1nc(C(N2CCC(F)(CNC(=O)CC3NC(=O)NC3=O)C2)=O)sc1C 87024,c1(C(=O)NC(C2CCCC2)CNC(C(C)c2ccsc2)=O)c(F)cccc1F 87025,C1(C)(C(=O)Nc2cccc(C(C)C)c2F)COC(C)(C)OC1 87026,c1(SC)nccc(N2CC(CNC(=O)C(c3cccc(F)c3)C)CC2C)n1 87027,C#CC1(C(=O)NOCC2CCCO2)CN(C(=O)C=CCF)C1 87028,Cc1cc(CC(N2CC(C(C)(C)O)(CNC(C3(C)CC3(F)Cl)=O)C2)=O)c(C)s1 87029,CC1CC(C(N2CCC(CCNC(=O)CC3CCCCO3)CC2)=O)CCO1 87030,Cn1nccc1C1CC1C(=O)NC(C)(CNC(=O)COc1cccnc1)CO 87031,C(CN=C(NCC(F)(F)CO)N1CCN(Cc2ccc(Cl)cc2)CC1)OCC=C 87032,Cn1cc(CN2CCCC(NC(C3CNC(=O)C3)=O)CC2)c2ccc(F)cc12 87033,Cc1cc(CNC2C3CN(C(=O)CSc4ccccc4)CC23)c(C)s1 87034,N1(C(C(C)NC(CC)=O)=O)CC(OC)C(NC(=O)CCc2cncs2)C1 87035,C(=O)(CCC(C)(C)C)NCCN(C(=O)Cn1cc(C2CCOC2)cn1)CCOC 87036,c1(C(C)C)ccc(C(=O)NCC2CCN2C(=O)CC2CCCCC23CC3)cc1F 87037,C(=O)(C(O)C(C(C)C)OC)N1C(C(=O)NCC(=O)NC)CC1 87038,Cc1ccc(F)c(CNC2(C)CCCCC2C(=O)OC(C)(C)C)n1 87039,c1(N(CC(CN(C)C)(C)C)C)nc(N2CCN3CCCCC3C2)nc2cc[nH]c12 87040,C1(NC(CC2CC(C(=O)OC)C2)=O)CCCC12CN(C(=O)C(O)Cc1ccccn1)C2 87041,C1(NC(CCOCCOC(C)(C)C)=O)CC2CC(NC(C3(O)CCSC3)=O)CC12 87042,C(=O)(C1=COCCO1)N(C)CC1CCCN1C(C1(C)CCCO1)=O 87043,c1(OC)cc(CN2C(C(=O)Nc3ncc(F)cc3Cl)CC3CC23)cc(O)c1O 87044,C1(CNC(C(CC)(C)O)=O)CC(F)CN(C(=O)CCc2cncc(Br)c2)C1 87045,C(=O)(CC(C)C(C)C(C)C)N(CC(CC)NC(c1[nH]c(C)cc1C)=O)CC 87046,C1(OCC)CN(C(c2ccn(CC)c2C)=O)CC1CNC(=O)CC(C)(C)O 87047,c1(OC)cnc(C(=O)NCCCNC(c2cc(-c3cccs3)on2)=O)nc1 87048,C12(CNC(C3N(CC)C(=O)CC3)=O)CN(C(C3CCCO3)=O)CC(F)(C1)C2 87049,CC(C)C(O)C(=O)N(C1CN(N2CCC2)C1)C.C1(CC=O)(C(F)(F)F)COC1 87050,C(=O)(CS(=O)(=O)C1CCCC1)N(C1CCN(Cc2cccc(F)c2)CC1)CC#C 87051,CC1(CNC(c2cnn(CCF)c2)=O)CCCN(C(C23CCC(CC2)CO3)=O)C1 87052,c1(C(=O)NCCNC(=O)Cc2ccccc2OC(F)F)cc(Br)cnc1S 87053,C1(NC(CC2(C=C)CC2)=O)CN(C(c2cc(CC)ccn2)=O)CC1C 87054,N1(CCC)CC(C(=O)NCCC2CN(C(c3cc(O)cs3)=O)C2)CC1=O 87055,C1(C(=O)NC2(CC3CCC3)CC2)OCCC1C(F)(F)F 87056,c1(C(N2C(CNC(C(CCC)CC(C)C)=O)CC2)=O)cccc2nc(O)ccc12 87057,CCC(CC(=O)NCC1(CNC(=O)C(C)(C)c2cccs2)CC1(F)F)SC 87058,CN1C(=O)C(N(C(=O)CNC(=O)C(C)(C)C)C)CCc2ccccc21 87059,N1(C(C(CC=CC)OC)=O)CC2CC1CN(C(=O)C(C)NC(C)(C)CC)C2 87060,C1(NC(COCCC#C)=O)CC2CC(NC(c3ccc(C=CC(=O)OC)o3)=O)C1C2 87061,C(N=C(NC1CCC1)N1CCC(NC(C)=O)C1)c1ncc(CC)s1 87062,C(=O)(C(C)(C)CCS(C)(=O)=O)NC1CCN(C(c2cc(CC)n(C)n2)=O)C1C 87063,c1(C(N2CCC3(CC2)CC3CO)C(=O)NCC(C)C)nccc2cc(Cl)ccc12 87064,C=CCC(C)(CC)C(=O)N1CCCN(Cc2cn(-c3ccccn3)nn2)CC1.OCC 87065,O=C1Cc2c(C(N3CCC(CNC(c4cnc(O)o4)=O)CC3)=O)cccc2N1 87066,C(=O)(C(Cn1cccn1)NC(=O)C(c1ccccc1)=O)N(C)C 87067,N1(C(CC(C)OCC)=O)CCN(C(c2ccc(OC(C)C)nc2)=O)CC12CC2 87068,C1(C(N2CC(O)(C(C(=O)N(C(C)C(=O)NC)CC)F)C2)=O)CC12CCOCC2 87069,C1(NC(c2cccc(C(C)=O)c2)=O)CCN(C(=O)CN(C)C2CC2)CC1C 87070,CC(CCC(C)(C)C)C(=O)NCC1CC(C(N2CC3(CC(F)C3)C2)=O)C1 87071,C1(NC(c2c(C)n3c(s2)cnc3)=O)CCCC2CN(C(c3ccccc3)=O)CC12 87072,c1(CS(=O)(=O)NC2(COC)CC(O)C2)cccc(C(F)F)c1 87073,Cc1sc(C(=O)NC(C)(CNC(=O)C(C(C)O)N(C)C)CO)nc1O 87074,C1(COC)(NC(c2cc(C)nn2C)=O)CCN(C(C2CC23CCC3)=O)CC1 87075,c1(C(=O)NCc2cc(C(=O)NCCSCC)no2)cc([N+](=O)[O-])n[nH]1 87076,C=CCC(C(=O)NC1CC1NC(=O)Cc1sccc1C)NC(=O)OC(C)(C)C 87077,C1(NC(C2CC(CNC(C(n3ccc(C)n3)C)=O)OC2)=O)CCC=CCCC1 87078,CC(CC(F)F)C(=O)N1CC(NC(c2cnc(Cl)s2)=O)C(C(F)F)C1 87079,C1(C(=O)NC2CCN(C(C(CCC)NC(N)=O)=O)C2)CCC2(CCCCC2)CC1 87080,c1(C(N2CCC(COC)(NC(=O)CC34CC(C3)C4)CC2)=O)cc2c([nH]1)CCCC2 87081,c1(NC(C2(C#C)CN(C(C3CCCCC(=O)C3)=O)C2)=O)ccc2c(c1)CCC2 87082,CC1CN(C(C2(CNC(=O)C(C3(O)CCCC3)F)CCCCC2)=O)CC1O 87083,Cc1cc(C)c(C=CC(=O)NC2CN(C(c3cc(C)[nH]c3C)=O)C2)c(C)c1 87084,O=C(CC1=CCN(C(C2CC(=C3CC3)C2)=O)CC1)Nc1coc(CO)c1 87085,C1(NC(c2nnc(C)s2)=O)CN(C(c2ccc(N(C)C)cc2F)=O)CC1C1CC1 87086,C12(C(=O)NC34C(CN(C(c5cc(CC)ncc5)=O)C3)C4)CCC(CC1)OC2 87087,C1(C(C#C)C)CCN(C(C2CCC2CNC(C2(C)SCCCS2)=O)=O)CC1 87088,C1(C(=O)NC(CC(C)NC(c2cc(C)n(C)c2)=O)C)CN2CCN1CC2C 87089,CON(CCC(=O)Nc1cn(C2CC2)nc1C)C(=O)CC1CCC(O)C1 87090,c1(CC(=O)NC(C2CCN2C(=O)CCc2cn(C)nn2)C)noc2ccccc12 87091,N1(C(C(C=C=C)C)=O)CC(C2CCN(C(=O)Cn3ccc(=O)n(C)c3=O)CC2)C1 87092,C#Cc1ccc(NC(C23CC(C)(CN2C(=O)C(C)(C)CCCOC)C3)=O)c(C)c1 87093,C1(C2CN(C(C3CCC(C)O3)=O)C2)CN(C(=O)CCc2ccncc2)CCO1 87094,C12(NC(CC(C(=O)OC)C)=O)CCC(CN(C(C3(CCF)CCC3)=O)C1)C2 87095,C(=O)(CCCC(=O)NC(CNC(=O)CSCc1cccs1)C(C)C)NCCC 87096,CS(=O)(=O)c1ccccc1NC(C1CSCCN1Cc1cncc(Cl)c1)=O 87097,N1(C(C(=O)N(CCC)CCNC(=O)C(c2ccccc2)OC)C)C(=O)CCC1=O 87098,Cc1nnc2n1CC(C(N1CC3(C1)CN(C(=O)CC(C)C)CC3CO)=O)N(C)C2 87099,c1(N2CC(N)C2)ccc(C2SC(=O)CS2)cc1 87100,C1(CNCc2cc(F)cc(C(F)(F)F)c2)CCC2COCCC2C1 87101,C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CCCC=C)C(=O)N1CCOC(C)C1C 87102,c1(C(N(C)CC2OCCN(C(C(CC)(C)F)=O)C2)=O)ccc(S(N)(=O)=O)s1 87103,c1(C(=O)NCC2N(C(C(C)=C3CCC3)=O)CC(C)CC2)ccc2sccc2c1 87104,c1(C(=O)NC(C2CCCN2C(=O)Cc2cncs2)C)nc[nH]c2ncnc1-2 87105,C(=O)(C1CCc2nccn21)N(C1CCN(C(c2cc3cc(N)ccc3s2)=O)C1)C 87106,CON(C(=O)C1=CCC(NC(c2ccc3occc3c2)=O)C1)C1CCC1 87107,c1(CN2CC(NC(C(CCC)C)=O)C(F)C2)cc(Br)cc(Cl)c1O 87108,c1(C(c2n(CC=C)nnn2)NC(Cc2ccccc2)CC)nc(F)ccc1Br 87109,c1(C(=O)NCC2(CN(C)C(C3(CCF)CCC3)=O)CC2)ccc2n[nH]cc2c1 87110,N1(CC)CCC(N=c2[nH]c3c(c(=NCCSC)[nH]2)COCC3)C(C)C1 87111,N1(C(Cc2cc(C)on2)=O)CC(NC(C2(C)CC2(C)C)=O)C(C)C1 87112,n1(CC)ccc(C(=O)NCC(C)CNC(c2scc(C)c2Cl)=O)cc1=O 87113,CN1CCOCC1CC(N1CCC(O)(CNC2(c3cccnc3Cl)CC2)C1)=O 87114,Cc1nsc(N2CCN(CCNC(C3CC(=O)N(C)C3)=O)CC2)c1C#N 87115,N1(C(c2ccnc(C)n2)=O)CCCC2C1CCN2C(C1CCCCC1)=O 87116,C=CC1(C(=O)NCC2C3CCCCCC23)CCN(C(C2CCC(C)(O)CC2)=O)C1 87117,c1(C(=O)NCC(=C)CCNC(c2cc(-c3cccnc3)on2)=O)oc(C)cc1C 87118,C1(C(=O)NCCCCC(=O)NC)CCC2(CC2)N1C(C12CCCC1OCC2)=O 87119,C1(CN(C(=O)CC2CCCC2C)C)COCCN1C(=O)CCC1(C)N=N1 87120,Cc1nn(C)c(C)c1C(=O)NCCCN(CCCNC(c1ccsc1)=O)C 87121,c1(C(N2CCC(CC#C)(C(=O)N(CCF)CCOC)C2)=O)cc(F)ccc1F 87122,N1(CC)CCOC(C(=O)NC(C)CNC(=O)C(c2ccc(F)cc2)C2CC2)C1 87123,C=CCC(C)C(=O)NC1COCCC1NC(=O)C=CC(C)(C)SC 87124,C1(NC(CCC#CC)=O)C2CCN(C(=O)Cn3cc(Br)cn3)CCC12 87125,n1(C23C(C)OC(CC2)C3)c(-c2ccccc2)csc1=Nc1ccc(Cl)c(F)c1 87126,C1(C(C)NC(C=CC(CC)C)=O)CCCCN1C(=O)CCN(C)CCOCCO 87127,c1(C(=O)NCCn2cc(CNC(CC(C)OC)=O)nn2)cccnc1S 87128,C1(F)(CNC(c2cn[nH]c2)=O)CN(C(=O)C(F)(F)c2c[nH]nc2O)C1 87129,c1(NC(C2CCN(C(=O)CCF)C2)(C)C)cnc(C(=O)OCC)s1 87130,N1(C(C(CNC(C2CCCC(F)C2)=O)N(C)C)=O)CCn2cncc2C1 87131,c1(C(=O)OC)ccc(OC(=O)NC2COC(C(F)F)C2)c(OC(F)F)c1 87132,c1(CC(C)C)ccc(C(N2CC(NC(C3CSCCS3)=O)C(F)C2)=O)cc1 87133,c1(C(C(N2CCC(CNC(C(CC)(C)C)=O)C2)=O)(C)C)ccc2ccccc2c1 87134,N1(C(C(CC)=CC)=O)CC2C=CC1C(C(N1CC(CCC)C1)=O)C2 87135,C1(C(N2CC(CC(C)NC(=O)COCCCN(C)C)C2)=O)CCC12CCOCC2 87136,C=CC1CN(C(=O)C(C(C)C)SCC)CC1NC(c1c(C)c[nH]c1CC(N)=O)=O 87137,n1(CCC(=O)OCC)nnnc1C(c1cnccn1)NCC(C)C(C)C 87138,C(=O)(C#CC1CCCOC1)N1CCC(C)C(NC(c2cc(O)cnc2N)=O)C1 87139,C1(C(=O)NCC=CCSC)CCC(C)(C)N(C(C2CCCO2)=O)C1 87140,c1(CNC(C=CCNC(c2cc(C)c(C)o2)=O)=O)nn(C)c(=O)n1C 87141,N1(C(c2cc(C)c(C)o2)=O)CC(O)CC1(C)C(=O)NCCCCF 87142,c1(CCC(=O)NC(C)CC(C)NC(c2cncc(F)n2)=O)ccc(C#N)cc1 87143,O=C(C1CCCc2c[nH]nc21)NCC1CN(C(=O)Cc2ccc(Cl)cc2)CCO1 87144,N1(C(c2ccc(CNC(Cn3ncc(C)c3)=O)cc2)=O)CC(O)CC12CCC2 87145,c1(CC)cc(C(=O)NC2COCCN(C(C3C(C)(C)C3(F)F)=O)C2)c(C)nn1 87146,C1(C(N2CC(C#C)(F)C2)=O)CC2C=CC1N(C(=O)CC1C(C)(C)C1(C)C)C2 87147,O=C(CCS(=O)(=O)c1ccc(F)cc1)NC1CCOC(C2CCOCC2)C1 87148,c1(CNC(c2cnn(C)c2)CC)cccc(CC(F)(F)F)c1 87149,C(=O)(C(CCCCCCO)N1CCC1(C)CCO)NCCSC 87150,c1(C(N(CC)CC2CCCO2)=O)oc(CNC(=O)CC(C)C2CC2)nc1C 87151,C1(NC(COCCCC#C)=O)CCCC(C(N2CCC(C)(C)C2)=O)CC1 87152,N1(C(c2cnc(CC)nc2)=O)CCCC(C)(C)C1C(=O)NCC(F)C(C)(C)O 87153,c1(N2C(CC)CN(C(C3CCC(=O)N3)=O)CC2)ncnc2c1ccn2C(C)C 87154,c1(C(=O)NCC(CCNC(C(CCC)N(C)C)=O)O)cc(C)c(Cl)c(C)c1 87155,C1(CNC(C(CC)NC(c2n[nH]cc2Cl)=O)=O)C2CCCCCC12 87156,N1(C(C(CC)(C)OC)=O)CCC2(C1)CN(C(c1ccc3nn[nH]c3n1)=O)CCO2 87157,N1(C(COCC=C)=O)CCC(CCNC(c2cc(C)nnc2O)=O)C(F)(F)CC1 87158,c1(C(=O)NC2C(NC(C=C(C)Cl)=O)CCC2)[nH]c2ccc(Cl)cc2c1Cl 87159,C1(F)(C(=O)OC)CC1C(=O)NCC(=O)NC(=O)C1CC1.C(C)(=O)O 87160,CC1(C)CCOC1NC(=O)CC1CC(C(=O)OC(C)(C)C)C1(C)C 87161,c1(C(=O)NCC(CCOC)NC(=O)C(C)OC)cncc2nc(C)[nH]c12 87162,C(C)(C)(C(C)NC(=O)C(C)(C)F)NC(C=C(C)C(C)C)=O 87163,C(C(=O)NCC(CO)NC(=O)COCc1cccc(C)c1)(C(C)(C)C)NC(C)=O 87164,c1(C(=O)NC2C(OC)CN(C(c3csc(CC(C)C)n3)=O)C2)cnc(C)c(C)c1 87165,CP(C)(=O)c1cncc(C(N2CCCC(NC(=O)COC3CCOC3)C2)=O)c1 87166,N1(C(CNC(CC)=O)=O)CC(CNC(c2cnccc2Cl)=O)C2(CCC2)C1 87167,C1(C(N(CC(=C)C)CCOC)=O)CCCC(NC(c2ccncc2)=O)C1 87168,c1(NC(C2N(Cc3cnc(OC)c(Br)c3)C3C(C2)C3)=O)ccc(F)cc1[N+](=O)[O-] 87169,N1(C(c2c(C)nccc2)=O)CCC2C1CCN2C(c1cc2cccnn2n1)=O 87170,c1(OC)cc(F)c(C)cc1NCc1ccnc(Br)c1Br 87171,C(CCCC(=O)N1CCC(F)(CNC(c2cc(C(C)(C)C)no2)=O)C1)OCC 87172,N1(C(C2(C#N)C(C)C2)=O)CC2CCC1CN2C(c1nc(C2CC2)cs1)=O 87173,O=C1CCC(O)CN1c1cn(CCOCc2cccnc2OCC(F)F)nn1 87174,C(C(CC(F)(F)F)NC(c1snc(O)c1Cl)=O)NC(C(C(C)C)OC)=O 87175,C1(O)(C(C)NC(CCOCCC)=O)CCN(C(=O)CNC(=O)C(F)(F)F)C1 87176,CCC(C(=O)NC1(CNC(=O)Cc2ncoc2C)CCCC1)NC(C)=O 87177,C1(NC(CC2(C#N)CC2)=O)CC(O)CN(C(=O)Cc2csc(C3CC3)n2)C1 87178,N1(C(CCCCOCCC=C)=O)CCC2CN(C(=O)CC(COC)COC)C2C1 87179,C(=O)(C(CCS(C)(=O)=O)c1ccccc1)N(C(C(C)O)C)CCO 87180,C1(NC(C2(C)CCN(C(c3cc(C(N)=O)[nH]n3)=O)C2)=O)(CO)CC2CCCC12 87181,C1(CNC(c2c(C(C)C)ocn2)=O)CCCC2CN(C(C3(C#N)CCC3)=O)CC12 87182,CC(C)CC(O)C(=O)NCC1(F)CCCN(C(=O)CN2CCCCCC2=O)C1 87183,Cc1ccc(O)cc1C(=O)N(CCC(=O)NC1CCCCC1(C)O)CC1CC1 87184,CCC(C(=O)NC1CC(NC(C2(CC(C)C)CCC2)=O)C1)C(C)(F)F 87185,N1(C(c2cc(C(C)C)no2)=O)CCC(C(=O)NC(c2cncc(F)c2)C)C12CC2 87186,N1(C(C2CCC(C(=O)OC)O2)=O)CC2(CNC(=O)C(O)C(C)(C)C)CCC1CC2 87187,N1(C(C(Br)=C(C)C)=O)CC2CCC(NC(=O)Cc3cccc(F)c3F)CC2C1 87188,c1(C(=O)NC(C2CCCCN2C(=O)Cc2ccccc2)C)cc2c[nH]cnc-2n1 87189,c1(CC(=O)NCCN(C(=O)C=C2CCN(C)CC2)CC)cc(F)cc(Br)c1 87190,C12(CNC(c3n(CC)ccc3)=O)CCCC1CN(C(=O)Cc1ccn(C)n1)C2 87191,N1(C(CC=CC)=O)CCC2CCC12CNC(c1c(O)cccc1Cl)=O 87192,C(CCCC(=O)NCC(C)(Cn1cccn1)NC(=O)CCc1ncco1)SC 87193,C(=O)(C(C(=O)NC1(C(=O)NC2C=CCCCC2)CCCCC1)OC)OCC 87194,c1(C(=O)NC(CNC(CC(=C)Br)=O)C)cn(C)nc1OCC(F)F 87195,C=CC(C)(CC)C(=O)NCc1csc(CNC(c2[nH]c(C3CC3)nc2C)=O)n1 87196,N1(C(C)C)CC(C(=O)NC2CC(NC(C34CC(CCO3)C4)=O)C2)CCC1=O 87197,C1(NC(CC2N(C)CCC2)=O)CCC2(CC1)CN(C(=O)CC1CC3(CCC3)C1)C2 87198,C1(C(N(C2CCCN(C(CCn3ccc(C)n3)=O)C2)C)=O)CN2CCC1(C)CC2 87199,Cc1oc(C#N)cc1C(=O)NC12CC1CN(C(c1ccnn1C(C)(C)C)=O)C2 87200,C(=O)(C(C(C)C)NC(N)=O)N(CCCN(C(C(C)=CC)=O)C)C 87201,c1(C(=O)NCCCOCCC(=O)NCC2(CCC)CCC2)cc(C)ncc1C 87202,N1(C(CCC(CCC)CC)=O)CCC2CCCC(C1)N2C(=O)CC(O)CC(C)C 87203,C(CCC(=O)NC(c1cn(C)nn1)C(=O)NCc1ccn(CC)n1)=CCC=C 87204,N1(C(CCCOCC)=O)CCN(C(c2ccc(C)cn2)=O)C2CC12 87205,N1(C(c2[nH]nnc2C2CCCN2C(=O)C(F)(F)F)=O)CCSCC1C1CC1 87206,C1(C(N(C)CC2CN(C(=O)C(O)c3ccsc3)C2)=O)CCCN1C1CCCCC1 87207,[N-]=[N+]=NC1CCN(C(=O)NC2C=CCC2)C1 87208,c1(C(=O)NCC2CCCNCC2)cc2cc(Cl)cc(Cl)c2[nH]1 87209,N1(C(c2c(C)[nH]nc2Cl)=O)CCN(C(=O)CC2CNC(=O)C2)C(CC(F)F)C1 87210,N1(C(c2ccn(C)n2)=O)CCC(NC(c2cnn(CC(F)F)c2)=O)C(CO)C1 87211,c1(N(C(C)=O)C2CC2)ccc(CN2CCC(Nc3ccnc(C)n3)CC2)nc1 87212,CC(C(=O)NCC1CC(NC(=O)Cc2cccs2)CCO1)C(F)(F)F 87213,C(=O)(C(C)S(C)(=O)=O)N(C(C)C(N1CCCC(CN=[N+]=[N-])C1)=O)C1CC1 87214,C#CCC(CC(=O)OC)NC(=O)CC(CCC)NC(=O)C1=C(C)CC1 87215,C1(CNC(=O)C(C(F)(F)F)C(F)(F)F)CN(C(=O)C2CC2)CCC12CCOC2 87216,c1(C(N2CCN(C(C3CC(C#C)(O)C3)=O)CC2)=O)cc(Cl)c(Cl)n1C 87217,c1(OC)c(C(N2CC3CCN(c4nccc(SC)n4)C3C2)=O)cccc1[N+](=O)[O-] 87218,c1(C(=O)NCC(CN(C(=O)CC23COC(C)(C2)C3)C)O)c(N)cccc1Cl 87219,C1(CC)C(C(=O)N(C(C)CN(C(=O)C=Cc2ccco2)C)C)CCN1C 87220,CC1=NNC(=O)C1C(=O)NC(c1ccccc1)Cc1ccc(F)cc1 87221,N1(C(C2=NNC(=O)C2)=O)CC2(CCC2)CC1CNC(C1CCOCC1)=O 87222,C(C(=O)NNC(=O)C#CC1CCCOC1)CCN(C)C(=O)OC(C)(C)C 87223,Cc1noc(C(=O)N(C)CC2CCCCN2C(=O)COC2CCOC2)c1C 87224,C1(C(N(C(C)CNC(=O)COC2CC=CC2)C)=O)CCN(C)S1(=O)=O 87225,c1(C(=O)NC2CCCCC2NC(=O)COCC2CCOC2)cnc(OC2CC2)cn1 87226,C#CCCN=C(NC1CC(OC)C1(C)C)N1CCC(C(=O)OC)(CC)C1 87227,Cc1n[nH]c2cc(C(=O)NC(CNC(=O)CCC3CCCO3)C(C)C)ncc12 87228,C(=O)(C(=O)N(C)C)N(CC(C)N(C(C1C(CC(C)C)C1)=O)C)C 87229,c1(CN2CCC2=O)ccc(OC)cc1.c1(CCN(CC=C)C)ccon1 87230,N1(C(c2ncoc2C(F)(F)F)=O)C2CCCC1CC(NC(C1(O)CCCC1)=O)C2 87231,C(C)(C)(CCC(=O)NC1CC(C)CCC1O)NC(c1ncn(CC)c1)=O 87232,C1(C(C)C)CN(C(=O)C2=NNC(=O)C2)CCCN1C(c1coc(C(C)(C)C)n1)=O 87233,Cc1ccc2c(CC(=O)NC(C)(C)CCNC(C3CC(F)C(=O)N3)=O)c[nH]c2c1 87234,c1(C(=O)NC2C(NC(C(CC)OCC)=O)C2)ccc(-n2cccc2)nc1 87235,C#CC(CNC(=O)C(C(C)(C)C)n1cc(C2(O)COC2)nn1)CC(C)(C)C 87236,C(=O)(C(C)S(N)(=O)=O)NCC1(O)CC(NC(c2c(C)ccn2C)=O)C1 87237,n1(CC(=O)NC2CC(NC(CCCn3c(C)ncc3)=O)C2)ncc2ncccc12 87238,N1(C(C2C(C)C2C)=O)CCN(CC2CCCN(C(C3CC(F)(F)C3)=O)C2)CC1 87239,CC(C(=O)N1CC(n2cc(C3(O)CCOC3)nn2)CO1)N1CCOC1=O 87240,c1(C(N(C(C)CNC(C2CCCCS2)=O)CC)=O)cccn2cc(C)nc12 87241,c1(C(=O)NCC2N(C(C(C)NC(=O)O)=O)CCC2)n[nH]c2c(F)cccc12 87242,N1(C(CC(C)(C)CC(F)F)=O)CCC2(CCC(CN=c3ccnc[nH]3)O2)CC1 87243,N1(C(=O)CC2CCCOC2)CCC2(C1)CN(C(c1cc3occc3s1)=O)C2 87244,CCC(COC)C(=O)NCCC(C)N(C(=O)CC1CC=CCC1)C 87245,C1(O)(C(C)NC(=O)C=CC(=O)N(C)C)CCN(C(C2CC(=O)CO2)=O)CC1 87246,O(C1CCc2c(Br)cccc21)C(c1ccc(C2CCC2)cc1)=O 87247,C1(C(=O)NCCN2CCCC(C)C2)CC2(CCN1C(c1n[nH]c3c1CCC3)=O)CC2 87248,C(c1c(F)ccc(Cl)c1F)=CC(N1CCC(NC(C(CC)=CC)=O)C1CC)=O 87249,c1(C(N2C3CC(C(=O)NCCC(O)CO)C2CC3)=O)ccc2nccc(Cl)c2c1 87250,N1(C(C=Cc2ncc(C)[nH]2)=O)CCOC(C)C1C(=O)NCCC(CO)C(C)C 87251,CCC(CCC(=O)NCc1cc(C)ns1)NC(C1(CCN(C)C)CCC1)=O 87252,C(=O)(C#CC1CCCCO1)N1CCCC(CNC(c2c(C)cn(C)c2)=O)CC1 87253,Cc1nccc(CN(C)CC2CCCCN2C(c2nc(Cl)oc2C)=O)n1 87254,C1(NC(C(CC#C)C2CC2)=O)CC12CCN(C(c1ccc(Cl)c(C)c1N)=O)CC2 87255,c1(C(=O)NCCN(C(=O)CCc2cnoc2)CC(C)O)cccc2ccccc12 87256,Cc1cc(N2CCOC(CN(C)C(C3CC3Cc3ccccc3)=O)C2)nc(Cl)n1 87257,Cc1cnccc1C=CC(N1CCOC(CNC(c2nnc(O)cc2O)=O)C1)=O 87258,C12(C(=O)NC(c3cccnc3O)C)CCC(NC(=O)Cc3cncs3)(CC1)C2 87259,N1(C(C2C(C)N(C)CCC2)=O)CCCC2(CCc3ccccc3O2)C1 87260,C(=O)(CC(C(F)(F)F)S(=O)(=O)N(CCC(F)F)C1CC1)OCC 87261,CC(CC(C)(F)F)C(=O)OCC1OCCCO1 87262,N1(C(CCc2cc(C)no2)=O)CC2CCC(C1)N2C(c1cc(C)c(Cl)cc1C)=O 87263,N1(C(CC(C)=C(C)C)=O)CCC2(CC2C(=O)NCc2nnc(O)n2C)C1 87264,C12(C(=O)NCC(CC)C#N)CCC(CC1NC(C1CC3(C1)CC(O)C3)=O)C2 87265,c1(C(N2C(CNC(=O)C3=COCCC3)CC(C)(C)C2)=O)ccc2c(c1F)CCC2 87266,C(=O)(CCCCN(C)C(c1ncccc1Cl)=O)NCC(CC1CC1)OC 87267,C(C(=O)N(CCC(=O)NCCCn1ccnc1)CCO)(C(C)C)NC(C)=O 87268,c1(C(=O)NC(CN(C(C2CC(=C)C2)=O)C)(C)C)cc(CC)nnc1C 87269,c1(CNC(C2(COCC)CCC2)=O)c[nH]nc1OC.C12C(C1(F)F)CNC(=O)C2 87270,C#Cc1ccc(C(=O)OCC(C2CC3C=CC2C3)=O)cc1 87271,CS(C)(=O)=Nc1ccc(C(N2CCN(C(=O)CC3CCOC3)C(CF)C2)=O)cc1 87272,Cc1nc(O)nc(C)c1CC(=O)N(CCNC(C1CCCN1C(C)C)=O)C(C)C 87273,c1(N2CC(C(=O)Nc3ccc(-c4cn[nH]c4)cc3)C(O)CC2)ncnc2occc12 87274,c1(CC)ncncc1C(=O)NC(C1CCN(C(=O)CCc2cccnc2)C1)C 87275,C(C(C)C(F)C(=O)Nc1cn(C)nc1C#N)NC(c1ccnc(OC)n1)=O 87276,c1(C(=O)OC)ccnc(NC(C2CCCC(NC(c3cscc3C)=O)C2)=O)c1 87277,C12(C(N3C(C)(C(=O)NC)CC3)=O)C(NC(=O)C(C)C#N)C3CC1C2C3 87278,C1(NC(C2(C)CC=CCC2)=O)CN(C(c2cc(Cl)cnn2)=O)CCC1F 87279,C1(NC(C(C)N(C)C)=O)CCN(CC2CCC(C)C2)CC1(C)C 87280,c1(C(=O)OCC)ccccc1N.c12cncc(c1)OCC(=O)N(C1CC1)C2.OC 87281,Cn1nccc(C(=O)NC2CN(C(=O)Cn3nccn3)CC2O)c1=O 87282,N1(C(CC=C)=O)CC(NC(c2ccnc(CC(C)C)n2)=O)CC(F)C1 87283,N1(C(CCc2c(C)ncs2)=O)C2CCCC1CN(C(=O)CC1CCC3CC13)C2 87284,c1(OC)c(CN(C)Cc2ccc(-c3cccs3)cc2)cccc1Cl 87285,C1(C)(C(=O)NCC(=C)CCNC(c2cc[nH]c2C(=O)OC)=O)CC(O)CN1C 87286,C1(c2nnnn2Cc2nocc2Br)(NCCSC)CCC(c2ccccc2)C1 87287,C12(C(N3CCCCC(NC(CC4N(C)CCC4)=O)C3)=O)CCC(CO)(CC1)CC2 87288,N1(C(C2N(CCCC)CCCC2)=O)CCC(C)(C)C(C(=O)N(C)C)C1 87289,C(C(C(=O)N(C)CC1(O)CCOC1)C(C)(C)C)NC(C(C(=O)OCC)(C)C)=O 87290,c1(C2(C(=O)NC(CC(C)NC(=O)C(C3CCCC3)N(C)C)C)CC2)ccc(O)cc1 87291,c1(CC)cccc(C(=O)NC2CC(NC(=O)Cc3c(Cl)cnn3C)C2)c1F 87292,[N-]=[N+]=NC1CN(C(=O)CC2CC(=O)NC2=O)CC1NC(=O)Cc1cncnc1O 87293,N1(C(c2cccc(OC)n2)=O)CCN(C(=O)C(C)OC(C)(C)C)C(C)C1 87294,CC1(C)CCCC(CC(N2CCN(C(c3ccnc(S)c3)=O)CC2C2CC2)=O)O1 87295,c1(C(N2C(CNC(C(C)CC(C)(C)C)=O)CCCC2)=O)c2c(nn1C)CCCC2 87296,C(=O)(CC(C)C)NC1(C(=O)OCC)CC1.C12(CSC1)C(=O)NC2 87297,c1(CC)nc(O)c(C(N2CCC3(NC(=O)CC4CCSCC4)CC3C2)=O)cc1C 87298,N1(C(c2ccc(C#C)o2)=O)CCCCC2C1CCCN2C(=O)C(F)C(C)C 87299,C1(C(=O)NCC2(C#C)CCOCC2)CC2(CCC2)CN1C(=O)CC1CCCCO1 87300,Cc1scc(C(=O)NCC2CN(C(C3(Cl)CC3(F)F)=O)CC2O)c1N 87301,C(=O)(C(CNC(=O)CN1CCCCC1C)(CC)CC)NC(C#C)C(C)(C)C 87302,C1(CCC(=O)N(CC(C)O)CC)CCCCN(C(=O)Cc2cc[nH]c2)C1 87303,Cc1nc(N)cnc1C(=O)N(C)CCOCCNC(=O)CC(C)n1ccnc1 87304,C1(NC(c2cnn(C)c2F)=O)CN(C(C2CC3CCC2O3)=O)CC2(CCC2)C1 87305,c1(C(C)C)cc(N2CCC(NC(=O)C3=CCCCC3)C(C)C2)n2ncnc2n1 87306,C(=O)(C#CC1(C)CCCO1)N(C1CCN(C(C2CCC3(C2)N=N3)=O)CC1)C 87307,C=C=C(C)CC(=O)N1CCC(N(C(=O)CCSc2ccccc2F)C)C1 87308,C1(CN(C(C(C)OCCC(C)C)=O)C)CN(C(=O)CC=CC(C)(C)C)CCO1 87309,CC1CCN(C(=O)CC(C2CC2)NC(=O)CS(C)(=O)=O)CCS1 87310,c1(C(C(N2CCC(N(C(=O)Cc3ccnn3C)C)C2)=O)(F)F)cccc(F)c1F 87311,c1(C(=O)NC2CCC(C(N3CCCC(F)(F)C3)=O)C2)c(F)c(F)c(O)c(F)c1F 87312,C1(NC(CN2C(C)CCC2)=O)CCC2(CC1)CC2NC(C1C2CC3C(C2=O)C13)=O 87313,c1(OC)ccc(C(=O)NCC#CC(=O)NCC(=O)NC2CCCC2)s1 87314,N1(C(C2(C#C)CCC2)=O)CCOCC(C)(CNC(=O)CCC2CCCCN2C)C1 87315,c1(C(=O)NCC2(F)CCC(CNC(C3(CO)CCCO3)=O)C2)ccc(F)cc1Cl 87316,c1(N(C(=O)C(=O)NCC(C2CC2)N(C)C)CC=C)c(CO)cc(Br)cc1C 87317,N1(CC)CC(C(=O)NCC2(NC(c3ncc(C)o3)=CC3CCC3)CC2)CC1=O 87318,N1(C(CCNC(=O)OCC)=O)CCCCC1N(C(=O)CSCC)CC 87319,C(CN=c1[nH]c(=NCCC2CCCCO2)[nH]c2cc[nH]c12)c1ccc(SC)cc1 87320,c1(CN2C(C(=O)Nc3ccc(Br)nc3I)CCC2)cc(F)c(Cl)c(Cl)c1 87321,N1(C(C(C2CCOC2)NC(C(C)OCC#C)=O)=O)CCCC[Si](C)(C)C1 87322,CCCCN=c1ncc(-c2ccnc(NC(=O)CCN3CCCCC3)c2)c[nH]1 87323,c1(C(=O)NCC2CCCCN2C(c2n[nH]cc2F)=O)c[nH]cc(Br)c1=O 87324,N1(C(CC(C(F)F)NC(c2cc(C)c(F)cc2)=O)=O)CCC2CCCC2CC1 87325,Nc1sc2c(c1C(N1CCC3(C1)CN(C(=O)C1=C(Cl)CCOC1)C3)=O)CCC2 87326,[N-]=[N+]=NCCCCCC(=O)N1CSCC1C(=O)NC1(C2CCC2)CC1 87327,c1(C(=O)NCC2C3N(C(C4C(CCC)C4)=O)C(CC3)C2)ccc2oc(O)nc2c1 87328,c1(CC=C)ccccc1C(N1CCC(CNC(=O)C(C)n2cccn2)(OC)C1)=O 87329,C1(NC(=O)C=CC=C(Cl)Cl)CCCCC12CCN(C(=O)C=Cc1cccs1)C2 87330,c1(OCCC)ccc(C(N2CCCC2C(C)NC(=O)CC2CN(C)C2)=O)cc1 87331,C(=O)(CCC=CBr)N1CC(CC(C)NC(CCc2ccc(SC)s2)=O)C1 87332,Cc1nc(CC(N2CC(N3CCN(CCOCc4ccco4)CC3)C2)=O)c(C)s1 87333,N1(C(c2cc(C)c(Cl)s2)=O)CC2CC1CN2C(C1CC(C2CC2)=NO1)=O 87334,N1(C(C2CNC(=O)N2)=O)CC(C2CC2)(C(=O)NC2C3C=CC(C3)C2CO)C1 87335,c1(CC(=O)N(C(C)CCNC(C2CCCCO2)=O)C)c(F)ccc(Br)c1F 87336,c1(C(N(CCCCNC(C2CCC2)=O)C)=O)csc(C2CC2)c1 87337,N1(C(c2ccc(NC)cn2)=O)CCCC(CC(=O)NCC2(C)CC(O)C2)CC1 87338,C(C1=CCN(C(c2cc[nH]c2C2CCC2)=O)CC1)NC(C(F)OC)=O 87339,c1(CNC(C2(C(N(c3ccccc3)CC)=O)CC2)=O)cn(C)c(=O)nc1O 87340,C1(F)(CNC(C(C)OCC=C)=O)CCN(C(c2cccs2)=O)CC1 87341,N1(C(C2N(C(CCC)=O)CCCC2)=O)CC2(CCCCN(C(=O)C(C)CO)C2)C1 87342,C1(=CC(N2C(C)C(NC(=O)Cc3ccncc3F)CC2)=O)CC2CCC(C1)N2C 87343,C(=O)(CC(O)CC(C)(C)C)NCC(=O)N(CCCOCC)C(C)C.C1(=O)CN1 87344,C1(CNC(C(C)c2cncs2)=O)CC(O)CN1C(=O)CCc1cc(Cl)no1 87345,N1(C(C2CCC(=O)C2)=O)CCC2(CCCN2C(C2CC2c2ccccc2)=O)C1 87346,C(=O)(CCCCCN(C)C)N1CC(CCC)C(C(N2CC(F)C2)=O)C1 87347,c1(NC(CCC)CCCNC(C2CCC2(C)C)=O)c([N+](=O)[O-])c(CC)nn1C 87348,CC1(C(N2CC(O)(CCNC(=O)C(N)=O)C2)=O)CC1(F)F 87349,N1(C(CN(C)S(N)(=O)=O)=O)CCC2(CC1)CC2NC(=O)CCSc1nccn1C 87350,N1(CC(CC(=O)OC)Sc2noc(C3CC3)n2)CCCN(C)CC1.C(C)=O 87351,C1(CNC(CN(C)C(c2ccccc2)=O)=O)CCCCC1NC(=O)CC(F)F 87352,c1(OC)ccc(C2(C(=O)NC(C)CC(C)NC(C3CCC(=O)N3C)=O)CC2)cn1 87353,CC(C)(CCC(=O)N1C2CCC1C(CNC(=O)C#CC1CCOC1)C2)[N+](=O)[O-] 87354,CC(CC(=O)NC1CCN(C(C2CC2(F)F)=O)CC1C)C(F)F 87355,c1(C(C(=O)N2CC(F)C2)NC(CCOC(C)C)=O)cnn(C)c1 87356,C12(NC(=O)CCSCc3ccccn3)CCC1CN(C(c1c[nH]c(=O)cn1)=O)C2 87357,c1(C(=O)NC2CC(NC(C3C(C(N(CC#C)C)=O)C3)=O)C2)cc2occc2n1C 87358,N1(CC(=O)O)CCCC(N2CC(NC3CSC3)C2)C1=O 87359,C(CN=c1cc(C)nc(C)[nH]1)C1(O)CCN(C(C=CC=CC=CC)=O)CC1 87360,c1(C(C(=O)NC)N(C)Cc2cnnn2C)ccc(C)cc1 87361,CC1c2ccc(F)cc2CCN1C(c1cnsn1)C(=O)Nc1cccc([N+](=O)[O-])c1 87362,c1(C(=O)OCC)c(OC)ncnc1Cl.c12cc(ncn1)NCCN2.C1(N)CCOCC1 87363,CC(CC(C)NC(C1CCCN1c1cnccn1)=O)NC(=O)C(C)(C)C 87364,c1(C(=O)OC)nn(C)cc1NC(C1CCCN1C(=O)C=CC(C)(C)SC)=O 87365,c1(C(N(CCC(=O)N(CCC)C)CCO)=O)c[nH]nc1COC 87366,C1(C(=O)NC(c2ccccc2)CC)CC2(CCC2)CN1C(=O)C(CO)C(F)(F)F 87367,C1(C(=O)NCC2(F)CN(C(C(N3CCCCC3)C)=O)C2)CCC(=O)NC1 87368,C1(C2CCCN(C(=O)C(C)(C)CC#N)C2)(NC(C(c2ccncc2)C)=O)CC1 87369,CC1CN(CC(=O)NCc2nccs2)c2cc(C(F)(F)F)ccc2O1 87370,C(=O)(C(CNC(C1CNC(=O)N1)=O)CC1CC1)N(CC(C1CCC1)OC)C 87371,c1(C(=O)NC(CC)CN(C)C(C2(CCF)CC2)=O)cc(C)c(Cl)c(C)c1 87372,CC(CNC(c1ccc(O)cn1)=O)C(F)C(=O)NCCc1cccnc1F 87373,N1(C(C)C)CC2CC1CN2C(=O)C(c1ccnn1C)NC(=O)CC1(O)CCOC1 87374,c1(COC)nc(OC)cc(NCC2CN(C(=O)CCc3c(C)noc3C)C2)n1 87375,c1(C(C)NC(C(CC)NC(c2ccccc2)=O)=O)cc2ccccc2s1 87376,C1(C(N2CCN(C(CCOC)=O)CC2C)=O)CC2CC1C1C2C1(F)F 87377,C1(CC(=O)NCCC2(O)CN(C(COCC=C)=O)C2)CCOC(C)(C)C1 87378,C1(C(=O)N(C(C=C)C2CCC2)CC)CN(C(=O)C(CC)=CC)CCC1(C)C 87379,c1(C(N2C(C(C)NC(c3cc(Cl)cnn3)=O)CCC2)=O)cncc2nc[nH]c12 87380,CN1CC2(CN(C(=O)NC3CC3c3cccc(OC(F)(F)F)c3)C2)OC1=O 87381,C1(NC(NC(COC)C)=NCC2CC(=O)N(C(C)C)C2)CCOC(C)(C)C1 87382,CON(CCCO)C(=O)C1(CO)CCCN(C(c2cnnc(C)c2)=O)C1 87383,C1(CCCNC(C2(CSC)CC2)=O)CCCN1C(=O)C=CC1CC1 87384,CC1CN(C(c2cccc(O)c2)=O)CC1(C)C(=O)NC1CCC(C)(C)CC1 87385,c1(NC(C2(C)CCN2Cc2ccc(O)c(O)c2)=O)ccc(OC(F)(F)F)cc1Br 87386,C=C(C)C1CCC(C)CC1NCCCOc1ccc(Br)cc1 87387,c1(CC)oc(C(=O)NC2(C(=O)N(CC)CC34CCCCC3C4)CCOCC2)cc1C 87388,C1(CC)CCN(C(=O)CCC2(C)CC2)C1C(=O)N(CC(C)(C)COC)C 87389,c1(CNC(C(C)Cn2ccnc2)=O)ncccc1C(=O)O 87390,c1(C(=O)NC23CN(C(C(CC=C)C)=O)C(CC2)CC3)cc(C#N)c(O)nc1N 87391,C1(N(C(=O)Nc2ccc(COC)cc2)C)CCC(=O)N(c2cccc(F)c2)C1 87392,N1(C(C(CC)CC)=O)CC2CC1CC2NC(c1cnc(C)nc1C(C)C)=O 87393,C1(C(=O)NCC(CC)N(C)C(c2nnc(C)s2)=O)CCCC(C)C1 87394,N1(C(C2CC(CC)(CC)C2)=O)CC(C(=O)NCC2C=CCCC2)CCC1C 87395,C1(C)(OC)CCCN(C(=O)CC=CCNC(=O)C2=C(C)OCC2)CC1 87396,Cc1c(C(=O)NCC2COCCN2C(=O)Cn2cc(Br)cn2)cncc1Br 87397,C1(C(N2CCC(C(CNC(C3C(=C)CC3)=O)F)CC2)=O)CN2CCC1CC2 87398,c1(C(N2CCC(F)(CNC(C(CC)OCC)=O)C2)=O)cccc(S(N)(=O)=O)c1 87399,C(=O)(CCCCN(C(=O)C(C)(F)c1ccon1)C)NC(c1cc[nH]n1)C 87400,c1(OC)ccc(CCC(=O)N(C2CN(C(=O)CC3CC(C)C3)C2)C)cn1 87401,CC(CC(=O)N(C)CC1(O)CCN(C(=O)C(F)(F)CO)C1)C(F)(F)C(F)(F)F 87402,c1(C(N)=O)ccc(C=CC(=O)NCC2CC(NC(c3cscc3Cl)=O)C2)o1 87403,N1(CC2(NC(C=COCC)=O)CC2)CCN(C(=O)C(F)(F)c2ccccn2)CC1 87404,Cc1cc(C(=O)NCC(=C2CN(C(=O)Cc3ccn(C(C)C)n3)C2)F)n(C)n1 87405,C(CO)(CCCCNC(C1(C)COC(=O)OC1)=O)NC(C=COCC)=O 87406,C1(CNC(CC=CC=C)=O)(CNC(=O)CCNC(=O)CC(C)C)CC12CCC2 87407,CC(C)CCCCC(=O)NC1CC1CNC(c1ccnc(OC(C)C)c1)=O 87408,CC1(C)CC(C)(C(=O)NCCC2(CNC(C3CNC(=O)C3)=O)CC2)C1 87409,Cc1cc(C(C)C(=O)NC2CC(c3ccc(=N)[nH]c3)C2)ccc1Br 87410,c1(C(N2CC(OC)CC2(C)CNC(=O)CNC(N)=O)=O)nnc2ccccc2n1 87411,C12(C(=O)NCCCCNC(Cc3cc(C(C)C)no3)=O)CCCC1CC2 87412,c1(C(N(CCCc2cccc(C)c2)C)=O)c2c(nn1C)CCCC2 87413,CCCC(C)C(CC)(c1nnnn1C(C)C)NCC1(c2ccc(OC)cc2)CC1 87414,N1(C(C(C)=C(CC)C)=O)CCC2CN(C(c3cn(CC4CCOC4)nn3)=O)CC12 87415,c1(CC(=O)NCC2C(CNC(CSCC=C)=O)C2)ccc(C)nc1 87416,c1(C(c2nnnn2CCCC2CC2)NCCC(=C)C)ccc(S(C)(=O)=O)c(NC)c1 87417,CS(=O)(=O)CC(=O)NC1CCCCC1NC(=O)CNC(=O)C(F)(F)F 87418,C12(CNC(c3n(C)cnc3)=O)COCCN1CCN(C(c1cnsc1)=O)C2 87419,CCC(CC(C)C)C(=O)N(CC(C)(C)CNC(=O)CC1CCC(C)(C)CC1)C 87420,c1(CC)ccoc1C(=O)NCC1(CNC(C2CN(C3CCC3)C2)=O)CCC1 87421,N1(C(CC2(CC(=O)OC)CC2)=O)CCCC(C2CC2NC(=O)CC(C)(C)O)C1 87422,C1(NC(C2CCC(=O)S2)=O)CCc2nncn2C1 87423,C(=O)(C(C)(C)CCCNC(=O)Cc1ccnc(O)c1)NC1C(C)(C(F)F)C1 87424,N1(C(C2C(C(C)C)CCC2)=O)CCCC(C)(C)C1C(=O)NC1CCC2(CCC2)C1 87425,c1(C(=O)NC(C2CCN(Cc3cccnc3Br)CC2)C)cc(Cl)cnc1Br 87426,C1(NC(C(CC)NC=O)=O)C=CCN(C(=O)COc2cccc(OC)c2)C1 87427,N1(C(CCCC=C)=O)CC(C2CC2)(C(=O)NC2CCCOC2)C1 87428,Cc1ccc2c(c1)C(C(=O)NC(C)(C)CNC(C1CC1c1ccccc1)=O)C2 87429,c1(OC)ncccc1CN1CCC(C)C1.C1(N(C)CC)CCN(C)CC1 87430,C(=O)(NNc1ncc(Br)c2ccccc12)C(C)(C)CNC(=O)OC(C)(C)C 87431,C1(CCC(N2CC(CC(C)NC(=O)CN(c3ccccc3)C)C2)=O)CCCN1C 87432,C12(C(=O)NCC(C)(C3CC3)NC(=O)CC34COCC(C3)C4)CCC(CC1O)C2 87433,N#CCCCC(=O)NC1CCN(C(=O)COc2ccc(Cl)cc2)C1 87434,c1(CC(N2CC(CNC(C3(C)CC(C#N)C3)=O)OCC2)=O)ncn2c1CCCC2 87435,c1(C(N2CCC(C(C)C(N3CC(CO)(CF)C3)=O)C2)=O)nnn(C)c1N 87436,C=CC1(C(N2C3C=CCC2CC3)=O)CCN(C(=O)C(C)COC(C)=O)C1 87437,c1(C(=O)NCCCCCN(C)C(c2sccc2F)=O)ccc2n[nH]cc2c1F 87438,C1(NC(C2CC(C)(F)C2)=O)CC2CCC1N(C(c1ccc(F)cc1N)=O)C2 87439,C(CCCCCO)NC(CC(C)N(C(CN1CCC(C)C1)=O)C)=O 87440,C(=O)(C(C)C(C)c1ccc(F)cc1)N(CCNC(=O)CCc1ccc(Cl)s1)CC 87441,CN1CCOC(CC(=O)NC(CCN(C)C(c2ccco2)=O)c2cccs2)C1 87442,Cc1cc(S(=O)(=O)NCC2COC3(CCCC3)O2)c(Cl)cc1Cl 87443,N1(C(CN(C(=O)OC)C)=O)Cc2ccnn2CC(NC(=O)CNC(N)=O)C1 87444,C12(C(=O)NC(C#C)CC(C)C)CCC(NC(C3CC34CCCCC4)=O)(CC1)C2 87445,Cc1cc(Cl)cc(C(N2CCCC(NC(c3cncc(O)c3Cl)=O)C2)=O)c1C 87446,CN1CCOC(C(=O)NCC(O)CCNC(c2cnoc2-c2ccco2)=O)C1=O 87447,c1(CC)ccsc1C(=O)NC(C1CC1C(=O)N(C(CO)C(C)C)C)C 87448,Cc1ncc(N)cc1C(=O)NCC(C)N(C)C(c1nc(Cl)c(Cl)s1)=O 87449,c1(C(N(CCCCNC(C(CC)C(C)(F)F)=O)C)=O)noc2c1CC(C)CC2 87450,c1(C(N2C(c3nnc(C)o3)COCC2)=O)cnc2scc(C)n2c1=O 87451,c1(CCC(=O)NCC(C(C)C)NC(C2(C(N)=O)CC2)=O)cncc(F)c1 87452,c1(CC(N2CCC(C(C)NC(c3nc(C)sc3)=O)C2)=O)ccc2c(c1)ncn2C 87453,c1(OC)cc(CN2CC(OCC(=O)Nc3nc[nH]n3)C2)cc(OC)c1OC(F)F 87454,C(=O)(C(C)(C)C(N)=O)N1CC(NC(C2C(C)OCCC2)=O)C1 87455,CN1CCN(C(=O)C(O)CCn2cncn2)CC1CNC(=O)C=CCN(C)C 87456,c1(SCC(=O)NC2CCN(C(CC(CCC)C)=O)C23CC3)nnc2ccccn12 87457,c1(C(=O)NCCN(C(=O)C(C2CCC(=O)N2)C)C(C)C)ncc(F)cn1 87458,Cc1cc(=O)n(CC(C)C(=O)NCC2CCC(C)(C)CC2)cn1 87459,C1(NC(C=CCC)=O)CCC12CN(C(=O)C(CC)NC(=O)OC(C)(C)C)C2 87460,N1(C(C(C)c2ccsn2)=O)CCCN(C(=O)C#CC2CC2)C(C)C1 87461,Cc1ccc(C(C)C(=O)N(C2CCN(C(=O)CC(O)C3CCCC3)C2)C)s1 87462,N1(C(C(C)(C)OC)=O)Cc2occ(C(=O)NC3CN(C)CC3(C)C)c2C1 87463,C#CCCCC(C)C(=O)N(CCN(C)C(C1(C)COC(C)(C)CO1)=O)C(C)C 87464,C(CCCCCNC(C1CCC(C#N)C1)=O)NC(c1ccn(C)n1)=O 87465,n1(CC)ncnc1CN1CC(C(C)NC(C2CCCCS2)=O)C1 87466,CC1CN(C(=O)C=Cc2ccncc2)CC(C(=O)NCc2ccon2)O1 87467,c1(C(c2n(CC=C)nnn2)NCC2(OCC)CCSC2)ccnn1C=C 87468,Cn1cc(C(=O)NC23CCCC(NC(=O)C(F)C(F)(F)F)(C2)C3)ccc1=O 87469,CN1CCCCC(C(=O)N(C)CCN(C)C(c2cn(CC(F)(F)F)cn2)=O)C1=O 87470,C(=O)(CCCCN1CCCC1)N1CC(OCCNC(C(C)CC2CCCO2)=O)C1 87471,c1(C(N(CCOC)CCNC(C2(C(F)F)CC(O)C2)=O)=O)cc(O)n(C)n1 87472,N1(C(Cc2cccc(C#C)c2)=O)CCCC2(NC(C3CC(=C)C3)=O)CC2C1 87473,Cc1cc(C)n(C(C)CC(=O)N(C)CC2CCN(C(c3ccc(F)o3)=O)C2)n1 87474,C1(NC(C(C)CO)=O)C2CC3C1C3C2C(=O)Nc1cc(O)cc(F)c1 87475,Nc1c(C(N2CC(NC(=O)Cn3ncnn3)CC(F)(F)C2)=O)ccc(Cl)c1Cl 87476,S(=O)(=O)(c1c[nH]ccc1=NC1COCc2cccnc21)NCC(CC)OC 87477,C1(C(N(CCCCCC)CC(N)=O)=O)CCC(CC2CCCN2C(C)=O)CC1 87478,C(=O)(C(C)(C)C(C)(F)F)N1CC2C(C(N(C3CCOCC3)C)=O)C2C1 87479,N1(C(C2(SC)CC2)=O)CCC(C)C(NC(=O)C(C)(c2ccccc2)OC)C1 87480,C(=O)(C(CC)C(C)(C)CC)N1CCCC(N(C(CCCC(=C)C)=O)CCO)C1 87481,C(CC(C)C)(C(C(=O)Nc1ccc2c(c1)OCO2)N1CCOCC(CO)C1)OC 87482,c1(OC)cc(C)c(CN(c2cc(NCC(C)CC3CC3)nc(C)n2)C)cc1C 87483,S(=O)(=O)(c1ccc(Br)s1)N1C(C(=O)Nc2cc(C(C)(C)C)no2)CCCC1 87484,C(=O)(C(CC(C)C)N(C)C(C1(CC)CC1)=O)N(CC(=O)OCC)C 87485,CCCCCC(O)C(=O)NC1(CCC(=O)N(C(CO)C2CC2)C)CCC1 87486,CN1CC2C(CCCN2C(=O)NC2CCCN(Cc3ccccc3)C2)C1=O 87487,CC1(C)CCC(C(=O)NC(CCO)C2CC2)CN1C(C1(O)CCCC1)=O 87488,CCC(C)(COC)C(=O)NC1CC1CNC(=O)Cc1nn(C(C)C)cc1Br 87489,C(=O)(C=C1SCC(=O)N1C)NCCC(C)N(C(=O)CC1CC(=O)NC(=O)C1)C 87490,C1(CNC(C(C)C)=O)CN(C(C2CCCN(S(C)(=O)=O)C2)=O)CCCO1 87491,N1(C(C)=O)CCCCC1C(C)(C)CNC(c1ccc(N(C)C)cn1)=O 87492,C1(F)(CNC(C(C)OC)=O)CN(C(=O)CCNC(c2ccsc2)=O)C1 87493,N1(C(CNC(N(c2cc(C)on2)C)=O)=O)CCN(C(=O)CNc2ccco2)CC1 87494,c1(CN(C(CC)CC(C)C)C=O)ccc(C#N)n1C 87495,C1(NC(C(CCC)C)=O)CN(C(c2ccn(-c3cccnc3)n2)=O)CCC1(C)C 87496,c1(C(N(CC(C)N(C(COC(CC)(C)C)=O)C)C)=O)ccc(-n2cnnc2)cc1 87497,C1(C(N(CC(=Cc2ccccc2)C)C)=O)CN(C(c2ccc(Cl)s2)=O)CC1(C)C 87498,c1(C(N2CCC(N(C(C3C(C=C)C3)=O)CC)C2)=O)cc(Cl)ncc1N 87499,C=C=CC(C)C(=O)NCC1CCCN(C(C2(C)COC(=O)N2)=O)C1 87500,c1(CC)noc2ncc(C(=O)NC3CCN(C(=O)CNS(C)(=O)=O)CC3O)cc12 87501,O=C(C1=CCCCCC1)Nc1nnc(CSCCNC2OC(=O)CC2O)s1 87502,CC(C)S(=O)(=O)CC(=O)NC1CCN(C(C2CCCCCS2(=O)=O)=O)CC1O 87503,c1(C(N2CCC(C(=O)Nc3ccc(C4CC4)cc3)(CF)C2)=O)cccc(Cl)c1 87504,Cc1cc(C(=O)NCCN(C(=O)CCCF)C2CCCCC2)cc2c[nH]nc12 87505,c1(C2(NC(CCC(=O)Nc3cccc(C)n3)=O)CCC2)c(F)cccc1F 87506,CC(C)CCCC(=O)N1CCC(NC(=O)C=CC2CCCCC2)C(O)C1 87507,CC(C)C(C)(CNC(C1CCC(=O)C1)=O)NC(c1ccc(C2CC2)nn1)=O 87508,C1(C)(C(=O)NCCC2(C(N(CC(C)OC)C)=O)CCC2)CCCOC1 87509,N1(C(c2scc(OC)c2)=O)CCCC(CC(=O)NCC(C(C)C)C(C)C)CC1 87510,Cc1nnc2c(C(N3CCCN(C(C4CCCSC4)=O)C(C)C3)=O)nccn12 87511,O=C(CC1NC(=O)c2ccccc21)NCCC1CCN(C(C2SCCS2)=O)C1 87512,C(CCC(C)CC(=O)N(C)CC1(NC(=O)COC(C)(C)C)CC1)=C(C)C 87513,c1(COC(C(COC)C)=O)cc(Br)ccc1C(=O)OC 87514,N1(C(CNC(CC(c2c(C)n[nH]c2C)C)=O)=O)CCOC(C)(C(F)F)C1 87515,N1(C(C(CC#C)O)=O)CC(NC(c2ccn(C)c(=O)c2)=O)CCC1C 87516,CC(CN=c1[nH]cnc2c(C(F)(F)F)cccc12)N(C)C(c1ccc(C2CC2)o1)=O 87517,N1(C(C(C2CCOC2)NC(Cn2ncc(C)c2)=O)=O)CCCC2(CC1)CC2 87518,C(=O)(C1=CC2C=CC(C1)C2)NC(C1(C(N2CCCC(C)(N(C)CC)C2)=O)CC1)C 87519,C(C)(CCS(C)(=O)=O)NC(=O)NCc1ccc(CC)nc1 87520,c1(C(C)(C)C)cccc(NC(=O)CC2CCC(C(=O)NC3CC(O)C3)CC2)n1 87521,C(=O)(C1Cc2ccc(F)cc21)NC1(CNC(CC(C)C2CCCO2)=O)CCCC1 87522,Cc1cccc2nc(NC(=O)CC3CCCN3C)[nH]c12 87523,N1(C(C2N(C)CCOC2)=O)C2CCC1CN(C(c1ccc(C(F)F)c(F)c1)=O)C2 87524,N1(C(C)=O)CCC(CC(=O)NCCCN(C(c2cncn2C)=O)C(C)C)C1 87525,C=CCCC(=O)N(C(CNC(c1cscc1Cl)=O)Cc1ccccc1)C 87526,C1(C(=O)O)COC2CN(C(c3ccccc3-n3cc(C4CCCC4)nn3)=O)CC12 87527,N1(C(C(C(C)O)C)=O)CCCCC(NC(=O)CCc2ccsc2)C1 87528,C1(C(=O)NCCC(=O)NC)CCOCC1NC(c1ccc(O)cn1)=O 87529,C#Cc1cnc(C(N2CCCC(C(=O)N(CCC)CCSC)(CC)C2)=O)c(C)c1 87530,c1(OCC(=O)N(CCNC(C2(CC(C)C)CCCC2)=O)C2CC2)cccc(O)c1 87531,Cc1nc2[nH]ccc2c(=NCC(O)CNC(c2cnn(C3CCCC3)c2)=O)[nH]1 87532,c1(C(=O)NC2CN(C(C(CCC)N(C)C)=O)CC2O)ncnc2cc[nH]c12 87533,C12(C(N3CCCC(CNC(C4CC5(CCO4)CC5)=O)C3)=O)CC3CC1C2C3(F)F 87534,c1(CC)nc(C(N2CCCC2CNC(=O)C=CCOC)=O)c2ccccn12 87535,CCC(F)(F)C(C)(C)C(=O)NC1CN(C(=O)C=C(Cl)Cl)CCC12CCC2 87536,C(CN=C(NCC(c1cccc(Br)c1)C)N1CCC2(CCOC2)C1)OC 87537,C1(COC)CC(CNC(=O)C=C2CCSCC2)N(C(C2CSCN2C(C)=O)=O)C1 87538,c1(NC(C2CC(=C)C2)=O)cccc(C(N2CCOC(C(=O)N(C)C)C2)=O)c1 87539,C1(C(F)(F)F)(C(=O)NCCC(C)NC(C2OCCC2C(F)(F)F)=O)CC(F)(F)C1 87540,c1(SC)nc(C(F)F)cc(=NCNCC(C)(C)C2(O)COC2)[nH]1 87541,C(=O)(C1=C(SC)CCCC1)NCC1CCN(C(c2c(CC)csc2)=O)CC1C 87542,C1(OC)(OC)CCN(Cc2ccc(Cc3ccccc3)cc2)CC1O 87543,c1(CCC(N2CCCC(N(C(c3ccns3)=O)CC)C2)=O)cccc(C#N)c1 87544,c1(CC)ncc(C(=O)NC2CN(C(C3CCC(C)(C)CO3)=O)CCC2C)c(O)n1 87545,C1(CN(C(C(c2cnccn2)C)=O)C)CCCN(C(c2ccc(=O)oc2)=O)C1 87546,N1(C(CCCC#CC)=O)CCC2(CC1)CC(NC(=O)CSC)CCO2 87547,Cc1cc(=NCC(=O)N(C2CCCCC2)C)[nH]c(=NCC2CN3CCN2CC3)[nH]1 87548,C1(CNC(C2(C)CCC2)=O)C2CN(C(=O)CCc3cccs3)CC12 87549,C1(C)(CNC(N(C2CCC(F)(F)C2)C)=O)CCC2(CC1)CC2 87550,N1(CC)CCC(NC2CCC(CC(F)(F)F)CC2)CC1 87551,CC1=C(C(=O)N2CC=CC(NC(c3ccc(C(N)=O)c(Cl)c3)=O)C2)CCO1 87552,C(c1cc(Cl)c2c(c1)OCO2)=CC(N1CCC(C)C(NC(=O)C(C)N(C)C)C1)=O 87553,C(c1ccc(C#N)cc1)=CC(=O)NC1(CN(C(C2CC(C)OCC2)=O)C)CC1 87554,Cc1cc(O)cc(C)c1C(N1CC(F)(CNC(C2(C)CC3CC3C2)=O)C1)=O 87555,C(=O)(C(C)(C)CC(C)C)N1CC(C(N2CCC(C=C)(O)C2)=O)OC(C)C1 87556,C1(C(=O)OC)CC(C(F)(F)C(F)(F)F)CN(C(C2(c3ccccc3I)CC2)=O)C1 87557,C(N=c1cccc(S(=O)(=O)N(C)SCC)[nH]1)c1ccc(CC2(OC)CCOC2)o1 87558,N1(C(=O)NC(C2CCC2)C2CC2)CCC2(CC1)CC2(C)Cn1c(C)ncc1 87559,Cc1cc(Cl)c(C(N2CCC(O)(C(C)NC(c3cccc(F)n3)=O)C2)=O)cc1C 87560,c1(OC)cc(COC(c2cc(C)ccc2N2CCCC2=O)=O)ccc1O 87561,c1(C(COC)N(C)C(N2CCC(c3noc(C)n3)(C(=O)O)C2)=O)ccc(Br)cc1 87562,C1(NC(C(CN=[N+]=[N-])NC(=O)C(=O)NC2CC2)=O)CC2(C1)CC21CCC1 87563,CC1(C)CC(CO)CN(C(CCc2ccccn2)C(=O)NCC2CCOCC2)C1 87564,N1(CC#C)CCN(C(C2CSCN2C(=O)CCc2cnoc2)=O)CC1=O 87565,c1(C(N(CCCOCCN(C(CN2CC(C)(OC)C2)=O)C)C)=O)cc(Cl)ccn1 87566,C(=O)(C#CC(C)(C)CNC(=O)C(F)C1CCC1)NC(c1ccc(C)s1)C 87567,N1(C(C(C)OCC#C)=O)CCN(C(c2cnn(CC)c2C)=O)C2CS(=O)(=O)CC12 87568,C1(NC(c2cc(OC)c(O)c(Cl)c2)=O)CN(C(C2CCC2)=O)C2(CCCOC2)C1 87569,C(=O)(CCCS(C)(=O)=O)NC1(C)CCN(C(C2CC2F)=O)CC1 87570,C1(NC(C(CSC)OC)=O)CCC2(CC1)CN(C(=O)C1=COCC1)C2 87571,N(S(=O)(=O)N(C)C)CC(=O)NCCOCCNC(c1cc(C(CC)CC)no1)=O 87572,C(COC)(CC(=O)NCC1(CC)CC1)NC(C(C)=CC=C)=O 87573,c1(C(N2CCCC(C)(NC(C(C)=C3CC3)=O)C2)=O)ccn2cc(C)nc2c1 87574,C1(F)(C(N2CCN(C(C(C(C)C)SC)=O)CC2)=O)CCC(F)(F)CC1 87575,c1(N2CCCN(CCC)CC2)nc(=NCc2cnn[nH]2)[nH]c2cc(C)ccc12 87576,CCCCC(O)CC(=O)NCC(C1CCCC1)NC(c1ncccc1Cl)=O 87577,C1(n2cc(CN(CC(C)(C)OC)C)nn2)CCCCCC1O 87578,N1(C(CCC(C)OC)=O)CC2CC1CCC2NC(=O)CC1CCCCC1O 87579,C(=O)(CC(C)(C)C(F)F)NC(CCCC)CNC(c1cc(C2(O)COC2)on1)=O 87580,C(c1cn(C)cn1)=CC(=O)NC1(CC)CN(C(C2C(OCC)CCC2)=O)C1 87581,Cc1nc[nH]c1CC(=O)NCC1(CCNC(c2cc(C(F)F)cs2)=O)CC1 87582,c1(C(N2CC(C)C(n3cc(CCC4CC4)nn3)C2)=O)cccc2ncsc12 87583,Cn1cc(NC(C2CCN(C(=O)C(F)(F)C(F)F)CCO2)=O)c(O)nc1=O 87584,c1(C(N2CCC(C3N(C(CC(CC)C)=O)CCC3)C2)=O)ncc(F)c(OC)n1 87585,C#Cc1ccc(CC(N2CCC(NC(c3c(C)csc3Cl)=O)C(CC)C2)=O)cc1 87586,c1(C(=O)NC2CCN(C(=O)Cn3ccccc3=O)C2)ccnc(C(F)(F)F)c1F 87587,C1(C(=O)NC2C(NC(c3cc(C(C)C)[nH]n3)=O)C2)CCC(C(F)(F)F)CC1 87588,N1(C(c2cc(C)ncn2)=O)CCN(C)CC1CNC(c1ccoc1CC(N)=O)=O 87589,c1(CCC(=O)NCCCCNC(CC2C(CC)C2)=O)cccc(O)n1 87590,Cc1cnc(F)cc1C(N1CCCC(CNC(=O)C(C)(C)n2cnnn2)C1)=O 87591,c1(OC)cc(C(=O)Nc2cccc(N(C)C)c2)c2ccccc2c1 87592,C1(CNC(N(CCCN(C)C)C)=O)CCN(C(=O)C(C)(C)C)CC1.C1CO1 87593,c1(CCC)cc(=NC(CNC(c2coc(COCC)n2)=O)C2CC2)[nH]c(Cl)n1 87594,c1(CNC(=O)CCC2CC2)ccc2c(c1)CCC2NC(c1cccc(O)n1)=O 87595,C=Cc1cncc(C(N2CC(O)(C(F)C(=O)NCC(c3ccncc3)O)C2)=O)c1 87596,N1(C(C(CC)COC)=O)CCC(O)C(N(C(=O)CCC=CBr)C)C1 87597,C(=O)(CC(C)(C)NC(c1sccc1CC)=O)NC(C1CCOC1)C#C 87598,CC(Cn1cccn1)N=c1cccc(S(=O)(=O)NC2CC3CCCCC23)[nH]1 87599,C(=O)(CC1=CCN(CC2(C)CCCN2C(C)=O)CC1)OC 87600,c1(OC)cc(C(=O)NC2CCC(NC(C3CC(CF)C3)=O)C2)ccc1C 87601,Cc1sc(C(N2CCCC2C(C)NC(=O)C2=NOCC2)=O)cc1Br 87602,N1(CC)CCC(C)N(Cc2ccccc2)CC1.C12(CCCCC1)N(C)C2=O 87603,c1(SC)ccc2nc(S(C)=O)[nH]c(=NCCC(C)(F)F)c2c1 87604,c1(CN(CC)CC)ccc(Cl)cc1Cl.N12CCN(CC1)C2=O 87605,C(=O)(C(C)(C)CS(N)(=O)=O)N1CC(NC(C(C2CC2)OC)=O)C(C(F)F)C1 87606,Cn1cncc1C=CC(=O)NCC(C1(O)CN(C(C2C3CNC(=O)C23)=O)C1)(C)C 87607,Cc1ccc(NC(C2CCCC2CNC(c2cnn3c2CCC3)=O)=O)cc1C 87608,C#Cc1cnn(C)c1C(=O)NCC1COCCN1C(C1C2CCC1CC2)=O 87609,C1(NC(c2cc(Cl)ccc2F)=O)CN(C(=O)CCCC(F)F)CC1C1CC1 87610,c1(C(N(C2CC(NC(C(C(CC)CC)C)=O)C2)C)=O)cnn2cccc(OC)c12 87611,CN1CCc2ccc(C(=O)NCC(CO)NC(=O)C3=NNC(=O)CC3)cc21 87612,CCC(C)C(C(=O)NCC1CN(C(c2cn3ccnc3s2)=O)CC1(C)C)N(C)C 87613,C(=O)(C(C)CC(F)(F)F)NCC1CN(c2cc(C)nc(C(C)(C)C)n2)CC1(C)C 87614,C(=O)(CCS(C)(=O)=O)NC1(C(=O)NC(CC)CN2CCCC2)CCSC1 87615,c1(C(=O)NC2CC(NC(=O)C=Cc3cc[nH]n3)C2)ccc(C2CC2)nc1 87616,N1(C(c2c(C)n(C)cc2)=O)CCC(NC(=O)C(O)C(F)F)C2(CCC2)C1 87617,c1(OC)ccc2nc(OC)[nH]c(=NCC3OCCc4sccc43)c2c1 87618,N1(C(c2c(C)n(C3CCOC3)nn2)=O)CCC(CNC(C2CC2(Cl)Cl)=O)C12CC2 87619,c1(CC(=O)NC2CC2NC(c2csc(-c3ccccn3)n2)=O)ccc(O)cn1 87620,c1(C(=O)NCC2(C(N(C)CC3CCC3)=O)CC2)ccn(CCF)n1.C1(C)CCC1 87621,O=C(C1=CS(=O)CCC1)NCCN(CCOCCO)C(C1(OC)CCC1)=O 87622,O=[N+]([O-])c1ccc(Br)c(Cl)c1NCc1nccs1 87623,c1(CC=CC)ccccc1C(=O)NCC(C)CNC(c1snnc1C1CCC1)=O 87624,Cc1cc(O)nc(C(C)N(C(=O)CN2CC=CC2C(C)C)CC(C)(C)C)n1 87625,N1(CCC(=O)NCC2CCCC2NC(=O)CCN2CCOCC2)CCOCC1=O 87626,C(N=c1ccnc(C)[nH]1)C1CCCC(NC(Cc2cc(C)cc(C)c2)=O)C1 87627,c1(C(=O)NC2C3(CN(C(C4(CC)COC4)=O)C3)CC2)coc(S(=O)(=O)NC)c1 87628,N1(C(C(c2ccc(OC)nc2)(F)F)=O)CCC2(NC(=O)CC(C)(C)O)CCCC12 87629,N1(C(c2cc(C)c(C)s2)=O)CC2(CC(NC(=O)CS(=O)(=O)N(C)C)C2)C1 87630,N1(C(Cc2ccc(C)cc2)=O)CC(NC(=O)C(C)CC(C)(C)C)CCC(O)C1 87631,C1(CC(=O)N(CC)Cn2cccc2)CN(C(=O)CC2CCC(C3CC3)O2)CCO1 87632,c1(OC(CCSC)=O)ccc(OCC(N)=O)cc1.c1(CO)ccc(F)cc1 87633,O([Si](C)(C)C(C)(C)C)CCCCCNC1(COC(C)=O)CC=CC1 87634,CCC(CNC(=O)C(C(=O)OC)OC)(CC)C(=O)Nc1ccc(O)cc1Cl 87635,C(=O)(C#CC1(C(F)(F)F)CC1)NC1C(CNC(CCCN(C)C)=O)CCC1 87636,N1(C(c2c(CC)ncs2)=O)CCCC2(C1)CN(C(c1cccc(C)c1Cl)=O)C2 87637,CC1CN(C(=O)CS(=O)(=O)N(C)C)C(C)CN1C(c1cnn(CCN(C)C)c1)=O 87638,CN1CCN(C(C2CC(C3CC3)=NO2)=O)C(C(=O)NC2(CCF)CCC2)C1 87639,CCCCN=C(NCC(C)Sc1ccccc1)N1CCC(C(C)C)C1 87640,C1(C)(C(=O)NCC(C#C)CC2CC2)CCCN(C(C2CCC2(OC)OC)=O)C1 87641,c1(C(N(C2CCCCN(C(C3(C)CC=CC3)=O)C2)C)=O)cc(Br)cnc1O 87642,N1(C(CC)=O)CCCCC1C(=O)NC(C)CCNC(c1cnc(NCC)cn1)=O 87643,c1(OC)cc(NC(N2CC3CC2CN3S(=O)(=O)CC)=O)c2ccccc2c1 87644,C1(C)(CNC(CN(C)C(=O)C2CC2)=O)CCN(C(C2C3CNC(=O)C23)=O)CC1 87645,N1(C(c2c(CNC(c3c(C)nccn3)=O)c[nH]n2)=O)CC2NC(=O)OC2C1 87646,C1(NC(C(CN(C)C)(F)F)=O)CC2(C1)CC(CNC(c1ccc(Cl)c(F)c1)=O)C2 87647,c1(-c2nnc(CN(C)CCc3c[nH]c4cnccc34)o2)sc2ccccc2c1Cl 87648,c1(C(=O)NCCC(C)N(C(c2c(CC)csc2)=O)C)cc[nH]c(=N)c1 87649,C(=O)(C#CC1CCCOC1)NCC1(C)CCN(C(c2c(N)ccc(CC)c2)=O)C1 87650,C12(C(N(C3CN(C(c4cccc(C(F)F)n4)=O)C3)C)=O)CCOCC1C2 87651,C(C1CN(C(=O)C(O)CC2CCCC2)CC1C(=O)NCC(C)C(C)C)=CC 87652,Cc1cccc2[nH]cc(CC(N3CC(NC(=O)Cc4ccsc4Cl)C(C)C3)=O)c12 87653,c1(C(N2C(C)(C(=O)Nc3ncc(OC)nc3)CC2)=O)c(OC)ccnc1F 87654,N1(C(C(N2CCSCC2)C)=O)CC(NC(c2ccc(F)s2)=O)CCC1C 87655,C1(CCNC(C2CCC(C)S2)=O)(OC)CN(C(=O)CC(C2CC2)C2CC2)C1 87656,N1(C(CCC2(C)N=N2)=O)CC2CC1C2C(=O)NCC1CC(F)C1 87657,C1(CNC(=O)NC2(CC)CCOCC2)Cc2nccn2C1 87658,c1(CC=CCNC(c2[nH]cc(CC(C)C)c2)=O)nc2c(cc1C#N)CCC2 87659,C1(CC(=O)NCC2(OC)CN(C(CNC(CC)=O)=O)C2)COc2ccccc2O1 87660,c1(C(=O)NC2CN(C(COCCCC)=O)CC2O)sc2ncccc2c1Cl 87661,N#Cc1cccc(OCC(=O)NCCCCNC(=O)CC2CCC(F)(F)C2)c1 87662,CC1(C)OC(=O)CC1C(=O)NC1(CCCNC(=O)CCN2CCC2)CC1 87663,C(=O)(C(F)(F)C(F)(F)F)N1CC(CC)C(NC(c2cnn3ccccc23)=O)CC1 87664,c1(C(=O)NCCN(CCC)CCc2cccc(C)c2)cccnc1S 87665,C1(CC(=O)NCCNC(c2nc(C)sc2)=O)CCCC(C)C1 87666,C(CC1=CCN(C(c2cccc3c2NCC3)=O)CC1)NC(CC1C(C)CCO1)=O 87667,c1(C(=O)NCc2ncc(C(C)C)cn2)cc(Cl)c(Cl)c(Cl)c1 87668,N=S1(=O)CCCC2(CCCN2C(=O)CC(N)Cc2ccc3ccccc3c2)C1 87669,CCC(C)(O)C(=O)N1CCCC1c1nc(C(N2CC(n3cnnc3)C2)=O)cs1 87670,C1(OC)CCCN(C(C2(C(NOCC(=C)Cl)=O)CC(=O)C2)=O)CC1 87671,N1(C(c2c(C)noc2C)=O)CCC2(CC1)CC2C(=O)Nc1c(C)ncnc1C 87672,C1(COC)C=CCCN1C(c1occc1CNC(c1c[nH]cc1C)=O)=O 87673,C1(NC(c2cc(C(C)C)[nH]n2)=O)CCC2(CC1)CN(C(c1cncc(F)c1)=O)C2 87674,N1(C(c2c(CNC(C3(C(=O)OC)CC3)=O)cco2)=O)CC(C)CCCC1C 87675,N1(C(C(SC)SC)=O)CCCC1C(C)NC(=O)CC1CCC1 87676,Cc1cc(CCC(=O)NC2C=CCN(c3ncc(C(F)F)cn3)C2)nn1C 87677,N1(C(c2cncc(N(C)C)c2)=O)CCOCC(NC(C2CC=CCC2)=O)C1 87678,N1(C(CC2(OC)CCCC2)=O)CCN(C(=O)CCN2CCC(O)CC2)C(CF)C1 87679,N1(C(C(C)=C2CCCC2)=O)CCN(C(c2cc(-c3ccccc3)no2)=O)C(C)C1 87680,Cc1nc(NCCCCC(N)=O)cc(=NCC2CCC(=O)NC2)[nH]1 87681,N1(C(c2oc(C)c(Br)c2)=O)CC(C)CN(C(=O)C(F)=C2CCC2)C(C)C1 87682,N1(C(C2(C#C)CCC2)=O)CC2COCC(C1)C2NC(C12CCCN(CC1)C2)=O 87683,C(CC(C(C)C)NC(=O)OC(C)(C)C)NC(C1CCCCC1)CC 87684,c1(C(=O)NCC(CCC)NC(c2ncccc2O)=O)cccc2nccn12 87685,C(C(C)(C)CCNC1(CO)CC1)NC(c1nnnn1C1CCOC1)C.C1CC1 87686,c1(C(=O)NC2C(NC(C3(CCOCC)CCC3)=O)C2)cnc2c(c1)NC(=O)CO2 87687,c1(C(=O)NCCC2CCCCN2C(=O)CC2CCOC2=O)cncc2nc[nH]c12 87688,CCCCCCN(CCC(=O)NCC1CCN1C(c1cnc(NCC)s1)=O)CC 87689,N1(C(c2cnc(OC)s2)=O)CC2CC1C2NC(=O)Cc1sc(C)nc1C 87690,Cc1cc(OCC(=O)NC(CNC(=O)CC(C)(C)C#N)CO)cc(C)c1 87691,N1(C(CCC=CCC=C)=O)CC=CC(C(=O)NCc2ccccc2C)C1 87692,c1(C(=O)NC2CN(C(C(c3ccncc3)C)=O)CC2(C)C)cc2c(o1)CCCC2 87693,c1(C(=O)NCC2(C)CCN(C(CCCCCSC)=O)C2)cc2nc[nH]c2cc1F 87694,CC(CN=C(NCC(c1cccc(C#N)c1)O)NCC1CCC1)c1cccnc1 87695,CCCCC(C(=O)OC(C)(C)C)NC(=O)NCc1cc(CCCOC)cs1 87696,Cc1cc(C(=O)N(CC(O)CNC(c2ocnc2C(F)(F)F)=O)C)sc1Cl 87697,C1(NC(C2(C3CCCO3)CC2)=O)(CO)COc2ccccc2C1 87698,C(CCCCn1cc(Cn2ccnc2C)nn1)NC(C1(CCC)CC1)=O 87699,N1(C(CC2(NC(=O)CC3CCCC34CC4)CC2)=O)CC2CCCC(O)C2C1 87700,CC1CC(NCc2nn(C)c3c2COCC3)c2ncnn21 87701,N1(C(C2CCN(CC)C2)=O)CCC2(C(=O)NC(CO)CC(C)C)CCCC12 87702,n1(CC(=O)NC2C3(CCN(C(C(C)C4CC4)=O)CC3)C2)[nH]cc2c(=O)ncnc1-2 87703,C1(O)(CNC(CCC(C)NC(c2ncnc(O)c2F)=O)=O)CC2C=CC1C2 87704,CC1(C)CC(CC(N2CCC(CF)(NC(c3cc([N+](=O)[O-])n[nH]3)=O)C2)=O)NC1=O 87705,c1(CN(C(C(CN(C(C)C)C)N)=O)C)ccccc1N 87706,N1(C(CCCOCC=C)=O)CCC2(CC1)CCN(C(c1ccc(Cl)c(O)c1)=O)C2 87707,N1(C(C(CC=C)CNC(=O)C(C)(O)C2CCC2)=O)CCOCC2(CCC2)C1 87708,C12(NC(C3C(COC)C3)=O)CCC1CN(C(c1ccc(Cl)cc1Cl)=O)C2 87709,C(CCC(C(=O)NCC1(F)CC1)NC(=O)Cc1cncnc1O)OC 87710,CC(CC(=O)NC(C1CN(C(c2cnoc2-c2ccoc2)=O)C1)C)n1ccnc1 87711,CC(C)C(C)C(=O)NC1(CCNC(=O)Cc2coc(-c3ccccc3)n2)CC1 87712,CN1CCCC(O)(CC(=O)NC2CCC(NC(c3cccc(F)c3O)=O)CC2)C1 87713,C1(NC2(c3nnnn3C)CCC(C(C)C)C2)CC2C=CCC(C1)C2 87714,C1(CNC(CN2C(C)CCC2)=O)CCC(F)(CNC(=O)C(C)CC(N)=O)CC1 87715,c1(C(N2C3(CNC(C(C)=CC)=O)CCC3CC2)=O)ccc2ccccc2n1 87716,C(=O)(CCCN(C)C)N(C1CCC(NC(C2(F)CCC2)=O)C1)C 87717,C1(F)(CNC(C(COC)OC)=O)CCC(CNC(=O)C(c2cnccn2)C)CC1 87718,C1(NC(Cc2n(C)nc(CC)c2Cl)=O)C(C)CN(C(C2CN(CC)C2)=O)CC1C 87719,C1(NC(C(C=CC)O)=O)CCN(C(c2ccnc(F)c2Cl)=O)CC1F 87720,N1(C(C)=O)CCCC(CCNC(c2sc(F)cc2C)=O)CC1 87721,C(C(=O)N1OC2CCC1C2)C1(C)N(CC)CCC1.C1CCCC(=O)N1 87722,CC1OC2(C(=O)NCC(N3CCN(C(=O)C(F)F)CC3)C(F)F)CC1C2 87723,N1(C(C=C2CCC(C)C2)=O)CCCN(C(=O)Cc2cncc(Br)c2)CCC1 87724,N1(C(c2ncn(C(C)C)n2)=O)CCC2(CCC2NC(c2cnncc2O)=O)CC1 87725,c1(C(=O)NC(c2cnc[nH]2)C)coc(CNC(c2ccsc2Cl)=O)n1 87726,Cc1cc(C(=O)NCCN(C(=O)Cc2cncc(C#N)c2)C2CC2)ccc1Cl 87727,O=C1CC(C(=O)NC23CCN(C(c4cccc(Cl)c4F)=O)CC2C3)CC(=O)N1 87728,c1(C(=O)NCC(C)CNC(=O)C(c2ccccc2)O)cc(Cl)c(Cl)cc1N 87729,C1(C(=O)OCC(C(=O)NCC)C)(C(=O)OC)CCNCC1 87730,Cc1cn2cc(C(=O)NC3CCC3CNC(c3cnc(C(C)(C)C)s3)=O)nc2s1 87731,N1(C(C(CCC)O)=O)C2CCCC1CN(C(=O)C(O)C1CCC1)C2 87732,c1(C(N2CC(NC(CC3(C(=C)F)CCC3)=O)C(OC)C2)=O)ccc(C#N)c(C)c1 87733,N1(C(C2N(C(CC)=O)CSC2)=O)CCCC(O)(CNC(C23CCC(C2)C3)=O)CC1 87734,CCCCCC(C)(C)C(=O)NC(CO)CCCCNC(c1c[nH]nc1[N+](=O)[O-])=O 87735,C=CCC(C(=O)N1CC(N(C)C(c2ccn(CCC)n2)=O)C1)c1ccccc1 87736,C=CCCCCC(=O)NCC1CC1NC(c1cnn(-c2ccccc2F)c1N)=O 87737,c1(OCC)cccnc1C(=O)NC1CCCC1NC(C1(C)CCC(=O)N1)=O 87738,CC(C)CCC(O)C(=O)NCCCCC1CCN(CC(=O)OCN)CC1.C(C)(C)(C)O 87739,c1(N(C)C)n[nH]c(=NC(=O)N2CC(CN)C(c3ccccc3)C2)s1 87740,N1(C(C(CC)COC)=O)CCCC(C)(C(=O)NCc2nocc2C(C)C)C1 87741,c1(C(N(CC(C)CNC(c2cncc(N(C)C)c2)=O)C)=O)ccccc1S(C)=O 87742,C1(C(=O)NCCN(C(=O)CC(C)(F)F)CCOC)CCc2cncn2C1 87743,C1(NC(c2occ(C)c2)=O)COC2C(NC(=O)C(F)F)COC12 87744,C1(NC(=O)CCCC2CC2)COC2C(NC(c3cn(CCF)nn3)=O)COC12 87745,c1(CC)nc(C(=O)NCC2CN(C(=O)C(c3ccccc3)C)CC2O)c(C)o1 87746,c1(C(=O)NC2(CNC(c3n[nH]cc3F)=O)CCOC2)cnn2c1OCCC2 87747,c1(SCC)cc(C(=O)NCCC2(NC(=O)CC(CC)SC)CCC2)ccc1F 87748,N1(C(c2n(C)ncc2)=O)CC2CC1(C(N1CCC(C(F)F)CC1)=O)C2 87749,C1(C(=O)NC2(CNC(c3occ(C)c3)=O)CCOC2)COC(C)(C)CO1 87750,C1(CCNC(C(C)(C)Br)=O)CCN(S(=O)(=O)Cc2cccc(Br)c2)CC1 87751,c1(CC)ccc(C(N2CC(CNC(=O)CCc3n[nH]c(=N)s3)C(C)C2)=O)c(F)c1 87752,C1(C(N(CCO)CC)=O)CC2CN(C(C3CCCCC3)=O)CC2C1 87753,CC1CN(C(c2ccc(C3CC3)nn2)=O)CCN(C(c2cnnn2C)=O)C1 87754,n1(CCC(=O)NCC(C2CCC2)NC(C23CCC2CC3)=O)ccc(O)nc1=O 87755,N1(C(c2c(OCCC)cccc2)=O)CC(NC(=O)C(C)n2cccc2)CC(C)C1 87756,C=CCC(CC(C)C)C(=O)N1CCOC(CN(C(=O)CCc2cnn[nH]2)C)C1 87757,c1(CC(=O)NCC(C)N(C(Cc2ccc(C)cc2)=O)C)nn(C)cc1[N+](=O)[O-] 87758,Cc1cc(C(=O)NC(CNC(=O)C(c2ccccc2Cl)(C)C)C2CC2)ncc1F 87759,C1(NC(CCCCOCC)=O)CCN(C(=O)C(C)(C)C2CC2)CC1C 87760,N1(C(C2(C#N)C(C)(C)C2)=O)CCC(C=CC(=O)NC2CC(N3CCCC3)C2)CC1 87761,C1(C)(C(N2C(C)C(NC(c3cccc(CO)n3)=O)CCC2)=O)CCS(=O)(=O)CC1 87762,C1(C(=O)NCCc2ccc(C)s2)(NC(COCCOCC)=O)CCN(C)C1 87763,C(CN=c1[nH]c2c(c(=NCc3nc(C4CC4)cs3)[nH]1)CSC2)C1(CO)CC1 87764,C1(C(=O)NCCNC(C)=O)CN(C(=O)C(C)(C)COC(C)(C)C)CCCO1 87765,N1(C(C2C(CC)CCC2)=O)CC(NC(=O)CC(=O)NC2CC2)CC2(CCC2)C1 87766,c1(OC)ccccc1C=CC(=O)NCC(C)(CO)NC(c1cc(F)ccc1C)=O 87767,C1(C(=O)NCC(C(C)C)NC(c2cc(CO)on2)=O)CCC(C)CC1 87768,c1(CC(=O)NCCC2(CNC(CSCCC#N)=O)CC2)ccc2ccoc2c1 87769,c1(OC)nc(NC(c2n[nH]cc2NC(c2scc(C)c2Cl)=O)=O)cnc1C#N 87770,c1(C(N(C(C)CNC(=O)C=Cc2ccnn2C)C)=O)ccc2c(c1)OCCCO2 87771,N1(C(C2(C)CCCCO2)=O)CC2CC(NC(=O)C(O)C3CC3)CC2C1 87772,C1(CN(C)C2CC2)CCN(C(=O)CCOC2CN(C(=O)CC3CC=CC3)C2)C1 87773,N1(C(C(CSC)OC)=O)CC2(CCCN(C(=O)CCN3CCC3)C2)C1 87774,C1(C(N2CCC(NC(=O)CSCCc3ccccc3)C2)=O)CCn2nccc2C1 87775,c1(N2CC(C)N(CC#N)C(C)C2)nc(NC(C)CC(F)(F)F)c2cnn(C)c2n1 87776,C1(N(C(CC(C=C)c2ccccc2)=O)C)CCCN(C(=O)C=CC=CC)CC1 87777,c1(C(c2nnnn2C2CC2)NC(CCC)CC)ccc(OC)c(F)c1F 87778,CC1CC(C(=O)NCc2nocc2C(=O)N(C)CC2CC(F)(F)C2)CCO1 87779,N1(c2nccc(C(=O)OC)n2)CC2(CCCC2NC(=O)CCC(C)C)C1 87780,Cc1cc2ccc(C(=O)N(C3CCCCC3NC(C3CC3Br)=O)C)cn2c1 87781,Cc1cnc(N2CCC(N(C(=O)Cn3nc(O)ccc3=O)C)C2)nc1O 87782,c1(C(N(CCNC(c2cccc(C)c2)=O)CC2CC2)=O)ccc2nn[nH]c2n1 87783,C1(C(=O)NC2CCN(S(C)(=O)=O)C2)CN(C(C2(C)CCCCC2)=O)CCN1 87784,CCC(C)C(C(=O)N(C)CC1(CNC(c2cc(N)ccc2OC)=O)CC1)OC 87785,N1(C(C(=O)NCc2nnn(C)n2)CCC2CCCO2)CCC(S(=O)(=O)C(F)F)C1 87786,c1(C(N2CC(C(N(C)CC3CCCC4CC34)=O)OCC2)=O)c(F)cccc1F 87787,c1(OC)cc(CN2CC(NC(c3scnc3C)=O)CC(C)C2)cc(I)c1O 87788,C12(C(C)NC(c3coc(CNC(=O)CCc4cn(C)cn4)c3)=O)CCC(CC1)C2 87789,Cc1cccc(C(C2CCC2)NC(=O)Cc2ccnn2-c2ccccc2)c1 87790,CCC(CC(=O)N1CCN(C(=O)CCc2ccc(C)s2)CC1COC)C(F)F 87791,c1(OC)cccc2c(CC(=O)NCCCN3CC(C)CC(C)C3)c[nH]c12 87792,Cc1cccc(N)c1C(=O)NCC1C(C)CCCN1C(=O)Cc1cccc(F)c1 87793,c1(CCC)onc(C)c1C(N1CC2CC2(C(=O)NCc2cccc(Br)n2)C1)=O 87794,c1(C(N2CCCC(OC(C)(C)C)C2)C(=O)NC(CC)(C)C)ccc2c[nH]nc2c1 87795,c1(C(N(CC(C)NC(c2cnc(C(C)O)s2)=O)C)=O)cnn(C)c1C1CC1 87796,C1(C(N(C2CCC2O)C)=O)CC(O)C(O)CC1CNC(C12CCC1C2)=O 87797,C1(NC(C2CCn3ccnc3C2)=O)CCCC12CCN(c1nncs1)CC2 87798,Cc1cc(N)c(C(=O)NCC2CN(C(c3cccc(F)n3)=O)CCO2)cc1F 87799,c1(CN2CCC(C(=O)OC)(C(C)C)C2)ccc2c(c1O)CCCC2 87800,C1(NC(C(CC#C)C)=O)CC2(C1)CN(C(c1ccnc(OCC)c1)=O)C2 87801,c1(C(N2CCCC(N(C(C(CC)OC)=O)C)C2)=O)cc2ccccc2o1 87802,c1(NCC(N2C(CN(C(C(CC)OC)=O)CC)CCC2)=O)ccc(C)cc1 87803,c1(OC(CC)C)cc(N2CCC(C3CC(N)CCO3)CC2)nc(C)n1 87804,C1(NC(CC(c2ccc(NC)cc2)C)=O)CCNCC12CC2 87805,CC(CCCNC(=O)N(c1cccnc1)CCCCO)c1nn[nH]n1 87806,C(C1c2ccccc2CN1C(=O)CSc1nncs1)NC(C1C2CCCOC12)=O 87807,c1(C(N2C(C)CN(C(C3CCC(=O)N3)=O)CC2)=O)ccnc(P(C)(C)=O)c1 87808,C1(CN(C)C(c2cccc(O)n2)=O)CCCCN1C(C1(C)CCC(=O)C1)=O 87809,c1(C(=O)NCC2C(C(=O)NCC(=O)N(C)CC)CCC2)ccccc1C1CC1 87810,C1(C(=O)NC2CCC(NC(Cc3ccc(C)o3)=O)CC2)CC2CCCCCCC12 87811,c1(C(=O)OC2(C(N)=O)CCOC2)ccc(CC#N)cc1.C1(=O)CCN1C 87812,c1(CCC(=O)NCCOc2ccc3cccnc3c2)cccc2c1OCCO2 87813,C1(NC(=O)COC2CCCCC2)C=CCOC1 87814,N1(C(C2CCC(=O)N2)=O)CC2(CCCC2NC(c2ccc3ncsc3c2)=O)C1 87815,c1(OC)cccc(C(F)F)c1C(=O)N(CCCNC(C12CC(C)(C1)C2)=O)C 87816,C1(C(=O)NC2CCN(C(CC3C(C)(C)C(O)C3)=O)CC2F)CC2C=CCC(C1)C2 87817,N1(C(CNC(CC)=O)=O)CCC(C(C)NC(c2sc(C)nc2CC(C)C)=O)CC1 87818,C(=O)(C1=NOC2COCC12)N(CCNC(C(C)SC)=O)CC1CC1 87819,C=CCCCCC(=O)NC1COCC1CNC(c1c[nH]c(Br)c1)=O 87820,N1(C(c2occ(C)c2)=O)CC2OCCN(C(C3C=CCCC3)=O)C2C1 87821,C(C1=CCCOC1)NC(CC(C1CC1)NC(C)=O)=O 87822,Cc1cc(C(=O)NCc2cc[nH]c2C(=O)NCC(c2cnc[nH]2)C)[nH]c1C 87823,c1(NC(C(=O)NC(C2CC3CCC2C3)CC)=O)cncc(SC)c1 87824,N1(C(C(C(C)C)O)=O)CC2CN(C(=O)C(C)NC(C3CCCCC3)=O)CC2C1 87825,c1(CC)ccccc1C(N1CC(CCCCNC(=O)CC2CC3CCC2C3)C1)=O 87826,C1(NC(C2CC2(F)F)=O)CC2(C1)CN(C(c1nc(Br)sc1C1CC1)=O)C2 87827,Nc1ccc(C(=O)NCC2CCCC2NC(C2COCCN2C)=O)nc1 87828,C1(CNC(C2(C(=O)OCC)CC2)=O)CN(C)CCN1C(c1csnc1C1CC1)=O 87829,N1(C(COCCC#C)=O)CC(CNC(C2CCCCN2C)=O)C(O)C1 87830,c1(CCC(=O)N(C2CCN(C(CCC(=C)C)=O)C2)C)cn2ccccc2n1 87831,c1(OC)cc(OC)[nH]c(=NC2CCC(C)N(C(c3ccc4scnc4c3)=O)C2)n1 87832,c1(C(NC(=NCC2CN(C)CCO2)NC2CCC2)C)ccc2c(c1)CCCC2 87833,c1(C(N2C(CNC(Cn3c(C)cnc3)=O)C(C)CC2)=O)cccc(O)c1F 87834,C=Cn1nccc1C(=O)NCC(C)CN(C)C(C1CCN(C2CC2)C1=O)=O 87835,CCCCCCCCC(=O)NC1(C(N2CCOC(CF)C2)=O)CC1 87836,c1(OC)ncc(S(=O)(=O)NCC2(O)CCCOC2)cc1C 87837,c1(NC(c2cc(Br)cnc2OC)c2n(C(CC)C)nnn2)cccc2c1OCC2 87838,C1(CC)CN(C(=O)CCOCC(F)(F)F)CCN1C(c1ccnc(C)c1N)=O 87839,N1(C(C2C(C)(C(C)C)C2)=O)CCC(O)(CNC(c2ccc(Cl)c(CO)c2)=O)CC1 87840,Cc1csc2ncnc(N3CCCC(C(=O)NCC(C)O)C3)c12 87841,c1(CC(=O)NC(C)CCNC(c2csc(-c3cnc[nH]3)n2)=O)c[nH]c(=N)nc1O 87842,C12(CNC(C=Cc3ccc(C)o3)=O)CCCC1N(C(=O)Cc1nc[nH]n1)CC2 87843,C(CC(F)F)(C(=O)N(C(C)C(=O)NC)C)N(C(CCN(C)CC)=O)C 87844,C=CCC(C(=O)NCC(F)C1CCC1)NC(=O)CCCN(C)C 87845,Cc1nc(NCC2CCC3(CC3)CO2)cc(=NCc2nnc(-c3ccccc3)s2)[nH]1 87846,C1(C(=O)NC(CCNC(c2cnn(C(C)C)n2)=O)C)CCCCC1C 87847,c1(C2C(C(=O)NC3CC(CCNC(C=CCC)=O)C3)CC2)nc(S)n[nH]1 87848,c1(NC(C)=O)ccc(C(N2CCCC(NC(C3CCCS3)=O)C2)=O)c(Cl)c1 87849,c1(C(N(CC(C)NC(=O)CC2(CO)CCCC2)CC)=O)coc2c1COC2 87850,N1(C(C2CC(C)(C)C2)=O)CC2CC1(C(=O)NCC1CC3CCC1C3)C2 87851,c1(-n2cc(C3N(C(c4cnn(CC)c4Cl)=O)CCC3C)nn2)cc(F)cc(Cl)c1 87852,c1(OCCCC(=O)Nc2cccc(CNC(CSC)=O)c2)ccc(C#N)cc1 87853,c1(CC)nn(C)c(CC)c1CC(=O)NCCCCNC(c1cc(N)cnc1C)=O 87854,N1(CC(=O)N(C(CNC(C(CC)C#N)=O)C)C)C(=O)NC2(CCCCC2)C1=O 87855,C(c1c(C)nn(C)c1Cl)=CC(=O)NC(CC)(C)CNC(C1CN2CCC1CC2)=O 87856,C1(CC(C)NC(c2cc(OC)no2)=O)CCN(C(C2CCCCC2OC)=O)CC1 87857,N1(C(C2CCN(C(CCC(C)SC)=O)CC2)=O)CCC2(CC1)CN(C)C2 87858,c1(C(=O)NC(C(C)C)C(C)NC(=O)Cc2cncs2)cccc2c1OCC2(C)C 87859,CC1CCN(C(C(=O)Nc2ccc(Cl)cc2F)c2cc[nH]n2)CCS1 87860,FC1(F)CCCC(c2nc(-c3ncccc3Br)no2)CC1 87861,C(=O)(C1CCCc2ccccc21)NC(CN=c1[nH]nc(C(=O)OC)s1)C 87862,CCC(C)C(O)CC(=O)N1CCC(CC(=O)NCC=C(Cl)Cl)CC1 87863,C(CO)(CCCNC(c1ccc(=N)[nH]c1)=O)NC(c1c(CC)cco1)=O 87864,c1(OC)ccccc1OCC(N1CCC(NC(C2C3COCC23)=O)C1)=O 87865,C1(NC(CCc2cnc(C)o2)=O)CCCC(C(=O)N(CC(C)O)CC(C)O)CC1 87866,Cc1cnn(C)c1CC(=O)NCC1(CNC(C2CC2C)=O)CCCC1 87867,CCC(C)(C(=O)O)n1nnc(CCCCCO)n1.n12cc(nn1)CN1CC2C1 87868,c1(CNC(c2cnn(C)n2)=O)ncc(C(=O)N(C)CCOCC2CC2)cn1 87869,C(CNC(=O)C(C)Oc1ccc(F)cc1)(CC(C)C)NC(c1c(CC)ocn1)=O 87870,c1(NC(C2(CC)CN(C(=O)Cc3ccoc3C)C2)=O)cnccc1CO 87871,C(C)(CCCCNC(=O)C(F)CC1CCOC1)NC(c1ccc(C)o1)=O 87872,C1(C(N2C(C(N(CCO)CC)=O)CC2)=O)CCCSC1 87873,Cc1cc(C)c(C(=O)NCC(C)(C(C)C)NC(C2CCNC2=O)=O)o1 87874,c1(CC)nc(=NC2CCN(CCNC(c3cccnc3CC)=O)CC2)s[nH]1 87875,c1(OCC(=O)NCC23CC(NC(=O)CC4C=CCC4)(CO2)C3)cccc(Cl)c1 87876,CC1(C(=O)NC2CC(NC(C3CCCS(=O)(=O)N3)=O)C2)CCc2ccccc21 87877,N1(CC(CC)CC)CC2C3CCC(C2C1)N(C(c1cnn(C2CCCC2)c1)=O)C3 87878,N1(C(c2c(CC)nccc2)=O)CCC2(CCCN2C(C23CCC2CC3)=O)C1 87879,N1(C(c2c(C)c[nH]n2)=O)CCC(CN(C(=O)COC2CCCCC2C)C)CC1 87880,CC1(C)CC(NC(c2coc(C3CC3)n2)=O)CN(C(=O)Cc2n[nH]c(=N)s2)C1 87881,C1(C(=O)NCCCOCC2CCC2)CN(C(C2CCCSC2)=O)CC12CCC2 87882,c1(OC)ccc2cc(C(N3CCN(C(=O)C(C)N(C)C)CC3)=O)ccc2n1 87883,C1(CC(=O)N(CCNC(=O)CCn2cncn2)CC)CC(C2CC2)C1 87884,Cc1ccc(C#N)cc1C(=O)NCc1ncoc1CCNC(C1C=CCCC1)=O 87885,CC#CCC(C(=O)N1CCCC(CC)(CO)C1)NC(=O)C=CCOC 87886,c1(NC(=O)NCCNC(CCNC(CN(CCC#C)C)=O)=O)ccc(O)cc1F 87887,C(=O)(CS(=O)(=O)CCOC)NCC(CCOC)CNC(C1CC2CCC1CC2)=O 87888,c1(C(=O)NCC2C3CN(C(=O)CC4C=CCCC4)CC23)cc(F)cc(F)c1 87889,C1(C(=O)NCC(O)CO)(OC)CCN(Cc2ccc(F)cc2)CC1 87890,C1(CCC)CN(C(C2CCCSC2)=O)CCN1C(=O)CC1CCC1 87891,c1(C(N2C(CCNC(c3c(CC)nn(C)c3)=O)COCC2)=O)ccc(F)cc1Cl 87892,C1(NC(c2c(CC)cccc2)=O)CC2CC1N(C(c1cn(C)nc1Br)=O)C2 87893,C(=O)(C(CCC1CCC1)NC(=O)CC1CCC(=O)NC1)NCc1ccn(C)n1 87894,c1(NC(C23C(CN(Cc4ccc(OC)nc4)C2)C3)=O)cccc2c1OCC(=O)N2 87895,C1(C(N2CC(NC(=O)OC)C2)=O)CCC(O)CN1C(=O)CC1CCN(C)CC1 87896,N1(C(CS(CC)(=O)=O)=O)CCCN(C(C2CCC(=O)N2C)=O)C(C(C)C)C1 87897,C(=O)(C(C)(C)S(=O)(=O)C1CC1)NC1C(CNC(c2cccc(C)c2F)=O)CC1 87898,c1(C(C(=O)NCCc2cccc(C#C)c2)C)ccc2c(c1)OCO2 87899,N1(C(=O)NCC=C(CCC)C)CCC(C)(C(=O)OC(C)=O)CC1 87900,N1(C(CC(C(=O)OC)C)=O)CCC(C)(C)CC1C(=O)NCC(CO)OC 87901,c1(OCCCNC(CNC)=O)ccc(Br)nc1 87902,C12COCCN(C1)C(=O)C2.C(C(=O)NCCSCCOC)=CCC 87903,c1(SC)cccc(C(N2CCC(CCNC(=O)C(C)CF)C2)=O)n1 87904,c1(-c2nc(CCNC(=O)NCC3(CO)CCOCC3)sc2)cccc(F)c1 87905,Cn1c(C(N2CCCC2CCc2cn(CCCO)nn2)=O)cc2ccc(O)cc12 87906,C(C)(C)(CC(F)C(=O)NC1(C)CC2CCC1C2)NC(C(CCCC)O)=O 87907,CC1(C)CC(CNC(C23CCC2C3)=O)CN1C(=O)CC=Cc1ccccc1 87908,C1(C(=O)NC2(C)CN(C(=O)CC3(O)CCOC3)C2)Cc2c(F)cccc2O1 87909,N1(C(c2c(C)c[nH]c2)=O)CCN(C(=O)CCc2cncnc2)CC(C)C1 87910,C1(C(N2C(CNC(C3(N(C)C)CCC3)=O)CC2)=O)CCCOC1c1cn(C)nn1 87911,C=CC1(O)CCN(C(=O)CC(C(C)OC)NC(c2cncnc2CC)=O)C1 87912,C(=O)(C(C1=CCSC1)N(CCS(=O)(=O)C(C)C)C)NCCC 87913,c1(OCC)ncc(Cl)cc1CNC(=O)Nc1oc(C2CCC2)nc1C 87914,C(C(C)(C)CC1COC1)N(C(=O)C(C)(C)C)C(C)=O.C12CC1OC2=O 87915,c1(OCC)cccc(C(N2CC(F)CC2C(=O)NCc2cnc(C)cn2)=O)c1 87916,C(C(CC(=O)N1CC(NC(N)=O)C1)NC(C1C=CCS1)=O)OC 87917,c1(NC(CCC)=O)cncc(CCC(N2CCN(CCC#N)CC2)=O)n1 87918,c1(CCCC)ccc(CC(=O)N(C2CCC(SC)C2)C)cc1 87919,C1(C(=O)NC(c2ccc(OC)cc2)C)CC12CCN(c1nc(Cl)ncc1Cl)CC2 87920,CC(C(=O)Nc1cnc(F)nc1)C(C)NC(c1ncc(F)cn1)=O 87921,CCCC(C)(C)C(=O)NCC(CNC(c1cnn(C)c(=O)c1)=O)OC 87922,CC1C(NC(C2CCN(C(C34CCC3C4)=O)CC2)=O)CCCN1C(N)=O 87923,N1(C(C(c2ccc(C)cc2)F)=O)CCC2C(CCCN2C(C2CCS2(=O)=O)=O)C1 87924,N1(C(C=CC=CCC)=O)CCC2CCN(C(=O)Cc3nc(C)sc3Cl)C2C1 87925,N1(C(C=C(COC)C)=O)CCN(C(=O)CC2CCC(C)C2)CC(O)C1 87926,CC(C)C(CNC(C1(C)CC1(C)C)=O)C(=O)NCc1c(F)cccc1F 87927,c1(CCC)ccc(CC(N2CC=CC(N(N3CCC(F)C3)C(=O)CC)C2)=O)cc1 87928,c1(OC(=O)NCC(CC(=O)OC)C2CC2)cccc(OC)c1 87929,C1(C(=O)OCC)CN(C(=O)CC2CCC(O)C2O)CC1(C)C 87930,C(N=c1[nH]c(=NCC(C(C)C)N(C)C)[nH]c2c1CCCCC2)c1snc(C)n1 87931,CC1(CC(=O)NC2CN(C(=O)CCCNC(N)=O)C2)CC1(F)Cl 87932,c1(C(=O)NC2CCN(C(C3CC4C(C3)C4(F)F)=O)CC2F)occ2c1CCOC2 87933,C(c1cccc(F)c1F)=CC(=O)NCC(O)CNC(c1n[nH]c2c1CC1CC21)=O 87934,N1(C(C2(C)C(C)(C)C2)=O)CC2COCC(C1)C2NC(=O)C1=C(Cl)CC1 87935,N1(C(C(CC)OCC)=O)CCCC2CN(Cc3ccc(S(C)(=O)=O)cc3)CCC12 87936,c1(C(N2CC3C(CNC(C(COC)O)=O)(C3)C2)=O)nc2n(c1Cl)CCCC2 87937,c1(CNC(=O)CC(C)NC(C2(C(=O)OC)CC2)=O)cccc(F)c1F 87938,C1(NC(c2nnc(CC)o2)CC)CCCC1C(=O)O 87939,c1(C(N2CCC(N(C)C(c3[nH]ccc3COCC)=O)C2)=O)cccnc1S 87940,CCC(C)(CC)C(c1nnnn1-c1ccccc1C)NCc1ccc(OC)nc1C 87941,N1(C(C(C)OC(C)(C)C)=O)CCC2(CCOCC2)C(NC(=O)C=CCO)C1 87942,C1(CC)CCN(C(=O)C=Cc2ccncn2)C1C(=O)NCC1COCCO1 87943,N1(C(C(C)OCCOC)=O)CCC(CNC(=O)C(C)(C)N2CCOCC2)C(C)C1 87944,C(CCCCCC(=O)NC(C1CCN(C(c2ccc(C(N)=O)cc2)=O)C1)C)SC 87945,N1(C(c2cn(C)nc2O)=O)CC(CO)C2(C1)CN(C(=O)C(C)(C)n1cncn1)C2 87946,Cc1ccc(C=CC(=O)NC(C)CN(C(=O)CC23CCCC2C3)C)cc1 87947,CCS(=O)(=O)CC(=O)N1C2CCC(C2)C1C(=O)NC(CO)C1(C)CC1 87948,C(CC(C)(C)C)(C(=O)N1CCC(C)(C(N2CCCCC2)=O)C1)OC 87949,C12(C(N3CCC(CCNC(c4c(C)nc(CO)s4)=O)C3)=O)CCC(CC1)CC2 87950,c1(C(=O)NC2CC(C(=O)NCc3ccc(Br)cc3)C2)cc2cccnn2n1 87951,C(CCCCC(=O)NCC1CCC(C#N)C1)n1cc(C2(CC)CCC2)nn1 87952,N1(C(c2c(Cl)cc(C)s2)=O)CCC2(CC1)CC2NC(=O)CCC1CCCN(C)C1 87953,N1(C(c2c(OC)nsc2)=O)C2CCC1C(C)C(NC(c1n[nH]cc1C(C)C)=O)C2 87954,C1(CNC(c2c(C)nn(C)c2)=O)CC(N=c2ccnc(S(C)(=O)=O)[nH]2)C1 87955,c1(C(=O)NC2CCC(C)N(C(=O)Cn3ncnn3)C2)ccn2c1CSCC2 87956,C1(NC(C(=Cc2cccnc2)C)=O)CCN(C(=O)CC2(C)CCC2)CCC1CO 87957,c1(OC)ccccc1-c1n[nH]cc1C(c1nnnn1C)NCC(C)NS(C)(=O)=O 87958,C(=O)(N=c1ccn(CCF)[nH]1)C1(C=C)CCN(C(=O)CCC2CCCOC2)C1 87959,c1(NC(C(n2cc(C(C)OC)nn2)C)=O)ccccc1[N+](=O)[O-] 87960,C(c1ccccc1)=CC=CC(N1CC(N(C(=O)COCCF)C)C1)=O 87961,c1(C(N(CCNC(=O)C(F)OC)CC)=O)n[nH]c(C(C)C)c1[N+](=O)[O-] 87962,C(=O)(C1=C(Cl)CCC1)N1CC(CNC(c2c(CC)n(C)nc2)=O)C(C(F)(F)F)C1 87963,N1(c2nnc(C(C)(C)C)s2)Cc2nccn2CC(NC(C2(C)CC2(F)Cl)=O)C1 87964,C=CCC(C)(CC)C(=O)NC1CCCC1CNC(c1cnnn1C)=O 87965,c1(OCC)nc(C)ccc1CNC(C1CCCN1C(=O)CCC(C)C#N)=O 87966,c1(C(N2CCC(N(C(c3cc(C)on3)=O)C)C2)=O)c(-n2nccn2)cccc1F 87967,C1(CC=C)(NC(=O)CCC2(C)CC2)CN(C(=O)COC(F)(F)F)C1 87968,Cc1nc(C(C)C)ccc1C(=O)NC1CCCC(NC(c2cc(F)n(C)n2)=O)C1 87969,C(=O)(C(C)(C)C(=O)NC1CCCC(C(=O)NCC2CCCCC2)CC1)OCC 87970,c1(C(C(=O)OC)N(C(=O)COC2CCCOC2)C)ccccc1F 87971,C1(CCC)CN(C(=O)CCNC(=O)COC)CCN1C(C1CCCOCC1)=O 87972,C(=O)(CS(=O)(=O)C1CCCC1)NCC(C(C)(C)C)NC(C1CC2(C1)CC2(F)F)=O 87973,Cc1ccc2snc(C(=O)N(CC(C)NC(C3CC4CCCCN4C3)=O)C)c2c1 87974,C1(C(N2CC(C)(C)C2)=O)COC2(C1)CN(C(=O)CC1CCCOCC1)C2 87975,CC1OCCCC1C(=O)NC1(C(=O)NCC(C)(O)C2(C)CC2)CCCCC1 87976,Cc1ncnc(C)c1CC(=O)Nc1ccc(N2CCN(C)CC2)nc1 87977,CCC(COC)C(=O)N(C(C)(C(=O)NC(C)C(C)(C)CN(C)C)C1CC1)C 87978,C(CN=C(NCC1CC=CCC1)NC(C)CC(F)F)OCC 87979,Cc1cccc([N+](=O)[O-])c1C(=O)NCC(n1cc(CCCO)nn1)C 87980,N1(C(CC(C)OC)=O)CCCC(CC(N2CCC(CC3CC3)CC2)=O)C1 87981,O(NC(=O)C(F)C(C)CNC(c1c(C)ccnc1O)=O)CCCC#C 87982,CC1(NC(=O)CC2CCSCC2)CCCN(C(c2coc(CC3CC3)n2)=O)C1 87983,C1(O)(CNC(c2cc(OC)no2)=O)CCN(C(=O)C(C)(C)Sc2ccccc2)C1 87984,C1(C(=O)NC(CNC(C2(C(C)(C)O)CCC2)=O)CC)(COCC)CCC1 87985,N1(C(c2c(OC)ncnc2)=O)CCC2(CCSCC2)C1 87986,CC1(CNC(C2(NC(=O)CCc3nccs3)CCCCC2)=O)CC2CCC1C2 87987,C1(CC(=O)NCC(C)NC(C(COC)C)=O)(CNC(C)=O)CCCCC1 87988,c1(OC)cc(C)c(C(=O)NC2CCC(C(=O)Nc3onc(C)c3C)C2)c(C)c1 87989,C1(C(N(CCNC(=O)Cc2csc(S)n2)Cc2ccccc2)=O)CCCC1(F)F 87990,N1(C(C(CCSC)OC)=O)CC2CC1CN2C(c1ncn(C(C)(C)C)n1)=O 87991,Cc1cc(Cl)ncc1NC(=O)C(N1CCOCC1c1noc(C(C)C)n1)=O 87992,C1(CC)CCC(O)(C(=O)NCCC2(CNC(=O)C=Cc3ccc[nH]3)CC2)C1 87993,C#Cc1cc(F)c(C(=O)NC(CO)C(C)NC(c2cnnn2C2CC2)=O)cc1F 87994,C12(c3ccn(C)n3)CCC(C1)C2C(N1CCCC1CNC(c1ccnnc1)=O)=O 87995,C(CCC(=O)N1CCCC1C(C)NC(=O)C(C)N1CC(C)C1)OCC 87996,CP(C)(=O)C(O)C(=O)NCCOC1CCN(C(=O)CCC2CCCC(=O)N2)CC1 87997,c1(C(=O)NC(C)CCNC(C2(CCF)CC2)=O)cc([N+](=O)[O-])ccc1OC(F)F 87998,c1(C(c2nnnn2Cc2ccccc2)NC(C=C)C2CC2)cc(F)cc(C#N)c1 87999,c1(OCC(=O)NCCN(C(=O)Cc2cnsc2)CCOC)ccc(Cl)c(C)c1 88000,Cc1cc(C(=O)NCC2CCN(C(=O)C=Cc3cncs3)C2)no1 88001,CC(C(F)F)N(C)N(C)CCc1c[nH]c2ccccc12 88002,c1(CN(CC(CC)NC(C#C)=O)C(C2CCCC2)=O)cn(C)nc1OC 88003,Cc1cncc(C)c1C(=O)NC(CC(=O)NCC(C)N(C)C)C(F)F 88004,N1(C(c2c(CN=[N+]=[N-])ccs2)=O)CCN(C2CCN(C(C3(CF)CC3)=O)C2)CC1 88005,c1(CC(N2C(C)C(C(=O)NCC3(CO)CC(C)(C)C3)CC2)=O)ncc(F)cc1F 88006,Cc1nc(C(N2CC(O)C(O)C2CNC(=O)CCCc2nccs2)=O)cc(O)n1 88007,CC1=C(C(=O)N2CC=CC(NC(C3CCCSC3)=O)C2)CCCO1 88008,c1(N2CC(C(=C)C)OCC2)nc(-c2ccccc2)nc(=NC2CCSC2C)[nH]1 88009,C1(C(N(CCOC)CCO)=O)CCC2(CC2)N1C(C1Cc2nccn2C1)=O 88010,N1(C(Cc2cccc(C#C)c2)=O)CCC2(CCCN(C(=O)CCCOC)C2)C1 88011,N1(C(c2cc(OC)no2)=O)CC2(CCOCC2)CC1CNC(C1CCCS1)=O 88012,C1(C(=O)NCC(CNC(c2c(C(C)C)sc(Cl)n2)=O)F)Cc2cccnc2C1 88013,C1(NC(C(C=CCCC)O)=O)CCCC(NC(C2CC(=O)N(CC)C2)=O)C1 88014,c1(C(N(CCC(C)NC(=O)CN2CCOCC2)C)=O)cc2c(F)c(F)ccc2s1 88015,c1(C(C(N2CC(CCNC(CCCN(C)C)=O)C2)=O)O)ccc(Cl)c(F)c1 88016,C1(CNC(CNC(CNC(CC=CC)=O)=O)=O)CCCC(C#C)C1 88017,c1(OCC(=O)N(CCN(C(C2CCC2(C)C)=O)CC)CC)ccc(C#N)cc1 88018,C1(CNC(c2cc(C)n(C)n2)c2n(C(C(=O)OC)C)nnn2)CCN(C)CC1 88019,c1(Nc2c(C(=O)NCc3ccc(O)nc3)cc(OC)nc2)ncc2[nH]ncc2n1 88020,c1(C(N2CCC(C)(NC(C3CCC4CC4C3)=O)C2)=O)cc2n(n1)CCNC2=O 88021,C(=O)(C(F)CCC(C)C)N(CC(=O)NCC(CC)OC)CCC(C)(C)C 88022,C1(c2nn[nH]n2)(C(=O)NC(C(C)C)Cc2ccccc2)CC12CCCC2 88023,c1(C(=O)NCCOCCNC(c2c(C)nncc2)=O)cccc(CO)c1C 88024,c1(OC)cc(S(=O)(=O)N2CC(CNC(c3cc4cccnc4[nH]3)=O)C2)ccc1Br 88025,n1(CC(=O)NCC2CC(NC(C3CCC(=O)O3)=O)C2)c(=O)cnc2ccccc12 88026,c1(C(=O)NC(C2CCCC2)CNC(c2n(CCC)ccc2)=O)ncccc1CC 88027,C=CC1(C(=O)NCC(c2ccc(F)cc2)NC(C2CC2C)=O)CCOCC1 88028,C1(C)(NC(CC2(N(C)C)CCCC2)=O)CCN(C(=O)C(c2cccnc2)O)CC1 88029,CC1CCCC(n2nc(-c3ccc(N(C)C)nc3)nc2CCF)C1 88030,c1(C(C(=O)NC(C(=O)NCC(=C)Br)C2CC2)C)cncnc1 88031,N1(C(C(CCC)N(C)C)=O)CCC2(CC1)CN(C(=O)Cc1ccc(CC)cc1)C2 88032,N1(C(C=CCOC)=O)CCCCC12CC(NC(=O)CCCSc1ccccc1)C2 88033,C1(CNC(c2c(C)cc[nH]2)=O)CC2CCC(C1)N2C(=O)Cc1nonc1C 88034,CCC(CC)C(C)C(=O)NCCC1(OC)CN(C(=O)COCC(C)C)C1 88035,Cn1cnc2nc(N3CCN(CCCO)CC3)nc(NCc3cc(Cl)sc3Cl)c12 88036,CN1CCC(NC(=O)NC2CCCCC2)C1c1cccs1 88037,N1(C(c2nccc(OC)c2)=O)CCCC(O)(CNC(C2CC3(CCC3)CO2)=O)C1 88038,C12(CC(N3CC(NC(C(C4CC(F)(F)C4)OCC)=O)C3)=O)CCC(CC1)CC2 88039,n1(CC(=O)NC(CC)CNC(=O)CCSc2nccn2C)cnc([N+](=O)[O-])c1 88040,CC1CC(NC(=O)Nc2ncccn2)c2nccn21 88041,c1(C(=O)NC(C)CCNC(c2nnn(C(C)(C)C)n2)=O)cc(Cl)ccc1[N+](=O)[O-] 88042,C(=O)(C(CO)C(F)(F)F)NC1C2C(C(=O)NC(C(=O)NC)CC3CC3)C3C(C2)C13 88043,C1(C2(C(C)Cc3nn[nH]n3)CCC2)NC(=O)N(c2ccccc2)C2=C1C(=O)OC2 88044,c1(C(=O)NCCN(C(C(=O)NC)C)C2CC2)cc(Cl)ccc1OC(C)C 88045,c1(CC(N2C3CCC2CC(CO)C3)=O)ccc(OC(F)(F)F)cc1[N+](=O)[O-] 88046,c1(CC)ncoc1CNC(=O)C(C1CC1)NC(=O)C(C1CC1)C1CC1 88047,c1(CNC(CCN(C)CC)=O)cn(CC(=O)N(CCC(C)(C)O)C)nn1 88048,Cc1c(NCC2CCCC(F)(F)C2)ncnc1N1CC(C)SC(C)C1 88049,C1(C(=O)OC)CCOC1C(=O)N(C)CC1(O)CN(C(=O)C(C)CN(C)C)C1 88050,c1(C(=O)NCC2(COC)CN(C(=O)CC(C)(C)C)C2)cc(F)ncc1OC 88051,C1(C)(CNC(C(C(C)C)OCC)=O)CCN(C(=O)CCc2ccoc2)CC1 88052,Cc1nc(CCC(=O)NCC2C(C)CCN2c2nnc(C3CC3)o2)[nH]c1C 88053,CCCCC(C)CCC(=O)NC1CCCC1(C)CNC(=O)CNC(=O)CC(C)C 88054,C1(C(N(C)CCNC(=O)Cc2cncnc2)=O)CCNC(=O)C1 88055,N1(C(C(=O)NCC=C)C)CCC(O)(C(=O)NCC(C2CCCCC2)C)CC1 88056,c1(CNC(C2(F)CCN(C(c3cncc(Cl)c3)=O)C2)=O)ccnc(F)c1F 88057,Cc1ccc(Br)c(C(=O)NCCC2(O)CN(C(=O)C(O)C(C)(C)C)C2)c1F 88058,C1(C#N)(CN(C(C(=O)NCc2ccccc2)C2CC2Cl)C)CCOCC1 88059,CON=CC(=O)N1CC(CCCCNC(c2csc(C(C)(C)C)n2)=O)C1 88060,C1(C(=O)NCCC(=O)N(C)C)CSCCN1C(c1cc(Cl)n[nH]1)=O 88061,n1(CCC)ncc(-c2nc(C3CCCCCC3)nn2C(C)C(C)C)c1C 88062,Cc1[nH]c(C)c(C(=O)NCCCN(CCCCNC(C2(C)CCN(C)C2)=O)C)c1C 88063,C1(CNC(Cc2cc(C)ns2)=O)CCCCN(C(=O)C(N2CCSCC2)C)C1 88064,CC#CCCCC(=O)N1CCCC(N(C(=O)C(CC(C)C)NC(N)=O)C)CC1 88065,CC(C)(C)CCCC(C(=O)NCc1cccc(Br)c1)N1CCC(C(N)=O)CC1C 88066,N1(C(c2cnc(C)c(C#N)c2)=O)CC(C)CN(C(C23CC2C3)=O)CC1C 88067,C(CCC(C)C(=O)NC1CCN(C(=O)CCCC2(C)N=N2)C1C)OC 88068,C1(F)(C(=O)NC(C2CCOC2)CC)CCN(C(c2ccn(COC)n2)=O)CC1 88069,N1(C(C(=O)Nc2c(OC)cc(Cl)c(C)c2)=O)CCC(C2CCC(F)(F)CC2)C1 88070,N1(C(CCCCN(C(C)=O)C)=O)CC2(CCCN(C(=O)C(C)(C)S(C)(=O)=O)C2)C1 88071,C(=O)(C1=C2CCCN=C2NN1)NC(C1CCCN(C(CCC=CCC=C)=O)C1)C 88072,C1(CC(=O)NCCOCCN(C)C(c2cc(C#N)on2)=O)SC2=NCCN2C1=O 88073,C(=O)(CCCC(F)(F)F)NC(CSCC)C(=O)NCCC1CCN(C)C1 88074,C1(NC(CC2(N(C(c3ccc(C#C)o3)=O)C)CC2)=O)CCC(C)(C)CC1 88075,c1(C(C(=O)NCC(CNC(c2c(OC)n(C)nc2)=O)CO)=O)cc(F)ccc1C 88076,N1(C(CCC#C)=O)CCC2CC2(NC(=O)CCNC(c2ccc(F)cc2)=O)CC1 88077,CN1CC(CN(C(c2ccc(I)cc2)C(=O)NC2(C)CC2)C)C(O)C1 88078,N1(C(c2nnn(CC)c2C)=O)CC(C)N(C(c2cccc(COC)c2)=O)CC1C 88079,C(=O)(C(C)(C)C(F)F)N(C1CC(NC(c2ccn(CCOCCOC)n2)=O)C1)CC 88080,O=C(C1=CCCC1)NCC1(O)CC(C(N2CC(N3CC(F)C3)C2)=O)C1 88081,C1(CNC(c2n(C(C)C)nnc2)=O)CN(C(=O)CNc2ccccn2)CC12CC2 88082,N1(C(c2n(CC(C)C)ncc2)=O)CC2CN(C(=O)Cc3cnc[nH]3)CCC12 88083,c1(OC)c(C(N2C3CCC2CC(NC(c2ccnn2C)=O)C3)=O)ccc(Cl)c1C 88084,C1(C(=O)NC2C(CC(=O)NC(C#C)CCC)C(O)C2)NC(=O)OC1C 88085,C1(NC(C(CC)OCC)=O)CCN(C(=O)C(C)=C(C)CC)CC1 88086,C#CC1(C(=O)N(C)Cc2nnc(CC)o2)CCN(C(c2csc(C)c2)=O)C1 88087,Cc1nc2ccc(C(=O)NC3CCCN(C(C4(C)COC(=O)OC4)=O)C3)cc2o1 88088,C12(C(=O)NC3C(CN(C)C(c4ccc(C(N)=O)nc4)=O)CCC3)CCC(CC1)C2 88089,C(=O)(C(C)(C)CCS(C)(=O)=O)NC(Cc1ccc(OC)cc1)(C)C 88090,N1(C(CSCCC)=O)CC2CC(C1)C(CO)C2NC(=O)C(CC)N(C)C 88091,CC1(C)CCCCC(C(=O)NCC2CN(C(c3ncccn3)=O)C2)C1 88092,CC1CN(C(c2ccc(OCC(N)=O)cc2)=O)CC1NC(c1cnc[nH]c1=N)=O 88093,C1(C(=O)NC(c2cn(C)nn2)C(=O)NCc2c(OC)n(C)nc2)CCC(C2CC2)C1 88094,C12(NC(C3(C(=O)OC)C(=C)CC3)=O)CC1CN(C(c1cnc[nH]1)=O)C2 88095,N1(C(C2C(C)(C)C2)=O)CC2CCCC(NC(c3csc4cc(Cl)cnc34)=O)C2C1 88096,C1(CC)CCCC1(C)C(=O)NCC1CCN(C(=O)Cc2cccc(OCC)c2)C1 88097,C1(OCC#C)CCCN(C(=O)CONC(=O)C(C)c2cccs2)C1 88098,c1(C(=O)NC(C2(C(=O)NC3CCN(C)C3)CC2)C)ccc(F)nc1 88099,Cc1ncc(C(N2CCC(C)C(CNC(c3ccc(O)cc3O)=O)C2)=O)c(C)n1 88100,c1(C(N(CCNC(c2cc(S(=O)(=O)NC)oc2)=O)C)=O)ccc2sc(C)nc2c1 88101,n1(CCC(N2CC3(C(NC(C(C)SC)=O)CC3)C2)=O)ncc(=O)c2ccccc12 88102,Cc1ncnc(C)c1OCC(N1CCN(C(C2CC2F)=O)C(CO)C1)=O 88103,c1(CC)cnc(C(N2CCC(NC(c3ncccc3C(F)F)=O)C2C)=O)cn1 88104,C=CCC(C(=O)NCCc1cc(C)ns1)NC(C1CCCC1C(C)C)=O 88105,c1(CC(=O)N(C)C)cccc(NC(=O)NCC2C3CN(C(N)=O)CC23)c1 88106,c1(C(=O)NCC(CNC(c2c(C)onc2)=O)(C)C)nn2c(c1Br)CCC2 88107,CCCC(CC(=O)Nc1cscc1C)NC(C1CCCN(C)C1)=O 88108,c1(NC(N(CCCCCCCO)CCOC)=O)cc(NCC2CC2)nc(Cl)c1 88109,C1(NC(CSC)=O)CCCC(CN(C(=O)CC2CN(C)C2)C)C1 88110,N#Cc1cnn(CC(N2CC3C(CNC(C4CC5CCC4O5)=O)C3C2)=O)c1N 88111,c1(C(=O)NCCCCC(C)NC(CSCCCC)=O)cccc2c1OCCN2C 88112,Cc1ncnc(C(N2CCSCC2C(=O)N(CCCCC(C)C)C)=O)c1C 88113,Cc1cc(-c2ccsc2)ncc1C(=O)NC1CCC(NC(c2cocn2)=O)CC1 88114,N1(C(CC2CC(NC(CC3N(C)CC=CC3)=O)C2)=O)CC(=O)NCC12CC2 88115,N1(C(c2n(C)cnc2)=O)CC2C(NC(=O)C(c3cccc(Br)c3)O)C2C1 88116,c1(OC)ccc2c(c1)CCC2C(=O)NCC(CNC(C12CC(C1)C2)=O)C(F)(F)F 88117,C1(NC(C2CC(=C)C2)=O)CCCN(C(c2ccc(C#N)c(O)c2)=O)CC1F 88118,Cc1cc(C(N2CCSCC2CCNC(c2cnn(CC(C)C)c2)=O)=O)ncn1 88119,c1(C(=O)NCC(n2cc(CC3(O)CCC3)nn2)C)ccc2c(c1)CC(C)O2 88120,C1(NC(c2ncc(C)nc2)=O)CC2CC1CC2C(=O)NC1COCC1F 88121,Cc1nc(C)n(CCC(=O)NC(CO)C(C)NC(C2CCN(C3CC3)C2=O)=O)n1 88122,C1(C(C)C)N(C(c2cnc3c[nH]nc3c2)=O)CC12CCN(C(=O)C1CC1)CC2 88123,c1(CC(=O)NCCC(C)CCNC(C2(F)CC=CC2)=O)cccc(Cl)c1Cl 88124,N1(C(c2c(OC)n[nH]c2)=O)CCCC(C)(C)C1C(=O)NC1C2CCCOC12 88125,CC(C)CCC(C(=O)NC1CCS(=O)(=O)C1)NC(C1CCCC(=O)N1C)=O 88126,CC(CCCNC(c1cnc[nH]1)=O)NC(=O)CCc1nccn1C 88127,C1(CCCC)CCN(C(C2CC(CCNC(=O)C(F)OC(F)(F)F)C2)=O)C1 88128,C1(C(=O)NCC(CNC(C(Cn2ccc(C)n2)C)=O)O)CC(C2CC2)=NO1 88129,C1(OC)CC(NC(C2(OC)CCSC2)=O)CN(C(=O)Cc2occc2C)C1 88130,c1(CNC(CCC(C)N(C)C)=O)cccc2nccnc12 88131,CC(C)CC(C)(O)C(=O)NCC1CCN(C(c2ccc(CN(C)C)[nH]2)=O)C1 88132,N1(C(CCCCOC)=O)CC(NC(C2(C(=O)N(C)C)CC2)=O)CC(F)(F)C1 88133,Cc1ccc(O)c(C(N2CCC(O)C(NC(C3CC4(C3)CC4F)=O)C2)=O)n1 88134,C1(NC(c2ccc(C#C)cc2)=O)CC2CN(c3nccc(C(F)(F)F)n3)CC2C1 88135,N1(C(CCC)=O)CCC2(C=C(C(=O)N(C)Cc3cn[nH]c3)C2)C1 88136,N1(C(=O)COc2cccc(Cl)c2)CC(NC(C2(F)CC=CC2)=O)C2CC2C1 88137,C1(C(=O)NCCn2ccnc2)CN(C(c2ccnc(-c3ccccc3)c2)=O)CCN1 88138,CP(C)(=O)c1ccc(C(=O)NC2COCC2NC(=O)Cc2cn3ccsc3n2)o1 88139,c1(C(N2CC=CC(NC(CCCCSC)=O)C2)=O)cnc2n1CCCCC2 88140,CC1(C)CCCN1CCC(=O)NCCn1cc(C(c2ccccn2)O)nn1 88141,c1(SCNC(C(c2ncc(CC)o2)N(CCC2CC2)CC)=O)ccc(Br)cc1 88142,c1(C(=O)NCC2CCN2C(C23CC(F)(C2)C3)=O)cnc2ccsc2c1 88143,C=C(C)CC(C)C(=O)NC1CN(C(c2csc(CO)n2)=O)CC1O 88144,c1(NC(=O)NC2C=CCN(C(C3CCCO3)=O)C2)ccc(Br)cn1 88145,CCCCC(=O)C(=O)NCC1CN(C(c2cc(C)sc2C)=O)CCC1C 88146,c1(C(N(CCOC)C)=O)cc(CNC(C2CC2(C)C(F)F)=O)on1 88147,N1(C(C(C)OCCCC)=O)CCCN(C(=O)C=CSc2ccco2)C(C)C1 88148,C(=O)(C1CCCc2ncnn21)N1C(CCN(C(C=C(C)Cl)=O)C)CCCC1 88149,c1(CCC(=O)NCC(CNC(c2n(CC=C)ccc2)=O)F)nc2ccccc2s1 88150,C=C(Cl)CCC(=O)N(CC(C)NC(=O)C(C)(C)c1cscc1Cl)C 88151,Cc1cccc(C(C)(C)C(=O)NCCCC(C)NC(c2nc(C(C)C)cs2)=O)c1 88152,C1(CNC(c2ncsc2Br)=O)CN(C(=O)CNC(=O)C(F)(F)F)CCO1 88153,Cc1ncccc1CCCNC(C1(NC(=O)COc2ccccc2)CCCC1)=O 88154,N1(C(=O)C(O)Cc2ccccn2)CCN(C(=O)Cc2ccsn2)C(CO)C1 88155,c1(CN2CC(CC(=O)NCCOCCCC)C2)ccc(Cl)nc1C 88156,c1(COC)ccc(C(N2CCC(N(C(=O)C(CO)NC(N)=O)C)CC2)=O)cc1 88157,c1(C(c2n(CCOCC)nnn2)NC(C2COC2)C)cccc(F)c1OC 88158,Cc1ccc(-c2ccc(C=O)cn2)c(CN2CCCC(C)CC2)c1 88159,N1(C(c2cc(C)c(N)cn2)=O)CCN(C(C2CN(C)CC(C)O2)=O)CC12CC2 88160,c1(C(N(C2CCCN(C(=O)Cc3ccccc3)CC2)C)=O)cnc2ccnn2c1 88161,C1(C)(C(=O)NCCC2(OC)CN(C(=O)C(F)(F)CN(C)C)C2)CCOCC1 88162,c1(C(N2CCC(NC(C3(CC#C)CCCC3)=O)C(C)C2)=O)cc(O)cc(C#N)c1 88163,C=CC(CC)CC(=O)NN(C(C)C(=O)N(C)CCOC(C)=O)C 88164,N1(C(C(C(C)O)(C)C)=O)CC2CCC1CN2C(=O)CCc1ccccn1 88165,C1(CNC(c2ccc(C(=O)OC)o2)=O)CCCCN1C(=O)C(C1CCOCC1)F 88166,c1(C(N2CC(NC(c3ccc(CO)cc3)=O)C(F)(F)C2)=O)cc(Br)cc(Br)c1O 88167,Cc1nc(O)nc(C)c1CC(N1CCCCC(CNC(=O)C(N)=O)C1)=O 88168,c1(C(N2C3(c4cn(CCCSCC)nn4)CCC2CC3)=O)ccccc1[N+](=O)[O-] 88169,N1(C(CN(C2CCC2)C(c2n(C)ccc2)=O)=O)CCOCC(CO)C1 88170,C(C)(C)(C(=O)NCC=CC(=O)NCC1CC1CC(C)C)SC 88171,c1(C(=O)NCC2C(C(=O)NCc3cn(CC)nc3)CCO2)cncc(OC)n1 88172,C(=O)(C1COc2ccccc21)N1CCC(NC(CC2(CSC)CC2)=O)C12CC2 88173,C1(CC)(NC(=O)CCc2ccoc2)CCN(C(c2n[nH]c3c2CCC3)=O)CC1 88174,c1(C(=O)NC2CC(C)N(C(c3cnc(C4CC4)s3)=O)C2)ccc(P(C)(C)=O)o1 88175,CCCCN=C(NCCc1ccc(F)cc1F)NCC1CC(=O)N(CCC)C1 88176,CC(C)C(C(=O)NCC1CCC(F)(F)C1)C(C)NC(=O)CC1C=NN(C)C1=O 88177,Cc1csn1CC(=O)NCCN(C(=O)CC1CCCC1)C1CC1 88178,N1(C(C(C)(F)CC2CCCC2)=O)CC2(CCN(C(c3cncs3)=O)C2)C1 88179,C(CC(=O)NCC1CN(C(=O)C=C2CCCCC2)CC1O)(C(C)C)OCC 88180,S(=O)(=O)(c1cnn2ccc(=NC(C)CCOC)[nH]c12)NC(C(CC)CC)C 88181,C1(C(=O)NC2CC(C)(NC(C(c3cn(C)nc3)=O)=O)C2)C2CCN(CC2)S1(=O)=O 88182,c1(C(N2C(CCCNC(c3cnc(S)[nH]3)=O)CCCC2)=O)ccc2nc[nH]c2n1 88183,N1(C(=O)Nc2ccnn2C2CCC2)CCC2(CCCCO2)C1 88184,C(c1ccc(F)cc1Cl)=CC(N1CC2CN(C(CCCC#C)=O)CC21)=O 88185,Cc1c(NC(C2CC(F)(F)CN2Cc2cn3ccccc3n2)=O)ccc(Br)c1Br 88186,n1(CCC)nc(C)cc1C(=O)NC1CCC1NC(c1cccc(C(N)=O)c1)=O 88187,c1(C(=O)NCC2CCCN(C(C3(C)N(C)CCC3)=O)C2)ccc2nc(O)[nH]c2c1 88188,N1(C(c2cncc(NC(CC)=O)c2)=O)CCC(C)C(NC(=O)CC(C)(C)F)C1C 88189,C1(CNC(CC2(C)CCC2)=O)CC(F)CN1C(=O)CN(C1CCCC1)C 88190,c1(C(N2CCC(c3cnccn3)C2)C(=O)N(C2(C)CC2)C)cnccn1 88191,Cc1ccc(F)c(C(=O)NCCC(C)(C)NC(=O)CC2CCC(O)C2)c1F 88192,CCC1=NOC(C(N2CC=CC2CNC(c2cnoc2COC)=O)=O)C1 88193,CCCCC(C(=O)NC1CCN(c2cc(F)ncn2)C1C)NC(N)=O 88194,N1(C(c2n(C)ccn2)=O)CC2CCOC2(CNC(c2ccsn2)=O)C1 88195,c1(NC(Cn2cc(C(=O)NC)nn2)=O)ccc(C)c(N(C)C)c1 88196,c1(CNS(=O)(=O)Cc2ccccc2N2CCCCC2)cc(I)ccc1O 88197,c1(OCCCC)ccc(C(=O)NCC2(C)CC2(Cl)Cl)cc1OCCC 88198,c1(CC(=O)NCC2C(C(=O)NCC(N3CCOCC3)C)C2)cn(C)nn1 88199,C1(C(=O)NCC2N(C(CC=CC(C)(C)C)=O)CCOC2)CCC(C2CC2)CC1 88200,N1(CC(CC)C)CCS(=O)(=O)C(CCNC(=O)Cc2nnn(C(C)(C)C)n2)C1 88201,N1(C(CC=CCC)=O)CC2CCC(C1)C2CNCc1ccc(-n2cncn2)cc1 88202,C1(CC(=O)Nc2ccc(O)c(Cl)c2)CC(N=c2ccnc(N3CCCC3)[nH]2)C1 88203,CC(C)CCC(O)C(=O)NC(CC1CC1)C(N1CC(=O)NCC1C(N)=O)=O 88204,c1(OC(CNC(=NC)NCCc2cnccn2)(C)C)ccccc1C#N 88205,N1(C(COCCC)=O)CCC(C)(C(=O)NCC2CN(C(C)C)CCO2)CC1 88206,C1(C(N(CCCCCNC(c2c(C)ocn2)=O)C)=O)CC12CCC(F)(F)CC2 88207,Cc1ccc(N)c(C(=O)NC2CN(C(=O)C(n3nc(C)cc3C)C)CC2(C)C)c1 88208,C1(N(C(=O)CCc2csc(C)n2)CC#C)CCN(C(C2CCC(C)S2)=O)CC1 88209,c1(C(=O)NCC2CC3(CC(NC(CC4(C)CC4F)=O)C3)C2)ccc2n[nH]cc2c1 88210,N1(C(CC(C)(C)C)=O)CC2CCCC(NC(c3coc4c(F)cccc34)=O)C2C1 88211,N1(C(COC(C)C)=O)CC(NC(=O)Cc2cc(C(C)C)no2)CC(O)C1 88212,c1(C(=O)NCC2C(NC(CCC=C)=O)CC2)c(C)ccc(F)c1O 88213,c1(N2CCC(NCCCOC)C2)oc(Cc2ccccc2)nc1C#N 88214,c1(C(N2C(CNC(CCc3c(C)c[nH]c3C)=O)COCC2)=O)nc(Cl)ccc1F 88215,C(=O)(C1CCc2c(Cl)cccc21)N(CCCNC(=O)COC1CC1)CC 88216,CC(C)CC(C)(C)C(=O)NC1CN(C(c2ccncc2Cl)=O)CC2(CC2)C1 88217,C(C)(C)(CCCC(=O)N1CCC2C(O)CC12)NC(CCc1n(C)cnn1)=O 88218,C(=O)(C(F)CC(C)(C)NC(c1cc2ccccn2n1)=O)N(C)CCc1cccs1 88219,C1(C(=O)NCC2C(C)CCCN2C(C2CC2C(C)O)=O)CCCC2C1C2(F)F 88220,C(C(COC)C(=O)N1CCCC(CCCO)C1)OC 88221,CCC(C)C(O)C(=O)N1CCCC(NC(c2ccnc(Br)c2N)=O)C1 88222,c1(C(=O)NC2CCC(N(C(c3ncc(CC)s3)=O)C)C2)ccc(C2CC2)cc1 88223,C(=O)(C(C)(CSC)NC(=O)C=CC1CCOC1)N1C(C)(CC)CC1 88224,N1(C(C2C(C)(C)C2)=O)CCC2CC1CN2C(=O)CNC(=O)CC1CCCCC1 88225,C(=O)(CC1OCCc2ccccc21)NC(CNC(c1cc(C(C)C)on1)=O)(C)C 88226,C1(C(N2C(CCNC(c3[nH]cc(C(C)=O)c3)=O)CCCC2)=O)C(C)(C)OC1(C)C 88227,Cc1cc(C(N2CCCC2CC(=O)NC(C)CC2(O)CCC2)=O)c(N)s1 88228,C(C(=O)NCC1CCCN1C(=O)CC1OCCO1)(C(C)C)n1cc(C)nc1 88229,C#CCC(CC(F)F)NC(=O)CC1CN(C(=O)CCN2CCOC2=O)CC12CC2 88230,C(=O)(CCCCCC#N)NCC1CC2(CN(C(C3CN(C)C(=O)N3)=O)C2)C1 88231,CC(c1cccnc1)=CC(=O)NC1CCN(C(c2conc2C)=O)CC1F 88232,Cc1cc(C(N2CCC(C(N3CC(C(=O)OC(C)C)C3)=O)C2C)=O)c(C)nn1 88233,N1(Cc2c(OCC=C)cccc2)CCC(O)C(C(N2CCOC(O)C2)=O)C1 88234,C(CCN=C(NCCC(C)C)N1CCC(OC(F)F)C1)Oc1cccc(C)c1 88235,CC1CC(CC(=O)OC2(C)CN(C(=O)CSC(C)(C)C)C2)CN1C(=O)OCO 88236,C(=O)(C(C)P(C)(C)=O)NC(CNC(C(C)(F)F)=O)C(C)(C)C 88237,N1(C(C(CCCC)=O)=O)C(CNC(=O)C(c2cnn(C)c2)C)CC2CCCCC12 88238,C(CO)(C(=O)N1CC(CN(C)CCF)C1)O.C(=O)(CCNC(=O)CO)OC 88239,CN(C)NC(=O)CCC(=O)NC1(C)CCN(C(c2cnoc2C2CC2)=O)CC1 88240,c1(OC)c(C(=O)NC2CC(C)(NC(C3CCOC3C)=O)C2)sc(Cl)c1Cl 88241,C1(C(N(C2CCN(C(=O)C(=O)N3CCCC3)C2)C)=O)CCc2cncn2C1 88242,C1(CCNC(c2sc(F)cc2Cl)=O)CCCN(C(c2ccc(CCO)cc2)=O)C1 88243,C(=O)(CC(C)(F)F)NC(C=CC(=O)N(CCCC#C)CC)(C)C 88244,c1(CC(N2CCC3CN(C(c4c(C)coc4)=O)CC32)=O)coc2cc(O)ccc12 88245,n1(CC(N2CC(N(C)C(c3cnsn3)=O)C(F)C2)=O)cc2ncccc2n1 88246,Cc1ccnc(O)c1C(=O)N(CC(O)CN(C(=O)CC1(N2CCCC2)CC1)C)C 88247,N1(C(c2c(C)cco2)=O)CC2C3CCC(C2C1)N(C(=O)CSCC(N)=O)C3 88248,Cc1c(N)ccc(C(=O)NC(C)(C)CNC(C2CCC(C)(C)O2)=O)c1C 88249,N1(C(CNC(CC)=O)=O)CCCC2C1CCCCN2C(=O)C(O)C(C)C 88250,CC(O)CCCCCC(=O)NC1CCCCC1NC(c1ncn(C(C)(C)C)n1)=O 88251,C=CCCCCCCC(=O)NC1CCC(NC(=O)C=C(C)c2ccccc2F)C1 88252,N1(C(C2C(COC)C2)=O)CCn2ncc(CN(C)C(c3nocc3C)=O)c2C1 88253,c1(C(=O)NCCCC(=C)C)ccc(CNC(C2(C)CCOC2C)=O)nc1 88254,c1(C(=O)NC2CN(C(COC(CC)(C)C)=O)CC2(C)C)nccc2cccnc12 88255,C1(CNC(=O)CCc2nccs2)CN(C(C2CC2F)=O)CCC12CCOC2 88256,c1(C(N2CCC3CN(C(C4(F)CCCC=C4F)=O)CC23)=O)cc(Cl)cc(Cl)c1O 88257,N1(C(c2ccc(C(F)F)o2)=O)CCC2CCN(C(=O)CCc3cccs3)C2C1 88258,CC1CN(C(c2cc(O)nc(O)n2)=O)CCCN1C(=O)C(c1ccccc1)F 88259,c1(OCC)cc(F)c(-c2ccc(NCc3cc(C(F)(F)F)ccc3Br)s2)c(F)c1 88260,C1(C(=O)NC2C(NC(c3cn(CCC4CC4)nn3)=O)CCC2)CC12CCOC2 88261,CCCC(C(C(=O)NC1CCC1)N1CCCC(C(O)C(F)(F)F)C1)OC 88262,CC1CN(C(=O)C(=O)NCc2cnn(C3CC3)c2)CCS(=O)(=O)C1 88263,C12(C(=O)NC3(C)CN(C(C(c4ccccc4F)C)=O)C3)COC(CCO1)C2 88264,c1(OC)cc(F)c(C(=O)NC(C)CCCCNC(c2cc(C)ncn2)=O)c(Cl)c1 88265,C1(NC(CCC(C)=O)=O)CC2(C1)CC(C(=O)Nc1cccc(C(=O)N(C)C)c1)C2 88266,c1(C(N2C(CC)CN(C(=O)C(C)(O)CC)CC2)=O)cn2cccc(Cl)c2n1 88267,c1(NCCOCCNC(c2ccco2)=O)cccc(Cl)c1.O=C1CCN1 88268,c1(C(=O)NC2CC(NC(C3CC3Cl)=O)C2)cccc(C)c1.CC 88269,c1(C(=O)OC(c2c(OC)cccc2)C)c(C)ncnc1O 88270,N1(C(c2nn(C)c(CO)c2)=O)CCC(NC(C2CC3C=CC2C3)=O)C(C(N)=O)C1 88271,c1(C(=O)NC2(C)CC(NC(c3c(OCC)cccn3)=O)C2)ccc(C#N)cn1 88272,N1(C(C(=O)N(C2(CNC(CC#N)=O)CCOC2)CCl)C2CC2)CCS(=O)(=O)CC1 88273,N1(C(C2C3CN(C(C(COC)NC(C)=O)=O)CC32)=O)CCc2c(Cl)cccc2C1 88274,N1(C(=O)C2=CCCO2)CCC(C2CCCN(C(C3CC4(CCOCC4)C3)=O)C2)C1 88275,N1(C(C(COC)COC)=O)CCN(C(=O)CC2CN(C(C)=O)C2)CC1CC(F)F 88276,CN1CCCC(NC(=O)NNC(=O)C2COCCN2)CC1 88277,Cc1c(Cl)c(C(N2CC3(C2)CN(C(c2c(Cl)nn(C)c2Cl)=O)C3)=O)nn1C 88278,CCC(N=c1[nH]c(=NC(C)c2ccncn2)c2ncccc2[nH]1)c1ccncc1 88279,N1(C(C)=O)CCC(C(=O)NCCCNC(=O)Cc2cccs2)CC1 88280,c1(C(=O)NCC(C)N(C(=O)C(C2CCCCC2)=O)C)csnc1C1CC1 88281,C1(C2(O)CCOC2)(CNC(c2c(OC)cc(NC(C)=O)cc2)=O)CC1 88282,c1(OCC(N2CC(NC(c3c(C)csc3)=O)C(C)(C)C2)=O)ccc2c(c1)CCC2 88283,C1(NC(CCN(CCC)C)=O)CCC2CCN(C(=O)CC3CNC(=O)C3)C12 88284,C(=O)(CC(O)CC(C)(C)C)N1CCC(=C)CC1C(=O)NOCC1CCC(OC)CC1 88285,C1(NC(c2c(C)nc(CNC(C3CC(=C)C3)=O)o2)=O)CCOC(C)(C)C1 88286,C(C)(CCC(C)(C)C)(C(=O)O)NC(C(C)S(N)(=O)=O)=O 88287,C(C(Cc1ccc(F)cc1)C(=O)O)NC(c1cccc(N2CCOCC2)n1)=O 88288,Cc1ccccc1-n1ccc(C(=O)NC2(CN(C)C(c3[nH]cnc3C)=O)CC2)n1 88289,Cc1nnccc1NCCNC(N1CCOC(C2CC(F)(F)C2)C1)=O 88290,Cc1nc(C)c(C(=O)NC(C)(CNC(=O)Cc2cscc2Br)CO)[nH]1 88291,c1(C(=O)NCC2C(CNC(C=CCCC)=O)C2)c(Cl)cncc1Br 88292,c1(OC)ncc(NC(C2CCN(C(=O)CC3CC(OC)C3)C2C)=O)cn1 88293,N1(C(C(CN(C)C)(F)F)=O)CCCC(CCNC(c2ccc(Cl)s2)=O)CC1 88294,C1(NC(Cc2coc(C)c2C(F)(F)F)=O)CCN(C(=O)CNC(N)=O)C1(C)C 88295,c1(C(N(C(C)CNC(=O)C(O)C2CCC2)CC)=O)cccc(-c2nc(=O)o[nH]2)c1 88296,c1(C(N2CCC(NC(CSCC=C)=O)C2(C)C)=O)ccc(C)c(C)c1O 88297,CC(CNC(=O)CC1CCOC1(C)C)CC(=O)NCCC1(C)CCCC1 88298,C1(NC(C2N(C(C(C)NC(=O)OC)=O)C3(CC2)CC3)=O)CCN(C)CC1C#N 88299,O=C1CC2C(C(N3CCCC(NC(C4(C5CC5)CCCO4)=O)C3)=O)C2C1 88300,CN1CC(NC(C2CCC2NC(=O)CCN2CCOC2=O)=O)CC1=O 88301,N1(Cc2ccc(C(=O)Nc3cc(C)cc(C)n3)cc2)CC2CC3CCCN3C2C1 88302,CC(C)C#CC(=O)NC(C)C=CC(=O)NCC1(C)COCCO1 88303,[N-]=[N+]=NCCCCCCNC(=O)C(C1(O)CCCCC1)NC(=O)CCC1CC1 88304,CCCC(C)(O)CC(=O)NC(C)CCNC(c1cc(Br)cnc1N(C)C)=O 88305,c1(OC)cc(C(N2CC(OC)CC2CNC(c2ccc[n+]([O-])c2)=O)=O)cc(Cl)n1 88306,c1(OCC=C)cccc(C(c2nnnn2CC(F)F)NCCC(C)CO)c1 88307,N1(C(c2c(SC)nccn2)=O)C2CCC1CN(c1nc(C)cc(C#N)n1)CC2 88308,n1(CC)ncc(C(N2CC=CC(NC(c3cnc(N(C)C)cn3)=O)C2)=O)c1C 88309,c1(C(=O)NC2CC(O)(CNC(C(C3CC3)OCC)=O)C2)cnc2c(c1)COC2 88310,N1(C(CN(C(C)C)C)=O)CCC(CCCNC(=O)CCc2ccc(F)cc2)CC1 88311,C1(C(=O)NCCCOCCN(C(c2cn(CCC)nn2)=O)C)CCCOC1C 88312,C1(CNC(c2nc(CNC(CNC(C(C)(C)C)=O)=O)oc2)=O)CC[Si](C)(C)C1 88313,C12(C(=O)NCCCCC(C)NC(C(C)c3ncco3)=O)CC3CC(CC(C3)C1)C2 88314,c1(C(=O)OC)ccc2oc(CNc3nccc(C)n3)cc2c1 88315,N1(C(CCC#CC)=O)CCC2(CC1)OCCC2NC(c1cc(OC)n[nH]1)=O 88316,c1(C(N2CC3C(CCNC(c4c(C)cco4)=O)(CC3)C2)=O)cccc([N+](=O)[O-])c1 88317,C1(NC(C(c2cn(C)nc2)=O)=O)CN(C(C2CCC(N(C)C)CC2)=O)CCC1F 88318,N1(C(c2ncc(C)cc2F)=O)CC2CC(NC(=O)C(C)C)CC2C1 88319,CC1(C)CCCC(CNCCCn2ncc3ccccc23)CC1 88320,c1(CN2C(CC)CCC2)cc(C)cc(N)c1 88321,C(=O)(C(F)(F)C(F)F)NCC(CNC(C1(CC#C)CCOC1)=O)F 88322,C12(C(=O)NCC3CC(NC(=O)Cc4cccc(O)c4)C3)CSCC1C2(F)F 88323,c1(OC)ccc(C(=O)CCC(=O)N2CCCC2(C)CNC(=O)C(C)SC)cc1 88324,C1(CNC(=O)CC2CN(C(=O)CCN3CCC3)CCO2)CCC(C(=O)O)CC1 88325,C1(C(=O)NCCC2(O)CN(C(c3cc(CC)[nH]n3)=O)C2)CCS(=O)(=O)N1C 88326,Cc1cnn2cc(C(N3CCCC3CN(C(=O)CCSCC(N)=O)C)=O)cnc12 88327,c1(CCC(=O)NCC2CCN(C(c3c(C)cco3)=O)C2)cccc2c1OCCO2 88328,c1(CC)cc([N+](=O)[O-])ccc1N(CCNC(=O)C(C)C(C)(C)C)C1CC1 88329,C12(NC(CC(C)C3CCCC3)=O)CC1CN(C(=O)Cc1csc(Cl)n1)C2 88330,C1(CC(N2CC(CC)(NC(=O)CC(=O)NCC3CC3)C2)=O)CCN(C)CC1 88331,c1(CC)[nH]c(=N)sc1C(=O)N(CC(C)N(C)C(c1cncnc1C)=O)C 88332,N1(Cc2c(C)nc[nH]2)CCc2nc(C(=O)NC3CCC(N(C)C)CC3)cn2CC1 88333,N1(C(C=Cc2n(CC)ccn2)=O)CCCC2(NC(=O)C=CC(=O)OCC)CC2C1 88334,c1(SC(C2CCCN(c3nccs3)C2)C)cccc(OC(F)(F)C(F)(F)F)c1 88335,c1(C(N(CC(O)CNC(=O)C#CC2CC2)C)=O)cnc2c(F)c(F)ccc2c1 88336,c1(C(N(CCC(C(C)C)NC(C(C)OC)=O)C)=O)cccc2ncc(Br)n12 88337,C1(CC(=O)Nc2cc(CC)no2)CCCN(C(C2CCC(=O)O2)=O)C1 88338,CCC(C)(C)CC(=O)N1CCC(C)(C(=O)NC2CC3(CC3)C2)C1 88339,c1(NC(C)=O)cccc(C(=O)NC2CCCC(CNC(c3scnc3Cl)=O)C2)c1 88340,c1(C(N(C)CC2(O)CCN(C(=O)Cn3cnnn3)C2)=O)cc2c(ccn2C)[nH]1 88341,N1(c2c3ncn(CC)c3nc(Cl)n2)CCc2cc(C)ccc2C1C 88342,N1(C(C(CN(C(COCCC#C)=O)C)(C)C)=O)CC2OCCN(C)C2C1 88343,N1(C(CSc2c(C)cccc2)=O)CCC2(CCN(C(C3(C)CC4CC4C3)=O)C2)C1 88344,c1(C(=O)NC2CCC(NC(c3c(OC)cc(Cl)nc3)=O)C2)cc(C)c(F)cc1Br 88345,c1(C(C(=O)NCC2(C)N(C(c3onc(CC)n3)=O)CCC2)C)cc(C)cc(F)c1 88346,C1(C(=O)NC(C)(C)CNC(C2CC(C)(F)C2)=O)CCCC1(F)F 88347,c1(C(N2C(CCNC(=O)C3=CCCCC3)CCC2)=O)cc2cccn2cn1 88348,C#CC1CN(C(=O)CCc2ccnn2C)CCN1C(c1cnn(C(C)(C)C)c1)=O 88349,CCC(CC(C)C)C(=O)N1CCC(CC(C)NC(=O)C(C)(C)c2nccs2)CC1 88350,c1(CNC(C=CC)=O)nn(C)c2c1CN(C(c1ccnc(C)c1)=O)CC2 88351,C1(C(=O)NCC(CCNC(=O)CCc2cnco2)O)CCc2ccccc2C1 88352,C1(C(=O)NCC2(O)CC(NC(Cc3ccc(C)o3)=O)C2)CCCCN1S(N)(=O)=O 88353,C1(C(=O)NC2(CC=C)CCOC2)CCCC(NC(=O)CNC(=O)CN(C)C)C1 88354,c1(C(=O)OCC)cnc(NC2CC3(C2)CC3NC(c2[nH]nc(OC)c2Cl)=O)cn1 88355,C1(C(F)(F)F)(C(=O)NC(CC)CNC(c2ccnnc2)=O)CC=CCO1 88356,N1(c2nccc(N3CCC(CC(N)=O)C3)n2)CCC(O)(CC2CC2)CC1 88357,N1(c2nnc(C)s2)CCOC2(CCN(C(=O)Cc3ccc4ncnn4c3)CC2)C1 88358,N1(C(CC=CC)=O)CCCCC1CCN(C(=O)C(C(=O)OC)OC)C 88359,c1(OC)nn(C)cc1N(C)C(C1CC(CNC(=O)CCCC2CC2)C1)=O 88360,N1(C(CCCOCC)=O)CCC(NC(c2ccc(SCC)cc2)=O)C12CCCC2 88361,N1(C(C=CCC)=O)CCCCC1CN(C(C1(C)COC1)=O)CC 88362,N1(C(c2cc(CCNC(c3cnc(C)o3)=O)on2)=O)CCOC2CC12 88363,c1(CC(CNC(C2CCCCC2)=O)NC(=O)CCC2CCCO2)ccccc1 88364,C1(CC)CC(C(=O)NCC(C)CC(=O)OC)CCN1C(c1c[nH]c(=N)c(C)c1)=O 88365,N1(C(CSCC#C)=O)CCC(O)(CCNC(=O)C(c2nc(C)cs2)C)C1 88366,C1(C(=O)NCCC2CN(C(C3CC(C4CC4)C3)=O)C2)(CC)CCCCO1 88367,C1(C(N(CC)CC2CCCO2)=O)C2CN(C(=O)CC3COCCO3)CC12 88368,N1(C(CC2CCN(C(C3C(CCC)CCC3)=O)C2)=O)CC(NC(C)=O)C2(CC2)C1 88369,n1(CC)nc(C(=O)NCC(C)NC(C2COCC3(CCC3)O2)=O)c2c1CCOC2 88370,n1(CC)cnc(C(=O)NCC2(NC(c3ccn(CC(C)C)n3)=O)CCCC2)n1 88371,c1(C(=O)NCCn2ccnc2)cc2ccc(-c3cnn(C4CC4)c3)cc2s1 88372,N1(C(c2c(CC)non2)=O)CCC2(CCCN(C(C3CCN(CC)C3)=O)C2)C1 88373,C1(C2CN(C(=O)C(C)CC=CC)C2)(NC(C(C=CC)O)=O)CC1.C(CCC)=C 88374,N1(Cc2cn(C3CC(C(=O)NCC(CO)CO)C3)nn2)CC(=O)NC1=O 88375,c1(CC(N2CC(NC(C3N(CC)CC3)=O)C(O)C2)=O)cc(C)ccc1OC 88376,C1(C(N2C(CC)CN(C(=O)CCCF)CC2)=O)CCC(C2CC2)CC1 88377,C1(CCNC(c2csc(C3CC3)n2)=O)CCCCN1C(c1cc[nH]n1)=O 88378,C#CC1(O)CC(C(=O)N(CC(C)N(C(C2(OC)CCSC2)=O)CC)C)C1 88379,CCC(C(=O)NCC1(OC)CC1)N(C(=O)C(C)(F)c1ccon1)C 88380,c1(NC2(C)CCN(C(C(C=CC)O)=O)C2)ncc(C(=O)OCC)cc1[N+](=O)[O-] 88381,C1(NC(=O)C2CC2)CCCC1C(=O)NC1CC(F)(F)C1 88382,CC(CN1CCOCC1)C(=O)NC(C)CCN(C)C(c1ccco1)=O 88383,c1(NCC(CC)(C)OC)ccc(S(=O)(=O)NCC(C)(C)COC)c(Cl)c1 88384,c1(C(=O)NC2CCC(CNC(CS(N)(=O)=O)=O)C2)cnc2nccn2c1 88385,C1(CNC(CSCC(C)C)=O)COC(CNC(=O)COCCC(C)C)C1 88386,C1(C(=O)NC(C2(CNC(c3cc(C)n(C)c3)=O)CC2)C)CCC(C)(C)OC1 88387,N1(C(COCCOC)=O)CC2CC2(C(=O)NC(CO)C(=O)O)C1 88388,N12CC3CC1CN3C(=O)C(O)C1CN(C3CN2C3)C1.C(=O)NC 88389,N1(C(c2cncc(C#C)c2)=O)CCC2(CCCC2CNC(=O)C=CCO)CC1 88390,N1(C(=O)OCC)CSCC1C(C(=O)CCCc1ccccc1)=O.C1(CN)(O)CC1 88391,C1(NC(C(CNC(C2(CC#C)CC2)=O)OC)=O)CC(C)(C)C12CCC2 88392,N1(C(C(=Cc2ccco2)C)=O)CC2(CCN(C(=O)CC(C)(C)C(=O)OC)C2)C1 88393,CC1OC2(C(=O)NC3CCN(C(c4cc(C(N)=O)co4)=O)C3)CC1C2 88394,C#CCCCCC(=O)NC1CCC(NC(C2(CCOC)CC2)=O)C1 88395,CCC(CC)CCC(=O)NC(c1ccccc1OC)C(C)NC(C1CCCC1)=O 88396,Cc1ccn2ncc(C(N3CC4(CCC4NC(c4ccco4)=O)C3)=O)c2c1 88397,N1(C(COCCC)=O)CCC(C)CC1CNC(=O)CCc1cccnc1 88398,N1(C(C=CCOC)=O)C2CCCC1CC(NC(C1CC(n3cnnc3)C1)=O)C2 88399,c1(CNc2c(OC)cc(C(F)F)cc2)cc2ccccc2o1 88400,C1(F)(C(N(CCCNC(C2(F)CCOC2)=O)C)=O)CCCCC1 88401,CC1(C)CCC(NC(c2cncnc2)=O)C(CNC(=O)C2=CCCOC2)C1 88402,c1(C(=O)NC(C)CNC(=O)CCN2CCSC(C)(C)C2)cccc2c1COCC2 88403,C1(C(N2CCC(N(C(C(C)=CC)=O)C)C2)=O)CC2CCC(C1)C2F 88404,N1(CC(=O)NCC2C(C)CN(C(=O)C=CC3CCOC3)C2)CCCCCCC1=O 88405,Cc1cc(F)ccc1C(=O)N(C1C2CN(C(C3CCCOC3C)=O)CC12)C 88406,CCC(C)(C(=O)N1CCC1CNC(c1cncc2[nH]ccc12)=O)C(F)F 88407,CN1CCC2CCC(C1)N2C(=O)CC(O)CNC(=O)C(C)(C)C(N)=O 88408,C1(NC(C2(OC(C)C)CCOC2)=O)CN(C(=O)Cc2cccs2)CCC12CCC2 88409,N1(C(C(=O)NC(CC)C)CCC2CC2C)CC(C(=O)OC)C(C2CCCCC2)C1 88410,c1(NC(C(F)=CC)=O)ccc(NC(c2cc(CC(C)C)c[nH]2)=O)cc1C 88411,N1(C(C(C)C(C)(F)F)=O)CCC(C2(O)CN(C(=O)CNS(N)(=O)=O)C2)CC1 88412,N1(C(c2cnc(C(C)=O)s2)=O)CC2CC1CCC2NC(=O)C(C)SC(F)(F)F 88413,c1(CC(=O)NCCN(C(C(C=CCCC)O)=O)C2CC2)ccc(C)cc1Cl 88414,c1(OC)ccc(F)cc1CC(=O)N(C1CCCN(C(C2CCCO2)=O)CC1)C 88415,N1(C(C2C(C#C)C2)=O)CCOCC1CN(C(=O)C=CCOC)C 88416,CC(F)(F)C(C)(C)C(=O)NCC1CC(F)(F)CN1C(C1COCCN1C=O)=O 88417,c1(C(N2CCC(N3CCOC3=O)C2)C(=O)NCCOC)cnc(OC)c(Cl)c1 88418,C(=O)(C(O)C(F)(F)F)N(CC(CC)NC(=O)C(O)Cc1ccccn1)CC 88419,c1(C(=O)NC(CCN(C(c2cc(=NC)[nH]cc2)=O)C)C)cnc2c(c1)COC2 88420,N1(C(C(CCC)F)=O)CC(CNC(c2c(C)csc2C)=O)CC(C)C1 88421,C(CO)(C(O)c1cccnc1)NC(c1nc(Br)c[nH]1)=O 88422,c1(OCC(N2C3CC(NC(C4N(C)C(=O)OC4)=O)(C3)C2)=O)ccc(Cl)cc1F 88423,C(C(C(C)(C)C)NC(=O)COC1CCOCC1)NC(COCCC#C)=O 88424,CCC(C)C(=O)NC(C)CCCNC(c1cnoc1-c1ccco1)=O 88425,CCCCCC(C)C(=O)N1CCN(C(=O)COc2ccc(Br)cc2)CC1C#N 88426,C(=O)(C(F)C(F)(F)C(F)(F)F)NC1C(CNC(C(=O)N(C)C)=O)CC1 88427,N1(C2CN(C(CC3(CC(C)C)CC3)=O)C2)CC(NC(=O)C(=O)NC(C)C)CC1=O 88428,C1(NC(=O)CCc2cc(C3CCC3)on2)(CO)CCN(C(=O)CC(F)F)C1 88429,c1(C(=O)NCC2CN(C(C3C(C(=O)NCC#C)C3)=O)C2)n[nH]c2c1CCCCC2 88430,C1(CC(=O)NCC2N(C(C3(O)CC(C)(C)C3)=O)CC2)Cc2ccc(Br)cc2C1 88431,C1(C(=O)NCCN(C(C2CCCN2C(=O)NC)=O)CC)(CSC)CC(F)(F)C1 88432,c1(NC)cnncc1C(=O)NCC1CCC(NC(c2cc(O)ncn2)=O)C1 88433,CC(CC(=O)NCc1ccccc1CNC(=O)C1=NNC(C(F)(F)F)C1)C(C)(C)C 88434,C1(C(=O)NC(CC(C)NC(c2cnc(C)s2)=O)C)Cc2ccccc2N1 88435,CCC(CC)CCCC(=O)N1CCCC1C(N1CCCC(N=[N+]=[N-])C1)=O 88436,C1(NC(c2cc(C(N)=O)[nH]c2)=O)CC2CCC1(NC(C1CC=CC(O)C1)=O)C2 88437,C(=O)(C1c2c[nH]nc2CN1C(=O)C#CC1(C)COC1)N(CC(C)O)CC1CC1 88438,c1(C(=O)NC2CN(C(COc3cn(C)nc3)=O)CC2F)c[nH]c2ccc(Cl)cc12 88439,O=C1CCCC(C(N2CCCC(NC(c3cnn(C4CC4)c3)=O)C2)=O)CC1 88440,CON(C)C(=O)C(C)NC1CCCCC1n1cc(Br)cn1 88441,N1(C(C(C)C2CC2)=O)CC2(CCC(CNC(=O)Cc3ccc(Cl)c(F)c3)O2)C1 88442,c1(C(N2C(CNC(CNC(C)=O)=O)C(C)CC2)=O)ccc2n[nH]c(C)c2c1Cl 88443,N1(C(CCNC(C)=O)=O)CCOC2(C1)CN(C(c1cc(C)cc(Cl)c1)=O)C2 88444,CC1CCc2[nH]c(C(N3CC(C)C(C)(C(=O)O)C3)=O)cc2C1 88445,N1(C(CC)=O)CCOCC2(COCCN2C(=O)C(O)C(C)c2ccccc2F)C1 88446,CC(C)C(C)CC(=O)NC(CC1CC1)C(=O)N(C1(c2cc[nH]n2)CC1)C 88447,c1(C(N(CCC(=O)NC2CCSC2)CC#C)=O)ccnn1C 88448,c1(C(=O)NC(CCN(C(C(C)=C2CC2)=O)C)C)ccc(C2CNC(=O)C2)cc1 88449,N1(C(C(C)NC(N)=O)=O)CC(C(=O)NCC2CCC=CCCC2)CC1(C)C 88450,CN1CCC(NC(=O)C(CN(C)C)NC(c2cncc(Cl)c2)=O)C(C#N)C1 88451,c1(N(C2CCN(C(c3ccccc3Cl)=O)C2)C)cnc(C#N)cn1 88452,C12(CNC(C(CCO)N(C)C)=O)CCC1CN(C(=O)Cc1c[nH]nc1O)C2 88453,N1(C(Cc2cc(C)cc(C)c2)=O)CCC(NC(C2CC2C)=O)CC(C)(C)C1 88454,CC(C(C)(C)C)=CC(N1CCC(NC(=O)CCCc2csc(C)n2)C1)=O 88455,CCC(CO)C(=O)NCCC1(O)CN(C(=O)C(F)(F)C2CCOCC2)C1 88456,N1(Cc2c(OC)cc(Br)cn2)CCC(F)(F)C(NC(=O)Cc2ccsc2)C1 88457,C(CCC(=O)NC1CCOCC1(C)C)(C(C)C)NC(Cn1c(C)nc(C)n1)=O 88458,c1(CC(=O)NCC2CCCC(NC(c3csnn3)=O)C2)nc([N+](=O)[O-])n[nH]1 88459,N1(C(C2(C)CCC2)=O)CCN(C(=O)CCCN=[N+]=[N-])C(CC(F)(F)F)C1 88460,c1(NC(C)C)ccc(C(N2CC(F)(CNC(C3CC3Cl)=O)C2)=O)cc1 88461,C1(N(C(=O)CCN2CCOCC2)C)CCC2CN(C(c3ccoc3Cl)=O)CC12 88462,n1(C2CC(C(N3CC(C4CCCCO4)C3)=O)C2)cc(C2CCCOC2)nn1 88463,O=C(CC1=CCCCC1)N1CCC(F)(CNC(=O)C(F)(F)C(O)C2CC2)CC1 88464,C1(CNC(C(CC=C)NC(=O)C2=C(Cl)CC2)=O)CCCC12CCC2 88465,C1(CC)(NC)CCN(C(C2CCC(CO)CC2)=O)CC1 88466,CC(O)(CNC(c1conc1CNC(C1(CO)CCOC1)=O)=O)C(F)(F)F 88467,c1(C(N2CCC(N(CCC)C(c3ccc(C)cc3)=O)C2)=O)cc(F)c(N)cc1F 88468,N1(C(C2CCC(C)C2)=O)CCN(C(=O)CC2CC2)CC1 88469,C1(C(=O)NCCCc2cn(CCC(F)(F)CO)nn2)CCC(C(F)F)CC1 88470,C1(C(N(C)Cc2scc(C)c2)=O)C2CC1N(C(=O)Cc1ncoc1C)C2 88471,c1(C(=O)NCC2(CCCNC(COC(C)C)=O)CCCC2)cc2sccc2cn1 88472,CN1CCN(C2CCCC2c2ccc(OCCCOc3ccccn3)cc2)CC1 88473,c1(C(=O)NCC2CN(C(CC)=O)CC2(F)F)ccc2c(c1)C(CC)C(=O)N2 88474,N1(C(CCN(C)CCO)=O)CCC2CN(C(C3OCCN(C)C3=O)=O)CC12 88475,C1(CC)CCCN(C(c2ccccc2F)=O)C1C(=O)NCCC(C(C)C)N(C)C 88476,c1(N2C(=O)CC(C(=O)NCC(CN(C(=O)C(C)(C)O)C)O)C2)ccc(F)c(F)c1 88477,C1(C(=O)NCC2C(NC(C3CC(OC)C3)=O)C2)COCCN1CC(F)(F)F 88478,C1(C(=O)NCCOCC2CC2)(CNC(C(C)OC2CCCC2)=O)CCCO1 88479,C(=O)(CS(=O)(=O)C1CC1)NC1C(C2CCN(C(C(F)=C(C)C)=O)CC2)OCCC1 88480,CN1C2CCC1CN(C(C1COCCN(C(C3CCCO3)=O)C1)=O)CC2 88481,c1(N(C(c2cnc(C)[nH]2)=O)CC2CC2)ccc(Cl)cc1 88482,C(=O)(C1=NOC(C)C1C)N(C)CC1(O)CN(C(Cc2nc(C)[nH]n2)=O)C1 88483,CC1(C(=O)Nc2cnccc2Cl)CCCN(C(=O)CCc2cnccn2)C1 88484,c1(C(=O)NC2CCN(C(CSCCCC)=O)CC2)ccnc2c1ccn2C 88485,N1(C(Cc2c(C)cccc2)=O)CCC2CCC12CNC(c1c(C)[nH]c(C)c1C)=O 88486,C(=O)(CS(=O)(=O)CCO)NCC1(CO)CCN(C(C(COC)O)=O)C1 88487,C(CCCC(C)NC(c1cnn(CC)n1)=O)NC(C(C)(C)OCC)=O 88488,c1(NCC(C)Cc2ccccc2F)nccc(=NCC2(CC(N)=O)CC2)[nH]1 88489,c1(C(C)OCCCCCC)nc(-c2cncnc2)nn1C(c1ccccc1)CC 88490,N1(CC(=O)NCC(N(C(CCCCC#C)=O)C)C2CC2)CCc2ccccc21 88491,C1(c2nnnn2C)(N(C(=O)C(F)CC)C(C)CCF)CCN(C2CCCCC2)CC1 88492,N(C(=NC1CCS(=O)(=O)C1)NCC1CC(C)(C)C1)C1CC(OC)C1 88493,C#CCCCCCC(=O)NCC1C2CN(C(=O)CC(C)N(C)C)CC12 88494,S(=O)(=O)(CC(=O)NC1CCCC1NC(c1nccn1C(C)C)=O)NC 88495,C1(CC(=O)N(CCCC=C)C)CCCN(C(C2CCCN2CC)=O)CC1 88496,C(=O)(C1CCCc2ncnn21)N1CC(O)CC(NC(C2(C)CCCCC2)=O)C1 88497,Cc1nn(CC(=O)NC2C3CN(C(=O)C(C)CC4CC4)CC23)c(C)c1Cl 88498,Cc1cc(CNC(=O)COC(=O)C(C)N(C)C(C2CCCC2)=O)ncn1 88499,c1(C(N2CC=CC(NC(CCOCC#C)=O)C2)=O)ccc(S(N)(=O)=O)s1 88500,N12CCCC(C1)C2.C(=O)(CC(F)F)NS(CC)(=O)=O.C1(=O)CCN1 88501,Cc1n[nH]c2cnc(C(=O)NCC(C(C)C(C)C)NC(c3nocc3Cl)=O)cc12 88502,N1(C(C(CSC)OC)=O)CC(NC(=O)CCc2cncc(O)c2)C(C2CC2)C1 88503,C1(CC)CC(C(=O)NCc2cccc(Cl)c2)CCN1C(c1ccn(C2CC2)n1)=O 88504,N(C1CCCc2cc(CNC(=O)C=Cc3ncco3)ccc21)C(CCOC)=O 88505,C1(OC)(OC)CCC1C(=O)NC(Cn1cncn1)C(=O)NCC1SCCS1 88506,C(=O)(C(=O)CCC(C)(C)C)NCC1C(C)CN(C(c2cc([N+](=O)[O-])n[nH]2)=O)CC1 88507,N1(C(C2C(OCC)C2)=O)CCN(C(c2cc(O)nc(O)n2)=O)CC1CC(F)(F)F 88508,N1(C(C(C(C)(C)C)O)=O)CCC2(CC1)CN(C(C1Cc3cccc(F)c3O1)=O)C2 88509,c1(C(N2C(C(N(CCCO)C(C)C)=O)CC2C)=O)ccc(CO)cn1 88510,C1(C(=O)NC2(CCOC)CC2)COCCC1NC(=O)CC1CSC1 88511,Nc1ccc(C(N2CCC(O)(CCNC(C3CCS(=O)(=O)N3)=O)C2)=O)c(O)c1 88512,C1(NC(CN2CCC(C)CC2)=O)CC(F)CN(C(c2cc(C(N)=O)no2)=O)C1 88513,CC(CC(F)(F)F)C(=O)Nc1ncc(C(C)(C)O)s1 88514,c1(OC)ccc(C)c2c1CCN(C(c1ccc(C)nc1N)=O)C2 88515,c1(C(=O)OCC(C2C(C)C2(F)F)=O)cc(-n2ccnc2)ncn1 88516,C1(OCC(=O)NC(C)CN(C(=O)CC2(CO)CCOCC2)C)CCC(F)(F)CC1 88517,c1(-c2nc(CC(CCC)C)n(CC(C)C3CC3)n2)ccc2ccccc2n1 88518,N1(C(=O)Cn2ccc(C3CC3)n2)CCCN(C(c2n[nH]cc2[N+](=O)[O-])=O)CC1 88519,CC1=C(C(=O)N2CCC(NC(C34CCCC3C4)=O)CC2C)C(=O)OC1(C)C 88520,c1(CC(=O)NCCCN(C(c2csc(Br)c2)=O)CC)cc(OC)no1 88521,C1(OCC)CN(C(C2(CC)CC2(F)F)=O)CC1CNC(c1ncccc1NC)=O 88522,CCC(CC(F)F)C(=O)N1CCN(C(c2cscc2SC)=O)CC1 88523,N1(C(C(C=C)C)=O)C2CCC(C(N3CC4(C)CCC4(C)C3)=O)C1CC2 88524,CC(CN(C)C)N=c1[nH]c2c(c(=NC(C)c3ncc(C(F)(F)F)[nH]3)[nH]1)CCC2 88525,n1(C(C(=O)NCCN(CC(=O)OCC)CCNC(N)=O)C)cc(Br)cn1 88526,c1(CNC(CC2(OC)CN(C(C3OCCCC3(C)C)=O)C2)=O)ccnc(F)c1F 88527,c1(CC)[nH]nc(C(=O)NCCC(C)NC(=O)C(c2ccnn2C)C)c1[N+](=O)[O-] 88528,N#CC1(C(=O)NCC2(NC(=O)Cc3ccccc3)CCC2)CCOCC1 88529,Cc1cc(CNC(c2conc2C(C2CC2)NC(C)C)=O)n(C)n1 88530,Cc1cnc2c(C(=O)N(C3CCN(C(=O)CC4CC(F)C4)C3)C)cnn2c1 88531,Cc1c(F)cc(C(N2CCCC(N(C)C(C34COCC3C4)=O)CC2)=O)c(F)c1N 88532,Cc1nc(C(N2CCC(n3cc(CNC(=O)C(F)C4CCC4)nn3)C2)=O)c(C)o1 88533,c1(CNC(c2cc(CCNC(COCC(=C)C)=O)on2)=O)ccc(O)c(F)c1 88534,c1(NC(C2C(C)C2)=O)ccc(COCC(=O)NC(C2SCCS2)C)cc1 88535,C(C(=O)OC(C)(C)C)(C(C)OC)OC(C1CCC(CSCC)C1)=O 88536,Cc1nc(CO)sc1C(=O)NCC(C)NC(c1nc(=N)cc[nH]1)=O 88537,c1(C(N(CCOCCNC(C(C(C)O)C)=O)C)=O)ccc(F)c2ccoc12 88538,Cc1nc[nH]c1CC(=O)NC(C)(CNC(c1cccnn1)=O)C1CC1 88539,C1(NC(CCC=C)=O)C=CCN(C(=O)C(C)NC(C2CCCCC2)=O)C1 88540,Cc1[nH][nH]c1C(=O)NCCCc1cn[nH]c1Br 88541,C1(O)(CN(C(C(C2CC2)SC)=O)C)CCCN(C(c2ccn(C(C)C)n2)=O)C1 88542,C=CCC(C)(C)CC(=O)NCCCCNC(c1c(C)ncnc1O)=O 88543,C1(NC(C(C=C)(C)O)=O)CN(C(c2cc3ccccc3o2)=O)C2(CCC2)C1 88544,Cc1cnc(Cl)c(S(=O)(=O)N2CCCC2CC(=O)Nc2ccnc(Cl)c2I)c1 88545,C=C(C)C1OCCC1C(=O)NC(CCNC(c1cc(C(C)(C)C)n[nH]1)=O)C(C)C 88546,c1(NCc2ccc(C(C)C)cn2)cc(Br)ccc1S(=O)(=O)N1CCOCC1C 88547,Cn1cnc2cc(C(N3CCCC(NC(=O)C4=CCCOC4)C3)=O)ccc12 88548,c1(-n2cc(C3C(C(N(c4cnn(C)c4)C)=O)C3)nn2)ccnc(F)c1 88549,C1(COC)CCN(C(c2cc(=O)cc[nH]2)=O)CC1.CCC(C)=CC(=O)NCC 88550,c1(NC(=O)COC2CCCCC2)cccc(-c2nc(O)n[nH]2)c1 88551,N1(C(CC2(OCC)CC2)=O)CCN(C(c2cn(C3CC3)nc2C)=O)CC(C)(C)C1 88552,c1(OC)cc(C(N2CCC2CNC(c2cccc3ccoc23)=O)=O)cc(N)c1N 88553,C12(C(=O)NC3CCC(NC(C4C=CCC4)=O)CC3)C3CC(CC13)C2(F)F 88554,CC1CN(C(=O)CNC(c2ccccc2)=O)CC1NC(C1(F)CC=CCC1)=O 88555,N1(C(CCOCC)=O)CCSCC1CCNC(C1CCCN1C1CC1)=O 88556,N1(C(C)=O)CC2CN(C(=O)CCn3cc(-c4ccc(C5CC5)cc4)nn3)C2C1 88557,Cc1cc(F)ccc1C(=O)NCC1CCCN1Cc1cc(I)c[nH]1 88558,C(CC(F)F)(C(=O)NC1CCCC1C#N)NC(COCCSC)=O 88559,c1(C(N2C3CCC(CNC(C4CCN(C)C4=O)=O)(C3)C2)=O)ccc2nccn2n1 88560,CC1COCCN(C(=O)CCN(C(=O)COC2(C)CCC2)C2CC2)C1 88561,N1(C(c2n(OC)cnc2C)=O)CCC2(CCOC2)C(CNC(=O)COC(C)C)C1 88562,N1(C(C(CCOC)NC(=O)CCCCNC(N)=O)=O)CCNC(=O)C1C 88563,c1(C(=O)NC2CC(CNC(C(C)C3CCC3)=O)C2)n[nH]c2ccc(Cl)cc12 88564,c1(C(=O)NCCC2N(C(CC(C)NC(N)=O)=O)CCC2)nn(C)nc1Br 88565,C(C(=O)NC1(c2cccs2)CC1)(C(C)(C)O)NC(CC(CC)SC)=O 88566,CC1(C)CCOC1CS(=O)(=O)NC(c1cnc(CN2CC(N)C2)o1)=O 88567,Cc1cccc2c1CCOC2C(=O)N(CCCOCCNC(=O)CCNC(N)=O)C 88568,C(=O)(CC(C)(C)C(=O)OCC)NC1C(NC(CCC=C)=O)CC1 88569,C=Cn1ncc(C(N2CCC(C)(C)C2CC(=O)NC2(C)CC(C)C2)=O)c1N 88570,C1(CNC(CCCC(C)=O)=O)CN(C(=O)C(C)(C)C2CCCCO2)CCC1(F)F 88571,c1(OC)coc(C(=O)NC2CC(CCNC(=O)Cn3cc(C#N)cn3)C2)cc1=O 88572,C(CC(C)(C)C)(C(=O)N1CCC(C)(C(=O)N(C)CC2(C)CCC2)C1)OC 88573,C#Cc1cccc(C(N2CC(CNC(c3cnn4ccn(C)c34)=O)C2)=O)c1F 88574,c1(C(N(CC(CN(C(=O)CCC2CCCO2)C)O)C)=O)nccc2cccnc12 88575,CCCCCC(F)C(=O)N1CC(NC(=O)CCCCCn2cnnn2)C(C)(C)C1 88576,C1(N(C(C2(C#C)CC2)=O)C)CCCN(C(c2cc(C)n(CCO)n2)=O)C1 88577,N1(C(CC)CC)CC(C(=O)N(C2CCC(CNC(=O)C(F)CC)CC2)C)CC1=O 88578,c1(C(=O)NCCC2(O)CN(C(CC3CC(=O)OC3)=O)C2)cc(C2CC2)ccn1 88579,C(=O)(CC(C)(F)F)N1C(C2(CCC(=O)NC3(C)CCC3)CC2)CCC1 88580,C1(NC(C(CC)NC(N)=O)=O)CCC2CC1CN2C(=O)COC(=O)CO 88581,N1(C(C(CC)(F)F)=O)CCc2ccccc2C(NC(c2ccncc2Cl)=O)C1 88582,C1(C)(NC(CC2C=CC(NC(c3cc(C(C)C)on3)=O)C2)=O)CC(F)(F)C1 88583,c1(C(C)=O)[nH]c2ccccc2c1C(=O)NCC1CC1F.C12CCCC1NC2=O 88584,Cc1ncnc(C(=O)NCC(CC2CC2)C(=O)NC2(c3nn[nH]n3)CC2)c1C 88585,C12(NC(C(C)C3CCCC3)=O)CCC(CNC(=O)CN3C(=O)CCC3=O)(C1)OC2 88586,C(=O)(C(O)CC(C)(C)C)NCC1C(CC)CN(C(=O)C2=COCCC2)CC1 88587,C1(C(=O)Nc2coc([Si](C)(C)C)c2)CCc2ccc(O)cc2C1.CC12CN(C1)C2 88588,N1(C(=O)NC2CC(c3ccccc3)(OC)C2)CCCc2cc(OC)ccc21 88589,CC(C(=O)NC1CC(CC(N2CCOCC23CC3)=O)C1)S(N)(=O)=O 88590,C1(C)(c2cn(CCc3ncn(C)n3)nn2)COCCN1C(=O)Cc1nc(=N)[nH][nH]1 88591,C(=O)(C1CCCc2ncnn21)N1CC(=C(CNC(c2csc(S)n2)=O)F)C1 88592,C(CC(C(C)(C)C)NC(=O)CC1CN(C(C)=O)C1)N(C(C(COC)(C)OC)=O)C 88593,N1(C(c2ccnc(F)c2Cl)=O)CC(CO)C2(CCN(C(C3CC34CC4)=O)CC2)C1 88594,c1(C(N(CCCN(C(=O)CCc2ccnc(Cl)c2)C)C)=O)cnn2ccn(C)c12 88595,C(=O)(C(C)(C)C(C)C)NCCC(N1CCC(N(C(CCCOC)=O)C)C1)=O 88596,c1(COC(CC2ON=C(CC)C2)=O)ccc2c(c1)CCCO2 88597,c1(OC)ccc2c(c1)CC(C(=O)NCC(C)(CO)NC(=O)C1=CCOC1)O2 88598,c1(N(C)C)ccc(C(=O)NC2CC(CNC(=O)CNC3CCSC3)C2(C)C)cn1 88599,C(=O)(CCC(=O)N1CC(CC(C)NC(=O)CCCC2CC2)C1)NCCC 88600,Cc1cc(C(N2CCCC2(C(=O)N(C(CO)C2CC2)C)C(C)C)=O)nc(O)c1 88601,c1(CNCC(=O)N(CC(=O)N(C)CC2(CO)COC2)C)ccccc1 88602,N1(C(C(C)=C2CCCC2)=O)CCC(O)C(NC(c2cc(=O)n(C)cn2)=O)C1 88603,CCCCC(CC(=O)N1CCC(C)CC1C)NC(=O)CC1CC2CC2C1 88604,S(=O)(=O)(c1ccc(NC2CCC(CO)C2)cc1Cl)NCCc1nc(C)sc1 88605,N12CCCC(C1)C(=O)N(CC)C(CC)C2=O.C1(F)(NC(C2CCCC2)=O)CCC1 88606,N1(C(CCCOCCC)=O)CC(C(=O)NC(CF)C(F)(F)F)C(F)(F)C1 88607,C1(C(=O)Nc2ccns2)CCN(C(c2ccc(O)c(I)c2)=O)CC1O 88608,CC1=C(C(=O)N(C)CCC2CCN(C(C3(C(=O)N(C)C)CC3)=O)CC2)SCCO1 88609,C1(C(N(C)Cc2ccc(Cl)s2)=O)C=CCN(C(C2CCCCO2)=O)C1 88610,C1(NC(COCCOC)=O)CC12CCN(C(=O)Cc1cnc(C)s1)C2 88611,C1(C)(NC(CC2C(C)CCN(C(C3CNC(=O)O3)=O)C2)=O)CC(C)(C)OC1=O 88612,C1(NC(CC(C)(C)C2CC2)=O)CCCN(C(c2ccc(Br)c(O)n2)=O)CC1 88613,Cc1cnccc1C(N1CCC(NC(=O)COC(c2nccn2C)C)C1)=O 88614,c1(C(N2C(CNC(Cc3ccc(OC)nc3)=O)CC2)=O)cc2n(n1)CC(F)C2 88615,C1(NC(c2cncnc2)=O)C(CC2CC2)CCN1C(=O)CCC1CC1 88616,C(=O)(CCC(F)(F)C(=O)N1CCN(C(C2C=C2C)=O)CC1COC)OCC 88617,Cc1cccc2c1OCC2C(=O)N1CC(CCCCNC(=O)CCOC(C)C)C1 88618,c1(CN(CC)CC)ccc(OC)c(OC(=O)Cc2ccc(OCC(C)C)cc2)c1 88619,C1(C(=O)NCCCCCCNC(C2(C)CC(C)C2)=O)Cc2ccncc2N1 88620,C(C(CC(C)C)NC(=O)CSc1ccc(C)cc1)NC(COCCCC#C)=O.O 88621,C1(C(=O)NCC(C(C)(C)C)NC(C2ON=C(CC)C2)=O)Cc2cc(C)ccc2S1 88622,N1(Cc2cnc(CCC)s2)C(C(N2CCOC3(CC3)C2)=O)CC2CCCCC12 88623,c1(NC(=O)C(CC2CCC2)OC(C(CCCOC)C)=O)cccc(C#N)c1C 88624,C(C)(C(C(=O)NCCc1cnn[nH]1)C(C)C)NC(CCCOC(C)C)=O 88625,C(CC1CCCCC1)(C(=O)NCCCCCN(C(=O)C=Cc1cscn1)C)OC 88626,N1(C(C(CCOC)(C)C)=O)CCC2CC(NC(C3(O)CCSC3)=O)CCC2C1 88627,Cc1cn2c(n1)CC(C(=O)NCC(C(C)C)NC(c1cc(C3CC3)on1)=O)CC2 88628,C1(OCC(=O)NCC2C(CC(=O)OC)C2)CCN(C(C2(C)CCOC2)=O)C1 88629,c1(C(N2CCC(C)(NC(CN(CCOC)C)=O)C2)=O)[nH]c2ccc(Cl)cc2c1Cl 88630,CCC(C(=O)NC1(C(=O)OC)CC1)NC(=O)Cc1cn(C)nn1 88631,c1(C(N(CCOCCN(C(c2cn(CC=C)nn2)=O)C)C)=O)cc[n+]([O-])cc1 88632,c1(OC)ccc(Br)c(F)c1S(=O)(=O)N1CCC(c2ccc(Br)s2)C1 88633,N1(C(C(CC(C)(C)C)NC(c2cccc(F)c2O)=O)=O)CC(C2CCCCC2)C1 88634,C(CC(=O)N1CCCCC1CCN(C)C(C1CCC(=O)O1)=O)(C(N)=O)NC(C)=O 88635,C1(CNC(C=C(COC)C)=O)CN(C(c2cccc(C#N)c2)=O)C2(CCC2)C1 88636,C1(CC)(NC(c2cc(CNC(C3CC(C)(C)C3)=O)on2)=O)CCCC1 88637,c1(C(=O)NC(CNC(CC(C)OC)=O)(C)Cn2cccn2)cccc(N)n1 88638,c1(SC)c(C(=O)NC(C(=O)NOCC(C)(C)O)C2CCOCC2)cnn1C 88639,C(=O)(C(CC=C)CC(C)C)NC1(CC=C)CCN(C(c2cccnn2)=O)CC1 88640,NS(=O)(=O)c1ccc(C(=O)NC2CN(C(=O)C(O)C(F)F)C2)cc1F 88641,CCC(C)(CNC(C1COCC(C)O1)=O)C(=O)N(C1CCN(C)C1)C 88642,c1(OC)ccc(NC(=O)CCC2CCN(C(C3CC3F)=O)CC2)cc1C 88643,N1(C(C(COC)C)=O)CCN(C(c2nc(Cl)c(Cl)s2)=O)CC(C)(F)C1 88644,Cc1cc(C(N2C3CCC2CC(C)C3)C(=O)NC2CCCCC2)nc(Cl)c1Br 88645,C#CCC(C)(C(=O)NCCC1(O)CCC1)NC(c1cc(C)sn1)=O 88646,Cc1cc(C(=O)N(C)CC2(O)CCCN(C(C3CSCC(=O)N3)=O)C2)ncc1N 88647,C1(CNC(c2c(Cl)cn(CCC)n2)=O)CN(C(C2C(C#N)C2(C)C)=O)CC12CC2 88648,c1(C(N(CC)CC2CCCN2C(C2CC(CCO)C2)=O)=O)ccc(N(C)C)cn1 88649,C(=O)(CCCC(C)(C)NC(=O)COC1CCCOC1)NCC1(CC)CCC1 88650,N1(CCNC(C(C)NC(=O)NC)=O)CCN(c2ccc(-n3cnnn3)cn2)CC1 88651,N1(C(COC2CC(C(C)C)C2)=O)CC2(CC2)C1 88652,C1(CN(CCNC(c2ncccn2)=O)C2CC2)CC12CCOC2 88653,c1(OC)cc(F)c(CC(=O)N(CC(C)NC(c2csc3nccn23)=O)C)c(Cl)c1 88654,c1(C(=O)Nc2ccc(-c3nnc(Br)o3)cc2)ccn2cccc2c1 88655,N1(CCc2cn(C(C(N3CCC(O)(CC)C3)=O)C)nn2)C(C)CCCC1C 88656,C1(C(=O)NCc2cncc(CC)c2)CC12CCN(C(=O)C(C1(O)CCCC1)F)C2 88657,C1(CNC(CN(C)C(N)=O)=O)CN(C(=O)CC2C=CCCC2)CCC1(F)F 88658,Cc1cc(N(C)C(C2C3CN(C(C4CS(=O)C4)=O)CC23)=O)cc(C)c1 88659,N1(C(COCCC)=O)CCC2(CC1)CN(C(C1COCCO1)=O)C2 88660,C1(CCNC(c2ncccc2C2CC2)=O)CCN(C(C2C3CCC(=O)C23)=O)CC1 88661,c1(C(=O)OC(C(=O)OC)C2CCCC2)cc(C(F)(F)F)nc2c1CCCC2 88662,C1(COC)(NC(c2cc(C(C)(F)F)on2)=O)CCN(C(C2CCC=CCC2)=O)C1 88663,C(=O)(CCC(F)(F)CN=[N+]=[N-])N(CCNC(C1CCc2nn[nH]c2C1)=O)CC 88664,n1(CCCSCC)nnnc1C(C(C)(C)C)NCC(C)C1CCC1 88665,c1(C(N2CCC(NC(c3ccc(O)nn3)=O)CC2)=O)cc2cc(F)ccc2o1 88666,C1(C)(N(C(C=CCN(C)CC)=O)C2CC2)CN(C(=O)CCCF)C1 88667,C(=O)(CC(C)CC(=O)N(C(C)C(=O)NCC(F)C1CCC1)C)OC 88668,c1(C(=O)NCC(C)N(C)C(c2cncc(Cl)c2Cl)=O)cccn2nncc12 88669,C1(CC(=O)NC2(CC=C)CC2)CCCC1NC(c1ccsn1)=O 88670,n1(CCNC(=O)NCC(C)CN(C)C(=O)OC(C)(C)C)cccc1C=O 88671,c1(C(N2CCC(N(C(C3(C4CC4)CC3)=O)CC)C2)=O)cccn2c(C)nnc12 88672,N1(C(CC(C(CC)C)O)=O)CC2(CCN(C(=O)CC3CC(F)C3)CC2)C1 88673,Cc1cc(CNC(=O)NC2CCC(C(=O)O)CC2)c(F)cc1Br 88674,c1(C(C(=O)NCC2CCOC2)N(CCSC)CC)ccc(OC)c(C)n1 88675,CN1CC2(CC2)CC1C(=O)NC(C(=O)NC12CC(C1)C2)C1(C)CC1 88676,S(=O)(=O)(C1CCS(=O)(=O)C1)NCC1CC(F)(CNC(=O)OC(C)(C)C)C1 88677,C(CCC(=O)NCC(O)C(=O)NCC1(SC)CC1)OCC 88678,N1(C(C=Cc2nc(C)sc2)=O)CCN(C(=O)Cc2csc3nccn23)CC(C)(F)C1 88679,C1(C(=O)Nc2n(C)nc(-c3cccs3)c2)CC(O)CCN1Cc1cnccn1 88680,N1(C(c2[nH]cc(C)n2)=O)CCCC(CCn2cc(C(C)O)nn2)CC1 88681,c1(CC)ccc(CCCNCc2nc(CO)n[nH]2)cc1 88682,N12CC(CC1(C)C)CC2=O.C(=O)(C(F)C(C)(F)F)NCC1CC(N(C)C)C1 88683,Cc1c(C(=O)N(CC(C)NC(c2ccc(C(F)F)cn2)=O)C)cnn1C(C)(C)C 88684,C1(NC(C(C(C)C)c2cnn(C)c2)=O)CN(C(c2ns[nH]c2=O)=O)CC12CC2 88685,C(=O)(CCCC(C)(C)C)N.c1(OC(CC)C)ccc(C(=O)NC2CN(C=O)C2)cc1 88686,C(=O)(C1=CCCCC1)N1C(C(N2CCC(C(C)(C)C)C2)=O)CC(OC)C1 88687,C(CC(C(=O)N1OC2CCC1C2)OC)NC(c1c(CC)cno1)=O 88688,C1(CNC(c2cccc(CC)c2)=O)CC2(CO1)CN(C(=O)C(C1CCC1)OC)C2 88689,c1(N(C)CC2COC(=O)O2)nc(N2CC3CC2C3)c2cnn(C)c2n1 88690,C1(NC(c2c(C)nn[nH]2)=O)CN(C(c2ccc(-c3ccc(Cl)cc3)[nH]2)=O)CC1C 88691,CC(C)C(CCN(C)C(c1ccn(C2CC2)n1)=O)NC(=O)CC(C)(C)O 88692,Cc1[nH]c(=N)ccc1C=CC(=O)NCCC(C)NC(C1CCCC12CC2)=O 88693,C1(CNC(C2CCC2(F)F)=O)CC2(CCN(C(c3cccc[n+]3[O-])=O)CC2)CO1 88694,C(=O)(C1=CCOC1)NC(C(C)CCC(N=C1CCCC1)c1nn[nH]n1)=O 88695,C12(NC(C=C(C)Cl)=O)CCN(C(C3(n4cnnn4)CC3)=O)CC1C2 88696,C#CCCCC(C)C(=O)N1CCN(C(c2cnoc2C)=O)CC1CS(C)(=O)=O 88697,Cn1nc(Cn2cc(CN3CCCC(F)CC3)nn2)c2c1CCC2 88698,c1(OC)ccccc1OCCC(=O)NC1(CCNC(C2COCC(C)O2)=O)CC1 88699,c1(NC(C2(F)CCN(c3ncc(OCCOC)cn3)C2)=O)nc(C)c(Br)c(Cl)n1 88700,N1(C(C2C(C)C2)=O)CCCC(N(C(=O)CCC2CCCOC2)CCO)C1 88701,c1(C(=O)NCCCS(C)=O)ccc([N+](=O)[O-])cc1C(F)(F)F 88702,C1(C(N(C)CCC2CCCCN2C(c2cncc(Cl)c2)=O)=O)CCC(C)(C)CC1 88703,n1(CC(=O)OC)cccc(NC(C2CCC(O)(C(F)(F)F)CC2)=O)c1=O 88704,c1(CC(=O)NCC2N(C(C(N3CCC(O)CC3)C)=O)CC2)cccc(F)c1F 88705,CCCC(C)(CCC)C(=O)NCCC12CCC1CN(C(C1(C)CCSCC1)=O)C2 88706,C(c1ccsc1Br)=CC(=O)NC1CCC(CNC(c2ccon2)=O)C1 88707,N1(C(c2c(CC)con2)=O)CCN(C(C)CNC(C2CCC(O)C2)=O)CC1 88708,N1(C(C(C(C)C)c2ccncc2)=O)CCN(C(c2cnc(=N)[nH]c2)=O)C2(CC2)C1 88709,C(C(C)(O)CC(=O)NC1CCCN(C(c2cc(C#N)cs2)=O)C1)OC 88710,c1(NC(Cn2c(C)cc(C)n2)=O)ccc(NC(c2cnc(CO)cn2)=O)c(F)c1 88711,C=C(C)CN=C(NCCN1CCN(C(C)=O)CC1)NCC1CCC=CO1 88712,N1(C(c2cc(OC)ncc2)=O)CCN(C(C2CC(CCO)C2)=O)C(C2CC2)C1 88713,C(=O)(CC(CC)CC(F)(F)F)N1C(CN(C(CC(=O)NCC)=O)C)COCC1 88714,N1(C(CNC(c2n(C(C)C)ccc2)=O)=O)CCN(C(=O)CN(C)C(N)=O)CC1 88715,C12(C(N3CCCC(NC(CN(S(C)(=O)=O)C)=O)C3)=O)CCCN1S(=O)(=O)CC2 88716,C12(C(N3CC(NC(CSC(C)C)=O)C(CC4CC4)C3)=O)CCCCCC1OCC2 88717,C(CC(CC)C(=O)NC1CCCN(C(c2ncccc2C(F)F)=O)C1)=CC 88718,C(C(=O)N1CCC(C2CCCN2C(=O)CC2CC2)CC1)(C(C)C)OC 88719,C1(OC)(CNC(=O)CSCc2ccccn2)CCN(C(C2(C)CC2C)=O)C1 88720,N1(C(CP(C)(C)=O)=O)CC2(CCCN(C(=O)Cc3cccc(C(F)F)c3)C2)C1 88721,C1(C(N(CC#CC)C(C)C)=O)C2CC3C(C2NC(=O)CC2CC(CC)C2)C13 88722,C1(F)(C(N2CCC(NC(c3cc(CN4CCCCC4)on3)=O)C2)=O)CC=CCC1 88723,c1(NC2CC(NC(NCc3cncc(C)c3)=S)C2)ncnc2ncc(Br)cc12 88724,N1(Cc2cc(OC)c(C)cc2)CCCC(C2CCCN(C(c3cn[nH]c3)=O)C2)C1 88725,Fc1ccc(C(c2nnnn2CCCF)NC2CCCC(F)(F)C2)c(F)c1Cl 88726,Cc1ccc(NC(C2CCCC2NCc2cc(F)c(O)c(Br)c2)=O)c(Cl)c1O 88727,CCC(CCN1CCCCC1)(c1nnnn1C1CC1)NC(C1CCOCC1)C 88728,O=C(C1=C(F)CN(C(C2CN(C3COC3)C2)=O)CC1)NCC(F)CO 88729,n1(CCCC)nccc1C(=O)NC(C1CCN(C(=O)C(O)C2CC2)C1)C 88730,N1(C(C(N2CCN(CCF)CC2)=O)=O)CCCN2CCCC12 88731,c1(C(N(C(C)CNC(C2SCCS2)=O)CC)=O)ccc(C)o1 88732,C1(C(=O)OC)CN(C(=O)Nc2nnc(C(F)(F)F)s2)CCC1C(=O)OC(C)(C)C 88733,C(C(C)(C)CC(=O)N1CCN(CC2CCC(C)(C)C2)CC1)OC.C12(CC1)C(=O)N2 88734,CC(C)(O)C(F)(F)C(=O)N1CC2(CC(C(=O)NC(CC3CC3)C3CC3)CO2)C1 88735,N1(C(c2cnn(CCC)c2Cl)=O)CCN(C(=O)C(F)n2cccn2)C(CCO)C1 88736,N1(C(C)C(=O)NCCCCNC(=O)CC(C)c2cnn(C)c2)CCC(O)CC1 88737,CCC(C)C(O)CC(=O)NCCN(C)C(c1ccn(-c2ccccc2OC)n1)=O 88738,CC1CCC(NC(=O)CCC2CC2)CN1C(c1cc(C2CC2)ccn1)=O 88739,c1(C(C(=O)NCC(n2cc(-c3cccnn3)nn2)C)(C)C)ccc(F)cc1 88740,C1(NC(Cc2nc(C)oc2)=O)CC2CCC(C1C)N2C(C1CN(S(C)(=O)=O)C1)=O 88741,Cc1ccc(CC(=O)NCC2CC3CN(C(C4CCSCC4)=O)CC23)c(Cl)n1 88742,c1(CC(C)C)ccc(C(=O)NC2CC(CCNC(c3cnc(N(C)C)s3)=O)C2)o1 88743,N1(C(c2cn(CC)nc2)=O)CC(C2CC2)(C(=O)NC(c2cccc(C)n2)C)C1 88744,Cc1cc(C)c(C=CC(=O)N(CC(C)NC(c2cnc(Cl)[nH]2)=O)C)cc1C 88745,N12CCC3(CCN(C3)N(CC)C(=O)C1)C2.C1(CCC(=O)OC)CCC(=O)N1 88746,C1(CCC)CN(C(=O)CSC(C)(C)C)CCN1C(c1ncn(C(C)C)n1)=O 88747,C1(C(N2CC(NC(c3ccc(C(C)(C)C)[nH]3)=O)C2)=O)C2CCC(F)(F)C12 88748,c1(OCCC)ccc(C(N2CCC(CN(C(=O)Cc3ccon3)C)C2)=O)cc1 88749,N1(C(c2cccc(C)n2)=O)CC2CCN(C(C3CC34CC4)=O)CCC2C1 88750,N1(C(C(N2CCOCC2)C)=O)CCCC(C)(C(N2CCC(OCC3CC3)C2)=O)C1 88751,c1(-c2cccc(C(=O)OC(CCCOC)C(=O)OC)n2)ccc(C#N)c(C)c1 88752,c1(C(=O)NC2(CNC(CCSCC(C)C)=O)CCOC2)n[nH]c2c1NCCC2 88753,C12(C(=O)NC(CNC(CNC(C)=O)=O)C3CC3)CC(C1)C(C)(C)O2 88754,CCCCC(CNC(c1scc(C)c1OC)=O)NC(C1(C)CC1(F)Cl)=O 88755,c1(CNC(=O)NC2C(c3cccc(C)c3)C2)cc(F)ncc1OC(C)(C)C 88756,Cn1ccc(CC(=O)NCCCCNC(C2CC2(C)C)=O)n1 88757,C(=O)(C(CN=[N+]=[N-])NC(c1cc(Cl)n[nH]1)=O)NCCCN(C)C 88758,O=C1Cc2c(NC(c3cc(Cl)ccn3)c3nnnn3C3CC3)cccc2N1.C1CO1 88759,CC1(C)CCCCC1CC(=O)NC1CC2CN(C(c3cc(C(N)=O)no3)=O)CC12 88760,N1(C(C2N(C(C)C)C(=O)CC2)=O)CCC(CNC(=O)C2=CCCCC2)C(F)(F)C1 88761,N1(C(CSC)=O)CCN(C(=O)CCOc2cccc3ccccc23)C(C)CC1C 88762,c1(C(=O)NC2(CNC(=O)CCc3cncc(F)c3)CC2)cc(O)cc([N+](=O)[O-])c1 88763,Cc1cc(-c2ccc(=NCc3noc(C(F)F)n3)[nH]n2)c(C)cc1CO 88764,C1(NC(CCCOCC)=O)CCN(C(C2CN(C3COC3)C2)=O)CC1F 88765,C1(OC)CN(C(c2sccc2C)=O)CC1NC(=O)CCNC(C)=O 88766,C1(C(=O)NC2CCCC(CNC(c3ccc(SC)s3)=O)C2)CCC(C)(F)CC1 88767,N1(C(C2(OC)CCCCCC2)=O)CC(C)CN(C(=O)CCCCO)C(C)C1 88768,Cc1cc(CNC(=O)C(CNC(C2(C)CCNC2=O)=O)CC2CCCC2)sc1C 88769,C(N=c1[nH]c(Cl)nc2c1SCC2)C1CN(C(C2(C(N)=O)CC2)=O)C1 88770,C(N=c1[nH]cc(C#N)c2ccsc12)N1C2(NC(=O)OC(C)(C)C)CCC1CC2 88771,C1(CNC(C)=O)(COC)CCN(C(=O)Cn2ccc(C)n2)C1 88772,O=C(C1=CCC2CCC1N2C(C1CN2CCC1C2)=O)NCc1cccc(F)n1 88773,c1(C(=O)NCCC2N(C(COCCC)=O)CCC2)ccc(Cl)c(C)c1Cl 88774,C#CC1CCN(C(C2CCN(C(c3sccc3C)=O)CC2)=O)C1 88775,c1(C(N2CCOC(CCNC(C3(F)CC=CC3)=O)C2)=O)cccc(Br)c1 88776,N1(C(C(C)C#N)=O)CCC(C)(NC(=O)CCc2ccc(NS(C)(=O)=O)cc2)C1 88777,C1(CC(=O)NCC2(NC(C(CC)=CC)=O)CCC2)CCN(CC2CC2)CC1 88778,c1(N(CC(CN(C(=O)CCOCC(F)(F)F)C)O)C)nccc(OC)n1 88779,c1(C(N2CC(CNC(c3c(C)scn3)=O)OCC2)=O)c(O)cccc1O 88780,C1(C(NOCC(=O)NCC2(O)C(C)CCC2)=O)CC2CC1CC2O 88781,Cc1cc(CNc2csc(-c3cc(O)ccc3F)n2)c(O)c(Br)c1 88782,C1(C(=O)NCc2csnn2)CC2(CCN1C(=O)CCC1CCCCC1)CC2 88783,N1(C(c2c(N)ccc(C(C)C)c2)=O)CCC2(CCC2)C(NC(c2cnsc2)=O)C1 88784,C12(NC(CCC(=O)NCC)=O)CCC(CC1NC(=O)CCn1ccnc1C)C2 88785,C=CC(CC)CC(=O)NCC1CC(OC)CN1C(C1CC1c1sccc1C)=O 88786,c1(C(C(=O)NCCN(C(C2C(C(=O)OCC)CC2)=O)C)C)ccc(Br)cc1 88787,C(=O)(CC(C)CC(=O)NC(C)(C)C(C)NC(c1cnccc1C(F)(F)F)=O)OC 88788,C12(NC(C(C)SC)=O)CCC(C(=O)NCc3ccnc(F)c3)(CC1)C2 88789,N1(C(CCC(=C)Br)=O)CC2CC1CN(C(c1ccccc1OC1CC1)=O)C2 88790,c1(C(N(CCCNC(=O)CCN(S(C)(=O)=O)C)CC)=O)cncn1C 88791,c1(COC)ccc(C(=O)NC2CCN(CCNC(=O)NC(C)=O)CC2)c(F)c1 88792,C1(CC=C)(C(=O)N(C)C(C2CCCO2)C)CN(C(=O)CCOC2COC2)C1 88793,N1(C(c2cccc(C(N)=O)c2)C(=O)NCC)CCC2(CC1)OCC(C)(C)CO2 88794,c1(C(N2CCN(Cc3c(C)ncs3)CC2C)=O)cc(=O)c2ccccc2o1 88795,CCCC(C)C(=O)NC(C)CCCNC(c1cnn(CCN(C)C)c1C)=O 88796,CC(C(C)C(=O)NCc1cnc[nH]1)NC(=O)C=Cc1cnccn1 88797,c1(C(CC(=O)OONC(CC2ON=C(C)C2)=O)C2CC2)ccc(F)cc1 88798,c1(C(=O)NCC(CNC(CNC(C(C)(C)C)=O)=O)CO)ccnc(O)c1F 88799,CC(CF)CC(=O)NC(C1CCN(C(c2[nH]nnc2-c2ccccc2)=O)CC1)C 88800,C(C#Cc1cnn(C)c1)NC(C1C(NC(C2CC(C)(CC)C2)=O)CC1)=O 88801,Cc1cc(C#N)cnc1C(N1CCOCC(NC(=O)C2=COCCO2)C1)=O 88802,C1(F)(C(N(C2CC(C)OCC2)C)=O)CCCN(C(C2COC(=O)NC2)=O)C1 88803,c1(C(=O)NCC(C)NC(C(C)SCCCC)=O)ccc([N+](=O)[O-])cc1 88804,Cc1cn(C)nc1C(N1CCCC1C1CCN(C(c2cc[n+]([O-])cc2)=O)C1)=O 88805,C1(NC(CC(C=C)c2ccccc2)=O)(CO)CCCN(C(=O)C(C)C(O)CC)C1 88806,Cc1nn(COCc2ccccc2)c(C)c1C(=O)NC1CN(C(=O)C(N)=O)CC1C 88807,CC1(C)CC(O)CN1C(=O)CC1CN(C(C2CCC(O)C2)=O)C1 88808,C(=O)(C1=CCCN(C(=O)CNC(=O)CC(C)C)C1)NC(CC=C)C(=O)OC 88809,N1(C(C(C)S(C)(=O)=O)=O)C2CCC1C(F)C(NC(c1ccn3nccc3n1)=O)C2 88810,Cc1scnc1C(=O)NCCC(C)N(C)C(C1CSCCS1)=O 88811,c1(C(N2CC(C)CC(NC(C(C)SC)=O)C2)=O)c[nH]c2nccc(Cl)c12 88812,c1(C(N2CCC(NC(Cc3c(C)con3)=O)C2)=O)nccc2c1CNC2=O 88813,N1(C(C(C)=C(CC)C)=O)CCC2CCN(C(c3ccc(Br)c(O)c3)=O)CC12 88814,CCC(C(=O)NCc1cc[nH]c1C(=O)NC(c1ccccn1)CO)NC(C)=O 88815,N1(C(=O)Nc2n(CC)nnc2)CCC2(CCN2)CC1 88816,C(N=c1cc[nH]c(=NCCC2COCC3(CCC3)O2)[nH]1)c1c(C)cc(Br)cc1 88817,C(C(C)(O)C(=O)NCC1CN(C(=O)C(F)n2cccn2)CC1C)OC 88818,C(N=c1[nH]cnc(NCCCNC(=O)OC)c1C)c1cn(CC=C)nn1 88819,c1(CC)cc(C(=O)NCC2(O)CCN(C(c3cc(C4CC4)ns3)=O)C2)c(C)nn1 88820,c1(CN2CC(C)(C)C(O)CC2)csc2ccc(F)cc12 88821,C(=O)(CCCN(C)N=O)N1CCN(CC(C)NC(Cc2cc(C)ns2)=O)CC1 88822,N1(C(COc2ccc(C(C)(C)C)cc2)=O)CCCn2nc(C#N)cc2C1 88823,N1(C(C=CC=CC)=O)CC2CCCC(NC(=O)Cn3cc(C#N)cn3)C2C1 88824,c1(C(=O)NC2CC2NC(C2CCCO2)=O)nccc2ccccc12 88825,C(=O)(C1=NOC2(CCC2)C1)NCCCOCC(=O)NCCNC(C)=O 88826,C1(C(=O)NCC2(C)CCN(C(CCc3cncc(C)c3)=O)C2)CN2CCC1CC2 88827,c1(C(N2CCC(OCCNC(c3cnc(CC)[nH]3)=O)C2)=O)nnccc1C 88828,C1(C(=O)NC2CN(C(C=C(C)C)=O)C(C)(C)C2)CN2CCN1CC2C 88829,C1(N(C(c2c(C)ocn2)=O)C)CN(C(=O)CC2CCC(C)CO2)CC12CC2 88830,C1(C(=O)OCC)(C(=O)NCC2CC(NC(C3CCCC3(F)F)=O)C2)CCOCC1 88831,N1(C(C2CC(C#C)(O)C2)=O)CCOCC(C(=O)NCCC2CCCC3CC23)C1 88832,CC(C)CC(O)C(C)C(=O)NC(C)(C)CNC(c1nnn(C(C)(C)C)n1)=O 88833,C1(NC(c2n(CC)ncc2Br)=O)CCN(C(=O)Cn2ncnn2)C(C)C1 88834,CC(C)CCC(O)C(=O)NCC1(C)CCCN1C(c1ccn(CC(C)C)n1)=O 88835,c1(CC)nc(C)c(C(=O)NCC(C)CNC(c2cnn(C3CCC3)c2C)=O)o1 88836,c1(C(N2CC(CNC(C(CCC)C)=O)C(C)C2)=O)cc(C)cc(Br)c1 88837,C12(C(=O)NCC3(CCNC(C(N4CCCC(O)C4)C)=O)CC3)CCOC(C)(C1)C2 88838,C(=O)(C(CC1CCCCC1)NC(=O)CCc1ccccc1)NCCC(=O)NC 88839,c1(OC)ccc(OCCC(=O)NC(C)CCNC(=O)C(C#N)C2CC2)cc1 88840,C1(NC(c2cnc(CCC)s2)=O)CCC(C)(CNC(c2c(C)n[nH]c2C)=O)C1 88841,c1(C(N2C3CN(C(CSc4ccc(C)cc4)=O)C(C3)C2)=O)cnc2occc2c1 88842,CCC(O)C(C)C(=O)NC(C)CCN(C(=O)CNC(c1ccccn1)=O)C 88843,CC(C(=O)N1N=Cc2ccccc2OC1)S(C)(=O)=NCC(=O)NCC(=O)O 88844,N1(C(C(C(CC)CC)C)=O)CCN(C(c2ccc(CO)o2)=O)CC2(CC2)C1 88845,C(=O)(C1(C)CCc2ccccc21)NCC1(F)CCN(C(CCC=C)=O)CC1 88846,c1(OC)ccc(F)c(C(=O)NC(C)CNC(=O)C=CC2CCOC2)c1 88847,N1(C(C2(c3c(C)cccc3C)CC2)=O)CCS(=O)CCC1C 88848,CC(C)(C(=O)NCC1CCC(NC(C2CC2C2CCCO2)=O)C1)c1ncco1 88849,CC1CC(CO)(NC(C2(F)CN(C(C3CCSC3)=O)C2)=O)C1 88850,Cc1cnn(C)c1CC(=O)N(CC(O)CNC(=O)C(CN(C)C)N(C)C)C 88851,C1(C(=O)NCC(=O)NC2CC2)CC2CCC1N(C(=O)C=Cc1cnc[nH]1)C2 88852,C1(CC(=O)NCc2cc(C(N(C3CSC3)CC#C)=O)no2)CC(O)C1(C)C 88853,C=CC1CN(C(=O)CC2CCC2(C)C)CC1NC(c1ccc(N(C)C)cc1F)=O 88854,C#Cc1cnc(C(=O)NC2CC(CCNC(=O)C=C(C3CC3)C3CC3)C2)c(C)c1 88855,Cc1c(C(=O)N(C)Cc2ccc(C#N)cc2F)sc2ccccc12 88856,c1(SC)ccc(C=CC(=O)NCCC(C)NC(C2CC(C#N)C2)=O)s1 88857,Cc1ccc(C)c(CN2CCCC2CC(=O)NC(c2ccc(C#N)cc2)C)c1 88858,CC1CC(C)(C(=O)NC2COCC2NC(=O)Cn2ccnn2)CC(C)O1 88859,c1(OC)ccc(CC(=O)N(C)CCOCCN(C(=O)C(F)C2CC2)C)c(C)c1 88860,CC(C)C(O)C(C)C(=O)N1CC2C(C(=O)N(C)Cc3nnnn3C)C2C1 88861,C1(C(=O)NCC23CC(NC(CN4CCC(C)(C)C4)=O)(C2)C3)CC12CCCOC2 88862,C1(NC(=O)CCOC2CCC2)CCC2(CC1)CC2NC(c1cc(C2CC2)ns1)=O 88863,NC(=O)CC(C(=O)NCC1C=CCCC1)NC(C1CC(C2CC2)C1)=O 88864,CC1=C(C(=O)NCCC(C)NC(=O)CCC2=CCCCC2)S(=O)(=O)CCO1 88865,C1(CNC(CCCSC)=O)CC2CCC1N(C(=O)C(C)C(C)n1cccn1)C2 88866,CCC(C)C(O)CC(=O)NCC1CCCC1C(=O)NCC12CCC(CC1)CC2 88867,c1(NC(C(COCC)NC(C2CCCCC2O)=O)=O)cc(C)cc(C#N)c1 88868,CCCCCCCCC(C)CC(=O)N1CC(NC(=O)CS(=O)(=O)C2CC2)C(O)C1 88869,C1(C(N2CC(NC(CCSC)=O)C(CO)CC2)=O)C(C)(C)CCCC1(C)C 88870,C1(NC(C(CC)(C)COC)=O)CCCC2CN(C(C3CN4CCC3CC4)=O)CC12 88871,n1(CC(=O)NC(CCC)CNC(c2ccnc(CC)c2)=O)cc([N+](=O)[O-])cn1 88872,N1(C(Cc2cn(CC)nc2)=O)CCC(NC(c2nc(C)nn2C)=O)C12CCC2 88873,C1(n2cc(C3(NC(C)=O)CCC3)nn2)CCN(CCC2CCCC2C)CC1 88874,c1(C(=O)NCCN(C(c2c(CC)onc2C(F)(F)F)=O)C)cc(C)cnc1N 88875,C(C(=O)N1CCC(O)(CNC(C2(c3ccccc3Cl)CCC2)=O)C1)(C(C)C)OC 88876,c1(CC(=O)NC2C(NC(CC(C=C)C)=O)COC2)ccc(Cl)c(Cl)c1 88877,c1(C(N2CC(CNC(C(CC#C)(C)C)=O)OCC2)=O)ccc2cc(C)ccc2n1 88878,c1(C(=O)NC2CCC(Nc3ncncc3Br)C2)ccc(C(F)(F)F)c(I)c1 88879,N1(C(c2ccn(C(CC)CC)n2)=O)CCC(C)(C)C1CNC(=O)Cc1ccncc1 88880,C1(NC(c2onc(C)c2C(F)(F)F)=O)CC(C)CN(C(=O)CCNC(=O)CO)C1 88881,N1(C(CCN(C)CC)=O)CCOC2(CCN(C(=O)C(C(C)C)n3ccnc3)C2)C1 88882,c1(COC)nc(NCC2C(C)CCCN2C(=O)C=CC(C)(C)SC)cc(O)n1 88883,CCC(F)(F)C(C)(C)C(=O)NC1CCC(CNC(c2cc(Cl)c[nH]2)=O)C1 88884,C1(C(=O)OC)CCCC1(C)NC(=O)C(F)CC1CN(C(=O)CC(C)(C)OC)C1 88885,c1(C(N2CCC(NC(CC(C(C)C)C)=O)(CO)CC2)=O)cnn2c1CC(F)(F)C2 88886,C1(NC(CCC(C)O)=O)CCN(C(=O)CCCNC(N)=O)C(C)C1 88887,c1(C(N2CC(NC(C3CC=CCC3)=O)C(F)(F)C2)=O)cc(F)cc(F)c1F 88888,C1(CC(=O)N(CC(C)CNC(=O)CC2CCCC2C)C)Cc2ccccc2N1 88889,C(C(=O)N=S(=O)(c1ccccc1)c1cccc(Br)c1)C1CCC(C)CC1 88890,c1(C(N2CCCC(F)(CNC(C(C)(C)F)=O)C2)=O)cn2cccc(Br)c2n1 88891,C1(NC(C(N2CC3OCC(OC)C3C2)=O)=O)C2CC3CC1CC(O)(C3)C2 88892,C1(CN(C)C(C2CC(CF)C2)=O)CCCCN1C(C12CCC(C1)C2)=O 88893,N1(C(c2c(C)ncnc2)=O)CCC(C(F)(F)F)C(CNC(=O)CC2CCCO2)C1 88894,Cc1cnc2cccc(C(=O)NCC3CCN3C(=O)C=Cc3cc[nH]c3)n12 88895,C1(C(=O)NCCC(COC)OC)CN(C(=O)CC2CC=CC2)C(C)(C)C1 88896,Cc1csc(=NCC(=O)NCC2COCC2NC(c2c[nH]cc2C(C)(C)C)=O)[nH]1 88897,CCCC(CC)CC(=O)NCCC(O)CNC(c1cc(C)cc(C)c1C)=O 88898,C1(NC(C2C(C(=O)OCC)C2)=O)CCN(C(=O)Cc2cnn(C)c2C)C12CCC2 88899,C(=O)(C1=CCCC1P(C)(C)=O)NC1(C)CN(C(c2ncncc2Cl)=O)C1 88900,N1(C(COCC#C)=O)CCC2(CCC2)C(NC(=O)C(C)CC(C)(C)C)C1 88901,C(CCS(=O)(=O)c1ccc(F)cc1)N1c2c(cc(F)cc2)CC(CCC(=O)O)C1 88902,N1(C(C(CC)F)=O)CCC(O)(CN(C)C(C2CCCCN2C(=O)C(C)C)=O)CC1 88903,Cc1cc(C(N2CCC(C)N(C(C3SCCC3C)=O)CC2)=O)c(C)cc1Br 88904,C(C(F)(C(=O)NCC1(C#N)CC1)C(C)C)NC(c1c(C)scn1)=O 88905,C(=O)(C1=NOC(C)(C)C1)N1CC(OC)C(NC(c2cnc3n2CCC3)=O)C1 88906,CN1CC(O)CC1C(N1CCC(CCNC(=O)CSc2cccc[n+]2[O-])C1)=O 88907,C(CO)(CCCCNC(=O)CCN1C(=O)CCC1=O)NC(C(C)(C)C1CC1)=O 88908,c1(NC(C(C)C(=O)NCC(=O)OC(C)(C)C)C)cccc2cncn12 88909,c1(OC)cccc(Cl)c1CNC(=O)C(=O)NCC(c1ccc(Cl)c(Cl)c1)N(C)C 88910,Cc1c(C(N2CCSCC2C(=O)NCCc2ccncn2)=O)oc2ccccc12 88911,c1(C(=O)NC2C(C)CN(C(c3ncc(F)cn3)=O)CC2)cccc2c1ncn2C 88912,N1(C(C2COCCN(C(c3ccns3)=O)C2)=O)Cc2ccncc2C1 88913,c1(C(=O)NCC23CC(CN2C(C2CCCCS2)=O)C3)cc2occc2s1 88914,C(CNC(=O)C=CC(F)(F)F)(C(C)C(C)C)NC(C(c1cc(C)sc1)(F)F)=O 88915,N1(CCCC(=O)NCCNC(c2c(C(C)(C)C)con2)=O)C(=O)CNC1=O 88916,N1(C(c2c(CC)cns2)=O)CC(C(=O)NCC2CC23CCOCC3)CC(C)C1 88917,N1(c2nc(N3CCC4CCC(C3)S4)cc(C)n2)CC2CC3CC(C2)CC1C3 88918,Cc1coc(NC(=O)C(N2CCC(C)C(CCn3ccnc3)C2)=O)c1C#N 88919,N1(C(CCCOCCC)=O)CC2(CCC2NC(c2ccc(F)cc2CC)=O)C1 88920,CC(CN=c1ncc2ccccc2[nH]1)C1CCN(C(=O)C2=CC3CCCC23)CC1 88921,c1(C(N2CC(OC)C(F)C2)=O)cnc2c(-c3ccc(I)cc3)cnn2c1 88922,c1(C(N(CC(C)O)CCNC(=O)Cc2cc[nH]n2)=O)cccc2c1OCC(=O)N2 88923,C1(CNC(C(C2CCCCC2)OC)=O)CN(C(C2C=CC=CC=C2)=O)CCN1C 88924,C1(N(C(CC(C)NC(N)=O)=O)C)CCCCN(C(=O)COCP(C)(C)=O)C1 88925,c1(CNC2C(C(N(C3CCOCC3)CC)=O)CCC2)ccc2ccc(Cl)cc2n1 88926,C1(N(C(Cc2c(C)cccn2)=O)C)CN(C(C2CC3CCC2CC3)=O)CCC1C 88927,N1(C(c2cc(OC)ns2)=O)CCCC(N(C(=O)CN2CCC2C)CCF)C1 88928,C1(C)(OC)CC(NC(c2ccc(CNC(=O)C(C)SC)nc2)=O)C1(C)C 88929,C(C(CO)C(C)(C)C)NC(CC1N(C(C2CC(N(C)C)C2)=O)CC1)=O 88930,c1(N(C(C2CCC(C(C)C)C2)=O)CC2CCN(C)CC2)ccc(F)c(F)c1 88931,C=C=CCCN=c1[nH]c(N2CCC(C)(CN(C)C)C2)nc2c1COCC2 88932,C1(CC(=O)NCCC2(C(N3CC(O)(c4cc[nH]n4)C3)=O)CCCC2)COCC1O 88933,N1(C(C(C2CCOCC2)C)=O)CC2CCC1C(NC(=O)CCCCF)C2 88934,C(=O)(C(F)CC(C)(C)NC(=O)CC#N)NC(C(C(C)C)O)C 88935,c1(C(=O)NC2CC(NC(C(COC)(C)C)=O)C2)cc(OC(F)F)cc(F)c1 88936,N1(C(CC(C)N(C(c2cncc(C)c2)=O)C)=O)CC(C(C)C)CCC1C 88937,C(CN=c1[nH]c(=NCC2(F)CCC2)c2[nH]ccc2[nH]1)NC(=O)NCC(C)C 88938,C1(CCOC)(NC(COCC(=C)C)=O)CCN(C(=O)C(CCSC)NC=O)C1 88939,C1(CNC(C2COC2)=O)C2CN(C(C3CC=CCC3)=O)CC12 88940,Cn1ncc2c(N3CC4CC3CN4c3ncncc3F)ncnc12 88941,C(C)(CC(C)(C)C#N)(c1n(C)nnn1)NC(C)CCCCCCO 88942,c1(C(=O)NCCCCC(C)NC(CCCC#CC)=O)c[nH]c2cccc(C)c12 88943,c1(-n2cc(CCSCC)nn2)cccc(CO)c1.N1(C=O)CCOC(CC(=O)OC)C1 88944,C(c1ccccc1)=CC(=O)N(CCCCN(C(CC1(C(=O)OC)CC1)=O)C)C 88945,C1(C(N2C(CNC(CCC(C)(C)F)=O)CC(C)(C)C2)=O)CCCC12OCCO2 88946,Cc1nc2cc(NC(C3CC(O)CN3C(c3ccn(C)c3)=O)=O)ccc2s1 88947,c1(C(C)(F)F)ccccc1C(=O)NC1CC(C)(NC(c2cscn2)=O)C1 88948,n1(COC)nccc1C(=O)NC(C)CC(C)NC(=O)CC1CCCC1 88949,Cc1n[nH]c(C)c1C(C)NC(=O)C(CNC(=O)OC(C)(C)C)CC1CCCCC1 88950,CC1CCc2[nH]nc(C(=O)NC(C3CCCN3C(c3cc(O)n(C)n3)=O)C)c2C1 88951,C12(NC(C3N(C)CCCC3)=O)CCC(C(=O)NCC3CCC(O)CC3)(CC1)C2 88952,C1(C(=O)OCCCNC(CCC)=O)CC12CCOC2 88953,N1(C(C2(C#N)CCCC2)=O)CCC2CCN(C(C3(CO)CC(F)(F)C3)=O)CC2C1 88954,c1(C(N2C3(CNC(C4CC(=C)C4)=O)CCC2CC3)=O)cn2ccccc2n1 88955,N1(C(c2ccc(C)nc2)C(=O)NCC)CCc2cccc(OC)c21 88956,C1(C(N(C)CCc2nccs2)=O)CCCN1C(=O)C=Cc1ccc[nH]1 88957,N1(N(S(C)(=O)=O)C)CCCC1NCC.c12cn(nn1)C2.C1CC1 88958,C1(C#N)(C(=O)NCCCCCCN(C(=O)CCCC(C)(C)C)C)CC2CCC1C2 88959,C(=O)(C1=NOC2COCC12)NC1C(C(=O)NC(C(C)F)C)COC1 88960,C(CN=c1[nH]ccnc1F)(C1CC1)NC(c1cn(C(C)(C)C)nc1)=O 88961,CC1CN(Cc2cn(C3COCC3NC(C3CCCC3(C)C)=O)nn2)CC(C)O1 88962,N1(C(CC2CC(=C)C2)=O)CCN(C(C2(C)CC3CCC2C3)=O)CC(O)C1 88963,N1(C(C2(OC)CS(=O)(=O)C2)=O)CCCCC(CNC(c2cc[nH]n2)=O)C1 88964,C1(NC(=O)C(=O)N(Cc2ccccc2)CC2CCOC2)CNC2(CCC2)C1 88965,c1(C(=O)NCc2cn(C3CCN(C(=O)C(F)F)CC3)nn2)c(F)cccc1Cl 88966,C1(NC(C(COC)OC)=O)C(C)(C)C(NC(=O)C2=COCCC2)C1(C)C 88967,Cc1cccc(C(N2CCN(C(=O)C=C(Cl)Cl)C(CC(F)F)C2)=O)c1F 88968,c1(OC)ccc(F)c(Cn2nnnc2N(C2(C#N)CCOCC2)C)c1 88969,C(=O)(C=C1SCC(=O)N1C)NC1(CNC(c2ccc(C#C)cc2OC)=O)CCC1 88970,CC1(C)C(NC(C2CCCN2C(c2ccco2)=O)=O)CC1N=c1[nH]nco1 88971,N1(C(CC(C)c2ccco2)=O)CCC2(CCC2)C(NC(=O)C(=O)NCC(F)F)C1 88972,C(C(=O)N=c1ccn(C)[nH]1)C1(C)N(C(C(CCCC)CC)=O)CC1 88973,C1(C(N(C2(C(=O)NC(CC3CCC3)CO)CC2)C)=O)CC(F)CN1C 88974,c1(C(=O)NCC(CC)(CC)NC(CC(CCC)O)=O)cc2cccnc2cc1F 88975,Cc1cc(Cl)ccc1CNC(=O)NCC12CCCC1CCN2C(=O)OC(C)(C)C 88976,c1(NC2CC=CC(NC(=O)OC(C)(C)C)C2)cc(Br)cnc1Br 88977,N1(C(c2cnc(CCC)s2)=O)CC(NC(C2CC2[N+](=O)[O-])=O)CC12CCCC2 88978,CC1(F)CN(C(=O)CCNC(C2CCCOC2)=O)CCN(C(=O)CNC(N)=O)C1 88979,CCC(CCCC(=O)NCc1ncsc1C)NC(C1CCCCC1O)=O 88980,N1(C(C2CCCC23CC3)=O)CC2(CCN(CCOc3ccccc3F)C2)C1 88981,CC1ON=C(C(=O)N(C)CCC2CCN(C(=O)CCc3ccnn3C)CC2)C1C 88982,Cc1nc2cccnn2c1C(N1CC(N(C(=O)C(N2CCC(O)CC2)C)C)C1)=O 88983,CC1(C)CN(C(C2CC3(CCC3)C2)=O)CCN(C(C2CC2(F)Cl)=O)C1 88984,C=C=C(C)CC(=O)NC(CNC(c1ccccc1Oc1ccncc1)=O)C(C)C 88985,c1(CN(C(c2c(C)noc2)C(=O)NC2CCCC2)C)cncc2ccccc12 88986,C(=O)(C#CC1CCCCC1)N1CCC2(CC(NC(CCCCCC=C)=O)C2)C1 88987,C(CC(C(=O)NCCCNC(=O)C(F)OC(F)(F)F)OC)OC 88988,N1(C(C2CCCC(OC)C2)=O)CCCC2(C1)CN(C(=O)C(F)(F)c1cscn1)C2 88989,C1(NC(c2c[nH]nc2C(F)F)=O)CC12CCN(C(=O)C1=COCC1)C2 88990,c1(C(=O)NC(CNC(CCc2onc(C)n2)=O)C(C)(C)C)cc(C#N)ccc1N 88991,CCC(CC)C(=O)N1CCOC(C(=O)NC2CC(O)C(O)C2)C1 88992,N1(C(C(N2CC(C=CC)C2)=O)=O)CC(C)CC(C)C1 88993,CCC(C)C=CCOC(C1CC(Br)C1)=O 88994,C1(CNC(C(C=C)O)=O)COCCN(C(C2CCN(c3cccnc3)CC2)=O)C1 88995,c1(C(N2CCC(CNC(C3C(C)(C(C)C)C3)=O)C2)=O)cnn(C)c1Cl 88996,C1(NC(C2(N=[N+]=[N-])CC2)=O)C2CC(CN(C(C3CCC3)=O)C2)C1CO 88997,Cc1ccc(O)cc1C(N1CCCCCC1C(=O)NCC(c1cn(C)cn1)O)=O 88998,c1(CNC(N(C(C2CCCO2)C)C)=O)ccc2nccnc2c1 88999,C1(CN(C(C2C(C=C)C2)=O)C)CCCN(C(=O)C(C)(Cl)Cl)C1 89000,c1(C(=O)NC2CCN(C(=O)NC3(CC(=O)OC)CC3)C2)ccnc(C)n1 89001,C1(C(C2CCCC2)CNC(C2(C=C)CC2)=O)CCN(C(c2cc(CO)[nH]n2)=O)CC1 89002,N1(Cc2c(OCC)cccc2)CCC2(C=CCOC2)CC1 89003,C1(C(=O)NC(c2csnn2)C)N(C(=O)C2=CCCC2)CCC1(C)C 89004,N1(C(C(F)=CC)=O)CC2(CCC(NC(=O)CCOCC(F)(F)C(F)(F)F)CC2)C1 89005,c1(NC(C2C(NC(C=CC)=O)C2)=O)cc(Br)ccc1F 89006,c1(C(N2CC(CNC(CNC(CC)=O)=O)C3C2C3)=O)ccc(F)c(OC)c1F 89007,Cc1nn(C)cc1NC(C1(NC(c2c[nH]c(C#N)c2)=O)CCSC1)=O 89008,c1(COCCNC(C)=O)ncc[nH]1.C(C(=O)NCC(C)C)OCC1(C(N)=O)CC1 89009,N1(C(c2n(C)c(O)nc2)=O)CCCC1C1CCCN1C(=O)Cn1nnnc1N 89010,C(C(C)C)(C(O)C(=O)N1CC(C)(C(=O)NCCC2CCCC(C)C2)C1)OC 89011,C1(CC)CN(C(=O)C=Cc2ccnn2C)CCN1C(=O)CC(C)N1CCCC1=O 89012,c1(C(=O)OCC(=O)N(C2C=CCCC2)C2CCNC2)ccccc1 89013,c1(C(=O)NCC(CNC(c2ccc(C)nc2)=O)C)cc(Cl)ccc1O 89014,CC1CCC(C(=O)NCCC(C)(C)O)CN1C(=O)CC1CCC(=O)C1 89015,C(=O)(C1=C(Cl)CCCC1)N1C(C(=O)NC2CC(CO)C2)(COC)C=CC1 89016,c1(-c2nc(C3CCCN(C(=O)Nc4nnc(CC)s4)C3)on2)ccc(C)c(C)c1 89017,c1(OCCC(=O)NC2C(NC(=O)C=CCn3cncn3)C2)ccccc1F 89018,C(=O)(C1=CCC(F)(F)CC1)NCC1(O)CN(C(c2cncc(N)c2)=O)C1 89019,c1(-c2cn(C3C=CC(C(=O)NCC4C(SC)C4(F)F)C3)nn2)cnn2c1CCC2 89020,O=C(CC1=CCCC1)NCc1cn(C2CCCN(C(C3CCCCS3)=O)C2)nn1 89021,C12(NC(CSC)=O)CCCC1N(C(=O)COc1ccc([N+](=O)[O-])cc1)CCC2 89022,Cc1ncccc1CCC(N1CCCC(NC(c2ccncc2Cl)=O)C1)=O 89023,C(=O)(NNc1ccc(Br)cc1)c1cc(CCC)nc(O)c1 89024,c1(OC)cnncc1C(=O)NCC(O)C(=O)NCc1cccc(OC)n1 89025,c1(C(c2n(C(CC)C)nnn2)NCCS(=O)(=O)N(C)C)cc(F)ccc1Cl 89026,c1(C(=O)NC)ccc(C(=O)NCCCCC(C)NC(=O)CCn2ccnn2)cn1 89027,C(=O)(N1CCC(C(=O)NCCCn2cnnn2)O1)c1cc(OCC)no1 89028,C1(C2CCC2)(C(=O)OC)CCN(C(=O)Nc2ccccc2F)C1 89029,c1(C(=O)NC2CCC(F)(CNC(C(CC)(C)C#N)=O)C2)cc(F)cc2nn[nH]c12 89030,C1(C(N2CCC(CCCC)C2)=O)CCN(C(=O)CCCCC(C)=O)CC1(C)C 89031,Cc1cc(O)c(C(N2CCC(NC(c3ccc(CO)cc3)=O)C(O)C2)=O)nn1 89032,N(C1CCOc2ncccc21)C(=O)C(C1(O)CCCC1)F 89033,C1(CC)(NC(=O)CC(C)C(C)C)CCCN(C(c2csc(Br)c2C)=O)C1 89034,Cc1cc(C(=O)NCC(C)NC(=O)CC(C)(C)CN(C)C)cc(O)n1 89035,c1(C(N(C)CC2CN(C(C3CC3C#N)=O)C2)=O)ccc(SC2CC2)cc1 89036,CC1CC(N2CCOCC2)CN1C(=O)C(=O)Nc1ccc(-c2ccccc2)cc1 89037,Cc1ccccc1COCCN(C(=O)C(N1CCCC(n2ncnn2)C1)=O)C 89038,C(=O)(C#CC1CCOCC1)N1CCC(NC(c2cnc(OC)nc2C)=O)(CF)C1 89039,C1(NC(C(CCC)CC)=O)CCN(C(c2cc(CC(C)C)[nH]n2)=O)CCC1(F)F 89040,c1(-n2cc(C(C)NC3CCOC3)nn2)ccccc1C(=O)OCCSC(C)(C)C 89041,CC(C)(C)CCC(F)C(=O)NC1CCCC(NC(c2ccc(N)c(Cl)n2)=O)C1 89042,C12(C(=O)NCC3(F)CN(C(c4ccc(C)cc4C)=O)C3)CCCN(CCC1)C2 89043,c1(C(=O)NC2CC(CNC(C(C)NC(c3ccoc3)=O)=O)C2)cccnc1O 89044,CC(O)C(C(=O)NC(CNC(=O)Cc1ccccc1SC(C)C)C1CC1)N(C)C 89045,C1(C(N(CC(COC)(F)F)C)=O)CCN(C(C2CCC2C#N)=O)C(C)(C)C1 89046,C1(NC(C2C(NC(=O)OC)C2(C)C)=O)(CO)CCN(C(C2CC(C)CCO2)=O)C1 89047,C(=O)(CC(CC)C(=O)OC(C)(C)C)N1CCC(N(C(c2c[nH]nc2C)=O)CC)C1 89048,C(C1CCC1)=CC(=O)NCC=CC(=O)N(C(C)CC1CC1)C 89049,CP(C)(=O)C1(C(=O)NC2CCCCC2NC(C23CCN(CC2)C3)=O)CC1 89050,C1(NC(=O)Cc2cc[nH]n2)CC2(CNC(=O)C(O)C(F)(F)F)CC1CO2 89051,c1(CS(=O)(=O)NCC2CCN(C)C2c2ccccc2)ccc(Cl)c(Cl)c1Cl 89052,c1(C(N2CCC(N(C)C(C3CC(F)C3)=O)C2)=O)ccc2nn(C)cc2c1 89053,C1(NC(c2cc(C)ns2)=O)CCCC(Nc2cccc(COCC(F)(F)F)c2)C1 89054,CCC(C)C(C)C(=O)NCC1(F)CC(CNC(c2c(Br)c(C)nn2C)=O)C1 89055,C(=O)(CCC(=O)N1CCCCC1CCNC(C1CCC(C(N)=O)C1)=O)NC 89056,N1(C(C2CN(c3c(C)cccc3)C(=O)C2)=O)CCC2(CCOCC2)C1 89057,CCCC(C)N=c1[nH]c(=NC2CC(N3CCOCC3)C2)c2sccc2[nH]1 89058,C1(NC(C2CCN(CCC)CC2)=O)COCCN(C(c2cc(C3CC3)on2)=O)C1 89059,c1(OCCNC(c2n(C(CC)C)nnn2)c2cccn2C)cccc(C)c1C 89060,C(=O)(C(C)CC(C)CC)NC1(C(N(CCCO)CC#C)=O)CCCCC1 89061,CC#CCCCC(=O)N(C(CC(F)F)C(=O)N1CCC(C(C)CO)CC1)C 89062,C(CCC(CO)NC(C1CC1C1CCCO1)=O)NC(CCC=CC(C)C)=O 89063,CC(C)CCN=C(NCCS(=O)(=O)CC1CCC1)N1CC2C(=O)NC(=O)C2C1 89064,Cc1cc(C)n2cnc(C(N3CC(N(C(=O)Cc4cccc(F)c4)C)C3)=O)c2n1 89065,O=C(CCCC#Cc1ccccc1)NCC1CCN(C(c2sc(F)cc2Cl)=O)C1 89066,CC1CCN(C(=O)C(CC(F)F)NC(C2CC3CC(=O)C2O3)=O)CC1(F)F 89067,Cc1c(C(=O)NC(C)CCCNC(=O)CC2(C)OCCO2)sc(Cl)c1Cl 89068,C(=O)(Nn1ccccc1=O)C1(C(=O)CC2CC3(CC(=O)C3)C2)CCCCO1 89069,Cc1scc(C(N2CC(NC(=O)CCCn3c(O)nnc3O)C(C)C2)=O)c1N 89070,N1(C(C=NOC)=O)CCC2C(CCCN2C(=O)CCc2nc3ccccc3[nH]2)C1 89071,c1(C(=O)NC2(C)CCN(C(=O)Cc3ccsc3Cl)C2)ccnc2ccccc12 89072,C1(CNC(c2nc(COC)sc2)=O)CN(C(c2ccc(CC3CC3)s2)=O)CC1O 89073,CC1=CCCN(C(=O)COc2ccc(N3CCCCC3=O)cc2)C1 89074,C1(n2cc(N(CCN(C(C)(C)C)C(C)=O)C)nn2)CN(C(=O)CC2(C)CC2)CC1C 89075,C(=O)(C1=COCCO1)N(CCN(C(C1(CC)CCC1)=O)C)C(C)C 89076,n1(CCCCNC(C(=O)NCCC(N2CCOCC2)C)=O)cc(Br)cn1 89077,C(C(C)(C)C(=O)NCC1(F)CC(NC(c2[nH]nnc2C2CC2)=O)C1)N(C)C 89078,CC(C)CC(C)(C)C(=O)NCC1CCCN1C(C12CC(CO1)C2)=O 89079,c1(N2CCC(C(C)NC(=O)CSCc3ccc(F)cc3)C2)nc(C)nc(C)c1F 89080,C(=O)(CCC(C)(C)c1ccccc1)NC(C(C)C)C(C)NC(=O)Cc1cn[nH]c1 89081,C(C)(N=c1[nH]c(N2CCOC(C(N)=O)C2)nc(=N)[nH]1)c1scc(C)n1 89082,c1(OC)cccc(C(C2CC2)NC(N2CCC(N3CCCC3=O)C2)=O)c1Cl 89083,C(=O)(C(COC)CC(C)C)N(CCC)CCNC(C1CCCCC1(F)F)=O 89084,C(c1ccc(OCCF)cc1)=CC(=O)NCC(C1CC1)NC(C12CCC1CC2)=O 89085,c1(C(N2CCC(CNC(c3n[nH]c4ncccc34)=O)C2)=O)c(F)ccc(O)c1F 89086,C12(CNC(C3(NC(c4c(C)cns4)=O)CCCC3)=O)CCCCC1C2 89087,C1(C(N2CCCC(C)(N(C)C)C2)=O)(NC(c2c(C)con2)=O)CCC(C)(C)C1 89088,C1(NC(c2csc3nccn23)=O)CCOC12CCN(C(C1CCC3CC13)=O)CC2 89089,c1(CCNC(N(CC(C)(C)C)C2CCCC2)=O)nc(C(F)(F)F)cs1 89090,C(CCC(=O)NC(C1CN(C(C2CNC(=O)O2)=O)C1)CO)OC(C)(C)C 89091,Fc1cc(N(C(CCC2CCCO2)c2nn[nH]n2)C2CC2)cc(C(F)(F)F)c1 89092,C(=O)(C1CCCn2ncnc21)N1CCN(C(CNC(CC2(C)CCC2)=O)=O)CC1 89093,c1(C2C(CC(=O)NCCCN(C(c3cnsc3)=O)CC)C2)cccc(F)c1 89094,N1(Cc2[nH]ccc(=O)c2)CCCN(CC(O)Cc2cccc(Cl)c2)CC1 89095,Cc1c(C(=O)NCC2CCC(NC(c3ncoc3Br)=O)C2)cnn1C 89096,c1(C(=O)NCC2C(CNC(c3c(C(C)C)ncs3)=O)C2)cc(=N)[nH]c(Cl)n1 89097,CN1C2CCC1CC(C(=O)NCC1CCCN(C(C3CCC(C)(F)CC3)=O)C1)C2 89098,C1(CNC(C(c2ccc(Br)s2)N(CCN(C(C)=O)C)C)=O)CCOCC1 89099,N1(C(C(F)=CC)=O)CC2CCC2(CNC(c2cc(Cl)c(Br)[nH]2)=O)C1 89100,c1(OCC(=O)NCCCCC(C)NC(C2CC(CCC)C2)=O)ccc(C)cc1F 89101,N1(C(CN(C(c2cccc(OC)n2)=O)CCO)=O)CCC(O)C(C)(C)C1 89102,N1(C(C)=O)CC2(NCC(c3ccc(OC)c(OC)c3)C)CCCC1C2 89103,c1(C(N2C3C(CNC(C4CC(C)=C(C)CC4)=O)C(C3)C2)=O)c(C)nc2sccn12 89104,c1(C(=O)NC(C(C)NC(=O)CC(=O)NCC2CC2)(C)C)cc(O)nc(Cl)c1 89105,n1(CCC(=O)N(C2CCC(NC(=O)CC(O)C3CC3)CC2)C)ccccc1=O 89106,N1(C(c2ccc(CC)s2)=O)CCOCC1CC1N(Cc2nnsc2Cl)CCCC1 89107,N1(C(COCCOC)=O)CCCN(C(=O)CN2CCC(F)(F)C2)C(C)C1 89108,c1(C(N2CCC(O)(C(=O)NC(CCCOC)CO)CC2)=O)cc2cccnc2[nH]1 89109,Cc1cccn(CC(=O)NCC(C(C)C(C)C)NC(C2(CF)CC(=O)C2)=O)c1=O 89110,C1(C(=O)O)CCN(C2CCN(C(C3CCCN(C(c4ccco4)=O)C3)=O)C2)CC1 89111,C1(C(=O)NCC2(OCC)CC2)COC2(C1)CN(C(=O)C(C)N(C)C)C2 89112,C1(C(=O)NCCCC#C)C2CCC(C2)C1NC(C1(CO)CCOCC1)=O 89113,C1(NC(C=CCC)=O)CN(C(c2cc(OCC)no2)=O)C(C)(COC)C1 89114,CC1(C)CN(C(=O)C=Cc2ccc([N+](=O)[O-])s2)CCN(C(C2(C)CC2(F)F)=O)C1 89115,C(=O)(Nn1cnnc1)C1C(C)(C)C1N(C(=O)CC12CCCC1C2)CCO 89116,N1(C(c2nc(COC)oc2)=O)CCCCC1CN(C(=O)CC1(C)CCCO1)C 89117,c1(CNC(=O)Nc2cnc(C(=O)OC(C)(C)C)nc2)cc2n(n1)CC(OC)CO2 89118,C1(c2ccc(Br)cc2)(NC(C2CCS2)=O)CCCCC1 89119,Cc1cc(C(=O)NC2CC(O)CN(C(c3cc(C(N)=O)co3)=O)C2)ncc1F 89120,Cc1cc(C)c(C(=O)N(C)CC2CN(C(c3cn(C)[nH]c3=N)=O)CCO2)c(C)n1 89121,C(=O)(C1CCCc2ccccc21)N1C(C)CN(C(C2CC(C)(C)C2)=O)CCC1 89122,C1(NC(C(C(=O)OC)C)=O)CN(C(=O)CCN2CCCS2(=O)=O)CC12CC2 89123,N1(C(CCC=CC)=O)Cc2ccccc2C1C(=O)Nc1cncc(C(F)F)c1 89124,N1(C(C(CC#C)O)=O)CC2CCC1CN2C(=O)C(C(C)(C)C)SC 89125,c1(-c2nc(C(=O)NCCC3(CSC)CC3)sc2)cccc(C#N)c1 89126,c1(NCC(N2CCC(C(C)NC(CN3CC(C)C3)=O)C2)=O)ccc(O)cc1 89127,C1(NC(c2c(CC)ncnc2)=O)(CNC(=O)COCC(=O)NC)CCCCC1C 89128,c1(NCc2n(C)c(Br)nn2)nc2ccccc2nc1NCC1C(C)(C)C1(F)F 89129,CCC(C#N)C(=O)N(C(CC)CC(=O)N(C)Cc1scnc1C)C 89130,c1(C(=O)NC2(CC=C)CN(C(C3(c4cc[nH]n4)CC3)=O)C2)cccc(C(N)=O)c1 89131,C(=O)(C(CC)CC(C)C)NC1(CN(C(CN(CCC#C)C)=O)C)CC1 89132,CN1CC(C(=O)NC(CC2CCC2)C(=O)NCC2(C(C)(F)F)CC2)CCC1=O 89133,c1(C(=O)NCCN(CC(C)O)C(C2CCC2)=O)cc2sc(Br)cc2[nH]1 89134,N1(C(C(CC)OC)=O)CC(NC(=O)COC2CC2)C(C)C1.c1ccc(C(C)=O)cc1 89135,C1(NC(CC2C(C)C2)=O)CC2(C1)CC(NC(c1ncoc1C1CC1)=O)C2 89136,C1(CC(=O)NCC2(NC(=O)COCC3CCCO3)CCOC2)CC2(CC2)C1 89137,c1(C(=O)NCC(CN(C)C(c2cn(CC3CC3)nn2)=O)O)csc(C#N)c1 89138,O=C(CC1=CCCCC1)NC1CCCC(NC(=O)CCC2CC2)CC1 89139,Cn1cc(Cl)c(C(=O)NC2CC3(C2)CC3C(N2CCCC(F)C2)=O)n1 89140,c1(C(C)=O)ccc(SCCC(=O)NCCC2(CNC(=O)C=C(C)Cl)CC2)c(F)c1 89141,C1(CNC(C2(CC(C)C)CCNC2=O)=O)COCCN(C(=O)C#CC2(C)CC2)C1 89142,C12(CNC(C(C)N(C(=O)Cn3ccnc3C)CCC)=O)CCCC(CO1)C2 89143,C(=O)(N=c1cc(Cl)cn[nH]1)C1C(NCc2cc(C)ncc2)C1 89144,N1(C(c2ccc(SC)cc2)=O)CC2(C)CC1C2CNC(=O)Cc1ccc(C)nc1 89145,c1(OCC)cc(N2CCC(C(C)NC(=O)C(C)(C)O)C2)ncn1 89146,C1(C(N(CCOC)CCO)=O)C2CC1N(C(C1CN(C3COC3)C1)=O)C2 89147,C(=O)(C(C)(N)C(F)(F)F)NCc1n(CC)nnc1C 89148,N1(C(C(C)n2cnnn2)=O)CC2(C1)CN(C(c1c[nH]cc1C1CC1)=O)CCO2 89149,C1(CNC(C(C)C2CCOC2)=O)(CNC(C2(C)COC2)=O)CC1(F)F 89150,c1(C(=O)NC2C(NC(C=C(C)C(C)(C)C)=O)C2)oc(Br)nc1C 89151,C1(C(N2CCCN(C(Cc3ccc(C)s3)=O)CC2)=O)CCCCN(C)C1=O 89152,CS(=O)C=CC(=O)NCC1CC(NC(=O)Cn2cc(Br)cn2)C1 89153,C1(C#N)(C(=O)NCC2CN(C(c3cc(C)sc3)=O)CC2C(F)(F)F)CCOCC1 89154,N1(C(CSCC#C)=O)CCC(O)(CN(C)C(C2CCCN2C2CC2)=O)C1 89155,c1(C(N2CCC(NC(C(CCC)=CCC)=O)(CO)C2)=O)cc2ncccc2[nH]1 89156,C1(C)(CC)CC(NC(c2c[nH]nc2OC)=O)CN1C(=O)Cc1ccnn1C 89157,C1(C(=O)NCC2(CNC(c3c(N(C)C)ccnc3)=O)CCC2)CCCCNC1=O 89158,c12cncc(c1)C(=O)NC1CC(C1)CO2.C1(CC)CC(n2ccnn2)C1 89159,C1(C(C(=O)NCC=C)N(C(C)COCC)CC=C)CC2OC(C)(C)OC2C1 89160,N1(C(C(CC2CCC2)OC)=O)CC2CC(C1)N2C(=O)Cc1ccc(Cl)cc1 89161,c1(N2CC(CNC(c3cc(CCC)oc3C)=O)(OC)C2)cc(O)nc(COC)n1 89162,c1(CC)ccc(F)c(C(N2CC(C3(NC(C4CC45CC5)=O)CC3)C2)=O)c1 89163,CCC(C)(CCC(C)C)C(=O)N1CC2CN(Cc3c(OC)cccc3Cl)C2C1 89164,C1(C(=O)NC2(CC(=O)NCc3n(CCC)ccn3)CCC2)CCC(C)(CC)O1 89165,c1(C(=O)NC(CCCCC#C)=O)ccc2c(c1)CN(C(C1CCN(CC)C1)=O)C2 89166,c1(C(=O)NC2CC(C)(NC(C(C)NC(=O)NC)=O)C2)cccc(OCC(F)F)c1 89167,CC(CC(=O)NCC(O)CNC(=O)CS(=O)(=O)CC1CCCO1)C(F)(F)F 89168,n1(CC)c(C(=O)N(C(c2ccccc2)CNC(C2(F)CC2C)=O)C)cnc1O 89169,C#CCC(CC(=O)Nc1cc(OC)cc(Cl)c1)NC(C1(CF)CC1)=O 89170,CN1Cc2cc(NC(=O)NC3CCc4ncnn4C3)ccc2C1=O 89171,C(=O)(CCN=C(NCC1CCN(S(C)(=O)=O)C1)NC1CCOCC1F)NC 89172,c1(CCCC)nc(C(N2CC(NC(=O)C(C)NC(c3ccco3)=O)C2)=O)cs1 89173,c1(-c2nc(C3CCC(C)CC3)nn2C(C2CCOCC2)C)nccc2occc12 89174,C1(CNC(CC(=O)NCC#C)=O)CCCN(C(C2CC(C)CCO2)=O)CC1 89175,C1(C(N(CC(O)CNC(c2n[nH]cc2C2CCC2)=O)C)=O)CCC(C)CC1 89176,c1(OCC(=O)NCC(C)(C2CC2)NC(C2CC(C)(F)C2)=O)c(F)cccc1F 89177,N1(C(C(C=CC)O)=O)CCCC12CCN(C(C1CC(=O)CCO1)=O)C2 89178,c1(C(=O)NC23CN(C(Cn4c(C)cc(C(F)F)n4)=O)C(C2)C3)ccc(F)c(F)c1 89179,S(=O)(=O)(c1ccc(NCC2(C)CCC(=O)N2)c(F)c1)N1CCC(CC=C)C1 89180,C1(C(=O)NCc2ccc(C)s2)CC(N=[N+]=[N-])CN1C(=O)C(F)C1CCC1 89181,C#CC1(NC(=O)C(C)N(C(C2CCN(C)CC2)=O)CC)CCOC1 89182,N1(C(C(F)OC)=O)CC(CO)C2(CCN(C(C3COC(=O)N3C)=O)CC2)C1 89183,CC1(C)CC(C(=O)NC2CCCC2CNC(C2(Br)CC2(C)C)=O)=NO1 89184,C1(CC)CN(C(=O)CCc2cc(C)n(C)n2)CCN1C(=O)COc1ccncc1 89185,Cc1cc(C(=O)NCC2CCCC2NC(c2cnncc2O)=O)cc(N)c1O 89186,c1(C(=O)NCc2ccc(C(N3CC(O)(CO)C3)=O)cn2)n[nH]c2c1CCC2 89187,CCCCC(CNC(=O)CCOCc1ccccc1)NC(=O)C(O)CC 89188,c1(CNC(=O)CC2CCOC2C)n[nH]cc1C(=O)NC1CC(NC(C)=O)C1 89189,C1(CNC(C(C(CC)O)C)=O)CCC2CN(C(=O)Cc3nc(C)sc3C)CC12 89190,C#Cc1cccc(C(=O)NCC2CN(C(=O)Cn3cc([N+](=O)[O-])cn3)C2)c1F 89191,N1(C(=O)NCC)CCCC(C(=O)NCC2(OC)CN(C(C3(CC)COC3)=O)C2)C1 89192,C(CCC(=O)NC(Cc1ccccc1)CCNC(=O)COC1CCOC1)OCC 89193,CC(C)(CCF)C(=O)NC1CC(O)(CNC(C2CC(CC3CC3)C2)=O)C1 89194,c1(N2CCOCC(NC(C(c3cccnc3)OC)=O)C2)ccn2ccnc2n1 89195,N1(C(C2(F)CN(C(c3nc(COC)oc3)=O)C2)=O)CC(OC)C(O)C1 89196,O=C1OC2CC1N(C(C1CCCC(CC(F)(F)F)N1)=O)C2 89197,c1(CC)nc(CNC(C2(NC(C3CC(F)(CF)C3)=O)CC2(C)C)=O)n[nH]1 89198,C1(NC(C2CCCN2CC2CCN(Cn3ccnc3)CC2)=O)CCC2CCCC12 89199,C(CC1=CCN(C(C2CCc3ccnn3C2)=O)CC1)NC(C(C)(O)C1CC1)=O 89200,C(=O)(CCC(=O)NN(C)C)N1CC(C)N(C(=O)COc2cccnc2)CC1 89201,c1(C(=O)OC)ccc(F)c(C(N2CCN(C(c3cc(Cl)c[nH]3)=O)CC2CF)=O)c1 89202,c1(C(=O)NC2CC(NC(C3C4CC5C(C4=O)C35)=O)C2)ccc2c(n1)CCO2 89203,Cc1c(C(=O)NC(CN(CCO)C(C)C)C2CCC2)cccc1Cl 89204,c1(C(N(CCNC(C(CC)C)=O)C)=O)cc(C)n(C(CC)CC)n1 89205,N1(C(CCc2scc(C)n2)=O)CCOC(CCNC(C2(C)CNC(=O)C2)=O)C1 89206,Cc1cc(C)c(C(N2CC(N3CCN(C(C4CCCCC4F)=O)CC3)C2)=O)[nH]1 89207,N1(C(CSc2nc(C)[nH]n2)=O)C(CNC(C2(n3cnnn3)CC2)=O)CC2COCC12 89208,C(=O)(CC(C)C(F)(F)F)NC(CCN(C(CCCCOC)=O)C)C 89209,C1(O)(C(=O)NC2CC(C(N3C(C)(C(=O)OCC)CCC3)=O)C2)CCOC1(C)C 89210,Cn1c(C(N2CC(CNC(C3CC(C)(C)CO3)=O)C2)=O)cc2sccc12 89211,C(=O)(C(CCNC(C1(C2CC2)CCCO1)=O)OC)NC1(COC)CC1 89212,c1(N2CC(CC)(CC)S(=O)CC2)nc(C)cc(=NCC2CC3(CCOCC3)C2)[nH]1 89213,N1(C(c2c(C)nn(C(C)C)c2)=O)CC(NC(=O)CC=C(Cl)Cl)CCC1C 89214,C(c1c[nH]c2ccccc12)=CC(N1C(C(N2C(C)C(O)CCC2)=O)CC(O)C1)=O 89215,C1(CC(=O)N(CC#C)CC=C)CCN(C(=O)C(C)C2CCC2)C1(C)C 89216,c1(C(C)C(=O)NC(C2(N(C(=O)C3CC3)C)CC2)C)cnn(C)c1 89217,C(=O)(C(C)(CCF)NC1(c2ccn(-c3c(F)cccc3F)n2)CCC1)OC 89218,C1(NC(=O)Cn2cnnc2O)CC2(C1)CN(C(=O)Cc1ccccc1C1CC1)C2 89219,N1(C(c2c(C)ncn2C)=O)CCC2(CCCN2C(c2cncc(Cl)n2)=O)C1 89220,CC1CN(C(=O)COCC2CC2)CC(C)C1NC(=O)CCCN(C)N=O 89221,C1(C(N2CCC(CCNC(C3(CO)CC(F)(F)C3)=O)C2)=O)CC2CCCC(C1)C2 89222,c1(C(N(CCC)CCNC(c2sccc2Cl)=O)=O)ccc(F)c(C)c1C#N 89223,c1(NC(CCC)C)ncnc(NCCc2ncccc2C)c1C 89224,Cc1ncc(C(=O)NCC2CCCCN(C(c3cncs3)=O)C2)cc1N 89225,c1(C(N(CC(CC)NC(CC(CC)C2CC2)=O)CC)=O)c[nH]c2c(Cl)cccc12 89226,N1(C(CC2ON=C(C(=O)OC)C2)=O)CCOCC(C)(CNC(C2(O)CCC2)=O)C1 89227,Cc1cc(OCC(=O)NC2(CNC(=O)C3CC3)CCCCC2)ccc1[N+](=O)[O-] 89228,C1(CNC(c2c(OCC)oc(C)n2)=O)COC(C)(C)CN1C(c1ccns1)=O 89229,C1(NC(c2cnc(COC)s2)=O)CC2CC1CN2C(c1cn(C)c(C)n1)=O 89230,Cc1csc2ncc(C(=O)N(C)CC3CC(F)CN3C(=O)CC3(C)CC3)n12 89231,C=Cc1cnn(C)c1C(=O)NCC1CN(C(=O)C(F)(F)CC)CC1C(F)(F)F 89232,Cc1cc2c(C(N3CCSCC3CCNC(C34COCC3C4)=O)=O)cccc2o1 89233,c1(NCC2CCCN(C(C)=O)C2)[nH]c(=NCCCC2CCC2)nc2c1ncn2C 89234,Cc1nc(C)n(CCC(=O)NCC2(C(C)(C)O)CN(C(=O)CC(F)(F)F)C2)n1 89235,N1(C(C2CC3(C2)CC(F)C3)=O)CC2CCCC(C1)N2C(C1(O)CCCCCC1)=O 89236,n1(CCNC(=O)C(C)CC(N)=O)nnc2c(N3CCC(=CCOC)CC3)ncnc12 89237,N1(C(C(COCC)(C)C)=O)CC2(CNC(=O)CC(C)(O)C3CC3)CC1(COC)C2 89238,C1(C(=O)NCC2(F)CC(NC(C3(CF)COC3)=O)C2)CCCCCC1 89239,c1(NC(C2(OC)CCN(C(C(CCCOC)C)=O)C2)=O)cn(C)c(=O)nc1O 89240,C1(C2N(C(=O)CCCOC(C)C)CCC2)CCN(C(c2c[nH]c(=S)cn2)=O)CC1 89241,N1(C(c2ccncc2O)=O)CCCC2C1CCN2Cc1ccc(F)c(F)c1Cl 89242,C(CCCC(=O)NC1(CN(C)C(C2(OC)CC2)=O)CC1)OCC 89243,C1(NCCn2cnc(C)c2C)CCC2COCCC2(C#N)C1 89244,CC1(C)CC(C(=O)NC2CC2NC(=O)CCc2ccc(Cl)cc2)C(C)(C)O1 89245,CC(C)C(CNC(=O)CP(C)(C)=O)C(=O)NC(C)(CO)C(C)(C)O 89246,c1(COC)nn(C)c(Cl)c1C(N1CCC(O)(CNC(=O)CCF)C1)=O 89247,CC12CC(C(N3CCC(CNC(C4C5CC5C5CC45)=O)C3)=O)(CCO1)C2 89248,c1(-c2cn(CCN3CCC(C)CC3)nn2)ccc(Cl)cc1F.C1CC(=O)N2CCC12 89249,C(C)(C)(CCC(=O)N(C)CC1CN(C(=O)C(c2ccc(Cl)s2)C)CCO1)OC 89250,c1(OC)cc(CNC(=O)CC2(C)CN(Cc3cc(CO)ccc3O)C2)ccc1F 89251,c1(C(=O)NCC2C3CN(C(=O)CC4CC=CCC4)CC23)cc(O)ncn1 89252,Nc1cc(Cl)cc(Cl)c1C(=O)NCCC(O)CNC(c1cnc(C2CC2)[nH]1)=O 89253,c1(C(N2CCC(CNC(c3c(C)n(C)nc3)=O)C2)=O)cc(Br)cc2nc[nH]c12 89254,c1(SC)ccc(C(=O)NCC2(F)CC(CNC(=O)C=CC3CCCO3)C2)o1 89255,c1(C(=O)NCCN(C(COCCC#C)=O)CCCN(C)C)cnnc(O)c1 89256,C(=O)(CCCCN1CCOCC1)NC(CC(C)NC(c1[nH]cc(CC)c1)=O)C 89257,C1(C(=O)NC2CC3COCC3C2)C2CC(C(O)C2O)S1(=O)=O 89258,CCC(C)N(OC)C(=O)C1CC=CCN1C(C1CC2(C1)CC2(F)F)=O 89259,c1(C(C)C)nccn1CC(=O)NCC(O)CN(C)C(C1CC1C(C)(C)C)=O 89260,CC(C)C(C)C(CNC(=O)Cc1c(Cl)cnn1C)NC(=O)COCC1CCC1 89261,C(C(=O)NNC(=O)Cn1ccc(C2CC2)n1)(c1ccc(O)cc1)OC 89262,CC(C)C(C)(CNC(=O)C(C)Oc1ccc(F)cc1)NC(=O)C=Cc1cocn1 89263,N1(C(c2nc(C(c3ccccc3)C)sc2)=O)CC(C(=O)O)CCC1C(=O)O 89264,Cc1cccc(CCCNC(c2nc[nH]n2)C)c1 89265,c1(C(=O)NCC2CCN2C(c2ns[nH]c2=O)=O)ccc2ocnc2n1 89266,C(=O)(C1=CCc2ccccc21)NC1C(NC(C(c2ccc(Cl)cc2)C)=O)C1 89267,c1(OCC)ccc(C#CCN=c2cc[nH]c(C)c2Br)cc1 89268,C1(S(N)(=O)=O)(C(=O)NC(C(C)NC(C2CCCC(=O)N2)=O)CO)CCC1 89269,C(=O)(CC(O)CC(C)(C)C)N1C(C(C)NC(CCCn2ncc(C)c2)=O)CCC1 89270,c1(OC)ccc(O)c(C(c2ccccc2)NC(=O)CCCCCN(C)C)c1 89271,C1(CCOC)CN(C(=O)CN2CCC2C)CCN1C(=O)Cn1cncc1C 89272,c1(C(=O)NC(C2CCCN(C(=O)C=CS(C)=O)C2)C)cc(C(F)(F)F)ccc1Cl 89273,C1(NC(C(CC)C(C)O)=O)CCC2CCN(C(=O)C(C)(C)CC#N)C1C2 89274,c1(C(=O)NC2(CC=C)CN(C(C3(OC)CCOCC3)=O)C2)cnc(S(C)(=O)=O)s1 89275,c1(OC)n[nH]c(NC(C2CN(C(C3CCCC3C)=O)CCS2)=O)c1C#N 89276,N1(C(CSC(C)C)=O)CC2(C(N3CCOC(C(C)(C)C)C3)=O)CCC1CC2 89277,N1(C(c2cncc(C#C)c2)=O)CCC2CN(C(c3cccc(OC)n3)=O)CC12 89278,C1(C(N(N2CSCCSC2)CC(=C)C)=O)CCCN(C(=O)C2CC2)C1 89279,N1(C(C)=O)CC(CNC(C2(n3cc(COC)nn3)CCC2)=O)CC(O)C1 89280,CC1C(NC(C2CC(O)C2)=O)CC2CCC1N2C(C1(CF)CCC1)=O 89281,Cc1c(N(CC(C)(C)C(F)(F)F)C)nc(Cl)nc1O 89282,N1(C(C2(CC)CNC(=O)C2)=O)CC=C(C(=O)N(C)CC2(N(C)C)CCC2)C1 89283,C1(NC(c2ccc(COC)o2)=O)CCCCC1NC(C1CCCC1C(F)(F)F)=O 89284,C(CC(C(C)(C)C)NC(c1cc(F)cs1)=O)N(C(c1c(CC)n(C)nc1)=O)C 89285,C1(CNC(Cc2cccc(OC)n2)=O)CCC2(CCC2)C1NC(=O)C1CC1 89286,N1(C(c2cc(F)ccc2F)=O)CC2CC(C1)CN(C(C1CC=CCO1)=O)C2 89287,C1(C2(C(=O)NCCn3cccn3)CC2)CCCN1C(c1nc(Cl)cs1)=O 89288,c1(COC(C)C)cc(C(=O)NCCN(C)C(C2COC(C)(C)CO2)=O)ccc1F 89289,C1(NC(C(CC)O)=O)C=CCCC1C(=O)NCCC1CCCC12CC2 89290,c1(C(=O)NC23C(CCN(C(C4(CC)CC4)=O)CC2)C3)cc(O)nc2c1CCCC2 89291,CC(O)CC(=O)NCC1(C(=O)NCCCC2CCCC2O)CC1 89292,C1(NC(C(C)c2ccsc2)=O)C2CN(C(=O)CCc3ccc(N)cn3)CC12 89293,Cc1cc(F)c(C(=O)NC2CC(C)(NC(c3ccnc4c3CCC4)=O)C2)cc1F 89294,C1(NC(C)=O)CCN(C(C(=O)NCCN2CCOCC2)C2CC2c2ccco2)C1 89295,c1(C(=O)NC2C(NC(C3C(=C)C3)=O)C2)cncc(NC(C2(O)CC2)=O)c1 89296,N1(C(C2C(SC)CCC2)=O)CCC(C2(O)CN(C(c3coc(CO)c3)=O)C2)CC1 89297,c1(C(=O)NCC2CC(NC(C(C(C)O)N(C)C)=O)C2)ccc(C2CC2)c(F)c1 89298,c1(C(N2CCC(NC(C3(OC)CC3)=O)C(C(C)C)C2)=O)ccnc2c1ncn2C 89299,Cc1c(C(=O)NC2(C)CN(C(C3CCCN3C)=O)C2)cccc1Br 89300,c1(C(=O)NCCNC(Cc2c(C)ccc(F)c2)=O)cccc2c(C)ccnc12 89301,Cc1c[nH]cc(C(=O)NC(C(C)NC(c2cn(C)nc2C(F)F)=O)C(C)C)c1=O 89302,c1(C(N2C3CC(NC(c4c(C)nsc4)=O)C3CC2)=O)cccc2c1ncn2C 89303,N1(C(CC(=O)OC)=O)CCC(CC(N)=O)(NC(=O)Cc2ccsn2)CC1 89304,C(=O)(C1CCc2cccc(F)c21)NCC(C1CC1)NC(c1c(C)noc1C)=O 89305,CCC(CCCC(=O)N(CC(O)(CC)CC)C)NC(=O)CC1CCCC(=O)C1 89306,N1(C(c2c(C)n(C)nc2)=O)CCC(C(N2CC(O)C(C)(C)C2)=O)C(C)(C)C1 89307,N1(C(C2(CC=C)COC2)=O)CCC2CCC(C1)N2C(=O)C=CC1CC1 89308,N1(C(CCOCCC)=O)CCCC(C2CCN(C(=O)CC(F)F)CC2)C1 89309,N1(C(CN(C)C)=O)CCC(C)(CC(=O)NCC2(Br)CC2)C1 89310,N(C1CCCc2ccoc21)C(C1(NC(C(C)C2CCCO2)=O)CCC1)=O 89311,Cc1ccc(NCC(N2CC(CNC(=O)CN3CCCS3(=O)=O)CC2C)=O)cc1 89312,c1(C(N2CCC(NC(C=CCC)=O)(CO)C2)=O)nc2ncccn2n1 89313,C1(C)(CNC(C(c2cn(CC)nc2)=O)=O)CCCN1C(=O)CCOCC(F)(F)F 89314,C1(CNC(C2(C)CC2)=O)C=CC(NC(c2coc(Br)c2)=O)C1 89315,N1(C(C2CCC(C)O2)=O)CCc2cnccc21 89316,C1(C(=O)NC(C(C)NC(C=Cc2ccc(CC)o2)=O)CO)CCn2nnnc2C1 89317,N1(C(C(CC=C)CC)=O)CCCCC2C1CCCN2C(c1nccnc1N)=O 89318,N1(C(=O)CCSC(F)(F)F)CCC(N(C(=O)CC2(CO)CC2)CCO)CC1 89319,c1(CCN2CCC(N)C2)ccc(OC(F)F)cc1F.CC(CCO)c1cn[nH]c1 89320,N1(C(c2c(C)c(F)cnc2)=O)CC2CC(C(=O)NCCCN=[N+]=[N-])C(C2)C1 89321,c12cc(ccn1)NC2=O.N1(CCN(CCC(=O)O)C)CCCCCC1 89322,c1(C(N2CCC(C(=O)NCC(C(CC)C)(C)O)C(C)C2)=O)c[nH]c2nccc-2c1 89323,C(=O)(CCC(C(C)C)NC(C1CC(=O)C1)=O)Nc1ccc(C#C)nc1 89324,C1(CNC(CC2CCC(OCC)CC2)=O)CCN(C(=O)C(C)SC(C)C)C12CC2 89325,C1(CC(=O)NCC2N(C(CCCN(C(=O)OCC)C)=O)CC2)CCCC1(F)F 89326,N1(C(c2[nH]n(C)c(=O)n2)=O)CCC(F)C(NC(C2CCC(NC(N)=O)CC2)=O)C1 89327,c1(C(C)NC(=O)C(=O)N(C)CC2CCOC2C)cccc(Cl)n1 89328,N1(C(c2c(C(=O)OC)cccc2)=O)CCN(C(=O)CC2CC2C)CC(O)C1 89329,c1(C(N(C2CCCC(NC(C3CC(=C)C3)=O)C2)C)=O)cnn2cc(C)cnc12 89330,O=CN1CCCC1C(N1CC2C(CNC(c3csnc3Cl)=O)C2C1)=O 89331,Cc1c(Cl)sc(Cl)c1C(N1CC2CC(NC(=O)CCc3ncc[nH]3)C1C2)=O 89332,C1(NC(C(C)CC2CC2)=O)CC2CCC1CN(C(c1ccc(=O)n(C)c1)=O)C2 89333,CCCCCCC(C)C(=O)NCC(CCNC(=O)CSCCN(C)CC)OC 89334,N1(CC(=O)NCC2N(C(C(C)OCCN(C)C)=O)CC2)CCC(C)(C)C1 89335,CC1CCCn2c(C(N3CCCC(N4CC(O)C4)C3)=O)cnc21 89336,C1(NC(c2n(C)ncc2)=O)CCCCC1NC(c1ccncc1F)=O 89337,N1(C(C2C(CC)CCC2)=O)CC2CCCC(C1)N2C(c1ccc2cnsc2c1)=O 89338,C12(C(=O)NC3CCCN(C(c4ccc(NC)c(F)c4)=O)C3)CCCCN1CCC2 89339,N1(C(C(Cc2ccoc2)NC(c2c(OC)cnnc2)=O)=O)CC(O)CC(O)C1 89340,C1(C(N2CC(C)C(NC(=O)CC(=O)NC3CC3)C2)=O)C2CCCCCCC12 89341,c1(COC)nc(NC2(CO)CCCN(C(=O)C(C)C(C)COC)C2)cc(Cl)n1 89342,N1(C(=O)CCn2cncn2)CC2CCC(C1CO)N2C(=O)CC1CCCCCC1 89343,CC1CCN(C(C2CN(C)CCN(C)C2)=O)CCN1C(=O)Cn1ncccc1=O 89344,c1(C(C(=O)NC2CCCCN(C(CC(=O)NCC)=O)C2)C)cc2ccccc2o1 89345,CC1CN(C(=O)NCc2ccn(C(F)(F)F)n2)CC(C)S1 89346,C1(NC(c2ncn(C)c2)=O)CN(C(C2CC(=C(F)F)C2)=O)CC2(CCC2)C1 89347,c1(CC(=O)N(C)CC2C3CN(C(CC(C=C)C)=O)CC32)noc2ccc(F)cc12 89348,N1(C(=O)NC2CCc3nc[nH]c3CC2)CCCC1C1CCCN1C(C)(C)C 89349,C1(C(C)NC(=O)CN(C)C)CCCN(C(c2cc(N)cnn2)=O)C1 89350,Cn1cnc2cc(C(=O)NC3CC4(NC(=O)CC5(CO)CC5)COC3C4)ccc12 89351,C1(CN(C(=O)CC2OCCCO2)C)COCCN1C(=O)CC1CCCO1 89352,C(C#Cc1ccccc1)N1CC(C)C(NC(=O)CCCC(N)=O)C1 89353,C(=O)(C1=NNC(=O)CC1)N1CCN(C(C=Cc2cc(OC)ns2)=O)C2C1C2 89354,C1(C(N2CCC(CNC(c3onc(COC)n3)=O)C2)=O)CCCCNC1=O 89355,O=C(CC(C(F)F)NC(=O)CN1CCCC1)NC1CC2OC1C1CC21 89356,c1(C(=O)NC2CC(N(C(CC(C=C)C)=O)C)C2)cnc(O)n(C2CC2)c1=O 89357,C1(NC(C=COCC)=O)CN(C(=O)Cc2ccc(O)cc2)CC1N=[N+]=[N-] 89358,C1(C(=O)NC2CC(C)(NC(C(C(C)C)C)=O)C2)CC(F)(F)C1(C)C 89359,c1(C(N(CCCN(C(c2nccc(C)c2O)=O)C)C)=O)cc2cccc(F)c2o1 89360,C#CCC(O)C(=O)NC(C)(C)CNC(=O)C(=Cc1ccccc1)NC(C)=O 89361,C12(NC(C3CC3F)=O)CCC(CC1)N(C(C1(F)C3CCCCC13)=O)C2 89362,c1(C(N2C3CC(NC(c4c(CC)con4)=O)C(C3)C2)=O)ccn2nnnc2c1 89363,CC(C(=O)NCCCN(C(=O)Cc1ccc(Br)s1)C)C(F)(F)F 89364,c1(-c2cccc(NC(C)=O)c2)ccc2c(c1)CN(C(c1ccncc1CO)=O)C2 89365,C1(CC(=O)NC(CNC(C(c2ccccc2F)C)=O)(C)C)SC2=NCCN2C1=O 89366,Cc1c(C(N2CCC(N3CC(F)(F)C3)CC2)=O)cc([N+](=O)[O-])cc1[N+](=O)[O-] 89367,C1(NC(C(CC)OC)=O)CC2CCC(C1C)N2C(c1ccc(C(=O)CF)cc1)=O 89368,c1(C(N2CCCC3(CNC(c4ccc(Cl)cc4)=O)C2C3)=O)cc(F)cc(F)c1O 89369,c1(OCC(=O)NC2CC2NC(c2ccnn2C2CCC2)=O)cccnc1 89370,N1(C(CCOCCC)=O)CCC(O)(NC(C)=O)C1 89371,N1(CC(=O)NCCN(CCC)C(c2ccoc2Cl)=O)CCC(CO)CC1 89372,C12CN(CCO1)CC(=O)NC2.C1(NC(C(c2n(C)ncc2)(F)F)=O)CCC(C)CC1 89373,n1(CC)cc(C(=O)N(CCCCCCNC(=O)OC(C)(C)C)C)c(OC)n1 89374,n1(CC(=O)NC(CC)CN(C)C(c2cnn(C)c2OC)=O)cc(C)ccc1=O 89375,C1(NC(C(C)(C)OC)=O)(COC)CCN(C(=O)C(O)Cc2cccc(Cl)c2)C1 89376,C1(C(=O)NCCC2CC(NC(C=C(C)Cl)=O)C2)C2CCCC12 89377,c1(C(=O)NC2(CCNC(C3CCOC3)=O)CCCC2)cnc(-n2cccn2)cn1 89378,C1(CC(N2CCOC(CCNC(=O)CN3CCC3C)C2)=O)(OC)CCCCC1 89379,c1(CNc2c(C(=O)NCC(=O)NC)scc2)ccc(Cl)c(Cl)c1 89380,C(CCC(C(=O)N1CC=CC1CN(C)C)NC(c1ccc(=O)n(C)c1)=O)OC 89381,C1(C(=O)O)(NC(N2CCN(CC3CCCO3)CC2)=O)CC2(CC(F)C2)C1 89382,c1(C(=O)NC(CC(C)NC(c2nnn(C)c2C(F)(F)F)=O)C)cc2n(c1)CCC2 89383,C1(N(CC)Cc2cccs2)CCN(C(c2cnn(C)c2)C(=O)NCCCF)CC1 89384,C1(NC(C2C(NC(Cn3ncc(C#C)c3)=O)C=CCC2)=O)CCC12CCCC2 89385,C#Cc1cnn(C)c1C(N1CCOC(C(=O)NC(c2cn(C)nc2C)C)C1)=O 89386,C1(NC(c2cc(CNC(C34CCC(CC3)C4)=O)[nH]n2)=O)COCC1C1CC1 89387,c1(N2C(CN(CC)CC)CCC2)nc(NC(c2nnc(O)n2C)C)c2ncsc2n1 89388,c1(C(=O)NCCC(CNC(c2ccc(C)cc2Cl)=O)(C)C)ccn2nncc2c1 89389,c1(C(=O)NCC(CC=C)NC(=O)C(C)(CC)CCC)ccc(CC)c([N+](=O)[O-])c1 89390,c1(CC(N2CC(C(C)NC(c3cccc(OC)n3)=O)C2)=O)ccc(C)c(F)c1F 89391,c1(C(C(=O)NC(CN(C(C(n2ccc(C)n2)C)=O)C)(C)C)F)ccc(F)cc1 89392,C12(COC)COC(C(=O)NCCC3CN(C(=O)C(C(C)C)n4cnnn4)C3)(C1)C2 89393,c1(-c2c(C)ccs2)csc(=Nc2cccc(CO)c2)n1C(C1CCCC1)C1CCC1 89394,C(=O)(C(C(C)O)NC(=O)CCCCN(C)C)NCCOCCC=C 89395,c1(C(C)=O)cc(C(=O)N(CC(C)CNC(=O)Cc2cnc(C)o2)C)co1 89396,CC1CCC(C)(C(N2CCC(=CCNC(=O)CC3(C)OCCO3)CC2)=O)C1 89397,C1(C(=O)NCC(CC)N2CCCC2)CN(C(c2sccc2OC)=O)C(C)(C)C1 89398,Cc1cc([N+](=O)[O-])ccc1C(=O)Nc1nnn(C(C)(C)C)c1C(N)=O 89399,C1(OC)CC(N=c2[nH]c(=NC(C)c3ccncc3F)c3ncccc3[nH]2)C1 89400,N1(C(CNC(c2ccoc2)=O)=O)CCN(C(c2cc(O)ncn2)=O)C2COCC12 89401,n1(CC)cc(Br)c(C(=O)N(CC(C)NC(=O)CCc2ccncc2)CC)n1 89402,c1(CC(=O)NCC2CCC2NC(C2COC2)=O)ccc2c(c1)OCCCO2 89403,Cc1cc(C(N2CC(C(C)NC(C3CCC(C)(C)C3)=O)C2)=O)n(C(C)(C)C)n1 89404,CC(C(=O)N1CCC2(CCN(C(c3cc(Cl)n(C)n3)=O)C2)C1)C(C)S(C)(=O)=O 89405,C1(CN)CN(C(C2C=CC=CC=C2)=O)CC1(C)C.N1(C(C2(SC)CC2)=O)CCCC1 89406,C1(C)(C(N2CC(C(C)OC)C2)=O)CCN(C(=O)C=C(C)C(C)C)C1 89407,N1(C(c2c(CC)c[nH]c2)=O)CCC2CCN(C(c3cc(C)on3)=O)C2C1 89408,N1(CC)CC(C(=O)NC2(CNC(c3cccn3C3CCCC3)=O)CC2)CC1=O 89409,c1(C(=O)NCc2cn(C)nc2C(F)F)c(F)ccc(O)c1F 89410,c1(C(N(CCCCCNC(C2(CC)CCCC2O)=O)C)=O)ccc2occc2c1 89411,CC1(C)CCCC(C)(C)C1C(N1CCCC1CNC(C1CCN1S(C)(=O)=O)=O)=O 89412,C12(CNC(=O)CC3CCC(O)C3)CN(C(c3cc(C4CC4)on3)=O)CC(F)(C1)C2 89413,c1(C(N2C(C(N(CCCCO)CC)=O)CCC2)=O)ccc(C)cc1Cl 89414,C1(C(=O)NC(C2CC(NC(=O)C(C)Cc3cccnc3)C2)C)CCC(CO)CC1 89415,C(=O)(C(CCOC)OC)NCc1c(C(=O)NC(COCC)CN(C)C)nco1 89416,CC(C)C(CCC(=O)N(CCO)CCN(C)C)NC(=O)CSCc1nc[nH]n1 89417,N1(C(C(C)OCC#C)=O)CCOC(CC(=O)NCCc2ocnc2CO)C1 89418,c1(OC)c(C)ccc(C(N2CC3(C2)CN(C(C2CC(C(C)C)=NO2)=O)C3)=O)c1F 89419,c1(C(=O)NC(C2CCOC2)CNC(C=NOC)=O)c(N)cc(Cl)cc1F 89420,c1(OC)cc(C)c(C)cc1C(N1CC2(CCC(NC(c3sccc3I)=O)C2)C1)=O 89421,C1(NC(C23CCC(NC(C(COC)N(C)C)=O)(CC2)C3)=O)CC2(C1)CC(C#N)C2 89422,C1(CCNC(=O)CC2CCNC2=O)CN(C(C2(O)CCCCC2)=O)CCO1 89423,N1(Cc2c(C)n[nH]c2C)CCCC2(CCCN(C(=O)Cc3ccc(Cl)cc3)C2)C1 89424,Cc1cccc(Br)c1C(N1CC(NC(=O)C(C)Cc2ccccn2)C(O)C1)=O 89425,N1(C(C2(NC(C)C)CC2)=O)CCCC1C1CCCCN1C(=O)C=CC1CCC1 89426,CC1CCC(C(=O)N(CCNC(=O)CCc2cccnc2)C2CC2)C1 89427,N1(C(CN2C(C)CCC2)=O)CC(N(C(=O)Cn2ccc(O)nc2=O)C)C(C)(C)C1 89428,c1(C(=O)NC2CCCCC2F)c(Cl)ccc2ccncc12 89429,N1(C(CC2CC(C)C2)=O)CCNC(=O)c2c(Br)cccc21 89430,Cc1c[nH]nc1CNC(=O)CC1CCC(NC(=O)C(C2CCOCC2)O)C1 89431,C(=O)(C(C)C(O)C(C)C)NCCCCCCNC(c1sc(C(=O)OC)c(N)c1)=O 89432,CC(CO)C(C)N=c1ccnc(N(C)Cc2cccnc2)[nH]1 89433,N1(C(c2c(C)scn2)=O)CCCC(C(N2CCCC2CNC(N)=O)=O)(C(C)C)C1 89434,N1(C(C2=NOC(C)C2)=O)CCCN(C(=O)C(C)Cc2ccncc2)C(C)C1 89435,CC(C)(O)C(CCO)NC(C1CC2(CC2)CN1C(=O)CCc1cncs1)=O 89436,N1(C(C(C(C)C)C(C)NC(=O)C=CCF)=O)CCC(O)(C2CC2)CC1 89437,[N-]=[N+]=NC1CCN(C(C2CN(C(=O)COCC(F)F)CC23CC3)=O)C1 89438,N(C(=NCC1CCC(=O)NC1)N1CCC(CCC#N)CC1)C(COC)C 89439,C1(c2n(CCSC)nnn2)(NC2CC(CO)C2)CCN2CCCC2C1 89440,c1(CC(C(=O)NCCC(C)NC(c2cn(CC)nc2)=O)O)cc(Cl)cc(Cl)c1 89441,C1(CNC(C2N(C=O)CCC2)=O)CC2COCC2N1C(c1ccc(Cl)cn1)=O 89442,N1(C(c2c(CC)ocn2)=O)CCC2CN(C(c3ccc(N)cc3O)=O)CCC2C1 89443,C(=O)(C1=CCCOCC1)NCC1(F)CCN(C(c2cc(N)cc(F)c2)=O)C1 89444,N1(C(c2nc(C(C)=O)sc2)=O)CC(NC(C2CCC(C)(C)O2)=O)C2(CC2)C1 89445,N1(C(c2n(CC)ncn2)OC)CC(CC(=O)OC)CC12CCOCC2 89446,c1(CC)ncc(C(=O)NC(C2CCN(C(C34CCC(CC3F)C4)=O)C2)C)c(C)n1 89447,Cc1nc(C(=O)N(C)CC2CCCN2C(=O)C(C2CCCO2)C2CC2)c(C)o1 89448,c1(OC)cc(O)nc(CNC(=O)CC(C(C)C)OC(C)=O)n1 89449,C=CC1(CC(=O)OCC(=O)OC2CC2C#N)CCCCC1 89450,S(=O)(=O)(c1cccc2c1OCCC2)N1CC(O)CC(OC(C)(C)C)C1 89451,N1(C(C(CN(C(=O)C=CCF)C)(C)C)=O)CCC2OCCCC2C1 89452,c1(CC)cc2c(NCCCCCCNC(c3cccnc3Cl)=O)nc(C)nc2s1 89453,c1(C(=O)NCC2CN(C(CC(C)(C)OC)=O)CC2O)cc(=O)c2ccccc2o1 89454,c1(C(=O)NC2C(C)(C)CCN(C(C(C)OC)=O)C2)ccc(=O)n2c1CCC2 89455,N1(C(c2ccc(CC)cc2)=O)CCC2(C)CN(C(=O)CCOC(C)=O)CC12 89456,Cc1ccc(NC(C2(C(C)NC(=O)OC(C)(C)C)CC2)=O)cc1N=[N+]=[N-] 89457,N1(C(c2c(SCC=C)cccc2)=O)CC2(C1)CN(C(C1CCC3CC3C1)=O)C2 89458,N1(C(CCC)=O)CCN(C(=O)CCn2ccccc2=O)CC1CC(F)F 89459,C1(C(N2C(CC=C)CCCC2)=O)CN(C(C2CCCN2C)=O)C(C)(C)C1 89460,CCC(CNC(C1CCCCN1C(=O)C(n1ccnc1C)C)=O)C(C)C 89461,C=CCC(CNC(=O)C=NOC)NC(C1CC1C(=O)NCCO)=O 89462,c1(C(N2CCC(CNC(=O)CC(O)C3CCCC3)C2)=O)cc([N+](=O)[O-])cnc1O 89463,N1(C(C(n2cc(CCN(C)C)nn2)C)=O)CC2CC2(CO)C1 89464,C1(OC)CN(C)C(C)(C(N2CCC(CCNC(=O)CSC(F)(F)F)CC2)=O)C1 89465,C=C(CNC(=O)COc1cnn(C)c1)CCNC(=O)C(n1ccc(C2CC2)n1)C 89466,CCC1=C(C(=O)NCC2CN(C(C3CCCN3C(C)=O)=O)CCN2C)CCCO1 89467,N1(C(C(C)CF)=O)CCC2(CC1)CCN(C(c1cc(F)ccc1O)=O)CC2 89468,c1(CCC(=O)NCC(=O)NCc2ccc(Cn3cc(C4CC4)nn3)s2)nc(O)n[nH]1 89469,c1(C(N(CCC2CCN(C(C3(C)CC(=C)C3)=O)CC2)C)=O)ccc(C)c(C)c1Cl 89470,Cc1cc(C(=O)NCCCCN(C(=O)Cc2ccnn2C)C)c2cnn(C)c2n1 89471,N1(Cc2nc(C(=O)Nc3cccc(OC(C)=O)c3)sc2)CC(C2=NOCC2)C1 89472,n1(CC(N2C(CNC(COCCOCC#C)=O)CC2)=O)cc([N+](=O)[O-])cn1 89473,N1(C(C(=O)NCC)=O)CCC2OCCN(C(=O)CCOCc3ccccc3)C2C1 89474,N1(C(C(CO)NC(N)=O)=O)CC2CC1CN2C(c1cc(Cl)ccc1Cl)=O 89475,CCC(C)CC(=O)C(=O)NC(CO)C(=O)NCC1CCc2nccn21 89476,C(=O)(CC(C)NC(C1CCCC1)=O)N1CC(CCNC(COC(CC)CC)=O)C1 89477,c1(N2CCC(NC(c3c(C)ccc(C)n3)=O)C(C)C2)ccc([N+](=O)[O-])c(C#N)c1 89478,C#Cc1ccc(CNC(=O)C(O)CCNC(=O)CC2CC(C)C2)cc1 89479,C(CCCCC(=O)N1CC(CNC(=O)CS(=O)(=O)NC)C2(CC2)C1)OCC 89480,C#CCCC(C(=O)N1CCC(N=[N+]=[N-])C1)NC(=O)CC1CC(SC)C1 89481,Cc1nc(NC(=O)CCn2nnc3ccccc23)nc(Cl)c1Br 89482,C(C(C)(C)C(=O)N1CC(F)CC1C(N1CCCC1c1ccncc1)=O)SC 89483,C1(NC(CC=C)=O)CN(C(c2ccc(C(N)=O)o2)=O)CC1CO 89484,C1(NC(c2cn(CC)nc2)=O)(CO)CCN(C(=O)C(O)COC)C1 89485,N1(C(Cc2ncn(C)c2)=O)CC2CC1(CNC(C1CC13CCOC3)=O)C2 89486,c1(C(N(CC(C)NC(C(C=C)CC)=O)C)=O)ccn(C)c(=O)c1 89487,C1(O)(COC)CCN(C(=O)C(=O)Nc2cccc(-c3ccccc3)c2)CC1 89488,N1(C(c2n(CC)ncn2)=O)CCCC(NC(c2c(C)nnn2CC)=O)CC1 89489,CC1(C)C(CNC(C2(c3cc[nH]n3)CC2)=O)CCN1C(C1CCNC1=O)=O 89490,c1(CNC(=O)NCCSCC(F)F)ccc2c(c1)CCO2 89491,N1(C(=O)OC(C)(C)C)CCC2CC(NCC3CCOC(C(F)F)C3)CCC12 89492,c1(NC)cnc(C(C)C)nc1C(=O)NC(C)(CNC(c1ccc(O)nn1)=O)CO 89493,C1(NC(=O)C=CCN2CCCC2)CCC2CN(C(c3cnnc(O)c3)=O)CC2C1 89494,C(C1c2ccsc2CCN1C(C1CCCOC1)=O)NC(Cc1nc(CC)sc1)=O 89495,Cc1cn(CC(=O)NC(CNC(=O)CN2CCCCC2)CO)c2ccccc12 89496,C(C)(CO)(CC(F)(F)F)NC(c1cc(OC)c(OCc2c(C)noc2C)cc1)=O 89497,C1(OC(C)C)CCN(C(c2cc(CNC(=O)C=CC(F)(F)F)cs2)=O)C1 89498,C1(NC(CN(CC)CC)=O)CC2(CCCCN2C(c2ncccc2CSC)=O)C1 89499,c1(C(CC)C)nccc(=NCC23CC(NC(c4[nH]ccc4COC)=O)(CO2)C3)[nH]1 89500,C1(C(C(=O)O)Nc2ccc(C(=O)OC)cc2)CC(=O)N(C)C1c1cnn(C)c1C 89501,C(=O)(C1=CC2(CCOCC2)C1)NC1CC(C)N(C(c2cc(C(N)=O)cn2C)=O)C1 89502,N1(C(C(F)=C(C)C)=O)CCOC(CCNC(=O)CCc2nccn2C)C1 89503,C12(NC(CC3(NC(C)=O)CC3)=O)CCCN(C(c3ccc(O)c(N)n3)=O)CC1C2 89504,N1(C(C(CC)CCOC)=O)CC2CCOC2(CNC(=O)Cc2sc(C)cc2C)C1 89505,Cc1c(C(N2CC(CO)OC(CO)C2)=O)oc2cc(Cl)ccc12 89506,CCS(=O)(=O)c1ccc(Cl)c(C(=O)NCC2CCN(C(c3cc(F)c[nH]3)=O)C2)c1 89507,C1(CNC(C(Cc2ncn(C)c2)O)=O)CCC(NC(c2cnc(O)n2C)=O)CC1 89508,N1(C(COCP(C)(C)=O)=O)CCC2CCN(C(C3(CN(C)C)CC3)=O)C2C1 89509,c1(C(=O)NC2CCC(C(=O)NCC(C)(F)F)C2)c(Cl)cc(F)cc1Cl 89510,Cc1cc(C(=O)N(CCCN(C)C(C2CCOC2)=O)C)c2c(n1)CCCC2=O 89511,N1(C(C(C)NC(C)=O)=O)CCN(C(=O)CCCc2nccs2)C(c2cn[nH]c2)C1 89512,N1(C(c2cccc(NC)n2)=O)CCC2(CCCCC2NC(=O)CC(C)C2CC2)C1 89513,S(=O)(=O)(c1ccc(NCc2cnccn2)c(Br)c1)N1C(C)C(C)(C)CC1 89514,C12(C(=O)NC(c3ccccc3)CNC(Cc3cc(C)no3)=O)CC3CC1C2C3 89515,c1(C(CCO)NCCNC(c2n(CC)nnn2)(C)COC(C)C)ccc(F)cc1 89516,C1(CNC(C(C)=C2CCC2)=O)CN(C(c2cccc(Br)c2)=O)CCC1(C)C 89517,Cc1c(C(N2CC(NC(c3cnc(CC(C)(C)C)o3)=O)C2)=O)nn(C)c1C1CC1 89518,c1(C(N2CCN(C(C3CC4CCCCCC34)=O)CC2)=O)cc(O)ccc1Cl 89519,C(C(C)(C)C(=O)N(C)C1CC1)N(C(=O)C(C1CCOCC1)=O)C 89520,C(=O)(CC(C)(C)C(F)F)N1CCCC(C(=O)N(C2(CC)CCCCCC2)CC)C1 89521,c1(C(N(CC(CC)NC(=O)C(CC)N(C)C)C)=O)cc(C)c2c(O)n[nH]c2n1 89522,C(CC1=CCCCCC1)NCC1(C(=O)O)CCN(Cc2ccccc2)C1 89523,c1(CC)cc(=NC2CC(NC(=O)CC(=O)N(C)C)C2)[nH]c(SCC(F)(F)F)n1 89524,N1(C(C(CC=C)(C)O)=O)CC(C(N2CCC(C)(CCO)C2)=O)C2(CCC2)C1 89525,C(=O)(CC1=CCCCC1)N1CCC(C)C1CNC(c1cccc(C(N)=O)c1)=O 89526,CC1(C)CCC=C1C(=O)N1CCCN(C(=O)Cc2ccc(F)c(Cl)c2)CC1 89527,c1(C(=O)NCCN(C(C(=O)NC(CC)C)C)C2CC2)ccc2cccc(F)c2n1 89528,N1(C(C(C)(C)N2CCC2)=O)CCOCC(C(N2CC(SC(F)F)C2)=O)C1 89529,c1(C(N(C2CCN(C(=O)CCc3cccnc3)C2)CC)=O)ccn(C(C)(C)C)c1 89530,c1(C(=O)NCc2cccc(C(N(C(CC(=O)OC)C)C)=O)n2)c(O)cccc1F 89531,N1(C(CC(CNC(=O)C(=CC2CCCC2)C)OC)=O)CC2CC1CC2CF 89532,c1(C(=O)NC(CCNC(c2ccc(CC)[nH]2)=O)C)ccc2c(=O)n(C)cnc2c1 89533,Cn1ncc(C(N2CC(CNC(=O)CCOCC(F)(F)F)C(O)C2)=O)c1Cl 89534,c1(C(=O)NCC2CCN(C(Cc3cccc(C)c3)=O)C2)cc(=O)n2nccc2[nH]1 89535,C(CCNC(C1(NC(C2C(C)(C)C2(C)C)=O)CC(O)C1)=O)(C(C)C)OC 89536,C(CC(=O)N(C)CC1COCCO1)(C(F)(F)F)NC(C1C(C(C)C)C1)=O 89537,C1(CCNC(c2cnc(C(C)O)s2)=O)CCN(C(=O)CC(C)c2ccco2)CC1 89538,Cc1ccnc(CN2CCCC2CC(=O)NCc2cccc(-c3nn[nH]n3)c2)c1 89539,c1(NC2(C3CN(C(C4C5CCCC45)=O)C3)CC2)ccc2cnccc2c1[N+](=O)[O-] 89540,Cc1nnc2cnc(C(N3CC4CC3CCC4NC(=O)CC(C)(C)O)=O)cn12 89541,N1(C(C(C)Cc2cnn(C)c2)=O)CC2(CCCCN2C(C2CCC(CN)C2)=O)C1 89542,CC(C)C(CNC(C1CCCCO1)=O)C(=O)Nc1cccc(OC(F)F)c1 89543,N1(C(=O)Nc2c(Cl)cnc(SC)n2)CCCC2NC(=O)CCCC12 89544,C1(C)(CNC(C=CCCC)=O)CCCN(C(=O)C=Cc2nc(C)cs2)C1 89545,C12(C(N3CCN(C(C4C(CC)C4)=O)CC(C)(C)C3)=O)CCCCC1NC(=O)CC2 89546,c1(CC)c(C(=O)N(CC(C)NC(=O)C(O)(CC)c2ccccc2)C)nnn1C 89547,c1(C(CNC(=O)CCC2CCCO2)=O)csc(CCCn2cncn2)n1 89548,Cc1ccccc1NC(=O)C(N1CCOC(C(=O)N(C)C)C1)c1ccc(Cl)s1 89549,c1(-n2cc(CCC#N)nn2)ccccc1CC(N1CC(C(=O)O)C2CC12)=O 89550,c1(N(C(N(C)C)=O)C)ccc(C(=O)N(C2CC2)Cc2cn(CCCCO)nn2)cc1 89551,Cc1cc(C=CC(=O)NC(C)C(C)NC(=O)C(C)(Cl)Cl)ccc1C(F)(F)F 89552,C1(CC=C)(NC(c2sccc2C(C)C)=O)CCCN(C(c2cncc(N)c2)=O)C1 89553,c1(C(N(C(C(=O)O)C2CCOC2)C)=O)cccc(S(=O)(=O)NC(C)(C)C)c1 89554,N1(C(c2n(C)cnc2)=O)CCC(CNC(c2ccn3ncnc3c2)=O)C(F)(F)C1 89555,CC(C)CC(CNC(=O)C=Cc1cncn1C)NC(C1CN(C)CCO1)=O 89556,c1(OC)ccc(C(=O)NCC(O)CN(C(=O)C2=CCCSC2)C)cc1OC 89557,C=CCC(C(=O)N1CC(O)CC1C(=O)NC1(C2CCCO2)CC1)OC 89558,CC1C(C=CC(N2CC(O)(CNC(c3ccc(C(N)=O)o3)=O)C2)=O)C1(Cl)Cl 89559,C(CC(C)C(=O)NCC(C1CCCC1)NC(c1cccc(OC2CC2)c1)=O)OC 89560,c1(C(=O)NCCC2CCCN(C(CC#N)=O)CC2)c(Cl)ccc2ccncc12 89561,CCC(CC)C(F)C(=O)NC(CCC(=O)N(C1CCC1C)C)C(C)C 89562,C1(OC)CCCCC1NC(c1csc(CNC(C2CC(CF)C2)=O)n1)=O 89563,CCC(C)(CNC(C1CC1F)=O)NC(c1cc(CF)on1)=O 89564,c1(OC)ccc(CNC(C2CCCN(C(c3ccccc3CO)=O)C2)=O)c(F)c1 89565,c1(C(=O)NCC2(NC(C3CC3c3ccsc3)=O)CCC2)cccc2c1CCCN2 89566,c1(OC)cc(F)c(-c2ncccc2C(=O)NC(c2cccnc2)C2CC2)c(F)c1 89567,C1(CNC(CC(C)(C)O)=O)C2CCCCCC12.C12CCCCC1NC2=O 89568,C1(C)(C(N(C)CC2CCN2C(=O)CCCNC(c2cccs2)=O)=O)CCCS1(=O)=O 89569,C1(C(=O)Nc2cccc(NC(=O)C(F)Cc3ccccc3)c2)CCCCCCC1 89570,N1(C(C(COC)C)=O)CCC(C(=O)NCC2CC23CCOC3)CC1C 89571,N1(C(C2(CSC)CC2)=O)CC(CO)(NC(C2CC(=O)N2)=O)C1 89572,C=C1Cn2c(C(=O)NCC3(C(N)=O)CN(C(=O)C=CCn4cncn4)C3)nnc2S1 89573,c1(CN(C(=O)CC2CNCCO2)C)ccc(Br)cc1F 89574,c1(CC)occc1C(=O)NCCN(CC(C)O)C(c1cc(COC)on1)=O 89575,c1(CC(=O)NCCC(C)NC(=O)C=Cc2cnccn2)cn2ccsc2n1 89576,CN1CCOCC2(COCCN2c2nnnn2CC2CCC3(CNC3)O2)C1 89577,C1(C(=O)Nc2cccc(CNC(C(CCC)OC)=O)c2)COc2ccccc2C1 89578,C1(NC(C(C)=C(CC)C)=O)CC(N=c2[nH]cnc3c(C(=O)OC)nsc23)C1 89579,c1(CC)c(N2CCN(C3CCN(C(=O)C=CCF)CC3)CC2)nc(C)nc1Cl 89580,C1(C)(C(N2CC(OCCNC(C(c3cccnc3)OC)=O)C2)=O)C(C)(C)C1(C)C 89581,c1(C(=O)NCC2CC(c3ccccc3)CO2)ccc(Br)cc1 89582,N1(CCC(=O)NCCCN(C(c2cnc(C)o2)=O)C(C)C)CCCCC1=O 89583,C1(C2(NC(C(C)C3CCC3)=O)CC2)CCCN1C(=O)Cn1ccc(Br)n1 89584,C1(C(=O)NC2C(F)CCN(C(CC(C=C)(C)O)=O)C2)CN(CP(C)(C)=O)C1 89585,C(CC(C)CCNC(C1CCN(C(=O)NC)CC1)=O)NC(C=C(CC)CC)=O 89586,c1(OC)c(CNC(=O)NCc2cscc2C)cccc1C#N 89587,C1(C(=O)NC(CC=C)CO)CC(N=[N+]=[N-])CN1C(=O)C(O)CN(C)C 89588,C(=O)(C(CCSC)NC=O)NCCCCCN(C(CC)=O)C 89589,CCC(CC)CC(F)C(=O)NC(CNC(C1(C)CCOC1)=O)CCOC 89590,CN1CCCC1C=CC(N1CCOC(CCNC(=O)CSc2n[nH]c(=N)s2)C1)=O 89591,C1(C(=O)NC(CNC(CN(S(N(C)C)(=O)=O)C)=O)(C)C)CN2CC3CC2(CO1)C3 89592,c1(C2(C(=O)NC3(CNC(CC(C)SC)=O)CCC3)CC2)ccc(Br)cc1 89593,N1(C(CC2C(CC)C2)=O)CC2CN(C(c3sccc3SC)=O)CC2(C)C1 89594,c1(C(=O)NCC2N(C(CCOCC#C)=O)CC(C)CC2)cccc2nonc12 89595,N1(CCCC)CCN(C(=O)CC2CCCCN2C(=O)Cn2cccn2)CC1 89596,C1(NC(C=CC(=O)Nc2cccc(C)c2)=O)COCCN(C(C2CCC2C)=O)C1 89597,C1(C(=O)O)CC2CCC(C1)N2C(c1ccc(F)cc1)c1ccncc1 89598,c1(C(C(=O)NCCCCCC)N(C)CC2CCOC2)cc(C)nc(C)n1 89599,Cn1cc(C(=O)NCC2CC(NC(=O)C=CCO)CC2O)c(-c2nccs2)n1 89600,Cc1c(C(=O)NC(CNC(=O)CCC2CCCCN2C)C2CCC2)c(Cl)nn1C 89601,c1(N2C(C)C(NC(c3ccc(CO)cn3)=O)CCC2)ncc(C#N)cc1Cl 89602,C(C)(CC(=O)NC1C2CC1N(C(c1ccc(CO)s1)=O)C2)(C(F)F)N(C)C 89603,c1(CC)ccc2cc(C(=O)NCC(C)CNC(C3(c4cc[nH]n4)CC3)=O)[nH]c2c1 89604,CC1(C)CN(C(C2CCCN(C3CCCCC3)C2)=O)C1c1cccnc1 89605,C1(NC(c2cn(CC3CCOC3)nn2)=O)CC12CCN(C(c1cnns1)=O)CC2 89606,c1(CC)ccccc1C(CNC(C1CCC2CC12)=O)NC(C1(CCO)CC1)=O 89607,C#Cc1ccc(CC(=O)NCCN(C(=O)C(=Cc2cccnc2)C)CC(C)O)cc1 89608,C1(C(=O)NCC(C(C)C)NC(C2CCCCC2)=O)CCCCN1C 89609,CCCC(C)CCCC(=O)N(C1(C(=O)NC2(c3cc[nH]n3)CC2)CC1)C 89610,C1(C(=O)NCC=CCNC(C2(C)CCC(=O)N2)=O)Cc2ccccc2CO1 89611,c1(C(N2CC(CC=C)(NC(=O)Cc3ccsn3)C2)=O)c(C)cccc1[N+](=O)[O-] 89612,N1(C(COCC(C)C)=O)CC(NC(=O)CCCn2ccccc2=O)CC2(CC2)C1 89613,N1(C(C(C2CCC2)OCC)=O)CCc2ccc(C(=O)NC(CC)CO)nc2C1 89614,c1(CNC(C(CC)(C)O)=O)ccc2c(c1)CN(C(=O)C(C)(CO)OC)C2 89615,N1(C(C(C(C)c2ccccc2Cl)NC(C)=O)=O)CC(F)(F)C(F)(F)C1 89616,Nc1cc(Cl)ccc1C(N1CC2CC(NC(c3ccc(F)s3)=O)C2C1)=O 89617,C1(NC(c2c(N(C)C)ccnc2)=O)CCCCC1N=c1nc(C2CC2)[nH]s1 89618,C(=O)(C#CC(C)(C)CNC(=O)Cc1ccoc1)N1CCOCC(C(C)C)C1 89619,c1(C(=O)NCC2N(C(Cn3ncc(C)c3)=O)CCN(C)C2)cccc2c1CCC2 89620,c1(C(=O)NC2CCN(C(c3c(OC)ccnc3)=O)CC2)cnc2cnccc2c1 89621,C1(C)(C(=O)OCC)CCN(C(C(=O)NC2CC2)C(C)C2CCCOC2)C1 89622,CC1(CNC(c2ncoc2Br)=O)CCCN1C(C1CC(F)C(=O)N1)=O 89623,C1(C(=O)N(C(C)C(=O)N(C(C)COC(C)=O)C)C)(CC)CCNC1=O 89624,c1(C(=O)OCC)cccc(NC(=O)Nc2cnc(OCC(C)C)cn2)c1 89625,c1cc(=NCCCc2nccs2)[nH]c(NC2CCC(C3CC3)C2)n1 89626,c1(C(=O)O)cccc(CN2CCC(F)(C(N3CCS(=O)CC3)=O)CC2)c1F 89627,CN1CC(O)(COCCNC(=O)CC2(N(C)C(=O)OC(C)(C)C)CC2)C1 89628,CC1CCN(C(=O)C(C)(C)N2CCCC2)CCN1C(C1CC2(CCCCC2)C1)=O 89629,N1(C(C(CC)N(C)C)=O)CCCC(CN(C)C(c2csc(COC)n2)=O)C1 89630,c1(C(N(CCCNC(C(CCOC)C)=O)C)=O)cnc2nc(O)nc(O)c2c1 89631,c1(CC(=O)NC2C(OC)CN(C(c3ccsc3OC)=O)C2)cc(F)ccc1O 89632,C1(CNC(Cn2c(=O)sc(C)c2C)=O)CN(c2nncs2)CCC12CCOC2 89633,N1(C(CC2CC(CC(=O)N(C3CC(C#N)C3)C)C2)=O)CCC(C(C)(C)C)CC1 89634,c1(C(N(CC(CNC(C2(CC)CC2(F)F)=O)O)C)=O)nn(C)c2c(=O)[nH]cnc12 89635,c1(C(N(C)CC2CCCN2C(C2CN(C(=O)N(C)C)C2)=O)=O)cn2ccsc2n1 89636,c1(CNC(C(F)=C(C)C)=O)ncoc1C1CN(C(C2CC(C)CO2)=O)C1 89637,C1(CN(C(=O)CCC2CCCC(=O)N2)C)COCCN1C(C1CC2(CC2)C1)=O 89638,c1(C(C)C)ccc(N)c(C(N2C3CCC2C(NC(C2(C)CCCC2)=O)C3)=O)c1 89639,c1(C(C(=O)NC(C(=O)NCC2(CCNC(C)=O)CC2)=O)C)cccnc1 89640,Cc1nn(C)c(N2CCOCC2)c1CN1CCCN(c2ncc(C(=O)O)s2)CC1 89641,N1(C(CN2CCCC(CC)C2)=O)CC2(CCCC2NC(C2C=C2C)=O)C1 89642,N1(C(CC2C(C)C2)=O)CCC(OCCNC(=O)CSc2ccoc2)CC1 89643,C(CC(C(=O)NOCC1CCCC1)OC)NC(c1c(CC)[nH]cc1)=O 89644,C1(C(=O)NC(c2ccnn2C)C(N2CC(OC(C)C)C2)=O)C=CC=CC=C1 89645,CCC(C)(C)OCC(=O)NCC(C)(C)C1CC1.C1=CCNC(=O)C1 89646,Cn1cc(-c2cccc(CC3CCN(n4ccnn4)CC3)n2)c(C(F)(F)F)n1 89647,C1(C(N2CCC(NC(c3c(C(=O)OCC)c[nH]c3)=O)C2)=O)OCC2COCCC12 89648,N1(C(C2(OC)CCCOC2)=O)CC2CC(NC(=O)Cc3n[nH]c(C)n3)C(C2)C1 89649,Cc1ccc(CNC(C)CCc2ccc(Br)cc2)c(Br)c1 89650,C12(C(=O)OCC(c3ccc([N+](=O)[O-])cc3)=O)CC=CCN1CCC2 89651,N1(C(c2ccnn2CC)=O)CCCC(CCC(=O)NC2C(OCCC)CCC2)C1 89652,N1(C(c2c(CNC(c3c(CC)noc3)=O)occ2)=O)CC2CCC2(OC)C1 89653,C1(C(=O)NC2C(NC(COc3cccc(CC)c3)=O)CCC2)C(F)(F)C12CCC2 89654,C1(OCC)CC(F)CN(C(C2C=CC(NC(c3ccc(CC)o3)=O)C2)=O)C1 89655,c1(CCC(=O)NC2CCN(C(c3cc(C4CC4)[nH]n3)=O)C2)cc(F)cc(F)c1 89656,C1(CNC(CCC=C)=O)CN(C(=O)C(C)CCO)CCC12CCOC2 89657,c1(NC(CNC(c2c(CC)cno2)=O)=O)cccc(C#N)c1 89658,O=C(CCCC1CCC1)NCCn1cc(C(N2CC(c3cc[nH]n3)C2)=O)nn1 89659,N1(C(c2ccc(CCCC)cc2)=O)CCC(NC(C2COCC2(C)C)=O)C(O)C1 89660,C1(C(N(C2CCN(C(c3csc(O)n3)=O)C2)C)=O)CCS1(=O)=O 89661,C1(C(=O)NC(CC)CCC(=O)N(CCCN(C)C(C)=O)C)CCCC(C)(C)CC1 89662,N1(C(CC)CO)CC(=O)N(CC(=C)F)C1 89663,c1(C(N2C(CCCNC(c3n(CC#C)cnn3)=O)CCC2)=O)cccc(CC)n1 89664,N1(C(C(C)OCC(C)C)=O)CCOCC(C(=O)N(C(C)(C)C)CCN)C1 89665,N1(CCC(N2CC(CCNC(Cc3c(C)occ3)=O)C2)=O)C(C)CCCC1C 89666,C(=O)(C(O)CC(C)C)NC(C1CNC(=O)C1)C(=O)N(CC(CC)(C)OC)C 89667,Cc1cc(C(=O)NCC2CC(F)(CNC(=O)CC(C)F)C2)ns1 89668,C1(C)(C(=O)NCCCOC)CCCN(C(=O)Cn2nc(C)cc2C)C1 89669,C1(CNC(=O)C=Cc2ccccc2)CC(N=c2[nH]cnc3cnccc23)C1 89670,c1(OC(C)C)ccc(F)cc1C(=O)NC1CCCC(NC(C2(CCO)CC2)=O)C1 89671,C12(CN3CCC(c4cccc(Br)n4)C3)CCCCCC1NCC2 89672,Cc1cncc(C)c1C(=O)NC1CN(C(c2cnc(O)o2)=O)CC1C 89673,C12(C(=O)NCC(=O)CCC3CC3(F)F)CCC(O1)c1ccccc12 89674,CCCC(O)CC(=O)NC(C)CNC(=O)COC(C)CC 89675,Cc1cc(CC(=O)NC23CC(C2)N(C(=O)CCn2cccn2)C3)cc(C)c1 89676,c1(OCC)ncc(S(=O)(=O)Nc2ccc(OCc3ccccc3)cc2)s1 89677,c1(-c2nn(C)c(C(=O)NCC(C)(O)C3CNC3)c2)cc(F)cc(F)c1 89678,C1(CNC(c2ccc(CC)o2)=O)CN(c2nncs2)CCO1 89679,C(=O)(C1=CCSC1)NCc1c(C(=O)NCCC(CC)C)cco1 89680,C(CC(C)C)(C(=O)NC)NC(CC)CN(C)C(c1ccc(OCC(C)C)cc1)=O 89681,C(C)(C(O)C(F)F)NC(C(C)(N(C(C(CC)O)=O)C)C1CC1)=O 89682,C1(n2cc(C3CCOCC3)nn2)(C(N(CCC2CC2)CC)=O)CCOCC1 89683,C1(CNC(C2C(CC)C2)=O)CC(C)N(C(=O)C=Cc2cncs2)C1 89684,C(=O)(C(C)C(C)(C)O)NC1C(NC(c2c(C)[nH]c(C(C)(C)C)c2)=O)COC1 89685,N1(C(CC2CC(C)C2)=O)CCC(C(=O)NCCC(O)C(F)F)C(O)C1 89686,C(=O)(CCC(=O)N1CCCC1C1CCC1)Nc1nnc(CC(=O)OC)s1 89687,C#CC1(C(=O)NC2CC2c2ccn(C)n2)CN(C(=O)C(C)c2cc[nH]n2)C1 89688,CC1(C(N2CCC(N3CCN(C(C4CCCCC4)=O)CC3)C2)=O)CC2CCC1O2 89689,c1(C(C(=O)N(CC(=O)NCC)C)NC(=O)CCOCCCOC)cnn(C)c1 89690,c1(CCC(=O)NCC(=C2CN(C(c3cc(Cl)no3)=O)C2)F)nnc(O)nc1O 89691,N1(C(c2c(C)cc(C)[nH]2)=O)CCC(NC(c2cnc(C(F)(F)F)nc2)=O)C12CC2 89692,N1(C(C2(C)CCC(C)C2)=O)CC(CNC(=O)CNC=O)C(F)(CO)C1 89693,N1(C(CCc2onc(C)n2)=O)CCC(O)C(N(C(=O)CSC(C)C)C)C1 89694,c1(C(=O)NCCC(C)NC(C=C(C)c2cccs2)=O)cnc(O)cc1C 89695,c1(C(=O)Nc2cc(OC)c(Br)cc2C)c(Cl)nc2cc(Cl)ccn12 89696,O=C(CCCC1CC1)NCCCCC1CN(C(c2ncoc2C2CCC2)=O)C1 89697,C1(CC(=O)NC2(C)CC(NC(C(C)Cn3ccnc3)=O)C2)CCC(C)(C)C1 89698,N1(C(c2c(CC)n(C)nn2)=O)CCC(C2CCCN(C(c3cc(Cl)ns3)=O)C2)C1 89699,O=[N+]([O-])c1ccc(CNc2ccccc2-c2ccccc2)cc1C1CC1 89700,N1(C(c2nc(CC)sc2)=O)CCC(CC(=O)NC(C)C(C)C)CC1 89701,C1(NC(=O)COC2COC2)CCC2CC1CN2C(C1(CCF)CC1)=O 89702,c1(CN(C(c2cccnc2)C(=O)OC)C)cc(Br)ccc1OC 89703,c1(C(=O)NCC(CO)NC(c2coc(C3CCC3)n2)=O)ccnc(C(F)(F)F)n1 89704,CCC(C)(COC)CNC(=NCc1ccccc1Cl)NC(C)C 89705,C(=O)(CC(F)F)NCCOCCCN(C)C(c1ncccn1)=O 89706,c1(CC)nc(C)cc(=NCCC2CC(NC(C3CCNC3=O)=O)C2)[nH]1 89707,C(=O)(C1=CCN(C)C1)NC1CC(F)(c2cn(CCC(=O)OC)nn2)C1 89708,Cc1ccc(=N)[nH]c1C(N1CC(NC(=O)CC2(C)CC2)C2(CC2)C1)=O 89709,Cc1ccc(C(C)(F)F)cc1C(N1CCC(C)(NC(c2ccccc2)=O)C1)=O 89710,c1(C(N2CCCCC(CNC(c3ccc[nH]3)=O)C2)=O)ccc2c(=O)ccoc2c1 89711,[N-]=[N+]=NCCCCC(=O)NC1(C(=O)NCC2CCCC2O)CCC1 89712,C#CC1(C(=O)NCc2nccn2CCC)CCN(C(=O)C(C)N=[N+]=[N-])C1 89713,C#CC1(CO)COCCN1C(c1ccncc1-c1cc(F)ccc1CO)=O 89714,c1(OC)ccc(CCC(=O)NC2CCC(NC(c3cnc(S)n3C)=O)C2)cc1F 89715,c1(N2CCC(CC=C)(COC)CC2)nc(=NC)[nH]c(=NC2COCC2F)[nH]1 89716,N1(C(C2CC2Cl)=O)CCC12CN(Cc1cccc(C(F)(F)F)c1O)C2 89717,Cc1noc(C)c1C(C)(C)C(=O)N(CCCNC(=O)C(C)NC(C)(C)C)C 89718,C(C(=O)NN1CCCC1C(=O)N(C)C(c1cnnn1C)C)OCC=C 89719,C1(NC(=O)Nc2c(OC(C)C#N)cc(F)cc2)CCCC2OCCC12 89720,C12C=CCN(C1)CC(=O)NCC1CC(C1)C(=O)N2.c1(C(N)=O)ccnc(C2CC2)c1 89721,C#Cc1ccc(C(=O)NC(Cc2cn[nH]c2)C(=O)NCCCN2CCOC2=O)o1 89722,CN1CCOC(N(C(C(=O)NCCC#N)C(C2CC2)C2CC2)C)C1 89723,CC#CCC(C)N=c1[nH]c(=N)[nH]c(=NCC(c2cccs2)N(C)C)[nH]1 89724,c1(C(=O)NCCC2(OC)CN(C(C3CCC3CF)=O)C2)ccc(Cl)c(O)c1 89725,c1(C(N2CC=C(CNC(C(CC)(C)C)=O)CC2)=O)ccc(S(N)(=O)=O)c(Cl)c1 89726,C1(CCC(=O)NCC(C)(C)F)CCN(C(c2cc(Cl)ncn2)=O)CC1 89727,CC1c2nnc(C3CC3)n2CCN1C(=O)NC(c1cncc(Br)c1)C1CC1 89728,c1(CC(=O)NCC(CNC(=O)C(CO)C2CC2)OC)ccc(C(F)F)cc1 89729,Cc1ccc(SCC(=O)NC(C2CCCN2C(c2nccnc2Cl)=O)(C)C)cc1 89730,C(=O)(C(C)(C)CCCN=[N+]=[N-])NCCOC1CCN(C(C2(C)CCCCC2)=O)C1 89731,CC1(C)COCCC1CC(N1CC2CC2(NC(c2ccnc(C3CC3)n2)=O)C1)=O 89732,c1(CC(=O)NCCC(C)NC(C2CC3CCC2C3)=O)c[nH]c2ccccc2c1=O 89733,c1(C(C(F)F)NC(CCn2cc(CN(C(C)C)C)nn2)=O)c(F)cccc1F 89734,C1(C(N2C(CNC(CC=CCC)=O)CC(C)(C)C2)=O)Cc2cncn2C(=O)N1 89735,c1(OC)cc(C(=O)NCC(Cc2ccc(F)cc2F)CO)ccc1Br 89736,CCCCC(C)CCC(=O)N(CCCN(C(=O)CCc1c(F)cccc1F)C)C 89737,c1(C(N2CC(SC)C(NC(c3csc(Cl)c3)=O)C2)=O)ccc2cc[nH]c2c1 89738,Cc1coc(C2CC2)c1C(N1CCCCC1c1cn(Cc2cscn2)nn1)=O 89739,Cn1c(CNC(C2CCC(CNC(c3nccs3)=O)C2)=O)nnc1O 89740,Cc1c(C(=O)NC2CC2NC(=O)CCCOC2CCCCC2)cnn1CC(C)C 89741,C1(C2CCCN(C(=O)CCNc3ccccc3)C2)(NC(CC(COC)C)=O)CC1 89742,n1(CC)cnnc1CN(C(=O)CC(O)C1CC1)C 89743,N1(c2nnc(COC)s2)CCC(NC(=O)CC2CCOC2)CC(C)(C)C1 89744,N1(C(=O)CC2CCC(O)C2)CCN(C(c2ccns2)=O)C2CCCCC2C1 89745,N1(C(C2C(CC)C2)=O)C2CCC(C(=O)N(C)CCC3CCCCC3)C1CC2 89746,c1(OC)noc(C)c1C(=O)NC(CNC(=O)C(C)(C)COCC(F)F)C1CCC1 89747,c1(C(=O)OC)cc(N2CCC(CNC(=O)Cn3cncc3C)C2(C)C)nc(C)n1 89748,N1(CC)CCOCC1C(=O)NCc1cccc(CN2CCOCC2)c1 89749,N1(S(CCC)(=O)=O)CCC(C(=O)OCC(=O)Nc2ccccc2SCCF)CC1 89750,N1(Cc2cccc(C)n2)CCCC2CN(Cc3cccnc3)CCC12 89751,N1(C(=O)COC2CCN(C(C3(C(=O)C4CC4)CC3)=O)C2)CCCN2CCCC2C1 89752,Cc1ccc2snc(C(=O)NC(CNC(C3CCC4CC3CO4)=O)C3CC3)c2c1 89753,CC1=C(c2cnc(CC(=O)NCc3ccc([N+](=O)[O-])c(Cl)c3)nc2)CCCC1 89754,N1(C(C(CC)CC)=O)CC(NC(C23CCCC2C3Br)=O)C2(CCC2)C1 89755,N1(C(C(C)OCC#C)=O)CCC2(CC1)CCN(C(c1ccc(Cl)c(Cl)c1)C)CC2 89756,c1(COC)ccc(F)c(C)c1F.C12CN(C(=O)OC(C)(C)C)CC1O2 89757,C12(CNC(c3cc(CC)on3)=O)CCC1CCN2C(=O)C=Cc1ccc(C)nc1 89758,Cc1ncc(Cl)cc1C(N1CC(CO)(NC(=O)C(C)C(F)(F)F)C1)=O 89759,C1(NC(CC2(C=C)CCC2)=O)CC2CC(NC(=O)C=COCC)CC12 89760,c1(NC(c2ccnc(C)n2)C)ncc(Cl)cc1C(N)=O 89761,Cc1ccc(CC(=O)N(C(C)C(=O)NC(CC2CCCC2)CO)C)cc1 89762,N1(C(c2cc(Br)cs2)=O)CCC2(CC2C(N2CCOCC23CC3)=O)C1 89763,C(=O)(CC(O)C(C)C)NC(COCC)C(=O)NCc1[nH]cnc1C 89764,C(=O)(C(F)(F)CF)NCCOC1CN(C(C(C)N(CC)CC)=O)C1 89765,N1(C(C(CC)F)=O)CCC(CNC(C2CCCS(=O)(=O)C2)=O)C1(C)C 89766,C(=O)(C1=C(C)OCCC1)N(CCNC(Cc1cccc(OC)n1)=O)C1CC1 89767,Cc1ccc(Br)cc1CN1CCCC(C(N2CCCC(C)(C)C2)=O)C1 89768,C(=O)(CCC(F)(F)C(F)F)N(C)CC1CCN(C(=O)CC2CCC2C2CC2)CC1 89769,CCC(C(=O)NCc1n[nH]cc1C(N1CCC(C(=O)NC)C1)=O)OC 89770,CN1CCN(C(C2CC3(CCO2)CC3)=O)C(C(N2CCCC(C#N)C2)=O)C1 89771,C(=O)(C(C)(C)C1=CCN(C(c2cnc(OC)nc2)=O)C1)N1CCCC(CCC)C1 89772,CCCC(C(=O)NCCN(C1CCCC1)C(c1ccsc1)=O)OC 89773,Cc1cnc2cc(C(N3CCN(C(C4CC=CC4)=O)C(CO)C3)=O)ccn12 89774,C#Cc1ccc(Br)c(C(=O)NC(C)CN(C)C(C2(C)C=CCCC2)=O)c1 89775,C1(C(=O)O)CN(C(c2cnco2)=O)CC12CN(C(c1ccccc1O)=O)C2 89776,c1(CC(N2CCC(NC(C(C)C)=O)CC2)=O)c(F)c(F)c(F)c(F)c1F 89777,N1(C(C(C)CN(C)C)=O)CCN(C(C2(CC3CC3)CC2)=O)CCC1C 89778,c1(NC(=O)NCCCn2cnc(=N)[nH]2)ccc(N2CCOCC2)c(F)c1 89779,N1(C(C(=O)NCCCOC)NCC)CCC(NC(C)=O)C1.C(C)(C)(C)OC=O 89780,c1(C(N2CCN(C(CC=C)=O)CC2CC2CC2)=O)cc2ccc(F)cc2cn1 89781,CCC(CC)(CCNC(c1ccon1)=O)NC(=O)C(Cc1ccccc1)N(C)C 89782,C1(NC(CC(C)c2ccccc2)=O)CN(C(c2ccc(O)nc2Cl)=O)CC12CC2 89783,c1(OC)ccc(CNC2CCC(C(N3CC4CC3CN4C)=O)OC2)cc1OC 89784,C1(N(C)CC=CC(=O)N(CC)Cc2c(C)cnn2C)(OCC)CC(F)(F)C1 89785,CC(C(=O)N1CC(NC(=O)CNC=O)C(c2ccccc2)C1)C(F)F 89786,N1(C(CC(C)(C)C(F)F)=O)CCC2CCN(C(C3CNC(=O)N3)=O)C2C1 89787,c1(OC)cccc(C=CC(=O)NC2CC2NC(=O)CC(C)(C)C)c1 89788,C1(c2cccc(C)c2)CCCN1NC(=O)c1cnn(C2CCCCC2)c1C 89789,C(=O)(C(C)(C)c1cccs1)N(CCOCCNC(CSCC)=O)C 89790,C1(NC(=O)NCC=CCCOC)CC12C1CC3CC(C1)CC2C3 89791,C1(COC)CN(C(c2cc(O)ncn2)=O)CCN1C(=O)C(C(C)C)n1ccnc1 89792,CCC(COC)C(=O)N1CCCC(NC(=O)C=Cc2cncn2C)C1 89793,C1(n2cc(-c3cn(CC)nc3)nn2)CN(c2ccccc2)CCC12CCC2 89794,C(=O)(C(O)CCC(C)C)N1CCN(CC(C)NC(C2(C#C)CC(=O)C2)=O)CC1 89795,c1(OCC)cccc(NC(C2CCC2NC(c2cc(C)n(C)c2)=O)=O)c1 89796,c1(C(N(C(C)(C)CC(=O)Nc2cnccc2CO)C)=O)ccccc1O 89797,c1(N2CC(CNC(C3(C)CCNC3=O)=O)OCC2)cncc(C#N)n1 89798,c1(C(N(C)CCOCCCN(C)C(C2CCCC2O)=O)=O)cc2ccccn2c1 89799,C1(COC)CCCCN1C(=O)CC1CN(C(C2COCCO2)=O)C1 89800,N1(C(c2ccn(C(F)F)n2)=O)CCOC(C2CC2)C1 89801,c1(C(=O)OC)cccc(C(N2CC3(CC3)CC2CNC(=O)C=CSC)=O)c1C 89802,N1(C(c2cnn(CC)c2C)=O)CCCC(NC(=O)CC2(CO)CC2)C(F)C1 89803,c1(C(N2CCC(NC(c3c(C)ncnc3)=O)C2)=O)ccc(N)cc1C(C)(C)C 89804,N1(Cc2c(F)cc(OC)cc2F)CCCC12CCNC2=O 89805,N1(C(C2CN(Cc3cccs3)CCC2O)=O)CCc2ncncc2C1 89806,C(CN=c1cccc(S(=O)(=O)NC(CO)CCC2CC2)[nH]1)c1ccc(C)cc1 89807,Cc1c(C(=O)NCC(C)CN(C(=O)CC2CCC2)C)c(-c2ccccc2)cn1C 89808,c1(C(=O)NCC2C(CNC(C3(C)C(C)(C)C3)=O)C2)cc(O)cc(O)n1 89809,N1(CC)C(=O)NC(c2c(OC#N)ccnc2Cl)C(C(=O)Nc2ccccc2)=C1C 89810,C1(CN(C)C(C2CC(C(F)(F)F)C2)=O)CCCN(C(C2C3CC(=O)CC23)=O)C1 89811,C(=O)(C1CCCn2cncc21)NC(C(C)C)CNC(c1c(Cl)ccc(O)c1N)=O 89812,C#CCC(C)(CC)C(=O)N1CC(C(=O)NC(c2ccc(F)cc2)C)C(C)(C)C1 89813,C1(C(=O)NC2(CCNC(COCC)=O)CC2)Cc2ccc(Br)cc2C(=O)O1 89814,N1(C(C2OCCN(C(CCCOC)=O)C2)=O)CCC(C2CCC2)C1 89815,Cc1c(CC(N2CCC(CCNC(=O)C(C3CC3)C3CC3)C2C)=O)cnn1C 89816,C(C(C)N=c1ccc(C#N)n[nH]1)NC(Cc1c(C)nc[nH]1)=O 89817,N1(C(c2n(C)ncc2C#N)=O)CCC2(CCCN2C(=O)CCS(N)(=O)=O)C1 89818,C(CN=c1[nH]c(N(CCC(N)=O)C)nc2c1SCC2)(c1ccccc1F)OC 89819,O=C1CC(CC(=O)N(C2CCCC2)CCCNC(c2cccc(Cl)c2)=O)C(=O)N1 89820,C1(CNC(c2c(C)cc(C)o2)=O)CN(C(=O)CNC(=O)CC(C)C)CCC1(F)F 89821,N1(C(C2CC23CCCCC3)C(=O)NCC=C)CCCC2(CCCNC2=O)C1 89822,c1(CNCC(C)CF)ccc2nonc2c1 89823,c1(C(N(C2CCN(C(C3CC(O)C3)=O)C2)CC)=O)cnn(CC2CCCCC2)c1 89824,c1(C(=O)NC2C=CC(CNC(C=CCCC)=O)C2)c(C)cc(O)nc1C 89825,CC(O)(C(=O)NCC1CC2CN(C(=O)CCCc3ncco3)CC12)C(F)(F)F 89826,C1(C#N)(C(=O)NC2C(C)N(C(=O)CSc3cccnc3)CC2)CC12CCC2 89827,Cc1nnn(CC(=O)NC(C2(O)CN(C(=O)C(C)NC(N)=O)C2)C)n1 89828,c1(C(N(C)CC2CN(C(=O)CC3COC(=O)N3)CCO2)=O)ccc2[nH]ccc2n1 89829,c1(C(=O)NCC2N(C(c3n(CC)ccn3)=O)C3C(C2)C3)cccc(Cl)c1F 89830,C#Cc1ccccc1CC(=O)NCC1CC(CNC(C2C=CC=CC=C2)=O)CO1 89831,C(=O)(C1CCCc2sccc21)NC1CCC(CNC(c2ccc(N)cc2F)=O)C1 89832,n1(C(C(=O)NC2CCCN(C(C)=O)C2)C)cc2ccccc2n1 89833,N1(C(=O)OC(C)(C)C)CCCCC(NC(=O)NC(CO)C2CC2)C1 89834,C(=O)(C1Cc2ccc(Cl)cc21)N(CCCN(c1ncnc2c1CCC2)C)C 89835,C(=O)(C1=CCC(F)(F)CC1)N(C(C1CC(CCNC(=O)OC(C)(C)C)C1)=O)C1CC1 89836,c1(CC(N2CCCC2CNCC23C=CC(CC2)C3)=O)cccc(O)c1F 89837,c1(C(N(CCNC(C2(CCOC)CCCC2)=O)C)=O)ccc(-n2ccnc2)cn1 89838,C1(C)(C(=O)NCCN(C(C(C)Cc2cccnc2)=O)CC(C)O)CCCN(C)C1 89839,N1(Cc2cc(OC)cc(C)c2)CCC2CN(c3nccc(C)n3)CC2C1 89840,c1(C(N2CCCC(C3N(C(COC)=O)CCC3)C2)=O)cncn(C)c1=O 89841,C(C)(CNC(=O)CC1CCSCC1)(CO)NC(C(C)=CC)=O 89842,C#Cc1cccc(C(N2CCC(O)(C(C)NC(=O)CCC3CCCOC3)C2)=O)c1 89843,Cn1cnnc1CC(N1CC(CO)(NC(c2ccc(C3CCOC3)s2)=O)C1)=O 89844,c1(NC(C(=O)Nc2c(C)nc3sccn32)=O)cccc2nc(O)oc12 89845,C(=O)(C1=CCN(C(C2C(C)C2C)=O)C1)Nc1cn(CC#C)nc1 89846,N1(C(=O)CC2CC3(CC3)C2)CC(C2CN(C(C3C4(CC4)C34CC4)=O)C2)C1 89847,N1(C(CS(=O)(=O)N(CC)CC)=O)CCCC2(NC(=O)CN3CC(C)C3)CCCC12 89848,C1(C(N(C2CCN(C(C3C(C(C)C)CCO3)=O)CC2)C)=O)CC2(CCCC2)CO1 89849,c1(CC)cnccc1C(=O)NC12CC(C(N3CCCCC3CCN(C)C)=O)(C1)C2 89850,C(=O)(N=c1ccnc(C(C)(C)C)[nH]1)C1CCN(Cc2n(C)cnc2)C1 89851,C1(C(N2C(C(=O)NCC3(O)CC3)(CC)CCC2)=O)C2CCC(C2)C1C 89852,CC(CC1CCC1)C(=O)N(CCC(N1CC(O)(C(N)=O)C1)=O)CC1CC1 89853,C=CC1(C(=O)NC(CC)CC(F)(F)F)CCN(C(c2cc(C)ccc2O)=O)C1 89854,Nc1cc(C(N2CCCC2CNC(C2CCCC23CC3)=O)=O)cnc1Cl 89855,Cc1cnn(C)c1CC(=O)NC(CC(F)(F)F)c1ccccc1 89856,c1(C(=O)NCC2C3CN(C(c4c(NC)c(C)cs4)=O)CC32)cccc2c[nH]nc12 89857,CCCC(C(=O)NCC1(F)CN(C(=O)CCC23CCC(CC2)C3)C1)OCC.CCC 89858,N1(C(C23C(C)OC(CO)(C2)C3)=O)CCC(NC(=O)C(F)(F)CO)C(C)(C)C1 89859,c1(OC(C)C(F)F)ccc(-n2cc(-c3cccc(C(F)(F)F)n3)nn2)cc1 89860,c1(C(=O)NC(CC(C)NC(C(F)=C(C)C)=O)C)n[nH]c2ccccc12 89861,C=C(C)c1ccccc1NC(C1CC1CNC(C1CCC1)=O)=O 89862,n1(CC)cc(Cl)c(C(=O)NC2CCCC(N(C(=O)Cc3ccns3)C)C2)n1 89863,N12CCC3(CC1)CC3C2.N1(C(c2nc(SC)sc2)=O)CCCC(C(N)=O)C1 89864,c1(C(N2CC(C)C(NC(c3cc(N)c(Cl)cn3)=O)C2)=O)ccc(C2CC2)nc1O 89865,O=C1NCC2CN(C(C3(CCNC(=O)CC4CC(F)(F)C4)CCCC3)=O)CCC12 89866,c1(C(N(C(CC)C(=O)NC2CN(C)NC2=O)C)=O)ccc2c[nH]nc2c1 89867,C1(CC(N2CCC(CC(C)NC(=O)CSCCN(C)C)CC2)=O)CCC(C)(C)CO1 89868,O=C1Nc2cc(Br)cnc2N2CCN(Cc3ccc(-c4ccc(F)cc4)s3)CC12 89869,CN1C(=O)CN(CC(=O)NCCC2(NC(=O)Cc3ccsn3)CCC2)C1=O 89870,C1(C(N2CC(NC(c3c(Cl)cn(CCC)n3)=O)C2)=O)CC2CCCC(C1)C2 89871,c1(C(N2CC(C3(NC(c4c(SC)ccs4)=O)CC3)C2)=O)c(C)ccc(C)c1O 89872,n1(CC(=O)OCC=C(C)C)cc(N(C(=O)CSC(C)(C)C)CC)c(O)nc1=O 89873,c1(N(C2CCN(C(c3c(OC)ccs3)=O)C2)CCO)nc(C)cc(C#N)n1 89874,c1(C(=O)NCCN(C(=O)C(C)(C)n2cnnn2)CC)cccc(S(C)(=O)=NC)c1 89875,c1(OC)nc(NC(C2C3CN(C(c4cc(Br)ncc4Br)=O)CC23)=O)cc(O)n1 89876,C1(CNC(c2cc(C)n(C3CC3)c2C)=O)CN(C(=O)C(N)=O)CCC12CCC2 89877,n1(-c2c(OC)ccs2)cc(S(=O)(=O)NC(c2cc(C)ccc2C(F)(F)F)=O)cn1 89878,Cn1nc(C(=O)NCC=CCNC(=O)CCC2CCOC2)cc1-c1ccc(Cl)cc1 89879,N1(C(CCC2N(C(C(C=C)OC)=O)CCCC2)=O)CCC(C)(CC)CC1 89880,C(=O)(C#CC1CCOC1)NC1CC(CNC(C(C(CC)C)NS(C)(=O)=O)=O)C1 89881,C1(CNC(C(CCC)(C)O)=O)CN(C(C2(C(=O)NC)CCC2)=O)CC(C)(C)C1 89882,C=CC1(CC(=O)NC(C)C2CC2)CN(C(=O)C(C)NC(=O)OC2CCC2)C1 89883,C12CCCCN(C1)C(=O)CC2.CC1OCCC1N(CCO)C(C1CC1C(F)F)=O 89884,N1(C(C(N2C(CCC)CCSC2)=O)C)CCC(C)CC1 89885,CCCCC(C)(F)C(=O)NC1CC(C(=O)NC2C(=O)OC3CCCC23)CC1O 89886,CCCC(C)C(=O)NCC1CCCC1NC(c1coc(C)n1)=O 89887,CC1C2C(CCN2C(=O)CC2(O)CCOCC2)CN1C(=O)C=CCF 89888,c1(CC(N2C(CNC(=O)CC3CNC(=O)O3)CCC2)=O)c[nH]c2cccnc12 89889,N1(C(C(CCCC)CC)=O)CC2(C1)CN(C(=O)C(CC)CCOC)CCO2 89890,CC(O)(CC(=O)N1CC2CC1CC2NC(C12CC(F)(C1)C2)=O)CC(=O)O 89891,c1(C(N(C(CCNC(CCC(CC)C)=O)C)C)=O)ccc(=NCCOC)[nH]c1 89892,Cc1cc(N(C(=O)CCCCCNC(c2cnc3n2CCC3)=O)C)cc(F)c1 89893,C1(CCC)(NC(=O)CC)CCCN(C(C2CCC(OC(F)F)CC2)=O)C1 89894,Cc1cc(Br)ccc1CC(N1CCOC(C(C)NC(=O)C2=C(Cl)CC2)C1)=O 89895,C(=O)(CCCC(=O)N(CC(C)NC(c1ccc(OC)c(Br)n1)=O)C)OC 89896,C1(CN(C(C(CC)n2cccn2)=O)C)CCCN(C(c2oncc2C)=O)C1 89897,c1(C(=O)NCCN(C(C2N(S(C)(=O)=O)CC2)=O)C2CC2)ccc2[nH]nc(Cl)c2c1 89898,C(=O)(C1=C(Cl)CCOC1)NCC1CCC(NC(=O)Cn2nc(O)ccc2=O)CC1 89899,c1(C(N2CCN(C(CNC(C(C)SC)=O)=O)CC2)=O)ccc(Cl)c(F)c1O 89900,C1(C(N(C)CCNC(=O)C2=CCC2)=O)CC(C)(C)CCO1 89901,C12(CNC(c3cncc(C)n3)=O)CCC1CN(C(=O)CC1CNC(=O)C1)C2 89902,c1(CC)cc(C#N)c(NC(C2(F)CN(Cc3cnccn3)C2)=O)s1 89903,CCC(C(=O)N(C1CN(C(=O)Cc2sc(C)cc2C)CC1(C)C)C)C(C)C 89904,C(C(N=[N+]=[N-])C(=O)NCC1CC(C)N(C(=O)CCCC2CCOCC2)C1)OCC 89905,O(NC(=O)C(C)N(C(=O)Cc1ccccn1)C1CC1)CC(CC)C 89906,c1(C(N(C2CN(C(C3CC3c3cccnc3)=O)C2)C)=O)cccc(O)c1 89907,N1(C(c2c(Br)ccc(N)c2)=O)CCC(NC(C2CCOC2)=O)C2(CCC2)C1 89908,N1(C(C(CC)SC)=O)CCC(CNC(=O)C=Cc2cccc(OC)c2)C(C)C1 89909,CC1(CNC(=O)C2=COCCO2)CC(F)(F)CN1C(c1cn2ccnc2cn1)=O 89910,CS(=O)(=O)c1cc([N+](=O)[O-])ccc1NCC1CCCC1NC(C1(C(N)=O)CC1)=O 89911,N1(C(CCC2CCCC(=O)N2)=O)CC2CCC(C1)N2C(C1C=CCC1)=O 89912,CC1=C(C(=O)NCCCN(C(=O)C(C)Cc2ccnn2C)C(C)C)COCC1 89913,CC(C)(C)CCC(=O)N1CC(C)(C)CC1CNC(=O)Cn1ccc(C2CC2)n1 89914,N1(C(CCc2c(C)cccn2)=O)CCCN(C(C23CCC(C2)OC3C)=O)CC1 89915,N1(C(c2ccc(OC)s2)=O)Cc2ccccc2C(NC(c2ccc(Cl)cc2)=O)C1 89916,N1(c2n(CCOCC=C)c(C3CC4(C3)OCCO4)nn2)CCc2c(Cl)cccc21 89917,N1(C(C2CCCN(C(C(C(=O)OC)(C)F)=O)CC2)=O)CCC(C)C(C)(C)C1 89918,c1(OC)ncc(C)cc1-c1ccc(CC(=O)NC2CONC2=O)cc1F 89919,CN1CCC(C(=O)NCC=CCNC(=O)CCC(=O)c2ccccc2)CC1=O 89920,c1(C(=O)NC2CC(F)(CNC(CC3(C)CC3F)=O)C2)ncn2ccccc12 89921,N1(C(c2cn(C)c(O)n2)=O)CC2(CCC(NC(=O)CN3CCOCC3=O)CC2)C1 89922,N1(C(C2C(OC)(OC)CC2)=O)CC(C)(C(N2CC(F)CC2CO)=O)CC1(C)C 89923,Cc1cncc(C(N2CC(C(C)NC(=O)C(C3CC3)C3CC3)C2)=O)n1 89924,CC1CC2(CO1)CC(Nc1nccc(N3CC4CC3CS4)n1)C2 89925,CCC(CC)=CC(=O)NC1(CC(=O)N(C(C)C(F)F)C)CCC1 89926,C#CC1CCCC(NC(C2(CNC(c3cnn(C4CC4)c3)=O)CCC2)=O)C1 89927,C(=O)(C(C)S(N)(=O)=O)NC1(CNC(c2cnc(OC)s2)=O)CCOC1 89928,C(CCC(C)(C)C(=O)NOC(CC(C)C)C(=O)N1CC(N=[N+]=[N-])C1)OC 89929,C1(C(=O)NCC(CNC(C2(C)CC(C)C2)=O)F)C2CCC3C(C2)CC13 89930,Cc1nc(Cl)ncc1CNCCC(N1CCCCCC1)=O 89931,N(C1CC2CCCc3cccc1c32)C(C=Cc1ccc(C(N(C)C)=O)cc1)=O 89932,C1(NC(C2(CC#C)CCCO2)=O)CC2(CCN(C(=O)CC3CCCC34CC4)C2)C1 89933,c1(C(=O)NCC2C(C)CCN(C(C3(C)CC(=C)C3)=O)C2)cnc2ccccc2c1 89934,c1(CNC2N(C(=O)NCc3ccc(C)cc3)C(C)CC2)cc(C)ccc1O 89935,C1(N(C(CC(C)O)=O)C)CCCCC1N(C)C(c1cc(CNC2CC2)ccn1)=O 89936,c1(C(=O)NCCCCNC(C2(C3CC3)CCC2)=O)cnc2cc[nH]c2c1 89937,c1(C(CC)C)nc(N2CCC(NC(=O)COCC(F)F)C(C)C2)cc(C)n1 89938,Cc1nscc1CC(N1CC(CCCCNC(c2cc(Br)n[nH]2)=O)C1)=O 89939,C=CC(C)(C)CC(=O)N1CCOCC1CN(C)C(C1(C)CCN(C(C)=O)C1)=O 89940,c1(COC)nc(=NC(C)CN(C)C(c2ccc(OCCO)cc2C)=O)s[nH]1 89941,c1(C(=O)NC2CN(C(Cc3c(C)ocn3)=O)C(C)C2)cc(N)ccc1C(F)(F)F 89942,C1(CC)C(C(=O)NCc2ccsc2C)CCN1C(=O)Cc1cc[nH]c1 89943,c1(OCCC(=O)NC2CC(C)N(C(C3CC34CC4)=O)C2)ccc(Cl)cc1Br 89944,c1(SCC)ccc(C(=O)NC(C)(CNC(C2OCC2(C)C)=O)C(C)C)cn1 89945,c1(-n2c(C(O)C(F)(F)F)nc(CC(C)OC)n2)cccc2nc[nH]c12 89946,CC1(CO)CCN(C(c2sccc2Nc2ncc3ccsc3n2)=O)CC1O 89947,c1(C(N2CC(CNC(c3c[nH]cc3Br)=O)OCCC2)=O)cc2n(n1)CCCC2O 89948,CC1CN(C(c2ccncc2)=O)CC(C)C1NC(c1cnns1)=O 89949,c1(C(=O)NCC(C)N(C(C(C(C)C)NC(=O)OC)=O)C)cc(Cl)cc(Cl)c1 89950,c1(OCCn2c(N(CC)Cc3cscc3Cl)nnn2)cnn(C)c1C 89951,C#CCC(O)C(=O)N1CC(C)(C(=O)N(C)Cc2cc(=O)cc[nH]2)C1 89952,C1(CNC(C=CCOC)=O)CN(C)CCN1C(=O)CCCn1cnc(C#N)n1 89953,Cc1ncc2n1CCC(C(=O)NCC1CCCN(S(C)(=O)=O)C1)C2 89954,Cn1ncc(C(N2CCC(C(F)C(N)=O)CC2)C(=O)NCCCC2CC2)c1Br 89955,C1(C(N(CC(F)F)CCC)=O)CCCC2(CCC2)O1 89956,N1(C(C)C(N2C3CCCC2CC3)=O)CCC2CC(N(C3CCCC3)C)C2C1 89957,C1(C(=O)NCC2CCC(NC(c3c(C)nns3)=O)C2)CC(c2ccncc2)=NO1 89958,c1(CCN=C(NC(C)C)NCC2C3COCC23)cc(Cl)c2c(c1)OCCO2 89959,c1(OC)ncc(CN2CCCC(C(=O)N(CCO)CCO)CC2)cc1Br 89960,C1(C(=O)NCCCCC2CN(C(=O)CNc3ccccc3)C2)CC1C1CCCC1 89961,Cc1cc(C(=O)NCc2c[nH]nc2C(=O)NCC(N2CCCCC2)C)nc(C)c1 89962,C(=O)(CC(C)CC(C)C)NC(CCC)CC(=O)NCC1(OC)CCCC1 89963,c1(C(N(C2(CNC(C3CC(=O)N(C(C)C4CC4)C3)=O)CC2)C)=O)cccnc1N 89964,CC1CC(NC(=O)CC2CSCCS2)CN(C(=O)CCN(C2CCCCC2)C)C1 89965,c1(OCC)ccc(F)c(C(N2CC(Cc3cn(CCSC)nn3)C2)=O)c1F 89966,C#CC1(C(=O)NC2(C=C)CCCC2)CN(C(C2CCCN2C=O)=O)C1 89967,c1(C(N2C(CNC(CCSC)=O)CC2)=O)ccc(NCc2nc[nH]n2)cc1 89968,C1(N(C(=O)Cn2ccnn2)CCOC)CCN(C(=O)C(F)C2CCCC2)CC1 89969,C1(C)(C(N(CC(C)NC(Cc2ccc(C)cc2)=O)C)=O)CCCS1(=O)=O 89970,C(=O)(CC(C)(C)CNC(=O)CCc1ccco1)NCC(CC(C)C)O 89971,c1(C(=O)NCC2C(NC(C3(N=[N+]=[N-])CC3)=O)CCC2)c(Cl)ccc2c[nH]nc12 89972,c1(C(=O)NCCOC2CN(C(=O)C3=C(Cl)CC3)C2)cc2n(n1)CCO2 89973,C1(CNC(C(C)=CC)=O)(NC(=O)COC)CCC(F)(F)CC1 89974,c1(CC)nc(C)c(C(=O)NC(CCF)C(=O)NC(C)CCN(C)C)o1 89975,c1(C(N2CC(F)(CNC(c3n(CC)ncc3)=O)C2)=O)cn2ccn(C)c(=O)c2n1 89976,N1(C(CNC(N)=O)=O)CCCC2CCN(C(c3cn4c(n3)CCC4)=O)CC12 89977,C1(CNC(C(C)n2cccn2)=O)CCCC2(CN(c3ncccc3[N+](=O)[O-])C2)O1 89978,Cc1cc(F)c2cc(C(=O)NCCCN(C(=O)CC3CC=CC3)C)[nH]c2c1 89979,C(CN=c1cc[nH]c(C(N)=O)n1)(c1ccc(F)cc1)NC(C)=O 89980,c1(C(=O)NC2C(CNC(C(C)(C)F)=O)CC2)ccc(Br)c(N)n1 89981,c1(C(=O)NC2C=CC(CNC(c3n(C)ncc3Cl)=O)C2)ncn2c1CCCCC2 89982,C1(NC(c2c(COC)ncs2)=O)(CO)CCN(C(C2CCCC2)=O)C1 89983,CCCCC(O)C(=O)N1CCN(C(c2cc(I)ccc2Br)=O)CC1 89984,C(C(C(=O)NC(C)C(=O)OC)N1CCCC1CC)(N1CCC(N(C)C)C1)OCC 89985,C=CCC(C)(C)CC(=O)N1CC(CNC(C2CCN(C)C2=O)=O)OC(C)(C)C1 89986,Cc1ccccc1Cn1cc(CNC(c2cccnc2O)=O)nn1 89987,CCCCCC(O)CC(=O)NCC1CC1CNC(c1ccc(Cl)cc1O)=O 89988,CCC(C)CC(C(=O)NCC(C)(F)C(C)C)NC(=O)CCOCC1CC1 89989,Cc1cnc(C(=O)NCC(c2ccccc2)NC(C2COC(=O)O2)C2CC2)nc1 89990,N1(C(C(=O)N(C)C)=O)CCCC(C2CCN(C(C3(O)CCCCCC3)=O)CC2)C1 89991,C1(C(=O)NC(C(=O)N(C)CC)C)CCN(C(=O)c2c[nH]c(=N)c(C)c2)O1 89992,c1(C(NNC(=O)C2N(CC)CSC2)=O)nc2ccccc2[nH]1 89993,C1(N(C(CN(C(=O)OC)C)=O)C)CC2CCC(C1)N2C(c1c[nH]nc1[N+](=O)[O-])=O 89994,c1(C(=O)NCC(CC(C)C)NC(=O)CC(C)F)cn2c(n1)CCC2 89995,C1(NC(c2c(CC)nns2)=O)CC2CN(C(=O)C(N3CSCSC3)C)CC2C1 89996,N1(C(COC)=O)CCC2(CC1)CC(NC(C13COCC1C3(F)F)=O)C2 89997,c1(C(=O)OCC)cnc(NC(c2sccc2NCc2ccc(F)cc2)=O)c(Br)c1 89998,C1(O)(CC#C)CC(C(=O)NCC2CCN(C(c3occc3C3CC3)=O)C2)C1 89999,C1(NC(CCCC(=C)C)=O)C(C)CN(C(c2cccc([N+](=O)[O-])c2)=O)CC1C 90000,c1(NCc2cccc(OCC)c2OC)c(C)ccn2ncnc12 90001,N1(C(C2(SC)CCC2)=O)CCC(c2cn(CCCOCc3ccccc3)nn2)C1 90002,Cc1nc(C(=O)NC2CN(C(c3ccc(Cl)cn3)=O)CCC2C)c2ccccn12 90003,CCCCCCC(C)CC(=O)NCCN(C(C1CCC2CC2CC1)=O)CC1CC1 90004,C(C(F)(F)C(F)(F)F)OCCC(=O)NCC(C1CC1)NC(=O)C(F)OC(=N)O 90005,C=CCC(CC)C(=O)NC1(C)CCN(C(c2c(C)cccc2O)=O)C1 90006,c1(C(N(C2CCCN(C(C=Cc3occ(C)n3)=O)C2)C)=O)cccc(C)c1N 90007,C1(C(=O)NC(CNC(c2nc(O)c(C)s2)=O)CO)(COC)CCCCO1 90008,C1(C(=O)NC2C(NC(C(C)(C)OC)=O)CCCC2)CC2C=CC1CCC2 90009,Cc1ccc(SCC(=O)NCC(C)(O)CNC(c2ccccc2CO)=O)c(C)c1 90010,c1(C(N(CC(N2CCN(C(C=CC=CC)=O)CC2)=O)C)=O)ncc([N+](=O)[O-])n1C 90011,C(=O)(CC(CC)C(=O)OC(C)(C)C)NCC(CNC(C(CC=C)(C)C)=O)OC 90012,N1(C(C(C)(Cl)Cl)=O)CC2(C)CN(C(=O)C(O)C3CCC3)CC2(C)C1 90013,O=C(N1CCS(=O)(=O)CCN1)C1(COC(F)F)CCCC1 90014,n1(CC)cc(CN(C(=O)C(CC2CCCC2)NC(C2CCOC2)=O)C)cn1 90015,c1(C(N2C(CNC(c3ccccn3)=O)CC2)=O)ccc(Br)c(F)n1 90016,c1(C(=O)NC(C)CN(C(=O)CSC(F)(F)F)C)cccc(N2CCCC2)n1 90017,c1(OC)ccc(NC(=O)C(C(C)C)NCC(Cc2ccccc2)C(C)C)c(OC)c1 90018,c1(C(=O)NCC(N2CCCN(C(c3cccs3)=O)CC2)=O)cc2cccnc2o1 90019,C1(N(C)C(C2CC(n3ccnc3)C2)=O)CCCN(C(=O)Cc2ccc(Cl)s2)C1 90020,C1(CCNC(c2cnc(CC(C)C)[nH]2)=O)CCCN(C(=O)CCCC#N)CC1 90021,C(C(C)(C)CNC(C1CC1C)=O)N(C(=O)CNC(=O)NC)CC 90022,Cc1cc(C(=O)NCC2(C)CCN(C(c3cc(Cl)c(C)cn3)=O)C2)c(C)nc1C 90023,c1(C(N(CCC(C)NC(c2cc(CO)ccn2)=O)C)=O)cncc(Cl)c1 90024,Cc1cc(CC(N2CCC(OCCN(C(=O)C(F)(F)CF)CO)C2)=O)ccc1O 90025,c1(C(=O)NC2CC(NC(C3C(CC)CCC3)=O)C2)cnn(C)c1Br 90026,c1(OC)ccnc(O)c1C(=O)NC1CC2(C1)CC2NC(C1C2CCCC12)=O 90027,C#CC1(C(=O)NCCCCCC(=O)OC)CCN(C(=O)Cc2cc[nH]n2)CC1 90028,n1(C(F)F)cccc1C(c1cnccn1)c1nnnn1C.C1(CN)CCCS1 90029,c1(CCCC(=O)NCC2CN(C(CC3(C)CC3(F)Cl)=O)C2)c[nH]c2ccccc12 90030,C(=O)(C(C)(C)CCCNC(=O)C(=O)NC(C)C)Nc1ccc(OC)cc1 90031,c1(C(N2CC(C(=O)NC3(C)CC(C)(C)C3)C(F)C2)=O)ccnc2[nH]cnc12 90032,c1(CCCC(=O)N(C)CCNC(C2(C)CC2(F)F)=O)nc2ccccc2[nH]1 90033,Cn1ccc2sc(C(=O)NC3CC(NC(=O)C=CCN4CCCC4)C3)cc12 90034,N1(C(c2c(N(C)C)nccc2)=O)CC2(CCN2C(C2(C)CCCC2)=O)C1 90035,CCCCCCC(C)(CC)C(=O)NCC1CN(C(c2sccc2Cl)=O)CC1(C)C 90036,Cc1nc(CO)sc1C(=O)NC1COCC1CNC(C1CC(=O)N(C)C1)=O 90037,C1(NC(CN(C)C)=O)COC2(CCN(C(=O)C(N)CN)CC2)C1 90038,N1(C(C2(C)CCC(C)CC2)=O)CCCC2CN(C(C3CC(=O)C3)=O)CCC12 90039,c1(N2CC3(CCN(C)C3)OCC2)nc2c(c(=NCC3CCCN3C)[nH]1)CCC2 90040,C(=O)(C1=CCCOCC1)NC(C1(O)CCN(C(c2c(OC)n[nH]c2)=O)C1)C 90041,C1(C(C)NC(C2(C(=O)NC)CCC2)=O)CCN(C(=O)CCc2nncs2)C1 90042,N1(C(C2(CC(=O)OC)CC2)=O)CCC(O)(C(C)NC(=O)C(C2CCCCC2)F)C1 90043,c1(CC)nc(C#N)cc(=NCC2C(C)CCCN2C(c2cnnc(O)c2)=O)[nH]1 90044,C12CCCN(C1)C2=O.c1(CNC(=O)Nc2cnsn2)nc(C(F)(F)F)cs1 90045,N1(C(C2(SC)CC2)=O)CC(NC(=O)C(CC)c2ccccc2)CC2(CC2)C1 90046,N1(C(C(=O)NC)C)CC(O)(C(C)NC(c2cn(CCC(C)C)nn2)=O)C1 90047,n1(CC)ccc(C(N2CCC(NC(=O)C(C)N3CC(C)C3)C2C)=O)c1C 90048,Cc1cc(C(C)C(N2CCC(Cn3cc(CCCO)nn3)C2)=O)c(C)o1 90049,CCCCC(CC)CC(=O)NCCCOCCNC(=O)C=Cc1cscn1 90050,C1(CC(N2CC(C)(NC(CC(CC)CC)=O)C2)=O)Cc2ccc(Cl)cc2C1=O 90051,c1(OCC)c(F)ccc(C)c1NC(C1(CNCc2c(NC)cccc2)CC1)=O 90052,C12(CCNC(CCC=C)=O)CCC1CN(C(c1csc(O)n1)=O)C2 90053,CCCCCCCC(=O)NC1CC(NC(=O)C(C)(C)C2CCCO2)CC1O 90054,CC1CC(=O)NCC1C(=O)NCC=C1CCN(C(C2(CCN(C)C)CC2)=O)CC1 90055,CC(O)(C(=O)NCC1CCC(NC(=O)Cc2nccs2)C1)C1CCC1 90056,N1(C(C23CSC(C2)C3)=O)CCC2(CCCN(C(=O)C3=CCCC3)C2)CC1 90057,C1(C)(CNC(C2(CCN(C)C)CC2)=O)CN(C(=O)CC2CCCO2)CCO1 90058,c1(CC(N2C(CNC(Cc3c(C)n[nH]c3C)=O)COCC2)=O)ccc(C#N)cc1 90059,CN1CC=C(CC(=O)N2CC3(CCC3NC(c3csc(Cl)c3)=O)C2)CC1 90060,N1(C(c2ccc(C)c(O)c2)=O)CC2CC(C(=O)NCCN3CC=CC3)CC2C1 90061,N1(C(c2c(CCC)occ2)=O)CCC2(CCCC2NC(C2CC=CC2)=O)CC1 90062,n1(CC)cc(C(=O)NCC2CC(COC)CN2C(=O)CC2CCC(=O)C2)c(C)n1 90063,C1(NC(CC(=O)OCC)=O)CC2CN(C(c3n[nH]cc3[N+](=O)[O-])=O)CCN2C1=O 90064,C=Cc1ccc(C(N2CC3CC2CC3NC(=O)CNc2ccc(F)cc2)=O)cc1 90065,N1(C(CCC2CCN(C)CC2)=O)CCC(NC(C2CC3CC3C2)=O)C(C(N)=O)C1 90066,C1(CC)(CC)CC(NC(=O)C(C)C(C)C)CN1C(c1cnc(OC(C)C)nc1)=O 90067,C=CC1(CC(=O)NC(C)(CNC(=O)Cc2cncs2)C2CC2)CC1 90068,N#CC1(C(N2CCN(C(c3ccc(F)s3)=O)C(CC(F)(F)F)C2)=O)CCOCC1 90069,c1(C(=O)NC(CNC(C(CC)(C)CO)=O)CO)ccc2c(c1)OCO2 90070,N1(C(c2c(OC)nccc2)=O)CC(C(=O)N(C2(C)CC2)C)OC(C)C1 90071,c1(CC(CN(C(=O)NCC(COC)F)C2CC2)CO)ccc2ccccc2c1 90072,Cc1cccc(Cl)c1CC(N1CCC(C(=O)O)C(C(F)(F)F)C1)=O 90073,C1(CNC(C(=O)N(CC=C(C)C)C2CC2)=O)CC(CO)CO1 90074,c1(CC)ccc(C(=O)NC(CNC(=O)CCc2cnn(C)c2)CC)cc1Cl 90075,c1(OC)cnccc1C(=O)NCCc1n[nH]cc1C(=O)NCC(C)(O)CCO 90076,c1(C(N2CCC(C)N(C(=O)CCCN(C)C)CC2)=O)noc2ccc(Cl)cc12 90077,N1(C(c2c(CC)c[nH]c2)=O)CC2CCCCC2(CNC(=O)CSCC(F)(F)F)C1 90078,C1(NC(c2csc(-c3cn[nH]c3)n2)=O)CN(C(c2cc(Cl)no2)=O)C2(CCC2)C1 90079,CC1CC(CNC(=O)CCC2CC2)CN(C(C2C3COCC23)=O)C1 90080,N1(C(CCNC(C)=O)=O)CC(CN(C(=O)CC2CC=CCC2)C)C2(CC2)C1 90081,C1(C(=O)NCCN(CC(C)O)C(c2cnsn2)=O)CCn2c(O)nnc2C1 90082,C1(NC(c2n(C)ccn2)=O)CCN(C(C2OCC2(C)C)=O)C12CCC2 90083,CC(F)(F)CC(=O)NCc1ccoc1C(=O)NCc1ncsn1 90084,C1(NC(C(C)=C2CC2)=O)CCC(CNC(=O)C(C)Cc2cnn(C)c2)C1 90085,c1(C(=O)NC(C2(n3cc(C(CC)CC)nn3)CC2)=O)c(Br)c(C)nn1C(C)(C)C 90086,C1(CC(=O)NC2CCOCC2NC(C2CC3(CCC3)C2)=O)CCC(=O)NC1 90087,C#CCC(C)(CC)C(=O)NC1CCN(C(=O)Cc2ccc(O)c(C)c2)CC(O)C1 90088,N1(C(CCOCC(C)C)=O)CCCC(C2(NC(C3CCNC3=O)=O)CC2)C1 90089,S(=O)(=O)(c1ccc(=NCC2CCCCCC2(F)F)[nH]c1)NCC(C)F 90090,c1(C(N2CC(C(=O)NCC(C)(C)C3CC3)(CC)C2)=O)cc(C)ncc1C 90091,c1(C(=O)NCC2N(C(CSCCC)=O)CC(F)C2)c(C)cc(OC)cc1F 90092,N1(C(C(c2ccccc2)OC)=O)CC(NC(c2cc(C)cc(C)c2)=O)CC(F)C1 90093,CCC(C(=O)N(C)CCC1CCN(C(c2snc(O)c2Cl)=O)CC1)C(C)C 90094,c1(OC(CC)CNCC2CCC(c3nnc(C(C)(C)C)o3)CC2)ccccc1Cl 90095,N1(C(Cc2c(C)cc(C)s2)=O)CCC2CN(C(=O)C=CS(C)=O)CCC12 90096,CC1Cn2nc(C(N3CC(CNC(C4CCCC(F)(F)C4)=O)C3)=O)cc2C(=O)N1 90097,c1(C(=O)NC2CC(NC(CNS(C)(=O)=O)=O)C2)cccc(-c2ccccc2)c1O 90098,N1(C(C2(C)CCCN(S(CC(C)C)(=O)=O)C2)=O)C2CCC1CC(CO)C2 90099,N1(C(C(C)n2ccnn2)=O)C2CCC(C2)C1C(=O)NCC1(F)CCOCC1 90100,C(C(C(=O)NC(C)C)N1CCCC(c2ncc(C)s2)C1)(C1CC1)OC 90101,N1(C(C(C)OCC#C)=O)CCN(C(=O)C(C)OCC2(c3ccccc3)CC2)CC1 90102,N1(C(CN2CCN(CC)CC2)=O)CCN(C(=O)Cc2cccn2C)CC1CF 90103,C1(NC(C=CC(C)C)=O)CCCN(C(=O)CC2(C)CC2(F)F)CC1 90104,N1(C(c2cc(CNC(c3[nH]cc(C)c3)=O)sc2)=O)CCC(C)(N(C)C)C1 90105,C1(CNC(Cc2c(C)nsc2)=O)CC2(C1)CN(C(C1CCCN1C)=O)C2 90106,c1(C(N2CCC(C)(NC(C3CCC(CC)C3)=O)CC2)=O)[nH]nc2c1CCC2(C)C 90107,C1(C(=O)NC2CC(CNCc3cnc(C(C)(C)C)o3)C2)Cc2ccccc2N1 90108,c1(CN2CC(C#N)N(C(c3ccccc3S)=O)CC2)ccc(F)c2ccoc12 90109,C(=O)(C(O)CCCNC(=O)CC1CCOCC1)N1CCN(CC=C)CC1 90110,Cc1cscc1NC(C1CCC(CNC(=O)CCc2cnn(C)c2)C1)=O 90111,C1(NC(CC(C)c2ccncc2)=O)CN(C(=O)CSc2nncs2)CC1C 90112,N1(C(CSCCC)=O)CCN(C(=O)C(O)CC(N)=O)C(C(C)(C)C)C1 90113,c1(C(N2C(=O)CC(COC(CC(C)(C)O)=O)C2)=O)cc(C#N)c(O)nc1N 90114,c1(C(CC)C)ccc(=NCCCOCCc2ccccc2)[nH]n1 90115,C(=O)(CCCC(CC)NC(C1CC(C#N)(OC)C1)=O)NC1(C=C)CCCC1 90116,c1(C(N2C(CNC(C3(CCOC)CC3)=O)CC2)=O)cc(C)c2c(c1)CCC2 90117,CN1CCN(C(C2CC23CCCCC3)=O)C(C(=O)NCC2CCNC(=O)C2)C1 90118,Cc1cn2cc(C(=O)NCCOCCNC(c3ccn4ccnc4c3)=O)nc2s1 90119,N1(C(C(c2cccc(OC)c2)C)=O)CC2(CC(NC(=O)CCC(C)OC)C2)C1 90120,c1(C(=O)OC)nc(NC2C3CC2CN(C(c2ccccc2)=O)C3)cnc1C 90121,N1(C(c2c(C)noc2)=O)CCCC(C(N2CC=CC2CN(C)C)=O)C1 90122,c1(OC)nn(C)cc1C(=O)NCC1(NC(=O)C=CS(C)=O)CCOC1 90123,Cc1c(CC(N2CCOCC(C)C2)=O)sc2ccccc12 90124,C1(C)(CNCC(C2CCOCC2)NC(C2CC(C(=O)OC)C2)=O)CCCCCC1 90125,C(=O)(CC(C)CNC(C1CCS(=O)CC1)=O)N(C(C#C)C1CCC1)C 90126,c1(NCC2N(C(c3cc(C4CC4)ncn3)=O)CCC2)c(F)cccc1[N+](=O)[O-] 90127,Cc1ccc(C(=O)NCC(O)CC(=O)NCc2nn(C)cc2CO)n1C 90128,N1(S(CC)(=O)=O)CCCC(C(N2CC3CC3(NC(=O)CCCCC3CC3)C2)=O)C1 90129,c1(C(N2CC3C(NC(C4C(C)C4C)=O)C(CC3)C2)=O)csc2c(Cl)cccc12 90130,c1(NC(=O)CCc2cccc(F)c2O)ccc(-c2ccc(Cl)cc2CO)cc1F 90131,C(=O)(C1=NOC(C)(C)C1)N1C(C(=O)NC(C#C)CC2CCC2)CSCC1 90132,C1(NC(C(CC#C)(C)NC(=O)CC2(O)CCCCC2)=O)CCc2n[nH]cc2C1 90133,N1(C(CC2C3CN(C(c4n(CC)ccc4)=O)CC32)=O)CC=CC12CCOCC2 90134,C#CC1CCCCN1C(=O)CSCCNC(=O)C(=O)CC(C)C 90135,c1(C(=O)NCCC2(C)CCN(C(COCCC=C)=O)C2)cccc2c1OC(C)C2 90136,C(=O)(C#CC(C)(C)O)N1C(C(=O)NC(c2ccncc2F)C)CC(OC)C1 90137,N1(C(CCOC)=O)C(C(=O)N(CC(=O)OC)CCN(C)C)CC2CC12.C(C(C)C)O 90138,c1(C(=O)NC(C2CC=CCC2)C(N2CCC(=C)C2)=O)cnc(O)cc1C 90139,c1(CC)nc(C)c(CC(=O)NC(C)(C)CCNC(=O)Cc2csc(C)c2)c(C)n1 90140,C1(NC(CC(CCC)C)=O)CCSC12CN(C(c1ccc(N)cc1OCC)=O)C2 90141,N1(C(CCc2cccc(C)c2)=O)CCCC(C(=O)NCC2CSCCO2)CC1 90142,C=CCCC(C(=O)NCC1(C2CC2)CCC1)NC(=O)CC1COC(=O)C1 90143,c1(C2(C(N3CCC(NC(C(COC)C)=O)C3)=O)CC2(C)C)cccc(Cl)c1 90144,C1(CNC(Cc2c(C)noc2Cl)=O)CN(C(C2(C)CC(=O)N(C)C2)=O)CCCO1 90145,c1(C(=O)NCCC(C)(C)NC(C2CC2(Cl)Cl)=O)cnc2occc2c1 90146,N1(C(C(C(C)(C)C)OC)=O)CCC(C(=O)NCC(CC(C)C)N(C)C)C12CCC2 90147,C(C)(C(C)(C)C(=O)NC1CC2CCCC2C1)NC(C(C)C)=O 90148,Cc1cc(NC(=O)CCN2CCC2)ccc1NC(C1CCCC1CF)=O 90149,N1(C(C2=C(C)OCC2)=O)CCC2CCC(NC(C3CC4(C3)CS(=O)(=O)C4)=O)C1C2 90150,CC(C)CC(C)CC(=O)N1CCCCC1CNC(c1cscc1C(N)=O)=O 90151,C1(CNC(C#CC(C)C)=O)CCCC12CCN(C(=O)CC1OCCC1C)CC2 90152,C1(NC(C2(SC)CC(O)C2)=O)CN(C(c2ccc(F)cc2)=O)C2(CCC2)C1 90153,N1(C(C(CC)C)=O)CC(CO)C2(C1)CN(C(=O)Cc1cccc(Cl)c1F)C2 90154,c1(-c2ccc(NCc3c(Br)ccc(C#N)c3)c(F)c2)cc2ccccc2cc1O 90155,CC(C)C(C(C)NC(=O)CCn1cncn1)NC(=O)Cc1ccc(O)cc1 90156,C1(CN(C(=O)C=Cc2ccco2)C)CN(C(C2CC2C#N)=O)CCO1 90157,CCC(C(=O)N(C(C)CCNC(c1ccc(S(N)(=O)=O)o1)=O)C)C(F)(F)F 90158,CN1CCC(O)C(NC(c2cc(CCNC(c3ccncc3)=O)on2)=O)C1 90159,c1(C(N(CCCNC(C(C)c2cncs2)=O)CCO)=O)cc([N+](=O)[O-])ccn1 90160,C1(C(=O)NCCN(C(=O)C(O)CC(F)F)C)CC12CCCCCC2 90161,CN1CC(C(=O)NC(C)(C)C(=O)NCCC(=O)OC(N)=O)CCC1=O 90162,C1(C)(c2ccc(NC(c3c(C)non3)=O)cc2)NC(=O)NC1=O 90163,c1(-c2scc(Nc3nc(C)cc(OC)n3)n2)cc(F)c(Cl)cc1Cl 90164,N1(C(Cc2ccnc(OC)n2)=O)CCN(Cc2ccccc2)C(C(C)C)C1 90165,C1(NC(C2C(=C)CC2)=O)CN(C(c2cc3c(s2)CCC3)=O)CCC1C 90166,C1(CNC(=O)CC2CCOC2)COCCN(C(=O)CCOCC2CCCO2)C1 90167,C1(c2c(C=C)cccc2)CCCCN1S(=O)(=O)N=S(C)(=O)CCO 90168,c1(C(N(CCN(C(Cc2c(C)noc2)=O)C)C)=O)cc2c(F)c(F)c(F)cc2[nH]1 90169,CC1(C)CN(C(C2(Cl)CC2)=O)C1C1CCN(C(C2CCS(=O)(=O)N2)=O)CC1 90170,c1(C(=O)NC(CCNC(C(CCC)C)=O)(C)CC)cc([N+](=O)[O-])c[nH]1 90171,S(=O)(=O)(c1cc2c(cc1Cl)CCCC(=O)N2)N1C(C)(COC)CC(N)C1 90172,CC(C)(CS(C)(=O)=O)C(=O)NCC(F)CNC(c1cnc(N)c([N+](=O)[O-])c1)=O 90173,Cc1cc(F)sc1C(=O)NCC1(NC(C2CCC(CC(C)C)C2)=O)CCCCC1 90174,Cc1cccc(C(O)CN(c2cc(C#N)no2)Cc2ccccc2)c1 90175,Cc1cc(=NCCC(C)(O)c2ccccc2)[nH]cc1S(=O)(=O)N1CCCC1C1CC1 90176,c1(OCC(=O)NOC2CCOCC2)cccc(NC(C2CC2CO)=O)c1.C(C(F)F)S 90177,c1(OC)ccc(-c2ccccc2)cc1NCC1CC(C(=O)O)CO1 90178,C=CCC(CC(F)F)NC(=O)COC1CCN(C(=O)C(C2(O)CCCC2)F)C1 90179,Cc1ccn2ncc(C(N3CCC4CC3CN4C(c3ccc(Cl)cc3)=O)=O)c2c1 90180,C(=O)(CCC(CF)CF)N1C(C)C(NC(=O)CN2CCOCC2=O)CCC1 90181,c1(CC)nc(Cl)[nH]c(=NC2CC(NC(=O)Cc3ccc(C)cc3C)C2)c1Cl 90182,C(C(CC(=O)NCCNC(N)=O)C1CCC1)NC(C(CC)N(C)C)=O 90183,C12(C(N(C3CC4(CC4)C3)C)=O)CCC(NC(C3CC4CCC4C3)=O)(CC1)C2 90184,C1(C(C)C)CN(C(=O)CC(C)(C)F)CCN1C(=O)CC1CCC(=O)N1 90185,Cc1cc(C(=O)N(C2CCN(C(c3ccc(C#N)cc3)=O)C2)CCO)ccc1Br 90186,C1(NC(c2cc(CC)on2)=O)CCCCC1CNC(C1(c2cc[nH]n2)CCC1)=O 90187,N1(C(C2(CCNC(C(CC(CC)C)=O)=O)CCCC2)=O)CCn2cc(C)nc2C1 90188,N1(C(c2c(C)c([N+](=O)[O-])cc(Cl)c2)=O)CCCCC(C2CN(C(=O)CO)C2)C1 90189,c1(C(N(C)CC2(C)CCCC2NC(=O)C2=NOCC2)=O)cc2n(n1)CCNC2=O 90190,CCC(C)C(C)C(=O)NCC1(F)CC(CNC(=O)CCc2ncc(F)cn2)C1 90191,CC(C)CC(O)C(=O)NC(C)CC1CN(C(=O)CCCn2ccccc2=O)C1 90192,C(=O)(CC(C(F)(F)F)NC(c1ccccc1F)=O)NCc1n(CC)ncc1 90193,N1(C(c2ccc(SCC)cc2)=O)CCC(F)(F)C(CNC(=O)CC(C)C)C1 90194,N1(C(CCOCCOC(C)(C)C)=O)CC=CC(NC(C2CCCN2C=O)=O)C1 90195,C1(CC(=O)NCCCN(C(C)C)C(c2ccc3c(c2)CC3)=O)CCCS(=O)(=O)C1 90196,c1(C(N2C(CNC(C3C4CC5C(C4=O)C35)=O)CC2)=O)ccc2c(c1)CCOC2 90197,C(=O)(C(C(C)C(C)C)NC(C)=O)NCCC(=C)CNC(=O)CCOCC(C)C 90198,c1(C(=O)NCC(C(C)(C)C)CO)cnc2cnc(Cl)cc2c1 90199,CC1(C)CN(C(=O)CCn2cccnc2=O)CC1NC(c1c[nH]cc(F)c1=O)=O 90200,c1(C(N2C(CNC(COCC=C)=O)COCC2)=O)cccc(C(N)=O)c1F 90201,c1(N2C(CNC(CS(CCOC)(=O)=O)=O)CCC2)cc2c(cn1)C(=O)CCC2 90202,N1(C(=O)OC(C)(C)C)CC(c2ccccc2)(NC(C2CCCS2)=O)C1 90203,c1(C(N(CC(C)NC(=O)C(C)(C)c2ccns2)CC)=O)ccc(Br)cn1 90204,N1(C(c2[nH]nc(OC)c2Cl)=O)CCCN(C(c2ccc(C(C)O)cc2)=O)C(C)C1 90205,CCC(C)(CCNC(=O)Cc1ccccc1F)NC(=O)CC1CCCCO1 90206,Cc1ncc(CC(=O)NCC2CN(C(=O)CC3CNC(=O)C3)C2)c(O)n1 90207,C(=O)(C1=CCCC(C)(C)C1)NC(C1CCCN(C(c2ccc(SC)cc2)=O)C1)C 90208,N1(C(CCCC(=O)OC)=O)CC2CN(C(C3CCC(C)CC3)=O)CC2(C)C1 90209,c1(C(N)=O)cccc(N(C(C2CN3CCC23)=O)Cc2ccccc2)n1 90210,c1(C(N(CCNC(c2ccc(-n3ccnc3)nn2)=O)CC)=O)cc(Cl)nnc1O 90211,C1(NC(CCNC(C)=O)=O)CCN(C(=O)CCS(C)=O)C1C 90212,c1(OCCC)cccc(-c2cccc(OCC3(C)CC3)c2)c1 90213,CC(C)(C(=O)NC1CCC(CNC(C2(CO)CCCO2)=O)C1)S(C)(=O)=O 90214,c1(C(C(=O)N(CCC)CCNC(=O)Cc2ccno2)N(C)C)ccccc1 90215,CC1(C(=O)NC2CC(CNC(=O)Cn3nnc(-c4ccccc4)n3)C2)CC(F)C1 90216,C1(N(C(CCC=CC)=O)C)CN(C(C2(COC)CC2)=O)CCC1O 90217,N1(C(CCCOCCC)=O)CC2CC(NC(c3cnsc3C)=O)CC2C1 90218,N=c1nc(CCNC(=O)C(N2CCCC(C(=O)O)C2)=O)cc[nH]1 90219,C1(C2CCCN(C(=O)C3=CCC(C)CC3)C2)(NC(C2C(C3C(C)C3)C2)=O)CC1 90220,c1(C(=O)NCC2OCCN(C(CC3(C=C)CCC3)=O)C2)cc(C#N)c(O)nc1N 90221,Cc1cccc(NC(=O)CC2CCC(NC(=O)Cc3nc(C)sc3C)CC2)n1 90222,N1(C(C2(CC)CC(C)(C)C2)=O)CC(C)OC2(CCN(C(=O)CSC(C)C)CC2)C1 90223,C(=O)(C1=NOC(CNC(C2CCSCC2)=O)C1)NCc1cc(COC)on1 90224,N1(C(=O)Cc2nc(Cl)cs2)CCN(C(c2ncncc2Cl)=O)CC(O)C1 90225,N1(C(C2CC2C(N2CC3OCC(CO)C3C2)=O)=O)CCc2ccccc2CC1 90226,C(=O)(C(CC(C)C)NC(c1ncn(C(C)C)n1)=O)Nc1c(C)nsc1 90227,C(C(C(=O)NCCC(C)CO)C(C)(C)C)NC(C(CC)(C)CC)=O 90228,C1(NC(C(C=C)(C)CC)=O)CC2CCC(C1F)N2C(c1conc1CC)=O 90229,c1(C(N(CC(C)NC(=O)C=Cc2ccoc2)CC)=O)cnc2[nH]ncc2c1 90230,C1(NCCNC(C2CCCCC2)=O)COCC1F 90231,N1(C(C2C(CC)OCC2)=O)CC2CCC(C1)N2C(C1CCC(C)(C)O1)=O 90232,C1(CNc2c(OCCC)cccn2)CCCC2(CC(C(=O)O)C2)O1 90233,C1(C(CNC(COCCOC)=O)NC(C2CN(C)C2)=O)CCCCC1 90234,C(=O)(C1Cc2ccccc21)NCC(=C)CCNC(c1cccc(C)c1CC)=O 90235,CCC(C)CCC(=O)N1CCOC(CNC(c2ncoc2C(F)(F)F)=O)C1 90236,Cc1nn(C)c2cc(NC(C3CC4CC4N3C(c3cc[nH]c3)=O)=O)ccc12 90237,C(CC1CCCC1)(C(=O)NCC#CCNC(C1CCCSC1)=O)OC 90238,c1(C(=O)NCC(C)NC(CCC=C=C)=O)cc2c(nc1O)CCCC2 90239,C1(CC(=O)NC2(C)CN(C(C(C)CC3CC3)=O)C2)CCCC1(F)F 90240,Cc1cncc(C=CC(=O)NCCC2CCCCN2C(c2oncc2C)=O)c1 90241,c1(C(N2CCCC(CNC(c3sccc3I)=O)C2)=O)cccc(F)c1I 90242,Cc1cc(C(=O)NCC(C)(C2CC2)NC(=O)CSC(F)F)cc(C)c1N 90243,N1(C(c2c(OC)c[nH]n2)=O)CC2CC(O)C1C2NC(c1ccc2nnnn2c1)=O 90244,c1(N2CCC=C(C)C2)[nH]c(=NCCc2cccs2)nc2c1ncn2C(C)C 90245,C1(CCNC(c2n(CC)ncc2)=O)CN(C(c2snnc2C)=O)CCCO1 90246,N1(C(C(CC)n2cccn2)=O)CCN(C(=O)CCCCC2CC2)C(CCOC)C1 90247,N1(C(C(C)(C)C2CCN(C(C3CCOC(=O)CC3)=O)C2)=O)CCC2(CCC(O)C2)C1 90248,N1(C(c2c(C)cnnc2)=O)CCC(C)(C)C(CNC(C2CCOC(C)(C)C2)=O)C1 90249,N1(C(C(COC)O)=O)CCC(C2CCN(C(=O)C(C)(C)C(C)(F)F)C2)CC1 90250,CCCC(C)(C)CC(=O)N1CCC1CNC(=O)CCc1cn(C)nc1C 90251,c1(C(N2CC3C(NC(C(F)=CCC)=O)(CCC3)C2)=O)c(C)[nH]c2ccc(Cl)cc12 90252,C1(C(=O)NCC2CN(C(C(C(CC)C)C)=O)CC2C)CN2CCN1CC2C 90253,c1(C(=O)NCC(CCOC)NC(C2CC2(Cl)Cl)=O)ccc(C(F)F)c(OC)c1 90254,c1(N(C)C)cccc(S(=O)(=O)C(=O)NC(C2CCCOC2)CO)c1 90255,C=CCCCC(C)(C)C(=O)NC1CC1NC(c1cccs1)=O 90256,c1(NCC(C(C)C)(C)NC(=O)CCn2ncn(C)c2=O)ncc2c(n1)COC2 90257,C1(C(=O)NCC(CNC(=O)C(C)CN(C)C)OC)CC2CC1CC2(F)F 90258,c1(C(=O)NC(C)CCCNC(C2CC2C)=O)cnn2c1S(=O)(=O)NCC2 90259,c1(C(=O)NC2(CCNC(C(C)(C(C)C)OC)=O)CCC2)cc(F)cc(N)c1F 90260,C1(C(=O)NCCCCC#C)CCC2(CC2)N1C(=O)CC1CC(CC)C1 90261,c1(C(=O)OC(c2cccc(Cl)c2Cl)C)ccc([N+](=O)[O-])nc1 90262,C1(NC(CCNC(CN(CCC#C)C)=O)=O)CC2CC2C1 90263,c1(OCC#C)ncccc1C(=O)NCCN(C(C1CC1Cl)=O)Cc1ccccc1 90264,CCC(C#N)(CC)C(=O)NC(C)CCNC(C1CC2(C1)CC1(CC1)C2)=O 90265,C1(F)(C(=O)NC2C(NC(C3N(C)CCCC3)=O)COCC2)CCC(F)(F)CC1 90266,C=CCC(CC(C)C)C(=O)NCC1CCCC1NC(C1(C(=O)NC)CCCC1)=O 90267,C=CC(C)(C)CC(=O)N(C(C)CN(C(=O)CC1C(C)C1(F)F)C)C 90268,C12(C(N3CC(NC(C4CC5(CCC5)C4)=O)C3)=O)CC3CC(CC1C3)C2 90269,c1(C(N2C(CNC(CN=S(C)(C)=O)=O)CC2)=O)cc(Cl)ccc1[N+](=O)[O-] 90270,C#CC1CC2(CC2)CN1C(=O)C(C)N(C(c1cc(C(C)=O)c[nH]1)=O)CC 90271,C1(NC(CCCCC(CO)NC(=O)OC(C)(C)C)=O)CS(=O)(=O)CC12CC2 90272,c1(C(=O)NCC2CCCC(NC(C3N(CC#C)CCC3)=O)C2)cc(Cl)nnc1Cl 90273,c1(C(=O)NC2CCC(NC(C3CCCCS3)=O)C2)ccccc1SCC(F)(F)F 90274,N1(C(C2CCC(=C)CC2)=O)CC2CCOCC2(NC(=O)CCC(C)C)C1 90275,C1(NC(=O)CN2CCS(=O)CC2)CN(N2CC(=C)C2)CC12CC2.C1(C=O)CCC1 90276,C=CC(CCC)CC(=O)N1CC(N(C)C(c2ccc(F)cc2F)=O)C(O)C1 90277,c1(C(=O)NCC(CNC(C2C(CC)CC2)=O)O)nccc(C)c1N 90278,c1(C2(NC(=O)NCc3ccc(-c4cccnc4)cc3)CCC2)ccc(Br)cc1F 90279,N1(C(c2n(CC)nnc2)=O)CC(NC(c2cc(N(C)C)ccc2F)=O)C(C)(C)C1 90280,c1(C(=O)NCC2CC(NC(c3c(C)coc3)=O)C2(C)C)ccc(C)c(C(C)=O)c1 90281,C=C(C)CCC(C)NC(C1C=CCN(C(c2nccn2C(C)C)=O)C1)=O 90282,c1(OCC)cc(N(C2CCN(C(=O)CC3CC(C)(C)CO3)CC2)C)ncn1 90283,CC(C(=O)N1CCC(C(C)(O)CNC(=O)C#CC2CCC2)CC1)C(C)(F)F 90284,c1(OCC(N2CCC(Oc3ccc(C)cc3)C2)=O)c(F)cc(I)cc1F 90285,c1(OC)nc(Cl)c(C)cc1C1CC(NC(C2C3CC(N)CC23)=O)c2ccccc21 90286,C1(NC(CN2CCC(C)CC2)=O)CCC2(CC1)CN(Cc1ccncc1C#N)C2 90287,CCCCC(C)C(=O)NC1CCCCCC1C(N1CC[Si](C)(C)CC1)=O 90288,N1(C(CCC#C)=O)CCCCC(C(=O)NC2CC23CCCCC3)C1 90289,S(=O)(=O)(c1cccc2ccccc12)N1CCOCC(NC(C(C=C)O)=O)C1 90290,C(=O)(C(O)CC(F)(F)F)N1C(C)(CNC(=O)NCc2cc(F)ccc2F)CCC1 90291,N1(C(C2C(C)CCCC2)=O)CC2(CCCCN2C(c2cnc3[nH]cnc3c2)=O)C1 90292,N1(C(=O)Cc2cnns2)CCCC(O)(CNC(C2(O)CC(F)(F)C2)=O)C1 90293,N1(C(C(C2CN(C(c3c(OC)nccn3)=O)C2)O)=O)CCC12CCSCC2 90294,c1(NC(C)=O)ccc(C(C(=O)NCCC#N)N(C)CC2CCCCC2O)cn1 90295,c1(C(N2CC3C(CNC(c4ccc(C#N)s4)=O)(C3)C2)=O)cnc2ccc(F)cn12 90296,C1(N(C)C(C2CC(F)(CF)C2)=O)CCCN(C(=O)COCCCF)C1 90297,c1(C(C(=O)NC(c2cnn(C)c2)C)O)ccc([N+](=O)[O-])cc1 90298,C(=O)(C(C)C1OCCc2sccc21)N1C(CNC(C2CC(OC)C2)=O)CC1 90299,C1(C(N2CC(NC(C(C3CCOC3)OC)=O)C(C)C2)=O)Cc2cc(F)ccc2O1 90300,CC1(NC(=O)CCc2cc(Cl)cc(Cl)c2)CCC(NC(C2CC(C)(O)C2)=O)CC1 90301,c1(CC(=O)NC2CC(NC(=O)Cc3cnc[nH]3)C2)csc2ccc(Cl)cc12 90302,c1(C(=O)NC(C(=O)NCCc2ccncn2)C2(C)CC2)nc(Cl)cs1 90303,Cc1c(C(=O)NCC2CCC(NC(C3CCCN(C)C3)=O)C2)nnn1C(C)C 90304,Cc1c(C(=O)NC(C)C(C)NC(c2ccc(Br)o2)=O)cncc1N 90305,N1(C(c2c(C)nc(-c3ccccn3)s2)=O)CCC(C)C(NC(=O)C=CCF)C1 90306,c1(C(=O)NCC2(OC)CCN(C(=O)CO)CC2)ccc2c(c1)CCC(=O)N2C 90307,C(CCCCNC(=O)CN1CCCC1C(=O)OC)N(C(C(C)OCC#C)=O)C 90308,C1(CNC(c2c(C)cno2)=O)N(C(C2CCS2(=O)=O)=O)CCC1(C)C 90309,N1(C(Cn2ccc(C)n2)=O)CC2(C1)C(NC(C1C=CCC1)=O)CCS2(=O)=O 90310,c1(C(=O)NC(CCCNC(C(C(C)C)OC)=O)(C)C)ncn2c1COCC2 90311,C1(C(C)N(C2(CN3CCCC3)CSC2)C)CCN(C)CC1 90312,C12(C(=O)NCCCCC3(NC(CCCC)=O)CC3)CCC(CC)(C1)OC2 90313,C(C1=NOC2OCCC12)NC(=O)Nc1ccc(CNCC2CCOC2)cc1 90314,C#CCC(C)(C(=O)N1CC(F)CC(F)C1)NC(=O)CC1CSCCO1 90315,C1(NC(C(CC)N(C)C)=O)CCCCC12CCN(C(C1(C#N)CCCC1)=O)CC2 90316,C1(C(=O)NCCCCCCC2CC2)COCCN(C(=O)CNc2ccccn2)C1 90317,c1(C(=O)NCC2(F)CCC(NC(CS(C)(=O)=O)=O)C2)ccc(F)c(Cl)c1N 90318,N1(C(CC)=O)CC2(CCCC(CNC(c3cnsc3)=O)O2)C1 90319,c1(Cc2ccc(OC)cc2)ccnc(SC)c1F.C12(CC1)C(=O)O2 90320,c1(N2CC(CNC(c3ccc(CC)c(F)c3)=O)OCC2)ncc2ccsc2n1 90321,C1(c2cn(C3CN(C(C4(F)CC(C(=O)OC)C4)=O)C3)nn2)C(C)(C)C1(C)C.C1(C)CC1 90322,CCC(CC(=O)NCCC1(O)CCN(C(C2CN3CCCC2C3)=O)C1)C(C)(C)C 90323,CC1(C)COC(CC(=O)NC2CCC(NC(=O)CCOC3CCOCC3)C2)C1 90324,c1(CC(=O)NCC2C3CN(C(C=C(C)C(F)F)=O)CC32)ccc([N+](=O)[O-])cc1F 90325,N1(C(C(CC)=CC)=O)CC2CC2C1C(N1CC(NC(C)=O)C1)=O 90326,c1(CC)nocc1C(=O)NC1CC(C)(CNC(=O)CCc2cc(C(N)=O)no2)C1 90327,CCCS(=O)(=O)CC(=O)NCC1(F)CCN(C(C2Cc3nc(C)cn3C2)=O)C1 90328,c1(OC)cccc(CC(=O)NCC2(O)CCN(C(=O)C(C)C)C2)c1Cl 90329,C(=O)(CCC(C)(C)C#N)NC1CC(C)N(C(=O)CSCc2ccccc2)C1 90330,C#CCC(C(=O)NN1CCOC1=O)c1cccc(Cl)c1 90331,N1(Cc2c(N)cccn2)CCc2c(Cl)cccc21 90332,N1(C(C2(C)C(C)(C)C2CNC(=O)CSc2n[nH]c(=N)s2)=O)CCC2CCC12CO 90333,c1(CC=C)cccc(C(=O)N(C(C)C(=O)NCC2=NOC(C)C2)C2CC2)c1 90334,c1(C(=O)NC(CC)C)cnc(N2CCC(F)(c3ccccc3)C2)nc1 90335,Cc1cc2c(cc1Cl)C(NC(c1ccc(NC(=O)NC3CCC3)c(Br)c1)=O)CO2 90336,C1(CC(=O)NCC2CC(OC)C2)CCN(C(c2cn(CCO)nn2)=O)C1(C)C 90337,Cc1ccc(C(=O)NC2CCCC(NC(=O)C(F)(F)c3nccn3C)C2)n1C 90338,C1(NC(=O)CCN2CCOCC2)CN(C(C2(c3cc[nH]n3)CCC2)=O)CC1O 90339,C1(CNC(C(C)Cc2cnn(C)c2)=O)(CNC(=O)CSC2CC2)CC(F)(F)C1 90340,Cc1nc(O)ccc1C(=O)NC(C)CCNC(c1ccc(-n2cccn2)cc1)=O 90341,c1(C(=O)NCC2C(NC(CCCC)=O)CCC2)cnc(OC)cn1 90342,c1(C(N(CC)CC)=O)ccc(OC(C)C)cc1.c1(CC(C)N)ccc(Cl)s1 90343,C1(CC)(CC)CC(NC(=O)CC2CCC(=O)N2C)CN1C(=O)CCC1CCCC1 90344,S(=O)(=O)(c1cccc(=NC(CCO)c2cccc(C)c2)[nH]1)NC(CC)CCO 90345,CC1C(NC(=O)CCn2ccccc2=O)CCCN1C(c1ccc(C#N)s1)=O 90346,N1(C(C(C)NC(CC)=O)=O)CCN(C(C2CC3(C2)CC3(F)F)=O)CC1C 90347,Fc1ccc2scc(CNC3CCCCC3c3cccc(Cl)c3)c2c1 90348,C1(NC(C2CCN(C)C2)=O)CC2CC(C1)N(C(C1SCCS1)=O)C2 90349,N1(C(c2cc(CC(C)C)on2)=O)CCCCC1CNC(=O)CCN1CCCC1 90350,c12cc(ncn1)N2.N1(C(C)=O)CC(CNC(C2(n3ccnn3)CC2)=O)C1 90351,CC#CCCC(=O)N1CCC(C(N2CC(C)C(F)C2)=O)CC1 90352,CC(C)CC(CNC(c1csc(O)n1)=O)C(=O)N(CC(O)CF)C 90353,N1(C(c2c[nH]c(=N)s2)=O)CCC2(CCC(NC(=O)C3=CC4(CCOC4)C3)C2)CC1 90354,N1(C(C(C)SC)=O)CCC(NC(=O)C(C)(C)NC(C)=O)C(F)C1 90355,c1(CC)ccc(F)c(C(N2CC(NC(c3cn(C)nc3COC)=O)C2)=O)c1 90356,c1(C(=O)NCC2C(NC(C3(COC)CC3)=O)C2)cc2cnc(Cl)cc2s1 90357,C1(C(=O)OC)CCCN(N2CCN(c3nc(C(C)=O)c(C)s3)CC2)C1C 90358,c1(C(N2CC(O)(CCNC(c3nc(C#C)sc3)=O)C2)=O)nc(O)nc(O)c1N 90359,C1(C(N)=O)(NC(=O)CN(C(=O)CC2C=CCC2)CC2CC2)CCCCC1 90360,N1(C(C)C)CCN(C(=NCC2CCCS(=O)(=O)C2)NCC2CCOC2)CC1=O 90361,c1(C(=O)NC)ccccc1OC1CCN(C(=O)NC2CC23CCC3)C1 90362,c1(OC)cc(C(C)CC(=O)N(C)CCN(C)C(N2CC3CC3C2)=O)ccc1C 90363,C(CCC(CCC)NC(c1cnc(S)n1-c1ccc(F)cc1)=O)NC(C=CC)=O 90364,c1(C(=O)NCC2CCN2C(C23CC(O)C2C3)=O)ccc2c[nH]nc2n1 90365,Cc1ncc(=NC(=O)Cc2c(C)[nH]c3ccc(C(C)C)cc23)[nH]c1Br 90366,CN1C(=O)CCCC1C(=O)NC1CCC1NC(=O)Cn1cc(C#N)cn1 90367,C(CCC(O)C(=O)NCCN1CCOCC1C)NC(C1(SC)CC1)=O 90368,C(=O)(CS(=O)(=O)N(C)C)N(CC(F)CNC(c1cnc(CC(C)(C)C)s1)=O)C 90369,C(C)(C)(CCCC(=O)NCc1cncs1)NC(CCc1ccn(C)c1)=O 90370,C1(CNC(CN(C)C2CC2)=O)CCCCC1NC(C1CCCOC1c1cn[nH]c1)=O 90371,c1(CNC(=O)NCC2(CC)CCC2)cc(C(F)(F)F)ccc1Br 90372,C1(OC)(CO)CCN(OC)C1.C1(C(=O)N)CC=CCC1C.c12cc(cs1)C(=O)NC2 90373,N1(c2snc(CCC)n2)CCC2(CCC(CNC(C3CCCCC3)=O)OC2)CC1 90374,Cc1cc(C(N2CCOC(C(N3CCOCC3CN(C)C)=O)C2)=O)ccc1C#N 90375,N1(C(C=Cc2cncc(OC)c2)=O)CC2CCCC2(NC(=O)CS(N)(=O)=O)C1 90376,CCS(=O)(=O)c1ccc(F)c(C(=O)NCC2(F)CCC(NC(=O)C(O)CF)C2)c1 90377,CC1CC(C(=O)N2CCOCC2(c2ccc(F)cc2)c2ccccc2)=NO1 90378,c1(OC)cc(C(=O)NC(C)(CNC(c2ccc(C)cc2C)=O)C(C)C)c(F)cn1 90379,Cc1cccc(Cl)c1C(=O)NC(C)CC(C)NC(C1(N(C)C)CCC1)=O 90380,c1(C2N(C(c3nn(CC)cc3Br)C(=O)NCCC)CCC2)cc(OC)nc(Cl)c1 90381,C1(NC(c2ccc(C)c(C)n2)=O)CC2CC1CN(C(=O)C=CC(C)(C)C)C2 90382,C1(C#CC(=O)NCCOC2CCN(C(=O)CCOCC(F)F)C2)(CC)COC1 90383,C1(C(=O)CC2C(NC(c3ccc(-c4cc[nH]n4)s3)=O)CC2)CC(F)(F)C1 90384,CC1CCC(C)N(C(=O)CCOC2CN(C(c3cc[nH]c(=N)n3)=O)C2)C1 90385,c1(C(N2C(C)(CC(=O)NCc3ncn4c3CCC4)CC2)=O)ccc2nccn2c1 90386,O=C1CN(CC2CC23CCC3)C(=O)N1CCCCN1CCCC1 90387,C(C(C)C(F)C(=O)N(C(CF)CF)C)NC(CCCC)=O 90388,c1(C(N2CC(CNC(c3cncc(C)c3)=O)C3C2C3)=O)coc2c1CS(=O)(=O)C2 90389,N12CCC(O)C(C1)C2=O.Cc1ccc(CS(=O)(=O)NCC2CCN(C)CC2)cc1 90390,c1(OC)nccc(=NCCOC2CN(C(=O)C=Cc3cccnc3)C2)[nH]1 90391,C1(c2cn(CC3(OC)CN(C)C3)nn2)CCN(C(C2(C)CC2)=O)C(C)C1.C(C)(=O)O 90392,C1(C(=O)NC2CC(NC(C3CC34CC(F)(F)C4)=O)C2)CCc2nncn2C1 90393,c1(C(=O)NC2(C)CN(C(C(CSC)C)=O)C2)ccc2cncn2c1 90394,c1(C(C(=O)NCC(COCC)C)N(c2ccccc2)C)cccc(OC)c1 90395,C1(CC#C)(C(=O)NCCc2cnn[nH]2)CCN(C(=O)C(COC)CC)C1 90396,CC#CC1CCN(C(=O)CCOC2CN(C(c3cc(CC)sn3)=O)C2)C1 90397,C1(NC(c2cnc(C(=O)OCC)s2)=O)CC(C)N(C(=O)CCSC2CCCC2)C1 90398,Cc1cc(C(N2CCC(CF)(NC(c3ncccc3Cl)=O)C2)=O)c2c(c1)CCC2 90399,N1(C(C2C(=C)C2)=O)CCOCC1CN(C(=O)CSc1n[nH]c(O)n1)C 90400,c1(OC)ccc(C(=O)NC2CCCC2CNC(c2ccc(Cl)cn2)=O)c(F)n1 90401,C1(NC(C(C=C)O)=O)CCN(C(=O)C(C)NS(C)(=O)=O)CC1(C)C 90402,C(=O)(C(C)(C)CC(=O)OC(C)=O)NCCn1cc(C(=O)NC2CC(OC)C2)nn1 90403,c1(C(N(CCCNC(C2C(C)CC2C)=O)CC)=O)nc(C)oc1C 90404,C(C(F)C(=O)N(C1CC1)CC1CCOC1)C1CN(C(=O)CO)C1 90405,C1(CC)CCCC(CNCc2cc(Br)cs2)C1 90406,N12CCC(CC1)OC1(CCCC1)C2=O.C(CC(=O)NCC(N1CCCC1)=O)OC 90407,c1(NC2C(NC(C(C)(C)c3nccs3)=O)CCCC2)nc(O)c2cnn(C)c2n1 90408,C(=O)(C(C(C)C)NC(C1CCC(NC(C2(C(=O)OC)CC2)(C)C)CC1)=O)NC 90409,C(=O)(C(C)(C)CC(=O)NCC=CC(=O)NCCN1CCC(CO)C1)OC 90410,CC1(C)CCC(CC(=O)NC2CC(C(=O)NCCCCCCO)CC2O)C1 90411,S1(=O)(=O)c2ccc(cc2)S(=O)(=O)N1CC#N.C(C(C)(C)N)N(C)CCO 90412,C1(NC(C2(N(C(C(COC)(C)OC)=O)C)CC2)=O)CCN(C)CC1(C)C 90413,C1(C(N2CCCC(CC)(NC(c3cccn3C)=O)C2)=O)CCCC1P(C)(C)=O 90414,N1(C(C2C(C)(COC)C2)=O)CCc2ccccc2C1CNC(c1nccn1C)=O 90415,C1(C(=O)NC2C(CC(C)(C)C)C2)CCCN(C(C23CCC(CC2)C3)=O)C1 90416,N1(C(CC)=O)CCC2CCC(NC(c3cccc(Oc4cccnc4)c3)=O)C1C2 90417,C1(C(=O)NC(C(C)C)(C)CNC(c2cnc[nH]2)=O)CCC2(CCC2)CC1 90418,c1(CCC)ncoc1C(=O)NC(C(=O)N1CC(O)C1)C1(C)CC1 90419,Cc1cccnc1CC(=O)NC1(CC=CC(=O)NCCC2CCC3CC23)CCC1 90420,c1(CCC(N2CCCN(C(C(C)C)=O)CC2CO)=O)ccc2c(c1)COCC2 90421,CC1(C)C=C(C(=O)N2CC(CNC(C3(c4cc[nH]n4)CCC3)=O)CC2(C)C)C1 90422,c1(OCC)nc(N2CCC(C)C(NC(c3cc(C)c(C)o3)=O)C2)ncc1Cl 90423,C1(C)(CNC(c2cccc(C)c2)=O)CCCN(C(=O)Cc2c(O)ncnc2O)C1 90424,C1(O)(CCNC(=O)C(=O)NCc2ccc(F)cc2)CCN(C(=O)C=CC2CC2)C1 90425,Cc1cc(=O)ccn1CC(=O)NCC1(O)CC(NC(c2ccc(C#N)cn2)=O)C1 90426,Cc1cc(C(=O)NC(C)(C)CCN(C(=O)Cn2ccccc2=O)C)[nH]c1C 90427,C(CC(C)(C)CNC(c1ccc(-n2cncn2)nc1)=O)NC(c1c(C)csc1)=O 90428,C1(C)(C2CC(C(N(C(C)(C)C)C(F)F)=O)C2)NC(=O)NC1=O.N1(C(=O)O)CCC1C1CCC1 90429,C(=O)(C1=NN(C)C(=O)CC1)NC1CC2CC(NC(C3(OC)CCC3)=O)C1C2 90430,c1(C(C)C)cc(=NCC2CCCN(C(=O)CSc3cccc[n+]3[O-])C2)[nH]c(Cl)n1 90431,N1(C(CN(CC)CC)=O)CC2CC(O)C1C2NC(c1cn(C2CCCC2)nn1)=O 90432,C1(C(N2CCCC(CCC(N3CC(C)C(C)C3)=O)C2)=O)Cc2ccccc2C1 90433,N1(C(CCNC(=O)NC)=O)CC(CC(=O)NCC(C)(C)SC)CC1(C)C 90434,CCC(C)(O)C(=O)N1CC(CN2CCN(C(C3(S(N)(=O)=O)CC3)=O)CC2)C1 90435,N1(C(CCCCCC)=O)CC2(C1)CN(C(C1CCC1OC)=O)CC2CO 90436,CCC(C)CC(C)C(=O)NCCN(C)C(c1ccc(CN(C)C)nc1)=O 90437,N1(C(COCC=C)=O)CC(NC(C2CC2CF)=O)C(C)C1 90438,N1(C(C(C)OC2COC2)=O)CCC(C)(C)C(CNC(c2ccc(=O)n(C)n2)=O)C1 90439,O=[N+]([O-])c1cccc2[nH]nc(CNc3nc4c(s3)CC(O)CC4)c12 90440,c1(C(N2CC3(OCC(NC(C(CC)=CC)=O)C3)C2)=O)ncc([N+](=O)[O-])cc1Br 90441,N1(C(C2(C#N)CCCC2)=O)CC(C2CN(C(C34CC(CO3)C4)=O)C2)C1 90442,c1(C(=O)NCC2(NC(C(CCSC)O)=O)CC2)c(C)ncnc1C 90443,N1(C(c2c(CC)con2)=O)CCN(C(=O)C(C)OCC(C)C)CC1CF 90444,c1(-c2nc(C(CC)C)nn2C2CC(OC(C)(C)C)C2)ccn2c1CSCC2 90445,C1(C(=O)NCc2cn(C)cn2)(NC(C(C)c2cc[nH]n2)=O)CC1(C)C 90446,C1(C)(COC)CC(NC(c2c(Cl)cccc2Cl)=O)CN1C(=O)CCC(C)C 90447,C1(OC)CC(CO)(NC(c2cn(CCNC(=O)C(C)C3CC3)nn2)=O)C1 90448,n1(CC(=O)NC(CC(C)C)CNC(=O)CCCN(C)C)nnc2c1CCCC2 90449,Cc1ccc(C(C)C)cc1C(=O)N(C(C)CCNC(=O)C(c1cnn(C)c1)O)C 90450,CON(CCC(=O)NC(c1nn(C)cc1O)C)C(=O)c1n[nH]c(C)c1C 90451,N1(C(C(COC)C)=O)CCN(C(=O)CNC(c2nccc(C)n2)=O)CC1 90452,N1(C(CC)=O)CCC(C(=O)NCC(c2cnn(C)c2)C)CC1C 90453,C1(C(N2CCCC(F)C2)=O)CCC2(CN(Cc3ccc(O)c(F)c3F)C2)O1 90454,c1(C(=O)NC(C2(C(=O)NC(C)(C)CCCF)CC2)C)ccc(C#N)cn1 90455,C=C1CCN(C(c2ccn(CC)c2C)=O)C(C(=O)NC2(c3ncc[nH]3)CC2)C1 90456,c1(CC(=O)NC2CC(F)(CNC(=O)C(O)CF)C2)c[nH]c2cccc(F)c12 90457,c1(C(=O)NC(CCCNC(C(CC)n2cccn2)=O)C)cnc(C(N)=O)cn1 90458,CC1OC(=O)NC1C(=O)N(C)CCOCCC(=O)NCCC1(CO)CCC1 90459,c1(CCC(N2C(C)CN(C(C3CC3(Cl)Cl)=O)CC2)=O)nc2cnccc2[nH]1 90460,c1(C(=O)NC(CN(C(=O)CCC2(C#N)CCC2)CC)C)cncc(C(N)=O)c1 90461,Cc1ncc(Br)cc1C(N1CC2C(NC(=O)CNC(C3CCC3)=O)C2C1)=O 90462,C12(C(=O)NCC3CCN(C)C3)CC(CO1)N(C(=O)CC1CCCC1)C2 90463,C1(CC)CCN(C(=O)C=CC2(C)COC2)C(C(=O)NCC2CCCC(C)(C)C2)C1 90464,C1(C(N(CC(C)NC(=O)CC2CNC(=O)C2)C)=O)CCC(=O)N(C)C1 90465,COn1cnc(C)c1C(N1CCN(CCNC(=O)Cc2cccnc2C)CC1)=O 90466,c1(C(C)C(=O)NC2CCCC2NC(=O)CN(C)C(N)=O)cccc([N+](=O)[O-])c1 90467,C1(C(=O)NCCC2(C(N3C(CCC=C)CCC3)=O)CCCC2)CCOC(C)(C)C1 90468,c1(C(=O)NCCC2(O)CN(C(c3cc[nH]n3)=O)C2)c[nH]c2ncc(Br)cc12 90469,C(C1CCCCCC1)=CCn1c(N2CCC(N(C(CC)=O)C)C2)nnn1 90470,c1(NCCC(C)S(C)=O)cc(=NCc2nc(O)n[nH]2)[nH]cn1 90471,C(=O)(CCC1=CCCCC1)N1CCC(C)(NC(=O)CC2CCC(=O)N2)CC1 90472,N1(C(CCN(C(C)C)C(C2CC(=O)CS2)=O)=O)CCCC(C(=O)NC)C1.N(C)C 90473,C1(NC(CCCC#C)=O)CCN(C(=O)Cc2ccc(Br)nc2)C(C)C1 90474,CN1CC2CCC(C1)N2C(C1CC(F)CN1C(=O)CC1CSCCO1)=O 90475,CP(C)(=O)c1cccc(C(=O)N=S2(=O)CCCCCC2)c1 90476,C1(NC(CC2N(CC)CCC2)=O)(CC)CCN(C(=O)CCC2CC2(Cl)Cl)CC1 90477,c1(C(=O)NCC(CC=C)NC(=O)CCC(C)CC)nccc2[nH]nc(C(C)C)c12 90478,N1(C(C(CC)(C)CO)=O)CC23CCCC2(C1)CN(C(c1c[nH]cc(C)c1=O)=O)C3 90479,c1(CC)cc(C(=O)NCC(O)CN(C)C(c2cnc(S)nc2)=O)nn1CCO 90480,C(=O)(C1=CCc2ccccc21)N1C(CNC(C2=CC(C)(C)C2)=O)C(C2CC2)CC1 90481,N1(C(c2c(C)nc(CC)o2)=O)CCC(C)(C)C1C(=O)NCC1CCCN(CC)C1 90482,C1(=CC(=O)NC2CC(F)(CNC(C3CCC(OC)C3)=O)C2)CCCCCC1(F)F 90483,N1(C(C(CCC)C#N)=O)CC2(CCN(C(=O)C(n3ccc(Br)n3)C)C2)C1 90484,n1(CCNC(c2c(Br)nnn2C)c2n(CCOCC)nnn2)nc(C)cc1C 90485,N1(C(c2nc(C)nn2C)=O)CC(C)(CNC(=O)C=CC(F)(F)F)CC1(C)C 90486,CCCC(C)(C)C(=O)NCC(=O)NCC1(C)CCC(O)CC1 90487,C(=O)(C(C)(C)CCC#N)N1CC(CCNC(C(CC)N2CCCC2=O)=O)C(C)C1 90488,c1(C(=O)NC(C)CNC(C2CCC2(F)F)=O)ncn2ccccc12 90489,c1(N(C)C(=O)OC(C)(C)C)cnc(N2CCC(C(=O)NC3COC3)CC2)cn1 90490,c1(C(=O)NC2C3CN(CC2)C3=O)c(Cl)nc2ccccn12.c1(CC)cccnc1 90491,CC1(C)CN(C(C2CC3CC3N2)=O)CCN1Cc1cc(Cl)c(Cl)c(Cl)c1 90492,N1(C(c2c(C(C)C)scn2)=O)CCC(NC(=O)CCCc2ccccc2)C1C 90493,CC(C)CCCC(=O)NCC(C(C)(C)C)NC(=O)CC1CCC=CCC1 90494,CC(C(=O)NCC1(F)CC(NC(=O)Cc2cc[nH]c2)C1)C(C)(F)F 90495,c1(CC(=O)NC2CCC(NC(=O)C(O)C3CC3)C2)ccnc(O)c1 90496,C(=O)(C(C)(C)N=[N+]=[N-])N1CC(C=C)(CC(=O)NCC(C)OCC#C)C1 90497,CC1CC(CNC(c2ocnc2-c2ccccc2)=O)CN1C(C1CC=CCO1)=O 90498,Cn1cc(N)c(C(=O)NCCC2CN(C(C3CC3Cc3ccccc3)=O)C2)n1 90499,C1(NC(C(C#C)(C)C)=O)CCC2(CCCN2C(=O)C2CCCn3ncnc32)CC1 90500,C1(=O)C(C(C)(C)C)CCN1.C1(n2cc(-c3cn(CC)nc3)nn2)CC2CCC1O2 90501,C(C(C)C(=O)N(CCNC(=O)Cc1sccc1Cl)Cc1ccccc1)OC 90502,c1(NC(CN2C(C(=O)OC)(CO)CCC2)=O)ccc(O)cc1O 90503,C(N=c1cc[nH]c(=NCCc2cncs2)[nH]1)C1(C)CC2CC2C1 90504,c1(OC2CN(C(=O)OC(C)(C)C)C(OC(F)F)C2)cnc(O)cc1O 90505,CC1Cc2cc(Br)ccc2N1C(c1cnc2c(c1)COCC2)=O 90506,N1(C(CC2CC(CC)OCC2)=O)C2CCC1C(CNC(C1CC1C(=O)OC)=O)C2 90507,N1(C(Cn2nc(C3CC3)n(C)c2=O)=O)CC(NC(C2(Cl)CC2)=O)C2CCCC2C1 90508,C(C(C)(C)C(=O)NC1CC2(C1)CC2C(N1CCC(F)(C(N)=O)C1)=O)OCC 90509,C(=O)(C1=CCC2(COC2)OC1)OCCc1c(C(=O)OCC)cccc1 90510,c1(C(=O)NCCC2N(C(C3C(=C)C3)=O)CCCC2)cc(O)ccc1[N+](=O)[O-] 90511,C1(NC(C)CCn2cccn2)COC(C(C)(C)C)C1 90512,CCC(C)CC(C(=O)NCCC1NC(=O)NC1=O)NC(c1cc(F)ccc1F)=O 90513,c1(Cc2nn(C(COC)C)c(-c3ccc(O)c(C)c3)n2)cc(F)cc(F)c1F 90514,c1(CC)nc(-c2ccc(C(=O)NCc3cccc(C(=O)O)c3)cc2)ncc1C 90515,N1(C(C2CCC(CCC)CC2)=O)CC2(C1)CN(C(c1nc(=N)cc[nH]1)=O)C2 90516,c1(NC(C(CC#C)NC(=O)C=Cc2ccncc2)=O)ccc(F)c(CC)c1 90517,C(CCC(=O)N(C)CCOCCCNC(c1cc(O)no1)=O)OCCOC 90518,N1(C(c2scc(C(C)=O)c2)=O)CCCCC1C(C)NC(C1(C(N)=O)CCC1)=O 90519,c1(C(N(C(CNC(c2ncc(C)c(C)c2)=O)C)C)=O)cc(Br)c(O)nc1C 90520,C1(C2CCCN(C(=O)Cc3nncn3C)C2)(NC(C(C)OCCC(C)C)=O)CC1 90521,C(C1=CCCN(C(c2cc(C)[nH]n2)=O)C1)NC(Cc1cn(CC)nn1)=O 90522,c1(OC)ncccc1C(=O)NCCCCC1CCN(C(=O)Cn2ncnn2)CC1 90523,C1(NC(Cc2n(C)nnc2)=O)CC2CN(C(C3(O)CCCC3)=O)CC12 90524,c1(OC)ccc(CN2CCC(O)(C(=O)NCC3CCC3)C2)c(Br)c1 90525,Cc1cc(=NCCCNc2ccccc2)[nH]c(=NCc2cc(Br)cnc2O)[nH]1 90526,c1(C(=O)NC(CC)(C)CNC(C2(S(C)(=O)=O)CCC2)=O)cnc(O)n(C)c1=O 90527,C1(C(=O)NC(C#C)CC(C)C)C2CCN(C(=O)CC(OCC)OCC)CC12 90528,S(=O)(=O)(c1ccc(NC2CCCn3nccc32)c(Cl)c1)NCCC(C)CO 90529,N1(C(C=C(C)Cl)=O)CCC(NC(=O)CCn2c(C)csc2=O)CC(O)C1 90530,N1(C(C(COCC)C)=O)CCCC(CO)(NC(=O)CCNC(=O)C=CCl)C1 90531,CC1(C)CCCCC1C(=O)NCCCC1(NC(=O)CCc2nc(=N)[nH][nH]2)CC1 90532,c1(NC(=O)CC(C(F)F)NC(c2cn(C3CC3)nn2)=O)cccc2c1OCC2 90533,c1(C(=O)NC(C)CCN(C)C(c2ccc(=N)[nH]c2)=O)cc2ccccc2c(O)n1 90534,N1(C(Cn2c(C(F)F)cc(C)n2)=O)CC(NC(C2CC23CC(O)C3)=O)C(C)(C)C1 90535,C(N=c1cc(F)nc[nH]1)C1C2CN(C(C3C(c4ccc(OC)c(F)c4)C3)=O)CC21 90536,c1(-c2cccc(NC(C)=O)c2)ccc2c(C(=O)NC3CCC(F)(F)C3)n[nH]c2c1 90537,Cc1ccc(F)c(N)c1C(N1CC(C(C)NC(C2CC2(F)Cl)=O)C1)=O 90538,Cc1nc(C(N2CC(C3(NC(=O)C(O)P(C)(C)=O)CC3)C2)=O)c2ccccn12 90539,C1(CN(C(CC=C)=O)CC)CCN(C(=O)C(O)C(C)c2ccccc2F)CC1 90540,C12(CNC(CC3(C)CCCO3)=O)CC(CO1)N(C(C1CCCN1C=O)=O)C2 90541,O=S(=O)(C1=CCCCC1)NCc1cccc(C(F)(F)C(=O)O)c1 90542,S(=O)(=O)(c1ccc(NCCC(C)C)c(F)c1)NCC(CC)(C)CO 90543,C1(C(=O)NCC2(CN(C(=O)CN3CCNC3=O)C)CC2)CC2(C1)CC2F 90544,C(=O)(CCP(C)(C)=O)N1CC(C)C(NC=O)C1.c1(CC(=O)N(C)C)ccccc1 90545,C1(NC(CC2(NC(c3n(CC)ccc3)=O)CCC2)=O)CC2CCCCN2C1 90546,CCCCC(C)CCC(=O)NC1CC1NC(=O)CCc1cncn1C 90547,N1(C(C2CCN(C(C(COCC)C)=O)C2C(C)C)=O)CC2OC(=O)N(C)C2C1 90548,C12(NC(C3CC=CCC3)=O)CC(C1)N(C(C1(C(F)(F)F)CCCC1)=O)C2 90549,C1(C(=O)NC2(CNC(c3ccc(CC)s3)=O)CCC2)CCCCC1F 90550,c1(-n2c(CCc3ccncc3)nc(CCCCC)n2)cccc2nc[nH]c12 90551,c1(CC(=O)N(CC(CNC(CS(CC)=O)=O)(C)O)C2CC2)cc(C)ccc1OC 90552,Cc1cc(Cl)c(CN2CCCC(C(=O)NCc3cncc(Cl)c3)C2)c(Cl)c1 90553,C(=O)(C(C(C)C)OC1CCCCC1)NCCCC(C)NC(CN(S(C)(=O)=O)C)=O 90554,C12(NC(Cc3ccc(OC)nc3)=O)CCC(C1)N(C(C1(C#N)CC1(C)C)=O)C2 90555,C(C1CCc2ncnn21)N(C)C(C1CCCN1S(=O)(=O)CCOC)=O 90556,c1(N2CCC(CN(C(=O)CCCn3c(O)nnc3O)CC)C2)ncnc(Cl)c1CO 90557,C1(C(=O)NCCC2(NC(C(CC=CC)C)=O)CC2)CC2(CCCCO2)C1 90558,c1(C(N(CC(=O)NCCc2cccc(O)n2)C2CCC2)=O)ccc2cccnn12 90559,C(c1ccc(Cl)cc1F)=CC(=O)NC1CN(C(C(C(C)C)C#N)=O)CC1C 90560,CCCCC(CCC)NC(=O)CC1(NC(c2cnn(CC)c2C)=O)CCC1 90561,C12(NC(C3N(C(CN(CCOC)C)=O)CC(F)C3)=O)CCC(CC1O)C2 90562,N1(C(c2c(C)nn[nH]2)=O)CC(N=c2[nH]c(Cl)nc3ccc(Cl)cc23)CC(C)(C)C1 90563,CN1CCC2(CCN(C(=O)C(Cc3cnc[nH]3)NC(=O)C3=C(Cl)CCC3)C2)C1 90564,C(=O)(C(O)CC1CC1)NCC(C)=CC(=O)NC(CO)C1(O)CC1 90565,c1(C(=O)NC2CN(C(CCSC)=O)CC2C(F)F)cc(C)nc(C)c1 90566,C1(C(=O)NCCCCNC(=O)C(O)Cc2ccccn2)CCc2nnc(O)n2C1 90567,n1(CC)ncc2cc(C(=O)N(CCC(C)NC(=O)C(O)C(C)(C)C)C)c(C)nc12 90568,c1(CNC(=O)NC(c2c(SCC)cccn2)(C)C)cnc2ccnn2c1 90569,N1(c2cc(OC)ncn2)CC2(CN(C(C3CN(C4CCOC4)C3)=O)CC2CO)C1 90570,N1(C(CN(CC(C)C)C(c2ccc(N(C)C)nc2)=O)=O)CCC2(CCC(C)C2)C1 90571,c1(CNC(C2CC(NC(c3ccc(O)nc3)=O)C2)=O)sc(Br)c2c1OCCO2 90572,c1(C(=O)NC2C(NC(c3ccc(C(C)=O)cc3)=O)CC2)nccc2cnn(C)c12 90573,Cc1csc2ncnc(NCC3(CCNC(=O)CC4CCCCC4)CC3)c12 90574,C1(C(N2CC(CNC(CC=C(C)C)=O)N(C)CC2)=O)CCC2(CC1)CC2(F)F 90575,N1(C(C(C)C2CCCC2)=O)CC2CCC(N=c3[nH]nc(C(C)(C)C)s3)CC2C1 90576,CCC(C(=O)NCC(C)(C)CNC(=O)C=CC(N)=O)N(CCC)CC 90577,Cc1cnc(N2CCN(C3CCCC3)C(=O)C2)cc1C(F)(F)F 90578,c1(OC)c(CN2CCC(NCCO)CC2)cccc1Cl 90579,N1(C(c2cncc(OC)c2)=O)CC(NC(=O)C(CO)NC(N)=O)C2CCCC12 90580,C(=O)(CC1=CCCC1)NCC1CC(C)N(C(c2cccc(CO)n2)=O)C1 90581,c1(C(N2C(C(=O)Nc3c(C)ccc(F)c3)CC2)=O)ccc2n[nH]cc2c1 90582,c1(OC)cc(C(=O)N(C)CCOCCNC(=O)C(C)CCOC)cc(C)c1 90583,C1(CNC(c2ccc(CC)s2)=O)CCN(C(=O)C2=NNC(=O)C2)CC1C1CC1 90584,c1(C(=O)NC2CC(NC(C(C)c3ncco3)=O)C2)ccc(SC(F)F)cc1 90585,C1(NC(C2CCC(=C)CC2)=O)CCC2(CCCN(C(=O)C3=C(Cl)CCC3)C2)C1 90586,c1(OC)ccc(N(C)C)cc1C(N1CCCC(C)(NC(C2CC23CC3)=O)C1)=O 90587,N1(C(CCc2ccc(C(=O)OC)nc2)=O)CCN(C(=O)CS(C)(=O)=O)CC1C1CC1 90588,C(=O)(C1CCc2c[nH]nc21)NCCCC1CCN(C(C(C)CC2CC2)=O)CC1 90589,CCC(C#N)(CC)C(=O)N(CCCCN(C(=O)CN1CCCS1(=O)=O)C)C 90590,c1(C(C(=O)NC2C=CC(CNC(C(c3ccc(C)o3)C)=O)C2)C)ccncc1C 90591,CC1CCN(C(C2(CF)CCC2)=O)CCN1C(C1C(c2ccccc2)C1F)=O 90592,C(=O)(C(O)CC(C)C)N(CCCN(C(c1sc(C)c(Br)c1)=O)C)C 90593,c1(N(C(c2c(C)nc(CC)nc2C)=O)C)cccc2cnccc12 90594,CC1c2ccccc2OC1C(N1CC2CC2(CNC(=O)CCC2CCCC2)C1)=O 90595,c1(NC(CC2(C(=O)OCC)CCC2)=O)cnc(C)c(NC(=O)CCc2ccoc2)c1 90596,C(=O)(C#CC(C)(C)C)NCCC(C)NC(C1(C)CCCC1(F)F)=O 90597,c1(C(=O)NC2C(C)CN(C(=O)COC3CC(F)(F)C3)CC2)cccc2c1CCC2 90598,c1(C(=O)NCCCC(CCC)NC(C2CCN(C(C)=O)C2)=O)cnc2ncccn12 90599,N1(C(CC=CC)=O)CCCCC1CCN(C)C(c1cc(C(=O)OC)nn1C)=O 90600,c1(C(=O)NCCc2ccc(COC)cc2)cnc(C)c(C#N)c1 90601,Cc1cc(C(N2CC(C)(NC(=O)CNc3ccccn3)C2)=O)ccc1O 90602,C1(C(N2CC(CCC)C(NC(=O)C(c3ccccc3)C)C2)=O)CC(C(C)C)=NO1 90603,C#CCCCC(C)C(=O)NCCn1cc(C(=O)NC2CCN(CC)CC2C)cn1 90604,CC1CN(C(c2cnc3[nH]nnc3c2)=O)CC(C)CN1C(=O)C1=CS(=O)CCC1 90605,N1(C(c2c(C)c[nH]n2)=O)CCOCC1CNC(c1csc(C(F)(F)F)c1)=O 90606,c1(C(C)NC(=O)CN(C(=O)CCCN(C)C)CC2CC2)nccc(O)n1 90607,c1(CC)nc(C)oc1C(=O)N(CCC(=O)NC(c1ccccc1F)C)C(C)C 90608,c1(CCC(=O)N(C(CNC(C(CCC)C#N)=O)C)C)ccc2c(c1)OC(F)(F)O2 90609,c1(C(=O)NC2CCC(NC(CC=CCC)=O)CC2)cnc2c(c1)CCOC2 90610,CC(CCNC(=O)CCOCC(F)F)CCNC(=O)Cc1c(Cl)cnn1C 90611,N1(C(C2(C(C)(F)F)CC2)=O)CCCC1CNC(=O)CCC1CCOC1 90612,c1(C(=O)OCCc2cc(OC)ncc2)ccc(C2CC2)c(Cl)c1 90613,C(C(CC(=O)NC(C)(C)CNC(c1cc(F)c(O)c(Cl)c1)=O)C(F)(F)F)N(C)C 90614,C(=O)(C(F)CC(C)(C)C)NC1(CC)CN(C(=O)CCc2cc(C)n(C)n2)C1 90615,c1(OC)ccc(C(=O)NCC2CC(F)(F)CN2C(c2cc(C)sc2C)=O)c(C)n1 90616,c1(CN2CCCN(C(c3ccc(C)cn3)=O)CC2)ccc(F)c(F)c1Br 90617,C(=O)(C1=C(Cl)CCC1)NC1C(CNC(c2nc(C)oc2)=O)CC1 90618,Cc1c(C(=O)Nc2ccc3c(c2)NCCCN3)sc2[nH]cnc(=O)c12 90619,C1(C(C)C)CN(C(=O)C(N2CCN(C)CC2)C)CCN1C(C1CCCS1)=O 90620,c1(C(=O)NC2C3CN(C(C(C(C)(C)C)SC)=O)CC32)cncc2nnn(C)c12 90621,C=CCCCC(C(=O)N1CC2COCC2C1)NC(c1[nH]ccc1CC)=O 90622,c1(OC)nc(C)c(C(N2CCOCC2CNC(c2cnc(C)[nH]2)=O)=O)s1 90623,c1(C(=O)NCC2C(NC(=O)CN3CCCC3=O)CCCC2)cccn2nccc12 90624,Cc1nn(C)cc1C(=O)NCC1(CO)CCN(C(=O)Cc2cocn2)C1 90625,CC(C(=O)N1CCCCC1CNC(C1(CC(C)(C)C)CC(F)(F)C1)=O)C(C)(F)F 90626,C(c1ccc(F)cc1)=C(C(=O)NCC1N(C(CC)=O)CC(O)C1)C 90627,CC1CCCCC1(C)C(=O)NCC1(NC(=O)C(C)(C)O)CCCC1 90628,c1(CNC(CC)=O)ccc(C(N2CCC(NCCN3CCCC(C)C3)C2)=O)cc1 90629,CC1CC(CNC(=O)CCN2CCCC2)CN1C(=O)CCc1ccn(C)n1 90630,C1(C(=O)NC2C(NC(c3ccc(-c4ncon4)cc3)=O)CC2)CC2(C1)CC2(F)F 90631,C(CCC(=O)NC1CCC(CCNC(c2cocc2Br)=O)C1)OCC 90632,NC1(CNC(c2cc(-c3ccc(F)cc3)ns2)=O)CCCCC1 90633,C1(NC(c2cc(Br)no2)=O)CC2CCCC(C1)N2C(c1cc(CF)on1)=O 90634,C1(C(N(C2CCCCN(C(c3cnccn3)=O)C2)C)=O)CCCC(C)(C)CC1 90635,c1(N2CC(OC)C3(C2)CC3)nc2cccnc2c(=NCCN2CCOC(C)C2)[nH]1 90636,C1(NC(C2CN(C(=O)Cc3nc(Cl)cs3)CCC2O)=O)CCc2ccccc2C1 90637,N1(C(C(CCSC)NC(N)=O)=O)CCCN(C(=O)C(C2CC2)N(C)C)CC1C 90638,C1(O)(C(C)NC(C=Cc2ccc(CC)o2)=O)CCN(C(=O)C#CC(C)C)CC1 90639,N1(C(C)=O)CC2CCOCC2(NC(=O)Cc2csc(S)n2)C1 90640,N1(C(C2(C(=O)NCC)CCC2)=O)CCCC(NC(=O)OC)C(O)C1.C12CN(C1)C2=O 90641,Cc1ccc(F)cc1C1(CN)CC1.N(S(=O)(=O)N(C)CC)CC1CC1 90642,N1(C(C2CCCN(CC)C2)=O)C2CCCC1CN(C(c1cccc(C)n1)=O)CC2 90643,c1(C(=O)Nc2scnc2C2CC2)n[nH]c2ccc(-c3ccccc3O)cc12 90644,N1(C(C2(NC(N)=O)CC2)=O)CC(NC(C2(c3ncco3)CCC2)=O)CC1CO 90645,N1(C(C(CC=C)C)=O)C(C(=O)NCCC(CCC)C2CC2)CCC12CC2 90646,C(=O)(C(O)CCC(C)C)NCC1N(C(CSCC=C)=O)CCC(C)C1 90647,c1(C(N2CCN(C(c3cc(C(F)(F)F)on3)=O)CC2)=O)ccc(O)c(Cl)c1 90648,N1(C(C(c2scc(C)n2)C)=O)CCCC2CN(c3ccnc(C4CCC4)n3)CC12 90649,c1(OC)ccccc1NC(=O)C(C1CCCN(C(=O)CC2CCCCC2O)C1)C 90650,C1(C(=O)OC)CCCCC1C(=O)NCCCCNC(=O)CCC1CCCC(=O)N1 90651,C1(NCCOC)CCOC2(CCC2)C1.c1(N2C(=O)N2)cccc(C)c1C 90652,c1(CC)cc(Cl)ccc1C(=O)N(CC(O)CN(C)C(c1ccnc(F)c1N)=O)C 90653,C(C(C(C)(C)C)NC(=O)CCCNC(c1cccnc1)=O)NC(C(CC)OC)=O 90654,O=C1CCCCC(C(=O)NCC2CCCN2C(=O)C2=NNC(C(F)(F)F)C2)C1 90655,Cc1nc(C(N2CC(F)(CNC(C3CC3(C)C)=O)C2)=O)c(C)s1 90656,N1(C(C(C)=C2CC2)=O)CCC2(CCCC2NC(C2CC(O)C2)=O)C1 90657,c1(N2CC(SC)C2)nc(N(C)CCN)c2c(ncn2C)n1.N1(CCC2CC2)CCCC1 90658,c1(C(N2CC(O)(CNC(=O)Cc3cccs3)C2)=O)ccncc1F 90659,C1(C(N2CCCC2CF)=O)(CC)CCN(C(c2cn(CC)nn2)=O)CC1 90660,CC1CCCCC1NC(c1coc(Cn2cc(CNC(=O)CC#N)nn2)c1)=O 90661,Cc1n[nH]c(=NCCC2CCC(NC(C3CCCC34CCC4)=O)C2)s1 90662,N1(CCC(=O)N(CCN(C(=O)CC2CCSCC2)C(C)C)C)C(C)CCCC1C 90663,Cc1ncnc(O)c1C(=O)N(C1C2CN(C(c3c(C4CC4)cnn3C)=O)CC12)C 90664,N1(CCNC(=O)NC(CC)CO)CCC(C)C1 90665,C1(COC)(CNC(c2csnc2C)=O)CCN(C(c2cc(C#N)cs2)=O)C1 90666,N1(C(C2(NC(=O)CC3CCOC3=O)CC(CO)C2)=O)CC2CCC(C1)O2 90667,CCC(O)C(C)C(=O)NCCCCC1CCN(C(=O)Cn2cnnc2O)CC1 90668,c1(C(=O)NCC2C(NC(c3ccc(CC)cc3F)=O)CC2)ccc(C#N)cc1F 90669,N1(c2cc(Cc3c(C)nc(CCC)o3)ncn2)CCc2cc(Cl)ccc2C1 90670,N1(C(CCCOCCOC)=O)CCCC(CCNC(c2cn[nH]c2)=O)C1 90671,C1(CNC(C2CC3(CC3)CO2)=O)CC2CN(C(c3cccnc3O)=O)CC12 90672,N1(C(C(CC=CC)NC(c2cncc(C=C)c2)=O)=O)CCN2CCCC2C1 90673,c1(-c2nccc(CC)c2)ccc(NC(c2cnn(C(C)C)c2)=O)cc1F 90674,c1(C(=O)NC(CCCNC(CC(=O)NCC#C)=O)(C)C)cccc2nc(S)oc12 90675,c1(CC(N2CC(C(=O)NC3(CC=C)CC=CC3)C2)=O)cc(C)cc(F)c1 90676,N1(C(CN2C(=O)NCC2)=O)CCOC(Cn2cc(CC(O)C3CC3)nn2)C1 90677,N1(C(CC(CC)CC)=O)CCOC2(CCN(C(=O)C(F)(F)CCn3cccn3)C2)C1 90678,C12(NC(c3cc(Cl)cs3)=O)CCN(C(c3ccn(CC(F)F)c(=O)c3)=O)CC1C2 90679,C(CCN=c1ccnc(C(F)(F)F)[nH]1)NCC(C1CCOCC1)OC 90680,Cc1nc(Sc2ncnc(N)c2N)c2ccccc2n1 90681,N1(C(c2c(C)cnnc2O)=O)CCC2CN(C(=O)CC(C)F)C2C1 90682,C1(NC(C2CCc3nccn3C2)=O)COCCN(C(c2cnc(S)nc2)=O)C1 90683,c1(OC)cc(C(=O)NC2CCN(C(c3ccnc(CO)c3)=O)C2C)ccc1O 90684,c1(-c2c(C)nc(F)cc2)cccc2c(C(=O)N=c3cco[nH]3)cnn12 90685,c1(C(=O)NC(C)CNC(=O)C(C)CCO)cc(C2CC2)nc(O)c1 90686,c1(C(N(CC(N2CC(=C)C2)=O)CC#C)=O)cc(F)ccc1C 90687,N1(C(C(C(COC)C)C)=O)CC(CO)C2(C1)CN(C(c1cccc(C)n1)=O)C2 90688,C(=O)(CCCN=[N+]=[N-])NC1CCC(C)(CNC(c2c[nH]c(=NC)s2)=O)C1 90689,c1(CC)[nH]nc(Cl)c1C(=O)NC(C)CC1CN(C(C2CCOC2)=O)C1 90690,c1(C(N2C(CNC(C3N(CC)CC3)=O)C(C)CC2)=O)cc2c(s1)CCCC2 90691,CC#CCCCCNC(c1cnc(CNC(=O)Cc2nonc2C)nc1)=O 90692,CC(C)CCC(=O)NC1CCCC1(C)CNC(=O)CC1CCC12CCC2 90693,C1(NC(CC2(COC)CC2)=O)CC2CCC(C1)N2C(=O)CS(=O)(=O)CC 90694,N#Cc1[nH]c(=NCC2(O)CCN(C(C3CCCSS3)=O)CC2)sc1Cl 90695,C1(C(=O)NCC(CO)NC(c2c(C(=O)OC)c[nH]n2)=O)COCCN1C 90696,CCC1=NOC(C(=O)NCc2nc(CNC(=O)CC(O)c3ccccc3)cs2)C1 90697,c1(C(=O)NC2(C)CC(NC(c3cc(CC)no3)=O)C2)snc(C)c1N 90698,C1(OCC)(OC)CC2(CC(CNC(C)CCc3ccsc3)C2)C1 90699,C(=O)(CCS(=O)(=O)C1CCCC1)NCCC(C)NC(C1SCCS1)=O 90700,C12(C(=O)OCC)COC(COCC3CCN(C(C4CCCCC4)=O)C3)(C1)C2 90701,C1(C(=O)NCCC#C)OCCC1NC(=O)CSCC 90702,C1(NC(c2ncccc2F)=O)CN(C(c2cccnc2)=O)CC2(CC2)C1 90703,N1(C(C2(CC=C)CC2)=O)CCC(COC2CCN(C(C3CCCSC3)=O)C2)CC1 90704,CCC(C)(C)CC(=O)N1CCCC(O)(CNC(c2ccnc(C3CC3)n2)=O)C1 90705,c1(C(=O)NCC(=O)NCC(C)N(C(C(C)N(C)C)=O)C)ccc(F)cc1F 90706,N1(C(C(N2CCSCC2)C)=O)CCN(C(=O)CN2CC(=O)N(C)C2=O)CC1C 90707,Cc1cc(C(N2CC(C(C)(C)O)(CNC(C3CN(C(N)=O)C3)=O)C2)=O)nnc1O 90708,N(C(=NCc1ccn(C(C)C)n1)NCC(F)F)CC(c1ccc(C)cc1)OC 90709,c1(C(c2nnnn2C)NCCCc2c(OCC)cccc2)c(F)cncc1F 90710,c1(OC)ncccc1CCC(=O)N(C)CC1CN(C(=O)C(F)CC2CCC2)C1 90711,c1(C(=O)NC2CN(C(Cc3cn(C)nc3)=O)C2)cc(Br)cnc1C1CC1 90712,c1(CC(=O)NCC2C(NC(C3C(C)(C)C3)=O)C2)c(Cl)cccc1Br 90713,C(=O)(C(CC(C)C)CC(C)C)NCC(=C)CCNC(C1CCC(O)C1)=O 90714,C1(CCC)CN(C(c2ccc(SC(F)(F)F)s2)=O)CCN1C(C12CC(F)(C1)C2)=O 90715,c1(C(=O)NCC(CNC(C(C)O)=O)O)cccc(Oc2ccccc2)c1 90716,c1(CCNC(CC2C(N)CCC2)=O)ccc(Br)c(F)c1 90717,c1(NC(N2C(c3n(C)ncc3)CCCC2)=O)ccc2ncsc2c1 90718,c1(C(N2CCCCC2CO)=O)n[nH]c2cccc(-c3cccc(C(F)F)c3F)c12 90719,C(=O)(CC1=CCCC1)NC1CC(O)(CNC(CC(N2CCCCC2=O)C)=O)C1 90720,C1(n2cc(-c3ncc(C)s3)nn2)CC2CCC1(NC(=O)C(C)n1ccnn1)C2 90721,C1(C(=O)NCC2(O)CN(C(c3cnn(C(F)F)c3)=O)C2)CC12CCC(F)(F)CC2 90722,N1(S(CCC)(=O)=O)CCC(C(C)C(=O)NCCc2cnns2)CC1 90723,c1(CNC(=O)NCCC(C)N(CCC)C)sccc1OC 90724,C1(C(N(C2CCC(NC(C(CC)(C)O)=O)CC2)C)=O)Cc2cc(F)ccc2O1 90725,C1(C)(CNC(C2CC(OCC)C2)=O)CCN(C(C2(C)CCC(=O)N2)=O)CC1 90726,Cc1nc2c(s1)CCN(C(c1nnn(C)c1C)=O)CC2 90727,N1(C(c2cncc(C)c2)=O)CCCC(NC(=O)C2=CCC2)C(F)C1 90728,C(c1cc(Cl)cc(Cl)c1)=CC(=O)NCC1CCCCN(C(C(=O)NC2CC2)=O)C1 90729,Cc1cc(NC(=O)C(CC(C)C)NC(=O)C(=O)C(C)C)c(C)cc1F 90730,N1(C(c2nc(CC(=O)OC(C)(C)C)sc2N)=O)CC(C(=O)O)CC1(C)C 90731,N1(C(Cc2c(C)nc(C)s2)=O)CCN(C)CC1CNC(=O)CN(C)C(=O)C1CC1 90732,N1(C(CC)C)CCN(C(C2COCC2NC(=O)Cc2cncn2C)=O)CC1 90733,C(=O)(C(F)C(C)(C)O)NC1CC(CCC(N2CC(OC(=O)NCC)C2)=O)C1 90734,CN1CC(O)CCC1C(=O)NCC1CCCC1C(=O)NC1(C)CCSCC1 90735,c1(C(CNC(C2CC(OC)C2)=O)NC(C2CCC(N(C)C)C2)=O)ccc(C)cc1 90736,C(=O)(C#CC1(C)CCCO1)NC1(CCC(N2CCC(CN(C)C)C2)=O)CCCC1 90737,n1(CCCN(C(=O)CSC(F)(F)F)C)cc(C(N2CCOCC2)(C)C)nn1 90738,CS(=O)(=O)c1csc(C(=O)NC2CC(C)(NC(C3CC3C#N)=O)C2)c1 90739,N1(C(c2c(CC)con2)=O)CC(NC(=O)Cn2ccc(C(F)F)n2)C(F)C1 90740,C(=O)(C1=CCOCC1)N(CCCNC(=O)C(c1ccc(Cl)cc1)(C)C)CC 90741,CC1(C)CC(NC(c2ccccc2SCCO)=O)CCN(C(C23CCC2C3)=O)C1 90742,C1(CCOC)(NC(C2CCCC2)=O)CCN(C(c2ccccc2COC)=O)C1 90743,c1(SC)ccccc1-c1cn(CCN2CCN(C(C3CC3F)=O)CC2)nn1 90744,C(C(=O)NOCC=CCl)=CC(C)N(C(=O)CN(C)C)C 90745,c1(Cn2c(NC(C)C(C)c3nn[nH]n3)ncc2)ccc(F)cc1 90746,c1(CCC(=O)NC2CC(C)(NC(CN3CCC(OC)C3)=O)C2)ncccc1C 90747,C1(NC(C(n2c(C)cc(C)n2)C)=O)C2CCC1CC(NC(c1ccco1)=O)C2 90748,C1(C(N(CCCNC(c2cc(Cl)c(F)cc2Cl)=O)C)=O)CCC2C(CC1)C2(F)F 90749,N1(C(c2c(C)ocn2)=O)CCC2CCCC12CNC(c1ccc(N)c(Cl)c1)=O 90750,c1(NCCN(C(c2ccc(C)cn2)=O)CC)nc(C(C)C)ccc1C#N 90751,c1(C(C(=O)N(C2C(C)CCNCC2)CC2CC2)=O)cncc2ccccc12 90752,CCCC(C(O)C(=O)NCc1csnc1C)NC(C1(C)COC(=O)N1)=O 90753,C1(CC)CCC(C)N(C(C2C=CCCN2C(=O)Cc2ccc(C)nc2)=O)C1 90754,Nc1cc([N+](=O)[O-])ccc1C(N1CCC(NC(=O)C(O)C(F)F)CC(O)C1)=O 90755,c1(C(=O)NC2CCCC(NC(C3(C)CC4CC4C3)=O)CC2)ccn2nccc2c1 90756,N1(C(c2cnn(C(C)C)c2Cl)=O)CCCC(NC(C2CCO2)=O)C1C 90757,C1(C(N2C3CC(NC(c4c(C)cc(C)o4)=O)C(C3)C2)=O)CCC(C2CCC2)CC1 90758,c1(OC)ccc(Br)cc1C(C1CC1)NC(=O)NCc1coc(C)n1 90759,c1(C(N(CCCN(C)C(C2CC(F)C(=O)N2)=O)C)=O)cnc2c(c1)NC(=O)CO2 90760,C1(C(N2C(CNC(C3(C(C)(C)C)CCC3)=O)CCC2)=O)C(C#N)C1(C)C 90761,N1(CC(C)NC(=O)CC2CCCCC2)CCN(C(C2CCC2C(C)(C)C)=O)CC1 90762,C1(C(=O)NC(c2ccc(C(C)(C)C)cc2)CCC)COC2(CCNCC2)C1 90763,N1(C(C2(CC)CCC2)=O)CC(C2CN(C(=O)CCCOC3CCOCC3)C2)C1 90764,Cc1cnc(CNC(C2CCCN(C(C3CCCCC3O)=O)C2)=O)nc1 90765,N1(CC)CC(C(=O)NC2(C)CC(NC(=O)CNC(c3ccoc3C)=O)C2)CC1=O 90766,CCC(CNC(c1c[nH]nc1CCNC(=O)CCN1CCOC1=O)=O)CCO 90767,C(=O)(C(CC)C(F)(F)F)N1CC(CC(=O)NCC2(OCC)CCC2)OCC1 90768,C(CC(=O)N1CCNC(=O)COCC1)SC.C1(SC)CC1.C(CO)O 90769,C(=O)(C1=CCCC1(C)C)NC1CC(NC(c2cn(CCC)nn2)=O)C12CCC2 90770,Cc1nc(NC2CC(F)(CNC(=O)C=Cc3ccccn3)C2)c(C)c(C)n1 90771,C(c1cccnc1C)=CC(=O)NC(CN(C(c1nncc(CCC)c1)=O)CC)C 90772,C12(C(=O)NC(CC#C)CO)CCCC1N(C(=O)Cc1cc(C)[nH]n1)CC2 90773,N1(C(c2cc(C#N)no2)=O)CCN(C(c2csc(Cl)c2Cl)=O)CC1C1CC1 90774,N1(C(C2N(CC)CCC2)=O)CC2COCCC2(NC(=O)C=Cc2nc(C)cs2)C1 90775,N1(C(CC(=O)NCC)=O)CCC(O)(CN(C)C(C2CSCN2C(C)=O)=O)C1 90776,CC1(C)CN(C(=O)Cc2ccco2)CCC1C(=O)N1OC2CCC1C2 90777,CCC(C)C(O)C(C)C(=O)N1CC2CC1C2NC(C1(CF)CC1)=O 90778,c1(C(=O)NCCCN(C(C2OC3CCC2C3)=O)CC)snc(Cl)c1Cl 90779,c1(CC(=O)N(CC(CNC(c2c(CC)[nH]cc2)=O)(C)C)C)ccc(C)c(F)c1 90780,c1(OCC)cc(C(N2CCC(CNC(=O)COc3ccccc3C)C2)=O)ccn1 90781,Cc1ccc(C(C)C(=O)NCC2CCC2C(=O)NC2(CCF)CCC2)o1 90782,c1(CNC(C2(CC=C)CN(C(c3cc(C)nn3C)=O)C2)=O)sc(C)nc1C 90783,N1(C(CN(C2(C)CCC2)C2CC2)=O)CCC(NC(=O)CC2COC(=O)N2)C(C)(C)C1 90784,C=CCC(CNC(c1ccc(=N)[nH]c1)=O)C(=O)N(CCCCC)C 90785,C(C(O)CC(C)C)NC(c1ccc(-n2cc(C3C(C)=C3)nn2)o1)=O 90786,CC(CNC(=O)CC(C(F)F)c1ccccc1)CN=c1nc(O)c(Br)c[nH]1 90787,N1(C(c2ncc(NC)nc2)=O)CC(C)(C)CC1C(N1CCC(c2cc[nH]n2)C1)=O 90788,C(=O)(C(O)CC[S+](C)C)N1CC(C(C)NC(C(C2CCCCC2)OC)=O)C1 90789,c1(C(N(C2CCN(Cc3cc(C#N)ccc3F)C2)C)=O)noc2c1CCCC2 90790,C(=O)(C#CC1CCCO1)NC1(CO)CN(C(C2CC(c3cn(C)nc3)C2)=O)C1 90791,Cc1cc(C(=O)Nc2cccc(NC(=O)CCN(C)C)c2)c2ccc(F)cc2n1 90792,C1(C(=O)NC2(CC)CCCN(C(=O)Cc3ccco3)C2)CCc2nccn2CC1 90793,c1(C(=O)NCC2C3CN(C(C(C(C)C)NC(C)=O)=O)CC32)c(OC)ccnc1O 90794,C1(C(N(C)CC2CCCN2C(C2CCC23CCC3)=O)=O)CCc2cn(C)nc2C1 90795,c1(C(=O)NC(C2CN(C(C=C(CCC)C)=O)C2)C)ccc2nncn2c1 90796,C1(C)(CNC(c2nc(CC(C)C)sc2)=O)CN(C(=O)C(O)CC2CC2)CCO1 90797,CC(C)CC(O)C(=O)N1CC2CC1CN2C(=O)Cc1cncnc1 90798,C(=O)(C(C)CC(N)=O)N1C(CNC(c2cnc(C)n2C)=O)CCC1 90799,c1(C(N(C)CC2CCCN(C(=O)Cc3ncc(F)cc3F)C2)=O)ccc(=O)n(C)c1 90800,C1(CCOC)CCCCN1C(C1CCC(NC(c2csc(C)c2OC)=O)C1)=O 90801,C1(CNC(Cc2cn(C)nn2)=O)CC(NC(=O)CN2C(=O)CNC2=O)C12CCC2 90802,c1(C(=O)NCC(C)CNC(C2COC(=O)N2)=O)cc(Cl)c(F)cc1Cl 90803,c1(CN2CCC(CNC(c3ccco3)=O)C2)ccccc1F 90804,CN=c1nc(C(N2CCCN(C(=O)C(O)COC)CC2CO)=O)cc(C)[nH]1 90805,C1(C(=O)NC(C#C)CC)CSCCN1C(c1cccc[n+]1[O-])=O 90806,C(C(C)(C)C(=O)N1CC(NC(C2CCCC2)=O)C(C)C1)SC 90807,C#CC(C(C)C)NC(=O)CCN(C(=O)CCC1CC1)CC 90808,CC(C)CC(CNC(c1ncccc1F)=O)NC(=O)CC1(CO)CCCCC1 90809,C1(CC=C)(C(=O)NCC2CC(F)CN2C(=O)CC(=O)OCC)CCOCC1 90810,CC(C)CCCCCC(=O)N1CC(N(C)C(C2CC3CCC2C3)=O)C1 90811,Cc1cc(O)nc(C)c1C(=O)N(CC(C)NC(C12CC(C)C1C2)=O)C 90812,C=CCC(CNC(=O)Cn1nnnc1C)NC(=O)CCNC(=O)C=CCl 90813,CCCCCS(=O)(=O)CC(=O)N1CC2CC1CC2NC(=O)CCc1nncn1C 90814,N1(C(CCCc2cc(C)no2)=O)CC2CCC(NC(=O)C=C3CCC3)(C2)C1 90815,C1(C(=O)NC(c2ccc(Cl)s2)C)CCCN1C1CC1 90816,CC(N=c1[nH]c(=NCC2CCOCC2)[nH]c2c1SCC2)c1nc(O)n[nH]1 90817,Cc1nc2ccccn2c1C(=O)NCC1CCN1C(=O)CC1(O)CCOCC1 90818,C1(C(N(C(CNC(=O)C(F)F)C2CC2)C)=O)(C(=O)NCC2CC2)CCC1 90819,CCCCCC(O)C(=O)NCCN(C(=O)C(=Cc1ccc(Cl)cc1)C)CC 90820,c1(C(N(CC(CC)NC(=O)CC2(O)CCOC2)C)=O)c[nH]nc1OC 90821,C(=O)(C1=COCCO1)NC(C)CCCNC(C12CC(CCO1)C2)=O 90822,c1(C(C(=O)NC2CCOC2)N(CC(COC)C)C)cc(S(C)(=O)=O)co1 90823,c1(CC(=O)NC(=O)CN(C(=O)C(F)(F)F)CCCCNC(N)=O)ccc(Cl)nc1 90824,C(CCN(C)C)(C(=O)NC1(C)CC(N(C)C)C1)NC(c1c(CCC)[nH]cc1)=O 90825,O=C(CS(=O)(=O)NCC1CCCO1)N1CC(NC(C2C3COCC23)=O)C(F)C1 90826,Cn1ccc2cc(C(=O)NC34COCCC3CN(C(C3(Cl)CC3)=O)C4)cnc12 90827,c1(C(N(CCC(C(C)C)NC(=O)COC2CCCOC2)C)=O)csc2cncn12 90828,C(CC(C)C)(C(=O)NCCOCC1CC1)ONC(c1ccc(CC)cn1)=O 90829,C1(C(=O)NC23CC(CNC(c4cc(C)[nH]n4)=O)(C2)C3)Oc2ccccc2OC1C 90830,N1(C(CCCOCCOCC)=O)CC(C)CN(C(C2(SC)CC2)=O)CC1C 90831,C(=O)(C1=NOC(CNC(=O)C(O)C2CC2)C1)N1C(C(N)=O)CC(O)C1 90832,c1(C(=O)NC2CCCC(NC(C#CC(C)(C)O)=O)CC2)ccc2nc[nH]c2n1 90833,C1(CC)CN(C(=O)C2=NOCC2)CCC1CNC(=O)CC1CCC(=O)NC1 90834,C1(CC(=O)NC2CCNC2=O)COCCN1C(c1cnn(C2CC2)c1)=O 90835,C12(C(=O)NC3C(=O)OCC3)COCC1CN(C(=O)CCc1ccccc1)C2 90836,c1(C(=O)NCC(CN(C(C(C=C)(C)C)=O)C)C)cn(CC(C)C)c2ccccc12 90837,C1(S(C)(=O)=O)(N(CCOCCN(C(CN(CCC#C)C)=O)C)C)CCCC1 90838,c1(OC)ccc(NC(=O)CNc2ccc(-c3nc(C)cs3)cc2)c(C)c1 90839,C1(CNC(C(C(C)C)OCC)=O)CN(C(=O)C=Cc2ccc(C)s2)CCCO1 90840,CON=CC(=O)NC(Cc1cnc[nH]1)C(=O)NCC(C)OCCO 90841,Cc1nc2c(N3CC(O)(CNC(c4ccc(Cl)nc4)=O)C3)ncnc2[nH]1 90842,O=C(NN1CCCCC1)c1cccc(NC(c2cccs2)=O)c1 90843,c1(C(N2CC(C)C(CCNC(=O)C=CC(F)(F)F)C2)=O)nccc2ncccc12 90844,C1(C(N(CCCN(C(=O)CNC=O)C)C)=O)CCCCC1F 90845,N1(C(CC(=O)NCC)=O)Cc2nccn2CC(NC(C2CCCSC2)=O)C1 90846,O=C1NCCn2ncc(NC(N3CCC(c4ccc(Br)s4)C3)=O)c21 90847,C1(C)(NC(c2ccn(CCCC)n2)=O)CCCN(C(=O)CCc2nc(=N)[nH][nH]2)C1 90848,C1(NC(=O)CCOCC2CCCO2)CCC(NC(c2coc(C(F)F)c2)=O)CC1 90849,C(CCC(=O)NC(c1ncc[nH]1)C)(C(C)C)NC(C(COC)N(C)C)=O 90850,c1(C(=O)NCC(C(C)C)(C)NC(=O)C(O)C2CCC2)cnc(Cl)cc1N 90851,Cc1cc(CN2CC(O)CC2C(N2CCC(C)C2)=O)cnc1F 90852,c1(C(=O)NCCC(C)(C)NC(c2c(C(C)C)noc2)=O)cn2c(n1)SCC2 90853,CC1(C)NC(=O)CC1C(=O)COC(=O)CCCCN1CCCCC1 90854,Cc1cccc2c(CNC3CCCC3C(=O)NCCc3cc[nH]n3)c[nH]c12 90855,C12(NC(C(CC=CCC)C)=O)CCC(CC1)N(C(=O)CCc1cc(OC)no1)C2 90856,CN1CCN(C(=O)CC2CCCC3CC23)CC1C(=O)NCCc1cnnn1C 90857,C(CC(C(=O)N(CC1CC1)CC1CC1)NC(c1ccncc1N)=O)SC 90858,C12(CNC(C(C)n3cccn3)=O)CC1CN(C(=O)C(CC1CC1)CC1CC1)C2 90859,N1(C(CS(C)(=O)=O)=O)CC(O)(C2(CNC(=O)CC=C(Cl)Cl)CC2)C1 90860,Cc1csc(CCC(=O)N(CC(C)NC(=O)CCn2cc(Cl)cn2)C)c1 90861,N1(C(C(C)CC2CCC2)=O)CCN(C(=O)Cc2cncnc2)CC1CCO 90862,C1(C(=O)NC(C(C)C)CNC(=O)CCc2cnn[nH]2)CCCN(C2CC2)C1=O 90863,C1(NC(C2(NC(N)=O)CC2)=O)CC(O)CN(C(C23CC4CC2C3C4)=O)C1 90864,C1(N(C(CN(C(C2C(OCC)CC2)=O)C2CC2)=O)C)CCC(C(C)O)CC1 90865,C1(F)(C(=O)NCC2CCCC2NC(C2CCC(C(F)F)CC2)=O)CCS(=O)(=O)C1 90866,c1(CC)cccnc1C(=O)NCC(C)CN(C)C(c1ccc(C(F)F)nc1)=O 90867,c1(C(N2C(CNC(c3cccc[n+]3[O-])=O)CC3CC32)=O)cc2c(cn1)OCCO2 90868,C1(NC2CCCC(C(C)(C)C)C2)CC2CC3CC(C2)C1C3 90869,C1(CC(=O)OCC)CCCN(C(C2CSCN2C(c2cccnn2)=O)=O)C1 90870,C(C(CC(=O)NCC1(O)CCC(C)C1)OC)NC(c1cnc(OC)s1)=O 90871,c1(N2CC(C(N(c3c(F)cccc3F)CC)=O)C2)nc(C)nc2c1CCC2 90872,c1(OC)ccc(C(=O)NCCCC(C)NC(c2c(N)cccc2F)=O)nc1OC 90873,C1(CC(=O)NCc2c(C(N(C)Cc3cc(C)on3)=O)occ2)CCCC(C)C1 90874,C1(N(C(C2C(C)CC2)=O)C)CCC2CN(C(=O)CCN3CCOC3=O)CC12 90875,CC1CN(C(=O)CC=C(Cl)Cl)CC(C(=O)NCC2CC=CC2)O1 90876,c1(OCC(C)C)ccc(CNC(=O)CCn2ncn(C)c2=O)cc1 90877,CCC(C)C(O)C(=O)NCCOCCC(=O)NCc1cnn(C)c1OC 90878,CC(C)CCCCC(=O)NCC1CCC1NC(c1cc(C(F)(F)F)ccn1)=O 90879,C1(C(=O)NCCCOc2ccccc2)CC(F)CN1Cc1ccncc1Br 90880,c1(C(=O)NC(CNC(CC2(OCC)CC2)=O)(C)C2CC2)cccn2c(C)nnc12 90881,CC1(CNC(=O)COCC2CCOC2)CCN(C(=O)C(F)C2CCCC2)CC1 90882,N1(C(c2nc(C)[nH]c2C(F)(F)F)=O)CC(NC(=O)Cn2cnnc2O)C(C)(C)C1 90883,C1(CCOC)CN(C(c2cncc(OC)c2)=O)CCN1C(c1cc(C)sc1C)=O 90884,CC(C)C(C)(O)C(=O)NCCCCCNC(=O)Cn1cnccc1=O 90885,CC(=O)C(C)(C)CC(=O)NC1(C)CCN(C(C2C(C)(C)C2(F)F)=O)C1 90886,C1(NC(COCC)=O)COC2(CNC(=O)Cc3nncs3)CC1C2.c1cccnc1 90887,N1(C(c2n(CC#C)cnn2)=O)CCC(CC=C)(NC(=O)CCCCOCC)C1 90888,CC(CNC(c1ccoc1)=O)C(=O)N(C)CCN(C)CCO 90889,N1(C(C(C)OC2CCCC2)=O)CC2C(NC(=O)C3=CCCC3)CS(=O)(=O)C2C1 90890,N#CCCCCC(=O)NCC1CC(O)CN1C(c1ccc(-n2cccn2)nc1)=O 90891,CCS(=O)(=O)C=CC(=O)NCCN1CCC(NC(c2cc(Cl)nc(Cl)c2)=O)CC1 90892,C(C)(C(C)(C)C(=O)N(C1CC(SC)C1)C)NC(CNC(=O)OCC)=O 90893,C1(O)(C(C)NC(=O)CC2(C3CC3)CC2)CCN(C(C2(C#N)CCSCC2)=O)CC1 90894,C1(O)(C(CNC(CCCC)C)(F)F)CCCCC1 90895,C1(C(N2CCC(NC(C(C(CC)C)N(C)C)=O)C(F)C2)=O)Cc2cccnc2C1 90896,c1(CCN(C)C)ccc(C(=O)NOCCC2CCCCC2)cc1 90897,Cc1nn(C)c2c(NCC(C)CO)nc(NC(c3ccc(F)cc3)CF)nc12 90898,C1(N(C(CCN(CC=C)C(C2C3COCC23)=O)=O)C)COC(C)(C)C1 90899,O=S(=O)(c1ccc(NCC(O)C2CC2)cc1Br)NCCc1cccc(C2CC2)c1 90900,Cc1cc(Br)cc(C)c1C(=O)NCCCN(C(=O)CC1CCCO1)C 90901,N1(C(c2cc(CCC)on2)=O)CC(C)CN(C(c2cc(Cl)nc(=N)[nH]2)=O)CC1C 90902,n1(CC(N2C(C(=O)OC(C)(C)C)CC2)=O)nccc1C(=O)OCC12CCCC1C2 90903,Cc1cn2nc(N(C(C)C(C)S(C)(=O)=O)C)ccc2n1 90904,c1(C(N2C(C3CCN(C(=O)CC4(CO)CC4)C3)CCCC2)=O)ccc([N+](=O)[O-])s1 90905,c1(CC)cccc(F)c1C(=O)NC(C1CCCCC1)C(C)NC(=O)COC 90906,c1(C(=O)NC2CCCCC2C(=O)NCC2C=CCC2)cccc(C(F)(F)F)c1F 90907,CCCC(CC)C(=O)NC1CCCC(NC(c2ncc(Br)cc2OC)=O)C1 90908,C(=O)(C(F)CCC(C)(C)C)NC(CC)CC(=O)NCCCN1CCOCC1 90909,CC1CCN(C(c2cc(C(F)F)[nH]n2)=O)C1CNC(=O)CCc1cccn1C 90910,S(=O)(=O)(c1c[nH]ccc1=NC1C=CC(C)(C)CC1)N(C)CCNC(=O)C1CC1 90911,c1(CCC(=O)NC2CC(C(C)NC(C(C)NC(=O)C3CC3)=O)C2)ccc(F)cc1 90912,c1(SCC(=O)NCC2C(NC(CC3(OC)CCC3)=O)CC2)c(Cl)cccc1Cl 90913,N1(C(C(n2c(C)cc(C)n2)C)=O)CCC(CC(=O)NCC(=O)N(C)O)C1(C)C 90914,C1(CNC(c2ccno2)=O)CCCC2(CN(C(=O)Cn3ncc(O)nc3=O)C2)O1 90915,N1(C(C2CC(C)(CC)C2)=O)CCCOC(CNC(c2cc(C(=O)OC)on2)=O)C1 90916,Cc1cccc(C(=O)NC(CNC(c2cnc(OC(C)C)c(Cl)c2)=O)CO)c1N 90917,C1(NC(c2cc(CNC(=O)CCOCC3CC3)no2)=O)CCCC1C1CC1 90918,C(c1cccnc1)=CC(C)NC(=O)CCCC1CCCC1 90919,O=S(=O)(c1ccc(N2CCN3CCC2C3)c(F)c1)NC1CCc2ccccc21 90920,c1(NC(N2CCC3(C(N4CC5(CCC5)C4)=O)CC3C2)=O)cc2cccc(Br)c2[nH]1 90921,CC1CC(N(C)C(c2ccc(CNC(=O)C=C3CCOCC3)nc2)=O)CCN1C 90922,N1(C(c2csc(C3CC3)c2)C(=O)NC2(C)CC2)Cc2ccc(Br)cc2CC1C 90923,C1(OC)CC(C(=O)NC(C2CSC2)C)N(C(c2snnc2C)=O)C1 90924,C(CC(C(=O)NC1CC(C)(O)C1)NC(c1cccc(F)c1)=O)OCC 90925,N1(C(C(C)(C2(C)CC2)OC)=O)CC(CO)C2(C1)CN(C(c1conc1C)=O)C2 90926,C(CCCN(C(=O)CC1CCC1C)C)NC(COCCOCC#C)=O 90927,C=CCCC(F)(F)C(=O)NCCCC(C)(C)NC(C1CCS(=O)(=O)N1)=O 90928,C1(CC(=O)NC(CCCCSC)CO)SC2=NCCN2C1=O.C1(C)(C)C=CC(=O)N1 90929,c1(C(N2CC(NC(C3(C(N)=O)CCC3)=O)CC(C)C2)=O)c(F)ccc2c1OCO2 90930,c1(C(=O)NCc2ccc(Cl)c(Cl)c2)cc2c(Cl)cc(F)cc2[nH]1 90931,N1(C(CCN(CC(F)(F)F)C)=O)CC(C(N)=O)(CNC(=O)C=C(Cl)Cl)C1 90932,C1(F)(CNC(C(CCC)(C)C)=O)COCCN(C(c2cc(O)cc(Cl)c2)=O)C1 90933,c1(C(=O)NC2(C)CCC(NC(c3ccsn3)=O)CC2)cc(Cl)c(F)cc1O 90934,CCCCCC(F)C(=O)N1CCC1CC(=O)NCCc1cccs1 90935,N1(C(C(C(CC)C)O)=O)CCOCC(F)(CNC(=O)C=Cc2sccc2C)C1 90936,c1(C(=O)NCCC(C)(C)NC(C(CC=C)CC)=O)cnn2c1OCC(OC)C2 90937,C(=O)(CS(=O)(=O)C1CC1)NC1C2CC(CNC(=O)Cc3cnc[nH]3)(C2)OC1 90938,C1(NC(C(CC)n2cccn2)=O)C2CN(C(=O)CCC(=O)N3CCOCC3)CC12 90939,C1(C(C)C)(C(=O)NCC(C)NC(c2ccnn2C2CC2(F)F)=O)CNC(=O)C1 90940,c1(C(=O)NCC(CC)NC(=O)Cc2nonc2C)ncc(F)cc1F 90941,c1(C(=O)OCC(CC(CC)C)=O)cc2cc([N+](=O)[O-])ccc2[nH]1 90942,c1(C(=O)NCCCCC2CN(C(CSCCCC)=O)C2)cc(Cl)c[nH]1 90943,CC1C(NC(=O)NCCOc2ccc(CC#N)cc2)C2CCN1CC2 90944,c1(CCNC(=O)NCCC)ccc2cnn(C)c2c1.c12ccc(cc1)[nH]c2=O 90945,C1(CNC(C=CC(C)C)=O)CCCCN(C(c2cc(C(N)=O)c[nH]2)=O)CC1 90946,C#CCC(CC(F)F)C(=O)NC(CC)CCC(N1CC2OCCOC2C1)=O 90947,c1(CN(CCN(C(c2c(CC)ccs2)=O)C)C)nccc(OC)n1 90948,CCC(C(=O)NC1(CN(C)C(C2CC2C(F)(F)F)=O)CC1)NC(C)=O.C(F)(F)F 90949,C1(NC(c2c(C)cnn2C(C)C)=O)CC(C)CN(C(=O)COC2CCC2)C1 90950,c1(CC(=O)NC2CC(F)(C(=O)OC)C2)cc(Br)ccc1C 90951,c1(CC(=O)NCCCOC(C)(C)C)ccnc(Cl)c1F 90952,N1(C(C2(C)N(C)CC(OC)C2)=O)C2CCC1CN(C(C1CN(C)C1)=O)C2 90953,c1(CCC)ccc(C(=O)N(CC(C)N(C)C(c2cc(C3CC3)nn2C)=O)C)cc1 90954,c1(NC(C2C=CCN2C(=O)CC(O)c2ccccc2)=O)nc(Cl)c(Cl)cc1Cl 90955,CCS(=O)CC(=O)N1CCCCC1CCCNC(=O)CC1OCCO1 90956,C1(CN(C)C(C2CCNC2=O)=O)COCCN1C(c1ccc(C(F)F)s1)=O 90957,c1(C(CNC(=O)CCC2CCCO2)N(C(=O)C(F)=CCCF)C)ccccc1 90958,c1(C(=O)NC2CC(C)(NC(C=C(CC)C)=O)C2)cccc(C(C)=O)c1 90959,C(=O)(C#CC1CCCCC1)N(C)CC1CCCN1c1nnc(C2CCCC2)s1 90960,N1(C(CC=CC(C)(C)C)=O)CCOCC1CCNC(C1CCC(F)CC1)=O 90961,c1(C(=O)NCC(CN(C(CCCC=C)=O)CC)(C)C)cc(C)nc2c1cnn2C 90962,CCCCC(C(=O)NCc1occc1C(=O)NC1CC2CCC(C1)N2C)C(C)C 90963,C1(C(N(C(CO)C2CC2)C)=O)CC(C)(C)CCN1C(c1csc(O)n1)=O 90964,CCCC(C)(C)CC(=O)NC(CCF)C(=O)N1CC(C)(C)C1C(C)C 90965,Cc1cc(C2CC2)ccc1C(=O)NCC1CCN(c2cccc(Cl)c2)C1 90966,c1(CNC(=O)NCC(C2CC2)N(C(c2c[nH]nc2CO)=O)C2CC2)ccccc1 90967,C1(C(=O)OC)CCC2(CCC2)N(C(=O)C(=O)CCC2CC(C)(C)NC2=O)C1 90968,c1(NC(c2c(OCC3CC3)cccc2F)=O)c(Br)cc([N+](=O)[O-])cc1Br 90969,C1(C(N(C)CC2CCN(C)C2)=O)C(C2CC2)CCN1C(=O)CC12CCC(CC1)C2 90970,CCCC(C(=O)NCC1=CCN(C(c2[nH]nc(OCC)c2Cl)=O)CC1)C(C)C 90971,c1(C(=O)NC2CN(C(CC(CC)O)=O)C2)cnc2c(c1)NCC2 90972,Cc1ccc(CCNC(C)(CNC(=O)CCCC2CCCO2)C2CC2)cc1 90973,c1(-c2scc(C)n2)cccc(NC(=O)N(CCCNc2cn(CCF)cn2)C)c1 90974,n1(CC(=O)NC2C=CC(CNC(C3CC(O)C3)=O)C2)nnnc1-c1ccsc1 90975,N1(C(C(CC=C)(C)C)=O)CCN(C(C2(c3ccc(Cl)cc3)CC2)=O)CC(C)(F)C1 90976,CS(=O)(=O)C1CN(C(c2csnn2)=O)CC1NC(c1cc2ccccc2[nH]1)=O 90977,c1(C(=O)NCC(N(C(C(N2CCOCC2)C)=O)C)C2CC2)cc(C(F)(F)F)no1 90978,Cn1ccnc1CCC(=O)NCCC(O)CNC(=O)COC1CC(F)(F)C1 90979,c1(C(=O)NCC2CC(C(=O)NC(C3CCCO3)COC)C2)cncc(NC)c1 90980,C(=O)(CC(C(F)(F)F)n1ccnc1)NCC(CC)NC(c1cc(C)c(C)nn1)=O 90981,c1(OC(C)=O)ccc(C(N2CC(NC(=O)CN3CCCC3C)C(O)C2)=O)cc1 90982,c1(C(=O)OC)cnc(N(C)CCN(C(=O)CC2CC2c2ccccc2C)C)nc1 90983,c1(C(N(CCC)CCNC(=O)C(F)C(C)(C)O)=O)cnc2onc(C3CC3)c2c1 90984,c1(OC(CC)C)ccccc1C(N1CCCCC1CNC(=O)CN(C)C(C)C)=O 90985,N1(c2nc(C)cc(NC3CCN(CCC)C3)n2)Cc2cnn(CCO)c2C1 90986,C1(NC(C=C(C)C)=O)CCCC(NC(c2ccn(CC(F)(F)F)n2)=O)C1 90987,N1(CCC(=O)N(C(C)C)CCNC(=O)CCCn2cncn2)CCOCC1=O 90988,C=CCC(C)C(=O)NCCn1cc(C(=O)N(C)Cc2cnco2)nn1 90989,C1(CC)CN(C(C2(c3ccccc3OC)CC2)=O)CCN1C(=O)Cn1cccc1 90990,c1(C(=O)NCCCN(CCCOC)C(C)C)ccc(Br)c(N)n1 90991,C(CC(C)C)(C(=O)NC(Cc1ccco1)CO)NC(C(CCOC)OC)=O 90992,c1(C(N(C)CC2N(C(C(CCC)N(C)C)=O)CCOC2)=O)cccn2cncc12 90993,C(C)(C)(C(=O)N1CC(OCC(=O)NC(C2CCOC2)CO)C1)SC 90994,C1(C(=O)Nc2c(CC)cccc2)CC(C)(C)CCN1C(=O)CCn1ccnn1 90995,CCCC(CC)CC(=O)N1CCC(C)CC1CNC(c1ncc(OC)cc1F)=O 90996,N1(C(C2CNC(=O)O2)=O)CCC(CNC(C2(CC3CC3)CC2)=O)C(F)(F)C1 90997,c1(CC)ccc(F)c(C(=O)NC2CCCC2CNC(=O)C(C)C2=CCCC2)c1F 90998,c1(C(N2C(CNC(C(C)OCCN(C)C)=O)CC2)=O)nc2ncccn2n1 90999,C12N(CC13CCOCC3)C(=O)C=CCn1cc2nn1.C(c1ccccc1)=CC 91000,N1(C(c2c(C)cns2)=O)CC(O)(C2(CNC(c3cc(F)cc(C)c3N)=O)CC2)C1 91001,CCCCC(CNC(=O)CN(C)CCC)NC(=O)COc1ccc(COC)cc1 91002,C1(CN(C(c2cc(CC)sn2)=O)C)COCCN1C(C1CCCSC1)=O 91003,CN1CCC2(C1)CN(C(=O)NCC1CC1(Br)Br)CCO2 91004,N1(C(C=C(CC)C)=O)CCC(O)(C(C)NC(=O)CN2CCCC(N(C)C)C2)CC1 91005,C1(NC(CCOC)=O)CN(C(c2cnc(C(F)(F)F)s2)=O)C2(CCOC2)C1 91006,C(=O)(CC(C(F)(F)F)OC)N1CC(CC)N(C(=O)C(O)C(C(C)C)OC)CC1 91007,N1(C(C(C2CCN(C(C3CCCOC3)=O)CC2)C)=O)CCc2cc(C#N)ccc21 91008,N(C1CCc2cc(CNC(c3cccnc3)=O)ccc21)C(C1(C)CC(C)C1)=O 91009,CC(C)C(O)CCNC(c1ccc(OCC2CC2)cc1)(c1nnnn1C1CC1)C 91010,C1(C(=O)NCC(CC)CO)(CNC(=O)C(C)C2CCC2)CC2(CC2)C1 91011,C(=O)(CCC(C)(C)N(C)C)NCC(C1CCCN1C(=O)CC1CCCCC1)(C)C 91012,C(CC(C(=O)N1CCCC1CCCNC(=O)C=C(Cl)Cl)NC(N)=O)SC 91013,C1(C(=O)NC(CC=C)CNC(C2CCCCS2)=O)Cc2ccccc2C1 91014,c1(C(N2CCOCC(NC(CC3(COC)CC3)=O)C2)=O)c2c(nn1C)CCCC2 91015,c1(C(=O)NC(C2CCOC2)C)n[nH]cc1NC(c1cc(Br)c[nH]1)=O 91016,Cc1nc(C(=O)N(C(C)CCNC(c2sc(C3CCCO3)nc2C)=O)C)c(C)o1 91017,N1(C(C(CCC)C)=O)CCC(C(F)(F)F)C(NC(c2ccc(Cl)c(O)c2)=O)C1 91018,CCS(=O)(=O)CC(=O)NC1CN(C(=O)CC2CC2C(F)(F)F)CC1OC 91019,C1(O)(CCNC(C(c2n(C)ncc2)O)=O)CCN(C(=O)CCc2c[nH]c(=N)[nH]2)C1 91020,N1(C(c2n(C)cc(Cl)c2)=O)CCN(C(=O)C(C)(C)c2ccccc2)CC1C(F)F 91021,N1(C(COCC=C)=O)CCCCC(F)C1.C1(C)(C(=O)NCCCCCC)CCCC1 91022,Cc1ccc(S(=O)(=O)NC(=O)C(C2CCCOC2)N)cc1 91023,C(=O)(C1=C(Cl)CCC1)N1C(CC)C(NC(C2(CCN(C)C)CC2)=O)CC1 91024,N1(C(=O)NCC2CC(F)(CNC(CC(C)c3ccco3)=O)C2)C(=O)CN(C)C1=O 91025,c1(C(=O)NC2CCC(CNC(c3ncc(C)nc3)=O)C2)ccc(C#N)cn1 91026,CC1CC(CNC(=O)C=CCN2CCCC2)CN1C(=O)CC(=O)NC1CC1 91027,c1(-c2cn(CCCCNC(C(C3CC3)OC)=O)nn2)cccc(C#N)c1 91028,C1(C(=O)NC2C(CNC(C3(C(=O)NC)CC3)=O)CC2)CCc2cnc(C)n2C1 91029,C(CC)(CCC(=O)NC1C=CCCC1)NC(c1nccc(CC)c1)=O 91030,C1(NC(CN(C(C(C)C)=O)C)=O)CC2(C1)CC2NC(C12CC(F)C1C2)=O 91031,N1(C(C2CCC(C)C2)=O)CCC2(CC1)CCN(C(c1ccc(C(F)F)nc1)=O)C2 91032,C1(C(N2CCC(C(C#C)C)CC2)=O)CCC(C)N(C(c2scnc2C)=O)C1 91033,N1(C(C(C2CC2)OC)=O)CC(C)(C)OCC1CNC(=O)C#CC(C)(C)C 91034,c1(C2(C(=O)NCC3(SCC)CC3)CC2)cccs1.C12CC1CNC2=O 91035,n1(C2CCN(C(C3(c4nnnn4C4CCCC4)CC3)=O)C2)ccc(O)nc1=O 91036,N1(C(COCC)=O)CCC(C)(C)CC1C(=O)N(C1CCSC1)CC 91037,N1(C(CC=C=C)=O)CCC(N(C)C(c2cnn(-c3cccnc3)c2)=O)CC1 91038,C=CCC(F)(F)C(=O)NC1(F)CC(NC(C2CCCN(C(=O)NC3CC3)C2)=O)C1 91039,C1(C)(CNC(CCC=C(C)C)=O)CN(C(C2C3CCCCC23)=O)C(C)(C)C1 91040,C(=O)(CC(C(C)C)OCC)N(CC(CN(C(c1ccc(C#C)o1)=O)C)O)C 91041,n1(CC(N2CC(NC(CC(C)c3cnn(C)c3)=O)C(F)C2)=O)cccc(O)c1=O 91042,c1(OC2CC(CCOC)C2)ccc(NC(=O)CC(C)O)cc1 91043,CCCC(C)(O)CC(=O)N1CCN(C(=O)C(=Cc2ccco2)C)CC(CO)C1 91044,Cc1ccc(OC(C)(C)C(=O)NC2CN(C(C3CC(O)C3)=O)C3CC23)cc1 91045,Cc1ccc(C(=O)N(C)CCNC(c2ncccc2N)=O)c(F)c1F 91046,C(=O)(C(C)(C)C(=O)N(C)C)N1CCCC(CN(C(C2C(=C)CC2)=O)C)C1 91047,N1(C(C(CC#C)C)=O)CCN(C(=O)CCC2CCC(=O)N2)CC12CCC2 91048,c1(C(=O)NC2CN(C(c3c(C)ncc(C)c3)=O)CC(O)C2)cnc2[nH]cncc1-2 91049,CC(C)C(F)C(=O)NCC1CCC(C(=O)NCCC2COCCO2)CC1 91050,c1(CC)c(C(=O)N(CCCN(C(=O)C=Cc2ccsc2)C)C)oc2ccccc12 91051,CC1CC(CN(C2CCN(NC(C=O)=O)C2)CCO)CCS1.C12CC3CC1C2C3 91052,c1(C(=O)NCC(CN(C(C2CC(C)OC2=O)=O)C)(C)C)cccc2c1CCC2 91053,c1(CC(=O)O)ccc(OC(F)(F)F)cc1.CC(C)CC1CC1NC1CNC1 91054,c1(C(N2C3CCN(C(CSC)=O)CC3CC2)=O)c[nH]c2c(F)c(F)ccc2c1=O 91055,S(=O)(=O)(c1cnccc1N1CCC(Cc2ccccc2)C1)N(C1CCS(=O)C1)C 91056,c1(C(=O)NCCN(C(=O)CC2(O)CCOCC2)C)ccc2ccncc2c1 91057,N1(C(CN(S(CC)(=O)=O)C)=O)CCC2CN(C(c3cc(C)c(N)cc3F)=O)C2C1 91058,C(=O)(C#CC1CCC1)NC(C(=O)NCC(c1nncn1C)C)C1CCC1 91059,C(=O)(C1=CCCCC1C)NCCCN(C(c1cc(OC)c(Cl)cc1)=O)C1CC1 91060,c1(C(N2CCC(N(C(=O)Cn3cncc3C)CCC)C2)=O)nccnc1CC 91061,N1(C(=O)CC2OCCO2)CCOCC(C(N2CC(n3cnnn3)C2)=O)C1 91062,C1(NCc2c(C(=O)OC)n[nH]c2)CN(C(C2(OC)CCSC2)=O)CC12CC2 91063,c1(C(=O)NCC(n2cc(-c3cccc(F)n3)nn2)C)cnc2ncc(Br)cc2c1 91064,C1(C#CC(=O)NC(c2ccc(C)cc2)CNC(c2cc[nH]n2)=O)(CC)COC1 91065,C(C(C)(C)CC(=O)NC1CCCC1NC(c1cncc(N(C)C)c1)=O)OC(C)=O 91066,C12(C(=O)NCCN(C(=O)C(F)C3CCOC3)CC)CCC(C(=O)OC)(CC1)CC2 91067,C(=O)(C1=CCC(C(F)(F)F)OC1)Nc1ncc(CCOC)s1 91068,N(C1CCOc2c(Br)cccc21)C(CCC)(CCC(N)=O)c1nnnn1CCC 91069,c1(C(=O)NCC2C(NC(=O)C3=CCCC3)C2)cc2ccccc2n1CC(F)(F)F 91070,C1(OCCNC(CC2CC(OC)C2)=O)CCN(C(=O)Cc2ccnc(O)c2)CC1 91071,c1(C(N2CC(NC(C(C3CCOC3)OC)=O)C2)=O)cnn(C(F)F)c1 91072,N1(C(C(CC=C)C)=O)CC(C(C)(C)C)CC(CNC(C2(n3cccn3)CCC2)=O)C1 91073,CC1CN(C(C)=O)C(C)CN1C(=O)CC(=O)OC(C)(C)C.C(C1CCOCC1)=C 91074,c1(C(=O)NC2C(CNC(=O)C=Cc3ccccn3)CCC2)cc2cccnc2s1 91075,CC1CCC(C)C1NC(=O)CC1CN(C(C2CC(CF)C2)=O)CC1C 91076,c1(C(=O)NCCC(C)N(C)C(c2ccn(C3CCC3)n2)=O)ccc(P(C)(C)=O)o1 91077,C(=O)(C(C)(C)CS(N)(=O)=O)N1CCCN(C(C2=CC(Cl)=C2C)=O)CC1C 91078,C1(CC(=O)NC)CN(C(=O)Cc2ccc(O)cn2)CCN1C(=O)CN(C)C 91079,N1(C(CCC(C)NC(c2n[nH]cc2Cl)=O)=O)C2CCC1CC(O)C2 91080,C1(O)(CN(C(C(CC)n2cccn2)=O)C)CCN(C(c2ncncc2N)=O)CC1 91081,CCCC(CNC(C1CN(C)CCO1)=O)C(=O)Nc1cnc(Cl)cc1C 91082,CCC(C)(C(=O)N1CCN(C(=O)C(=O)NCC(F)F)C(c2cn[nH]c2)C1)C(N)=O 91083,N1(C(n2cc(-c3cn(C4CC(O)C4)nn3)cn2)=O)CCCC(C(F)(F)F)CC1 91084,c1(C(N(C2CN(C(CCC=C)=O)CC2F)C)=O)ccc2nc(O)[nH]c2c1 91085,N1(C(C(C)(C)c2ccccn2)=O)CC(NC(c2ccc(F)cc2N)=O)CC(O)C1 91086,c1(OC)ccc(CN2CC3(CCN3C(=O)Cc3cc(C)n(C)n3)C2)cc1O 91087,C1(NC(C2(CC)CC2)=O)CCC2(CCN(C(c3cccc4oncc34)=O)CC2)C1 91088,Cc1c(CCC(=O)NC(CNC(=O)CN(C)C)C(C)C)c(O)nc2[nH]nc(O)c12 91089,c1(C(N(C2CCN(C(C34CCCC3C4)=O)C2)CC)=O)cnc2c(c1)CCC2 91090,c1(C2(C(N(C(CNC(c3nc(CCC)sc3)=O)C)C)=O)CC2)ccc(C)cc1 91091,C1(C)(C(=O)OC)C=CCN1C(C1OCCC1CNC(=O)Cc1cnn(C)c1)=O 91092,C1(C(=O)NC2CN(C(=O)NCC)C2)CCCCC1NC(=O)CC1CC(N(C)C)C1 91093,C1(C(C(=O)NCC(C2CC2)NC(c2ccncc2C(F)F)=O)F)CCCCCC1 91094,CC(C)C(CCN(C)C(C1CC2CCC2C1)=O)NC(=O)CN1CCNC1=O 91095,C=CCC(C)(C)C(=O)NC1CCCN(C(c2ccc(CC)c(N)c2)=O)C1 91096,C(=O)(CCN(OC)C(=O)C(C1(O)CCCCC1)NC(=O)CCC(C)(C)C)OC 91097,C(=O)(CC(C)CCc1ccccc1)NCC(CNC(C1CN(C(C)=O)C1)=O)(C)O 91098,N1(C(CC(CC)C2CC2)=O)CC2CCC(C1CO)N2C(c1cccnn1)=O 91099,C(CCC(CO)NC(=O)CC(C)(C)C)NC(c1scc(C)c1)=O 91100,c1(C(=O)OCC)onc(C)c1NC(C1CCCCN1C(=O)CCNC(C)=O)=O 91101,CCCCC(CN=c1nc2cccc(Br)c2c[nH]1)NC(C1CC2CC2CC1C)=O 91102,N1(C(c2cn(C(C)C)nc2)=O)CCC2(CC1)CC(CNC(=O)CC(C)CF)C2 91103,N#Cc1ccc(CCC(N2CC3C(NC(C4CCOC4)=O)C3C2)=O)c(F)c1 91104,c1(C(=O)OC)cc(I)cnc1NC(C1CC(O)CN1C(c1ccc(CO)o1)=O)=O 91105,CN(C)S(=O)(=O)N1CC(C(=O)NC2CC3(COC(C)(C)C3)C2)C1 91106,c1(CC)nc(C)c(C(N2CCC(C(=O)NCCC(C(C)C)OC)C2)=O)o1 91107,c1(C(N2C(CNC(C3CC4CC4C3)=O)CC(O)C2)=O)ncc(Cl)cc1Cl 91108,S(=O)(=O)(c1ccc(Cn2cc(C)cn2)cc1)N1C2CN(C(C(CC)=O)=O)CC21 91109,c1(SCC(=O)NC(C(C)C)C(C)NC(c2cocn2)=O)ncnc2[nH]cnc12 91110,CN=c1ccc(C(=O)NC2C3CC(NC(c4cnn(CC5CC5)c4)=O)CC23)c[nH]1 91111,C(CCCC(=O)NCC#CC(=O)NOCC1CCOC1)NC(N)=O 91112,c1(CC)c(C(=O)NC(C)CCCCNC(c2cnc[nH]2)=O)csc1C 91113,c1(C(=O)NCC2CCN2C(C2CCCO2)=O)ccc(C23CC(OC)C2C3)cc1 91114,C1(C)(COC)CC(NC(=O)Cc2ccc(Cl)c(Cl)c2)CN1C(=O)CN(C)C 91115,c1(C2(NC(CCC3CCCC(=O)N3)=O)CCCC2)ccc2c(c1)OCCO2 91116,C=Cn1ncc(C(N2CCC(O)CC2C(=O)NCCC2CC2)=O)c1N 91117,N1(C(C2C(C)(C(C)C)C2)=O)CCCC(NC(c2ccc(=O)n(O)c2)=O)C1C 91118,c1(C(=O)NCC(N(C)C(c2cocn2)=O)C2CC2)cccc(F)n1 91119,C1(NC(c2c(C)snn2)=O)CC2(CCN(C(c3sc4ccsc4c3C)=O)C2)C1 91120,C1(C(=O)NCCC(CC)C)CC2(CC2)CN1C(c1cc(C)sc1N)=O 91121,N1(C(C(CC)CN(C)C)=O)CCN(C(=O)COC2CC=CC2)CC1CF 91122,c1(OC)ccnc(C(=O)N(CCCNC(c2c[nH]c(=N)o2)=O)C)c1C 91123,Cc1cc(OC2CN(C(=O)NCc3ccc(I)cc3C)C2)cc(C)c1 91124,c1(NC2(CC(=O)OC)CCOC2)ccc(C2(C(=O)O)CC2)cc1 91125,C1(NC(C2C(C)OCC2)=O)CC2CCC1CN(C(c1cc(F)ccc1O)=O)C2 91126,C(C(C)(O)C1=CCC2CC1C2(C)C)NC(Cc1cn(CC)nn1)=O 91127,C(=O)(CCCCC(N)=O)N1C2CC(CNC(C(C)CC3CC3)=O)C1CC2 91128,c1(C(=O)NCC2N(C(c3c(CC)ocn3)=O)CC2)cc(F)ccc1-n1cccn1 91129,N1(C(CC2C(C)CCN(C(=O)CCCC3CCCC3)C2)=O)C2CCCC1COC2 91130,C1(C(=O)NCC2=CCN(C(CC=CC=C)=O)CC2)Cc2cc(C)ccc2S1 91131,Cc1ccc(C2CC2C(N2CCN(C(=O)CN3CCSCC3)CC2)=O)cc1 91132,N1(C(C2N(C(CC(C)C)=O)CCC2)=O)CCN(c2cncc(Cl)n2)CC1 91133,CCC(C)CC(=O)C(=O)NC(c1ccccc1)C(C)NC(c1cscc1Cl)=O 91134,C1(NC(C2C(C(C)C)C2)=O)CC2CC(NC(=O)C(C)(Cl)Cl)CC12 91135,c1(C(=O)NCC(c2ccccc2)NC(C=CCN(C)CC)=O)ccc(N)cc1C 91136,C1(C(=O)NC(C(=O)NCCNC(=O)OC)CN(C)C)COCC1(C)C 91137,c1(C(N)=O)ncccc1NC(C1CCC(NC(c2cnn(C3CC3)c2)=O)C1)=O 91138,Cc1cc(OCC(=O)NCCC(C)CCNC(C2CC(C)(O)C2)=O)cc(C)c1 91139,C1(CC)CC(C(=O)Nc2cccc(C(F)(F)Br)n2)CCC1=O 91140,c1(C(=O)OCC(=O)NC(c2ccco2)C)cn(C)c2ccc(Cl)cc12 91141,c1(C(=O)NCCCCCCC(C)C)cc(F)ccc1S(C)(=O)=O 91142,CCCC(C(=O)NC1CCCC(C(=O)NC(C)(C)CCCO)C1)OC 91143,c1(C(=O)NC2CCCC2NCc2ccccc2)cccc2nc(Cl)sc12 91144,C#CCCCC(C)C(=O)NC(C1(O)CN(C(c2ccsc2C)=O)C1)C 91145,C1(COC)(NC(=O)CCn2ccc(C)n2)CCN(C(C2CC(C#N)C2)=O)C1 91146,C1(C(=O)NCCNC(C2CCN(C3CC3)C2=O)=O)CCCc2ccccc2C1 91147,N#Cc1cc(F)c(C(N2CC(F)CC2C(=O)NCC2CCC2)=O)c(Cl)c1 91148,CCC(F)C(=O)NC1CCC1NC(=O)Cn1cc(C(=O)N(C)C)nn1 91149,N1(C(C=CC)=O)CCC2(CC1)CC(NC(=O)CC1CC3(C1)CC31CCC1)CCO2 91150,C1(C(N2C(C)(C)CCC(C(=O)OCC)C2)=O)CCc2ncc(Br)n2C1 91151,C1(C(N2CC3CC2CN3C(=O)OC(C)(C)C)C(=O)NC)CC2OC(C)(C)OC2C1 91152,c1(C(=O)NCC(Cl)Cl)cc(CNC(c2cnn[nH]2)=O)cs1 91153,C1(C(=O)NCC2N(C(c3nc(CC)oc3)=O)C3C(C2)C3)CCC(C)(F)CC1 91154,C1(C(=O)NCC(C)CNC(C2CC23CCC3)=O)CCc2ccccc2C1 91155,N1(C(CCc2c(C)n(C)nc2)=O)CC(CO)C2(C1)CN(C(C1CC(C)(O)C1)=O)C2 91156,C1(NC(CCSCC)=O)CN(C(=O)CSc2nncn2C2CC2)C2CC12 91157,C1(C)(COC)CCCN(C(=O)C(CCCOC)NC(=O)C(CC(C)C)OC)C1 91158,N1(C(C2N(C(C3=CCC(C)CC3)=O)CC=C2)=O)CCc2nncn2CC1 91159,N1(C(C2CCN(C)C2)=O)CC2CN(C(=O)CC3CCC(=O)NC3)CC2C1 91160,C1CC(O)C(=O)N1.c1(C(c2nnnn2C(C)C)NCCOC)cnnn1C 91161,C1(C(=O)NCC2(NC(c3cc(OC)ns3)=O)CC2)(COC)CCCO1 91162,N1(C(C(C(C)C)N(C)C)=O)CCCC(C)(CNC(=O)CC2(C)CCCC2)C1 91163,c1(C(N2CC(CN(C(=O)Cc3ncc(Cl)s3)C)C2)=O)ccc(OC(F)(F)F)cc1 91164,Cn1cc(C(=O)NCC23CCC(C)(CC2)OC3)c(O)nc1=O 91165,N1(C(C(C2CCOCC2)C)=O)CCN(C(=O)CC2OCCO2)CC12CCC2 91166,N1(C(=O)C(F)CC2CCOC2)C2CCCC1CN(C(C13CCC(CC1F)C3)=O)C2 91167,C1(C(=O)NCC2(CNC(C(C)C(=O)N3CCOCC3)=O)CC2)CCS(=O)(=O)N1C 91168,N1(C(c2ccc(OCCCl)cc2)C(=O)NCCOC)CCCC(N=[N+]=[N-])C1 91169,CCC(C)C(C)C(=O)N1CCC(C)C(c2ccccc2)C1 91170,N1(C(c2c(C)noc2)=O)CCCC(NC(c2nnc(C(F)(F)F)s2)=O)C1C 91171,c1(C(=O)NCCCC(C)NC(C2C(C)C2c2ccccc2)=O)cccnc1F 91172,C1(NC(=O)Cn2ccnn2)CCC(CCNC(C2(CCF)CCC2)=O)C1 91173,c1(C(=O)NC2CCC(C(=O)NCC3CCCC34CC4)CC2)cc(F)cc(F)c1 91174,C(=O)(CCN=C(NCC1(CC(N)=O)CCCCC1)NC1CC(O)C12CCC2)NC 91175,C(c1cccnc1)=C(C)C(=O)NC1CC1CNC(c1ccc(F)cc1)=O 91176,C1(C(=O)NC(CC=C)CNC(c2sc(F)cc2C)=O)CCC2CC2CC1 91177,CC1=C(C(=O)NCC2CCN2C(c2cc(Cl)ccc2Cl)=O)CCC1 91178,CC1(C)C(O)CCN1C(C1CCOCC1)C(=O)NCCC#N 91179,C#Cc1cccc(NNC(=O)NC2CC3CCCCN3C2)c1 91180,N1(C(C2N(CC)CCCC2)=O)CCN(C(c2c(N)cc(Cl)cc2F)=O)CC(O)C1 91181,C(=O)(CCCS(C)(=O)=O)N1CCC(NC(c2c(C)n[nH]c2)=O)CC1C1CC1 91182,C1(NC(c2cn[nH]c2)=O)CN(C(c2ns[nH]c2=O)=O)CC(F)(F)C1 91183,N1(C(C(C)NC(CC)=O)=O)CCCC(N(C(=O)CSc2nncs2)CC)C1 91184,N1(C(c2c(C(C)C)nn(C)c2)=O)CC(NC(C2CC2C(F)F)=O)CC2(CC2)C1 91185,c1(CC)cnccc1CNC(=O)N(C1CCC(C)(C)C1)C 91186,C1(NC(c2cnn(C)n2)=O)CN(c2snc(Cl)c2C#N)C2(CCOCC2)C1 91187,c1(CN2CCCS2(=O)=O)cncc(C(=O)NC2(CN)CC=CC2)n1 91188,C1(C)(CNC(C(CC)n2ccnc2)=O)CCN(C(C2CC3C=CC2C3)=O)CC1 91189,c1(C(N2CC(CCOC)N(C(=O)C3=C(C)CCC3)CC2)=O)c(C)cc(C)oc1=O 91190,c1(SC)ncc(C(=O)NCCCN2CCCC2C)cn1 91191,C1(NC(CC2(NC(CCc3ncn(C)c3)=O)CC2)=O)CCS(=O)(=O)C1 91192,c1(C(C)=O)cccc(OCC(=O)NC2(CNC(C3CCCN3C)=O)CC2)c1 91193,C1(OC)CC(CCNC(=O)Cc2ccc(O)cc2)N(C(c2snc(O)c2Cl)=O)C1 91194,c1(C(CSCCC)(C)NCC2CC=CC2)nnnn1C(C)C 91195,C1(NC(C=CCNC(=O)CCOCC2CC2)=O)CC2(CCC2)C1O 91196,c1(CCC(N2CC(CN(C(CCCC)=O)C)OCC2)=O)nc2cc(Cl)ccc2s1 91197,Cc1ncc(C(N2CC3C(CNC(=O)Cc4ccns4)C3C2)=O)n1C 91198,c1(OC)cc(OC)cc(C(=O)NC2CC3CCC2N3C(=O)C(C)(C(C)C)OC)c1 91199,NS(=O)(=O)c1ccc(CCC(=O)NC2(CNC(=O)C3=CCC3)CCOC2)cc1 91200,N1(C(COCCCC)=O)CCC(CC)C1CNC(=O)C(CC)OCC 91201,c1(SCC)cnccc1C(=O)NCC(C)(O)CNC(c1ccc(O)cn1)=O 91202,C(C)(CN=c1[nH]cnc2c1COC2)NC(C1(COC)CCOCC1)=O 91203,c1(SC)nc2c[nH]c(=NCc3cnc4n3CCS4)nc2s1 91204,N1(C(c2c(C)nc(C)[nH]2)=O)CC2CC(NC(C3CCCCS3)=O)CC2C1 91205,c1(C(C)=O)cc(C(N2CC(C(=O)NCC(F)CO)CC(F)C2)=O)ccc1O 91206,C1(NC(CC2CC(NC(=O)CN3CC4CC4C3)C2)=O)CCN(C(=O)CO)CC1O 91207,c1(C(N2C(CNC(C(CC)c3ccccc3)=O)CC2)=O)noc(C)c1[N+](=O)[O-] 91208,C12(NC(CC(=O)N(C)C)=O)CCCC1N(C(=O)C=CC=C(Cl)Cl)CC2 91209,Cc1ccnc(C(=O)N(C)CC2(CNC(=O)CCn3cc(C)cn3)CC2)n1 91210,c1(C(N2CCN(C(C(Cc3ccccc3)OC)=O)CC2)=O)ccc(N)c(C)c1Cl 91211,c1(C(=O)NC2C(NC(C3(O)C(C)(C)C3)=O)CCC2)cccn2ncc(Br)c12 91212,C1(C(C)C)CCC(C(=O)NCC#CC2CC2)N1C(=O)CC1OCCO1 91213,N1(C(C(F)=CCC)=O)CCCC(C)(C)C1CNC(=O)CC1C=CCC1 91214,C1(CCNC(C(C)OC2CCCC2)=O)CCN(C(=O)Cc2ccc(F)nc2)CC1 91215,C1(C(=O)NCCC2(C)CCN(C(C3(C)CCC(=O)NC3)=O)C2)SC2C=CC1CC2 91216,c1(C(C)C)conc1C(=O)NCCC(C)NC(C1CCOC1C1CC1)=O 91217,c1(N2CCC(c3c(OC)cccc3)C2)nc2cccc(Br)c2[nH]1 91218,C(=O)(CCCC(C)CC)NC(CC)C(=O)NCC1(CO)CCN(C)C1 91219,Cc1[nH]c2ccnn2c(=O)c1CC(=O)NC1CN(C(=O)C2=CCOC2)CC12CC2 91220,C(c1ccc2occc2c1)=CCO.CC1CN2C(C)CN1C(=O)C2=O.C(C)(C)(C)O 91221,c1(OC)ccc(COCCOC(=O)COc2ccc(O)cc2I)c(Cl)c1 91222,c1(OC)cncc(C=CC(N2CCC(NC(=O)Cc3ccoc3C)C2(C)C)=O)c1 91223,c1(CC)ccc(C(=O)NCC2CCC2NC(=O)C=CSc2ccccc2)c(O)c1 91224,c1(C(=O)NCCc2c[nH]c(=NCc3cc(Cl)ccn3)s2)[nH]nc2ccncc12 91225,N1(C(CC(CC)SC)=O)CC2(CNC(c3cn4c(n3)CCC4)=O)CCC1C2 91226,CC(C)(CCC#N)C(=O)NC1CC(NC(C2CCCN2C=O)=O)C1 91227,Cc1coc(C)c1C(N1CC(CNC(=O)CCNC(=O)CO)C2CC12)=O 91228,c1(CNC(C(C)n2ccnc2)=O)cc(Cl)ccc1O 91229,N#Cc1ccc(CCC(N2CCC(Nc3ccccc3F)C2)=O)cc1 91230,Cc1cc(C)c(C(N2CCOC(C)(CNC(c3cnsn3)=O)C2)=O)c(C)n1 91231,N1(C(c2cncc(Cl)c2Cl)=O)CCC2(CC(NC(C3(O)CC3)=O)CO2)C1 91232,c1(C(C(=O)N(C2CCCCC2=O)C)C2CC2)ccc(Br)cc1 91233,C1(N(C(CC(C)SC)=O)C)CCN(C(c2oc(C)nc2C)=O)CC1 91234,N1(C(C2(COC)CCOC2)=O)CCCCC(C2CN(C(=O)CSCC(N)=O)C2)C1 91235,N1(C(C(COC)O)=O)CCC2(C1)CN(C(=O)CC(C)Cc1ccc(Cl)cc1)C2 91236,CC1(C)C(C)(C)C1(F)C(N1CCC(F)(CNC(c2ccc(CO)o2)=O)C1)=O 91237,Cc1cc(-c2cnc(C(=O)Nc3[nH]cnc3C#N)nc2)cc2c[nH]nc12 91238,N#Cc1ccc(SCC(=O)NC2(CNC(C3CCC3CF)=O)CCOC2)cc1 91239,c1(CC)nc(C(=O)N(C2CCCN(CC)C2)c2ccccc2)c(C)o1 91240,CC(C)CC(CNC(c1cnco1)=O)NC(=O)CCc1ccncc1 91241,N1(C(Cn2c(C)ccn2)=O)CCCC12CCC(NC(=O)C=Cc1cnc[nH]1)CC2 91242,CC1CCC(C(N2C3CCC2C(CNC(=O)CC2COC(C)(C)C2)C3)=O)CC1C 91243,C1(NC(=O)Cc2cnoc2)CCCN(C(=O)C(O)Cc2cnc[nH]2)C1 91244,C(=O)(C(C)(C)C(F)F)OC(C)C(N1CCCCC(CO)C1)=O 91245,c1(CC)occ(C)c1C(=O)NCC1CC1NC(=O)C=CCc1ccsc1 91246,c1(OCC)cc(-c2ccc(C(N3CC4CCC(C3)O4)=O)nc2C)ccc1F 91247,N1(C(c2cc(C)c(Br)o2)=O)CCc2cc(CNC(=O)CC3CC3C)ccc21 91248,c1(C(=O)NC(C(=O)N(CC(C2CCC2)OC)C)C)cncc(O)c1 91249,C1(NC(n2ncccc2=O)=O)CN(C(=O)CSC(F)F)C2(CCCOC2)C1 91250,c1(-c2n(CC)ncc2)cncc(-c2nccn2C(N2CCC2)=O)c1 91251,c1(C(N(CCCNC(C2COCC(C)O2)=O)CCO)=O)cc2cccn2c(O)n1 91252,c1(CNC(N2CCC(NS(=O)(=O)C3CC3)CC2)=O)ccc2nonc2c1 91253,c1(C(N2CC(C)C(NC(=O)C(CO)NC(N)=O)C2)=O)c[nH]c2c(F)cccc12 91254,C1(NC(c2c(C)sc(Cl)n2)=O)CCN(C(=O)COCC2CCCOC2)CC1F 91255,c1(OC)cc(C)cc(C(=O)N(C2CC(NC(=O)CN(C)C3CC3)C2)C)c1N 91256,CCCCCCC(C)CC(=O)NC1CCN(CCOc2cccc(F)c2)CC1 91257,C1(CNCc2cc(OC)c(OC3CC3)cc2)(COC)CCCNS1(=O)=O 91258,C(=O)(CS(=O)(=O)CCO)NC1(CNC(c2c(OC)cnnc2)=O)CCCCC1C 91259,CN1C(=O)CN(CC(=O)NCC2(F)CN(C(C3(c4cccs4)CC3)=O)C2)C1=O 91260,N1(C(CC(C)(C)OC)=O)C2CCC(C2)C1CNC(c1ccc(C2CC2)o1)=O 91261,CCCCC(C(=O)NC1CCCC1NC(c1cccn1C1CC1)=O)C(C)C 91262,c1(OC)ccc(CC(O)C(=O)NC(CNC(c2cnc(O)o2)=O)C(C)(C)C)cc1 91263,C1(C(N2C(C(=O)OCC)CN(C(=O)C(F)(F)F)CC2)=O)CC(=O)CC12CCC2 91264,c1(-c2cc(C)no2)ccc(S(=O)(=O)N2CCCN(C(=O)CNS(C)(=O)=O)CC2)s1 91265,C1(C(=O)OC)CN(C(=O)C(N2CCOC(CSC)C2)=O)CCN1C 91266,c1(C(N(C)CC2CCCN(C(C3CC4(CC(=O)C4)C3)=O)C2)=O)ccc(Cl)c(Cl)c1 91267,C1(NC(C(C)O)=O)CCCC(NC(c2ccc(N3CCCCC3)cc2)=O)CC1 91268,CC(C)CC(CNC(C1(c2ccccc2F)CC1)=O)NC(C1CCS1(=O)=O)=O 91269,N1(C(CC2ON=C(C)C2)=O)CCC(C(=O)N(c2cc(F)ccc2C)C)C(O)C1 91270,CC(C(=O)N1CCC(CN(C)C(c2cc(C(C)(C)C)nn2C)=O)C1)C(F)(F)F 91271,C#Cc1cncc(NC(C2(CNC(c3cc(C4CC4)no3)=O)CC=CC2)=O)c1 91272,N1(C(C(CC)NC(N)=O)=O)CC2CCC1C(CNC(C1(F)CC=CC1)=O)C2 91273,O(C1CCc2c1cccc2[N+](=O)[O-])C(C1=NOC(C)C1)=O 91274,c1(C(=O)NCCN(CCOC)C(C2(C)CCCO2)=O)ccc(F)cc1C 91275,Cc1cc(C)n(CC(=O)NCCCOCCNC(=O)CC2CCCCC2)c(=O)n1 91276,c1(OC)cccn2ncc(C(N3CC4C(N(C(=O)C(F)CC5CC5)C)C4C3)=O)c12 91277,N1(C(C2C(C)(C)OCC2)=O)CCC(F)CC1C(N1CC(C(N)=O)C1)=O 91278,C1(CC=C)(C(=O)N(C)Cc2nc(C)ns2)CCCN1C(C1CC1C(C)(C)C)=O 91279,Cc1ccc(C#N)cc1C(=O)NC1CN(C(c2cc3n(c2)CCOC3)=O)CC1C 91280,C1(C(=O)NCCCNC(c2ccn(C3CCC3)n2)=O)CC2(CCCO2)C1 91281,c1(CC(C(=O)NCC(c2c(F)cccc2Cl)N(C)C)O)cc(Cl)ccc1Cl 91282,Cc1cccc(C)c1C(=O)N(CCC(C)NC(=O)C(C)SC(C)C)C 91283,C1(NC(c2c(SC)scc2)=O)CCN(C(c2[nH]nnc2C)=O)C(C)C1 91284,C1(NC(C=CC)=O)CN(C(=O)CCc2ccccc2N2CCOCC2)CC1(C)C 91285,c1(C(N2CC3(CCN(C(CSCCOC)=O)C3)C2)=O)ccc(S(=O)C(C)C)cc1 91286,Cc1ccncc1C(N1CC(N(C)C)C(CNC(C2C=CCCC2)=O)C1)=O 91287,O=C(C1=C(c2ccccc2)CCC1)NC1(C2CN(C(C3CCOC3=O)=O)C2)CC1 91288,N1(C(c2ncc(NC)nc2)=O)CC2CCC(N(C(=O)Cn3cc(Cl)cn3)C)C2C1 91289,Cc1cccc(C(=O)N(CCCNC(c2cnn(CC(F)F)c2)=O)C(C)C)n1 91290,C1(NC(=O)Cc2cc[nH]n2)CCCC(NC(=O)Cc2nc(C3CC3)cs2)C1 91291,C1(OC)CN(C(=O)C(C)N(C)C(=O)OC(C)(C)C)CC1CO 91292,C1(OC)(CF)CCN(C(=O)Cc2csc(C3CC3)n2)CC1 91293,N1(C(C2C(CC)OCC2)=O)CCC(O)C(NC(c2cc(C)n(C(F)F)n2)=O)C1 91294,C1(NC(=O)C=Cc2cocn2)CC12CCN(C(c1cnn3c1CCCC3)=O)CC2 91295,O=C(CC1CN(C(=O)CC2CCOC2=O)CC12CC2)Nn1cnc2ccccc12 91296,C1(NC(C2COCCO2)=O)CCN(C(c2ncc(Cl)cc2Cl)=O)CC1F 91297,C1(CC)CCC(O)(CC)C1.c12cc(on1)CC(=O)NCCOCCNC2=O 91298,c1(C(C)(C)C)ccc(NNC(=O)NCc2ccc(NC3CCOCC3)cc2)cc1 91299,C(CC1CC1)(C(=O)NC(C)C(=O)NCC(C)F)OC 91300,c1(NCC(N2CCCC2)C)ccc(S(=O)(=O)N2CCC(c3ncno3)C2)c(Br)c1 91301,N1(C(CONC(=O)C2(OC)CC2)=O)CCC(C2(C)CC2)C1 91302,N1(C(c2nnc(C(C)C)s2)=O)CCC(NC(=O)CCC2CC2(C)C)C(CO)CC1 91303,C1(CNC(=O)COc2cccnc2)CCN(C(=O)CCCc2ccsc2)CC1 91304,Cc1c(-c2cn(CC(=O)NCC3CCC=CCCC3)nn2)cccc1C#N 91305,Cc1[nH]c(C(C)(C)C)cc1C(N1CC(C)(NC(C2CCCSC2C)=O)C1)=O 91306,c1(NC(C2N(C(C=Cc3ccc(C)cc3)=O)CC2C)=O)cnc2[nH]cnc2c1 91307,C1(=O)CCC(=O)NC23CC1(C2)C3.C1(C(=O)NC(C)C)CC(C)OC1=O 91308,Cc1cc(C(=O)NCCSCC(N2CCC(c3ncco3)C2)=O)nc(O)c1 91309,C(c1cc(C(=O)N(C)CCN(C(=O)C(F)(F)C2CC2)C)cc(OC)c1OC)=CC 91310,N1(C(c2cn(CC)nc2)=O)CCCCC1CNC(c1[nH]nc(OC)c1Cl)=O 91311,CCC(C)CCCC(=O)NC1CN(C(c2ccc(C(=O)OC)cn2)=O)CC12CC2 91312,Cc1ccc(C(N2CCC(CNC(C3CCC(C(N)=O)CC3)=O)C2)=O)n1C 91313,c1(C(N(CC(CC)NC(=O)COC(c2ccn(C)c2)C)C)=O)ccc(OC)nc1 91314,C12(CNC(C=CCN(C)CC)=O)CC(CO1)N(C(c1ccc(C)nn1)=O)C2 91315,c1(C(=O)NC2CC(C)N(C(=O)CCc3cnoc3)CC2)cccc2ccncc12 91316,C1(C2CCCN(c3nc(C)cc(C#N)n3)C2)(NC(C(CC(C)C)OC)=O)CC1 91317,N1(CC(=O)NC2CCC(N(C)C(c3cnn(CC(F)F)n3)=O)C2)C(=O)CNC1=O 91318,N12CCC(NC(c3cnn(C)c3F)=O)(C1)C(=O)NCC2=O.Cc1ncsc1C=O 91319,N1(CC)CC(NC(=O)CC2CC(NC(=O)C=Cc3cn(C)nn3)C2)C(C)C1 91320,C#Cc1ccc(C(=O)NC(C(=O)N(C(C)C(=O)OC)C)C(C)(C)C)cc1 91321,C1(C(=O)OC)CC2CC(C1)N(c1nnc(C(C)C)s1)C2 91322,Cc1sc(=O)n(CC(=O)NCC(C2CC2)NC(=O)CC2CCCS(=O)(=O)C2)c1C 91323,Cn1c(CC(=O)NCC2(F)CN(C(=O)CNC(=O)NC3CC3)C2)nnc1S 91324,c1(CC(N2CCCCC(NC(C(CCSC)O)=O)C2)=O)c(F)c(F)cc(F)c1F 91325,C1(NC(c2nn(CC)c(O)c2)=O)CC(NC(=O)Cn2nc(C)nc2C)C12CCC2 91326,C(=O)(CCC(=O)c1ccccc1)N1CCC(CCNC(c2ccc(Cl)nc2)=O)C1 91327,N1(C(C(Cn2cccn2)NC(c2ccccc2F)=O)=O)CCCC2(CCCC2)C1 91328,c1(OC)cc(-c2nc(C(=O)Nc3cncc(C#N)n3)ccc2F)ccc1C 91329,Cc1cc(C(=O)NC(c2ccsc2)CO)nc(Br)c1 91330,N1(C(=O)NCCOC(C(=C)C)=O)CCC2(CCN(Cc3cc(Br)ccc3C)C2)C1 91331,N1(C(c2ccnc(C)c2C)=O)CCC(C(=O)NCc2nnnn2C2CC2)=C(F)C1 91332,Cc1cn2c(C(N3CCC(CNC(c4sc(F)cc4C)=O)C(C)C3)=O)cnc2s1 91333,CC1CN(C(=O)CCc2nccn2C)CC1NC(c1cnncc1C(F)(F)F)=O 91334,c1(C(=O)Nc2cccc(NC(c3cnccc3Cl)=O)c2)cc2n(n1)CC(O)CO2 91335,C(N=c1cc(Cl)nc(C)[nH]1)C1N(C(C=CCOC)=O)CCCC1C 91336,N1(C(CCCC=C)=O)CC2CC(C1)C(CO)C2NC(=O)C(Br)=C(C)C 91337,C1(CC(=O)NCC2CC(NC(CC=CC)=O)C2)CCn2cncc2C1 91338,C1(C(N(CC(C)NC(c2cc(-c3ccccc3)cs2)=O)CC)=O)CC2(CCC2)C1 91339,C(=O)(CC(C)(C)C(=O)N1CC(OC)C(NC(=O)C(C)CC)C1)OCC 91340,Cc1nc(N(C)C)sc1C(=O)NCCC1CN(C(C2CC(C)(C)O2)=O)CCO1 91341,C1(=CC(=O)OC(c2ccccc2)COC)CCC(C)(C)CC1 91342,C1(N(C(CSCc2nc(C)on2)=O)C)CN(C(=O)Cn2cnnc2O)CC1O 91343,CCC(C#N)(CC)C(=O)NCC1CN(C(=O)C(C2CCOCC2)O)C(C)(C)C1 91344,C1(C(=O)NC2(C(=O)OC)CC2)(NC(COCC=C)=O)CC(O)C1 91345,CP(C)(=O)CCC(=O)NCC1CC1C(=O)NC1CC(=O)N(CCF)C1.C 91346,C1(OC)CCC(C)(C(N2CCC(C)(NC(C3CC(=O)NC3(C)C)=O)C2)=O)CC1 91347,N1(C(C2CC(NC(C3CC(CCC)C3)=O)C(O)C2)=O)CC2CC2C2CC12 91348,N1(C(c2c(C(C)C)noc2)=O)CC(C(=O)NCC2(C)CCCC2O)C(F)(F)C1 91349,c1(C(=O)NC(C2CCN(C(=O)CCn3cnnn3)C2)(C)C)ccc(Br)cn1 91350,N1(C(c2c(C)oc(C(C)C)n2)=O)CC(CNC(=O)C(=O)NCCC#N)CCC1C 91351,c1(N2CCC(CCC)C2)ncccc1S(=O)(=O)NC12CCC(N(C)C)(CC1)CC2 91352,C(=O)(C(F)CC(C)(C)NC(=O)CCC1CC1(C)C)NCCSCC#C 91353,N1(C(C(CC)N(C)C)=O)CCC(O)(CCNC(c2[nH]c(C)nc2C)=O)C1 91354,C(CC(=O)NC1CN(C(c2nccc(Br)c2C)=O)C1)(C(F)(F)F)OC 91355,c1(OC)ccc2c(C(=O)NC3CC4CC3N(C(=O)Cn3cnnc3)C4)csc2c1 91356,CCC(C)C(C(=O)N(O)Cc1cn(C2CCCC2)nn1)Oc1ccc(F)cc1F 91357,C(=O)(CC(O)C(Cl)(Cl)Cl)NC(c1ccc(OC)cc1)CCCC 91358,c1(NC(C2(C)CCN(C(c3ccc(F)nc3F)=O)C2)=O)c[nH]c2ccc(Cl)cc12 91359,S(=O)(=O)(CC(=O)NCCCNC(=O)CC1OCCCO1)N(CC)CC 91360,CC1CC(NC(C2CCC(N(C)C)C2)=O)CN1C(c1ccc(OC2CC2)cc1)=O 91361,C1(C(N2CC(=C)C2)=O)CC(C)N1C(=O)CC1(COC)CC1 91362,CCC(O)(CC(=O)NCC=CCNC(c1cncc(Cl)n1)=O)c1ccccc1 91363,C#CC1(CNC(=O)NCC2(C)CC(C)=NO2)CCOCC1 91364,c1(OCC)ccc(C(=O)NCC(CC)NC(c2nc(Cl)c(Cl)s2)=O)cc1 91365,C1(CC(=O)NCCCC(C)NC(C2CCSCC2)=O)CCCC(C#N)C1 91366,Cc1sc(N)c(C(N2CCCC(CO)(CNC(=O)C(F)OC(F)(F)F)C2)=O)c1C 91367,C1(C)(NC(c2cc(CC)no2)=O)CCN(C(=O)C(n2cnc(C#N)n2)C)CC1 91368,N1(C(c2ccc(CC)[nH]2)=O)CCC2(CC1)CN(C(=O)CC1CCC3CC13)CCO2 91369,c1(C(N2CCNCC2)=O)ccc2c(c1)CC(OC)CN2C(c1c(F)c(C)nn1C)=O.CO 91370,N1(C(C(CO)NC(C(C)C)=O)=O)CC(NC(c2nnc(S)n2C)=O)CC2(CC2)C1 91371,C#CCCCCCCC(=O)NC(C)CN(C)C(C1CCCN(C(C)C)C1)=O 91372,Cn1cnc(C=CC(=O)NC2CC(F)(CNC(C3CCCC(F)C3)=O)C2)c1 91373,C(=O)(C1Cc2ccccc21)NCC1N(C(c2cn(C3CC3)cn2)=O)CCC(C)C1 91374,CCCCCC(C)(C)C(=O)N(CC(C)CNC(=O)CC1CC(O)C1(C)C)C 91375,N1(C(C(CC)OCC)=O)CC(F)(F)CC1CNC(c1ccn(C2CC2)c1C)=O 91376,N1(C(CSCCOC)=O)CCC(C)(CNC(=O)CN(c2ccccc2)C)C1 91377,c1(C(=O)NCC(CNC(C(C2CCCCCC2)C)=O)(C)C)cn(C)c(O)n1 91378,C#Cc1ccc(CC(=O)NC(CNC(c2cncc(C)n2)=O)CCCC)cc1 91379,N1(C(c2cc(C(CC)C)no2)=O)CCC(NC(=O)CCCF)C(C(N)=O)C1 91380,C(=O)(C(CCO)N(C)C)NC1CCC(NC(CC(=O)NCC)=O)C1 91381,C1(CC)CN(C(=O)COCC(=O)N(C)C)C(C)CO1 91382,c1(C(=O)NCC2CCCC2NC(C2CC(F)(F)C2)=O)nc2ccccc2cc1Cl 91383,C(=O)(CS(=O)(=O)C1CCCC1)N1CC(NC(C(C(CC)C)O)=O)C(OC)C1 91384,C(CC(C)C)(C(F)(F)F)NC(N1CCC(C(=O)NC(C)C)CC1)=O 91385,C(=O)(CCCCCF)NCCNC(C1(SC)CCC1)=O 91386,c1(OC(C)C)cnc(C(N2CC(CC(C)NC(C3C=CCCC3)=O)C2)=O)cn1 91387,N1(C(c2ccnc(C)n2)=O)CCN(C(=O)CC2CS(=O)(=O)C2)C2CC12 91388,C1(NC(c2ccncc2O)=O)COC2(CCN(C(c3cc[nH]c3)=O)C2)C1 91389,C1(CNC(C)=O)CCCCN(C(=O)Cc2cc(=O)n(C3CCS(=O)(=O)C3)[nH]2)C1 91390,c1(SC)cc(C(=O)NC(CCNC(C2(C(F)F)CC(O)C2)=O)C(C)C)ccc1N 91391,N1(C(CNC(=O)OCC)=O)CCN(C(c2cccc(Cl)c2OC)=O)C(CCO)C1 91392,c1(CC(=O)NC2CC3(C(NC(C(F)OC)=O)C3)C2)c(C)nc(O)nc1O 91393,c12cnc(nc1)C(=O)N1CCCC(C1)Cc1cn(nn1)C2C.n1(CO)cccc1 91394,N1(C(C2CC(=C)C2)=O)CC=CC1C(N1CCC(N2CCC2)C1)=O 91395,C1(NC(C(COC)C)=O)CCN(C(=O)Cc2ccc(OC)c(OC)c2)CC1O 91396,N1(C(c2c(C(=O)OC)c(C)[nH]n2)=O)CCCC(C)(NC(C2CC2(C)C)=O)C1 91397,CC(C)C1=CCC(C(N2C3CCC2CC(CCNC(=O)CSC2CC2)C3)=O)CC1 91398,N1(C(C(C)=C(CC)C)=O)CCC2(CCC2NC(C2COCCN2C=O)=O)CC1 91399,Cc1nccn1C(C)C(=O)NC1CCCC1NC(=O)CSCC(N)=O 91400,CN1CCn2ncc(C(=O)NCC3CN(C(=O)C(C)(C)C)CC3(F)F)c21 91401,c1(C(N2C(CNC(C(CC#C)C)=O)COCC2)=O)ccc(OCCCC)cc1Cl 91402,c1(CC(N2CC(CCNC(C(CC)(C)C#N)=O)C2)=O)c(C)[nH]c2ccc(F)cc12 91403,S(=O)(=O)(c1cncc(Br)c1)N1CC(N(c2cc(Br)nc(Br)c2)C)C1 91404,C1(NC(c2ccc(C(C)=O)cc2)=O)(CO)CCCN(C(C2CC(O)C2)=O)C1 91405,Cn1nc(C(=O)N(C2CCCN(C(C3(n4cccn4)CCC3)=O)C2)CCO)cc1Cl 91406,c1(C(N2CC(OCCNC(C3C(OCC)C3C)=O)C2)=O)cnnc(C)c1 91407,C1(C(=O)NCc2ncccn2)CC(F)CCN1C(c1cncc(Cl)c1)=O 91408,n1(CC)cnc(NC(=O)CCc2cc(C)no2)c1 91409,c1(C)cc(C(=O)N(C(C)C)NC(CCNC(CCSC)=O)=O)no1.C(C)C 91410,c1(C(=O)NC(C(=O)NCCC(CC)O)C2(C)CC2)c[nH]c2ccccc12 91411,c1(NC(CN2CCN(C(C(CCC)NC(C)=O)=O)CC2)=O)ccc(Cl)c(Cl)c1 91412,C(=O)(C(C)C(C)NC(=O)COCCCOC)N(CC(=O)NC)CC=C 91413,CC(C)C(CC(=O)NC1(CCO)CCCCC1)NC(C1CCC2(CCC2)C1)=O 91414,N1(C(c2c(CC)cno2)=O)CCC(C)(C(=O)N(CC(C)C(F)(F)F)C)C1 91415,c1(CC(=O)NC2CN(C(=O)C3=CCCCC3)CC3CC23)ccc(F)cc1[N+](=O)[O-] 91416,N1(C(C2(CC#C)CCC2)=O)CCC(CO)(NC(=O)CCc2ccc(Cl)s2)C1 91417,CC1CN(C(=O)CCC(N)=O)CCC1N(C)C(C12CC(c3ccccc3)(C1)C2)=O 91418,C1(C(=O)Nc2ccnc(F)c2Br)Cc2cc(O)ccc2CN1Cc1cnc(Br)s1 91419,C(=O)(C#CC1CCCCC1)N1CCC(C)(NC(C(CCCC)ON=C(C)C)=O)CC1 91420,C1(C(N(CC(COCC)O)C)=O)C2CN(C(C3(F)CC=CCC3)=O)CC12 91421,N1(C(C2(N(C)C)CCC2)=O)CCCC(C)(C(=O)NCc2ccccn2)C1 91422,N1(C(c2cc(C)c(C)s2)=O)C(C(=O)N(C2CCCC2)CCO)CC2CCCCC12 91423,N1(C(C2C(C)C2C)=O)CCC(C(C)C(=O)N(CCC(N)=O)C)C1 91424,c1(C(N2C(CN(c3nnc(C)o3)C)CCCC2)=O)c(O)nnc2c1CCCC2 91425,Cc1ccc(CCC(=O)NC2CC2NC(c2c(C)noc2N)=O)cc1C 91426,C1(CNC(C2(C)C=CCCC2)=O)CN(C(c2cc(O)ncn2)=O)C2CCCCC12 91427,N1(C(COCCCCC)=O)CC2CCN(C(c3ccc(F)c(F)c3N)=O)C(C2)C1 91428,Cc1cc(=O)n(C)cc1C(N1CCN(C(=O)CCOCC2CCCO2)CC1C)=O 91429,c1(NC(C(C2CCN(C(C3C(C)(C)C3(C)C)=O)C2)F)=O)ccc(O)cc1F 91430,c1(NCC(N2CCN(CC)CC2)(C)C)ccc(S(=O)(=O)N(C)C)cc1C#N 91431,c1(C(=O)NC(CNC(c2c(C)nc(CC(C)C)s2)=O)C2CC2)cn2c(n1)CCC2 91432,c1(CNC(c2cccc(F)c2F)c2n(C(C)(C)C)nnn2)nnc2n1CCS2 91433,Cn1ncc(C(=O)NCc2occc2C(=O)NCC2CCCSC2)c1N 91434,c1(CN2CC(NC(=O)C=Cc3ccsc3)C2)cccc(C(=O)O)c1F 91435,C(=O)(C(C)CCCC(C)=O)N(CC(=O)NCC(n1cnnc1)C)CC 91436,c1(C(=O)NC23C(CN(C(Cn4c(C)cnc4)=O)C2)CC3)nc2nccc(C)n2n1 91437,C(=O)(C1=CCCCC1C)NCc1ccc(C(N2CC=C(C)C2)=O)cn1 91438,C1(NC(C(c2n(C)ccc2)=O)=O)CCCC(NC(c2cnsn2)=O)C1 91439,C1(C(N2CC(N(C)C(=O)OC(C)(C)C)C2)=O)(NC(=O)C=CSC)CCC(C)(C)C1 91440,Cc1cc(Br)c(CN2CCN(c3ccc(CO)cc3)CC2)cc1O 91441,C(=O)(NN1CCC(F)(F)CC1)C1(C)CC1Br 91442,N1(C(C2CC(CC)C2)=O)CCCC(C2CN(C(=O)C=Cc3c(C)noc3C)C2)C1 91443,CC1CCC(CO)(NC(c2cncc(CNC(=O)C(C)OC(C)(C)C)c2)=O)C1 91444,C(=O)(C1Cc2ccccc21)NCC(CCNC(C1CC2(CC(=O)C2)C1)=O)O 91445,C1(CCC)(NC(C2CC3(CCC3)C2)=O)CCCN(C(C2CS(=O)C2)=O)C1 91446,N1(C(C2CC3CC(OC)C3C2)=O)CC23CCCC2(C1)CN(C(=O)C1=COCC1)C3 91447,c1(CNC2(c3nnnn3C3CCCC3)C(CC)CC2)cc2cccc(OC)c2o1 91448,CC(C)C(C(=O)N1CCC(CCNC(=O)C(C)N(CC(F)(F)F)C)C1)C(C)C 91449,c1(C(=O)NC2CCN(C(C3C(C=C)CC3)=O)CC2CO)cccc2c1CCC2 91450,C(=O)(C1=CC2(CCOC2)C1)N1C2C(NC(CC(CC)C3CCC3)=O)(CCC2)CC1 91451,c1(C(=O)OCc2cccc(F)n2)cc2ccc(Cl)cc2c(O)n1 91452,C1(C(N2CCCC(O)(CNc3ncc(F)cn3)C2)=O)CC2CCC1CC2 91453,C1(CNC(C2(CNC(C(CC#C)C3CC3)=O)CC2)=O)CCCOC1(C)C 91454,C1(CNC(c2ccc(CC(C)(C)O)s2)=O)CCCCN(C(C2CC=CCC2)=O)C1 91455,c1(NC(C(C)(O)C2CCCCC2)=O)ccc[n+]([O-])c1 91456,O=C1CCc2cc(C(=O)CCC(CCC(=O)N=c3cncc[nH]3)=O)ccc2N1 91457,C1(NC(=O)CSCc2ccccc2)CCN(C(C23CC(F)(C2)C3)=O)C12CCC2 91458,N1(C(CCS(CC)=O)=O)CC2(CCC(NC(=O)C(C)CSc3ccccc3)CC2)C1 91459,C1(NC(c2cccnn2)=O)CCC2CN(C(=O)C=CC=C(Cl)Cl)CC2C1 91460,N1(C(C(CC)N(C(=O)C(F)(F)c2nccs2)CC)=O)CCCCC1COC(C)=O 91461,c1(C(=O)OC)ccc(C(N2CCCC2(C)C(=O)Nc2nnc(Br)s2)=O)cc1F 91462,Cc1cc(NC(C2CCN(C(c3cnn4cc[nH]c34)=O)C2)C)ncc1[N+](=O)[O-] 91463,C#CC1(C(=O)N(C)CC2CCCC2(C)C)CCN(C(=O)C(O)CC(F)(F)F)CC1 91464,c1(C(N(CCCn2cc(CC(O)C3CC3)nn2)C)=O)cccc(F)n1 91465,c1(C(C(=O)NCC(C)C)N(C)CC2C3CCCC23)cnc(N(C)C)cc1Cl 91466,N1(C(C2CCCCO2)=O)CCNC(C(N2CCCC(F)C2)=O)C1 91467,N1(C(CCNS(c2c(C)nn(C)c2C)(=O)=O)=O)CCc2ncc(C3CC3)cc2C1 91468,C1(C(=O)NC2CCSC23CN(C(=O)CC(F)F)C3)CCCCC12OCCO2 91469,c1(C(N2CCOC(C(N3CC(F)(F)C(F)(F)C3)=O)C2)=O)cc2cc(F)ccc2[nH]1 91470,C1(C(N(C(C)(C)CC(N2CCC(F)CC2)=O)C)=O)CCCCC(=O)N1 91471,c1(CNC(N2CC(C#C)OCC2)=O)nc2c(COC)cccc2s1 91472,CN(C)NC(=O)CCC(=O)NCCCOCCNC(C1(C#N)CC2(CCC2)C1)=O 91473,c1(C(=O)NC(C(CO)NC(c2c(CC)scc2)=O)C)cc(F)cc2cc[nH]c12 91474,C(=O)(C(CC(C)C)C(C)C)NC(C(=O)N1C(C)CC1)CCN(C)C 91475,c1(C(N(C)CC2OCCN(C(C3(C=C)CCC3)=O)C2)=O)cnn2cccc(Cl)c12 91476,C(=O)(CCCCCF)N(CC)CC1CCN(C(C2CN(C)CC2C)=O)CC1 91477,N1(C(c2c(-c3cn(C)nc3)c[nH]c2)=O)CCC(O)(CNC(C2CC23CC3)=O)CC1 91478,c1(C(=O)NCC(CNC(C(CC=C)C(C)C)=O)(C)C)cnn2ccnc(C)c12 91479,C12(C(N(CC#C)C)=O)CCCC1N(C(CC(C)(C)C)=O)CC2 91480,C12(CNC(C(CC#C)C)=O)CC(CO1)N(C(=O)CC(C)(C)C=C)C2 91481,c1(OC)cccc(C)c1C(=O)NC(C)C(c1ccccc1)NC(C12CC(C1)C2)=O 91482,CCN=C(NCCC1(C)CCCC1)N1CCC(CN(C)NC(=O)OC(C)(C)C)C1 91483,C1(CNC(CCC=CC)=O)CCN(C(c2cnc(C(F)(F)F)s2)=O)CC1C 91484,N1(C(c2cc(C(=O)OC)sc2C)=O)CCC2C(C1)CN2C(=O)CSc1cn[nH]c1 91485,Cc1ccc(Cl)cc1C(=O)NCC(C)CNC(C12COC(C1)C2)=O 91486,c1(C(N2CCC(NC(C(CC)O)=O)CC2)=O)c(Br)sc(C)c1C 91487,n1(CC)ccc(=NC(=O)C(CCOC)NC(c2coc(C(F)F)c2)=O)[nH]1 91488,N12CCCC(C1)NC(=O)C=CC2=O.C(=O)(C(C)NC=O)N(CCCC)CC 91489,C1(N(C(c2n(CCOC)ncc2)=O)CC)CCCN(C(C2CC=CCO2)=O)CC1 91490,C(CCC(C)C)(C(=O)N(C1CCCN(C(=O)CC2OCCO2)C1)C)NC(C)=O 91491,c1(C(=O)NC2CN(C(Cn3nc(C)oc3=O)=O)CC2(C)C)ccc2c(c1)CCC2 91492,C(=O)(C(CC(C)C)ONC(=O)CC1CC(F)C1)N(CC)CC1CCC1 91493,C12(NC(COCC(=C)C)=O)CCCC1N(C(=O)Cc1ccc(O)cn1)CC2 91494,CCC(C)CC(=O)NCC(O)CNC(=O)CCN(C)CCO 91495,c1(C(N2C(CNC(=O)CCCCC(F)(F)F)CC2)=O)ccc2c(c1)OC(F)(F)O2 91496,C(c1ccc(C(F)(F)F)c(O)c1)=CCN(C(=NCC)NCC(C)OC)C 91497,N1(C(c2c(SC)cccn2)=O)CC(NC(c2csc(C)c2)=O)CCC1C 91498,c1(CO)cc(C)c(C(=O)NC2CCCC2n2cc(CNC3CCOC3)nn2)o1 91499,c1(C(=O)NC2CCC2NC(C2CCCC2)=O)cnc2[nH]nnc2c1 91500,CCCCCCC(CC)C(=O)NC(C)CCCNC(=O)C(C)C(C)S(C)(=O)=O 91501,c1(C(=O)NCCN(C(c2c(OCC)nc(C)cc2)=O)CC)c([N+](=O)[O-])cnn1C 91502,CCCC(C#N)C(=O)NCC1(NC(=O)C=Cc2ccc(C(=O)NC)cc2)CC1 91503,C1(C2CC2)(C(=O)Nc2n(C)nc(C(N)=O)c2)CN(C(=O)C(C2(O)CCCC2)F)C1 91504,Cc1ccc(CNC(=O)CC2C3CN(C(c4nc(C)c(C)s4)=O)CC23)cc1 91505,c1(C(N2C(C(N(CC#C)CC#C)=O)CC2C)=O)coc2c1COC2 91506,C1(NC(=O)C=CCO)CC2CC1CN(C(c1coc(Sc3ncccn3)n1)=O)C2 91507,c1(C(=O)NC2C3CN(C(c4c(C)cc(C)[nH]4)=O)CC32)cc2c(ccn2C)s1 91508,N1(C(C(CC)(F)F)=O)C(C(=O)NC(c2cc(C)on2)C)C2CC(O)C1C2 91509,CCC(CC1CCCC1)C(=O)NC(C)CC1CN(C(c2c(C)[nH][nH]c2=N)=O)C1 91510,c1(C(N2CC(C)N(C(c3ccc(Cl)[nH]3)=O)CC2)=O)ccc2c(c1)NC(=O)C2 91511,N1(c2onc(C)n2)CC(C(N2CC(NC(=O)CNS(C)(=O)=O)C(C)C2)=O)CC1=O 91512,N1(C(CS(N)(=O)=O)=O)CCC2C1CCCN2C(c1c(Cl)ccc(F)c1F)=O 91513,c1(CN2CCN(CC(=O)Nc3n(CC)ncc3Br)CC2)ccc(Br)c(OC)c1 91514,CC(C)CCC(=O)N1CC(O)CC1C(=O)N(C)C.c12cc(cs1)C(=O)NC2 91515,N1(C(c2ccc(COC)cc2)=O)CCN(C(C2CC2(F)F)=O)CC(C)(F)C1 91516,Cc1csc2ccc(CC(=O)NCCC(C)(C)NC(C3C4COCC34)=O)cc12 91517,C1(NC(c2c(C)cno2)=O)CCC2(C1)CN(C(C1(C)CC1)=O)C2 91518,C1(C(=O)NCc2ccsc2)CC12CCN(CCC1(F)CC1)CC2 91519,N1(C(CC2C(C)CC2)=O)CC(NC(C2CC3(CCC3O)C2)=O)CC12CCCCC2 91520,C1(NC(c2ccnc(OC)n2)=O)CN(C(=O)C(C2CCC2)OC)CCC1F 91521,CS(=O)c1ccccc1C(=O)NCC1(O)CN(C(=O)C=CC2CCCO2)C1 91522,CC(C)CC(CNC(=O)CC(C)(C)C(F)F)C(=O)NCC(C)CCCO 91523,c1(C(=O)NCCCCCC)n[nH]c2ccc(-c3ccc(-c4cncs4)cc3)cc12 91524,C1(C(=O)NC2C(O)CCN(C)C2)CC2(CCC2)CN1C(C1CC1(C)C)=O 91525,c1(CC(C(=O)N2CCC(C(C)NC(=O)CC3CC3)C2)(C)C)ccc(C#N)cc1 91526,CCCCCC(O)C(=O)NC(C(=O)NCCc1cc(C)ns1)C1(O)CCC1 91527,N1(CCNC(=O)Cc2cncs2)CCN(C(C2(CO)CCOCC2)=O)CC1 91528,Cc1nc(C)c(C(N2CCC(C)(CNC(C3(CC#N)COC3)=O)C2)=O)nc1C 91529,C12(CCC(C)(C)C1)NC2.c1(C(CNCC2N(CC)CC2)O)cc(C)cc(C)c1 91530,Cc1nn(C)cc1C(O)C(=O)NC1CCN(C(=O)C(=Cc2cccnc2)F)C1C 91531,c1(NC(C(C)N(C(c2ccc(OC)nc2)=O)C2CC2)=O)cc(CO)cc(F)c1 91532,c1(CCC(=O)NCCN(C(C)C)C(C23CCCCC2C3)=O)ccc(F)cc1Cl 91533,c1(CN2CCCC(C(=O)OC)C2)cccc([N+](=O)[O-])c1.C12CC(CN1C)NC2=O 91534,C1(F)(CNC(CN(c2ccccc2)CC)=O)CC(NC(C2C3COCC23)=O)C1 91535,C(=O)(C(F)C(F)(F)C(F)(F)F)N(c1c(OC)c(Cl)ccc1)C 91536,c1(C(=O)NCC2(C(=O)NCC(C(C)C)(C)F)CC(C)(C)C2)cc(O)cc(F)c1 91537,Cc1cc(C)n(CC(=O)NCC(C)(CO)NC(c2cn(C)nn2)=O)n1 91538,Cc1cc(NC(=O)CCc2cscc2Br)ncc1Br 91539,CN1CCN(CC(N2CCCC(NC(c3cccc(N)n3)=O)CC2)=O)CC1=O 91540,C1(OC)CC(NC(N2CCN(c3cccc(C(F)(F)F)c3)C(=O)C2)=O)C12CCC2 91541,C1(NC(C2CCCOC2)=O)CCN(C(=O)COc2ccc(Cl)cc2)CCC1CO 91542,C1(C(N(CCN(C(=O)CCOCC2CCCO2)C(C)C)C)=O)CCCCS1 91543,C(=O)(C1=CCCSC1)NC(C(C(=O)NCCN1CC=C(C)CC1)C)C 91544,C1(C)(NC(C(n2cc(-c3cccnc3F)nn2)C)=O)CC=CCC1 91545,C1(NC(c2ccnn2CCF)=O)CC2CCC(C1)N2C(=O)CC1CCCC(=O)N1 91546,c1(CC)c(C(=O)NC2CC2CNC(=O)Cn2nnnc2C2CC2)ccn1C 91547,c1(CC(C#C)NC(=O)N(c2cnn(C)c2)CC)cccc(Br)c1 91548,CCC(C(=O)Nn1ccnn1)N(C(=O)C#CC(C)(C)O)C 91549,c1(CCC)nc(C(N2CCCC2C(C)NC(C2(CC)CC2(F)F)=O)=O)cs1 91550,c1(C(=O)NCC(N(C(CCOC)=O)C)C2CC2)ccc(S(C)=O)cc1 91551,CCCCC(C)C(=O)NC1CN(c2ncccc2Br)C1 91552,c1(OC)cc(NCC2CC(NC(c3cncc(C)c3)=O)C2)nc(C(F)(F)F)n1 91553,C(CNC(c1cnn(CC2CC2)c1)=O)(CC(F)(F)F)NC(C1(C#C)CC1)=O 91554,N1(C(CCN(C)CC)=O)CCC2(CCC(NC(=O)CC(C)CC(F)(F)F)C2)CC1 91555,c1(OC)ncc(C(=O)NC2CC(C)(NC(=O)CCC3CC3C)C2)c(C)n1 91556,Cc1cn2c(C(=O)NC(C)C(CO)NC(C3(F)CCOCC3)=O)c(Cl)nc2s1 91557,C(=O)(C1=CC2C=CC(C1)C2)N1C(C(=O)NC2CCN(C)C(=O)C2)CCC(O)C1 91558,c1(COC)ccnc(C(=O)NCCCCC(C)NC(c2ccccn2)=O)c1 91559,c1(SC)ncc(C)c(N2CCN(CC(=O)Nc3cccc(C(F)F)c3Cl)CC2)n1 91560,C(=O)(CCC(C)(C)C#N)NC(C(C)NC(c1ccc(OC)c(C)c1)=O)CO 91561,C(=O)(CCCCCN=[N+]=[N-])N(C)CC.C(=O)(CCC1CCC1)N(C)CCOC(F)F 91562,c1(C(=O)NC2C(C)(C)CCN(C(C3(C)CCCO3)=O)C2)cnc2ccc(F)cn12 91563,N1(C(C2ON=C(C)C2)=O)CCN(C(=O)CC(F)F)CC1C(C)C 91564,C=CCCCC(=O)N1CC(CNC(c2cncn2C(C)C)=O)CC1C 91565,N1(C(c2cc(CC)n(C)n2)=O)CCC(CNC(c2cnn(C)n2)=O)C(F)(F)CC1 91566,C=CCC(CC(=O)N1CC(O)CC(O)C1)NC(C1(CC)CCCO1)=O 91567,c1cnc2ccc(-n3nc(C4CCCO4)nc3CC3CC3)cc2c1 91568,N1(C(C(=O)NCC)=O)CC(CNC(c2nn(C)nc2C(F)(F)F)=O)CCC1C 91569,C1(C(N(C)CC2CCN(C(=O)CN(C)C3CC3)C2)=O)CCCC(F)(F)C1 91570,N1(C(C)=O)CC2CCC1CN2N1CC(N2CCOCC2)CC1 91571,c1(C(=O)NCC(C)CN(C)C(c2cccc(F)c2)=O)cc2cnccc2[nH]1 91572,c1(C(C(=O)NC(CC)(C)C)N(C)Cc2cncnc2)ccc(C)c(C)c1F 91573,C(CC1C(=O)N1)SC.C1(C)(NC(N)=O)CCN(C(=O)CN2CCCC2)C1 91574,C12(C(N3CC4C(CNC(c5cnc(O)cc5O)=O)C4C3)=O)CC3CC1C2C3O 91575,C#CCC(C)(C)C(=O)NC(C)C(CO)NC(=O)C(c1ccccc1OC)OC 91576,c1(CC)nn(C)cc1C(=O)NC1(C(=O)NCC(O)CN(C)C)CCSC1 91577,CC1(C)CN(C(=O)CSC(F)F)CC1NC(C1(F)CCCC1)=O 91578,N1(C(C2C3CC(C)(C3)OC2)=O)CC(NC(c2cccnc2)=O)CC12CCOCC2 91579,N1(CC)C(C)CCC1C.CC(C)C(CNC(=O)C(=O)NCC)N1CCCCC1 91580,c1(CCC(=O)N(CC(C)NC(C2CC2(C)C)=O)C)ccccc1[N+](=O)[O-] 91581,C1(CNC(C(CN(C)C)NC(C2CC2C(C)(C)C)=O)=O)CCCC12CC2 91582,Cc1c(NCC2(c3ccccc3)CC2(C)C)ncnc1NC1CC(F)(F)C1 91583,C1(NC(Cc2c(C(=O)OC)csc2)=O)CC2CC(NC(=O)CCC3CCC3)CC12 91584,N1(C(C(C)N(C(C)=O)C)=O)CC(C2(NC(C3CN(S(C)(=O)=O)C3)=O)CC2)C1 91585,c1(CC)ocnc1C(=O)NC(CNC(c1ncc(C(F)F)s1)=O)C1CC1 91586,Cc1nc(C)c(C(N2CCC(CNC(=O)C(F)C3CCC3)C(F)(F)C2)=O)nc1C 91587,c1(C(=O)NCC(CO)NC(c2c(CC)nn[nH]2)=O)cccc(C2CC2)c1 91588,CN1CCN(C)CC(C(=O)N(CCCNC(C2(n3cncn3)CC2)=O)C2CC2)C1 91589,CC(=O)CCN=C(NCC(C)(C)C(=O)OC(C)(C)C)NC1CSC1(C)C 91590,N1(C(CC(CNC(=O)Cn2cc(Cl)cn2)O)=O)CCC(CO)=C(F)C1 91591,C(c1cncc(C)c1)=CC(N1CCC(C(=O)NCC(=O)OC)CC1)=O 91592,C1(CNC(C(C)(C)CO)=O)CCN(C(C2CCN(c3ncccn3)C2)=O)C12CC2 91593,c1(CNC2CN(C(c3n(C)cnc3)=O)CC2F)cc2c(Br)cccc2s1 91594,C(=O)(CCS(=O)(=O)c1ccc(C)cc1)N1CC2C(N(C(C(CC)C)=O)C)C2C1 91595,N1(C(C(CC)(F)F)=O)CCCOC(CNC(c2c(OC)ccnc2O)=O)C1 91596,C1(C)(C(N(CCCCN(C(=O)Cc2ccsc2Br)C)C)=O)CCCC1O 91597,N1(C(C(C)(C)NC(=O)NCC)=O)CCCC2(CCC(NC(=O)CCCOC)C2)C1 91598,c1(CNC(C2(NC(C(C3CCOCC3)C)=O)CC(O)C2)=O)ccc(C#N)o1 91599,CCCCS(=O)(=O)CC(=O)N1CCCC2(CNC(C3(C(C)C)CC3)=O)CCCC12 91600,CCS(=O)(=O)c1cccnc1C(=O)NCCCN(C)C(C12COCC(C1)OC2)=O 91601,c1(CSC(C)C(=O)NC(C)(CNC(c2nnsc2C)=O)CO)ccccc1Cl 91602,C1(CC(=O)NC2C(CC(C)(C)C)C2)C2CCCC2N1C(c1ccc(C(N)=O)o1)=O 91603,N1(C(C2CC(C)(C)C2)=O)CCCC2(CNC(c3ccc(C#N)o3)=O)CCCC12 91604,C1(CC(N2CC(OCC)C2)=O)CC(C)(C)CN1C(C1CCCOC1)=O 91605,c1(NC(=O)NCC2COC3CCCC3O2)c(C(F)(F)F)nc2n1CCCC2 91606,N1(C(C=CCOC)=O)CC(NC(C2CCN(C(=O)OC(C)(C)C)C2)=O)C(O)C1 91607,C#CC1(C(=O)NCCOCCOCC)CN(C(=O)C(CCSC)OC)C1 91608,Cc1cc(C)c(C(=O)NS(=O)(=O)CC2CCCC(C3CC3)O2)o1 91609,C(=O)(C(CC(C)(C)C#N)N1CCN(C)CC(O)C1)NCCCCCC 91610,CC(C)(C)CCC(F)C(=O)NCC1CN(C(=O)CC2CC2CO)CCC12CCC2 91611,C1(NC(C2C(C(C)C)C2)=O)CN(C(=O)C2=CC(C)C2)C2CCCC12 91612,c1(CNC(C2(OCC)CCC2)=O)cc(C(=O)NCCSCCO)no1 91613,C1(CCCNC(C=CC=CC)=O)CCCCN1C(=O)CN1CCCC1C 91614,CC1CCN(C(c2cc3ccsc3[nH]2)=O)CCN1C(=O)C=C1CCSCC1 91615,c1(C(N2CC(C)(NC(c3ccccc3)=O)C2)=O)cc(F)cc(N)c1F 91616,c1(C(N(C2CCN(C(C3CC3COC)=O)CC2)CC#C)=O)cccc2sccc12 91617,c1(OC)c(C(=O)NC2CC(NC(C3CCCC3O)=O)C2)cc([N+](=O)[O-])cc1Cl 91618,c1(OC)ccccc1C=CC(=O)NC1CCCCC1NC(=O)C=CCN(C)C 91619,CCC(CC)C(C)C(=O)N1CCC(CN(C)C(C23CCCN2CCC3)=O)C1 91620,Cc1ccc2c(C(=O)N(C(C)CCNC(=O)C(CN(C)C)C(C)C)C)csc2c1 91621,C1(NC2CC2)CCCC(N(CCCNC(C2(C(=O)NC)CC2)=O)CC)C1 91622,CCCC(CCCNC(C1(C)CC1C)=O)NC(C1CCN(CC(F)F)CC1)=O 91623,Cc1ccc2[nH]c(=NCC3(O)CN(C(C4CCCC5(C4)CC5(F)F)=O)C3)sc2n1 91624,C#CC1CN(C(=O)COC(C)CC)CCN1C(=O)Cc1n[nH]c(=N)s1 91625,N1(c2cc(C)nc(CO)n2)C2CCC1CC(CNC(c1cc3c([nH]1)CCC3)=O)C2 91626,CCCC(C(=O)NC1CCCC(NC(c2ccc(N)c(SC)c2)=O)C1)S(N)(=O)=O 91627,C=C=CC(C)C(=O)NC(c1ccc(F)cc1)CNC(c1ccn(C2CCC2)n1)=O 91628,C1(NC(C(C)c2ccsc2)=O)C2CC1N(C(=O)CNC(C1CCCCCC1)=O)C2 91629,CCCCCCC(F)C(=O)N1CCC(CN(C(=O)CC2(O)CCOC2)C)CC1 91630,N1(C(c2cn(-c3cnn(C)c3)nn2)CN(CCCC)C(C)=O)CCCCCC1 91631,c1(N2C(=O)CC(C(=O)NCCNC(c3ncn(CC)n3)=O)C2)ccc(C#N)cc1 91632,c1(C(=O)NCC(CNC(CCC(C)N(C)C)=O)O)cc(Cl)cc(Br)c1 91633,c1(CCOC)ccc(Br)cc1NC(=O)C=Cc1nnn(C)n1 91634,CCC(C)CCC(O)CC(=O)NC1CCN(C(=O)C=C2CCC2)CC12CCC2 91635,C12(CNC(Cc3cncc(C)c3)=O)CCC(C1)N(C(C1CCCCCCC1)=O)C2 91636,Cc1nnc2ccc(C(=O)NC3CCCC(NC(C4CC(F)C(=O)N4)=O)C3)cn12 91637,C(=O)(CC1C(=O)Nc2ccccc21)NC1CCN(C(c2ncn(C)n2)=O)C1(C)C 91638,Cc1ccc(C(=O)NC2CC(C(=O)NCCN3CCCCC3)C2)nc1 91639,c1(NC(CCC)CCO)[nH]c(=NCC23CCC(CC2)CC3)nc2c1ncn2C 91640,CS(=O)(=O)CCC(=O)NCC1CC(CNC(c2cn3ccnc3s2)=O)CO1 91641,N1(C(CC2CC(C)C2)=O)CCc2nc(CNC(=O)C(C)(C)C(C)(C)C)sc2C1 91642,N(C(=NCCN1CCCC1)NC1CC12CCC2)CC1(C#N)CCCC1 91643,C12(C(=O)NCCCCCNC(C(C)(C)c3cscn3)=O)CCCN(CCC1)C2 91644,C(=O)(CCC(C)(C)C#N)NCC1CC(NC(c2ccc(SC)o2)=O)C1(C)C 91645,N1(C(c2c(CN(C)C)cco2)=O)CCCC2(CCCN2C(=O)Cc2ccon2)C1 91646,C(=O)(CCCCCc1ccccc1)N1CC(NC(C(CC)=CC)=O)C(OC)C1 91647,N1(C(C=Cc2nc(C)c(C)[nH]2)=O)CCCC12CCN(C(=O)C=C1CCOCC1)C2 91648,N1(C(CN2C(=O)CC(C)(C)O2)=O)C(C(=O)NCCN2CCCC2)C2CC(O)C1C2 91649,C(=O)(C1=CC2CCCCCCC12)NC1C(C)(C)CN(C(=O)C=CC2CCCO2)C1 91650,N1(C(COC2(C#C)COC2)=O)CCN(C(=O)C(C)CC=C)C2COCC12 91651,c1(C(=O)NC(CC)CNC(c2ncn(C)c2C)=O)cnc2ncnn2c1C 91652,c1(CC(COC)N(C2CC3CNC2C3)C(C2(F)CCOCC2)=O)ccccc1F 91653,C1(CN2CCN(C(=O)Cn3ccnn3)CC2)CCCC2(CCC2)O1 91654,c1(CC)c(C(=O)NC2CCN(C(C3CC34CCCCC4)=O)C2)cnc2ncnn12 91655,C(CC(C)C(=O)NCC=CCNC(c1cc(SC)oc1C)=O)=CC 91656,c1(C(N(CCCNC(=O)C(C(C)O)N(C)C)CC)=O)ccc(S(=O)(=O)CF)nc1 91657,Cc1nc(C=CC(=O)NCC(C)CNC(=O)C=Cc2nnn(C)n2)cs1 91658,Cc1cnn(C(C)C(=O)NCC2CC(F)(CNC(c3cnn(CCO)c3)=O)C2)c1 91659,N1(C(C2C(C#N)C2)=O)CCC(NC(=O)C(c2ccccc2)N2CCCC2)CC1 91660,C1(CNC(c2c(OC)c(Cl)sc2)=O)CN(C(=O)CC2CC3(CC3)CO2)CC12CC2 91661,c1(OC)c(O)cc(C(=O)NCC2CC(F)CN2C(=O)C(C)OC)cc1C#N 91662,c1(N2CC(C(=O)Nc3nc(C(F)(F)F)cs3)SCC2)ccn2ncc(I)c2n1 91663,CCC(CC)(CCNC(=O)C(C)(CC)OC)NC(=O)CSC(F)(F)F 91664,C(=O)(C(C)(C(C)C)NCC1CC1)OCC(C)SC 91665,C(=O)(C(F)C(C)(C)O)NCCOC1CCN(C(CC2(C(=C)F)CCC2)=O)CC1 91666,C1(C)(NC(C(CC)n2cccn2)=O)CCCN(C(c2ccc(C)n2C)=O)C1 91667,N1(C(C(C)(C)CS(C)(=O)=O)=O)CCC2CCCN(C(=O)CSc3cccs3)C2C1 91668,CC1CN(C(C2(C)CCCN2C(=O)Cc2cncnc2)=O)CC1N=[N+]=[N-] 91669,C1(NC(c2cc(CC)[nH]n2)=O)CCN(C(c2cccc(C)c2O)=O)C(C2CC2)C1 91670,Cc1nn(CC(=O)NCC2(O)CN(C(=O)CSCc3ncc[nH]3)C2)c(=O)n1C 91671,C1(N)(COCC)CC1.C(C(=O)NC(=O)C1CC1)CCN(C(=O)OCC)C 91672,C1(COC)(NC(=O)CCNC(C)C)CCC(F)(F)CC1 91673,N1(C(c2cccc(S(C)(=O)=O)c2)C(=O)NC)CCCC2(CC1)CNC(=O)C2 91674,N1(C(CCC#CC)=O)CCN(C(=O)CSc2cccc(C)c2)C(C2CCCC2)C1 91675,Cn1nc(C(Cc2ccccc2)NC(C2CC3CC2CO3)=O)cc1C(=O)O.C(N)=O 91676,C(=O)(CCC[N+](=O)[O-])NC1(C)CCN(C(C2CCCCC2O)=O)C1 91677,c1(C(N2CCCC(CNC(CCCN(C)C)=O)CC2)=O)cnn2c1OCCC2 91678,c1(C(C)C(=O)N(c2cn(C)nc2Cl)CC2CCOCC2)ncc2ccccn12 91679,c1(N2C(CNC(CC(C)C3CC3)=O)CCCC2)ncnc2sccc12 91680,N1(C(C(C(CC)CC)F)=O)CCC2(CCN(C(c3cccc(F)c3)=O)C2)C1 91681,c1(NC(c2ncn(C)n2)C)ccc(S(=O)(=O)NCC2CSCCO2)cc1Cl 91682,C(=O)(C1=CCCSC1)NC(c1c(CC)cccc1)CNC(=O)C(F)OC(F)(F)F 91683,c1(C(N2CCN(c3nc(C)c(F)cn3)C(CC#N)C2)=O)cc(F)c(C)c(Br)c1 91684,c1(C(=O)NC2C3(CN(C(CC(=O)NCC)=O)C3)CC2)cccc2c1OC(F)(F)O2 91685,CC1CCN(C(C2(C)CC2(F)F)=O)CC1NC(c1ccc(-c2cnn(C)c2)o1)=O 91686,N1(C(C=CCOC)=O)CCC(NC(c2ncnc(OC)c2F)=O)CC1C1CC1 91687,C(=O)(C(C)(C)C(C)NC(=O)Cn1ccc(C)c1)NCCCCCOC 91688,c1(C(N2CC(NC(C3(C)N(C(C)=O)CCC3)=O)C2)=O)ccc(P(C)(C)=O)cc1 91689,C1(C(N(CCNC(C2CCCN(C(C)=O)C2)=O)C(C)C)=O)CCCCS1(=O)=O 91690,C=CC(C)(O)CC(=O)NC1(COC)CCN(C(=O)Cc2ccc(C(F)F)cc2)C1 91691,c1(-n2cc(NS(CC)(=O)=O)nn2)ccc(OCCN(C)C)cc1 91692,c1(C(=O)NC)nccnc1N.c12cc(cs1)C(C1CC1)N(C)C(=O)CCNC2=O 91693,c1(-c2n(CCOC)c(N3CC4CC3(C)C4)nn2)ccc2cn(C(C)C)nc2c1 91694,CC(C)(C)C1=NOC(C(N2CCCCC2CNC(C2(CO)CCC2)=O)=O)C1 91695,CCCCC(C(=O)N1CC2C(C(=O)OC)C2C1)NC(=O)CCCCCF 91696,N1(C(CCCCOC)=O)CC(F)(F)CC1C(N1CCN(CCF)CC1)=O 91697,C(CC(O)CC(=O)N1CCCC(NC(C2(C)CCOCC2)=O)C1)SC 91698,C1(C)(C(N2CC(CNC(CNC(CC)=O)=O)C2)=O)CCOC(C)C1 91699,C1(CNC(c2c(SCC)cccc2)=O)CCCCN(C(C2CC2(C)C)=O)C1 91700,C1(O)(CN(C(=O)C#CC(C)(C)O)C)CCCN(C(=O)CC2COCCN2C)CC1 91701,c1(C(N2CC=CC(NC(C(C)(CO)OC)=O)C2)=O)cccc(C)c1C#N 91702,C1(CC(=O)N(CC(CNC(CSCC(C)C)=O)C)C)CCC(=O)C1 91703,C1(CN)CC(C(=O)NC(C)CC(=O)NC)=NO1.CCCCCC(=O)C(C)=O 91704,C1(NC(CC(CC)SC)=O)CN(C(=O)CCc2ncco2)CCC1O 91705,C(=O)(C1=NOC(NC(c2coc3c2COC3)=O)C1)N1CC(OCC)(COC)C1 91706,c1(C(N(C2CCCN(C(CC(=C)C)=O)C2)CCO)=O)cc(C)c(OC)c(Cl)c1 91707,N1(C(c2c(C(C)C)[nH]cc2)=O)CC(CNC(=O)CC(C)N(C)C)CC(C)(C)C1 91708,c1(N2CCC(N3C(C)(C(=O)NC)CCC3)CC2)nc(C(C)C)nc(C)c1Br 91709,C1(NC(C2C(C)CCC2)=O)CC1C1CCCN(C(c2ncn3cccnc23)=O)C1 91710,c1(N2C(CN3CCN(C)CC3)CCC2)nc(=NC2CC2F)[nH]c2cccc(F)c12 91711,C1(NC(C(C)NC(C2CCC2)=O)=O)C2CC1N(C(=O)CCN1C(=O)CCC1=O)C2 91712,C1(C(=O)NCCC(C)N(C(=O)Cc2cc(Cl)ccc2O)C)CC(C2CC2)=NO1 91713,N1(C(C)C)CCN(C(=NCC2CCCCC2C)NCc2ccc(F)cc2)CC1=O 91714,N1(C(c2n(C=C)nnc2)=O)Cc2n[nH]cc2C1C(=O)N(CCC)OC 91715,N1(C(C=C(CCC)C)=O)CC(CNC(=O)C(C)CC)C(C)(C)C1 91716,N1(C(C2C(C)OC(=O)N2)=O)CC(NC(=O)CCc2ccccc2Cl)CC(C)C1 91717,CCC(O)CC(=O)NCC(C)C(=O)NCCc1ncccc1C 91718,c1(C(=O)NC2C(NC(C(CC)(C)OC)=O)CCCC2)cnc2[nH]cncc1-2 91719,C(C(CNC(=O)C(C)NC(=O)C1CC1)S(C)(=O)=O)NC(C(CC)(C)OC)=O 91720,C(=O)(CCCC(=O)OC(C)(C)C)NCC1C(NC(C2(CSC)CC2)=O)CCC1 91721,c1(OC(C)C)ccc(C(N2CC(NC(=O)CC3CCC(O)C3)C2)=O)cn1 91722,c1(C(=O)NC2CC(OCCC)C2(C)C)cc2cc(F)ccc2[nH]1 91723,Cc1cc(C(=O)NC2CC(CNC(C3(CO)COC3)=O)C2)c(C)c(C)c1 91724,C12(C(=O)NCC(C)(C)NC(c3c(C)c(O)ccc3)=O)CCCN1CC(O)C2 91725,N1(C(CCC2(NC(C(CC)C(=O)OC)=O)CCC2)=O)CCC(F)(F)C(C)C1 91726,c1(NC(C2C(C)(C)C(=O)C2)=O)c(C#N)cnn1C1CCC1 91727,N1(C(C(C(C)O)C)=O)CCOC2(CCS(=O)(=NC(=O)C3CCS(=O)(=O)C3)CC2)C1 91728,Cc1cc(C(=O)NCC2CCCN(C(C3CCC3(C)C)=O)C2)cc(O)c1 91729,c1(C(N2CC(CCCCNC(COC(C)C)=O)C2)=O)ccc2ncnc(O)c2c1 91730,Cc1cc(=O)c(C(=O)NC2(C3CCCN3C(C3CCCC34CCC4)=O)CC2)c[nH]1 91731,N1(C(C(C)O)=O)CCC(C2(O)CN(C(=O)CC3CCC4(CCC4)O3)C2)CC1 91732,C1(NC(C(CN(C)C)(C)C)=O)CN(C(=O)CCc2ncc(F)cn2)CC(C)(C)C1 91733,N1(C(CCC(C)C)=O)CCCC2CN(Cc3cc(Cl)ccc3F)CCC12 91734,c1(NC)ccccc1C(N1CCCC(C(C)C(=O)N(C2CCC2)C(C)C)C1)=O 91735,c1(C(=O)NC(C(C)NC(C(C(=O)NC)(C)C)=O)C)[nH]c2ccc(OC)cc2c1C 91736,N1(C(=O)NC(CCCC=C)C(=O)NC)CCc2c(cnn2C)C1C(=O)OC 91737,C1(NC(C2C(C(C)O)C2)=O)CCCN(C(=O)CC2(C(F)(F)F)CCC2)CC1 91738,C1(NC(c2cc(OC)nn2C)=O)CCN(Cc2cc3ncccc3[nH]2)CC1(C)C 91739,c1(C(N(C2CN(C(C(C)OC)=O)CC23CC3)C)=O)cc2sc(C)cc2[nH]1 91740,C(=O)(C(F)C(C)(F)F)NC(C(C)C)CCNC(c1ocnc1C1CC1)=O 91741,C(=O)(C1=CC2CCCCCC12)NCCCC(C)NC(c1cc(C(C)C)on1)=O 91742,N1(C(Cc2ccn(C)n2)=O)CCCC(NC(c2cc(-c3ccccn3)no2)=O)C1 91743,c1(C(=O)NCC(C2CCOC2)NC(C2(F)CCCC2)=O)cc2n(n1)CCO2 91744,C1(CNC(NC(c2cccs2)C)=NCCc2cn(C)nn2)Cc2ccccc2O1 91745,c1(C(N2CC(N(C(=O)C(F)CC3CCC3)C)C(O)CC2)=O)nccn2ccnc12 91746,N1(C(C2(OCC)CCOC2)=O)CC2(CC(CC(=O)NCCc3cc(C)[nH]n3)C2)C1 91747,N1(C(C=C(C)C(F)F)=O)CCC(NC(CN(C(=O)CCC2CCCN2C)C)=O)C1 91748,C(C)(C(C)(C)C(=O)NCCC(C)C(=O)OC)NC(CC=CC=C)=O 91749,N1(C(C2=NNC(=O)C2)=O)CC2CCCC(NC(c3noc4c3CCCC4)=O)C2C1 91750,Cc1ncnc(C)c1C(=O)NCC1CC(CNC(=O)Cc2ccsn2)CO1 91751,c1(OCC)ccc(C(=O)NC2CCN(C(=O)C(C)NS(C)(=O)=O)C2C)c(F)c1F 91752,C1(COC)CC(CNC(=O)CC2CC(=O)NC2=O)N(C(c2cc(Cl)c[nH]2)=O)C1 91753,N1(C(C(CC(C)C)F)=O)CCN(C(c2ncc(F)cc2F)=O)CCC1C 91754,C1(C#N)(OC)CC(C(=O)NCC#CC(=O)NCCC2CC=CCC2)C1 91755,C(=O)(C(F)CCC(C)(C)C)NC(C(N1CCCC(C)C1)=O)CO 91756,N1(C(CN(C)C2CC2)=O)CCN(C(c2cn(C)c(=O)n2C)=O)C2COCC12 91757,N1(C(C(CN)N)=O)CCC2(CC1)CC2NC(c1cc2ncccc2[nH]1)=O 91758,CC1(C)CC(CNC(=O)COCCCF)CN1C(=O)C1=NNC(C(F)(F)F)C1 91759,N1(C(COCC(=C)C)=O)CC2CCN(C(c3ccccc3CO)=O)C(C2)C1 91760,CC(C)(C)C(=O)N1CCCC1C(=O)NC1(CNC(=O)C=C2CCC2)CC1 91761,C(C(=O)N1CC(NC(c2ccc(Cn3cc(Cl)cn3)s2)=O)C1)(C(C)C)OCC 91762,c1(CNC(=O)CNC(c2cccnc2)=O)ccc2nonc2c1 91763,c1(C(=O)NCCC2CCCN(C(C=C(C)C(C)C)=O)C2)nc2c(s1)CCCC2 91764,CC1(C(=O)NCCC2CCN(C(=O)Cc3nncs3)C2)COc2ccccc2O1 91765,O(NC(=O)C1(N(C(=O)C=CC(C)(C)C)C2CC2)CCC1)C(C=C)C 91766,O=[N+]([O-])c1cccc2c(NCC(O)CC3CC3)nc(Cl)cc12 91767,C1(O)(CNC(C(c2cccc(OC)c2)C)=O)CCCN(C(C2(SC)CC2)=O)CC1 91768,c1(-c2nc(C(CC)CC(C)C)on2)ccc(S(=O)(=O)C(C)C)cc1 91769,C=CC(C)(CCOC)C(=O)N1CCCN(C(c2cc(CF)on2)=O)C(COC)C1 91770,N1(C(CC)=O)CCC(C2N(C(C3CCN(CC)C3)=O)CC2(C)C)CC1 91771,c1(C(=O)NCC(C23CCC(CC2)C3)O)ccccc1Br 91772,N1(C(C(C)C2CC2)=O)CCn2nc(CNC(c3cnn(CC(F)F)n3)=O)cc2C1 91773,N1(C(C2C(C(C)C)C2)=O)CCCN(C(c2ccc(CCF)cc2)=O)CC1 91774,c1(C(N)=O)ccc(C=CC(=O)NC2CCC(NC(C3(F)CCOC3)=O)C2)cc1 91775,C12(OC)CCC1CN(C(c1cn(C(C)(C)C)nn1)C(=O)NCCCSC)C2 91776,c1(OC)cc(OC)c(CN2CCN(C(c3ccnc(F)c3F)=O)C3CC23)c(Br)c1 91777,CC1(C)C(NC(c2cncnc2C2CC2)=O)C(C)(C)C1NC(C1CC(F)(F)C1)=O 91778,C#CC1(C(=O)NCCC(C)N(C(=O)CCc2ccncc2)C)CCC1 91779,c1(CC)cc(N)ccc1C(=O)N(C1CCCCC1N(C(=O)C(N)=O)C)C 91780,N1(C(C(C)C)=O)CCC(CC(C)NC(C2CCCN2C)=O)CC1 91781,N1(C(C=CC(=O)N(C)C)=O)CCCC1C(=O)NCCc1ccncn1 91782,C1(NC(CC2C(C)(C)N(C(=O)Cn3[nH]cnc3=N)CC2)=O)CCC(C2CC2)CC1 91783,C1(C(=O)Nc2ccc(COC)cc2)CC1C1CN(C(c2ccc(CO)o2)=O)C1 91784,c1(CN(C(=O)Nc2ncc(F)cc2Cl)CC)ccc(F)c(F)c1 91785,c1(C(Cc2ccccc2)NC(C(=C)Cc2ccccc2Cl)=O)cc(Cl)cc(Cl)c1 91786,c1(C(=O)NCC2OCC(CNC(=O)C=Cc3ccccn3)C2)cc(=O)c(O)c[nH]1 91787,C(C)(CNC(=O)Cn1cc(C(C)O)nn1)(CC(C)C)NC(C(CCOC)OC)=O 91788,CC1CC(NC(c2ccsc2C(F)F)=O)CCN1C(C1CCC(C#N)CC1)=O 91789,C1(C)(CNC(CCC=C)=O)CCN(C(c2ccc3c(c2)CC3)=O)CC1 91790,Cc1cc(O)nc(C)c1C(N1CCC2(C1)CN(C(C1(C)CCCOC1)=O)C2)=O 91791,C=C(CC)CN=c1nc(N(CCCN2CCOCC2)C)c2c([nH]1)CCC(C)C2 91792,CC1CCc2[nH]nc(C(N3CCC(NC(=O)C4=CCSC4)C3C(C)(C)C)=O)c2C1 91793,C1(NC(C2CC(C(C)C)C2)=O)CCOC(CNC(c2cccc(C(F)F)n2)=O)C1 91794,c1(C(C)CNC(=O)NC(C2CCOC2)COC(F)F)ccccc1Cl 91795,C1(C(=O)NC(CC)CO)CN(C(=O)C(C)NC(=O)Cn2cnnn2)CCC1O 91796,CC(C)CC(CNC(c1ccc(C(F)(F)F)cn1)=O)NC(=O)COC1CCC1 91797,c1(OCC(=O)NCC2C(NC(COCC#C)=O)C2)cccc(C(N)=O)c1 91798,c1(C(n2nnnc2C2(NC3CS(=O)(=O)C3)CCC2)C)ccc(F)c(Cl)c1Cl 91799,C1(NC(c2c(C(N)=O)nccc2)=O)CCCC(NC(=O)CCCCC2CC2)CC1 91800,C(c1ccncc1)=CC(N1C(C(=O)NCC(C)OCC#C)CC1C)=O 91801,Cc1cnc(C=CC(=O)N(C)CC2CCN(C(C3CCN3C3CCCC3)=O)C2)[nH]1 91802,C12(C(=O)NCCCCCNC(c3cc(CC)c(CC)o3)=O)CCCCN1CCC2 91803,C(CC(C)(C)C(=O)NC(CNC(c1ccccc1NC(N)=O)=O)CO)OC 91804,N1(C(CN(C(C#CC2(CC)COC2)=O)C2CC2)=O)CCCC2CN(C)CC12 91805,C1(N(C(=O)CCC2CC(F)(F)C2)CC)CCCN(C(=O)C(C)CNC(N)=O)C1 91806,N1(C(=O)OC)CCCC(C(=O)NC2(CNC(=O)Cc3csc(SC)n3)CCC2)C1 91807,C1(NC(CC=C=C)=O)COC2(CCCN(C(=O)Cc3cc(OC)ccc3Cl)C2)C1 91808,N1(C(c2nc(CCC)oc2)=O)CCC2(CCCC2NC(c2c[nH]c(=NC)o2)=O)C1 91809,N(C(=NCCC(C)CC(C)(C)C)NCc1nn(C)cc1C)C(C=C)C 91810,N1(CC)CCN(C(C2CCN(C(=O)C3=CCCC3C)CCO2)=O)CC1(C)C 91811,C1(C(NOCC=C)=O)CC(O)CN1C(=O)CC(C)(F)F 91812,c1(C(=O)NC(C)CNC(C2CC(NS(C)(=O)=O)C2)=O)nnn2c1CCCCC2 91813,c1(OC)ccc(Br)c(F)c1CN1CCOC(C)CC1 91814,c1(-c2onc(-c3ccc(-c4ccc(C)cc4)nc3)n2)ccc2ncccc2c1 91815,C1(C(C)C(=O)NCC(C)(C)F)CCN(C(=O)C(C)(C)n2ccnn2)C1 91816,C(C)(CO)(C(=O)NCC1(F)CC(NC(c2cc(Cl)n(C)n2)=O)C1)NC(C)=O 91817,CC1CN(C(=O)C(=O)NC2CC2)CCN1C(=O)Cc1ccncc1Cl 91818,Cc1cc(Cl)cc2cc(C(=O)N(CC(O)CNC(C3CS(=O)(=O)C3)=O)C)[nH]c12 91819,C(=O)(C1=CCCOCC1)N1CC(C)CC(NC(c2c(CCC)occ2)=O)C1 91820,N1(C(C(C2CC2)OC)=O)CC(C)(NC(=O)N(CCCF)CC)C1 91821,CC(C)C(C)CC(=O)NC1(CNC(C2CC3CCCC23)=O)CCOCC1 91822,N1(C(c2c(NC(C)=O)c[nH]c2C)=O)CC(NC(=O)C2=CCOC2)C2(CCC2)C1 91823,N1(C(C(C(=O)OCC)CC)=O)CCC2(CC(C(N3CCC3CC3CCCC3)=O)C2)C1 91824,C=CC(C)(O)CC(=O)N1CCC(CCNC(=O)C(n2cc(Cl)cn2)C)CC1 91825,C1(C(=O)OC(C)(C)C)CCN(C(c2ccc(SCc3nncs3)cc2)=O)C1(C)C 91826,c1(C(C)C)ccc(C(=O)NC(C2CN(C(=O)C(CN(C)C)N(C)C)C2)C)s1 91827,N1(c2nc(C)cc(C)n2)CCC(C2CCN(C(=O)CC(C)C(F)(F)F)CC2)C1 91828,C=CCCCCCCC(=O)NCC(=C)CCNC(C1CCCCC12CCC2)=O 91829,c1(Cn2cc(C3CCN(C(c4ccc(C(C)=O)s4)=O)C3)nn2)ccc(Cl)nc1 91830,c1(NC(C(C(C)NC(=O)C(C)(Cl)Cl)C)=O)cc(O)cc(F)c1 91831,N1(C(c2cc(C(N)=O)[nH]c2)=O)CCCC2(CCCN2C(c2cc(O)ncn2)=O)C1 91832,c1(CCC)ccc(S(=O)(=O)N2CC3CCC(C2)N(C(c2nnc(C)o2)=O)C3)cc1 91833,c1(C(N2CC3C(CNC(CCn4c(C)cc(C)n4)=O)C3C2)=O)ccc(Cl)cc1O 91834,c1(C(=O)NC2CCC(N(C(c3nccc(OC)c3)=O)C)C2)ccc(C)c(C)c1O 91835,C(=O)(C1CCCc2scnc21)N1CCC(N(C(=O)CC2C=CCCC2)CC)CC1 91836,c1(CC(=O)NCCC(C)N(C(=O)C(C)Oc2cccnc2)C)ccc(Cl)s1 91837,C1(C(=O)NCCCCNC(C(CC)n2cncn2)=O)CCC2(CCOCC2)CO1 91838,C1(N(C(COCCCCC)=O)C)CN(C(=O)C(CC)C(C)C)CC12CC2 91839,c1(CNC(c2cc(C)on2)=O)ccnc(C(N2CCC(C(C)O)C2)=O)c1 91840,C#CCCCC(=O)N1CC(NC(C2(c3cncc(Br)c3)CC2)=O)C(F)C1 91841,Cn1nc2c(c1C(=O)NCc1c(F)ccc(CO)c1F)CN(c1nnco1)CC2 91842,S(=O)(=O)(c1ccccn1)N1CC(NC(C2N(C)CCC2)=O)(CO)C1 91843,N1(CC(=O)Nc2snc(SC)n2)CC2CCC2(CCN)C1 91844,Nc1cc(C(N2CC(CNC(=O)Cc3cc(O)nnc3O)C2)=O)cc(O)c1Cl 91845,C1(C(=O)NCC(C)(CO)NC(c2cc(F)n[nH]2)=O)CC2CCCC(C1)C2 91846,C(=O)(C1=CC2(CCOC2)C1)N(CC(=O)NCC1(C)CC2CCC1C2)C(C)C 91847,CC1(C)CCCC(C(=O)NCC23CC(NC(C4CCS(=O)(=O)C4)=O)(C2)C3)O1 91848,C1(N(C)C)CCCC(NC(=O)C(c2cccc(C(F)(F)F)c2)N)C1 91849,c1(NC(C2(c3cccc(-c4cc(C)nnc4)c3)CCCC2)=O)cccc(Cl)c1C 91850,C=C(Br)CC(C)(C)C(=O)NCCC1CCC(NC(c2cnnn2CC)=O)C1 91851,CC(C)(O)C(C)(C)CNC(C1C=CC(NC(C2(C)CCCO2)=O)C1)=O 91852,N1(C(CC(C)=C(C)C)=O)CCC2(CC1)CC(CNC(c1ncn(C)n1)=O)C2 91853,C1(OC)(CNC(=NCC2CCCO2)NC2CCCN(CC(F)F)C2)CCSCC1 91854,C(=O)(CCCCC(C)CC)NCC(CCC)C(=O)NCc1nn(C)c(=O)n1C 91855,c1(C(=O)OC)ccc(OCCNC(=O)C(=O)N(C2CCCCC2SC)C)cc1 91856,CCCCC(O)C(=O)N1CCC(CNc2ncc(C)c(O)n2)C1 91857,c1(C(N2CCC(NC(CC3(OC)CCC3)=O)C(F)C2)=O)cc2nc(Cl)ccc2o1 91858,C1(CNC(c2nc(COC)sc2)=O)C2CCC(C2)N1C(=O)CC1C=CCCC1 91859,C(C)(C)(CC(F)C(=O)NC(C1CCOCC1)C)NC(C(NOC)=O)=O 91860,c1(C(N2CC(NC(c3ccc(C)c(N)c3)=O)C2)=O)cnc2ncnn2c1O 91861,N1(C(Cc2n(C)ncc2)=O)CC2CC2C1CNC(C1(c2ccsc2)CC1)=O 91862,Cc1nc2ncc(C(=O)NCC3CCN3c3ncnc4c3ncn4C)c(=O)n2[nH]1 91863,N1(C(c2c(C)n[nH]c2)=O)CCc2nc(O)cc(C(N3CCCC(F)CC3)=O)c2C1 91864,C1(C2CCN(C(C3(C(C)C)CCCCN3)=O)CC2)CCCC2(CCC2)O1 91865,c1(CCC(=O)NCCC2CN(C(C3CC4CCC4C3)=O)CCO2)cccc(O)c1 91866,C(CC(C(=O)N1CC(O)C1)NC(C1C(C)C1C)=O)=CC 91867,c1(C(=O)NCCC2CCC(NC(C(CSC)C)=O)C2)ccc([N+](=O)[O-])cc1F 91868,C=CCC(C)C(=O)N=S(C)(=O)c1cnn2c1CN(C(=O)CCCCO)CC2 91869,CC1(NC(=O)CC2CC23CC3)CCCN(C(c2cscc2Cl)=O)C1 91870,C12(C(=O)NC(c3ccccc3F)CNC(C3(CF)CC3)=O)CCN(CC1)C2 91871,C=CCCC(F)(F)C(=O)N1CC(C(=O)N(CC(C)O)C2CC2)C2(CC2)C1 91872,CC1(C)C(C(=O)NC(C2CCCCC2)C(N2CCC(F)(F)C2)=O)C1(F)F 91873,S(=O)(=O)(c1ccc(Br)cc1NCc1ccc(-c2ccccc2)cn1)NCC(=C)C 91874,N1(C(C(=CC2CCCC2)C)=O)CC2CCOC2(CNC(c2cncc(C)n2)=O)C1 91875,N1(C(C2C(CCOC)C2)=O)CCOCC(NC(=O)C(F)(F)CN(C)C)C1 91876,Cc1ccc(F)c(CNC(C2CCC(CNC(C3CC4CCC4C3)=O)O2)=O)c1 91877,c1(CC)ccc(C(=O)NCC2(C)CC(NC(=O)C(C)(C)n3cccn3)C2)nc1 91878,CCCC(CCC)C(=O)NC1CC(O)CN(C(=O)C(C2CCOCC2)F)C1 91879,N1(C(C2N(C(c3ccn(C(F)F)n3)=O)CC2)=O)CCC2(OC)CCCC12 91880,C(=O)(C(CC(F)F)c1ccccc1)N(CCCNC(C(C=C)(C)O)=O)CC 91881,N1(C(c2c(CCC)nco2)=O)CCC(C)(C)C1C(=O)N(C)Cc1nccn1CC 91882,CC(C)C(F)C(=O)NC1CCCC(C(=O)NCc2cn(C3CC3)nn2)C1 91883,C1(C(N(C2(C(NOCCCOC)=O)CCC2)C)=O)CC(=O)CCO1 91884,C1(N(C(=O)CC2CSCCS2)CC)CC2CCC(C1)N2C(=O)Cc1ccsc1 91885,N1(C(C2CC(CNC(=O)CSCC(F)F)C2)=O)CCOCC2(CC2)C1 91886,c1(C(N2CCC(O)(C(=O)OC)CC2)C(=O)NCCOCC)nc(Br)c(C)cc1Cl 91887,C#CCCN=C(NCC(C)Cc1cccs1)NC1CC(CNC(=O)OC(C)(C)C)C1 91888,C1(C(N(C(C)C)CCNC(C2CCN(CC(F)(F)F)C2)=O)=O)CCCOCC1 91889,Cc1cc(C(=O)O)cc(C)c1NC(=O)C(=O)NC1N(CC(C)O)CCCC1 91890,c1(C(C)C)ccc(C#N)c(NC2CCCCC2CNC(C2CC2F)=O)n1 91891,CCN=c1[nH]c(C)c(C(N2CCCCC2CNC(C2CCNC2=O)=O)=O)s1 91892,c1(C(N2CC(C)N(C(c3cnn4ccsc34)=O)CC2)=O)cccc2ccsc12 91893,CC1CC(CNC(C2(C(F)F)CCC2)=O)CN1C(=O)COc1ccccc1Cl 91894,Cc1cc(=NC(C)Cc2ccc(Cl)s2)[nH]c(=NCc2nnc3c(Cl)cccn23)[nH]1 91895,Cc1ccc(C)c(SCC(=O)NCCCC(C)NC(=O)Cc2nccs2)c1 91896,C1(C(N2CCC(N(C(CN(C(C)=O)C)=O)C)C2)=O)COCCN1C 91897,N1(C(C=CCCC)=O)CCC(NC(c2csc(CC)n2)=O)CC1C 91898,C=CC(CCC)CC(=O)N1CCN(C(=O)CN(C(=O)C(C)NC(=O)CC)C)CC1 91899,n1(CC)cc(Br)c(C(=O)NCC(C)(CO)NC(c2[nH]c(C)nc2C)=O)n1 91900,c1(CC)nc(C)c(C(=O)NCCC2CCC(NC(=O)Cc3cccn3C)C2)s1 91901,N1(C(Cn2ccc(C)n2)=O)CC2CN(C(c3ccc4nsnc4c3)=O)CC2C1 91902,c1(C(=O)NC(CNC(C2CC(O)C2)=O)C2CC2)cncc2c1CCCC2 91903,c1(C(=O)NCCC(CCNC(CC=CC)=O)C)c[nH]cc(Br)c1=N 91904,N1(C(c2nc(C(OC)OC)sc2)C(=O)NC(C)CC)CC(N(C)C)C(C(N)=O)C1 91905,C(CCC(C)(C)NC(=O)C(COC(C)C)N(C(C)COC)C)OC 91906,Cc1cccc(S(=O)(=O)CCCN2CCn3c(C(F)F)nnc3C2)c1 91907,C(=O)(C1CC=Cc2ccccc21)Nc1n(C)nnc1CN 91908,N1(C(C(C=CC)O)=O)CCCCC(N(C(=O)CN(c2ccc(Cl)cc2)C)C)C1 91909,C(=O)(C1=CCCCC1C)N1CC(O)(CN(C(CCCOC)=O)C)C1 91910,C1(CNC(c2c(COC)cco2)=O)CCCN(C(=O)C(F)(F)c2csc(Cl)c2)C1 91911,C1(CNC(C(CC)SC)=O)CCCN(C(=O)CSc2ncccn2)CC1 91912,N1(C(=O)Nc2c(C(=O)NC)n(C)nc2)CCC2NC(=O)NCC2C1 91913,N1(C(C(CC)C(C)(F)F)=O)C2CCCC1CN(C(=O)C(C)(C)S(C)(=O)=O)CC2 91914,C1(CNC(COCCC)=O)CC2COCC2N1C(c1c(F)ccnc1F)=O 91915,c1(C(N2CC3CC2CC3O)C(=O)NCCCC)ccc(C)c(Cl)c1 91916,C(=O)(C(O)C1=CCCCC1)NC1(c2cn(C3CC(C(=O)O)OCC3)nn2)CC1 91917,C1(NC(C2(CC)CCCCC2)=O)CN(C(=O)CC2CCN(C)C2)CC1N=[N+]=[N-] 91918,N1(C(C(C(CC)O)C)=O)CC=C(CCNC(c2ccnn2CC2CC2)=O)CC1 91919,CC1(C)CCN(C(=O)CC2CCC(=O)NC2)C1C(=O)NC1(CF)CCC1 91920,CC(O)(CC(=O)NC1CCCC1C(=O)NCc1cc(F)c(Cl)cc1Cl)CC(=O)O 91921,C(=O)(CC(C(C)CC)NC(C1(CO)CCOC1)=O)NC(C=C)CO 91922,C1(NC(C(CC(C)C)N(C)C)=O)CCN(C(=O)Cn2cnc(C#N)n2)CC(O)C1 91923,CCC(C(O)C(F)(F)F)N=c1cccc(S(=O)(=O)NCC2(C)CC3(CC3)C2)[nH]1 91924,c1(C(C(=O)Nc2cccc(OC3CC3)c2)O)cc(F)c(F)c(F)c1 91925,C1(OC)(OC)CCC1C(=O)NC1CCCC1CNC(=O)C(c1ccccc1)OC 91926,c1cc2[nH]c(=NCCCOC3CC3)[nH]c(=NCC3CCCOC3)c2[nH]1 91927,n1(COC)nccc1S(=O)(=O)N1CCCC12CCOC2 91928,C12COCCN(C1)C2=O.C1(OC2(CNC(CC3CC(C)C3)=O)CC2)CCOCC1 91929,CC(C)(C)CC(O)CC(=O)N1CC=CC(C(=O)NCC(c2ccccc2)F)C1 91930,C1(O)(C(=O)NC2C(C(c3ccccc3)NC(CCC)=O)COC2)CC(C)(C)C1 91931,CCC(C)(CC)C(=O)NCCC(CNC(c1[nH]ccc1C)=O)OC 91932,CCCC(O)C(CO)NC(c1cnn(CCNC(=O)CSCCC(C)C)c1)=O.C(C)=O 91933,c1(CC(=O)NCCC2CCN(C(C(CSC)OC)=O)C2)ccc(C(C)(C)C)cc1 91934,N1(CC(N2C(CNC(Cc3cc(C)ns3)=O)C=CC2)=O)CCNC(=O)C1 91935,Cc1ccc(C#N)c(NC(C2C3CC2N(S(=O)(=O)c2ccncc2)C3)=O)c1 91936,c1(OC)cc(S(=O)(=O)NC2CCC3(CN(Cc4ccsc4Br)C3)O2)ccc1Br 91937,Cc1nc(C(N2CCC3CCN(C(c4nccn4C)=O)CC23)=O)c2ccccn12 91938,N1(C(COC2CCCC(C)C2)=O)CCN(C(=O)Cc2ccc(F)nc2)CCC1C 91939,n1(CCC(N2C3C(NC(C(C)(C)F)=O)CC(C3)C2)=O)ccc2ccccc12 91940,c1(NCc2ccc(C)n(C)c2=O)sc2ccccc2c1C#N.c12ccc(cc1)C(=O)NOC2=O 91941,C1(NC(c2cnc(CC)s2)=O)CN(C(c2cc(C)nc(Cl)c2)=O)CCC1C 91942,c1(C(C(=O)NCC(C(C)C)NC(C2(CO)CCOCC2)=O)C)c(Cl)cccc1Cl 91943,C=CC(C)(CC)C(=O)N1CCN(CC(N2CCCN(C(C)=O)CC2)=O)CC1 91944,c1(C(=O)NC2CCN(C(CN(C(C)=O)C)=O)C2(C)C)nn(C)c2c1CCC2 91945,C(=O)(C(O)CC(C)(C)C)NCC12C(NC(c3c(CC)oc(C)c3)=O)CC(CC1)C2 91946,N1(C(CCC(C)OC)=O)CCCN(C(c2cc(C3CC3)nnc2O)=O)C(C)C1 91947,c1(N2CCN(c3ncc4c(n3)NC(=O)C4)CC2)ccc(C2=COCCC2)nn1 91948,N1(C(CC=C)=O)CC(CNC(=O)C(C2CC2)SC)CC12CCC2 91949,c1(NCCOC)cc(C(=O)NC2CCCC2CN)ccn1.c1(C(=O)N)nc(C)no1 91950,C1(C(N(C2(C(N(CC(CC)C)C)=O)CCC2)C2CC2)=O)C2CCC(F)C12 91951,C#CC1CN(C(=O)CC2(C=C)CN(C(c3cc(C(N)=O)c[nH]3)=O)C2)CCN1C 91952,C1(OCC)CC2(C1)CC2C(N1CCC(C(C)NC(c2nocc2C2CC2)=O)C1)=O 91953,C(=O)(C(CC)CCCC)N1CC(C(=O)Nc2cccc(CC=C)c2)C(OCC)C1 91954,C12(CNC(c3c(C)coc3)=O)CCC(CC1)N2C(c1cc2scnc2[nH]1)=O 91955,C=Cn1cc(C(c2nnnn2Cc2ccccc2OCC)NC2CC2CF)cn1 91956,C1(OC)CC2CC1CN(C(=O)CC1(N(C)C(c3cnncc3C)=O)CC1)C2 91957,c1(C(=O)NCCCOCCN(C(CC2CCC(C)O2)=O)C)cccc(Cl)c1 91958,C(C(=O)N=c1c(Cl)c[nH]cc1I)Oc1c(OCC)cccc1 91959,c1(NCC(CC(=O)NC)C)[nH]c(=NC(C)c2nncs2)nc2c1ncn2C 91960,c1(CC(=O)NCC(C)N(C)C(C2CN3CCC2CC3)=O)ccc(Br)cc1F 91961,c1(C(CNC(c2cnnn2C2CC2)=O)NC(C2CCCCC2)=O)ccccc1F 91962,C1(NC(C2C(C)C2)=O)CN(Cc2cc(Cl)cc(Cl)n2)CC1C#N 91963,C(=O)(C(C)(C)C(=O)N1CC(NC(C2C3CNC(=O)C23)=O)C(F)C1)OCC 91964,c1(C(=O)NC(CC=C)CNC(c2ncoc2CC)=O)n[nH]c(C)c1[N+](=O)[O-] 91965,Cc1cc(O)ncc1C(=O)NC1CC1CNC(c1ccc(O)c(Cl)n1)=O 91966,C1(C(=O)NCCCC(C)NC(c2nn(C)cc2Cl)=O)CC12CC(C)(C)C2 91967,N1(C(C23N(C(c4c(C)cn(C)n4)=O)CCC2C3)=O)C2CCC1CC1(C2)N=N1 91968,N1(C(CC(=C)C)=O)CCC2(C1)CN(C(c1ccnn1C(F)F)=O)C2 91969,Cc1nsc2ncc(C(N3CCCC4(C3)CN(C(C3CCCOC3)=O)C4)=O)cc12 91970,c1(CC)ccc(C(=O)NCC(C)NC(=O)COCCCC(C)C)c(OC)c1 91971,CC1CCC(C)(C(=O)NC2CC(NC(c3cncc(N)n3)=O)C2)C1 91972,c1(NC(C2CC(O)CN2Cc2ccc(Br)nc2)=O)c(F)cc(F)cc1[N+](=O)[O-] 91973,c1(-c2c(OC3CC(C)(O)C3)c[nH]n2)ccc(N)cc1 91974,c1(C(=O)NCC(C(C)C)NC(c2cc(OC)ncn2)=O)sc2cccnc2c1Cl 91975,C(CC(=O)NC12CC1CN(C(c1nc(Cl)sc1C)=O)C2)(C(C)C)OCC 91976,C(CCCCCNC(C1CC(O)CN1C(C1(OC)CCOC1)=O)=O)OC 91977,c1(N(C(=O)CC(Cc2ccccc2)C(F)F)C(C)=O)cc2cc(Cl)cnc2[nH]1 91978,c1(CC)ncncc1C(N1CCC(CNC(C23COC(CF)(C2)C3)=O)C1)=O 91979,c1(C(c2nnnn2C(C)C)NCC(CC=C)(C)C)c(F)cnc(Cl)c1C 91980,N1(C(c2cc(C)[nH]c2)=O)CC23CCCC2(C1)CN(C(=O)CCc1ncccn1)C3 91981,CN1CCc2cc(C(=O)N(C3CC(NC(C4CCCC(C#N)C4)=O)C3)C)ccc21 91982,c1(CN2CC(F)(C(=O)NCC)C2)csc2ccccc12 91983,C(N=c1[nH]c2cc(Br)ccc2o1)C1C(C)CN(C(C2CCOC2)=O)C1 91984,c1(Oc2ccc(C)cn2)ncnc(N2CCC(O)C(F)C2)c1C 91985,N1(C(c2c(C)cc(Cl)cc2)=O)CCCC(C2CCN(C(=O)C(O)C(C)C)CC2)C1 91986,N1(C(=O)C(F)F)CC2CCC(C1)N(Cc1ccc(C(F)(F)F)s1)C2 91987,c1(OC)ccc(OC)c(C(=O)NC2CCN(Cc3ccc(O)c(C)c3)CC2F)c1 91988,N1(C(CC(C)SC)=O)CCOCC1CC(=O)NOC1CCC(O)C1 91989,CCC(C(=O)N1CC(C)C(C)(CNC(C2CC(O)C2)=O)C1)C(F)(F)F 91990,CCC(C)C(O)C(=O)NCC12COC(CNC(=O)C(F)CC3CCCCC3)(C1)C2 91991,C1(NC(c2cc(C)[nH]n2)=O)CC(O)CN(C(c2ccc(-c3ccccc3)o2)=O)C1 91992,c1(NCCOCC=C)cc(=NC2CCOc3ccc(F)cc32)[nH]c(COC)n1 91993,C1(CCNC(C(C)C2CC2)=O)CCC(NC(=O)CN2CCOC2=O)C1 91994,c1(C(N2CCC(NC(c3n(CC#C)cnn3)=O)(CO)C2)=O)c(Cl)ccc(F)c1F 91995,c1(OC)c(C(=O)NCC(C)N(C(=O)COC2CCOC2)C)cc(Br)cc1F 91996,CN1CCOCC1CC(=O)NC12CC1CN(C(c1cn(-c3nccs3)nn1)=O)C2 91997,C1(CNC(C2CN(C(C)=O)C2)=O)CC(F)(CCCN(C)C)C1.C1C(=O)N1 91998,c1(C(=O)NCC(CO)NC(c2cc(CC)c(C)s2)=O)cc2c(ccn2C)[nH]1 91999,C1(C(N2CCCC(N(C(Cc3c(C)cco3)=O)CCF)C2)=O)CCCCC1(F)F 92000,C1(C(=O)NCC(CC)(C)O)COCCN1C(c1cc(=O)cc[nH]1)=O 92001,C=CCC(C)(C)CC(=O)N1CC=CC1CNC(c1ncnc(C)c1C)=O 92002,C1(CNC(CSCCC(C)C)=O)CN(C(=O)CC(C)(C)C#N)CC2(CCC2)O1 92003,N1(CC)CCN(CC(=O)NCCN(C(=O)C(N2CCN(C)CC2)C)C)CC1 92004,CC1=NOC(C)(C(N2CCC(Cn3cc(CCC#N)nn3)C2)=O)C1 92005,C1(C(=O)NC(C(C)C)C2CCC2)(CC)CCN(C(c2c[nH]nc2C)=O)CC1 92006,N1(C(C(CCC)OC)=O)CC2(C1)SCCC2NC(=O)Cc1cnoc1 92007,c1(CNC(C2CC(CCNc3cc(OC)ncn3)C2)=O)ccc(C)c(Cl)c1F 92008,C1(NC(C2(CC#C)CCCC2)=O)CCC(C)(NC(c2cc(Cl)ncc2O)=O)CC1 92009,Cc1noc(C)c1CCC(=O)NC1(C)CC(NC(C2CC23CC3(F)F)=O)C1 92010,N1(CC(C)NC(=O)OC(C)(C)C)CCC2(CC1)OCCc1ccccc12 92011,c1(NC(CCC)CCCNC(=O)CCC(N)=O)ccc(S(C)(=O)=O)cc1[N+](=O)[O-] 92012,C1(C(=O)NC2C(C(c3sccc3C(C)(C)C)NC(C)=O)C2)CCc2ccnn2C1 92013,Cc1ccc2[nH]c(C(N3CC(CCCCNC(=O)C#CC4CC4)C3)=O)cc2c1 92014,n1(CC)cc(Br)cc1C(=O)NC(C1(O)CN(C(C2CC23CCC3)=O)C1)C 92015,C1(CNC(C(CSCC)NC(C2COCC(C)O2)=O)=O)(OC)CCCCC1 92016,CC(C)CC(C(=O)NCCCNC(N)=O)ONC(=O)C1CN(C)C1 92017,C1(F)(C(=O)OCC)CN(C(=O)Oc2cccc(C#N)c2)CC12CCOCC2 92018,O=C1NCC2(CO1)COC(CF)CN2C(C1C2CC=CCC12)C(=O)OC 92019,C1(NC(C2CCCNS2(=O)=O)=O)CCN(C(C2CCCSC2)=O)CC12CCC2 92020,CC(C(F)C(=O)N1CCC(NC(=O)CC2CC3C=CC2CC3)C(O)C1)C(F)(F)F 92021,C=CCC(CNC(c1cc(CNC(C)=O)on1)=O)NC(=O)COc1cc(C)on1 92022,C1(C(=O)NC(CCC)CCO)CN(C(C2(SC)CC2)=O)CCC1(C)C 92023,c1(C(N(CC(=O)N(CC(CN(C)C)O)C)C2CC2)=O)c[nH]cc1C1CC1 92024,c1(NC(N2CCC(n3cc(CO)nn3)C2)=O)cc(Cl)cc2nccnc12 92025,N1(CC(COc2c(CC=C)cccc2)O)CCc2nc(C)n(C)c2C1 92026,N1(C(C2(CCC)CCC2)=O)CCC2C(C(=O)NCC(F)(CC)CC)C2C1 92027,CCCCCCCC(O)C(F)(F)C(=O)NCCN(C(=O)CC1CCCCCC1)C 92028,c12ccc(cc1Br)S(=O)(=O)NC1(C)CN2CCO1.C(CCCCC1CC1)OC 92029,c1(OC)c(Cl)nc[nH]c1=NCCC1CCC(NC(=O)C2=CCCOCC2)C1 92030,c1(C2(F)CC(C(=O)NC(C)CCN(C)C(C3CC3C)=O)C2)cccc(F)c1 92031,Cc1cccc(C(N2CCC(C(N3CCCCC(C)C3)=O)C2)=O)c1I 92032,N1(C(C(CSC)O)=O)CCC2(C1)CN(C(c1n[nH]c3c1CSCC3)=O)CCO2 92033,C(=O)(C(C)(C)CCC(C)=O)NCc1c(OC)ccc(F)c1 92034,c1(NC(C(CCC2CCC2)NC(C2CCCCO2)=O)=O)cccc2c1CCC2 92035,C1(CN(C(c2cc(C(F)(F)F)ncn2)=O)C2CC2)CCN(c2ncns2)C12CC2 92036,N1(C(CCN(C(=O)CC2C=CCC2)C)=O)CCCCC1CF 92037,c1(C(=O)NC(C(C)C)CNC(=O)C(c2ccnn2C)O)ccnc(C2CC2)n1 92038,c1(OC)cccc(C)c1NC(C1(CNC(c2cccn2C)=O)CCCO1)=O 92039,C12(CC)CCN(C1)C(=O)C1C=CC(C1)NC2=O.c1(C(=O)NC)ccn(CCF)n1 92040,CC1CN(C(c2cc[nH]n2)=O)CC1NC(c1ccc(-c2ncon2)cc1)=O 92041,c1(C(=O)NC(C(=O)NC2(C)CC(O)(CO)C2)CCF)cccc2occc12 92042,C(=O)(C(=O)CC(C)C)NC(C(=O)NCC(CC)C#N)(C)CO 92043,C12(C(CNC(=O)C(Cl)=CCl)NC(=O)CSCc3ncc[nH]3)CCC(CC1)C2 92044,N1(C(CC#CC)=O)CCCC(C(=O)NCc2cc(C)sc2C)C1 92045,C1(CC(=O)NCCOC(C)=O)CCCN(C(=O)Cc2cn(C)nn2)C1 92046,c1(C(N2C(C3CCN(C(C(CCC)O)=O)C3)CCC2)=O)coc2ccc(C)cc12 92047,Cc1cc(NC(C2CC(C)(C)CN2C(c2cccc(C)c2N)=O)=O)cnc1Cl 92048,c1(C(N2CCC3(CC(NC(c4occ(C)c4)=O)C3)C2)=O)ccc(C)c2c1CCC2 92049,c1(CC(N2CC(O)(C(C)NC(C3CC(CCC)C3)=O)C2)=O)c(C)nc(O)nc1O 92050,C1(C(=O)NCCC(CNC(=O)C(C)(C)n2cncn2)OC)CCc2c[nH]nc2C1 92051,C1(CC(=O)NCC(C(=O)OC)OC)CCCN(C(=O)C(OC)OC)CC1 92052,N1(C(C(C2CC2)SC)=O)CCCC(O)(CCNC(=O)CCC2CC2(F)F)C1 92053,N1(C(C2N(CCCC)CCCC2)=O)CCCCC(NC(C2(CC(C)C)CC2)=O)C1 92054,C(=O)(C(C(C)(F)F)NC(=O)CCc1ccc(F)c(CO)c1)OC 92055,c1(CCC)ccc(CC(=O)N(C)CCNC(=O)C(C)Cc2ccc(Cl)cc2)cc1 92056,C1(NC(c2c(C)ncn2O)=O)CN(C(C2CC3CCC2C3)=O)C2(CCCC2)C1 92057,c1(C(=O)NCC(C)CO)c(Cl)nn(C)c1Cl 92058,c1(CC)cc(C(=O)NCC(N2CCN(C(=O)C(O)COC)CC2)C)ccc1F 92059,C(=O)(C(C)NC(C)=O)NCCN(C1CCCC1)C(CSCC#C)=O 92060,CCC1=NOC(CC(=O)NC(C2CCN(C(C3C(Cl)(Cl)C34CC4)=O)C2)(C)C)C1 92061,c1(CC)ccc(N2CC(C(N3CCCC(CNC(=O)CO)C3)=O)CC2=O)cc1 92062,c1(C(=O)NC2CN(C(CSCC=C)=O)CC2N=[N+]=[N-])cnc2c(c1)ncn2C 92063,Nc1cccc(C(=O)NC2(CCO)CN(C(c3ccnnc3O)=O)C2)n1 92064,c1(C(N2CC(C)C(C)C2)C(=O)NC(CC)C)c(Cl)nc(Cl)n1C 92065,Cc1ccc(C(CNC(=O)CC(C)(F)F)NC(c2ccn(C3CC3)n2)=O)cc1 92066,N1(C(CCCC)=O)CCN(C(=O)COc2ccc(CC)cc2)CCC1C 92067,C1(C(N2CCC(C(C)C(=O)NCc3ncsn3)CC2)=O)CN(C)CCN1C 92068,C(CC(=O)NCCC(O)C1CCC1)(C(F)(F)F)NC(=O)CCc1nccs1 92069,C1(C(N2CCC(O)(CN(C(CCCC(=C)C)=O)C)C2)=O)Cc2ccc(F)cc2O1 92070,CC(C)C(C(=O)N1CC(CNC(=O)COc2ccc(C(N)=O)cc2)C1)C(C)C 92071,c1(C(N2CC(C)C(CNC(=O)C(C)C(C)(C)O)C2)=O)ccc(F)c(F)c1 92072,N1(C(=O)NC2CCCN(CCn3ccnc3)C2)CCOC2(CCCC2)C1 92073,N1(C(C(C)N(C(COCCC#C)=O)C)=O)CC2(C1)CC(C)(O)C2 92074,n1(CCF)nc(-c2ccoc2)nc1-c1ccc(OCC(F)F)cc1 92075,Cc1ccc2cc(C(=O)NCCCNC(=O)C(F)C3CC3)c(C)nc2c1 92076,N1(C(=O)C=CCOc2ccc(F)cc2)CCN(C(c2cccnc2)=O)C2CC12 92077,C#Cc1cccc(C(=O)NCc2cccc(CNC(c3cncs3)=O)c2)c1F 92078,C(=O)(CC(C)C(C)C)NC1(C(=O)NCc2ncc(CC)s2)CCCCC1 92079,Cn1cc(C#N)cc1C(=O)NC(CC1CCOCC1)C(=O)NCc1nnc(O)o1 92080,C1(CNC(CCN(C(C)C)C(C2CC3CC(=O)C2O3)=O)=O)CCCC2(CC2)C1 92081,CC(CCN(C(=O)CNC(C1CCCO1)=O)C)NC(=O)CSn1cncn1 92082,N1(C(CCOC(CC(C)C)C)=O)CCCC1(C)CNC(C1CN(C)C(=O)N1)=O 92083,c1(C(C)(C)C)ccc(CCC(N2CC(c3ccccc3)CC2C(=O)OC)=O)cc1 92084,c1(CC(=O)NCC(CC)NC(C2(OC)CC2)=O)c(C)nc(C)nc1O 92085,c1(OC)ccc2c(NCc3nc4cc([N+](=O)[O-])ccc4[nH]3)nc(Cl)nc2c1 92086,C1(C(=O)NC(CN(C(=O)C(C)SC(F)(F)F)CC)C)CC2CCC(C1)S2(=O)=O 92087,N1(C(Cc2cn(C)nc2)=O)CCOCC(NCc2cccc(O)c2Cl)C1 92088,C12(NC(C3CN(C)C3)=O)CCCN(C(=O)Cc3cc(F)cc(Cl)c3)CC1C2 92089,n1(CC(=O)NC2C(NC(CC(=O)N(C)C)=O)CC2)ncn(C)c1=O 92090,c1(-c2nc(C)nn2-c2ccn(CC(=O)OC(C)(C)C)n2)ccc2ccccc2n1 92091,c1(C(N2CCC(CNC(C3(C=C)CCCCC3)=O)C2)=O)nnn2ccccc12 92092,C(CC(C(=O)O)NC(=O)CCSc1ccccc1)NC(N)=O 92093,C#CC1(F)CN(C(c2ccoc2CNC(C2CC2(C)C(F)F)=O)=O)C1 92094,Cc1c(NC2CC2c2ccccc2)ncnc1N1CCC(C)CC1 92095,CC1C(C)N(C(c2cnc(F)c(F)c2)=O)CCN1C(=O)CCc1cnccn1 92096,N1(C(CCCn2cc(-c3ccc(NC(C)C)cc3)nn2)=O)CCOC(C#N)C1 92097,C=C(C)C1OCCC1C(=O)NC(C)(C)C=CC(=O)NCC12CCC(CO1)C2 92098,N1(C(CCC(C)OC)=O)CCC(C2(NC(c3ccccc3C#N)=O)CCC2)CC1 92099,C(CNC(=O)CC(=O)N(C)C)(CC(=O)NCC(C)CCC1CC1)OC 92100,c1(C(=O)NC2CCCN(C(C=CC)=O)CC2)cc(S(=O)(=O)NC)cs1 92101,N1(C(C=C(C)c2cnn(C)c2)=O)CCC(NC(=O)CCC2CC2)C12CCC2 92102,C1(C)(C(N(CCCCN(C(C(CC)NC(C)=O)=O)C)C)=O)CCCCC1 92103,C1(CNC(CN(CC(=O)NC(C)C)C)=O)CCCN(C(C2CC(N(C)C)C2)=O)C1 92104,C1(NC(=O)C(F)C2CCOC2)(CNC(C23CCC(C2)C3)=O)CCCC1 92105,C1(CNC(=O)CC2CC3(CCO2)CC3)CCC2CN(C(=O)COC(F)(F)F)CC12 92106,S(=O)(=O)(CCCN=c1nc2scnc2c(NCC2(COC(C)C)CC2)[nH]1)NCC 92107,C1(C(N2CCCC(N(C(=O)CC3CCCS3(=O)=O)C)C2)=O)CCCCC1(F)F 92108,c1(C(=O)NCC2(CNC(Cc3ccc(C)s3)=O)CCC2)cc2cn[nH]c2cn1 92109,c1(C(=O)NC2C(C)CN(C(=O)C(O)C3CCCC3)C2)cc2ccc(F)cc2[nH]1 92110,c1(CN2CCC(C(=O)Nc3n(C)cc(Br)n3)CC2)ccn2ccnc2c1 92111,N1(C(c2c(CCC)n(CC)nn2)=O)CCN(C(C2CSC2)=O)C(CC(C)(C)C)C1 92112,Cc1cnc(N(C2CCNCC2F)C(c2ncccc2C)=O)nc1 92113,C1(C(=O)NCCOCCSC)(C2CC2)CCCN1C(=O)C(C)NC=O 92114,N1(C(CC(COC)(C)O)=O)CCN(C(=O)CCOCC2CCCO2)C2CCCC12 92115,c1(CC(=O)NCC2(F)CC(NC(C3CC3F)=O)C2)cc(Cl)ccc1Cl 92116,N1(C(C2(COC)CC2)=O)CCC2(CC2C(N2CC(C#N)(COC)C2)=O)C1 92117,c1(C(=O)NCCCNC(C2(S(N)(=O)=O)CC2)=O)ccc(=O)n(CC2CCCO2)n1 92118,C1(NC(c2cc(COC)on2)=O)CCCN(CC(O)Cn2nc(C)nc2C)C1C 92119,Nc1nn2ccccc2c1C(=O)NC1CCC(F)(F)C1O 92120,C1(C)(CC)CC(C(=O)NCc2cc(C(=O)NC(C)Cc3cnccn3)no2)C1 92121,C(=O)(CC(C)CC(C)(C)C)NC(CC1CC2N(C(CC=CC=C)=O)C(CC2)C1)C 92122,c1(CC(=O)NCC2=CCN(C(COC(C)=O)=O)CC2)c(C)[nH]c2ccnn2c1=O 92123,CN1CCC(CCNC(C2CC(C)(NC(C3CCCCC3)=O)C2)=O)C1 92124,Cc1cc(N)c(F)c(C(N2CCCC(O)(CNC(C3(O)CC3)=O)CC2)=O)c1F 92125,C1(C#N)(C(=O)NCC(CNC(C(C)=C(CC)C)=O)OC)CCCC(=O)C1 92126,C1(NC(c2c(Cl)cc(C)s2)=O)COC2CN(C(=O)CCNS(C)(=O)=O)CC12 92127,c1(C(=O)NCC2(C)CC(NC(C(C3CCCCO3)OC)=O)C2)ccc(Cl)cc1 92128,C(c1ccc(F)c(F)c1)=CC(=O)NC(C)CCCNC(C1CCC1C)=O 92129,C1(NC(C(CC)N(C)C)=O)CCN(C(=O)CCC(C)(C)C#N)CCC1CO 92130,C12(NC(C3CCC(C(N)=O)CC3)=O)CCC1CN(C(=O)CC1CCCS1(=O)=O)C2 92131,Cc1cc(=O)n(CCC(N2CC(N(C)C(C3C4COCC34)=O)C(O)C2)=O)cn1 92132,Cc1ccc(C(N2CCN(C(=O)C(C)n3cncn3)CC2C2CCC2)=O)c(N)n1 92133,c1(C(N2CC(OCCNC(CCCCOC)=O)C2)=O)ccnc2c1nnn2C 92134,C(c1csc(Br)c1)=CC(=O)N(C1CCCC(NC(=O)CC2(C)CC2)C1)C 92135,N1(C(CC2(C)CCCCC2)=O)CC(CO)C2(C1)CN(C(c1ccc(=N)[nH]n1)=O)C2 92136,c1(C(=O)NCC(CC)NC(C(C=C)(C)O)=O)cc(OC)cc2c1OCC2 92137,c1(C(=O)NCCN(C(=O)C(C2CCCCCC2)C)CC)cncc(C2CC2)c1 92138,c1(C(=O)NCc2[nH]nc(C(C)(C)O)n2)ncn2c1COc1ccccc1-2 92139,c1(C(N)=O)ccc(CC(=O)NCCc2nccn2Cc2ccccc2)cc1Cl 92140,CC1CC(NC(C2(C(F)(F)F)CC(F)(F)C2)=O)CN1C(c1cncc(O)c1)=O 92141,N1(C(CC2CC(OCC)C2)=O)CCN(C(=O)C=Cc2nccs2)CC1C1CC1 92142,C(=O)(C1=CCC(C)(C)CC1)N(CCN(C(c1ccc(OC)cc1Cl)=O)C)C 92143,CC1CCC(C)(C(N2CC(O)(CNC(C3CCCCN3C(C)C)=O)C2)=O)CC1 92144,C1(C(N2CC(OCCNC(CCc3onc(CC)n3)=O)C2)=O)OC2CCC1C2 92145,N1(C(C(CN(C)C)NC(Cc2c(C)n(C)nc2)=O)=O)CCN(C2CC2)C(C)C1 92146,Cc1nc(NC(c2ccnc(F)c2)=O)sc1C(=O)Nc1ccc(C#N)s1 92147,N1(C(c2cc(-c3ccc(C)o3)[nH]n2)=O)CCCC1(C)CNC(c1cnccn1)=O 92148,Cc1cc(C(N2CCC(C(N3CCN(CCC(C)C)CC3)=O)C2)=O)ncc1Br 92149,c1(C(N2CC(Cc3cn(CCC(C)=O)nn3)OCC2)=O)cc2sccc2cn1 92150,CC1COCC(C(=O)NCCC2CCCN2C(=O)CCC2CCSCC2)O1 92151,c1(C(=O)NCC(CC)NC(c2cnc(OCC)s2)=O)noc(C)c1[N+](=O)[O-] 92152,N1(C(C#CC(C)C)=O)CC(C(=O)NC2CCCN(c3ncccn3)C2)C(C)(C)C1 92153,N1(C(C(C(C)NC(CC(C=C)CCC)=O)C)=O)CC2(CCOC(=O)N2)C1 92154,N#CC1CN(C(c2cc(O)ccc2F)=O)CCN1C(c1ccsn1)=O 92155,C1(NC(C(CC(C)=O)C)=O)CC2CC1CN(C(=O)CSc1ccccc1)C2 92156,N1(C(c2c(C)nc(C)[nH]2)=O)CC2CCN(C(c3c[nH]cc3C(C)(C)C)=O)CC2C1 92157,c12cncc(c1)OC(=O)CC2.c1(NC(=O)OC)ccc(NC(C)C)cc1 92158,CC(C(=O)N(C)CCNC(=O)CC1(O)CCCC1)C(C)n1cccn1 92159,CC1(C)CC(NC(C2(CO)CCCCC2)=O)CN(C(c2ncc(F)cc2N)=O)C1 92160,N1(C(c2n(C)nc(Cl)c2)=O)CCC=C(C(=O)N2CCCC2(C)C2CCC2)C1 92161,c1(C(=O)NCC(C)NC(c2cc3n(n2)CCCC3)=O)cc2nc(Cl)ccc2s1 92162,C12(C(=O)NC3C(CNC(c4c(C(C)=O)ccs4)=O)CCC3)CCC(F)(CC1)C2 92163,c1(CNC(C2(C3CCCN3C(C3CCCS3)=O)CC2)=O)ccc(O)nn1 92164,C1(CS(=O)(=O)OC)CN(N2CC(O)(CC#N)C2)CC1C(F)F 92165,C1(NC(CCCNC(C=Cc2ncn(C)c2)=O)=O)CC2(CCOC2)C1 92166,N1(CC)CC(C(=O)NC2CN(C(c3ccccc3C(F)(F)F)=O)CC2C)CC1=O 92167,N1(C(C=CC(CC)=CC)=O)CC(CNC(C2CCN(C3CC3)CC2)=O)C(O)C1 92168,N1(C(CCSCCC(=O)OC)=O)CCc2ccccc2C(NC(=O)C(C)(F)F)C1 92169,c1(C(=O)Nc2ccc(O)c(C)c2O)cnn2cccc(-c3c[nH]c4nccc-4c3)c12 92170,C=CCC(CC=C)c1nc(-c2cccc(F)c2)nn1CCCc1ccccc1 92171,Cc1nc(C(=O)NCC(C)(O)CNC(=O)C(N2CCCC(O)C2)C)cc(O)n1 92172,C1(C)(CNC(C=C(C)C(F)F)=O)CCN(C(C2(C)CC2(Cl)Cl)=O)C1 92173,C(=O)(CCc1nccs1)NCCN(C(CNC(C)=O)=O)C 92174,C1(CC)CN(c2ccccc2)CCN1C(=O)Nc1ccc(F)c(C)c1 92175,C(=O)(C(O)(C(F)(F)F)c1ccccc1)NCC1OCCN(C(CN(C)C)=O)C1 92176,Cn1cc2ccc(C(N3CCC(NC(=O)CS(=O)(=O)CCO)C(O)C3)=O)cc2n1 92177,c1(NC(C(C)OC(c2cncc(C3CC3)c2)=O)=O)c[nH]c2ccc(F)cc12 92178,c1(N2CCC(c3ncc(C)s3)CC2)ccc2ncccc2c1[N+](=O)[O-] 92179,CC1CCC(CNS(=O)(=O)c2ccccc2OC(F)(F)F)Cc2ccccc21 92180,c1(C2(C(=O)NCC3(F)CC(NC(=O)Cc4cscn4)C3)CC2)ccc(Cl)nc1 92181,N1(C(CCc2ccc(C)cc2)=O)CC(N(C)C(c2ccnnc2O)=O)C2(CC2)C1 92182,C(=O)(C1=COCCO1)N1CCC(C(=O)NC(CC=CC)CO)C1 92183,C(N=c1ccc(C#N)n[nH]1)C1CCCN(C(c2c(C)ccc(C(C)C)c2)=O)C1 92184,C1(CN(C(C2(CC)CC2)=O)C)CCCCN1C(c1cncc(N)c1)=O 92185,C1(NC(CSCC=C)=O)CC(C(=O)N(C)CC2CC(F)(F)C2)CC1O 92186,N1(C(c2[nH]cc(C)c2)=O)CCC(CNC(=O)C(C)OCCC(C)C)CC1 92187,Cc1nc(O)nc(C)c1CC(N1CCC(CNC(c2sc(CO)nc2C)=O)C1)=O 92188,CCC(CCOC)C(=O)N1CCCC(C)(C(=O)NCCCO)C1 92189,CC1CC=C(C(=O)NC(C(=O)NC2CC2(C)C(F)F)C(C)(C)O)CC1 92190,C1(NC(C2CCN(C)CC2)=O)C2CC3CN(C(=O)CC4CSCCS4)C1C3C2 92191,C1(C(NOC(C(=O)OC)(C)C)=O)CCCN(C(c2cnncc2C)=O)C1 92192,Cc1cccc(C2(C(N3CCC(CC(=O)N(C)C)C3)=O)CC2)c1 92193,c1(C(C)=O)ccc(Br)cc1NC(C1CCN(C(c2cc(C)n(C)n2)=O)CC1O)=O 92194,c1(CC(=O)NCCNC(=O)CC2CC(F)C2)cn2c(n1)CCCC2 92195,CC1(C)C2CCC1(C)C2C(N1CCC(O)(CCNC(=O)C(F)=C2CCC2)CC1)=O 92196,CCC(F)(F)C(=O)NC1CCC(NC(=O)Cn2cc(C3CCOC3)cn2)C1 92197,c1(C(=O)NCC2(CNC(C(C(=C)Cl)(C)C)=O)CC23CCC3)nnn2c1CCCC2 92198,c1(C(N(C2CCN(C(=O)COc3cccnc3)C2)C)=O)cc(O)c(F)cc1N 92199,c1(CC(=O)NCC2CN(C(C(COC)C)=O)CC2C(F)(F)F)c(C)cccc1Cl 92200,C(CC1c2ccccc2CCN1C(c1cc(C)cs1)=O)NC(COCCSC)=O 92201,CN=c1ccc(C(=O)NCCC2CN(C(=O)CN(C)S(N)(=O)=O)C2)c[nH]1 92202,C(C(C)CC(F)(F)F)NC(CC(C1CC1)NC(c1ccc(C)[nH]1)=O)=O 92203,C(CCCC(=O)NCC(O)CCNC(=O)CSC1CC1)N(C(C)C)C 92204,N1(C(C(CSC)OC)=O)CCC(C(=O)NCC2CCSC2)=C(F)C1 92205,CCCC(C)(CC)C(=O)N1CCC(N2CCCN(C(=O)COC3CC3)CC2)CC1 92206,N1(C(C(N)CCc2ccccn2)=O)CC2CNC(=O)C2C1 92207,c1(C(N(C)CC2(NC(C(CCOC)C)=O)CC2)=O)ccc(Cl)c2occc12 92208,C(CO)(C(=O)NCC1CCC(NC(C2CCN2C2CCCC2)=O)C1)N(C)C 92209,C1(CC#C)CCN(C(c2cn(C(C)C)nc2Br)C(=O)NC2COC2)CC1 92210,c1(CCC(=O)NCC2C(NC(CC3C(C)(C)C3)=O)C2)c(F)cccc1F 92211,c1(OCC)ccc(C)c(NC(C2C=CCN(C(C3CCC3C(N)=O)=O)C2)=O)c1 92212,c1(C2(C(=O)NC(CNC(C(COCCOC)F)=O)C(C)C)CC2)ccnc(Cl)c1 92213,Cc1cccc2c1CC(C(=O)NCC1CC13CCN(C(=O)CC1CCC1)CC3)N2 92214,c1(SC(=O)NC(CC(=O)O)CC2CCCCC2)cc(O)nc(C2CC2)n1 92215,N1(C(C(C)=CC)=O)CC(C)OC2(CCN(C(=O)CCNS(=O)(=O)CC)C2)C1 92216,C1(CC(=O)N(C)CC23CC(CN2)C3)CC(=O)CC(C2CNC2)O1 92217,C1(CC)CN(C(C)=O)CCO1.C12CC(C1)NC(=O)C(OC)C1CN(C1)C2=O 92218,C1(C)(CC)CC(NC(C2(CO)COC2)=O)CN1C(c1cc(OC)cc(Cl)c1)=O 92219,C1(C)(NC(CCOCCN(C(c2c(C)cco2)=O)C)=O)CC(C)(C)OC1=O 92220,c1(CC)nnc(C)cc1C(N1CCC(O)(CCNC(=O)C(C)SC(C)C)C1)=O 92221,c1(C(=O)NC2CCCCN(C(c3cc(C)nnc3)=O)C2)ccc2c(C)[nH]nc2c1 92222,C(=O)(C(C(C)(C)OC)c1ccccc1)NC(CC)C(F)F 92223,CC(C)CC(O)C(C)C(=O)NCn1ccc(C(=O)NCCC2CC2)c1 92224,CCC(Cc1ccccc1)CC(=O)NC1CN(C(=O)CS(C)(=O)=O)C(C)(C)C1 92225,C1(NC(COCCC)=O)CC(NC(C2CC2[N+](=O)[O-])=O)C(O)C1 92226,C(=O)(C1=CCCOC1)NC(C(=O)NCc1c(C)scc1)CC1CCC1 92227,c1(OCC(=O)NCC(CNc2cc(SC)ncc2)(C)O)cc(C)cc(C)c1 92228,C(CCCC(C)NC(=O)C(C)Oc1ccccc1)NC(C1(COC)CCCC1)=O 92229,c1(OCC)ccc(C(=O)NC2CCC(NC(=O)CS(C)(=O)=O)CC2)cc1 92230,C(=O)(C1CCc2cccnc21)NCC1(C(C)(C)C)CCN(C(C=COCC)=O)C1 92231,c1(CNC(CC2(C)CCN2C(=O)CC2CCOC2=O)=O)cncc(O)c1 92232,C#CC1(C(=O)NCc2cccs2)CN(C(C2CCSC(C)C2)=O)C1 92233,C1(N(C(c2cnc(N(C)C)nc2)=O)C)CCN(C(C23CC(F)(C2)C3)=O)CC12CC2 92234,c1(NC(C(CC2CC2)NC(C2CC3C=CC2CC3)=O)=O)cncc([N+](=O)[O-])c1 92235,c1(CN(C)CC2C(N3CCN(C)CC3)CCC2)cnc2ccc(Cl)cn12 92236,Cc1csc2ccc(C(=O)NNc3ccnnc3)cc12 92237,c1(CNC(C2(OC)CCC2)=O)cc(C(N2CCC(OC(C)C)C2)=O)ccn1 92238,C1(N(C(CN2C(C)CC2)=O)C)CCCN(C(c2sccc2C(F)F)=O)CC1 92239,Cn1nc2c(c1C(=O)NC1CCN(C(C3CCC3F)=O)CC1)CS(=O)(=O)CC2 92240,C1(CNC(c2cc(F)cc(F)c2Br)=O)CCN(C(c2cn[nH]c2)=O)CC1(F)F 92241,N1(C(C(=C)C)=O)CC(=O)Nc2c(Br)cccc21 92242,N1(C(CC(C=C)CC)=O)CC2CCC1C(CNC(=O)C=Cc1csc(C)n1)C2 92243,CC1(CNC(C2(C#N)CC3CC3C2)=O)CCN(C(=O)COC(F)F)CC1 92244,N1(CCn2c(C)nc(=O)[nH]2)CC=C(c2ccc(Cl)c(Cl)c2)CC1 92245,N1(c2ccnc(N3CCCC(C(C)C)CC3)n2)CCc2nncn2CC1 92246,c1(C(=O)OCC)cn(C)nc1Cn1cc(CN(C)C(C2CC2(F)F)=O)nn1 92247,C1(C)(C(=O)NCC(CNC(C(CC)F)=O)O)CNC(=O)C1 92248,C1(O)(CN(C(=O)C=C2CCCC2)C)CCN(C(c2nnn(C)c2N)=O)CC1 92249,Cn1nnc2c1C(C(=O)NCC#CCNC(C1CCOCC1(C)C)=O)CCC2 92250,CC1(C)CCC(C(=O)Nc2ccn3nccc3c2)CN1C(=O)CCCCCF 92251,N1(CC(COCC(c2ccccc2)OC(C)=O)O)CCCC(NC(C)=O)C1 92252,N#Cc1ccc2c(c1)N(C(C1CCC(CNC(=O)CCC3CCCO3)CC1)=O)CC2 92253,c1(OCC)cccc(C(=O)N(CC)CC2(O)CCC(C)C2)c1OC 92254,N1(C(C(C(=O)OC)(C)C)=O)CC2CC(C1)CN(C(C13CC1COC3(C)C)=O)C2 92255,c1(CC)ncncc1C(N1CCCC1C(C)(C)NC(=O)C(C)Cn1ccnc1)=O 92256,c1(C(=O)NCCN(C(=O)CCCCC(N)=O)C(C)C)ccc2[nH]cc(C#N)c2c1 92257,c1(C(=O)N(C(C(C)NC(CN(CCCCCC)C)=O)C)CC)cnc(OC)nc1 92258,CC1(C(=O)NCCc2ccsc2)CCCN(C(c2c[nH]c(=N)o2)=O)C1 92259,N1(C(C(N2CC(C)C2)C)=O)CCN(C(c2ccncn2)=O)CC1c1nccn1C 92260,Cc1cc(CN2CCN(c3ccc(C4CC4)c(C)n3)CC2)ccc1F 92261,C1(C(N2CC(CC=C)(NC(c3c[nH]nc3SC)=O)C2)=O)CCOC1C=C 92262,N1(C(C2CCCO2)=O)CC2(C(=O)NC(CO)C(F)(F)F)CC1CO2 92263,C1(CC=C)(NC(=O)C(O)C=CCN(C)C)CCCN(C(=O)C=Cc2ccco2)C1 92264,C(=O)(C(O)CCCc1ccccc1)N1CC(C)C(NC(=O)CC(C)(C)C)C1 92265,C(=O)(CCCS(C)(=O)=O)NCC1(CNC(C(C)Cc2cnco2)=O)CC12CCC2 92266,C=CC(C)(C)CC(=O)N1CC(C(=O)NCCNC(C2CCC(C)S2)=O)C1 92267,C(C)(C)(CC(F)C(=O)N(C)CC1COC(=O)N1)NC(c1c(C)c[nH]n1)=O 92268,C(=O)(C(C)(C)C(C)O)N(CC=CC(N1CCC(C)(NC(C)=O)C1)=O)C 92269,C(N=c1nnc(C)c(C)[nH]1)C1(C)CCN(C(c2ccc(C(C)=O)[nH]2)=O)C1.C1CC1 92270,c1(OC)cc(F)c(Cl)cc1C(=O)NC1CN(C(C2CCCC(=O)O2)=O)CCC1O 92271,c1(C(=O)NC(CC=CC)C(=O)Nc2cncnc2OC)c[nH]c(=N)c(C)c1 92272,N1(c2cc(NCc3n(C(C)C)cnc3)ncn2)CCCOC(C(C)C)C1 92273,CC(C)C(C(=O)NC1CC(C)(C)C12CC2)C(C)NC(=O)CCCn1ccnc1 92274,C1(C(=O)Nc2cn(CC=C)nc2)CC(C)CN(C(=O)CCn2cnnc2)C1 92275,N(C(=NCC1CC(OC)(CC)C1)NC1CCCC(c2ccc(F)cc2)C1)CC=C 92276,c1(CCC(=O)NCC2OCC(CNC(c3c(C)ccs3)=O)C2)ccccc1Cl 92277,c1(C(=O)NC2(CC)CCN(C(C3CCCC(O)C3)=O)CC2)cc(C#N)ccc1N 92278,C1(C(N(C2CCN(C(CCC#CC)=O)C2)C)=O)CC2(CCCC2)C1 92279,c1(OCC(=O)NC(CN(C(c2c(C(C)C)nco2)=O)C)C)ccccc1C#N 92280,Cc1cccc(NC(N2C(C(N3CCC(C)(C(N)=O)C3)=O)CC3CC23)=O)c1 92281,C1(C(N2CC3C(CC(=O)NCc4nc(C)c(C)s4)C3C2)=O)CC2(CCC2)CO1 92282,C1(CNC(C(CC)NC(C)=O)=O)CN(C(=O)C(F)(F)COC)CC1C 92283,C(C(O)C(C)(C)C)N(C(C(C)N(C(Cc1c(C)ocn1)=O)C)=O)C 92284,N1(CCN(C(CNS(CC)(=O)=O)=O)CCO)CCOCC1 92285,C=C(C)CCNC(=O)NCC(C)NC 92286,CC1CCn2ncc(C(=O)NC(CNC(c3ccncc3O)=O)C(C)(C)C)c2C1 92287,Fc1cc(Cl)cc(Br)c1N(c1ncc2cn[nH]c2n1)N1CC1.C1(C)CNC1 92288,C1(CC(N2CC(NC(c3coc(C4CCC4)n3)=O)C(O)C2)=O)CC2(CCC2)CO1 92289,c1(CC)cc(C(=O)NCC(O)CCNC(C2CCSC2)=O)cc(C)c1 92290,C(=O)(CC1=CCCCC1)NC1C(C)(CNC(CC2(OCC)CCC2)=O)CCC1 92291,C1(OCC)CC2(CCCN(c3nc(N4CC5CCC4CC5)c4ccsc4n3)C2)C1 92292,C#Cc1cc(C(=O)NCC2(C)CCCN2C(=O)CCC2CC2(C)C)ccc1Cl 92293,C1(CCCNC(C(C2CC(C)(C)C2)OC)=O)CCCCN1C(=O)C=CCO 92294,C12(C(N3CCC(N(C)C(c4nn(C)nc4C(F)(F)F)=O)C3)=O)CNCC1COC2 92295,c1(-n2cc(C34N(C(=O)C(F)F)CC(C3)C4)nn2)ccc([N+](=O)[O-])cc1F 92296,c1(C(N(CCCCN(C(=O)C(O)C2CCCC2)C)C)=O)c[nH]c(C#N)c1 92297,N1(C(C=CC(C)(C)C)=O)CCc2c(CNC(=O)CC34CCCC3C4)cccc2C1 92298,C(=O)(C(CN(C)C)CC)NCc1c(C(=O)NC(C(=O)OCC)C)[nH]cc1 92299,C(=O)(C(C)S(C)(=O)=O)NCc1c(C(=O)NC(c2nccs2)C)n[nH]c1 92300,N1(C(C2(OC)CC2)=O)CCCC2(CC(NC(=O)C=C3CCC(C)CC3)CO2)C1 92301,C1(C)(CNC2(n3cccn3)CCN(OC)CC2)CN(C(=O)OC(C)(C)C)CCO1 92302,Cc1nc(O)nc(C)c1C(=O)NCC(C)(O)CNC(=O)Cn1cc(C(C)O)nn1 92303,CC(C)CC(F)C(=O)NCCC1CCCCN1C(c1ccnn1C(C)C)=O 92304,c1(CCNC(=O)COCCNC(C2CCCS2)=O)ccncn1 92305,N1(C(C=CC=CC)=O)CC(N(C(=O)C(C)SC(C)C)C)CC1(C)C 92306,C#CC1(O)CN(C(=O)CSCCNC(C2(CF)CC2)=O)C1 92307,CC#CCCC(=O)N1CC(OCC)C(NC(=O)CCCN(C)C(C)C)C1 92308,C1(O)(CN(C(=O)CCC2CCC(=O)N2)C)CN(C(=O)CCc2cn[nH]c2)C1 92309,c1(SCC)ccc(C(=O)NC(C)(C)CCCNC(=O)Cn2cc(C#N)cn2)cn1 92310,C1(CC(=O)NCC(C)(CO)NC(C(C)=C2CCC2)=O)COC(C)(C)C1 92311,N1(C(CNC(C(C)(C)C)=O)=O)CCOC(C)(CNC(C2CC2(Cl)Cl)=O)C1 92312,C1(NC(C(COC)(F)F)=O)COC2(CNC(=O)COC(C)=O)CC1C2 92313,C#CCC(CC(F)F)C(=O)N1CCCC1CCC(=O)Nc1ccc(C)cc1CO 92314,CCC(CC)CC(F)C(=O)N1CCC2(CC1)CC2C(N1CCC1C1CCC1)=O 92315,N1(C(c2ccc(CC)cn2)=O)CC2(C)CC1(C(N1CC3CCC3(CO)C1)=O)C2 92316,c1(C(=O)NCC(C)NC(CC2CC(OC)C2)=O)ccc(N2CCCC(O)C2)cc1 92317,C(C1=CCN(Cc2cc(Cl)ccc2Br)CC1)NC(c1cccc(F)c1Cl)=O 92318,C1(NC2CC2)CC(C(=O)NC2C(c3n(C)ccn3)C2)C1(C)C 92319,N1(C(C(C)OCC=C)=O)CC(C(N2CCCC(C(C)(C)O)C2)=O)C(C)(C)C1 92320,N1(C(C2(N(C(c3n(C(C)C)ccn3)=O)C3CC3)CCC2)=O)CC2(CC(CO)CO2)C1 92321,C=CCCCCCCC(=O)N1CCN(C)C(CNC(=O)CC2CC(OC)C2)C1 92322,c1(OC)c(NC(=O)C(=O)NC2CNCCOC2)cc(F)cc1Br 92323,C1(S(C)(=O)=O)(C(=O)NC(C)CC(C)NC(c2ccncc2F)=O)CCC1 92324,c1(C(C(=O)NCC(CNC(=O)C=CCOC)OC)O)cc(F)c(F)cc1F 92325,C(=O)(CC(C)C(=O)NC1(C)CN(C(=O)CCn2cc(Cl)cn2)C1)OC 92326,Cc1nc(CO)ncc1C(=O)NCC1(C)CC(NC(C2(n3ccnn3)CC2)=O)C1 92327,N1(C(C2CC=C(C)CC2)=O)CCCC2CN(C(=O)CC3CC=CCC3)CC12 92328,N1(C(C(=O)N(C)C)=O)CCN(C(c2cccc3c2NCC3)=O)C2CCCCC12 92329,Cc1ccc(CC(N2CC(CNC(=O)CNS(N)(=O)=O)C(O)C2)=O)c(F)c1 92330,CCC(CCC(=O)N1CC(n2cccn2)C1)NC(=O)CC(C)C1CC1 92331,CC1CCN(C(=O)C(=O)NCC(F)F)C1CNC(c1c(Br)ncn1C)=O 92332,C(=O)(C(C)S(=O)(=O)C(C)C)NC(CC(C)C)CNC(=O)CCc1cnn[nH]1 92333,N1(C(C(C)=CC)=O)CC(CNC(=O)CC(CC)CCC)OC2(CCC2)C1 92334,c1(N(C)Cc2ccccc2[N+](=O)[O-])ccc(S(=O)(=O)NCC2CCCCS2)cn1 92335,C(CCCC(=O)N(C)Cc1nnnn1C)NC(C1C(CC)OCC1)=O 92336,C1(CC(=O)N(C2CCN(C(=O)COCCF)CC2)C)COC(C)(C)CO1 92337,N1(C(C=CC(=O)N(C)C)=O)CCOC2c3ccccc3OCC12 92338,C1(NC(C=C(C)C(F)F)=O)CCCN(C(C2CCC2(F)F)=O)CC1 92339,O1NC(=O)C(F)C2(O)CN(C(=O)C1(C)C)C2.c1(OC)ccc(=N)[nH]n1 92340,CC1CN(C(C2CCCN2c2cnccn2)=O)CCN1C(=O)C=CBr 92341,N1(CC2CCCC(C(=O)OC)C2)C(=O)NC(Cc2cc(C)cc(C)c2)C1=O 92342,C1(CC(=O)N(C)CC2N(C(C3CC(OCC)C3)=O)CCOC2)COCC(C)(C)O1 92343,N1(C(COCCCC)=O)CCN(C(C2(C)CCC(OC)C2)=O)CC12CCC2 92344,C1(OCCC)(OC)CCN(Cc2cccc(C(F)(F)F)c2)C1 92345,C1(CCNC(C(C)CC2CCC2)=O)CCCN(C(c2c(C(F)F)cnn2C)=O)C1 92346,C1(CNC(C2C(C=C)C2)=O)COCCN1C(=O)CC1CCSCC1 92347,c1(C(N2CC(C)N(C(=O)Cc3c(Cl)cnn3C)CC2)=O)cnn2c1N(C)CC2 92348,O=C(C=CCCc1ccccc1)NNc1ccc(Cl)cn1 92349,C1(NC(C=CC=CC)=O)CC2COCC(C1)C2NC(=O)CC1CCS(=O)(=O)C1 92350,C1(C(N2CCN(CCNC(=O)CC3=CCCC3)CC2)=O)CC2CCCCN2C1 92351,c1(C(=O)N(C2CC(C(=O)NOC3CCCCC3)C2)CCO)c[nH]c2cccnc12 92352,Cc1nc(O)sc1C(=O)N(CC(=O)N(CCCC(C)O)C)C(C)C 92353,C1(CC)CCN(C(C2CSCCS2)=O)C1CNC(=O)C(CCSCOC)N(C)C 92354,C1(CNC(C(c2cccc(O)c2)C)=O)CCN(C(=O)C=CC2CCCC2)CC1 92355,CCC(C)(CC)C(=O)NC(C1CCN(C(=O)C(C)Oc2cccnc2)C1)C 92356,c1(C(=O)NC(CN(C(c2cc(CN(C)C)c[nH]2)=O)CC)C)c(Cl)cnn1C 92357,c1(CCC(=O)NCC(F)CNC(C2(C(F)F)CC2)=O)ccc(F)c(Br)c1 92358,c1(C(C)C(=O)NC(C2(O)CN(C(c3ncccc3Cl)=O)C2)C)c(F)cccc1F 92359,C(=O)(C#CC1CC1)N1CCC(C(C)C(=O)NCC#CC(F)(F)F)C1 92360,c1(C(=O)OC)coc(C=CC(=O)NCC(C)N(C(=O)Cc2ccon2)C)c1 92361,N1(C(c2scc(C(C)=O)c2)=O)CCN(C(C2CC2(F)Cl)=O)CC(C)(C)C1 92362,c1(C(=O)NC23CC(NC(C4(C)CNC(=O)C4)=O)(C2)C3)ccc2nc(CO)[nH]c2c1 92363,C1(C(=O)NCC(=O)N(C(c2ccncc2)C)CC)CCC(OC)CC1 92364,Cc1ncnc(C(=O)NC2CCCC2C(=O)NCC2(F)CCOC2)c1C 92365,c1(OC)n[nH]c(C(=O)NC2(CNC(=O)CC3(O)CCCOC3)CCCC2)c1Cl 92366,N1(CCN=C(NCC(CC)CO)NC2CCC2)CCc2ccccc21 92367,C1(CNC(C(C=C)O)=O)CC(F)CN1C(C1CCC(C(C)(C)C)O1)=O 92368,C(=O)(CC1=CCN(C(c2c(F)cccc2F)=O)CC1)Nc1ccc(C)nc1C 92369,c1(C(N2CC=CC(NC(C3(CC=C)CCOCC3)=O)C2)=O)onc2ccccc12 92370,c1(C(C)N(C(=O)C(C)(C2CC2)N(C(=O)CN(C)C)C)C)ccccn1 92371,N1(C(C(n2cnc(C#N)n2)CC)=O)CC(CNC(=O)CCCF)C(C(F)(F)F)C1 92372,C(=O)(CCCCC(C)CC)NC(CCCC)CNC(c1ncoc1C(F)(F)F)=O 92373,C1(NC(CCCN(C)C)=O)CCC2CN(C(c3nc(Cl)cs3)=O)CC2C1 92374,C(CC(F)CN=[N+]=[N-])NC(c1cc(CNC(C(C)NC(CC)=O)=O)ncc1)=O 92375,Cc1nn(CC(N2CC3CCC3(CNC(c3cc[nH]n3)=O)C2)=O)c(C)c1C 92376,C1(C(N(C(CC)C2CC2)C)=O)COCCC1NC(c1cc(C)sn1)=O 92377,c1(N(C)Cc2cnn(CC)c2C)ncnc(NC2CC3CC(O)C2C3)c1C 92378,c1(C(=O)NC2CC3(C(NC(=O)CC4CCCS4(=O)=O)C3)C2)nc2cnccc2s1 92379,Cc1ccc(Cl)cc1NC(=O)CCCCCN(C(=O)Cn1cc(CO)nn1)C 92380,CCCC(CCCNC(=O)CSCCC(C)C)NC(c1coc(CC)n1)=O 92381,c1(OC)ccc(C(N2CC(CNC(=O)CC3CCOCC3)CC2(C)C)=O)c(F)c1 92382,CCC(O)CC(=O)NCCC1(CNC(=O)CCc2nc(-c3ccco3)no2)CC1 92383,CC1(C)CC(NC(C2(C)CCCC2(F)F)=O)CCN(C(c2cc(N)ccn2)=O)C1 92384,C1(CNC(C(N2CCOCC2)C)=O)CCN(C(C2CNC(=O)C2)=O)CC1 92385,c1(NC(CC)CNC(C23CC4CC(C(=O)N2)C3C4)=O)ncnc2c1nnn2C 92386,Cc1c[nH]c(C(=O)N(C)CC2(CNC(c3ccoc3C3CC3)=O)CC2)cc1=O 92387,C(CCC(C)C)(C(=O)NCCOCCN(C)C)NC(C(CC)n1cncn1)=O 92388,c1(C(N2C(C(=O)Nc3c(C(=O)OC)sc(Br)c3)CC3CC32)=O)cncc(Br)c1C 92389,C1(C(N(CC(=O)N(C)C)CCC)=O)CCCN(C(=O)C2=C(Cl)CC2)C1 92390,c1(C(=O)NCC2CC(NC(C(c3n(C)ncc3)O)=O)C2)ccc2c(c1)COC2 92391,c1(C(=O)NC(C2(C(=O)NC3CCCC3(F)F)CC2)C)ccc([N+](=O)[O-])o1 92392,C=CC1CN(C(c2ccns2)=O)CC1NC(c1ccc(C(C)C)c(F)c1)=O 92393,c1(C(=O)NC(C(C)NC(Cc2ccc(OC)cc2)=O)C(C)C)c(F)cccc1F 92394,C1(CCC(=O)NC)CCCN1C(=O)N(C)CCO 92395,c1(C(C)CN2CCN(C3(N)CCCC3)CC2)ccc(Cl)cc1 92396,CCC(CC(=O)N1CCC1CNC(C1(OC)CC1)=O)c1ccccc1 92397,C1(O)(C(=O)NC(C2CC=CCC2)C)CCN(C(c2cc[nH]c2)=O)C1 92398,c1(NC(C2CCCC2Cc2cnn(-c3ccccc3)c2)=O)cccc(Br)c1I 92399,c1(C(=O)NCC(C)(O)CNC(C2CC2(Cl)Cl)=O)cn2ccccc2n1 92400,c1(NC(C)CN(C(C(C(C)C)SC)=O)C)c(F)cccc1[N+](=O)[O-] 92401,c1(C(=O)NCC(C2CCCCC2)NC(C(C)N(CC)CC)=O)ncc(Cl)cc1Cl 92402,c1(OC)ccc(Cl)c(F)c1C(=O)NCCCCNC(C1CC1c1ccoc1)=O 92403,c1(OC)ccnc(NCC(=O)NCC(C)CNC(C2(C)CCCC2C)=O)n1 92404,C1(C(F)F)(OC)CCCN(C(c2nc(Br)cn2C)C(=O)NC(C)(C)C)C1 92405,N1(C(C(C(C)C)C)=O)CCn2ncc(CNC(C3C4CCOCC34)=O)c2C1 92406,Cc1c(C(=O)NCCC(C)(C)NC(=O)C(C)C2CCCO2)cccc1C#N 92407,C1(NC(c2ccc(C)cc2F)=O)CN(C(C2COC(C)(C)CO2)=O)C2CCCC12 92408,c1(C(=O)NC(CN(C(CCC(CCCC)C)=O)C)C)cc(F)c2nc(C)cn2c1 92409,CCCCC(O)C(=O)NCC1(C)CCN(C(c2cccnc2OC)=O)C1 92410,c1(C(CCC(=O)OC(c2ccc(Cl)cc2)c2ccccc2)=O)ccc(F)cc1F 92411,C(CO)(CC(C)(C)C)NC(C1C(CNC(Cc2nc(C)[nH]n2)=O)C1(C)C)=O 92412,C1(NC(c2cnc(CC)[nH]2)=O)C2CC(NC(C3CC3(F)Cl)=O)CC12 92413,C(C(CNC(C1CCS(=O)(=O)C1)=O)S(C)(=O)=O)NC(C1(CC#C)CC1)=O 92414,c1(C(=O)NC2CCN(C(C(C)NS(C)(=O)=O)=O)C2)cc(Cl)c(Cl)[nH]c1=N 92415,C=C=CCC(=O)N1CCC(C(C)(C)NC(c2cc(C(C)CC)no2)=O)C1 92416,C(C(CC(=O)N1CCC(CO)(NC(=O)C2=CCOC2)C1)C(F)(F)F)N(C)C 92417,N1(C(c2coc(C3CCC3)n2)=O)CCN(C(=O)C(F)(F)C(F)(F)F)CC2(CC2)C1 92418,CC(C)CCC(=O)C(=O)N1CC(C)(OCC(=O)NCC2(CO)CCOC2)C1 92419,C1(O)(CNC(c2cn(CCNC(CCC=C(C)C)=O)nn2)=O)CCC(C)C1 92420,C#CCC(C)C(=O)NCC(C)N(C(c1ccc(-c2cn[nH]c2)cc1)=O)CC 92421,c1(OCCCC(=O)NC(CNC(C(C)OCOC)=O)(C)CO)ccccc1Cl 92422,CC(CC(=O)N1CCC(O)(CNC(=O)CC2CN(C)C2)C1)C(F)(F)F 92423,c1(CC)cc(C(N2CC(CNC(c3cccc(F)c3F)=O)C(O)C2)=O)ccc1F 92424,C(C1CCCO1)=CC(=O)NCCC(C)N(C(=O)CCC1CCC1)C 92425,C(=O)(CCCN=[N+]=[N-])NCCCCC(C)NC(C1(CCOC)CC1)=O 92426,CCC(C(=O)NCCCCC1(NC(=O)Cc2csc(Cl)n2)CC1)C(F)(F)F 92427,CC(C)(C#N)CCCC(=O)NCC1C(CNC(c2c(F)cccc2F)=O)C1(F)F 92428,C1(NC(C2(C(F)(F)F)CCCC2)=O)CC2CN(C(c3csc(C(F)F)n3)=O)CC12 92429,C12(NC(=O)N(CCS(C)(=O)=O)C(C)C)CCC1CN(C(=O)OCC(C)(C)C)C2 92430,N1(C(COC2(C#C)COC2)=O)CCCC(C)(CNC(=O)C(=O)NC)C1 92431,C1(CNC(c2n(CC=C)ccc2)=O)C(C)CCCN1C(c1cc([N+](=O)[O-])n[nH]1)=O 92432,Cc1cc(C(N2CCC2C(=O)N(CC(F)F)C)=O)oc1C 92433,N1(C(C2CC(C)N2C(C2CC3CCC(C2)O3)=O)=O)CCc2ccccc21 92434,N1(C(c2cc(OCC)n[nH]2)=O)CCC2(CCCN2C(=O)CC2CCCCC2O)C1 92435,c1(C(N2CCC(C(CO)NC(c3c(C)onc3)=O)CC2)=O)ccc2nonc2c1 92436,C1(NC(C2(COC)CCC2)=O)CN(C(=O)COc2cccc(F)c2)CC2(CC2)C1 92437,C1(C(=O)OC)CCS(=O)(=O)C12CN(C(=O)C(=O)NC1CCN(CC(F)F)CC1)C2 92438,c1(C(N2CCCC(N3CCCC3=O)C2)C(=O)NCC(C)C)cnn(C(C)C)c1I 92439,C1(C(=O)NC(c2ccc(C)nc2)C)CCN(C(c2ccccc2F)=O)C(C)(C)C1 92440,C(=O)(C1=CCc2ccccc21)NC(C)CC(C)NC(c1cnc(Cl)n1C)=O 92441,c1(C(C(=O)NC2(CC(=O)NC(c3cccs3)CO)CC2)O)cccnc1 92442,C1(NC(CCC(N)=O)=O)CCC2CCN(C(=O)C(C3CC(F)(F)C3)O)C1C2 92443,N1(C(C(CC(C)C)=O)=O)CCC2CN(C(C3(C4CC4)CCC3)=O)CC2CC1 92444,n1(CCCOCC)cc(C)c(=NC(=O)c2cn(C(F)(F)CO)nn2)[nH]1 92445,N1(C(C(c2ccccc2)OC)=O)CCCOC(CNC(C2(SC)CC2)=O)C1 92446,c1(C(=O)NCCCN(C(C2CC(C)(F)C2)=O)CC)cc2n(n1)CCCNC2=O 92447,n12cc(nn1)C(=O)N(CCCC=C)CC(=O)NCC2.C(C)(C)(C)NC(N)=O 92448,N1(C(C2C(C)(C)CO2)=O)C2CCC1CN(C(C1CC3C=CC1C3)=O)C2 92449,C1(N(C(C(CCC)CC)=O)C)CC2CCC(C1)N2C(=O)C(F)(F)C(O)CC 92450,c1(N(CCC)CCNC(C2(C#N)CCC2)=O)cc(N2CCNC2=O)c(F)cc1F 92451,c1(C(=O)NCC2CCC(CNC(C(C)OC)=O)CC2)ccc(N)c(F)c1Br 92452,C1(O)(C(N(CCNC(=O)Cn2ccc(C3CC3)n2)CC)=O)CCC(C)(C)CC1 92453,Cc1ncc(CC(=O)N(C2CCCC2)CCNC(=O)C=CC2CCCO2)[nH]1 92454,N1(C(CC(CC)C(C)C)=O)CC2CCN(C(=O)C(C)OCC3CCCC3)C2C1C 92455,c1(C(C(N2C(C)(CNC(C(C3CC3)OCC)=O)CCC2)=O)=O)ccc(Cl)cc1O 92456,c1(C(N2CCN(C(c3cccc(F)c3)=O)CC2)=O)coc2c1C(O)CCC2 92457,c1(CC(N2CCN(C(C(C)(C)C#N)=O)CC2)=O)cc(F)cc([N+](=O)[O-])c1 92458,CC1CN(C(=O)Cc2cc(O)nc(O)n2)CCN1C(c1coc(Cl)c1)=O 92459,c1(C(=O)NC2CCN(C(CNC(=O)NC)=O)C(C)C2)cnc2[nH]c(C)nc2c1 92460,c1(C(=O)NCC2CN(C(CC3(C=C)CC3)=O)CC2O)nc2n(c1Cl)CCCC2 92461,c1(C(=O)NCC2(NC(c3ccsc3)=O)CC2)cccnc1-n1ccnc1 92462,N1(C(CCOC(C)C)=O)CCCC2(C1)C(NC(c1cc(F)n[nH]1)=O)CCN2C 92463,c1(C(=O)NCC(CC)(C)NC(c2csc(COC)c2)=O)nc(O)sc1C 92464,N1(C(COCCC#C)=O)CCCC(CNC(C2(CC(=O)NC)CC2)=O)C1 92465,c1(C(N2CCN(C(C3CC34CCC4)=O)CC2CCO)=O)ccc([N+](=O)[O-])c(Cl)c1 92466,C1(C(=O)NC(CC)(C)C(F)(F)F)CCN(C(=O)CN(C)C2CC2)C12CCC2 92467,C1(C(=O)NC2C(CNC(CNS(NC)(=O)=O)=O)CCC2)COC(C)(C)CO1 92468,Cc1cccn2c(CC(=O)NC(C)C(=O)NC(c3ccccc3)C(=O)O)cnc12 92469,c1(NC)cc(Cl)ccc1C(N1CCC(CO)C(NC(C2(C)CCCCO2)=O)C1)=O 92470,CCCCCC(C)NC(=O)C(c1cnn(C)c1)NC(c1ccc(F)s1)=O 92471,C1(C(=O)NCC(C)(C)NC(CCCC#C)=O)CSC(Cc2ccccc2)C(=O)N1 92472,CCC(=O)CCC(=O)N1CCCN(CCNC(=O)C(F)C2CCOC2)CC1 92473,N1(CCN(C)C)CCN(C(c2ccc3c(c2)CC3)C(=O)NCCC2CC2)CC1=O 92474,c1(C(=O)NCCC2CC(C(=O)NCC3(C)CCCO3)C2)cnn2c1OCC2 92475,C1(CC(=O)NCC2CCN2C(=O)C=CCOc2ccccc2)CCCCC1(F)F 92476,Cc1cc(C(=O)NC2CCC2CNC(=O)Cn2ccc(C3CC3)n2)ccn1 92477,c1(C(N(C)CC2N(C(c3c(C)nns3)=O)CCC2)=O)cnc2nc(O)ccc2c1 92478,N1(C(CC2CCC(C)C2)=O)CC23CCCC2(C1)CN(C(c1coc(CO)c1)=O)C3 92479,c1(C(C(N2C(C(=O)OCc3ccccc3)CSC2)=O)O)cc(F)c(F)cc1F 92480,C1(C(=O)NCc2ccn(C(C)C)n2)CCCC(NC(c2c[nH][nH]c2=N)=O)C1 92481,c1(CCNC(C(C2(C)CC2)NC(C(C)=CCC)=O)=O)ccn(C)n1 92482,CN1CCN(C(=O)C(C)(C)c2cnsc2)CC1CNC(C1(C)CC=CCO1)=O 92483,c1(CNC(C(=O)NCc2ccc(SC)cc2)=O)ccc2c(c1)CCO2 92484,Cc1cc(C(=O)NCCC2CC(NC(=O)Cc3ccsn3)C2)n2nc(C)cc2n1 92485,N1(C(CC2CC(=O)C2)=O)CC(NC(=O)C=CC2CCC2)C2CC12 92486,CC1(C#CC(=O)NC2CN(C(=O)C3=CCCCC3)CC23CC3)CC1 92487,Cc1onc(CC(=O)NC2CCC(CNC(C3CCCC(O)C3)=O)CC2)c1C#N 92488,CN1CCC(CN(C)C(C2CC(NC(C3(C)CC3)=O)C2)=O)CC1 92489,N1(CC(N2CCCCC2C(=O)NOC(C)C)=O)CCCC(O)(CO)C1.Cc1cc(O)no1 92490,C1(NC(Cn2c(C)ncc2)=O)CN(C(C2(Cl)CC2(C)C)=O)CC(C)(C)C1 92491,C(F)(F)(C(=O)NNC(=O)COc1cccc(C)c1)C1(CC)CCC1 92492,N1(C(c2cc(C(F)(F)F)cc(Br)c2)C(=O)NC(C)C)CCCC2CC(C)CCC12 92493,N1(C(C(C)(C)C2CC2)=O)CC2(C=C(C(=O)NOCCCCN3CCCC3)CO2)C1 92494,C1(NC(C(C)CCC)c2n(CCC)nnn2)CCC2(CCCCC2)CC1 92495,c1(C(=O)NC(CC)CN(C)C(c2cc(-c3ccoc3)[nH]n2)=O)cc(C)nc(N)c1 92496,C1(CNC(c2ccc(Cn3cc(C)nn3)o2)=O)CCCOCC1.C1(SC)CCOC1 92497,C1(CNC(C2(C)CCN(C)C2)=O)CC2(CC(NC(=O)CC3CC4(CCC4)C3)C2)C1 92498,C1(SC)CN(C(=O)CSc2nncs2)CC1NC(C1CC(C)C1)=O 92499,C1(NC(C=Cc2ncc(C)[nH]2)=O)CN(C(=O)C(C2CC2)C2CC2)CC1C1CC1 92500,N1(C(C23CN(C(CCC)=O)C(C2)CO3)=O)C2CCC1CC(CO)C2 92501,c1(N(C(CCNC(C2(OC)CCS(=O)(=O)C2)=O)C)C)ccc([N+](=O)[O-])cc1Cl 92502,N=c1nc2c(c[nH]1)CC(C(=O)NCCCCNC(=O)CC13CCCC1C3)CC2 92503,C1(CC(=O)NCC(C2CC2)NC(c2cncc(C=C)c2)=O)CCC2(CCC2)CO1 92504,C1(C(N(CC(CNC(CCC#C)=O)O)C)=O)CC(c2cn(C)nc2C)=NO1 92505,C1(NC(C(N2C(CC)CCC2)=O)=O)CCCCN(C(=O)CSc2ccccn2)C1 92506,CC1(C)NC(=O)N(CC(=O)NC2CC(NC(=O)C(CO)NC(N)=O)C2)C1=O 92507,C1(CNC(=O)Nc2nnc(-c3ccccn3)s2)CCCN2CCCC12 92508,c1(C(N(C)CC2CN(C(C34CC(F)(C3)C4)=O)C2)=O)cc2n(n1)CCNS2(=O)=O 92509,c1(C(N2CCC(C)(NC(C(CC(C)C)NC(N)=O)=O)C2)=O)cnn2c1NCCC2 92510,C1(NC(Cc2c(C)con2)=O)CCCCN(C(=O)C(F)C(C)(F)F)C1 92511,c1(C(=O)OCC)cnn(C)c1S(=O)(=O)NCC1OC(=O)CC1(C)C 92512,Cn1ncc(Cl)c1NC(C1(C(C)(C)C)CCN(C(C2CSC2)=O)C1)=O 92513,N#Cc1c(NC(C2CC2C(=O)NCCNc2ccc(Br)o2)=O)cccc1F 92514,C1(NC(c2c(C)nn(C)c2C)=O)CCC2CN(C(=O)CCCN(C)C)CC2C1 92515,C#CC1(C(=O)NC(c2ccc(O)nc2)C)CCN(C(C2C=C(C)CS2)=O)C1 92516,C1(CC)C(NC(c2ncc(F)cc2N)=O)CCCN1C(=O)C(CSC)OC 92517,C(C(C(=O)NCc1conc1C1CC1)NC(=O)CN1CCC(C)C1)SCC 92518,Cc1cc(F)cnc1C(=O)NC(CC1CC1)C(=O)NCC1CC2(CCC2O)C1 92519,N1(C(C=C(C)C)=O)CCC(N(CCO)C(c2cnco2)=O)C1 92520,C1(OC)CN(C(=O)COC2(C)CCCC2)CC1CNC(C1CCCN1N=O)=O 92521,C(N=c1cc(C)nc(C)[nH]1)C1CN(C(c2cc(C)ncc2)=O)C(C)C1 92522,C1(C(N2CC(CC)(NC(=O)Cc3cccnc3O)C2)=O)CCC2CC1C2(C)C 92523,C(CC1CCc2ccccc21)NC(N1CCCC1Cc1cc(F)ccc1Cl)=O 92524,C1(NC(C2N(C(CCC)=O)CCCC2)=O)CCN(C(=O)CCCC(F)F)C1(C)C 92525,c1(C(N(CCCNC(=O)CC(C)(C)F)C(C)C)=O)cc(Cl)cc(F)c1N 92526,N(C(=NCc1ccsc1)NC1CCOCC1)CC(C)(C)N(C)C 92527,C=C=CC(C)C(=O)NCCN(C(=O)C(C)CC=C)C1CCCCCC1 92528,c1(C(=O)NCc2cn(CCOC(C)=O)nn2)ccc(-n2cc(Br)cn2)cc1 92529,C=CCC(CC)C(=O)N1CC(NC(=O)CCSCC(C)C)CC1(C)C 92530,c1(C(=O)NCC(C)NC(C2CC2(F)F)=O)ccc2c(c1)B(O)OC2 92531,c1(C(=O)NC(CC(C)C)CNC(c2ccn(C)c2)=O)cc2ccc(Cl)c(F)c2[nH]1 92532,N1(C(C(C2CCCO2)OC)=O)CC2(CCN(C(c3cc(N)c(F)cc3C)=O)C2)C1 92533,N1(C(CCc2ccn(C)c2)=O)CCN(C(=O)CNS(=O)(=O)N(C)C)C(CCO)C1 92534,c1(C(=O)NC2CC(NCc3ccc(C(=O)OC)[nH]3)C2)nccn2nccc12 92535,C(=O)(CC1OCCc2ccccc21)N1CCC(C)(NC(=O)CC2(O)CCC2)CC1 92536,C(=O)(C(COC(C)=O)C(F)(F)F)NC12CCC(NC(C(CCCC)C)=O)(CC1)C2 92537,Cn1ncc(C(=O)NC2CCN(C(=O)CC3CC(C)(C)C3)C2)c1-c1ccccc1 92538,N1(C(CC2(NC(C3C4CCCCC34)=O)CC2)=O)CCC2(CCO2)C1 92539,c1(CC)ccc([N+](=O)[O-])cc1C(=O)NC1CCN(C(C2CSCC(=O)N2)=O)CC1 92540,CC(CC(=O)NC1(C)CCN(C(c2ncccc2O)=O)C1)C(F)(F)C(F)(F)F 92541,N1(C(C2CN(CC)C(=O)C2)=O)CC2(CCN(C(c3ccc(Cl)o3)=O)CC2)C1 92542,N1(Cc2ccc(C#C)s2)CC2(CN(C(=O)Nc3ccccc3F)CCO2)C1 92543,c1(OCC(=O)NC2C(NC(c3c(Br)ccc(C)c3)=O)C2)ccc([N+](=O)[O-])cc1 92544,c1(C(N2C(C)C(C)N(C(c3cncnc3)=O)CC2)=O)ccc(S(=O)(=O)CF)cc1 92545,CC1C2CC(C2NC(C2C3CC4C(C3)C24)=O)N1Cc1ccccc1 92546,C1(CN(C(c2c(C)cns2)=O)C)CN(C(=O)CCc2cccc(O)n2)CCO1 92547,c1(OCC)cc(F)c(C(=O)NCCC2CN(C(=O)C=CC3CCOC3)C2)c(F)c1 92548,c1(SCC(=O)NCC(C)N(C(=O)CCN(C)C2CC2)CC)ccc(F)cc1 92549,N1(C(=O)Cc2cncnc2)CCOC2(C1)CN(C(c1cc3c(s1)COCC3)=O)C2 92550,C(=O)(C1CNCc2n[nH]cc21)NCC1CCC2(CC(N(C)C)C2)CC1 92551,C(=O)(CC(C)(O)C(F)(F)F)N1CCN(C(CSCC#C)=O)CC1CO 92552,N1(c2nnc(C)s2)CC2(COC(CNC(C3CC(c4ccccc4)C3)=O)C2)C1 92553,C1(NC(c2ccccc2)CC)CCN(C(C2CC23CCC3)=O)CC1C 92554,C1(c2ccccc2)(CNC(COC(C)=O)=O)CCN(C(=O)CC2(C)CC2F)CC1 92555,c1(CCC)cc(C(N2CC(N(C(=O)CSc3nccn3C)C)C2)=O)n(C)n1 92556,c1(CNC(CN(C2CC(C#N)C2)C(C=C(C)C(F)F)=O)=O)csnc1C 92557,c1(OC)cc(Cl)ncc1NC(C1CC1C(=O)NC(c1ccc(C#N)cc1)CO)=O 92558,N1(C(C=Cc2c(C)ccs2)=O)CCC2CN(C(C3CC34CCSCC4)=O)CCC12 92559,C#Cc1cn(C)nc1C(=O)NCC1CN(C(c2cnc(S)n2C2CC2)=O)CC1C 92560,c1(CC(=O)NC2C=CC(CNC(C3N(C(C)=O)CCC3)=O)C2)ccc(O)c(C)c1 92561,c1(C(C)NC(=O)NC2CC(C)(COC)C2)cccc(SC)c1 92562,C1(C(=O)NC2C(C)(C)CN(C(=O)Cc3ccsc3)C2)CCc2nccn2CC1 92563,C#Cc1ccc(C(=O)NCCC(C)NC(C2CC(C#N)C2)=O)c(F)c1 92564,C(c1ccccc1[N+](=O)[O-])=CC(=O)NC1CCN(C(C2CCCCC2)=O)CC1F 92565,N1(C(C2(CC)CC2)=O)CCN(C(c2ccc(C3CC3)c(F)c2)=O)CC12CCC2 92566,CCC(C)C(O)C(=O)N1CC(n2cc(-c3ccnc(C)c3Cl)nn2)C1 92567,n1(C2CCN(C(c3n(Cc4ccc(C)nc4)ncc3)=O)C2)ccc2ccccc12 92568,c1(C(C)C)cccc(CNCC2(F)CC(CO)C2)c1NC(=O)OC(C)(C)C 92569,c1(OC)cc(C)ccc1N(C1CC(N)C1C)C(c1ccccc1)=O 92570,NC1CCN(C(c2csc(-c3cc(Br)cs3)n2)=O)C(CO)C1 92571,N1(C(C2CCN(CC)CC2)=O)CCN(C(C2CCSCC2)=O)C(CC#N)C1 92572,N1(C(C(C(C)C)SCC)=O)CCOC2(CCN(C(=O)CCCc3cncs3)C2)C1 92573,C(C(F)(F)CCNC(C1CC12CC2)=O)n1cc(CN(S(C)(=O)=O)C)nn1 92574,C1(NC(c2nc(C)n(C)n2)=O)CC2CC(NC(=O)C3=CCOCC3)CC2C1 92575,Cc1cn(-c2ncccc2Cl)[nH]c1=NC(=O)c1c[nH]c(C2CC2)c1C(N(C)C)=O 92576,C1(CNC(C2(C)CCCS2)=O)CCN(C(c2csc(CN3CCOCC3)n2)=O)C1 92577,CC1Oc2c(C(=O)NC(CNC(=O)C(C)(F)F)C3CC3)cccc2NC1=O 92578,O=CN1CCOCC1C(N1CC2CC2(CNC(C2CC(C3CC3)=NO2)=O)C1)=O 92579,N1(C(CCc2c(C)ncs2)=O)CCN(C(C2CCS(=O)(=O)N2C)=O)CC(O)C1 92580,C1(C(N2CCC(N(C(=O)C=CSC)CCC)C2)=O)CCc2nc(C)ncc2C1 92581,c1(OC)ccc(N(C(=O)C(C)N(C)Cc2ccc(Br)s2)Cc2ccco2)cc1 92582,CN1CC2C(C(=O)OCC3(C(=O)NCC4(NC(=O)N(C)C)CC4)CC3)C2C1 92583,Cc1cc(CNC(=O)NC(Cc2cccc(Br)c2)C(=O)O)ncn1 92584,C(C(C)(C)CN=c1[nH]c(=N)[nH]c(=NC(C)Cn2cc(C)cn2)[nH]1)OC 92585,c1(C(=O)NC(C2CCN(C(C3(OC)CCCOC3)=O)CC2)C)cnc(Cl)cc1N 92586,c1(C(=O)OC)cc(S(=O)(=O)N(C(c2ccccc2)CF)C)ccc1F 92587,C1(NC(Cc2c(C)occ2)=O)CCOCC1NC(C1(CCO)CC1)=O 92588,C=C(C)C(C)(O)C(=O)NC1CCN(C(=O)COc2cccc(Cl)c2Cl)CC1CO 92589,Cc1ncnc(C(=O)NC(C)CC(C)NC(=O)CCC(=O)c2ccc(Cl)s2)c1C 92590,c1(C(C(N2CC(C)OC(C)C2)=O)(C)C)ccc(Cl)cc1[N+](=O)[O-] 92591,C(=O)(C(CC(C)C)N(C1CC1)CC1CC1)OC.c1(C2C(=O)N2)ccccc1Br 92592,CC1CN(C(=O)C(C)(CO)NC(c2ccc(C(N)=O)o2)=O)Cc2nncn21 92593,N1(C(C(C(C)C)n2ccnc2)=O)CC2CCCN(C(c3cc(O)n(C)n3)=O)C2C1 92594,N1(C(C(CO)OC)=O)CCC(O)(CCNC(=O)COC2CC(F)(F)C2)CC1 92595,c1(C(=O)NCC(=CC(=O)NC(C(CCC)C)CO)C)ccc2cc[nH]c2n1 92596,c1(NC(CC2(C)CN(Cc3c(OC)c(F)ccc3)C2)=O)nccc2[nH]ccc12 92597,c1(CC(N2C(CNC(C=CCC)=O)CN(C)CC2)=O)ccc2c(c1)COC2 92598,Cc1cccc(C(=O)C(=O)Nc2cccc(CNC(=O)CC(C)C)c2)c1 92599,c1(CC(C)(C)C)cn(CC(C)C(=O)NCCCOCC)nn1.C(NCCO)NCC 92600,CP(C)(=O)c1ccc(C(=O)NC2C3CN(C(C45CCCC(C4)OC5)=O)CC23)nc1 92601,N1(C(Cn2ccc(C)c2)=O)CCC2(CC(NC(=O)CCCCC(N)=O)CO2)C1 92602,N1(C(c2ncnc(C)c2C)=O)CCCC2(CCN(C(=O)COCC(F)(F)F)C2)C1 92603,c1(C(N2CCC(C(C)(C)NC(C(F)OC)=O)C2)=O)cccc2ccc(O)nc12 92604,C1(C(=O)N(c2nnco2)C(C2CCC2)C2CC2)CCCN1C1CC1 92605,C1(C(=O)NC(C(=O)NCC(=O)OCC#C)CCSC)CC(=O)C12CCC2 92606,c1(CC(N2CC(CCO)(NC(c3cc(C)no3)=O)C2)=O)c(C)noc1Cl 92607,Nc1ncnc2c1ncn2CCCCC(=O)Nc1cccc2c1ncn2C 92608,c1(CCC)nc(C)c(C(=O)NCCC2CC(NC(=O)C=CC3CCCC3)C2)o1 92609,c1(CC(=O)NC(C)CCCNC(C2(C)CC2C)=O)ccccc1Br 92610,c1(C(=O)NC2C(C(=O)NCCn3ncc(C)c3)COC2)cncc(F)c1 92611,C(=O)(C(C)C(F)F)NCC(C)NC(=O)CCc1cnn[nH]1 92612,CC(C(=O)N(C(C)CCNC(c1ccc(C2CCOC2)cc1)=O)C)C(C)(F)F 92613,C1(C(=O)NCC)CCCN1C(c1ccc(CNC(=O)CCCNC(N)=O)s1)=O 92614,C1(C)(CNC(c2ccn(CC(C)C)n2)=O)CCCN1C(=O)COC1CCCCC1C 92615,n1(CC)ccc(C(=O)NCC2(CNC(=O)CC=CC(C)(C)C)CCCCC2)c1C 92616,C1(C(=O)NCC2C(NC(C3(COC)CCC3)=O)CCCC2)CCC2CCCCN12 92617,C#CCCCCC(=O)N1CCN(C(=O)CC(C)c2ccccc2)CC1CCO 92618,C(CC(CC)C(=O)NC(C1CC=CCC1)C(=O)NC1CCCC(CO)C1)=CC 92619,S(=O)(=O)(c1c[nH]c(C(N2CC(CCNC(=O)C(O)C(C)(C)C)(OC)C2)=O)c1)NC 92620,N1(C(C(CC)(C)F)=O)CC(NC(c2ccc(C(F)F)nc2)=O)C(N=[N+]=[N-])C1 92621,C1(C(=O)NC2CC(NC(c3ccccc3CO)=O)CC2O)(OC)CCC(C)(C)C1 92622,Cc1cc(C(=O)NC2CCCC2CNC(C2(F)CC2C)=O)cc2nc[nH]c12 92623,N1(C(C(C)OC2CCCCC2)=O)CCCC(CNC(=O)Cc2ccsc2Cl)C1 92624,C(=O)(C1=CC2(CCN(C(c3ccc(C(C)C)o3)=O)C2)C1)NCc1ccc(SC)o1 92625,c1(NC)cncc(C(N2CCCC(CN(C(=O)Cc3ccnc(C)c3)C)C2)=O)c1 92626,c1(NCC2(F)CCN(C(=O)C=C3CCSCC3)CC2)ccc(Br)cc1[N+](=O)[O-] 92627,c1(C(=O)NC2CCC(CNC(COCCCC)=O)C2)cc(OC)cc[n+]1[O-] 92628,C1(NC(CN(c2ccccc2)C(C)=O)=O)COCC1C(=O)NC(c1ccsc1)C 92629,C1(NC(c2c(C)snc2)=O)CCCC(C(=O)NCCOCC(O)CO)CC1 92630,c1(CC)nn(C)c(OC)c1C(c1nnnn1C1CCC1)NCC(C)CCO 92631,N1(C(C23N(C(c4n(OC)cnc4C)=O)CC(CO)(C2)C3)=O)CC(C2CCCCC2)C1 92632,c1(C(N2CCC(N(C(c3cnc(O)n3C)=O)CC)C2)=O)cccc2nccnc12 92633,c1(OC)ncccc1C(=O)Nc1cccc(CNC(=O)Cc2c[nH]nc2C)c1 92634,N1(C(C(CC)=CCCC)=O)CC(NC(C2(COCC)CCC2)=O)C(SC)C1 92635,N1(C(CS(CC)=O)=O)C2CCC1C(CNC(c1c[nH]cc(Cl)c1=O)=O)C2 92636,N1(C(C=CC=CC)=O)CCC(CC(=O)NC(CN2CCCC2)CC)C1 92637,N1(C(CCCCCC)=O)CC2CCCC2(NC(c2nnccc2C)=O)C1 92638,CCC(C)C(C(=O)NCC1(C)CCCC1O)NC(=O)C(=O)NC1CC1 92639,c1(-c2c(N3CCN(C(CC)=O)CC3)nccc2)ccc2[nH]c(C(=O)OC)cc2c1 92640,C=CCCN=C(NCC(C)C(F)(F)F)NCCc1ccc(C2CCCCC2)cc1 92641,C1(C(N(C)CC2CCCN2C(=O)C2=CCCO2)=O)CC2CCC(C1)N2C 92642,CCC(C)(C(=O)N1CCC(F)(C(=O)NC(C)C(C)(C)C#N)C1)OC 92643,c1(C(N2CCN(C(C=CC(CC)=CC)=O)C(C)C2)=O)cc(C#N)ccc1Cl 92644,C1(C(=O)NC(C)C(C)(C)NC(c2cncc(Cl)c2)=O)OCCOC12CCC2 92645,Cc1ncc(C(F)(F)F)cc1C(=O)NCC1CCC1NC(c1ccon1)=O 92646,CCC(CC(=O)NC1CCC(NC(c2conc2C2CCC2)=O)CC1)SC 92647,c1(C(=O)NCC(CN(C(=O)C2=CCOCC2)C)O)cnc2c(Br)cccn12 92648,N1(Cc2nc(C)[nH]n2)CCOCC(C(N2CCCC(C(N)=O)C2)=O)C1 92649,C(=O)(CCCC(=O)N(CCCOCCNC(=O)C(O)Cn1cncn1)C)N(C)C 92650,c1(C(N2C(CNC(c3cnn[nH]3)=O)CC(OC)C2)=O)cc(F)cc2c1NCCC2 92651,N1(CC(=O)NCC2CCC(NC(C=C(C)Cl)=O)CC2)CCCCC(O)C1=O 92652,N1(C(C=NOC)=O)CC(NC(c2cnc(C)c(C(F)(F)F)c2)=O)CC(O)C1 92653,C1(CC(=O)N(CC(C)NC(C23CC(CC)(C2)C3)=O)C)CCCN(C)C1 92654,CCC(C)(C)OC1(CC(=O)NN(CC(C)SC)C(=O)CC2CCC2)CCC1 92655,C1(CC)C(C(=O)NC(C)Cc2nc[nH]n2)CCCN1C(C1CC2(CC2)CO1)=O 92656,n1(CC(=O)N(C)CC2N(C(C(C)N(C)C)=O)CCC2)ccc2ccccc12 92657,Cn1cnc2c1CCC(C(=O)NCC1CC(NC(c3ccc(O)c(F)c3)=O)C1)C2 92658,C12(C(=O)NCC(=C)CCNC(=O)C(N3CCN(C)CC3)C)CC(C)(C1)OC2C 92659,C1(CNC(CSCCC(C)C)=O)C2CCC(C2)N1C(C1CC(=O)N(C2CC2)C1)=O 92660,C1(C(N2CC(O)(CN(C(C3C(C(=O)OC)C3)=O)C)C2)=O)C(C)(C)C1(C)C 92661,N1(C(C(=O)NC(C)CN2CCOCC2)=O)CC2CCC1C1CNCC21 92662,C1(NC(C(CC2CC2)NC(CC2OCC(C)(C)C2)=O)=O)CCCN2CCCC12 92663,Cc1ccccc1C(C)CC(=O)N1CC(O)(C(C)NC(c2nncn2C)=O)C1 92664,Cc1cccc2c1CCOC2C(=O)Nc1ccc(F)c(C#N)n1 92665,CC1CC(CNC(=O)CCC2CC2C)CN(C(=O)C=Cc2ncc[nH]2)C1 92666,CC(CF)CC(=O)N1CCC(C(C)CNC(c2ccn(C3CC3)n2)=O)CC1 92667,c1(N(C)C)nccc(C#N)n1.C12CCCN(C1=O)C2=O 92668,c1(OC)cc(NC(C2CC2NC(c2cccc(O)c2O)=O)=O)ccc1C 92669,CC(CCCCN=c1c(C#N)c[nH]c2cc(F)cc(F)c12)NC(=O)C1=CCCO1 92670,Cc1cc(F)ccc1C(N1CCOC(CNC(=O)C=CCOCC(F)(F)F)C1)=O 92671,C1(C(=O)NCc2c(C(=O)NCCC3CCN(C)C3)scc2)CCC(=O)NC1 92672,Cc1c(C=CC(=O)NCCCCC(C)NC(C23CCC(CC2)CO3)=O)cnn1C 92673,C(C(C)(CC(C)C)NC(C1CCOCC1(C)C)=O)NC(c1cccc(C)n1)=O 92674,N1(C(CCSC)=O)CC2CCCC(CNC(=O)CN3CCn4nccc43)C2C1 92675,C(C)(C)(CC(=O)N1C(C(=O)NCC2CCC2(F)F)CCC1C(C)C)OC 92676,S(=O)(=O)(c1c[nH]ccc1=NCCC1CC1C)N(CCCCOC)C 92677,N1(C(C2C(C)CC=CC2)=O)CCN(C(=O)CCn2ccccc2=O)CC1CCO 92678,n1(CC)ccc(=NC(=O)C2(CC)CCN(C(c3ncc[nH]3)=O)C2)[nH]1 92679,N1(C(CCN(C(c2c(CC)cco2)=O)C)=O)Cc2n[nH]cc2C1CO 92680,c1(C(=O)NCCC(=C)CNC(=O)C=CC=CC)[nH]c(O)nc1C 92681,Cc1nc2sccn2c1C(=O)NCC(O)CNC(C1C2CCC1CC2)=O 92682,C12(NC(C3CN(C(C)=O)C3)=O)CC(CNC(C3CCOC3=O)=O)(C1)OC2C 92683,C(=O)(CC(C)C(F)(F)F)N1CCCC(CC=C)(NC(=O)CCC=CC)C1 92684,N1(C(CC2OCCN(C(C(C3CCOCC3)C)=O)C2)=O)CCC2(CCCO2)C1 92685,C1(C(N2CCC(C)(CNC(=O)C3=NNC(=O)C3)C2)=O)CCc2nccn2C1 92686,c1(C(=O)NC2CCN(C(c3c(CC)cccn3)=O)C2)cc2c(C)c(C)ccc2[nH]1 92687,Cc1c(C(C)NC(N2CCC(C)(CC3CCC3)C2)=O)cnn1-c1ccccn1 92688,C1(CC(=O)NCCCCCCNC(=O)CC2CCC(=O)N2)CCCCCCC1 92689,C1(C(N2CC(C)C(CNC(=O)C3=C(Cl)CC3)CC2)=O)CN(C)CCN(C)C1 92690,c1(OCC)cccc(C=CC(=O)NC(c2ccccc2)CNC(=O)C=NOC)c1 92691,C(=O)(CCS(C)=O)NCC1(C(C)NC(c2nc(C(=O)OC)oc2)=O)CC1 92692,N1(C(CCS(C)(=O)=O)=O)CCC2(C1)CN(C(C1CS(=O)(=O)CC(=O)N1)=O)CCO2 92693,N1(C(c2ccc(C)nc2C)=O)CC2CCCC2C1C(=O)NCCCC(F)F 92694,C1(NC(C(N2CCCCC2=O)C)=O)CC12CCN(C(c1cnsn1)=O)CC2 92695,C(=O)(C(C)(O)C(C)(C)C)NC(C)CNC(=O)Cc1ccc(CO)cc1 92696,N1(C(c2[nH]c(=NC)sc2)=O)CCCOC(CNC(=O)Cc2ccc(Cl)nc2)C1 92697,CCC(CCOC)C(=O)NC1CC(CO)N(C(c2ccc(C(C)C)cc2)=O)C1 92698,N1(C(CCN(CC)CC)=O)CC2(CCCC2)C1C(=O)NC1CCCC(C)C1 92699,CC(CC(=O)NCC1C2CCCOC12)C(C)(C)NC(c1cscc1Cl)=O 92700,C1(NC(c2cc(C)sn2)=O)CC(NC(c2ccsc2C)=O)C12CCC2 92701,CC1(C)CN(C(C2CCOC2C(=O)O)=O)CCC1NC(C1(CCN(C)C)CC1)=O 92702,c1(C(=O)NCc2c(CNC(=O)CO)cccc2)cc(Br)ccc1Cl 92703,Cc1cc(C)c(C(N2CCC(CCNC(C3CC34CC4(F)F)=O)CC2)=O)cc1C 92704,C1(C(=O)NC2C(SC)CCC2)CCC(O)CN1C(=O)Cc1nonc1C 92705,C1(CCNC(CC(=O)NCC#C)=O)C(C)CCCN1C(c1sccc1C#N)=O 92706,CC1CCCC=C1C(=O)N(C(CC(F)F)C(=O)N1CCC(C(F)F)CC1)C 92707,N1(C(c2ccc(C)o2)=O)CC2COCC(C1)C2NC(C1CCC2(CC1)CC2)=O 92708,N1(CCC)CC2(CN(C(c3c[nH]cc3C)=O)C2)C1 92709,C12(C(=O)NC(CC#C)CC)CC1CCN2C(c1nccs1)=O 92710,C(=O)(CCC(CC)CCCC)NC(CC#C)CC(N1CCC2(CC1)CC2C#N)=O 92711,C1(C)(C(=O)OC)CCN(C(C2CCC2CNC(=O)C(C)SC)=O)C1 92712,c1(NC(c2cnc(NCC(CC)(CC)OC)nc2Cl)=O)c(C)cc(C)cc1C 92713,C(c1ccccc1F)=CCC(=O)NC(C1N(C(C(CCOC)C)=O)CCC1)C 92714,CN1CCC(CC(=O)NC2(C)CCN(C(C3CCOC3)=O)C2)C1=O 92715,N1(CCOC)CC(C(N2CCC(NC(=O)CCSCC(C)C)C2)=O)CCC1=O 92716,CC1OCCOC1C(=O)NC1C=CC(C(=O)NCCc2ccsc2)C1 92717,C1(CC(=O)NCCC(CNC(=O)CCOc2ccccc2)O)CCCC(=O)N1 92718,C1(CCCC)CCN(C(=O)NCC2(C)CCN2C(=O)OC(C)(C)C)CC1 92719,c1(C(=O)NCC(CNC(c2c(CC)sc(=N)[nH]2)=O)(C)O)cnc2ncnn2c1C 92720,C1(CC(=O)OCC)CN(C(C)C(N2CCC(N3CCCCC3)CC2)=O)CCO1 92721,N1(CCCCC)CCCC(c2nc(-c3ccc(OC)nc3)nn2C(C)C(C)C)C1 92722,CC(C)(C#N)CCC(=O)NC1CN(C(c2cc(F)c(F)c(F)c2)=O)CC12CC2 92723,C1(O)(CC(=O)NCC2CCC2)CCN(C(c2cc(F)cc(F)c2)=O)CC1 92724,N1(C(CC(=O)OCC)=O)CCCN(C(=O)CNC(=O)CC2CCCC2)C(CO)C1 92725,c1(C(N2CCC(C(=O)Nc3ccc(Cl)cc3I)CC2)=O)cc2cn[nH]c2cn1 92726,C1(C2(NC(CSCCC)=O)CC2)CCCCN1C(=O)CC1CCCSC1 92727,Cc1ccc([N+](=O)[O-])cc1NC(=O)NCC(c1ccc(Cl)cc1)O 92728,N1(C(c2cccc(NC(C)=O)n2)=O)CCC(C2(NC(=O)C(CO)N(C)C)CC2)C1 92729,C1(C)(CC)C=C(C(=O)NCC2(C(=O)NCC(C)(CO)OC)CC2)C1 92730,CC1(C(N2CCN(CCNC(C3CC(CF)C3)=O)CC2)=O)COC(=O)N1 92731,C(c1ccc(C)cc1C)=CC(=O)NC1CN(C(C2=CC(C)(CC)C2)=O)CC1F 92732,C1(C(=O)NCC(CC)NC(=O)C=CCN2CCCC2)(CC)CC1(F)F 92733,CCCCCS(=O)(=O)NC(c1cncc(-c2nn[nH]n2)c1)=O 92734,Cc1cc(N)c(F)c(C(=O)NC(CNC(=O)Cc2ccc(Cl)cc2F)CO)c1F 92735,Cc1cc(C(=O)NCCC(C)NC(C2COCCN2CC2CCC2)=O)ncc1F 92736,C1(C(=O)NCCN(C(=O)CC2CCCN2CC)CCC)CCC(=O)N(CC)C1 92737,c1(C(N2CCC(O)(CC(=O)NCC3(O)CC(C)(C)C3)C2)=O)ccc(F)c(F)c1 92738,C(=O)(C#CC1CCCCC1)NCC1CC2N(C(C3(CC)CCOC3)=O)C(CC2)C1 92739,C1(NC(C2(C(=O)NC)CCC2)=O)CCC(NC(=O)CC2CC(F)C2)C1 92740,N1(C(COCCC)=O)CCC(O)(C(C)NC(c2cnc(N(C)C)c(Cl)c2)=O)CC1 92741,c1(CC)ccc(C(=O)NC(CC2CCOCC2)CO)nc1C 92742,c1(C(N2C(C)C(NC(c3ccnc(O)c3)=O)CCC2)=O)ccc2ncccc2n1 92743,Nc1ccc2ccccc2c1-c1ccccc1Cl 92744,c1(OC)cc(C)c(C(C)NC(c2cc(F)ccc2C(C)C)=O)cc1OC 92745,c1(C(N2CCC(F)(CNC(C3(O)CCOC3)=O)CC2)=O)n[nH]c2c1CCCCC2 92746,N1(C(c2c(C)occ2)=O)CCN(C(c2ccc3c(n2)CCCN3)=O)C2CCCC12 92747,CC1CN(C(=O)CSc2nnc(S)s2)CC(C)C1NC(c1cccc(=O)o1)=O 92748,c1(OC)cc(CC(N2CC3(CCN3C(c3csnn3)=O)C2)=O)ccc1C 92749,C(=O)(CC(C)CC(=O)NCC1(C(=O)N(CC(O)C(C)(C)C)C)CC=CC1)OC 92750,C1(C(=O)NCC(C)CNC(c2ccc(C(F)F)cc2)=O)C(C2CC2)C1(F)F 92751,N1(C(C(C)C)=O)CCOC(CNC(C2CCOC(=O)N2)=O)C1 92752,CCCC(O)C(=O)N1CC(O)CC1CNC(=O)CCC1OCCO1 92753,c1(OC)cc(=NC(=O)C2CC3CCC2N3C(=O)CC2CC3CC3C2)[nH]n1C 92754,Cc1cc(C(F)(F)C(=O)NCC2(O)CN(C(=O)C(C)NC(N)=O)C2)cs1 92755,C12(C(N3CC(C#C)(N(C)C)C3)=O)CCC(CN(C(=O)C(C)CCOC)C1)C2 92756,N1(C(C=NOC)=O)CC2(NC(=O)COCC3CCCCO3)CCCC2(F)C1 92757,N1(C(C2C(C=C)C2)=O)CC(CNC(c2cc(C(C)(C)C)n[nH]2)=O)C2(CC2)C1 92758,C(C(CC(C)(C)C)C(=O)OC)Oc1c(OCC#C)ccc(F)c1 92759,c1(OCC)ccc(C(N2CC(c3cc(OC)ccc3O)C2)=O)cc1Cl 92760,C1(OC)CC(NC(C2(Br)CC2)=O)CN(C(c2ccccc2C2CCOC2)=O)C1 92761,CCCC(CCCNC(C1CCN1CC)=O)NC(c1cccc(Cl)c1N)=O 92762,CCCC(C(O)C(=O)NCc1nnc(CC)o1)NC(=O)CCc1nccs1 92763,O(NC(=O)CCNCC)C(C(=O)N(CC=C)CC=C)C 92764,C(N=c1cc(NCc2ccnnc2)nc[nH]1)C1(N(C)C)CCSC1 92765,c1(CC(N2C(CCNC(=O)C(O)c3ccsc3)COCC2)=O)cn2ccsc2n1 92766,C=Cn1nncc1C(N1CCCC1(C)CNC(C1CC1c1cccc(C)c1)=O)=O 92767,c1(OC)ccc(N2CCN(C(C)C(=O)NC(C3CCC3)C)CC2)c(F)c1 92768,N1(C(=O)NCCC(=O)OC(C)C)CC2CCCCC2(CCC(=O)O)C1 92769,N1(C(CNC(CC)=O)=O)CCCC(N(C(=O)C(CO)NC(N)=O)CCO)C1 92770,Cc1sc(C(F)(F)F)nc1C(=O)NC1CN(C(C2CCCOC2)=O)CC1C 92771,c1(C(N(CCNC(C2CCN(CCCC)CC2)=O)C)=O)ccc(O)nc1C 92772,C1(C(=O)NC2C=CC(C(N3CCC(NC(=O)OC)C3)=O)C2)(CC)CNC(=O)C1 92773,C1(NC(C2CCCN(CCC)C2)=O)CCCCN(C(c2ccco2)=O)CC1 92774,C1(NC(C(CC=C)c2ccccc2)=O)CCCN(C(C2CCC(=O)N2)=O)C1C 92775,Cc1ccc(C2CC2C(N2CC(N(C(C3C4CC5C(C4)C35)=O)CC)C2)=O)c(Cl)n1 92776,CC1(C(N2CCOC(CCNC(=O)COc3cccnc3)C2)=O)CNC(=O)C1 92777,C(=O)(C(C)(C)CCCO)N1C(CCNC(C2CN(CCOC)C(=O)C2)=O)CCC1 92778,CC1CN(C(C2CCC(CO)CC2)=O)CC1(C)C(=O)N(C1CCC2(CC1)CC2)C 92779,CCC(CC)(CC(=O)OC)C(=O)NC1CCCCN(C(c2cc(OC)n[nH]2)=O)C1 92780,CCCCCC(C)(C)C(=O)NCC1CCC(C(N2CCOC(C(=O)OC)C2)=O)C1 92781,c1(C(N(C(CNC(c2cc(C)[nH]n2)=O)C2CC2)C)=O)c(Cl)ccc(F)c1F 92782,CCC(CNC(=O)C(C1CCCO1)NC(=O)C(C)C1(O)CCC1)CC 92783,C1(C(CC)(C)C)CCCCN1C(c1cn(C2CCCC2)nn1)C(=O)NC1CCC1 92784,c1(CNC(C2(CNCC3N(CC)CC3)CC2)=O)ccc(Sc2nnnn2C)cc1 92785,C1(CNC(c2ccc(C)o2)=O)CC(NC(=O)CN=S(C)(C)=O)C12CCC2 92786,CC(CC(=O)N1CC(CNC(=O)CCNC(=O)CO)C(F)(CO)C1)C(C)(C)C 92787,CCC(CC)(C(=O)OC(C)(C)C)C(=O)N1CCN(C(c2nccn2C)=O)C2CC12 92788,CC(CCI)(c1nnnn1C1CC1)NC1(n2cc(CC3CCCCO3)nn2)CC1 92789,c1(N(C)C)cc(C(=O)NC2CCC2CNC(=O)CCCc2ccsc2)ccc1Cl 92790,C1(NC(CCC=C)=O)CCN(C)C12CCCN(C(=O)CC1CC(=O)NC1=O)C2 92791,c1(C(=O)NCCC(C)NC(c2cc(C(CC)C)no2)=O)c(C)nc(C)nc1C 92792,C1(CN2CCC(C(N(CC(F)(F)F)CC=C)=O)CC2)CN=C(C(F)(F)F)O1 92793,N1(C(Cc2cn(C(C)C)nn2)=O)CCCC(N(C(=O)C(=O)NC(C)(C)C)CCF)C1 92794,c1(C(=O)NC(C(C)C)CNC(=O)CCCc2cncs2)cnc2[nH]cncc1-2 92795,C1(CCN)(NC(C(C)Sc2ccccc2)=O)CCCCC1 92796,c1(C(N(CCCNC(C2(CC=C)CCOC2)=O)CCO)=O)cncc(C=C)c1 92797,CC(C)CC(CNC(=O)C(F)C(C)C)NC(C1(COC(C)C)CC1)=O 92798,c1(OC)cccc(NC(=O)C(c2ccc(Br)nc2)N(CCC#N)CCC#N)c1 92799,CC(CC(C)(C)C)C(=O)NC1(CCO)CN(C(=O)CC2NC(=O)NC2=O)C1 92800,C1(C(=O)NCCc2nc(C)[nH]n2)CN(C(C2CN(C(N)=O)C2)=O)CC1(F)F 92801,Cc1nn(C)cc1CC(N1CCC(CNC(=O)COC(c2cccs2)C)C1)=O 92802,N1(C(c2c(C)c(-c3ccccc3)[nH]n2)=O)CC2CCC(NC(=O)CSC)CC2C1 92803,C1(C(=O)NCC2N(C(CCOCC)=O)CCCC2)CCS(=O)(=O)C1(C)C 92804,C1(CNC(C2(CC(C)C)CCNC2=O)=O)COCCN(C(C2(F)CC2)=O)C1 92805,C1(NC(c2[nH]cc(CC)c2)=O)C(C)CCN(C(=O)CC2CCCC(C)C2)C1C 92806,c1(NC2(C(N)=O)CN(C(Cc3ccc(OCC)cn3)=O)C2)ccc(F)cc1F 92807,N1(C(=O)OC(C)(C)C)CC2(CCC(N)CC2)C1.CC1(C)OCC(C(O)C=O)O1 92808,c1(CN(C2CC3CCC2O3)C(C)C2CC2)ccc(OC(F)F)cc1 92809,Cc1ncncc1C(N1CC(O)(C(C)(C)CNC(C2(C)CCN(C)C2)=O)C1)=O 92810,c1(NS(c2cn(C)[nH]c2=N)(=O)=O)cccc(S(F)(F)(F)(F)F)c1 92811,Cc1cc(C2CCN2C2CC2c2cccnc2-c2n[nH]c(C)n2)cc(C)c1 92812,Cc1nccc(C(=O)NC2CCC(NC(c3ccn(C(C)C)c3C)=O)C2)c1O 92813,C1(CNC(C(CN(C)C)(C)C)=O)CC2(C1)CN(C(=O)CC1CN(C)CC1O)C2 92814,N1(C(C2CC(O)(CC#C)C2)=O)CC2(CCC(F)F)CC1CCO2.c1(=O)c(=O)[nH]1 92815,C1(C(=O)NCc2nccs2)CCC(n2cc(-c3cnccn3)nn2)CC1 92816,N1(C(CCC(C)c2ccccc2)=O)CC2(C1)CN(C(C13CC(CO1)C3)=O)C2 92817,C1(NC(C2CC(OC)C2)=O)(CO)CCCN(C(=O)COCCCN(C)C)C1 92818,N1(C(C(COC)(C)C)=O)CCCC(C2(NC(=O)C(F)C(F)(F)C(F)(F)F)CC2)C1 92819,c1(SC)nccc(N2CCC(CF)(NC(c3cc(Cl)n(C)n3)=O)C2)n1 92820,CC(C)C(O)CCN=c1nc2c(cnn2C)c(NCCc2ccc(N)cc2)[nH]1 92821,C1(CNC(c2[nH]ccc2CNC(C23CCCC2C3)=O)=O)CCC2(CC1)CC2 92822,Nc1c(F)ccc(Cl)c1C(=O)NC1CN(C(c2cc(Cl)c(F)cc2F)=O)CC1F 92823,C=CCCC(CC(C)C)C(=O)NC(COCC)C(=O)NCCC(CCC)N(C)C 92824,C1(N(C(=O)CC2CC(CN(C)C)C2)CC)CCCN(C(C2(CO)CCC2)=O)CC1 92825,N1(C(c2ccc(C(F)(F)F)cc2)=O)CCc2cc(-c3cc(F)ncc3F)ccc2C1 92826,C#Cc1ccc(CC(=O)NC2CC(NC(=O)C(C)CCCOC)CC2O)cc1 92827,C(c1ccccc1)=CC(=O)NCCC1CCC(NC(=O)C=C2CCCCC2)C1 92828,C1(C(=O)NC(CC)C(F)(F)F)CCCCN(C(=O)Cc2csnc2C)C1 92829,C#CC1(C(N2CCCN(C)CC2)=O)CCN(C(=O)CC2CCCCO2)C1 92830,C(=O)(CCCCCCC)N1CCC(CC#C)(C(=O)N(CC(O)C(C)(C)C)C)C1 92831,C1(NC(c2c(C)nccn2)=O)CC2(NC(c3ccc(CCF)cc3)=O)COC1C2 92832,CC(CCO)C(=O)N1CCC(CCNC(c2ccc(CCN(C)C)cc2)=O)CC1 92833,CCCC(C(O)C(=O)NCC(C)(C)CC(C)O)NC(=O)CCS(N)(=O)=O 92834,N1(C(CCc2ccc(C)nc2)=O)CC(O)CC1(C)CNC(=O)C=CC(C)(C)C 92835,C1(C)(C(N(CCC)CCOC)=O)CC12CCN(C(=O)CCCC(=O)C1CC1)CC2 92836,N1(C(CC2N(CC)CCC2)=O)CC(NC(C23COCC(C2)C3)=O)CC(O)C1 92837,O=S1(=O)CC2CC(N=c3[nH]c(=NC4CCC4)[nH]c4cc[nH]c34)CC2C(CO)C1 92838,C(=O)(C1=NOC2COCC12)NCC(C(=O)N(CC=C)C(C)C)(F)C(C)C 92839,C1(C2(O)CN(C(=O)C=C3CCOCC3)C2)(CNC(C2CN(C)C(=O)CC2)=O)CC1 92840,CCC(C)C(C)(O)CNC(=O)CN(C1CC(C#N)C1)C(c1ccnc(O)c1)=O 92841,c1(C(N(CC(CNC(C(C(C)C)SC)=O)C)C)=O)cc(Br)ccc1N 92842,n1(CC)nc(C(N2CC(CNC(=O)CCOC)C3CC23)=O)c2c1CCOC2 92843,N1(C(=O)CCC2CC(F)(F)C2)CCN2CCN(C(=O)C(F)C(F)(F)F)CC2C1 92844,c12cncc(c1)C(=O)NC2.C1(N)CCN(C(=O)CCC(=O)OC)C1C.C(C)(C)(C)OC 92845,CC(CCNC(C1(C)CC1)=O)CCNC(=O)C(C)(C)Cc1cnn[nH]1 92846,c1(C(N2CCN(C(c3ncc(C)c(C)c3)=O)CC2CF)=O)cnn2c1OCCC2 92847,c1(NC(CC)CN(C)C)ccc(S(=O)(=O)NCCC2CCN(C)CC2)cn1 92848,Cc1cc(C(N)=O)ccc1NC(CCCCCO)c1nnnn1C1CC1 92849,Cc1c(C(=O)NCC2CN(C(C3CCC4CC3CO4)=O)CCCO2)cncc1Cl 92850,C12(NC(c3c(C)cc(C)[nH]3)=O)CCN(C(=O)Cc3cncnc3O)CC1C2 92851,C(CCCC(C)C)NC(C(C1CN(C(c2scc(OC)c2)=O)C1)O)=O 92852,c1(CS(=O)(=O)NC)ccc(OCC(NOCC)=O)cc1 92853,C1(NC(COCCC(=O)NCC2(NC(CCOCCC)=O)CC2)=O)CCCOC1 92854,Cc1ncncc1C(=O)N1C(N)CCC1.C1(C(=O)N)CN(C(C2CCC(C)CC2)=O)CC1O 92855,C(=O)(C(C)(C)C(=O)NC(C(=O)Nc1c(CC)cccc1CC)C(C)C)OCC 92856,C1(CN(C(C(c2ccccc2)OC)=O)C)CCN(C(c2nc(Cl)sc2C)=O)CC1 92857,c1(C(N2C(CNC(C(CCCC)O)=O)CC(F)(F)C2)=O)cc2c(=O)[nH]ccn2c1 92858,N1(C(c2n(CC)ncc2)=O)CCN(C(=O)C(c2cccc(Cl)c2)SC)CC12CC2 92859,C1(C(=O)NC(C)CN(C(=O)CSC(=N)N)C)CC12CC(O)C2 92860,c1(NC)scnc1C(N1CCC(C(C)C(=O)NCC(CSC)OC(C)=O)C1)=O 92861,CC(C(=O)NC1CC(C(F)F)(NC(C2COC(=O)N2C)=O)C1)C(F)F 92862,N1(C(CC2CCCN(C(CCSC)=O)C2)=O)CCC([N+](=O)[O-])CC1 92863,c1(OCC)ccc2cc1OC2=O.N1(C(C)=O)CCC2C(C1)N2C(=O)C=CCBr 92864,N1(C(C(CC)O)=O)C2CCC1CC(NC(c1cccc(N)c1C)=O)C2 92865,N12CCCC(C1)CCc1cn(nn1)CC(=O)N(C(C(N)=O)C1CC1)CC2.CO.SC 92866,c1(C(N2CC(NC(c3cc(CC)on3)=O)C2)=O)c(Cl)cc(C)cc1Cl 92867,N1(Cc2nc(CCOC)on2)CCC2(NC(=O)CC3CCCC(=O)N3)CCCC12 92868,CN=c1nc(NC2CCCn3nc(C)nc32)[nH]c(=NCC(C)c2ccsc2)[nH]1 92869,c1(OC)ccc(Br)c(C(=O)NCCC2CCCN(C(C3COC3)=O)CC2)c1 92870,c1(N(CCOCC)C)nnc(C2CCC(=O)N2)n1Cc1sccc1C 92871,C1(NC(C(C)NC(C2CCCCC2)=O)=O)CCCCC1NC(=O)C(CCO)N(C)C 92872,N1(C(CCc2n(C)cnc2)=O)CC=CC(C(=O)NCC2CCOC2(C)C)C1 92873,CCC(C)C(C(=O)N1CC=CC1(C)C(=O)NCCc1cn[nH]c1)N(C)C 92874,C(=O)(CCCCCCNC(=O)Cc1csc2nc(C)cn12)N1CC(F)(C(=O)OC)C1 92875,c1(C(=O)NCCN(C(=O)Cc2csc(Cl)c2)CC)ccc(-c2cc[nH]n2)s1 92876,N1(C(=O)COc2cc(F)ccc2F)CCC2(CCN(c3cnc(F)cn3)C2)C1 92877,c1(C(N2C(C)CC(CNC(C3(C)CC3(F)Cl)=O)C2)=O)cccc(=O)n1O 92878,Cc1sc(Cl)nc1C(N1CC(CN(C(=O)C(C)Cn2ccnc2)C)C1)=O 92879,N1(C(c2c(C)cns2)=O)CCC2CCC12CNC(C1(N2CCCC2)CCC1)=O 92880,C1(NC(CC(CC)C)=O)COC2(CCN(C(C3CC4CCC3O4)=O)CC2)C1 92881,C1(C)(NC(c2scc(OC)c2)=O)CCN(CC(=O)N(C)Cc2nccn2C)C1 92882,c1(CN2C(C(=O)Nc3cccc(C4(C(=O)O)CC4)c3)CC2)ccc(Cl)c(Cl)c1 92883,C1(C(=O)NCC2CCN(C(c3cnc(O)s3)=O)C2)(CF)CC(F)(F)C1 92884,Cn1cccc1C(=O)NCCCCCNC(=O)CC1(C)CC1(F)Cl 92885,C(=O)(C(C)(C)C(C)C)NCC(C)(C)NC(CC(=O)NCC(=O)NC(COC)C)=O 92886,CC1(C)C(C(c2nnnn2C2CCCC2)NCCn2ccnn2)C1(C)C 92887,CCN=C(NCC(c1ccc(Br)cc1)F)NCC1(C2CC2)CCCO1 92888,c1(C(=O)NCC(C)(O)NC(=O)OC(C)(C)C)ccc(C(F)(F)F)c(F)c1 92889,C1(C2CC2)(C(N2C(CC(N)=O)CCC2)=O)CN(C(c2ncn3c2CCC3)=O)C1 92890,c1(C(N2CC(C(N)=O)(CNC(C3(F)C(C)OCC3)=O)C2)=O)scc2c1CCCC2 92891,O=S(=O)(c1c[nH]ccc1=NC1CCN(c2ccc(Cl)cc2)CC1)NCC1CC1Cl 92892,C1(NC(C(CSC)OC)=O)COCCN(C(=O)Cn2cc(Br)ccc2=O)C1 92893,C1(NC(C(c2cn(C)nc2)O)=O)CCCC2CN(C(c3cc(F)n(C)n3)=O)CC12 92894,c1(C(=O)NC2C(NC(c3nn(C)c(Br)c3)=O)C2)ccn2ccsc12 92895,C12(C(N3CCC(O)(CNC(C=C(CC)C)=O)C3)=O)CCC(C1)C(C)(C)O2 92896,c1(N2CC(C)CC(C)C2)nc2c(F)cc(F)cc2c(=NCCCCN(C)C)[nH]1 92897,C(CNC(=O)C=CC(=O)NC1CC1)(CC(F)(F)F)NC(CSc1n[nH]c(=N)s1)=O 92898,N1(Cc2cccc(OC)c2C)CC2CN(C(c3ccc(N(C)C)nc3)=O)CC2C1 92899,C12(C(=O)NCC3(CNC(=O)C=Cc4cncs4)CCCC3)OCCCC1C2(F)F 92900,C1(N(C)C(=O)C2CC2)CCN(C(c2c(F)cccc2Cl)=O)CC12CC2 92901,c1(C(N2C(C)(CNC(CCCSC)=O)CCC2)=O)cc2occc2n1C 92902,N1(C(=O)Cc2ccccc2)CCCC(c2cn(Cc3ccccn3)nn2)C1 92903,C(c1ccccn1)=CC(=O)NCCC(=C)CNC(=O)CC(C)c1ccncc1 92904,C12(C(=O)NCC(CNC(c3c(CC)n(C)nc3)=O)(C)O)CCC(C1)S(=O)(=O)CC2 92905,c1(NC2CCN(C(C3CCCC(C)C3)=O)C(C)C2)ncnc2c1ncn2C1CC1 92906,N1(C(C(C(C)C)SCC)=O)CCCC1C=CC(N1CC(F)C1)=O 92907,Cc1[nH]nc2c1CCC(C(=O)NCCc1coc3ccc(F)cc13)C2 92908,c1(C(N2CCCC(NC(C3(CC=C)CC3)=O)C2)=O)c[nH]c2cc(Br)ccc12 92909,CC1=CCSC1C(=O)N(C1CCN(C(c2cnc(Cl)s2)=O)C1)C 92910,CCC1=NOC(C(N2CCC(C(C)(C)C(=O)NCCCc3nccs3)C2)=O)C1 92911,c1(COCC)nc(C(=O)NC(C)CC2CN(C(c3cc(Cl)cs3)=O)C2)cs1 92912,N1(C(C(C)N2CCCC2)=O)CC2C=CC1C(C(=O)NCCc1cn(C)cn1)C2 92913,O=C(C1=CCCOCC1)NC(CO)C(=O)NCCCc1cnn[nH]1 92914,N1(C(C(C2CC2)OC)=O)CCN(C(c2cc(C)nc(C)c2)=O)C(C2CC2)C1 92915,C(=O)(CC(C)CNC(=O)C(C)(C)CC1CC1)NC(c1ccc(C)s1)C 92916,N1(C(=O)NC2CC2c2ccc3c(c2)CCC3)C2CCC1CC(C(=O)NC1CC1)C2 92917,C1(C)(NC(C(N2CCC(C)C2)=O)=O)CCN(C(=O)CC2CCC(F)(F)CO2)CC1 92918,N1(C(CCCCCC#C)=O)CC2CCCC(NC(C3CCNC3=O)=O)C2C1 92919,c1(C(N2CCC(NC(c3cc4sccc4[nH]3)=O)C2)=O)cccc(F)c1Cl 92920,c1(-c2cn(C(CNC(COCc3cc(C)no3)=O)C)nn2)ccccc1S(C)=O 92921,c1(C(C(F)(F)F)NCC(c2n(C)cnc2)O)cccc(C(C)(C)C)c1 92922,c1(C(=O)OC)ccc(C(N2CCSC(C)C2C)=O)cc1Br 92923,c1(NC2CCN(C(c3cc[nH]c3C3CCCC3)=O)C2)cc(O)nc(O)n1 92924,c1(-c2cn(CCC(C(C)C)NC(C(C(=O)N(CC=C)C)CC)=O)nn2)ccc2c(c1)CCC2 92925,c1(NC2CCN(C(C)C(=O)N(C3CCCC(O)C3)C)C2)ncc([N+](=O)[O-])c(=N)[nH]1 92926,C(=O)(CCC(C)C#N)NCC1CC(NC(c2c(CC)nn(C)c2)=O)C1 92927,C1(C)(C(=O)NCC(CNC(C2CC(CC)(CC)C2)=O)C)CCC(C)C1 92928,C(=O)(CCC(C)(C)NC(=O)C(C)CC#N)N(C1(C(=O)OC)CC1)C 92929,Cc1ccc(O)nc1CNC(=O)CC(C)(C)CNC(C1OCCC1C(C)C)=O 92930,C(C(CC(C)C)C(=O)NCC1COCCN1C)NC(c1c(C)nsc1)=O 92931,CC(C)C(C(=O)NCCC1CCN(C(c2nc(=O)n(C)[nH]2)=O)C1)NC(N)=O 92932,Cc1cc(C)c(C(N2CCCCCC2CNC(c2nccnc2N)=O)=O)cc1N 92933,c1(C(=O)NCC2CC(OC)CN2C(C2CC(SC)C2)=O)cc(Cl)cc([N+](=O)[O-])c1 92934,c1(C(C)NC(C(=O)NCc2c(OC)cc(C)s2)=O)cc(C)cc(C)c1 92935,c1(OC)cc(N)c(F)cc1CSc1ccc(OCC2Sc3ccccc3O2)cc1 92936,C(=O)(C(C)(C(C)C)OC)N1CCC(CCNC(CC(C)SC)=O)CC1 92937,c1(C(=O)NC2CC(CC(=O)N(C3CN(C(C)C)C3)C)C2(C)C)cc(C#N)cn1C 92938,C1(NC(C(CC)CO)=O)CC2(CCN(C(C3C=C3C)=O)C2)C1 92939,C1(CNC(Cn2c(CCC)nnc2S)=O)CCN(C(=O)C2=CC(C)(C)C2)C12CC2 92940,c1(C(=O)NC(C2(O)CCN(C(Cc3nc(C)[nH]n3)=O)C2)C)cccc2cncn12 92941,C(=O)(C(C)(C)CS(C)(=O)=O)NCCC1CN(C(c2c(SC)cccc2)=O)C1 92942,c1(NC(C2C(NC(C(C)S)=O)C2)=O)ccnc2cc(Br)ccc12 92943,Cn1nc(C(F)(F)F)cc1C(N1CCC1CNC(=O)CC1CCCS1(=O)=O)=O 92944,CC1CN(C(C2(CCF)CCOCC2)=O)CC(C)N(C(c2csc(Cl)c2)=O)C1 92945,c1(C(=O)NCC2C(NC(C3(C(N)=O)CCC3)=O)C2)cccc(F)c1F 92946,C=CCCCCC(=O)NC(C)C(C)NC(c1cc(C2CCCCC2)on1)=O 92947,c1(OC)ccccc1C1CC1C(=O)NCCC(C)(C)NC(C1C(Cl)(Cl)C12CC2)=O 92948,N1(C(C(CC)F)=O)CCN(C(=O)COC2CCCC2)CC1c1ccnn1C 92949,c1(CC(N2C(CNC(C3CC(O)C3)=O)CCC(C)C2)=O)nnc2n1CCOC2 92950,Cc1cc(CNC(c2[nH]ccc2C2CC2)=O)oc1C(=O)NCCC(C)F 92951,C1(C(C)C)N(C(C2(CO)CCN(C(c3ccc[n+]([O-])c3)=O)C2)=O)CC1(C)C 92952,N1(CCS(C)(=O)=O)CCCN(C(C2C3CN(C(=O)CNC=O)CC23)=O)CC1 92953,C(=O)(C(CC(C)(C)C)OC)NC1CC2(CC(NC(CN(C(=O)OC)C)=O)C2)C1 92954,C1(CC(C)C)CC(NC(=O)C(N2CC(c3ccccc3)C2(C)C)=O)CCO1 92955,C1(C(N(C2CCN(C(=O)CCc3ccco3)CC2)CC#C)=O)CC2(CCC2)CO1 92956,c1(SCC#C)cccc(C(=O)NC(C)CCCNC(=O)C(C)OCC(C)C)c1 92957,N1(C(c2n(C)ncc2)=O)CCC(C2(NC(c3coc(O)n3)=O)CC2)CC1 92958,CC1=CCN(C(c2cc(CCNC(C3(N(C)C)CC3)=O)on2)=O)CC1 92959,c1(C(=O)NCC2(C(=O)NC3(CC)CCCCC3)CCCCO2)n[nH]c2c1CCC2 92960,c1(CC(=O)NCCCCNC(C2(SCC)CC2)=O)ncnc2sccc12 92961,Cc1cnc(F)c(CNC(=O)C(c2ccoc2)NC(=O)C2=CCCCC2)c1 92962,N1(C(CN(C2CCC2)C)=O)CCCCC12CN(C(C1(c3ccno3)CC1)=O)C2 92963,c1(NC)cnc(Cl)cc1C(=O)NC(C1CCN(C(C2CCCC(=O)N2)=O)C1)C 92964,c1(SC)nc2nc(C)c(CC(=O)NC3COC4(CCN(C(C)=O)C4)C3)c(C)n2n1 92965,C1(C(N(C)CC2CC2(F)F)=O)C2CC3C(C2NC(c2cc(C(F)F)[nH]n2)=O)C13 92966,N1(C(C(C)OCC)=O)CCc2ccccc2C1CNC(=O)Cc1ccsc1Cl 92967,c1(NC(=O)NC(CC)COCCc2cccc(C)c2)cc(OC(F)F)c(Br)cn1 92968,c1(C2CN2)cccnc1.N1(C(=O)OC(C)(C)C)CC(NC(C2CCCO2)=O)C1 92969,Cc1cc(CC(N2CCC(NC(c3cc(-c4ccccc4)co3)=O)C2)=O)cs1 92970,N1(C(CC2CCC(NC(C3CC(C)(F)C3)=O)C2)=O)CC(CO)C(CO)C1 92971,N1(C(CCC2CC(C)C2)=O)CCN(C(c2ncoc2C(F)(F)F)=O)C(C)C1 92972,C=CCCCCC(=O)N1CCCOC(CCNC(=O)CC(C)NC(N)=O)C1 92973,c1(C(N(C2CCC(NC(=O)CCCn3cncn3)C2)C)=O)cnc2ccsc2c1 92974,N1(C(C2CC(SC)C2)=O)CCCC1(C(=O)NCC(CC1CC1)CO)C(C)C 92975,C1(O)(CNC(C(CO)N(C)C)=O)CCN(C(c2nn(C)cc2C(F)(F)F)=O)C1 92976,C1(CNC(COCCCC(C)C)=O)CN(C(C2CCCCS2)=O)CCO1 92977,Cc1nnc2cc(N3CCCC(NC(=O)C(C)c4cccs4)CC3)ncn12 92978,c1(-n2cc(CCN(CC)CC)nn2)cncc(CNC(=O)C(C(C)C)SC)c1 92979,c1(C(=O)NCC(CC)NC(C2N(CCC)C(=O)CC2)=O)ccc(F)c(C)c1Cl 92980,c1(C(N(CCN(C)Cc2nnc(CO)s2)C)=O)cc(Br)c[nH]1 92981,CC1CCN(C(=O)C=CBr)C1CNC(=O)C=CC1CCOC1 92982,c1(N(C)Cc2c(OC)nccc2)nc(N(C)Cc2cnn[nH]2)cc(C)n1 92983,Cc1ccc(C(N2CC(CC(F)C(=O)N3CC(O)(c4cnn[nH]4)C3)C2)=O)[nH]1 92984,C1(CNC(CC2C(NC(C=CC(C)C)=O)CCC2)=O)CC(O)C12CCC2 92985,C1(C2CCN(C)CC2)(C(=O)NC(CC)CNC(=O)CCC2CC2(F)F)CC1 92986,C(=O)(C1=C(Cl)CCCC1)NCC1C2CN(C(CCNC(=O)NC)=O)C1C2 92987,O=S(=O)(c1cccc(=NCc2cc(C(F)(F)F)ccn2)[nH]1)N1CC2CC2C1 92988,CC(C)CC(C)C(=O)NC1(C)CCN(C(c2ccc(N)c(N)c2)=O)C1 92989,c1(C(=O)NC(CC=C)CNC(=O)CCC2CC2(F)F)c(Cl)cccc1Cl 92990,C(=O)(C(C)(O)C(C)(C)C)NCC(CN(C(=O)CSc1ccccc1[N+](=O)[O-])C)O 92991,Cc1cc(C(=O)NC2CN(C(c3cncnc3C(C)C)=O)CC2O)c(C)s1 92992,n1(CCc2cccc(C(=O)OCC)n2)nc(C)c(C)c1C 92993,N1(C(C#CCNC(C2(C)CCCO2)=O)=O)CCCc2occc2C1 92994,N1(C(C2(CCC)CCNC2=O)=O)CCC(CNC(=O)C(CC)SC)(COC)CC1 92995,c1(C(C(=O)NCC2CN(C(C(c3ccc(F)cc3)OC)=O)C2)C)cccc(F)c1 92996,c1(C(N2C(CC)C(C(=O)N(C)CC3CCCC3)CC2)=O)cnn2c1CCC2 92997,N1(C(Cn2ncn(C)c2=O)=O)CCCC1C1CCCN1C(=O)OC(C)(C)C 92998,c1(C(=O)NCC2C(CC(=O)NCC(CC3CC3)OC)C2)ccn(CC)c1C 92999,C1(NC(c2cnc(OCC)s2)=O)CN(C(c2ccn(CCF)n2)=O)CCC1CO 93000,C12(C(N3CC(C(C)NC(=O)CCCN(C)C)C3)=O)CCCCC1C2 93001,Cc1c(CNC(=O)C=CCC(C)(C)NC(=O)Cc2cccnc2O)nnn1C 93002,C1(NC(c2ccc(C(C)C)s2)=O)CCC(NC(=O)CCC2CCCCN2C)CC1 93003,N1(c2nccc(N3CCC(C)CC3)n2)CC(NC(c2ccc(F)s2)=O)CCC1C 93004,N1(C(CC2(C)CCCO2)=O)CC2CCCC2(NC(c2cc[nH]c2C2CCC2)=O)C1 93005,N#Cc1cccnc1-c1nnn(-c2cc(CO)n(CCO)n2)n1 93006,c1(CO)ccc(-c2cc(CNN(CC(C)O)Cc3cccs3)ccc2C)cc1F 93007,C1(CNC(c2ccncc2)=O)CCC(C(=O)NC2CC2c2ccccc2)CC1 93008,c1(OC)csc(C(c2nnnn2Cc2cccs2)NCCCF)c1OC 93009,C1(NC(CSCC=C)=O)CN(C(=O)C(CO)OC)CC1(C)C 93010,C1(C(=O)NC(CNC(c2ncnc(C)c2C)=O)C(C)(C)C)CCCC(F)(F)CC1 93011,C(=O)(C(C)(F)C(F)(F)F)NCC(C(C)C)NC(c1cc(N)ccn1)=O 93012,c1(C(N2C(CCCNC(C3(C)CC3(Cl)Cl)=O)CCC2)=O)ncc(F)cn1 93013,C1(CC)CN(C(C23CCC(F)(CO2)C3)=O)CCN1C(c1ccc(NC=O)cc1)=O 93014,c1(OC)cc(O)c(NC(c2ccnn2CC2(C)COC2)=O)cc1C 93015,N1(S(CCOCC)(=O)=O)CCN(Cc2ccc(Cl)nc2OC)CC12CC2 93016,c1(C(N2CC(C(N)=O)(CNC(=O)C3=CCCCC3)C2)=O)nc[nH]c2ncnc1-2 93017,c1(C(N(CCCNC(C2CC(O)C2)=O)C)=O)ccc2c(N(C)C)ncnc2c1 93018,c1(C(=O)NCC(C)N(C(C(C)OC)=O)C)c2c(c[nH]c1=N)CCC2 93019,C1(NC(c2ccc(C(F)F)c(F)c2)c2n(CCCF)nnn2)Cc2cscc2C1 93020,N1(C(c2c(NCC)scn2)=O)CC(NC(=O)CCOc2cccnc2)C2CC12 93021,C=CCC(C(=O)NCCCCNC(c1cnn(C)c1Br)=O)NC(C)=O 93022,C1(COCC)(CN(C(=O)NCC2CC(F)C2)C)CCOCC1 93023,C12(C(=O)NC(CC)CNC(=O)CNC(C3CCCC3)=O)CCCC1C2Br 93024,C1(NC(C(C)OC)=O)(CNC(c2cnnn2C(C)C)=O)CCC(F)(F)CC1 93025,C(CCCCC(=O)N1CCC(NC(c2cn(C)c(C)n2)=O)CC1C1CC1)SC 93026,N1(C(C(C)C(C)O)=O)CCC2(CC1)CC(NC(=O)Cn1ncccc1=O)C2 93027,c1(C(N2CCN(C(CCC#C)=O)C(C)C2)=O)nccc2ccn(C)c12 93028,c1(OC)c(C(N2CC3CCC3(NC(=O)CC3(C4CC4)CC3)C2)=O)c(C)nn1C 93029,C1(C(=O)Nc2c(C)cc(NC(C34CC(C)(CO3)C4)=O)cc2)CCCC(F)(F)CC1 93030,c1(C(N2CCN(CCNC(C=CCC)=O)CC2)=O)cc(S(=O)(=O)NC)cs1 93031,C1(CNC(C(C)c2ncco2)=O)COCCN1C(c1sccc1Br)=O 93032,C(=O)(CC1=CCOCC1)NCC(CC(C)C)(C)NC(=O)Cn1ncnn1 93033,CC1(NC(=O)C(Cl)Cl)CCCCC1C(=O)NCCN(C1CCC1)C 93034,c1(C(=O)NC(CN(C(C(CC)NC(C)=O)=O)C)C)cccc(OC(F)(F)F)c1 93035,N#Cc1ccc(C(=O)N(CCCNC(c2cccn(O)c2=O)=O)C2CC2)cc1 93036,Cn1ncc([N+](=O)[O-])c1C(=O)NCCC(C)(C)NC(C1CC1c1cccnc1)=O 93037,N1(C(C=Cc2c(C)ccnc2)=O)CC2CCC1CC2NC(C1CC12CCOC2)=O 93038,C1(CC(C)NC(c2nc(C)[nH]n2)=O)CCN(C(=O)C(CO)NC(=O)C(C)C)CC1 93039,c1(SCC)ccc(C(N2CC(NC(C3(C4CCCCO4)CC3)=O)C(O)C2)=O)cc1 93040,Cc1ncc(C=CC(=O)NCC2(F)CC(NC(=O)CC(=O)N(C)C)C2)c(O)n1 93041,N1(C(CC2C(=O)NCCC2)=O)Cc2occ(C(N3CCC3C3CCC3)=O)c2C1 93042,C1(C(F)(F)F)(OC)CC(CO)CN(S(=O)(=O)CCCC#N)C1 93043,C1(C(N2CC(O)(CNC(=O)Cc3cc(Cl)sc3Cl)C2)=O)CNc2ccnn2C1 93044,CCCCC(CC(=O)NC(C)CCF)NC(=O)CC1CC2CCC1O2 93045,C(=O)(C(C)(C)CCCNC(C1CCCN(C)C1)=O)NCc1ccc(CC)o1 93046,c1cc(-c2cnc3cccnn23)c2c(c1)CN(c1ncnn3cccc13)CC2 93047,Cc1c(C(N2CCC(CNC(=O)C(C3CCOCC3)C)CC2)=O)cccc1O 93048,CON1CCC(C(=O)NC23CC(NC(C4CC5CCC4CC5)=O)(C2)C3)CC1 93049,C1(C(=O)NC2(CC=C)CN(C(=O)Cn3nc(C)cc3N)C2)CC(=O)N(CCC)C1 93050,c1(C(=O)NC23CC(NC(CC4(C=C)CCOCC4)=O)(C2)C3)ccc2cnoc2c1 93051,c1(C(=O)NCC(CCNC(C2(OC)CCCOC2)=O)O)cnc(C(F)F)c(C)c1 93052,Cn1cnc2c1CN(C(=O)COC(C)(C)CNC(c1ccc(N)c(F)n1)=O)CC2 93053,c1(CC)ccccc1OCCC(=O)N1CC(CNC(=O)C=Cc2csc(C)n2)C1 93054,N1(C(Cc2n(C)cnc2)=O)CC2CC(NC(c3ccc4nnnn4c3)=O)CC2C1 93055,c1(CC(=O)NC2(C)CC(NC(CCSCC)=O)C2)ccc(F)cc1F 93056,C1(C#C)(C(N(CCN(CC#C)C)CC)=O)CCN(C(C2CC2F)=O)CC1 93057,c1(CNc2cc(NCC(c3ccccc3F)C)ncn2)cccc(O)c1Cl 93058,C(c1cnn(C)c1)=CC(=O)OC.N1CC(CCNC(=O)CC2CCC2)C1 93059,c1(CC)cccnc1C(=O)N(C(C)CNCc1cccc(OC(C)=O)c1)C 93060,CC(C)(C(=O)NC1CC1CNC(C1CNC(=O)C1)=O)c1cscc1Cl 93061,c1(CNC(c2c(C(C)C)n[nH]c2)=O)cccc(NC(=O)CCc2cnccn2)c1 93062,c1(CNC(=O)NC23CCC(C(=O)OC)(C2)CO3)cccc2c(Br)ccnc12 93063,CC(CF)CC(=O)NC1CCCC1NC(C1(O)CCOCC1)=O 93064,C(=O)(C1=COc2ccccc2O1)NC1CC(NC(CCCC#C)=O)C12CCC2 93065,CCC(CC)C(=O)N1CCC(F)(CNC(C2CC2c2ccn(C)n2)=O)C1 93066,C(CC(C(C)(C)C)NC(=O)C=Cc1cocn1)N(C)C(C1CC(=O)CC(=O)N1)=O 93067,C(=O)(C#CC1CCCCC1)N1CCC(C(C)NC(C2(C#N)CCCO2)=O)CC1 93068,c1(C(=O)O)ccc(S(=O)(=O)NC2CC3(COC3)C2)c(Cl)c1 93069,c1(C(N(CCNC(C2(CC#C)CCOC2)=O)CCC)=O)cc(Cl)c(Cl)cc1O 93070,C(N=c1[nH]c(C)c(C(N2CCC(CCCO)CC2)=O)s1)c1ccc(C)c(Cl)c1 93071,CC1C(NC(c2ccn(CCF)n2)=O)CCN1C(C1C=CCS1)=O 93072,C12(C(=O)NC3C(SC)CN(C(=O)CC4=CCCC4)C3)CCCC(C)(C1)OC2 93073,N1(CC2(OC)CCCC2)CCCC(CNc2cc(OCC(F)F)ccn2)C1 93074,C(=O)(CCCC(C)NC(c1[nH]ccc1C1CC1)=O)NCC(C)NC(=O)OC 93075,CC1CCC(CNC(C)(C)C(=O)NCCCNS(C)(=O)=O)C1 93076,C(=O)(C(CC(F)F)C1CCC1)NC(CNC(=O)COc1cccc(F)c1F)CO 93077,C1(NC(c2ncn(CC)n2)=O)C2CC1N(C(C1(C3CCCCO3)CC1)=O)C2 93078,C12(NC(c3snc(O)c3Cl)=O)CCC1CN(C(=O)CCOc1cccnc1)C2 93079,N#Cc1ccc(CCC(=O)OCCc2cccc3sccc23)c(F)c1 93080,CC1=NOC(C)(C(=O)N(C)CC2CN(C(C3COC(C)(C)O3)=O)CCO2)C1 93081,N1(C(c2ccnc(Cl)c2)C(=O)NCC2CC2)CCC2(CC1)OCc1ccncc12 93082,N1(C(C(CC)C(C)C)=O)CCCC2C1CCN2C(c1cc(F)c(F)cc1O)=O 93083,c1(C(N2C3(CNC(CC(C=C)C)=O)CCCC(C2)C3)=O)ccc2oc(C)nc2c1 93084,C(=O)(CS(=O)(=O)CC(C)C)NC(C1(O)CCN(C(C(CC)C)=O)CC1)C 93085,S(=O)(=O)(c1cnc2ccccn12)NCC1(CC)CCOCC1 93086,N1(C(c2cnc(CC)[nH]2)=O)CC(C)N(C(=O)Cc2coc3ccccc23)CC1C 93087,Cc1noc(C)c1CCC(=O)NCC1(F)CN(C(=O)COCC2CCCC2)C1 93088,N1(C(COC(CC)(C)C)=O)C2CCC1C(NC(=O)CNC(=O)NC)C2 93089,c1(C(=O)NCCC(=C)CNC(=O)C(C)Oc2ccc(SC)cc2)csc(C#N)c1 93090,C1(NC(C2CC(=C)C2)=O)CS(=O)(=O)C2CN(C(c3nnn(C(C)C)c3C)=O)CC12 93091,C(=O)(C(CC1SCCS1)NC(=O)OC(C)(C)C)N1CC(C(=O)OC(C)C)C1 93092,C(CN=c1ccn2c(Br)cnc2[nH]1)C1(OC)CN(C(c2cn(C)nc2OC)=O)C1 93093,N1(C(C(CC#C)C2CC2)=O)C2CCC1CN(C(=O)C(C)C1CCC1)C2 93094,CCCC(O)C(=O)NC(C(N1CCC(CN(C)C)C1)=O)C1(C)CC1 93095,N1(C(C(C=C)OC)=O)CCN(C(c2c(COC)cccc2F)=O)CC1C1CC1 93096,c1(OC)ccc(CN2CCC(CC(N3CCCC3C(N)=O)=O)C2)c(Br)c1 93097,C1(CNC(c2n(CC)cnn2)=O)CCN(C(=O)CC23CCCC2C3)C1(C)C 93098,c1(CC(N2CC(NC(C3CCC3)=O)C3C2C3)=O)cc(F)cc(Br)c1 93099,CCC(O)C(C)(C)C(=O)N1CCC(CNC(=O)CCCN=[N+]=[N-])C1.n12cc(nn1)C2 93100,S(=O)(=O)(CC(=O)N1CCCC(N(C)C(C2CCCCN2CC(F)F)=O)C1)NCC 93101,CC1(C(N2CCC(CNC(C3(CF)CCOCC3)=O)C2)=O)CC=CCO1 93102,c1(CC(=O)NCC2CN(C(CN(C)C)=O)C2)csc(NC=O)n1 93103,Cc1ncc(Br)cc1C(N1CC(N(C(=O)CC2CCC(C)(C)C2)C)C1)=O 93104,c1(CNC2CC(C(N3CCN(CC#C)CC3)=O)C2)cccc2nc[nH]c12 93105,Cc1cc(N)cc(C(=O)NCC(c2ccccc2F)OC2CC2)c1F 93106,c1(C(C)C)cccc(C(N2CCCCC2CNC(=O)C(C)(C)c2cscn2)=O)c1 93107,C(CN=c1[nH]c(=NCC2CCCN(CC(F)F)C2)[nH]c2c1COC2)OCCO 93108,c1(C(N2CC(CNC(c3n(CC)ncn3)=O)C2)=O)cccc(OC(F)(F)CF)c1 93109,N1(C(C2CCCC2)=O)CCN(C(=O)C=CC2CCCCC2)C(c2ccncc2)C1 93110,c1(C(=O)NC2CN(C(C3(C#C)CCCC3)=O)CC2O)ccc(Cl)c(C)c1Cl 93111,N1(C(C(C)SCC)=O)CC(CNC(=O)Cc2ccc(C)c(OC)c2)C(F)(F)C1 93112,C1(C(=O)NC2C(CNC(=O)Cn3cnc([N+](=O)[O-])n3)C2)CCC2(CCCCC2)C1 93113,c1(OC)ccc(O)c(C(=O)NC2CC(CCNC(C3CC3Br)=O)C2)c1 93114,c1(C(N2CC=CC(NC(Cc3ccc(C)cc3Cl)=O)C2)=O)c(C)cc(O)nc1C 93115,N1(C(c2c(C)noc2)=O)C2CCC1CN(C(=O)C(C)CC1CCCO1)C2 93116,O(NC(=O)CC(C)NC(C1CCCN(C(C)C)C1)=O)CCOC(C)C 93117,N1(C(C2ON=C(C)C2)=O)CCCN(C(c2nc(=N)cc[nH]2)=O)C(CO)C1 93118,C1(NC(c2csc(C)c2N)=O)CC2(C1)CC(NC(=O)C(C)NC(=O)C(C)(C)C)C2 93119,C=C(C)C(CC(=O)N1CCCC(N(C(C)C(=O)N(C2CC2)C(C)C)C)C1)OCC 93120,c1(C(=O)NC(C(C)NC(=O)COc2ccc(O)cc2)C)c[nH]c2cc(Cl)ccc12 93121,CCC(CCOC)C(=O)N1CCOC(CN(C(=O)C#CC(=O)N(C)C)C)C1 93122,c12nc(C)ccc1C(=O)N2.c1(OC)cc(C(=O)N(C2CCCCC2)C(C)C)sn1 93123,Nc1nonc1NC(C1C(C2CN(C(CNn3ccnn3)=O)C2)C1)=O 93124,N1(C(CCn2cc(-c3ccc(C)c(F)c3)nn2)=O)CCCC2(C)CCCC12 93125,CC1OCCN(C(C2CCN(C(c3ccco3)=O)C23CC3)=O)C1C 93126,N1(C(CCSCCCC)=O)CC2CCCN(C(c3ncoc3C)=O)C2C1 93127,C1(NC(CC2C(C)(C)C2)=O)CC2(CCCN(C(c3c(Cl)csc3Cl)=O)C2)C1 93128,c1(N(C)CC)ccc(CN=C(NCC(C)(C)C)NC2CCC3CCC23)cn1 93129,c1(C(=O)NC2C=CC(CNC(C3CN(OC)C(=O)C3)=O)C2)ccn2c1CCCC2 93130,Cc1cccc2[nH]cc(C(N3CC(C)(NC(C4CCC(C5CC5)C4)=O)C3)=O)c12 93131,N1(C(C(C2CCC(C(C)(C)C)CC2)O)=O)Cc2ccccc2CC1c1ncc[nH]1 93132,c1(CC)ccc(F)c(C(=O)NCC2COCCN(C(=O)CC(C)C(F)F)C2)c1F 93133,C(=O)(C1CSc2ccccc21)N1CC(OCCNC(C2CN3CCN2CC3)=O)C1 93134,C1(CNC(C2(C)CC3CC3C2)=O)CC(C(F)(F)F)CCN1C(=O)CCCN=[N+]=[N-] 93135,C(=O)(C1=NN(C2CC2)C(=O)CC1)N1CCC(O)(CN(C(=O)Cc2ccon2)C)C1 93136,C(C(C(=O)NCc1nccn1CC)C(C)(C)C)NC(c1oc(CC)c(C)c1)=O 93137,N1(C(c2c(CC)[nH]nc2Cl)=O)CCC(NC(=O)CCn2ccnc2)C(C(C)C)C1 93138,CC(C)(C(=O)N1CCC1NC(=O)CN1C(=O)NC(C2CC2)(C2CC2)C1=O)C(F)F 93139,C(=O)(CCCC1CCCC1)N(C1CCN(C(=O)C(C)(C)F)C1)C.C1CCOCC1 93140,N1(C(=O)C2CC2)CCC(F)(c2cn(-c3cccc(Cl)c3Cl)nn2)CC1 93141,c1(NC(C2CCN(c3cc(OC)nc(OC)n3)CC2O)=O)ccc(C#N)nc1C 93142,N1(C(c2cnc(C)nc2C)=O)CCCC2(CCN2C(=O)C(c2ccccc2)O)C1 93143,CCC(O)C(C)(C)C(=O)NCC(C1CCC1)NC(c1ncc(OC)cn1)=O 93144,c1(C(=O)NCC(CCNC(c2ccc(C#C)cc2)=O)O)c(C)cc(C)cc1C 93145,c1(OC(C)C)cccc(C(=O)NCCCC(C)(C)NC(C2CC2Br)=O)c1 93146,C1(CNC(C(C)NS(C)(=O)=O)=O)(CO)CCN(C(=O)CN2CCC2C)CC1 93147,N1(C(c2nc(C)nn2C)=O)CCC2OCCN(C(=O)Cc3sc(C)nc3C)C2C1 93148,Cc1cccnc1C(=O)NC1(C2N(C(=O)CC3CCCN3C(C)C)CCC2)CC1 93149,c1(OC)cccc(Br)c1C(N1CCC2(CC2C(=O)NCC(C)O)C1)=O 93150,CCCCC(O)C(=O)N1CCCC1(C)CNC(=O)CCSc1n[nH]c(C)n1 93151,c1(C(N(C2CCCC2c2ccccc2)C)=O)cc(F)cc(F)c1O 93152,N1(C(c2c(C)cc(C)o2)=O)CCC(NC(=O)C(C)CN2CCOCC2)C12CC2 93153,C1(NC(c2cc(CSCC)on2)=O)CN(C(=O)C(C(C)(C)C)SCC)CCC1(C)C 93154,c1(N2CCN(C)CC2CNC(=O)CC2CC3CC3C2)cnc(C#N)c(C#N)n1 93155,S(=O)(=O)(c1ccc(C=CC(=O)OCC2=CCS(=O)(=O)C2)cc1)NCCC 93156,C(=O)(CCCC(=O)NC(C)C(CO)NC(C1NC(=O)OC1C)=O)NCCC 93157,c1(CC)nn(C)cc1C(=O)NCC(n1cc(CC2CCCCC2)nn1)C 93158,Nc1cccc(C(=O)NCCC2CCCCN2C(=O)CCC(=O)c2cccs2)n1 93159,c1(C(N2C3CC(NC(C4CCS(=O)(=O)N4)=O)C2CC3)=O)ccc2nnnn2c1 93160,C1(C(=O)NCC(NOC)=O)CN(C(=O)C(c2ccn(C)n2)C)CC12CC2 93161,c1(C(=O)NCC2(COC)CN(C(C3CN(C)C3)=O)C2)cc(Cl)cnc1OC 93162,c1(OCCC(=O)N(C2CCN(C(=O)C(F)OC)CC2)CCC)ccccc1F 93163,C1(NC(C2N(C(C(C(C)C)OCC)=O)CC(F)C2)=O)CC(C)(OC)C1(C)C 93164,C(=O)(CCC(C)(F)F)N1CCC(CN2CCN(C(C3C(C)OCC3)=O)CC2)CC1 93165,c1(C(N2CCC(N(C(=O)CSC(F)F)C)C2)=O)cc2cscc2s1 93166,c1(C(=O)NCCN2CCN(C)CC2)cc2ccc(Cl)cc2s1 93167,C1(C2CCCC2)(NC(C2C3CN(C(C(CCC)F)=O)CC32)=O)CCC1 93168,N1(c2nc(SC)c(F)cn2)CCC2(CCN(C(=O)CC(O)c3ccccc3)C2)C1 93169,c1(C(N2CCOCC(CNC(C(C)(O)C3CC3)=O)C2)=O)cccc2scnc12 93170,N1(C(C=CCC)=O)CCC2CCN(C(c3c(C)[nH]c4ccc(O)cc34)=O)CC2C1 93171,C1(C2CC2)(CNC(C(CCCC)C)=O)CCN(C(=O)C(F)OC)C1 93172,C(=O)(CC(C)(C)CNC(C1(C)CC(=O)C1)=O)NC(C(=O)N(CC)CC)C 93173,C1(NC(C(c2ncccc2F)C)=O)CCN(CC(O)COCc2ccco2)CC1C 93174,CC1OC2(C)CC1(C(=O)NC1CCN(CCOCC(F)(F)F)CC1)C2 93175,c1(CCC(=O)N(CCC(C)NC(=O)C(C)(C)c2cc[nH]n2)C)nnc(S)nc1O 93176,n1(Cc2c(C(N3CC(C)NCCC3)=O)cccc2)ncc2ncccc12 93177,Cc1ncc(N(C(=O)CCC2CCN2CC)C(=O)C=Cc2ccccc2)cc1Cl 93178,C(=O)(C(C)(C)Cc1ccccc1)NC1CC(N(C(=O)COCc2nccs2)C)C1 93179,Cc1ccc(C(=O)NCC2(C(C)(C)O)CN(C(C3CCOC3)=O)C2)nc1F 93180,c1(C(=O)NCC2N(C(C(C)CC3CCC3)=O)CCOC2)cc(Cl)nnc1O 93181,c1(SCC)cncc(C(N2CC(CCNC(c3cn(CC)nc3C)=O)C2)=O)n1 93182,C(=O)(CC1=CCN(C(=O)CN2CCCC2)CC1)NCCc1nccc(C)n1 93183,N1(C(CNC(c2c(C)ccs2)=O)=O)CC(CO)CC1C 93184,N1(C(c2c(C)cccc2C)=O)CC2CCC1C(CNC(C1CC(=O)N(C)C1)=O)C2 93185,C#Cc1ccccc1CNC(=O)C(=O)N(CC(c1ccc(Cl)c(Cl)c1)OC)C 93186,C=C=C(C)CC(=O)N1CCCC1CN(C)C(C1CC2(CSC2)C1)=O 93187,C(=O)(CC(CC(C)C)NC(=O)OC(C)(C)C)N1CC(CNC(C(C=CC)O)=O)C1 93188,c1(OC(C(N2C(C(C)NC(C(C)(C)OCC)=O)CCC2)=O)C)ccc(Cl)cc1 93189,c1(C(=O)NC2(COC)CCN(C(C3(C)CC3)=O)C2)ccc2c(c1)COC2(C)C 93190,c1(C(N2CCN(C(c3c(OC)c[nH]n3)=O)C(C)C2)=O)cn2nc(OC)ccc2n1 93191,CC1CCc2ncc(C(N3CC4CCC3CN4C(=O)C(C)C(C)(F)F)=O)n2C1 93192,C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)NC(CC)CNC(=O)CCOC(C)C 93193,N1(C(Cc2c(C)cnn2C)=O)CCCN(C(c2ccc(OC(F)F)cc2)=O)CC1 93194,C#Cc1ccccc1C(N1CC(CN(C)C(c2cnc(C)n2C)=O)C1)=O 93195,c1(OC)nccc(C(N2CC3(C2)CN(C(C2CCCCNC2=O)=O)C3)=O)c1F 93196,CCC(CNC(=O)C(CCOC)NC(c1ncc[nH]1)=O)(CC)C(N)=O 93197,c1(C(c2n(C(C)C)nnn2)NC2(CC3CCC(CO)O3)CC2)ccc(C#N)cc1F 93198,c1(C(N2CCCC(NC(C3CCC(C(N)=O)O3)=O)C2)=O)ccc2cccnc2c1 93199,C1(C(N2C(COC(C3(CO)CCCC3)=O)CCCC2)=O)CCc2[nH]nc(O)c2C1 93200,CCC(F)(F)CC(=O)N1CC(CO)(NC(C2CC2(C)c2cccs2)=O)C1 93201,C1(NC(C(N2CCCCCC2)C)=O)CC2CCC1N(C(=O)CCC(N)=O)C2 93202,C#CC1CCCN(C(c2c(C(N)=O)cnn2C)=O)C1 93203,c1(C(=O)NCC2(F)CCN(C(C(n3c(C)cc(C)n3)C)=O)C2)cc(C)c(C)nn1 93204,CN1CC(O)CC1(C)C(N1CC(O)(c2cn(CCN3CCOCC3)nn2)C1)=O 93205,CC(C)(C)S(=O)(=O)CC(=O)NCCC1CN(C(c2csnn2)=O)CCO1 93206,CC1OC2(C(=O)NCCCN(C(=O)CNC(C3CCC3)=O)C)CCC1C2 93207,N1(C(Cn2c(=N)[nH]nc2)=O)CC(NC(=O)C2=CCCSC2)CC12CCOC2 93208,N1(C(c2cn(C)c(Br)c2)=O)CC2CC(CNC(=O)C=C3CCOCC3)C2C1 93209,c1(NC(=O)NC(C)CCC(F)F)ncnc2c1CCCC2 93210,C(=O)(C(=O)CC(C)CC)N(C(CNC(C(CCCC)O)=O)CC)C 93211,N1(C(c2c(CC)n(C)nc2)=O)CCC2CCN(C(c3cscc3SC)=O)CC12 93212,c1(NC(C2C3CN(c4nc(C)cc(C)n4)C2C3)=O)nc(Br)cn2ccnc12 93213,N1(C(c2cn(C3(C(N)=O)CC3)nn2)C(=O)NC2(C)CC2)CCN(CCCF)CC1 93214,c1(CSC)ncc([N+](=O)[O-])cc1Br.C1CC(C)(O)Cn2ccnc21 93215,S(=O)(=O)(c1ccc(C(=O)NC2CCC(CNC(c3cncc(N)n3)=O)C2)o1)NC 93216,N1(C(C(c2ccc(OC(CC)C)cc2)OC)=O)CCC(O)C(C(=O)O)C1.C1CCCC1 93217,C(=O)(C(CN(C)C)CC)NC1C=CC(CC(=O)NCCCSCC)C1 93218,CC(C)(Cc1nn[nH]n1)C(=O)N1CCOCC1C(=O)OC1CCCCC1 93219,C1(NC(C(F)=CC)=O)CC(CNC(c2ocnc2C)=O)C1(C)C 93220,CC1(O)CCCN(C(=O)C(Cc2cnc[nH]2)NC(=O)CCN2CCCC2=O)C1 93221,C1(C(NOCCOCC)=O)CN(C(=O)C=CC(F)F)CC12CCC2 93222,N1(C(CC2CC(C)C2)=O)CCCN(C(c2ncc(F)cc2F)=O)CC1C 93223,C1(N(C(=O)CC2COC(=O)C2)C)CCCCN(C(C2CS(=O)(=O)C2)=O)C1 93224,c1(NCCCNC(=O)NC)ccc(S(=O)(=O)NC(C)CS(C)=O)cc1Cl 93225,c1(OC)cnnc(C(=O)NCC(C2CC2)NC(C2(OC)CCOC2)=O)c1 93226,C1(C(N2CC(C)(NC(C3N4CC(C)N(CC4)C3)=O)C2)=O)CCc2nnc(O)n2C1 93227,c1(C(=O)NCC(C(C)C)NC(C2CC3(C2)CC3(F)F)=O)cccc(C(N)=O)c1N 93228,c1(C(N(CC(CNC(C(=Cc2ccccc2)CC)=O)C)C)=O)cc(C)cc(Cl)n1 93229,C1(NC(N)=O)CCN(C(=NCc2ccc(-c3ccncc3)cn2)NCC(F)F)C1 93230,C1(F)(CNC(C(C)Cn2ccnc2)=O)CCN(C(=O)CN2CCCNC2=O)C1 93231,c1(CCC(=O)NCCC2N(C(C(C3CC3)SC)=O)CCC2)cccc(F)c1 93232,C1(C(=O)NC2(C)CN(C(CCC=C(C)C)=O)C2)CC(C(C)=NO)C1(C)C 93233,N1(CC)CCN(CC(N2CCN(C(=O)C(CN(C)C)NC(C)=O)CC2)=O)CC1 93234,c1(C(=O)NC2(CN(C(c3c(CC)oc(C)c3)=O)C)CC2)cnc(OC)c(Cl)c1 93235,C1(CCNC(CC=CC)=O)CC(F)(F)CN1C(=O)C(C)Oc1ccncc1 93236,C(C(N=[N+]=[N-])C(=O)N1CCOCC(NC(c2ccc(Cl)nc2Cl)=O)C1)OCC 93237,c1(CC)cnc(O)c(C(N2CCC(O)C(NC(C3SCC=C3C)=O)C2)=O)c1 93238,C1(c2noc(C)n2)(NC(C)=O)CCN(C(=O)C(C)NC(c2cccc(F)c2)=O)C1 93239,c1(CC(N2CC(NC(C(C(=O)OC)F)=O)C(OC)C2)=O)n[nH]c2c1CCCC2 93240,C1(O)(C(CC)C(=O)NC(CNC(C2CC2F)=O)Cc2ccccc2)CCCCC1 93241,C1(CNC(C2C(C)CC=CC2)=O)CC(C)(C)CN1C(=O)CCCSC(C)(C)C 93242,c1(CC(=O)NCCOC2CN(C(=O)Cn3nnnc3C3CC3)C2)ncc(Cl)s1 93243,C(=O)(CC(O)CCSC)NCC(CN(C(c1scnc1C1CC1)=O)CC)(C)C 93244,C1(OCC#C)CCCN(C(=O)Cc2nc(-c3ccc(F)cc3)oc2C)C1 93245,CC1(C)CC(O)C(O)CN(C(C2(c3cc(C(F)(F)F)cc(F)c3)CC2)=O)C1 93246,CC1CCC(NC(C2CC23CCSCC3)=O)CN1C(=O)CCN1CCCCC1 93247,c1(CN2CC(CC(N3CCC(O)(CC)C3)=O)C2)cc(Cl)ncc1C(=O)O 93248,c1(C(=O)NCCN2CCN(C(=O)COC3CCOC3)CC2)cnc2sccn12 93249,C1(NC(c2cc(C)[nH]n2)=O)CCCC1(C)NC(C1(c2cccs2)CC1)=O 93250,c1(CCNC(N(CCCO)C)=O)csc2ccc(Br)cc12 93251,N1(C(C2C(C)(C)C2)=O)CCC(O)(C2(NC(c3cc(C(N)=O)ccn3)=O)CC2)CC1 93252,C1(CNC(COCC)=O)CCN(C(=O)CCCCCOCC)CCC1(F)F 93253,C1(C(=O)N(C)Cc2cnco2)(COC)C=CCN1C(=O)CN1CCCC1 93254,c1(N(C(CNC(c2cc(CCC)[nH]n2)=O)C)C)ncnc(Cl)c1Br 93255,CONc1cccc(C(N2CCC2(C)CCO)=O)n1 93256,C=C(C)C1OCCCC1C(=O)NCC1C=CCN1C(c1ccnn1CC)=O 93257,C1(C(=O)NC(CC)CNC(c2snc(C)c2Br)=O)CC2(CCOCC2)C1 93258,c1(N(C)C)nc2ncnc(NC(C3CC(O)CN3C(=O)OC(C)(C)C)=O)c2s1 93259,Cc1cnc(O)c(CNC(=O)CC(C)N(C)C(C2CCCC(=O)CC2)=O)c1 93260,C1(O)(CNC(CSCC#C)=O)CCCN(C(=O)C(CC(F)F)c2ccccc2)C1 93261,c1(C(N2C(C)CC(NC(C=C(C)C)=O)C2)=O)ncnc2c1c(Br)cn2C 93262,N1(C(c2cc(NC)nc(Cl)c2)=O)CC2CCCN(C(c3cnsn3)=O)C2C1 93263,C1(CC)CN(C(c2cc(C)co2)=O)CCC1NC(=O)C(CC)c1ccccc1 93264,N1(CC2N(C(C3(N(C)C)CC3)=O)C(CC(=O)O)CC2)CC2CCCC(O)C2C1 93265,C1(N(C(C23CC(CCC)(C2)C3)=O)CC)CCCN(C(C2(O)CCSCC2)=O)CC1 93266,C1(NC(=O)C=C2CCCC2)CCCCC12CCN(C(C1(CF)COC1)=O)CC2 93267,C(c1cc(F)c(O)c(F)c1)=CC(N1CC2C(N(C(COC(CC)C)=O)C)C2C1)=O 93268,C1(OC)CCCC(C(=O)NCC(C)(C)CN(C(=O)CC2CC=CCC2)C)C1 93269,N1(CC(C)NC(C23CCC(CC2)O3)=O)CCN(C(c2cc(C(N)=O)c[nH]2)=O)CC1 93270,c1(C(=O)NCC#CCNC(c2cc(OC)no2)=O)cc(Br)c(C)nc1O 93271,c1(C(=O)NCC(C)(CC)NC(c2c(CC)cco2)=O)cc2oc(Br)cc2[nH]1 93272,c1(C(=O)NC(CC=C)CNC(c2[nH]ccc2COC)=O)cncnc1C 93273,N1(C(C(C=C)OC)=O)CCN(C(C2CC3CCCC3C2)=O)CC12CC2 93274,C=C1CCN(C(c2cc(CC)n(C)n2)=O)C(C(N2CCC(C)CC2)=O)C1 93275,Cc1cc(=NCCCOc2ccncc2)[nH]c(N2CC3COCC3(CO)C2)n1 93276,C1(NC(C2CC(=O)NC2)=O)CN(C(C2C=CCCC2)=O)C2(CCCCC2)C1 93277,C(=O)(C(O)C(C)(C)C)NC(CC#C)C(N1CCN(C(C)=O)C(C)C1)=O 93278,N1(C(C2CCN(C)C(=O)C2)=O)CCC2(CCCN2C(c2ccc(F)c(Cl)n2)=O)C1 93279,C1(CCNC(C2CCC(=O)O2)=O)CCN(C(=O)CC2CNC(=O)C2)CC1 93280,C1(SC)CCCC1N=c1cc[nH]cc1S(=O)(=O)NCc1csc(=N)[nH]1 93281,c1(C(N2C(CNC(CCCCOCCC=C)=O)CC2)=O)ccc(C)nc1O 93282,C1(CN(C(C2C(C)C2)=O)C)CN(C(=O)C(CO)c2ccccc2)CCO1 93283,CC(CC(N)=O)C(=O)N1CCCCC(NC(c2cc(-c3cccn3C)[nH]n2)=O)C1 93284,c1(OC)cc(C(=O)NC2CC(C(=O)NCCn3nncc3C)C2)on1 93285,c1(C(CC)(C)C)cccc(-c2nc(-c3occc3C)nn2CCF)c1 93286,C1(CCC#C)CCCN(C(C2COC(CNC(C3CSCC(=O)N3)=O)C2)=O)C1 93287,c1(OC)cc(N2CCCC(C(C)NC(=O)C(O)Cc3cnc[nH]3)C2)nc(C)n1 93288,CC(CCO)N=c1[nH]c2c(c(=NCC(CO)c3cccnc3)[nH]1)CCCCCC2 93289,C1(C(N(CC(C)(C)CNC(C2CN3CCC2CC3)=O)C)=O)CN(CP(C)(C)=O)C1 93290,c1(C(C)C)ccc(CCC(=O)NCC(CO)NC(=O)CCC2CCC2)cc1 93291,c1(SCC2N(C(C)(C)C)CCCC2)ncc(C=Cc2ccccc2)s1 93292,Cc1cccc(C(C#N)N(CC(=O)NC2C3CCCC23)Cc2ccccc2)c1 93293,C(=O)(C(C)CNC(=O)C(c1ccn(C)c1)C)NCCC(=O)NCC 93294,C1(C(=O)N)(C(n2cc(C(CCC)N(C)C)nn2)C)CCCCC1.C1CCCCC1 93295,C1(c2ccccc2)(C(=O)NC2(CNC(C3CC4CCCC34)=O)CC2)CC2(CC2)C1 93296,n1(CC(=O)NC2CN(C(=O)CCCC(F)F)CCC2F)cnc([N+](=O)[O-])c1 93297,C1(C(=O)NCC2OCCN(C)C2)COC2(C1)CN(C(c1cccnc1I)=O)C2 93298,C12(C(=O)NCC(=C)CCNC(=O)C=CBr)CCC(CC1)C(C)O2 93299,C1(C(=O)NCc2cccc(Oc3c(C)cccc3)c2)CCC(C2CCCO2)O1 93300,N1(C(C(C)OCCOCC)=O)CC(NC(C2CC2C(C)(C)C)=O)C(F)C1 93301,C1(CC(=O)OC)COC(C(F)(F)F)CN1Cc1ccc(-c2nnn(C)n2)cc1 93302,C1(C(=O)NCC(CNC(CCCC(C)(F)F)=O)O)CCS(=O)(=O)C12CCC2 93303,c1(C(N2CC(CNC(c3cc(C(C)=O)[nH]n3)=O)C2)=O)cc(OC(C)(C)C)ccn1 93304,C1(CNC(c2cc(CC)no2)=O)CCCCN1C(=O)Cc1ccccc1CC 93305,CN(C)C1CCc2cc(NC(c3ccc(F)cc3)c3nnnn3CSC)ccc21 93306,c1(C(C)=O)ccc(C(N2CCC(n3cc(COCCN(C)C)nn3)C2)=O)nc1 93307,C1(O)(CCNC(CC2CN(C)C2)=O)CN(C(c2ncoc2Br)=O)C1 93308,c1(OC(C(=O)NCCN(C(c2n(COC)ncc2)=O)C)C)ccc(Cl)cc1 93309,C1(NC(C(C2CC(F)(F)C2)OC)=O)CC12CCN(C(c1cc(C(C)C)sn1)=O)C2 93310,C(=O)(C(C(C)C)n1cnnc1)N1CC(OC(=O)Nn2cc(C(=O)OCC)nn2)C1 93311,C1(NC(C)=O)CC(=O)N(C2CN(C(=O)C(N3CCOCC3=O)C)C2)C1 93312,C(=O)(C(C)(O)CCC)NCC(C)(C1CC1)NC(c1c(CCC)n(CCO)nc1)=O 93313,Cc1nc(C)n(CC(=O)NCC2CCCC2NC(c2nn(C)nc2C(F)(F)F)=O)n1 93314,c1(C(N2CC3(CN(C(CCC(=C)C)=O)C3)C2)=O)cnn2c1OCCC2 93315,Cc1cc(C)c2c(c1)CCC2NC(=O)N=S(C)(=O)C1CCCCC1 93316,Cc1cn2cc(C(=O)NC3CCN(C(c4cc(CO)c(C)o4)=O)CC3F)nc2s1 93317,N1(C(c2cccc(CC=C)c2)=O)CCN(C)C(=O)C1 93318,c1(C2(C(N3CC(O)(CNC(=O)C(F)F)C3)=O)CC2)ccc(Br)cc1F 93319,Cc1cc(C(=O)NCCCN(C)C(c2ccc(-c3cc[nH]n3)s2)=O)cc(C)c1O 93320,c1(C(N2C(CNC(c3c(CC)non3)=O)C(C)CC2)=O)ccc2c(c1)CC2 93321,N1(C(CC2(COC)CC2)=O)CC2CCC1C1CN(C(C3CCC34CCC4)=O)CC21 93322,c1(C(=O)NCCN(C(CC(C)OC)=O)CC(C)O)n[nH]c(C(C)C)c1[N+](=O)[O-] 93323,c1(C(=O)NCCC2N(C(CC(C=C)C)=O)CCOC2)c[nH]c2c(F)cccc12 93324,c1(CC)ccccc1C(CNC(C1C2CC3C(C2)C13)=O)NC(c1csc(=N)[nH]1)=O 93325,CC1COCC(CNC(=O)CCCCN(C(=O)C=C2CCCCC2)C)O1 93326,CCCC(C(O)C(=O)N1CCC=C(C)C1)NC(=O)C(COC)N(C)C 93327,N1(CCN(C(Cn2cc(CC(=O)NC3(C)CCOCC3)nn2)=O)O)CC(O)CCC1=O 93328,Cc1ccccc1OCCC(=O)NCC(C)(C1CC1)NC(C12CCN(CC1)C2)=O 93329,c1(OC)c(C(=O)N(CC(C)NC(c2csc(C)c2C)=O)C)sc(Cl)c1Cl 93330,N1(C(CCCN(C(C)C)C)=O)C(C(=O)NC2(CC3CC3)CCC2)CCC12CC2 93331,c1(NC(c2nnnn2C(C)(C)C)(CC2(OCC)CCC2)C)cc(C)cc(Br)c1C 93332,C1(CN(C(CC=C)=O)C)CCN(C(C2OCC2(C)C)=O)CC1 93333,CC1(C)CN(C(=O)CCSC2CCCC2)CC1CNC(C1(C)CNC(=O)C1)=O 93334,N1(C(C=CSC)=O)CCC(C2CCN(C(C3OCCO3)=O)CC2)C1 93335,c1(C(N(C2CCC(NC(C(C(=C)C)(C)C)=O)C2)C)=O)ccc(C#N)cc1O 93336,N1(C(C2N(C)CCC2)=O)CC2CC1CN(C(c1nccc3nn[nH]c13)=O)C2 93337,c1(C(=O)NCCN(C(=O)CN=S(C)(C)=O)C)cc2ccccc2c(O)n1 93338,CCCCC(C(=O)NCC1CCC(C(=O)N(CC(C)(C)O)C)C1)C(C)C 93339,S(=O)(=O)(c1cccc(Cl)c1Br)N(CC(F)F)C 93340,Cc1c(C(=O)NC(C)CCNC(=O)C(C)(C)N(C)C)cnn1CC(C)(C)O 93341,N1(C(COC)=O)CC2COCC(C1)C2NC(=O)CCc1cncc(F)c1 93342,CCCCCCOC(C)C(=O)NCCC1(O)CN(C(C2CCN(CC)C2)=O)C1 93343,c1(OCC)ccc2nc(NC3CN(C(c4ccc(C)c(I)c4)=O)C3)sc2c1 93344,C1(NC(Cc2cc(C)on2)=O)CN(C(c2sc(CC(C)C)nc2C)=O)CC1C 93345,Cc1cc(N2CCC(C)C(NC(c3ccc(C)s3)=O)C2)c(C#N)cn1 93346,C1(OC)CCC(N(C)C(c2c[nH]nc2CNC(C2CCC(C)(C)C2)=O)=O)CC1 93347,C1(Nc2c(NS(C)(=O)=O)ccc(C)c2)CCc2nnc(O)n2C1 93348,C=C1c2ccccc2C(=O)N1CC(=O)NC1CC(C)N(C(c2cc(OC)n[nH]2)=O)C1 93349,Cc1cc2[nH]c(C(=O)N(C3CC3)CC3CCCN3C(=O)C=CI)cc2s1 93350,C1(C)(C(=O)NC(CC)COC)CCCN1C(=O)CC1CCOC1=O 93351,C(=O)(C1CCc2c(Cl)cccc21)N1C(CNC(C(C)S(N)(=O)=O)=O)CC(C)(C)C1 93352,C1(O)(C(=O)NCC2(NC(C3CC(=C)C3)=O)CC2)CC2CCC1C2 93353,C(=O)(C1COc2ccc(Cl)cc21)NC1(CCOC)CCN(c2cc(O)ncn2)C1 93354,C=CCC(C(=O)N1CCC(CCNC(=O)COCCCC(C)C)C1)C(C)C 93355,CC(C)P(=O)(CC(=O)N1CC(NC(=O)CCCC(N)=O)CC1C)C(C)C 93356,C(=O)(C(O)CC(F)(F)F)NC(C(C)(C)NC(CSc1c(OC)cccc1)=O)C 93357,N1(C(C(COC)N(C)C)=O)CC(NC(c2cc(OC)nc(C)c2)=O)CCC1C 93358,C(=O)(C(C)S(N)(=O)=O)NCC1C(C(=O)NCCCCC2C(C)C2)OCC1 93359,c1(C(N(C2CCN(C(=O)C(O)CC(C)C)C2)CCC)=O)cc2nc(F)ccc2o1 93360,c1(CC(=O)NCCN(C(=O)CC(C)OC)CC)cccc(OC(C)C)c1F 93361,N1(C(C(C)NC(CC)(C)C)=O)CCC=C(C(=O)Nc2n[nH]c3c2CCCC3)C1 93362,c1(N(C)CCN(S(C)(=O)=O)C)nc(N(C2CN(C)C2)C)nc2ccc(Cl)cc12 93363,C=CC1OCCC1NC(=O)CC1CCN(C(=O)Cn2ccc(C)c2)CC1 93364,CCC(CC)CCC(=O)N1CC(OC)CC1(C)CNC(C1(c2ccsc2)CC1)=O 93365,O=C1CC2C(C(=O)NC3CC(=O)N(C4CN(C(=O)CCc5nncs5)C4)C3)C2C1 93366,CC(C)(C#N)CCC(=O)NC1CC(C)(NC(c2ccn3cccc3c2)=O)C1 93367,c1(C(=O)NCC(CNC(C(C(=C)C)(C)C)=O)C)ccc2c(O)nccc2n1 93368,C1(F)(CNC(C(C)OCCC=C)=O)CCC(CNC(=O)C(C)SC)CC1 93369,C12(NC(=O)CC3(CO)CC3)CCCCCC1N(C(=O)CSCc1ccccn1)CC2 93370,c1(NC(=O)CO)cccc(C(N)=O)c1.C12CCN(CC1)C(=O)CCN(CC)C2=O 93371,Cc1cnc(C(N2CCCC(N(C(=O)COC(F)F)CCF)C2)=O)cc1C 93372,O=C1CCC2(C(=O)OCC3OCCCO3)CCCC2C1 93373,c12ccccc1CC(=O)N2.C(=O)(C(C)CC1CC1)NC1CC(OC(C)C)C1 93374,C1(N(C(=O)NCCCCSC)C)CCCN(Cc2ccccc2)C1C 93375,C(=O)(C1=NOC2(CCC2)C1)NC1C(NC(c2ccc(C(N)=O)c(Cl)c2)=O)C1 93376,C12(CNC(C(C)CN(C)C)=O)CCC(NC(C34CCCC3CC4)=O)(CC1)CO2 93377,c1(C(N(C)CC2N(C(CCCCC#C)=O)CCC2)=O)cc2ccccc2nn1 93378,C1(NC(CN(C2CC2)CC)=O)CCCN(C(=O)C(=O)NCC(F)(F)F)C1C 93379,c1(COC(Cc2cn(C(C)(C)C)nc2)=O)ccc(Br)c2cccnc12 93380,N1(C(CCN(CC#C)C(C2COC(C)C2)=O)=O)CCOC(CN=[N+]=[N-])C1 93381,CC(C)CC(CNC(c1cnc(-c2ccccn2)nc1)=O)NC(=O)C1=NOCC1 93382,N1(C(C(CSC)(C)C)=O)CCC(F)(F)C(CNC(=O)CC2CC2(C)C)C1 93383,N1(C(CSCC)=O)CCCC12CCN(C(c1nccn3cnnc13)=O)CC2 93384,c1(N2CCC(S(N)(=O)=O)C2)ncc(S(=O)(=O)NCCc2c[nH]c(=N)s2)cc1Cl 93385,N1(C(CSC)=O)CCC(C)(C)C1CNC(=O)CC1CCC1C 93386,c1(C(=O)NC2C=CC(CNC(C3(CC#C)CCOC3)=O)C2)cc(Cl)cn1C 93387,CN(C)S(=O)(=O)NCC(N1CCC(O)(CCNC(=O)C=C2CCN(C)C2)C1)=O 93388,c1(C(=O)O)ccc(CNCC23CC2CN(C(c2ccc(Cl)cn2)=O)C3)c(Br)c1 93389,c1(CC)[nH]ccc1C(=O)NCCn1cc(C(=O)N(CC(C)CO)C)cn1 93390,C1(NC(COCCC)=O)CN(C(C2CCC(CC)O2)=O)CC2(CCOCC2)C1 93391,c1(C(=O)NC2CC(CNC(c3nn(CC)c(C)c3)=O)C2)cccc(C(C)C)c1N 93392,N1(C(C2(C(C)C)COC2)=O)CCC2(CC2C(N2CCCCC2C2(O)CC2)=O)C1 93393,C(=O)(C(Cn1cncn1)NC(c1ccn(C)n1)=O)NCCCOC(C)C 93394,N1(C(c2ccc(CN=[N+]=[N-])cc2)=O)CCC2(CC1)CC2NC(=O)C(N)=O 93395,C1(CNC(c2cc(COC)no2)=O)C(C)CCN1C(=O)CSc1c(C)n[nH]c1C 93396,Cc1cc(C#N)nc(=NCC2CCNC2(C)C)[nH]1 93397,C1(CC(=O)N(CC(=O)OC)C2CC2)CN(C(=O)CCCC2CC2)CCC1C 93398,CC(C(O)C(F)F)NC(c1ccc(CNC(=O)C=CC2CCCCC2)cc1)=O 93399,C(=O)(C(C)CC#N)NC(C(C)c1ccccc1)Cc1ccccc1 93400,C1(C2CN(C(=O)CCc3nc[nH]n3)C2)(NC(=O)C(F)=CCCF)CC1 93401,c1(OC)nccc(N(C)C(=O)NC23CC(NC(=O)OC(C)(C)C)C(C2)C3)n1 93402,C1(CC(=O)NC2CN(C(=O)CC3CS(=O)(=O)C3)C2)CCCNC1=O 93403,CS(=O)(=O)c1cccc(CN2CCCC(CNC(c3cccc(Cl)c3Cl)=O)C2)c1 93404,c1(OC)cccc(C(C)CC(=O)NCC2CN(C(c3nc(O)sc3C)=O)C2)c1 93405,c1(OC)c(Cl)ccc(C(=O)NC(CNC(=O)CCc2cnn[nH]2)C(C)(C)C)c1F 93406,C1(C(=O)NC2C(CNC(C(CC)=CC)=O)COC2)CCC(N(C)C)CC1 93407,N1(C(C2(C)CC3(CCC3)C2)=O)CC2(CCN(C(C3CCC4CC4CC3)=O)CC2)C1 93408,c1cccc(F)c1.C1(C=O)C2CC3C(C2)C13.C1(=O)CN(C)N(C)CCN1 93409,CCCC(C)CC(=O)N(CCC(=O)NCCCN(C)C1CC1)CCO 93410,Cc1cc(F)ncc1C(=O)NC1(C(F)(F)F)CCN(C(=O)OC(C)(C)C)C1 93411,N1(c2nc(OC)c(Br)cn2)CC2(CCC2)CC1CNC(=O)Cc1coc(C)n1 93412,CCC(C)(C)C(=O)NC1CCOCC1NC(C1CC1C(C)(F)F)=O 93413,c1(C(=O)NCC(CN(C(CC(=O)OC)=O)C)O)c(NC(=O)C2CC2)sc(C)c1C 93414,c1(C2CCN(C(CNC3CC(NS(C)(=O)=O)C3)=O)C2)ccc(F)cc1F 93415,C1(C(CNC(C(F)OC)=O)(C)C)CCN(C(=O)CC2CCC(C3CC3)O2)CC1 93416,C1(CC(N2C(C(N(CC(N)=O)C)=O)C=CC2)=O)CC(O)C1(C)C 93417,O(N(CC)C(=O)C(CCNC(=O)CS(=O)(=O)NC)NC)CC 93418,C1(F)(CNC(C2(N=[N+]=[N-])CC2)=O)CCN(C(c2cc(C3CC3)cs2)=O)CC1 93419,c1(C(=O)NC(C)C(=O)N(C(C)CCO)C)ccc(=N)[nH]c1 93420,C1(Nc2ncc(CC)s2)CC(OC)C12CCN(C(=O)OC(C)(C)C)CC2 93421,c1(CNC(C2CCCN(C(N3CCCCC3)=O)CC2)=O)cc(Br)c(F)cc1F 93422,C1(CCNC(c2cn(CC=C)nn2)=O)CN(C(=O)C(F)=C(C)C)CC(C)O1 93423,C1(C)(CCC(=O)NC(c2ccccc2Br)C)CCN(C(=O)C(C)(C)O)C1 93424,C1(NC(c2cc(C)[nH]c2)=O)CC(C)N(C(=O)CCc2nnc(C3CC3)o2)C1 93425,c1(C(=O)NC2CCCCN(C(C3C(C)(C)OC(=O)C3)=O)C2)ccsc1S(N)(=O)=O 93426,C(=O)(N(OC)C1CCOCC1)C1CCN(C(C(C(C)C)NC(COC)=O)=O)C1C 93427,C1(C)(CNC(CCC=CC)=O)CCN(C(c2ccnc(OC(C)C)c2F)=O)CC1 93428,c1(C(C)C)cccc(C(=O)NCC(CO)NC(C2CCC(N(C)C)CC2)=O)c1N 93429,S(=O)(=O)(c1ccc(NC2CCCOC2)c(C#N)c1)NCC1(C)CC1(Cl)Cl 93430,N1(C(CCCC)=O)CC(NC(C2CCN(C)C2C)=O)C2(CC2)C1 93431,c1(CCC(=O)NC(C(C)NC(c2ccc(C)cc2)=O)C)c(Cl)cncc1Cl 93432,c1(C(=O)OCC)cc(C)c(C)c(Br)c1S(N)(=O)=O.O(P1(=O)OCCC1C1CC1)CC 93433,c1(NC(C2CN(S(=O)(=O)c3cccc(Br)c3)CCO2)=O)cc(F)cc2[nH]ncc12 93434,CCCC(CCC)CC(=O)NC1CC(=O)N(C2CN(C(=O)CC3OCCO3)C2)C1 93435,C1(C)(COC)CC(NC(C2CCC2)=O)CN1C(C1CCSCC1)=O 93436,C1(C(N2CCCC(CCNC(CSC)=O)C2)=O)CC2(C1)CC1(CC1)C2 93437,CC(C(F)F)NC(=O)CCOCCN(C(=O)Cc1cncs1)C 93438,C1(NC(c2c(COC)nn[nH]2)=O)CC2CC(NC(=O)CC(C)CN(C)C)C2C1 93439,Cc1cc(CN(C(c2ccn(CCC(F)(F)F)n2)=O)C2CC2)cnc1F 93440,C(=O)(C1CCCn2c(Br)cnc21)N1C2CC(NC(=O)C=CCF)C(F)C1CC2 93441,C(=O)(Nn1cnn(CC)c1=O)C1CN(C(CCC=C)=O)CC1C1CC1 93442,c1(OC)cccc(CN2CCCC(NC(C3CCCS3)=O)C2)c1O 93443,C1(C(N(C(C)CCNC(=O)COCCN(C)C)C)=O)CCOC2(CCCCC2)C1 93444,c1(NC(=O)NC(C(c2ccc(OC)cc2)O)C)cc(OC)cc2ccoc12 93445,CC1c2cc(Br)ccc2OC1CNC(=O)N(CC1CC1)CC1CC1 93446,C(=O)(CC1CN(C)c2ccccc21)NC1(C)CN(C(C(CC(C)C)C)=O)C1 93447,CC1(C(N2CCC(F)(CNC(c3ccnnc3)=O)C2)=O)CCCCC1(F)F 93448,CCC(C)CC1C(=O)NCC(=O)N1.C(C(C)(C)OCCF)NC(N)=O 93449,CN1CCCCCC1C(=O)NCC(O)CCNC(c1ccc(Cl)c(Cl)c1)=O 93450,c1(C(=O)NC(C2CCCN(C(c3nc(=N)cc[nH]3)=O)C2)C)[nH]nc([N+](=O)[O-])c1Cl 93451,N1(C(CNC(CNC(CC2(OC)CCC2)=O)=O)=O)CC(F)CC1C 93452,c1(C(N2CCCN(C(c3ccc(=N)[nH]c3)=O)CC2)=O)n[nH]c2nccc(Cl)c12 93453,Cc1ncc(CCC(=O)NC2CC2CNC(C2(C)CC2c2ccccc2)=O)o1 93454,N1(C(C(=Cc2ccco2)C)=O)CCN(C)C(C(=O)NCC2CCNC(=O)C2)C1 93455,C(=O)(C(C)CC(C)(C)C)NCCC(=O)NCc1c(COCC)cccc1 93456,N1(C(CN2CCC(OC)C2)=O)CC2CN(C(=O)C(C(C)O)NC(C)=O)CC2C1 93457,c1(C(=O)NC(C(C)NC(C2=NOC(C)C2)=O)C)cccc2sccc12 93458,c1(CNC(=O)C(=O)C2CC2)c(Cl)cccc1[N+](=O)[O-].C12(O)CCCN(C1)C2 93459,Cc1c(C(=O)NC2CCCC2C(N2CCC(CF)CC2)=O)cccc1C(F)(F)F 93460,N1(C(c2nc(C)n(C)c2C)=O)CC(NC(c2cn(C)cn2)=O)CC2(CCC2)C1 93461,N1(C(c2cc(CC)sn2)=O)CCN(C(c2cc(C)ccc2C)=O)C(C(C)C)C1 93462,C(=O)(C(CC(C)CC)NC(c1c[nH]nc1OC)=O)NCC(C(CC)C)CO 93463,N1(C(C(=O)NCCCC)C(C)C2CCC2)CCN(CC2(C(=O)OC)CC2)CC1C 93464,c1(C(=O)NCCOC(C)C)ccc2[nH]cc(-c3ccc4nccnc4c3)c2c1 93465,C(=O)(C(C)CC(=O)NC1CC2CC(NC(=O)Cc3cncnc3O)C1C2)OC 93466,C12(NC(COCCOC)=O)CCC(CNC(C3(S(N)(=O)=O)CC3)=O)(C1)OC2 93467,c1(CNCc2c(C)c(Br)cnc2)cc2c(cn1)OCCO2 93468,C1(C(=O)NC(CC)CCO)CN(C(=O)C=CC2CC2)CC1OC 93469,O=C(C1=CCc2ccccc21)NC1CC2CN(C(=O)CC3(O)CCCC3)CC2C1 93470,C1(NC(C(CC2CC2)OC)=O)(CNC(=O)Cc2ccc(C(C)=O)s2)CCCCC1 93471,N1(C(C=CCCCC)=O)CC(NC(C23CCCC2C3)=O)CC12CCCCC2 93472,n1(CC)ccc(C(=O)NCC2CCC(C)CN2C(C2CCCC(O)C2)=O)cc1=O 93473,C1(C(=O)NCC2CCCN2C(=O)CC2(C(F)(F)F)CC2)CCCC2CCCCC12 93474,c1(OC)cc(Cl)c(C(=O)Nc2cccc(NC(C3C4COCC34)=O)c2)cn1 93475,c1(C(C)C)ccc2c(c1)CC(N=c1ccc3c(Cl)ccc(F)c3[nH]1)CC2 93476,C(=O)(CC1=CCOCC1)NC1C2CCN(C(c3ccc(OC)cc3)=O)CC21 93477,N1(C(CCc2cc(OCC)no2)=O)CCOCC1c1cccc(OC)c1 93478,CC(C)C(O)C(C)C(=O)NCc1ccsc1C(=O)Nc1cncc(C#N)c1 93479,C1(C(=O)NC2C(NC(CCCCOC)=O)CCCC2)CCC2(CCC2)CO1 93480,C1(C(=O)NC(C)CCNC(=O)C(F)=CC2CC2)CC12CCS(=O)(=O)CC2 93481,c1(CC)cc(C(N2CCCC2C(C)NC(c2sccc2COC)=O)=O)oc1CC 93482,C(=O)(C(C)(C)C(F)c1ccccc1)NCC1C(C)CN(C(=O)C#CC2CC2)C1 93483,Cc1nn(CCC(=O)N(C2CCCCC2NC(=O)C(F)(F)CO)C)c(C)c1C 93484,CC(C)S(=O)(=O)CC(=O)NC1CN(C(=O)CCc2cncc(O)c2)CCC1C 93485,C1(C(=O)OC)CN(N2CCOCC2C(C)(C)C)CCO1 93486,O=NN1CCCC1C(=O)NCC(CO)NC(c1csc(-c2cn[nH]c2)n1)=O 93487,c1(OC)c(Br)ccc(F)c1CN1CC2C(C1)N2c1ncc(C)cn1 93488,C1(Nc2cc(OCC)nc(OC)n2)CC2CCCC(C1)N2C(=O)COCC(F)F 93489,CS(=O)(=O)c1ccsc1CN=c1[nH]c(CC(=O)NC(C2CC2)C2CC2)cs1 93490,C=CCC(C)C(=O)NC(C)(CNC(c1cc(C2CCCCC2)[nH]n1)=O)CC 93491,c1(NCC(NC(CCNC(CC(C)C)=O)=O)C2CC2)ncnc(-c2ccccc2)n1 93492,C(=O)(CCCCC#N)NC(C(C)NC(=O)Cc1ccccc1Br)(C)C 93493,C1(NC(c2ccc(CC)s2)=O)CC(F)CN(C(=O)C(CCSC)NC(C)=O)C1 93494,Oc1cccc2c1CN(c1nc(=NCC3CC4C(C3)C4(F)F)[nH]c3c1COC3)C2 93495,CCCC(C)(CCC)C(=O)NCC1CC2(CO1)CN(C(=O)CCC#N)C2 93496,C1(NC(C(CCC)NC(N)=O)=O)CC2CC1N(C(c1cnc(OC)c(C)c1)=O)C2 93497,c1(CC)ccc(-c2nsc(N(C)C)n2)cc1O 93498,C1(CNC(COC2C(C)CCCC2)=O)CCC2(CN(C(c3csc(O)n3)=O)C2)O1 93499,c1(C(=O)NC2(CNCC3(O)CCOCC3)COC2)c(Cl)ccc(Cl)c1F 93500,CCC(O)CC(=O)NC(C(=O)NCc1nc[nH]n1)c1ccoc1 93501,N1(C(Cc2cn(C)nc2)=O)CCCC1C1CCCN1C(=O)CCCc1cnn[nH]1 93502,C#CC(CC(C)C)NC(C1CCN(C(=O)CCc2csnn2)C1C(C)C)=O 93503,N1(C(c2cnc(CC)s2)=O)C2CCC1CN(C(c1cnnc(C)c1)=O)CC2 93504,CCC(O)C(C)C(=O)NCC1CC(NC(=O)CC(c2ccccc2)NC(N)=O)C1 93505,CC(C)C#CC(=O)NC(C)(CNC(=O)C)Cn1cccn1.O(C(F)(F)F)CCCN 93506,C1(C(=O)NCC(C(C)C)NC(C(C(=C)Cl)(C)C)=O)CCc2nccn2C1 93507,Cc1cc(C(=O)NC(C)CNc2ccccc2)c(Br)c(Cl)c1 93508,c1(C(=O)NCCN(C(=O)C(C)S(N)(=O)=O)C(C)C)cccc2c(O)nncc12 93509,c1(OCCOC)ncccc1C(=O)NCC1CCN1C(c1[nH]c(C)cc1C)=O 93510,c1(C(N2C(C(C)C)C(NC(=O)C(C)CN(C)C)CC2)=O)cc(F)cc(F)c1O 93511,N1(C(c2c(C)cc(CC)o2)=O)CCC(C)N(C(=O)C(C)CO)CC1 93512,Cc1cc(C(N2CCN(C(C3CCSC3)=O)C(CC(F)F)C2)=O)c(N)c(Cl)n1 93513,c1(C(N2CCN(C(CCCC#C)=O)CC2C2CC2)=O)ccnc2ncnn12 93514,N#CC1(C(N2CCC2CNC(=O)CC2CCSCC2)=O)CC=CC1 93515,C(=O)(N=c1[nH]sc2ncccc12)C1CC(C)CN1C(c1coc2ccccc12)=O 93516,c1(C(=O)OCC)cc(NC(=O)NS(=O)(=O)CC2CC3(CCC3)CO2)c(Br)c(C)c1 93517,C1(CNC(CC(=O)OC)=O)CCC12CN(C(=O)C(C)NC(=O)Cn1cnnn1)C2 93518,N1(C(C(CN(C)C)(C)C)=O)CCOC2(C1)CN(C(c1noc3ccccc13)=O)C2 93519,C(C)(CO)(C(=O)N1CCC(F)(CNC(c2cnc(O)n2C)=O)C1)NC(C)=O 93520,CC1CN(C(c2ccc(C(=O)O)o2)=O)CC1c1cn(CCOc2cnn(C)c2)nn1 93521,c1(N(C)C)ccc(N(C)C(C2CCOCCN2)=O)cc1 93522,C1(C(=O)NC(COCC)C)C2CCN(C(=O)CN3CCCCCC3)CC12 93523,C1(CC=C)(C(=O)NCCN(C(=O)C(O)CC)C)CCCCC1 93524,c1(OC)cc(C(=O)NCC2(CO)CCN(C(=O)CNC(=O)OC)C2)cc(F)c1 93525,c1(C(=O)NCC(CNC(C(C(C)O)N(C)C)=O)C(F)(F)F)ncc2n1CCCC2 93526,C1(C(N)=O)(NC(c2c(NC)cccc2)=O)CCCC(C)(C)C1 93527,Cc1oc(C(N2CCN(C(=O)CC3CC(=O)NC3=O)CC2)=O)cc1S(C)(=O)=O 93528,N#Cc1ccc(=NCC2CCCC2NC(C23CCC(CC2)C3)=O)[nH]c1 93529,c1(C(=O)NC(CC(C)NC(c2ccc(CCC)cc2)=O)C)ccc(OC)cc1F 93530,C1(C(=O)NCCCOCCOC)CCCCC1NC(=O)CN1CCCC1C 93531,C1(C(=O)NC(C)C(CO)Sc2csc(C#N)c2)CCCC(C(=O)NC(C)(C)C)C1 93532,Cc1nc(N2CCN(Cc3cc(C(=O)O)cc(F)c3)CC2)c2c[nH]nc2n1 93533,c1(OC)cccc(C(CNC(c2sccc2C)=O)NC(=O)CCNC(C)=O)c1 93534,c1(C(C(=O)NCC2N(C(C(COCC)C)=O)CC=C2)C2CC2)ccc(F)cc1 93535,C(=O)(C(C(=O)OC)C1CC1)NC(CCNC(COCC)=O)C 93536,CP(C)(=O)c1ccc(C(=O)NC23CCCC2CN(C(C2CCC2)=O)C3)cc1 93537,C1(C(N(CCOC)CCNC(=O)C=Cc2ccoc2)=O)CCCC(C)CC1 93538,c1(CC)ccnc(C(=O)NC(C2CCN(C(c3cnn(C)c3SC)=O)CC2)C)c1 93539,C12(NC(c3cc4ccccn4n3)=O)COCCC1CN(C(=O)Cc1cc[nH]n1)C2 93540,C1(CNC(c2n(CC(=C)C)nnn2)c2cnoc2)Cc2ccccc2C1 93541,C(=O)(CCS(=O)(=O)NC)N1C(CC)C(NC(c2cc(-c3ccoc3)[nH]n2)=O)CC1 93542,C1(C(N(C)Cc2nncn2C2CC2)=O)C=CCN(C(=O)CC2CC2)C1 93543,N1(C(CC(CC)C)=O)CC2(C1)C(NC(=O)Cc1ccc(C)cc1)CCS2(=O)=O 93544,CC(C)CCC(=O)N1CCCC1CCC1CCN(C(C2CC(C)CO2)=O)CC1 93545,c1(C(N2CC3C(CCNC(C(CC)CC)=O)(CC3)C2)=O)ccc2c(c1)COC2 93546,N1(C(C(CCC)C)=O)CC2CC1CC2CNc1ccc(C2(C(F)(F)F)N=N2)cc1 93547,CCCCC(O)CC(=O)N1CC2C(CC(=O)NC(c3ccccc3O)C)C2C1 93548,CN=c1ccc(C(=O)NC2CCCC2N2CCN(C(c3cnc[nH]3)=O)CC2)c[nH]1 93549,C1(C(=O)NCC(C)CCO)CC(C)(C)CN1C(c1cnc(Cl)n1C)=O 93550,N1(C(c2c3scc(C)c3ncn2)=O)CC(NC(=O)CCCF)CC12CCOCC2 93551,C1(CNC(C(C)Nc2scc(C)n2)=O)CCCCN(C(=O)C(C)CC(C)C)C1 93552,CC(C)(F)CCC(=O)NCc1cc(C(=O)NCCc2ccon2)co1 93553,c1(CC)n[nH]c(CC)c1CC(N1CC(CN(C)C(C2CCCOC2C)=O)C1)=O 93554,C1(C#N)(C(N(C)CC2CC(F)CN2C(C2CC(C)(F)C2)=O)=O)CC2CCC1CC2 93555,O=C1CN(C(C2CC3(CC3)CN2C(c2cc[nH]c2)=O)=O)CCCN1 93556,CC1CN(C(c2cnns2)=O)CC(C)N1C(C1CC(=O)NC1(C)C)=O 93557,CC1(C(N2CCC2CNC(c2cccc(C(F)F)n2)=O)=O)COCCO1 93558,N1(C(C(C)(C)NC(c2ccc(F)cc2)=O)=O)CCCC2CC12CO 93559,N1(C(c2cnc(C)n2C)=O)CC2(C(=O)NCCCC(C)CO)CC1CCO2 93560,N1(C(COc2c(C)cccc2)=O)CCC(N(C(=O)Cc2cscc2F)C)C(C)C1 93561,N1(C(C(C)(C)OCC(F)(F)F)=O)CC2CCC(C1)C(NC(=O)CCC1CCC1)C2 93562,C1(O)(C(=O)NCC=C)CCN(C(=O)C(C)N)CC1.c1(C=O)ccco1 93563,CCCC(CCC)C(=O)NC(CC1CC1)C(=O)NCC(F)(F)CC1CC1 93564,c1(CC)ccc(C(N2CC3C(NC(=O)CCC(=O)N(CC)CC)C3C2)=O)c(C)n1 93565,N1(C(C)=O)CSCC1C(=O)NC(C)CCCNC(C1(c2ccccc2)CCC1)=O 93566,N1(C(C(CN(C)C)NC(c2cc(C(C)C)[nH]n2)=O)=O)CC(C)OCC(C)(C)C1 93567,C1(C(=O)NCCC(C)SC)CCN(C(=O)CCC2(N(C)C)CCC2)O1 93568,CN1CCN(C(c2cn(C)c(=O)n2C)=O)C(CNC(=O)C2=COCCC2)C1 93569,C(=O)(C1Cc2c(Cl)cccc21)N1CCCC(N(C(=O)CCCN(C)C)C)CC1 93570,C1(NC(c2c(CC)cc[nH]2)=O)CCN(C(C2C=CCC2)=O)CC1CO 93571,N1(C(CP(C)(C)=O)=O)CCC2(CCC2)C(NC(=O)COc2cccnc2)C1 93572,C1(S(N)(=O)=O)(C(N2CCCC(NC(CNC(CC(C)(C)C)=O)=O)C2)=O)CCC1 93573,N1(C(CCOCC(C)C)=O)CCCN(C(=O)C(C)Cc2ccco2)CC1 93574,CC1=C(C(=O)N2CC(NC(c3ccc(O)nc3Cl)=O)CC(C)C2)C(C)(C)CCC1 93575,CC1(C)CN(CC(Cl)=CCl)CC(CNC(C2(F)CCS(=O)(=O)C2)=O)O1 93576,C1(CNC(c2cncc(-c3ccccc3)c2)=O)CCc2ccccc2N1 93577,N1(C(C(CC)O)=O)CCN(C(c2ccccc2Oc2ccccc2)=O)CC(O)C1 93578,CCC(CC)CCCC(=O)NCC1(COC)CN(C(=O)CCCc2cccs2)C1 93579,N1(C(c2nc(OC)oc2)=O)CCCC2CN(C(=O)CN(C)CCOC(C)=O)CC12 93580,C#CCC(C(=O)OCC)NC(=O)C(c1ccccc1)NC(C1CN(C(C)=O)C1)=O 93581,C(=O)CCCCCS(N)(=O)=O.c1(NC2CCCN2CC)nc(N(C)C)ncc1C 93582,C=CC1(NC(c2cn(C3CC3)cn2)c2nnnn2C2CCOC2)CCCCC1 93583,[N-]=[N+]=NCCCC(=O)NC1CC(NC(=O)CNC(=O)NC2CCC2)C1 93584,Cc1cc(C)nc(CN2CC(F)CC2CN=[N+]=[N-])n1 93585,C1(CNC(CCS(=O)(=O)NC)=O)CC2(CO1)CN(C(=O)CC(C)(C)C1CC1)C2 93586,C#Cc1cn(C)nc1C(N1CCC(CC(=O)NCc2ncc(C)cc2C)C1)=O 93587,C1(NC(=O)C2CC2)CCCN(C(C2CCN(C(c3ccnc(F)c3)=O)CC2)=O)C1 93588,c1(OC)cc(N)ccc1C(N1CC(NC(=O)Cc2cc(C)on2)C(C)C1)=O 93589,C(=O)(CCCN(C)N=O)N1CC(C)C(C)(CNC(C2(C)COC(=O)OC2)=O)C1 93590,c1(NC(c2c(CC)n(C3CCCC3)nc2)=O)ccc(=O)n(-c2cccc(F)c2)c1 93591,C1(NC(c2ccc(COC)o2)=O)CCN(C(c2oc(Br)nc2C)=O)CC1C 93592,c1(C(C(=O)NC(CNC(C2C(CCCC)C2)=O)C)OC(C)=O)ccccc1.C(C)(C)(C)O 93593,C1(CC=C)(NC(=O)C(O)Cc2ccco2)CCN(C(=O)Cc2ccc(Cl)cc2)C1 93594,CC(C)(O)CCC(=O)NCC1CN(C(=O)Cc2cnccn2)CC1C(F)(F)F 93595,c1(NC)ccc(C(F)(F)F)c(CNC(=NCC2CCCO2)NC2C(C)(C)C2(C)C)n1 93596,C12(C(C)(C)C)CC(C(=O)NC3(CO)CN(C(C4COC(=O)O4)=O)C3)(C1)C2 93597,c1(C(C(=O)NC(C)(C)C)N(C(c2cnn(C)c2)C)C)ccc(C2CC2)cc1F 93598,C(=O)(C1=CCSC1)N1C(C(=O)NC2CC2c2ccccc2Br)CCC1 93599,Cc1c(C(=O)N(C)CC2(NC(c3scnc3Cl)=O)CC2)oc2ccccc2c1=O 93600,C1(C(=O)NCCCCN(C(CCN(C)CC)=O)C)CCCCC1c1nncn1C 93601,O=S(=O)(c1ccc(Br)cc1N1CCC=C(c2ccncc2)C1)NC1CC2(CC2)C1 93602,C=CC1(C)COCCN1C(c1ccc(OC(C)C)nc1)C(=O)NCc1ccco1 93603,N1(C(C=CC(C)NC(CC2(CC)CCC2)=O)=O)CCC(CC2CCC2)C1 93604,CCC(CCCC(=O)NC(C)CCC(C)(C)C)NC(c1n[nH]cc1C)=O 93605,c1(OC)nc(NCC(C)=O)ncc1F.N12CC3C(C3C1)C(=O)N(C(C)C)CC2=O 93606,CC1(C)CC1(C(=O)NCC1CC(=C2CC2)C1)NC(=O)C=CCO 93607,C1(SC)CN(C(C2CCSCC2)=O)CC1NC(=O)CC1CCCN1C 93608,c1(CNC(Cc2c(C)nc[nH]2)=O)ncc(C(N2CCC(C(F)F)C2)=O)cn1 93609,n1(C(C)C)ccc(CC(=O)NC(CNC(c2csnc2Br)=O)C2CC2)n1 93610,C1(NC(c2c(C)ccs2)=O)CCCC(CNC(=O)CCC2CCCCC2)C1 93611,C1(F)(C(=O)NC(CC#CC)CO)CCN(C(c2scnc2C)=O)CC1 93612,C1(C(=O)NCCC2N(C(CCCCOCC)=O)CC(OC)C2)CC(=O)NC1(C)C 93613,N1(C(C=CC=CC)=O)CCN(C(=O)C(n2nnnc2C(C)(C)C)C)C(C)C1 93614,c1(C(N2CC(C)OCC2C(=O)O)=O)cc(Br)cc(S(C)(=O)=O)c1 93615,c1(CC(=O)NCC2OCCN(C(COCCC#C)=O)C2)ccc(C)cc1Cl 93616,c1(C(C)=O)ccc(C(=O)N(CC(C)CNC(=O)C(F)C(C)C)C)nn1 93617,c1(C(N2CCOC(CCN(C)C)C2)C(=O)NC(C)C)ccc2cccnc2c1 93618,c1(C(=O)NC2CCN(C(=O)C3=C(Cl)CCOC3)C2)cccc(C#CC2CC2)c1 93619,N1(C(C2CSCC(=O)N2)=O)CCN(C(=O)CC2CN3CCC2CC3)C(CCO)C1 93620,c1(CN(C)CCc2cccs2)cccc2c1CNC2 93621,C1(C)(NC(C(CC)=CCCC)=O)CCN(C(c2coc(C(=O)OCC)n2)=O)CC1 93622,Cc1cc(C)c(C(=O)N(C)CC2CCN(C(=O)CC(C)C3CC3)C2)c(S)n1 93623,C(N=c1[nH]c(=NCCC2CCOCC2)[nH]c2ccc(Cl)cc12)c1ccc(F)cc1 93624,N1(C(C(C)NC(N)=O)=O)CCC2CCCC12C(=O)NCC#CC(F)(F)F 93625,N1(C(C2CC(=C)C2)=O)CC2(CNC(=O)CS(=O)(=O)N3CCCCC3)CC(F)(C1)C2 93626,CC(C)CS(=O)(=O)CCC(=O)N(CC(C)CNC(=O)C(C)Cc1ccncc1)C 93627,C1(COC)(NC(=O)Cc2cscn2)CN(C(=O)CCNC(C2CCCO2)=O)C1 93628,c1(C(N2C3CC(C(N(C(C)C(N)=O)C)=O)(OC3)C2)=O)cc2ccccc2[nH]1 93629,c1(C(=O)NC2C(CN(C(CN3CCC(OC)C3)=O)C)CCC2)c(C)nc(C)n1O 93630,C#CCCCC(C)C(=O)NC(C)CC1CN(C(=O)CCc2ccc(Cl)c(Cl)c2)C1 93631,C(=O)(C1=C(Cl)CCCC1)NCCC(C)(C)NC(C(C1CC1)OC)=O 93632,C1(NC(c2n(C(CC)CC)ncc2)=O)CCCCC12CCOCC2 93633,c1(CC(=O)OCC)cc(NCCC2NC(=O)NC2=O)ncn1 93634,S(=O)(=O)(C1CCC(=O)CC1)NCc1c(C)csc1 93635,n1(CC)nc(C(=O)NC2(C(N3CC4C(C(N)=O)C4C3)=O)CCN(C)C2)cc1C 93636,N1(c2ccc(C(=O)OC)cn2)CCCCC(NC(=O)CC2CCOC(CF)C2)C1 93637,CC1(C(=O)NCC2(CF)CCC2)CCCN1c1cc(-n2ccnc2)ncn1 93638,C1(NC(CC(=O)OC)=O)CC2CCC(C1)N2C(=O)CCc1ccc(F)c(F)c1F 93639,N1(C(C(C(C)(C)C)=O)=O)CCn2nc(CNC(C3CCSC3)=O)cc2C1 93640,CC(C)(Cc1ccc(Cl)cc1)CC(=O)N1CCN(C(C2CCC2)=O)CC1C1CC1 93641,c1(C(=O)NCC2C(NC(c3cc(OC)ncc3)=O)C2)cc2cc(Cl)ccc2o1 93642,N1(C(c2ccc(CC)o2)=O)CCCC(C)(CNC(=O)C(F)(F)CC2CC2)C1 93643,C1(NC(CSc2cccc(C)c2)=O)CC(NC(=O)Cc2cnc(C)[nH]2)C12CCC2 93644,CC(CC(=O)NCC1CN(C(c2cnn3ccn(C)c23)=O)C1)CC(C)(C)C 93645,C(=O)(NNC(=O)N1CCSC1)c1c(C)ncs1 93646,Cc1csc2ncc(C(N3CCCC(C)C3CNC(C3CCNC3=O)=O)=O)n12 93647,N1(C(C(N2CCCC2C2CCCOC2)C)=O)CCC(NS(CC)(=O)=O)CC1 93648,C(=O)(C(O)CC(F)(F)F)NC1CC(NC(=O)CC(C(F)F)n2ccnc2)C1 93649,C=C(C)C(C)(C)C(=O)N1CCCC1CNC(c1csc(SC)n1)=O 93650,N1(C(C(C2CC2)OCC)=O)CC(NC(c2ccc(=O)oc2)=O)C(C)(C)C1 93651,C1(NC(c2c(CC)ocn2)=O)CC2CN(C(c3cc(C(C)C)on3)=O)CC12 93652,c1(C(=O)NC2C3CN(C(C(=O)Nc4ncc[nH]4)=O)CC32)csc2cncn12 93653,Cn1cc(I)c2c(NC(C3CC(NCc4c(F)cncc4F)C3)=O)ncnc12 93654,c1(N(C2CCCNC2)C)nc(Cl)nc2c1ncn2C(C)(C)C 93655,C1(OC)CC(C)CN(C(=O)CC2CN(C(=O)C(C)=NOCC#N)CCC2C)C1 93656,c1(-n2c(C)nnn2)cc(C(=O)Nc2ccc(N(C)C)nc2)ccc1Cl 93657,N1(C(C(C2CCC2)OCC)=O)CCC(F)C(NC(c2noc(C3CC3)c2C)=O)C1 93658,Cc1cn2c(C)c(C(=O)NCC3(CNC(C4OCC4(C)C)=O)CC3)nc2s1 93659,CC1CC(CCNC(=O)CCCCN2CCCC2)CCN1C(=O)CC#N 93660,C1(C(=O)NC(CC2CN(C(C(CCC)=CCC)=O)C2)C)CCc2n[nH]cc2C1C 93661,c1(C(N2C(C(=O)Nc3n(C)ncc3I)C=CC2)=O)cc2ccccc2[nH]1 93662,Cc1ncccc1C(N1CC(CNC(C2CCCN2C)=O)C(C(F)(F)F)C1)=O 93663,c1(OC(C)C)ccc(NC(c2cc(Br)nn2CC2CC2)=O)c(Cl)c1 93664,C(=O)(C1CCCn2ccnc21)NC1CC2(CN(C(CCC=C(C)C)=O)C2)C1 93665,C12(CNC(C(COC)O)=O)CCC(NC(=O)CCC#N)(CO1)C2 93666,C1(CNC(CNC(C2C(C)C2)=O)=O)(CO)CCN(C(C2CN(C(N)=O)C2)=O)C1 93667,CC(c1ccccc1C)=CC(=O)NC(C)CCCCNC(c1nc(=N)cc[nH]1)=O 93668,C(=O)(CCCCNC(c1cn[nH]c1)=O)NC(C)CCN(C)C 93669,C1(C(C(=O)NCCOC)NC(=O)CN2CCCC2)CCOCC1 93670,c1(CC)sc(C(=O)NCC2CC(NC(C3(C)CNC(=O)C3)=O)C2)cc1Br 93671,c1(CNC(C(CC)O)=O)cnn2c1CN(C(=O)C(C(C)C)n1cnnc1)CC2 93672,C=CCC(C(=O)NCCN(C(=O)C(C)(CC)C(N)=O)C(C)C)C(C)(C)C 93673,C(=O)(CC(C(=O)N1CCC(C)(NC(C2CCCCNC2=O)=O)C1)NC(C)=O)OC 93674,c1(NC(C2CC2NC(C2(O)CCCC2)=O)=O)nc(Cl)nc2n[nH]cc12 93675,n1(CC(=O)NCC(C)NC(c2cn3cnnc3cn2)=O)cnc2sccc2c1=O 93676,C(N=c1ncc2ccccc2[nH]1)C1CC(NC(=O)COc2ccccc2F)C1 93677,c1(C(=O)NC(C(C)NC(CCCOCC)=O)CO)cnc2c(c1)NC(=O)CN2C 93678,CC1(C)CCN(C(c2csc(Cl)n2)=O)CC1NC(c1csc2ccccc12)=O 93679,C1(C(=O)NCC2(CNC(CCOCCOC)=O)CC2)CCC(=O)N(CC(C)C)C1 93680,c1(C(=O)NCC(CNC(C(c2cccc(C)c2)O)=O)F)cccc2nn[nH]c12 93681,C1(C2CN(C(=O)NCC3C(C)CC3)C2)OCC1(F)F 93682,Cc1noc(C)c1CNC(=O)COC1CC(NC(C2(C(=O)NC)CC(O)C2)=O)C1 93683,c1(CN(C(=O)C(=O)NC(c2ccccc2C)C(C)C)CC)ccc2c(c1)CCN2 93684,N1(C(c2c(C)n[nH]c2)=O)CCN(C(=O)COC(F)(F)C(F)(F)F)CC12CCC2 93685,c1(OC)cc(OC)c(CN2CCC(C)(NC(c3nc(Cl)sc3Cl)=O)C2)c(Br)c1 93686,c1(C(N2CC(N(C(C(C)NC(N)=O)=O)C)C2)=O)cnc(O)cc1C(F)(F)F 93687,C1(NC(C#C)=O)CCN(Cc2ccc(-c3ccccc3)cc2)CC1F 93688,N1(C(c2nc(CCC)sc2)=O)CC(CNC(=O)C(C)(C)OC(C)C)OC(C)(C)C1 93689,c1(C(N(CC=C)CC=C)=O)ncccc1OC.c12ccc(nc1)C(=O)NC2C 93690,c1(C(C)=O)c(Br)ccc(NC(=O)CC2CCCN(C(C3CC3C)=O)C2)c1C 93691,c1(C(=O)NCC2CCN(C(c3c(CC)nccn3)=O)C2)c(C)sc(C)c1C 93692,N1(C(C2ON=C(C(C)C)C2)=O)CC2COCC2(C(=O)NC(C)(C)CO)C1 93693,C#Cc1cccc(C(=O)NC(C2CCN(C(=O)CSCC(F)(F)F)C2)C)c1 93694,N1(CCC(=O)N(CC(CN(C(=O)C=CC=C(Cl)Cl)C)O)C)Cc2ccccc2C1 93695,C1(CCNC(c2c(C)cccc2)=O)CCN(C(C2COCC(C)(C)O2)=O)C(C)C1 93696,N1(C(C2N(CC)CC2)=O)CC2CC(NC(=O)CCOc3ccc(Cl)cc3)C1C2 93697,c1(OC)cccc(C(N2CCOCC2C(=O)NCc2ccc(Br)c(F)c2)=O)c1O 93698,C1(NC(C2CCS(=O)(=O)C2)=O)CCN(C(C2CC(Cl)(Cl)C2)=O)CC12CCC2 93699,Cc1noc2ncc(C(N3CCN(C(=O)CC(C)CF)C(CO)C3)=O)cc12 93700,c1(C(=O)NC2CC(C(C)(C)C)C2)cccc(-c2cnn[nH]2)c1 93701,C1(C(=O)NC(CC)CNC(=O)Cn2cc(C(F)(F)F)cn2)CC2CCCCCC12 93702,C1(NC(c2c(CC)ccs2)=O)CN(C(=O)CCc2ccc(NC)cc2)C2CC12 93703,c1(SCC(=O)NCC2N(C(c3ccc(=N)[nH]n3)=O)CC2)nccc2ccccc12 93704,C1(C(=O)OC)COC2(CNC(c3cnc(N)c(Br)c3)=O)CC1C2 93705,c1(-n2cc(C(N(CC(C)NC(=O)CNC(=O)C3CC3)C)=O)nn2)cccc(Cl)c1 93706,N1(C(c2cccc(OCC)c2)=O)CC(NC(c2cnsc2)=O)CC12CCCOC2 93707,N1(C(C2(CNC(CC3CCN(C)C3=O)=O)CCCC2)=O)CC2(C1)CC1(CCC1)C2 93708,N1(C(C(CC)SC)=O)CCCCC(C2CN(C(c3ccc(O)c(Cl)n3)=O)C2)C1 93709,C(=O)(C1=CC2(CCOC2)C1)N(CC(N1CCOC(CCF)C1)=O)C(C)C 93710,c1(NC(=O)Cc2ccc(S(=O)(=O)F)cc2)ccc2c(=O)[nH]ccc2c1 93711,CCC(CC)(CCNC(=O)C1=C(C)OCC1)NC(=O)COC(C)(C)C(F)(F)F 93712,C12(NC(=O)CN(C)S(=O)(=O)N(C)C)C3C4C1C1C2C3C41C(=O)OC 93713,C12(NC(c3n[nH]c(C)c3Cl)=O)CCCN(C(c3cccc(Cl)c3Cl)=O)CC1C2 93714,c1(C(N2CC(CCC)C(NC(=O)COC(C)CC)C2)=O)cn2c(n1)CC(C)CC2 93715,C12(CNC(c3cc(C)oc3)=O)CCCC1CN(C(c1ccc(F)c(Cl)c1)=O)C2 93716,C=C(C)C(CC(=O)NC1CCC1CNC(=O)Cc1cn2ccsc2n1)OCC 93717,c1(SCC(=O)NC(CC(C)C)CNC(=O)CC2CCOC2)nnc2ccccn12 93718,CC1COC(C)(C)CN1C(C1CCCCC1CNC(=O)CCc1ccoc1)=O 93719,CC1(CNC(=O)C(=O)C(C)(C)C)CCN(Cc2nnnn2C2CCCCC2)CC1 93720,C(=O)(CC(C)C(F)F)NC(CCNC(CNC(c1cccc(C)c1)=O)=O)(C)C 93721,c1(OC)cc(O)ncc1C(=O)NC(C)(C)CNC(C1C2CCCCC12)=O 93722,C(C1CCn2ccnc21)NC(=O)NCCn1ncc(CC)c1 93723,C1(NC(c2c(CC)cccn2)=O)C(CNc2ncccc2C#N)CCC12CCC2 93724,N1(C(Cn2ncc(CC)c2)=O)CCOC(CN(C(=O)C=Cc2ccccc2)C)C1 93725,n1(C(C(=O)N(C2CCN(Cc3cscc3Br)C2)CC)C)cc(C)cn1 93726,C#Cc1ccc(CC(=O)NC2CCCN(C(=O)CCOC)CC2)cc1 93727,c1(C(=O)NC(CNC(COCC)=O)C)ccc2sc(C(=O)O)c(C)c2c1 93728,C1(CNC(CCCCOCC)=O)CN(C(C2CC2C(C)(C)C)=O)CC12CC2 93729,C1(NC(C2C(C(=O)OC)C=C2)=O)CC2CCCC(C1)N2C(=O)C(C)(C)CF 93730,C1(CNC(=O)CN)CC2(CCN(C(=O)C=C3CCC3)C2)CO1.c1(C=O)cscn1 93731,CC(C)CC(O)CC(=O)N1CCC1C(N1CC(c2nc(=O)o[nH]2)C1)=O 93732,C(=O)(C1CCCc2nn[nH]c21)N(C)CC1CCCN1C(C1(O)CC1)=O 93733,N1(CC(=O)NC(C2CCOCC2)CC)CCCC(C(=O)NC(C)(C)C)CC1 93734,c1(C(=O)NC2CN(C(C3C(=C)CC3)=O)CC(O)C2)ccc2c(c1)n(C)c(=O)n2C 93735,CC(c1ccco1)=CC(=O)NCCC(C)NC(=O)CC1CCC(C)CO1 93736,c1(COC)ccc(C(N2CC3C(N(C(=O)C=C4CCC(C)C4)C)C3C2)=O)cc1F 93737,N1(C(C2N(C(c3ccc(C)nc3C)=O)CCCCC2)=O)CCn2cnnc2C1C 93738,c1(C(=O)NCC2CCCC(NC(COCCC)=O)C2)cccc(O)c1Br 93739,c1(NC(c2ncc(-c3ccc(OCC)c(F)c3)cn2)=O)cc(C)cc(C#N)c1 93740,c1(C(N2CCC(N(C(c3ccc(CC)[nH]3)=O)CC)C2)=O)cnc(O)n1CC 93741,C(N=C(NCC(C)(C)C)N1CCCC(O)(CO)C1)c1cccc(CC)c1 93742,CC1(C(=O)NCC2CCCN(C(=O)CCCCC3CC3)C2)CC(F)(F)C1 93743,CC(CC(=O)NC1CCN(C(c2cccc(N)c2F)=O)C1(C)C)C(F)(F)F 93744,CCCCCCC(=O)NC(c1ccccc1)CNC(=O)CC(C)C(C)C 93745,N1(C(COC(C)C)=O)CCC2(CCC(NC(=O)C(c3cccc(F)c3)C)C2)CC1 93746,c1(C(N(C)Cc2cn(-c3ccccc3C#N)nn2)=O)ccc2nnnn2c1 93747,Cc1coc(C=CC(=O)NCC(CNC(=O)Cn2cccnc2=O)CO)n1 93748,N1(C(C(C)OCC)=O)C(C(N2CC(O)CC2CC)=O)C2CC(O)C1C2 93749,c1(C(=O)NCC2(NC(C(CC(C)C)C)=O)CCCCC2)ccc2ncsc2c1 93750,C1(CN(C(C(CC)OCC)=O)C)CN(C(=O)C(C)NC(N)=O)CCO1 93751,N1(CC(=O)NCC(C)NC(=O)Cn2nnc(C3CC3)n2)CC(=O)NC1=O 93752,CCC(C)C(O)CC(=O)N1CCCN(C(=O)CCC(=O)N2CCOCC2)CC1 93753,C1(C(=O)NCC2(O)CC(NC(c3c(C)cnn3C)=O)C2)CCC(O)CN1C 93754,N1(C(c2cnc(CCC)s2)=O)CC2CC(C1)CN(C(=O)C1=C(C#N)CCC1)C2 93755,C1(CC(=O)NC2C(CNC(Cn3cc(C(C)=O)nn3)=O)C2)NC(=O)NC1=O 93756,c1(OC(C(N2CC(NC(CC(C)O)=O)(CO)C2)=O)C)ccc(Cl)c(Cl)c1 93757,c1(NC(C2CCN2C(c2cc(I)cnc2Cl)=O)=O)ncc([N+](=O)[O-])cc1Cl 93758,c1(N(CC(C)CNC(=O)C(C)CC2CC2)C)ccc2c(n1)CC(C)(C)CC2=O 93759,N1(C(c2c(CC)n(C)cc2)=O)CC(C(=O)NCC(CC2CC2)CO)CCC1(C)C 93760,C1(CNC(C=CC(CC)C)=O)CCCC2CN(C(c3nc(C)nn3C)=O)CC12 93761,CC1(C)CC(CNC(C2(C)CCC(=O)N2)=O)CN(C(=O)CCCC2CC2)C1 93762,CC(C)(CC(=O)N1CCCCC1CNC(=O)C=C1CCCCC1)C1CC1 93763,C(C)(CN=[N+]=[N-])NCC(=O)NC(CN(C(C)C)C)C 93764,C1(n2c(-c3ccc(Cl)cc3C)nc(C)n2)CC2CCC1(C)C2(C)C 93765,C=CCC(C(=O)Nc1cccc(CNC(=O)CN2CCCS2(=O)=O)c1)C(C)(C)C 93766,C1(CNC(CCCNC(=O)OC)=O)CC(F)(F)CN1C(=O)C(O)C(F)F 93767,CCCCC(C(=O)NCC1SCCS1)NC(C1CCN1CC)=O 93768,Cc1ccc(F)cc1C(N1CCN(C)CC1CNC(C1CCOC(C)(C)C1)=O)=O 93769,c1(C(N2CC(CC(C)NC(C3(CO)CCCO3)=O)C2)=O)cc(O)c2ccoc2c1 93770,C(c1sc2ccccc2c1Cl)=CC(=O)NCC(CN(C(CCC=C)=O)C)O 93771,CCC(C)(C)C(C)NC(=O)C(C)CNC(=O)CN1CCOC1=O 93772,N1(C(CCCc2nc(C)sc2)=O)C2CCC1C(NC(c1nc(Cl)sc1C)=O)C2 93773,C12(C(=O)NCC(CC=C)NC(=O)CCOc3ccc(Cl)cc3)CC1COC2(C)C 93774,N1(C(C(C)O)=O)CCC(C(F)F)(CNC(c2cc(-c3cccc(Cl)c3)on2)=O)C1 93775,N1(C(c2snc(C)c2Br)=O)CCN(C(=O)C(C)C2CC2)C(C)C1 93776,C12(NC(CC(=C=C)C)=O)CCN(C(=O)CCN3CCOCC3)CC1C2 93777,N1(C(c2c(C(C)C)cccc2)=O)CC2(C1)CN(C(=O)Cc1csc(C(C)C)n1)C2 93778,N#Cc1cc(S(=O)(=O)N2CC(F)CC(F)C2)ccc1NCCOc1ccccn1 93779,N1(C(C)=O)CC(C(=O)NCC2(NC(=O)CCC3CC3(F)F)CC2)C1 93780,c1(N(CCCN(C(Cn2nnc(C)n2)=O)C)C)ncnc2cc(Br)ccc12 93781,C1(NC(c2cnn(CCC)c2C)=O)CCC12CN(C(=O)CCC(C)OC)C2 93782,C(=O)(N=c1ccc(C2CCCCC2)n[nH]1)NCC1OCC(C)(C)C1 93783,c1(C(=O)NCC(C)NC(CC(c2ccc(C)cc2)C)=O)ccc2oncc2c1 93784,CC1(C)CC(CNC(=O)CCc2cnn[nH]2)CN1C(C1CC(=O)OC1(C)C)=O 93785,N1(C(CCCCCC=C)=O)CCC2(CCN(C(=O)CC3CSCCO3)C2)C1 93786,C1(C(NOCCC)=O)COCCC1NC(c1cc(Cl)n[nH]1)=O 93787,N1(C(C(C=C)O)=O)CCC(NC(c2c(CC)ncnc2CC)=O)C(F)C1 93788,c1(C(N2CC(CNC(COC)=O)C(O)C2)=O)cc(C(F)(F)F)cc(C(F)(F)F)c1 93789,CC(CC(C)(C)C)C(=O)NC(C)(CO)C(=O)NCC1(CO)CCN(C)C1 93790,Cc1ccc(C)c(OCCC(=O)N(c2nnccc2C#N)CC#N)c1 93791,c1(CC)cnn(C)c1C(=O)NCC1(F)CC(CN)C1 93792,C(CCC(=O)NCC1(O)CC(CNC(=O)CC(C)n2ccnc2CC)C1)=CC 93793,c1(CNC(C(C)C)CO)ccccc1-c1cccc(C(=O)N(C(C)(C)CO)CCl)c1 93794,N1(C(CSCCCC)=O)CC2CC(NC(c3cc(C)c(C)c(C)c3)=O)C(C2)C1 93795,C#CCC(CC#C)C(=O)NCCCN(C)C(c1ccc(C)nc1N)=O 93796,c1(C(N2CCC(NC(CSCC=C)=O)C2C)=O)cc(C)n(C(C)C)c1C 93797,c1(C(N2C3C(NC(C(CC)n4cncn4)=O)C(C3)C2)=O)cnc2ncnn2c1O 93798,C=C(CNC(C1CC1(Cl)Cl)=O)CCNC(C1(C)CC1(F)F)=O 93799,CC1(C)OCCC1C(N1CCCC(NC(c2[nH]c(C3CC3)nc2C)=O)C1)=O 93800,C(=O)(C(CC(C)(C)C)OC)N1CCC(N(C(=O)CN2CCCNC2=O)CC)C1 93801,C=Cn1nccc1C(N1CC(OCC(=O)NCC)C1)=O.CCC(C)N1CCCC1 93802,C1(Cn2cc(C3CCN(C)C3)nn2)CC2CCCC2N1C(=O)COCCCF 93803,C1(C(=O)NCC(C)NC(C2CCS(=O)(=O)CC2)=O)CCc2nc(O)[nH]c2C1 93804,c1(OCC(=O)NCCC(CNC(c2n(CC)ncc2Cl)=O)O)cc(F)ccc1F 93805,C1(NC(CCC)(C)c2nnnn2CCCC2CC2)CCCS(=O)(=O)C1 93806,Cc1nc(C(=O)N(C)C)ccc1C(N1CCN(C(C2(C(F)F)CC2)=O)CC1C)=O 93807,Cc1nc(C2CC2)ncc1C(=O)NC1CC1NC(C1CCO1)=O 93808,C(CCN=c1[nH]cncc1I)N.N1(C(=O)CCc2cnn[nH]2)CCCCC1 93809,C(C)(C)(CCCNC(=O)COc1cccc(F)c1)NC(c1ccc(SC)o1)=O 93810,CC(CCN(C)C)C(=O)NC1(CC(=O)NCc2cncc(F)c2)CCC1 93811,C1(C(=O)NCc2c(C(=O)NC3C(OCC)COC3)c[nH]n2)CN(C)CCO1 93812,C(CC(=O)N1CCN(C(=O)C(F)F)C(CC(F)(F)F)C1)(C1=CCCC1)OCC 93813,c1(-c2cnc(CNC(CC(CC)O)=O)nc2)c(F)ccc(C(=O)OC)c1OC 93814,c1(NC(C2CC(F)(F)C2)C(=O)N(CC(=O)OCC)CCC)ccsc1CC 93815,Cc1cc(C2CCCN2C(=O)Nc2nc(C3CC3)oc2C)cc(Br)c1 93816,C(C(CCS(C)(=O)=O)OC)Nc1c(N(CC)CC)ccc(Br)c1 93817,c1(C(N(C)CCN(C)C(c2cnsc2)=O)=O)cc2c(Br)ccc(F)c2[nH]1 93818,N1(Cc2onc(CC(C)N(C)CC)n2)CCN(C(=O)C(C)(C)CF)CC1 93819,N1(C(C(CN(C)C)(F)F)=O)CC(C2CN(C(c3cccc(C4CC4)n3)=O)C2)C1 93820,CCCCCC(O)CNC(=O)C(C1CN(C(c2cc[nH]n2)=O)C1)OC 93821,C1(CNC(=O)CSc2ccccn2)CC(c2ccc(C(=O)O)c(Br)c2)=NO1 93822,N1(C(c2cnc(C)[nH]2)=O)CCc2nc[nH]c2C12CCN(C(C1(C)CCCO1)=O)C2 93823,c1(CC(=O)NC(CN(C(C(CCC)NC(N)=O)=O)C)(C)C)ccc2ncsc2c1 93824,c1(C(N2CC3C(CNC(=O)C(O)C4CC4)(C3)C2)=O)cnnc2ccccc12 93825,c1(N2CCC3(C(C(=O)Nc4cccc(CC)n4)C3)C2)ncnn2ccc(Br)c12 93826,N1(C(C2C=C(C)CS2)=O)CCCC1C=CC(=O)N(CCCC(O)CO)C 93827,C(CN=C(NCc1nnc(C2CC2)s1)NCC1(C)CCC(=O)N1)NS(C)(=O)=O 93828,c1(C(=O)NCCCCCCN(C)C(C2CC2(F)F)=O)ccc2c(n1)COCC2 93829,c1(OC)ccc(SCC(=O)NCCC(C)CCNC(=O)C=CC2CCC2)cc1 93830,C1(CC)C(C(=O)NC2C(C)C2C)CCN1C(c1ccncc1F)=O 93831,C1(CNC(c2cnn(C3CC3)c2)=O)CCCCN(C(C2(F)CCCCCC2)=O)C1 93832,CCCCCCn1cc(C2(C)CN(C(=O)C(C3CCC(=O)N3)C)C2)nn1 93833,Cc1cc(C(=O)NCC2(F)CN(C(=O)CN3CCC(C)(C)C3)C2)cc2nn[nH]c12 93834,N1(CC#C)CCOC(C)(CNC(=O)CC(Cc2ccccc2)CC)C1 93835,c1(C(C(=O)NC2(CC)CCN(C(c3cnco3)=O)CC2)C)c(C)nc(O)nc1C 93836,CC1=C(C(=O)NC2CCC(NC(C3CC3c3ccccc3)=O)C2)CCO1 93837,C1(CNC(C(C)(C)OC)=O)CC(C)(C)CCC1NC(=O)Cc1cc(C2CC2)no1 93838,c1(OC)ccc(C(=O)NC2CC(NC(=O)C=Cc3cccs3)C2)cc1F 93839,c1(OC)ccc([N+](=O)[O-])cc1NNC(=O)C1CCSCC1 93840,N1(C(COCCCCCC)=O)CCC(NC(c2ccoc2CCC)=O)C(CC)C1 93841,N1(C(c2scnc2Cl)=O)CCOC2(CCN(c3ncc4cccnc4n3)C2)C1 93842,C(=O)(CC(C)(C)C)NC(C)C(=O)N(C1CCN(C(=O)Cn2cncn2)CC1)CCO 93843,CC12CC(CC(=O)N(CCCNC(C3CCCC(C(N)=O)C3)=O)CCO)(CO1)C2 93844,c1(OC)ccc(C(=O)NCCCC(O)CC(F)(F)F)cc1OC(C)=O 93845,c1(CNC2C(C(=O)NCCC3CC3)CCC2)ccc(-n2cccn2)cc1 93846,C(CCN(C)C(c1ccc(-n2cncn2)cn1)=O)(C(C)C)NC(CSCC=C)=O 93847,CCCCC(CC)CC(=O)NC1(C)CCN(C(c2cc(O)ccc2F)=O)C1 93848,N1(C(CC2(OC)CCCCC2)=O)CC(CNC(=O)C(C)SC)C(C)(C)C1 93849,CC(C)CCC(O)C(=O)NC1(C)CCN(C(c2ccc(C(F)(F)F)s2)=O)C1 93850,c1(C(N2CCC(O)(CN(C)C(C3CCSCC3)=O)C2)=O)ccccc1S(C)=O 93851,c1(C(N2CC(C)N(C(=O)CC3CCCCN3C)CC2)=O)cnc2ccnn2c1O 93852,Cn1nc(C(N2CC(O)CCC2C(N2CCC3(CC2)CC3)=O)=O)cc1C#N 93853,c1(C(N(CC(CNC(c2cc(CCC)[nH]n2)=O)(C)C)C)=O)sc(C)nc1CC 93854,C1(CNC(C(C2CCCC2)OC)=O)CCN(C(C2CCCCS2(=O)=O)=O)CC1C 93855,N1(C(CCOC2CCN(C)CC2)=O)CCNCc2cc(F)c(F)cc21 93856,C1(NC(c2cc(C)sn2)=O)CCN(C(=O)Cc2cscn2)CC1(C)C 93857,CCC(Cc1ccccc1)S(=O)(=O)NCC(O)CCC1CC1 93858,C1(C(N(CC(CN(C(=O)Cc2ccon2)C)O)C)=O)CCc2ccc(F)cc2C1 93859,Cc1cc(C(=O)NC(CO)C(C)NC(=O)CC(C)C2CCCCC2)nnc1O 93860,c1(C(=O)NC(c2cn(-c3ccccc3C)nn2)C)cc(C#N)ccc1C(F)(F)F 93861,c1(C(=O)NC(c2nc(C(N3CCC4CC34)=O)co2)C)cc(C)nn1C1CC1 93862,C1(C(=O)NCCCC)CC12CCN(Cc1ccc(Br)cc1F)C2 93863,N1(c2nc(OCC)c(Cl)cn2)CCCC(C2CC2NC(=O)CSc2nncs2)C1 93864,C1(C(=O)NCCCC(=O)NC2CC2CSc2ccc(Cl)cc2)CCCC(=O)O1 93865,C=CCC(C(=O)NCC1CC2(CC2)CN1C(c1cnn(C2CC2)c1)=O)C(C)C 93866,c1(C(=O)NC2(CCNC(C#CC3(C)CC3)=O)CC2)cc2scc(Cl)c2[nH]1 93867,C(N=c1[nH]cnc2cc(Br)ccc12)C1OCC(CNC(=O)COC2CCCCC2)C1 93868,n1(CC)c(C)cc(C(N2CCCC(NC(C3(O)CCCCC3)=O)C2C)=O)c1C 93869,c1(NC(C2(COC)CC=CCC2)=O)cc(P(C)(C)=O)ccc1COC 93870,C1(O)(CCNC(C(C=CC)O)=O)CCN(C(=O)CCCCN(C)C(C)C)C1 93871,c1(C(N2CC(O)CC(NC(c3c(C)ncs3)=O)C2)=O)cc(F)c(Cl)c([N+](=O)[O-])c1 93872,c1(OC)cc(C)c(C(=O)NCCCN2CCS(=O)(=O)CC2)c(C)n1 93873,CC1CC(N=c2[nH]c3c(c(=NCC(c4ccccc4)N(C)C)[nH]2)COC3)CCO1 93874,C1(C(=O)NC2CCN(C(C3(c4ccsc4)CC3)=O)C2)CCC(CO)CC1 93875,CC1C(C)N(C(=O)CC(C)O)CCN1C(=O)Cc1nncn1-c1ccc(F)cc1 93876,CCC(C)C(C(=O)NC1CCCC1C(=O)NCC1(C)CSC(C)=N1)N(C)C 93877,CC(C)CC(CC(=O)NC(C1CCC1)C)NC(c1ccc(O)cc1)=O 93878,Cc1oc(C(N2CC(C)(NC(=O)C3=CC4C=CC(C3)C4)C2)=O)cc1S(C)(=O)=O 93879,C(C(C)(C)CC(=O)NCC(C)(C)n1cccn1)NC(C1CCC(CC)O1)=O 93880,N1(C(C2(SCC)CC2)=O)CCCC2(CCCN2C(c2ccncn2)=O)C1 93881,c1(NC(C)=O)ccc(N)c(C(=O)NCCN(C)C(C2CC2C)=O)c1 93882,C(C(=O)NOCC(N)=O)(C1CC1)NC(CCC#C)=O 93883,c1(CN(CC(Br)Br)C)ccc2c(c1)CCO2 93884,N1(C(COCCC=C)=O)CC2CCC1C(NC(c1ccc(Cl)c(F)c1O)=O)C2 93885,N1(C(C2(C)CCCO2)C(=O)NCCOCC)CC2CS(=O)(=O)CC2C1 93886,C12(C(NOCCOCC)=O)CC(CO)(CN1C(=O)CN(C)C)C2 93887,C(=O)(CS(=O)(=O)CC(C)C)NC1(C)CCC(NC(c2ccc(C#C)cc2)=O)CC1 93888,c1(C(N2CCC(CC(N3CC(CC(F)(F)F)C3)=O)CC2)=O)ncn2c1CCC2 93889,Nc1c(C(=O)NC2CCN(c3ccccc3)C2=O)nsc1I 93890,c1(C(CC)(C)C)cc(OC)nc(N2CCCCCC2C)n1 93891,c1(CC)nc(C(=O)NC2CC(CNC(C3CC3OC)=O)C2)c2ccccn12 93892,CCCC(C)(O)C(=O)NCC1(F)CCN(C(=O)CCc2ccc(Cl)nc2)C1 93893,CC1(C)CCCC(C)(NC(C2CC3CCC(C2)N3C(=O)CN2CCCCC2)=O)C1 93894,c1(C2CCN(C(C(CSCC)NC(C34CSCC3C4)=O)=O)C2)ccccc1O 93895,c1(C(=O)NC(C(C)(C)C)CNC(C2(CO)CCCC2)=O)ccc2cccnn12 93896,CCC(CCOC)C(=O)N1CCCC(CCNC(C2(O)CCSC2)=O)C1 93897,N1(C(=O)NC(CC#C)C)CCC(NC(=O)CC=O)C(CC)C1.C1CC1 93898,C1(CNC(=O)C2=CCOC2)CC2(CCC2)CN1C(=O)CCOc1ccccc1F 93899,C1(O)(CCNC(c2ccsc2)=O)CCN(C(c2coc(C(F)F)c2)=O)C1 93900,N1(C(C(C)n2ccnc2)=O)CC2(CCCCN2C(=O)C(N2CCOCC2)C)C1 93901,C1(CNC(CCCCC)=O)CC2(CCC2)CN1C(=O)CC1CCCCC(=O)N1 93902,CC1CCn2ncc(C(=O)NCC(C)(CO)NC(c3ccc(N)cc3O)=O)c2C1 93903,C(c1cccc(O)c1O)=CC(=O)N(C1CC(C)OCC1)C(C12CCC(N)(CC1)C2)=O 93904,Cc1c(Cl)c(C(=O)NCC2(C)CCC(NC(C3(C)CC(F)C3)=O)CC2)nn1C 93905,N1(C(c2ccc(COC)s2)C(=O)NCC(=C)C)CCc2c(C#N)cccc21 93906,CC(CS(C)=O)C(=O)NC1(CNC(=O)CN(C2CCC2)C)CCC1 93907,C(N=c1cc[nH]cc1S(=O)(=O)N(C)CC1CCOC1C)c1ccc(C(C)C)cc1 93908,c1(OC)cc(CN(CCO)Cc2cnc[nH]2)cc(C)c1 93909,C1(CNC(CC=C)=O)CCC2(CCN(C(=O)CNC(C3CCC3)=O)CC2)CO1 93910,c1(C(N(CCN(C(C(C(C)C)C)=O)C)C)=O)ccc2nnc(C(F)F)n2c1 93911,c1(NCC(=O)NC2C(SC)CCC2)cccc(Br)c1 93912,N1(CCN(C(=O)CCCNC(=O)CCC2CC2)C)CCOCC1 93913,N1(C(C2CC(NC(=O)CC(O)c3ccccc3)C2)=O)CCc2cc(Cl)ccc2C1 93914,C1(CNC(C(=O)NC(C)C)=O)CC2(C1)CN(C(=O)COCCCF)C2 93915,N1(C(CC(COC)COC)=O)CCC2(CCN(C(=O)CCc3cccnc3)C2)C1 93916,C1(CNC(Cn2c(=N)scc2)=O)CCC2CN(C(C3(CCO)CC3)=O)CCC2C1 93917,Cc1nc2n(c1CC(N1CCSC1c1ccccc1)=O)CCCC2 93918,c1(CN(C(=O)CSc2nccn2C)C)csc(C(C)(C)C)n1 93919,c1(-c2cn(C(C(=O)N(C(C)C(F)F)C3CC3)C)nn2)cccc(F)c1Br 93920,N1(C(CC(C(CC)C)O)=O)CCN(C(c2ccncc2F)=O)CC2(CC2)C1 93921,C1(C(C)NC(C(C2CC2)OCC)=O)CCN(C(=O)C(F)CC2CCC2)C1 93922,NS(=O)(=O)c1n[nH]cc1C(N1CCN(C(=O)C2=NOCC2)C(CC(F)(F)F)C1)=O 93923,N1(CC2CCC2)CCOCC1.C1(C(=O)N)CSCN1S(=O)(=O)CC1CCOC1 93924,N1(C(CSCC=C)=O)CCCN(C(c2c(C(F)(F)F)cccc2F)=O)CC1C 93925,CC1=C(C(=O)NC2CC(C(=O)Nc3cccnc3C)C2)CCO1 93926,C(CSC)(C(=O)N(CCC(=O)NCC1CC1(Cl)Cl)CC1CC1)OC 93927,N1(C(CCCNC(c2nc(O)n[nH]2)=O)=O)CCC2C(C1)C2(F)F 93928,CC1CC(C(=O)NC2(CC(=O)N(C3CC4(CC4)C3)C)CCC2)CCS1 93929,CC(C)CC(C(=O)NC(C)CCCNC(=O)CCCCN(C)C)C(C)C 93930,CC1=CCCN(C(=O)C(CO)NC(C2C(C#N)C2(C)C)=O)C1 93931,c1(C(=O)NC2CCN(c3nc(SC)c(F)cn3)CC2F)cc(F)c(Br)cc1Cl 93932,C1(N(C(C(C)C)=O)C)CCCCC1N(C(=O)COCCN(C)C)C 93933,CC1CN(C(C2(C(N)=O)CC2)=O)CC1n1cc(C2(O)CCOC2)nn1 93934,c1(CN2CC(OC)C(NS(=O)(=O)CCCl)CC2)cc([N+](=O)[O-])ccc1Cl 93935,C1(C(=O)OC)CCC(C2CCCCC2)CN1C(=O)NCC1(OC)CCOCC1 93936,C12(COC)CC(NC(C3CSCCS3)=O)(CN1C(c1cc(Cl)n(C)n1)=O)C2 93937,C=CC(CCC)CC(=O)NCCOC1CCN(C(c2[nH]nnc2COC)=O)C1 93938,CC(C)C(F)(CNC(=O)CCCC1CC1)C(=O)N(C(CO)C(C)C)C 93939,N1(C(C=CC2(C)COC2)=O)CCCN(C(=O)Cn2cnc(Br)n2)CC1 93940,c1(-n2nnc(C(=O)NCCCNC(C(C=CC)O)=O)c2C)ccc([N+](=O)[O-])cc1 93941,N1(C(c2ccc(C)o2)=O)CCC(NC(c2cc[n+]([O-])cc2)=O)C2(CCC2)C1 93942,C(=O)(C1=CC2CCCCCCC12)NCC(C)(C)OCCNC(CCCCCOC)=O 93943,C1(CNC(CSC)=O)CC(C(=O)N(CC(O)C(C)(C)C)C)=NO1 93944,CC(CC(=O)N1CCC(C(=O)NCCCCC(N)=O)O1)n1cccc1 93945,C1(NC(CC2(C)CCCO2)=O)CCC2(CCCN2C(c2ccoc2Cl)=O)CC1 93946,C1(CC=C)(NC(=O)CCCC2CC2)CCN(C(=O)CC2CCC(C)CO2)C1 93947,c1(CC(=O)NC2COCCC2NC(C2(F)CC=CCC2)=O)ccnc(Cl)c1F 93948,C1(C(=O)NC(CCOC)CNC(C2CCC2)=O)CCN(c2nccs2)CC1 93949,c1(CC(=O)NC2C(NC(C3N(C(CCC)=O)CCC3)=O)CC2)cccc(O)c1F 93950,C1(c2cn(CC(CC)CC)nn2)CC2CCC(C1)N2C(c1nc(CC)c(C)o1)=O 93951,N1(CC(=O)NCCN(C)C(c2ncsc2C2CC2)=O)CCCC(N(C)C)C1 93952,c1(C(=O)NC(CNC(CNS(CC)(=O)=O)=O)C2CCC2)c(S(C)(=O)=O)cnn1C 93953,N1(CC(=O)NCC2C(OC)COCC2)C(=O)CCC(N)C1=O 93954,N1(CC#C)CCC2(CCN(C(C3C4C5CCC(C5)C34)=O)C2)C1 93955,C1(C)(CC)CCCN(C(=O)COCCNC(c2csnc2Cl)=O)C1 93956,c1(C(=O)NCC2CC(NC(c3c(C)cc(O)nn3)=O)C2)c(O)ncc2c1CCC2 93957,C1(OC)CC(CNC(C2(C#N)CCC2)=O)N(C(c2c(C)csc2C)=O)C1 93958,N1(C(CC2CCCN(C(CC(=O)OC)=O)C2)=O)CCn2cnnc2C1C 93959,c1(CC2C(C3CCN(C(=O)OC(C)(C)C)CC3)OCCC2)cccc2[nH]ncc12 93960,c1(CC(=O)N2C(C)CNC(=O)CO2)cncc(F)c1.C1(CC)CCCO1 93961,O(N1CCC(N=c2nc(N(CCCC(F)(F)F)C)c3c([nH]2)CSC3)CC1)CC 93962,c1(C(=O)NCCN(C(c2sccc2CN(C)C)=O)CC)ccc2nsnc2c1 93963,N1(C(c2c(C)[nH]nc2Cl)=O)CCN(C(C2CC2F)=O)C(c2cc(F)ccc2F)C1 93964,N1(C(=O)Cn2nnc(C3CC3)n2)CCOC(CNC(C2C(C(=O)OCC)C2)=O)C1 93965,c1(C(N(C)CC2(O)CCN(C(c3nnc(C)s3)=O)CC2)=O)cc2ccccn2c1 93966,N#Cc1cc(C(N2CC=CC2CNC(C2(Cl)CC23CCC3)=O)=O)ccc1F 93967,c1(C(=O)NCCCC(C)NC(CC(C(C)C)O)=O)cc2c(Cl)ccnc2s1 93968,Nc1nccnc1C(N1CCC1CNC(c1c(Br)n[nH]c1Br)=O)=O 93969,N1(CC)CC(NC(=O)C(CO)NC(=O)C(C2CCCCC2)C)C(C)C1 93970,C1(NC(=O)Cn2cc(Cl)cn2)CCC2(CC1)CC2NC(C12CC3CC1C2C3O)=O 93971,N1(C(c2c(CC)nns2)=O)CCOCC(CNC(=O)C(C)n2cccn2)C1 93972,c1(N(C)CN2CC(Sc3ccccc3)CC2=O)ccc(S(=O)(=O)N(C)C)o1 93973,C1(Cc2ccc(O)cc2)CCN(N(C(CC(=O)OCC)=O)CNC(=O)OC)CC1 93974,c1(C(N2C(C(NOCC=CC)=O)CCC2C2CC2)=O)cccc(O)c1F 93975,N1(C(CCCOC)=O)CC(OC)C(NC(=O)CCCc2nccs2)C1 93976,CCC(C(=O)NCC(N(CC)CC)C1CC1)N(C(=O)CCN(C)CC)C 93977,C1(CC)CN(C(c2cc(C)n(C(C)C)c2C)=O)CCC1NC(C1CCCN1C)=O 93978,CC(CC(=O)NC1CCCN(C(=O)CCCC2CCCCC2)CC1)C(F)F 93979,c1(C(N2C(CNC(C(C)Cn3ccnc3)=O)CC2)=O)ccc2cc[nH]c2n1 93980,C=CCC(C(=O)NCC1CCC(N(C)C(c2cc(C3CC3)sn2)=O)CC1)C(C)C 93981,C(=O)(C(CCN(C)C)NC(=O)CCOC)NCC(C1CCCC1)OC 93982,C1(C(C)(C)NC(=O)CCN2CCC2)CCN(C(c2ccc(OCCF)cn2)=O)CC1 93983,c1(NC(c2c(C)cc(C)cc2C)C)nccc(=NC(C)c2n[nH]c(=N)s2)[nH]1 93984,N1(C(c2cc(C)c(Br)nc2)=O)CCC(C)(C#N)CC1 93985,C(CCN=c1nc(N2CCOCC2)cc[nH]1)N(C(C(C(C)S(C)(=O)=O)C)=O)C 93986,C1(CC)CC(OC)CN(CC(=O)NNC(=O)c2cccnc2)C1 93987,Cc1cc(CCC(=O)NCC(CC(C)C)NC(=O)Cn2nc(C)oc2=O)n(C)n1 93988,c1(C(=O)NC2CC(OC)CN(C(C(CC)SC)=O)C2)ccc2cn(C)nc2c1 93989,N1(C(C2C(OCC)CC2)=O)CCCC(CO)(NC(=O)CC(CC)C2CCC2)C1 93990,c1(C(N2CC(C)CC(NC(c3n(CC)c(O)nc3)=O)C2)=O)c(F)ccc(F)c1O 93991,c1(SC)cccc(C(=O)N(CCCCNC(c2occc2C2CC2)=O)C)c1 93992,N1(C(C(C(C)C)NC(C)=O)=O)CC2CCCN(C(=O)C(CC(C)C)C(N)=O)C2C1 93993,c1(C(N2CCC(CNC(c3ccccc3NCCO)=O)C2)=O)ccc[n+]([O-])c1 93994,c1(C2(C(=O)NC3CN(C(CC4CN(C)C4)=O)C3)CC2)ccc(Cl)c(F)c1 93995,C(N=c1[nH]c(=NC(C)C(C)F)[nH]c2cccnc12)c1cc(OC)nn1C 93996,C1(C(N(CCOc2nccc(C)c2)CCN(C)C)=O)CCCCNC1=O 93997,c1(CC(=O)NC(CN(C(=O)C=C(C)c2ccsc2)CC)C)cc[nH]c(=N)c1 93998,c1(OC)cc(CNC2C3CC4CCC3C(C2)CC4CN)cc(OC)c1OC 93999,Cc1ccc(C=CC(=O)N(CC(O)CNC(C2(C)CNC(=O)C2)=O)C)cc1Cl 94000,N1(C(C(n2ncc(C)c2)C)=O)CC=CC(C(=O)NCCN2CCC(O)C2)C1 94001,N1(C(c2ncc(C(C)C)s2)C(=O)NCCCCCC)Cc2ncsc2C1 94002,N1(C(c2cc(COC)no2)=O)CCCCC1CCNC(=O)C(C)CSC(F)(F)F 94003,CC(CC(=O)NCCCNC(=O)Cc1csc(-c2ncccn2)n1)C(C)(C)C 94004,C(=O)(CC(C)(C)C(=O)N1CC2CC(NC(c3cc(C4CC4)ns3)=O)C(C2)C1)OCC 94005,N=c1[nH]nc(CC(=O)NC2CCC(NC(=O)CCN3CCC(F)C3)C2)s1 94006,C1(NC(c2ccc(F)cn2)=O)(CNC(=O)C(O)Cc2ccccn2)CCOCC1 94007,C(CCCCCC=C)NC(C(CN(C(c1c(C#C)c[nH]n1)=O)C)C)=O 94008,N1(C(C2(c3ccccc3)C(C)(C)C2)=O)CCOC2(CCN(C(=O)C=CCF)CC2)C1 94009,C1(CC)CCN(C(=O)Nc2cccc(C3COC3)c2)C(CC)C1 94010,C(C1c2ccsc2CCN1C(c1ccc(F)cc1)=O)NC(CN(C)C)=O 94011,C1(C(N2CCC(N(CCO)C(c3cccc(=O)o3)=O)CC2)=O)C2CCC(C2)S1(=O)=O 94012,C1(OC)CCCC(C(=O)C(C#N)C(=O)NCCOc2cc(C)ccc2C)CC1 94013,c1(OC)ccc(C(N2CCC(NC(C3CC34CC4)=O)C2(C)C)=O)cc1CC1CC1 94014,N1(Cc2c(OC)ccc(O)c2)CCC2CN(C(=O)CSc3nc[nH]n3)CCC12 94015,C(=O)(CS(C)(=O)=O)NCC1(F)CCC(CNC(C(N2C(=O)CCC2=O)CC)=O)C1 94016,C1(C)(C(=O)NCC(c2cccc(OC)c2)NC(C=C(CCC)C)=O)CCC(C)C1 94017,C12(CNC(C)=O)CCCCC1CN(C(c1nsc3ccc(C)cc13)=O)C2 94018,C1(NC(CCn2ncc(C)c2)=O)CCN(C(=O)C(F)C(C)C)CC1(C)C 94019,Cc1nc(C(N2CC(C3(NC(=O)C(C)N(C)C)CC3)C2)=O)ccc1C(=O)N(C)C 94020,N1(C(c2csc(Cl)n2)=O)CCC2(CCN(C(C3CCC4(CCC4)CO3)=O)CC2)C1 94021,C1(C(N2CCC(N(C)C)(CC)C2)=O)CCC2(CC2)N1C(=O)C=C(C)C 94022,N1(C(C(C)n2cccc2)=O)CCCC(C(=O)NC2CCCC(O)C2)CC1 94023,C1(c2ccccc2)(CC(=O)N(C(C)CNC(C2COC(=O)N2)=O)C)CCOCC1 94024,Fc1cc(F)c(C(c2ccccc2)NCc2ccc3occc3n2)c(F)c1 94025,c1(CC)ncc(Br)cc1C(N1CCC(NC(=O)C(=O)N(C)C)C(C)C1)=O 94026,c1(C(=O)NC(C)CCNC(=O)C(C)c2cccs2)ccn2c1CSCC2 94027,c1(C(N2CCCC(CN(C)C(C3CC4(C3)CC4F)=O)C2)=O)c(F)cc(O)cc1F 94028,C1(S(=O)c2ccccc2)(C(N2C(c3cn(CCCC)nn3)C(C)CC2)=O)CCC1 94029,c1(C(N(C2CN(C(c3ncccc3Cl)=O)CC2F)C)=O)scc2c1OCCO2 94030,C(=O)(C(C)(C)C(N)=O)N(C1CCN(CC(=O)NCCC)C1)CCOC 94031,N1(C(C2C(CC)C2)=O)CCCCC1C1CCN(C(C23CC4CC2C3C4)=O)CC1 94032,c1(C(=O)NCCCCCNC(=O)C=C2CC2)ccc2c(c1)nc(O)n2CC1CC1 94033,c1(C(C)CNC(c2sccc2Br)=O)cccc(C(F)(F)F)c1 94034,Cc1cc(C(=O)NC2CCCC(CC(=O)NCc3ccnc(F)c3)C2)nc(C)n1 94035,c1(OC)ccc(C(=O)NCCC2(O)CN(C(=O)CC3C(C)(C)C3(C)C)C2)cc1F 94036,c1(NC(C2CCCN(C(CCNC(=O)OC(C)(C)C)=O)C2)=O)ccc(C#N)c(Cl)c1 94037,CC1OCCOC1C(=O)NC1(CO)CCN(C(c2c(Cl)nsc2Cl)=O)C1 94038,CCC(C(=O)NCC1CC1NC(c1cn2ccnc2cn1)=O)C(F)(F)F 94039,C=Cn1nncc1C(=O)NCC(CC(=O)NCC(C)C(F)(F)F)OC 94040,c1(CC(=O)NC2(CCNC(C3(C(=O)NC)CC3)=O)CCC2)cccc(F)c1Cl 94041,C1(CNC(c2scc(OC)c2)=O)CN(C(=O)C=C2CCSCC2)CCN1C 94042,c1(OC)ccc2c(c1)OC(C)(C)CN(C(C1CN(C)CCO1)=O)C2 94043,c1(CC(C(=O)NCc2cccc(N3CCC3=O)c2)NC)ccc(F)cc1F 94044,c1(C(=O)NCC(CNC(C2CC2C#N)=O)OC)cccn(C2CCC2)c1=O 94045,c1(CN2CCCC(C(N3CCC(CN(C)C)CC3)=O)C2)ccc(I)cc1F 94046,C1(CC)CC(O)CCN1C(C1COCC1NC(C1CC1C1CC1)=O)=O 94047,N1(C(C2(CO)CC(C)(C)C2)=O)CCCC(F)(C(=O)N(C2CCOCC2)CCO)C1 94048,n1(CC(=O)NCCOC2CN(C(CCC3(C)N=N3)=O)C2)ccccc1=O 94049,C1(C(N2C(CNC(=O)C3=CCCS3)CC3(CC3)C2)=O)CCc2nncn2CC1 94050,c1(N(C)C)sc(C)nc1C.C(CCC(=O)NCCOC1CCN(CC=C)C1)O 94051,c1(C(=O)NCCC2(CN(C(C3CCSC3)=O)C3CC3)CC2)cnn(C(F)(F)F)c1 94052,CCS(=O)(=O)CC(=O)NC(CCC1CC1)C(=O)NC1(CSC)CC1 94053,N1(C(C(C)OCC2CC2)=O)CCC(CNC(c2cc(O)n(C)n2)=O)C(O)C1 94054,C1(CCCCCNC(CCC#C)=O)CCN(C(c2ncn(C)c2C)=O)CC1 94055,N1(C(COCc2cc(C)no2)=O)CC(CNC(=O)C=C2CCSCC2)CCC1C 94056,c1(SCC)ccccc1CC(=O)NCC1CC(O)CN1C(=O)COC(F)F 94057,n1(C(CC)CCO)cnc2c(N(C3CCOCC3)CCF)ncnc12 94058,C12(C(=O)OC)CCCC1N(C(c1csc3ccccc13)C(=O)NCC(C)C)CC2 94059,C1(NC(C(F)=C(C)C)=O)CC1C1CCN(C(c2nccc3cccnc23)=O)CC1 94060,c1(CN(C)C)ccc(C(=O)NC2(C)CCN(c3nnc(C4CC4)o3)C2)cc1 94061,C1(C(=O)NC(CC)(C)C2CC2)CC12CCN(C(=O)C(O)CC(F)(F)F)CC2 94062,Cc1ccc(C(F)F)cc1C(=O)NC1CC(C)(NC(=O)CC2CC=CCC2)C1 94063,c1(CN(CCC)Cc2ccccc2)c(C)nn(-c2ccc(F)cc2)c1Cl 94064,S(=O)(=O)(c1cccs1)N1CCC(C(N2CCC2C(F)(F)F)=O)CC1 94065,C1(NC(C(COCC)n2cc(CC(=O)OC)nn2)=O)CCC2(CC1)COC2 94066,C1(C(=O)NC2(C)CC(C(=O)NC(CC)C(C)(C)O)C2)CCC2CC1CO2 94067,CC1CCN(C(C2(C)CCOC(C)C2)=O)CC1CNC(c1nccnc1Cl)=O 94068,C(C(C)C(=O)N=c1ccn(C)[nH]1)N(C(CCSC)=O)C 94069,C1(C)(C(N2CCC(NC(C3(CCOC)CC3)=O)CC2)=O)CCN(C)C1=O 94070,CCC(CNC(C12CC(CC(F)F)(C1)C2)=O)(CC)NC(c1cn(CCO)nn1)=O 94071,c1(C(=O)OC)sccc1S(=O)(=O)Nc1cc(C(=O)O)cc(C(C)C)c1 94072,C1(NC(C=NOC)=O)(CNC(=O)C(C2CC2)OCO)CCCCC1 94073,CCC(C)(C#N)C(=O)N1CC(NC(c2oncc2C)=O)C(C)C1 94074,Cc1ncc(C(N2CCC(CCNC(=O)Cc3csc(C)c3)C2)=O)c(C)n1 94075,c1(CC(N2C(CNC(C(CC)C(C)C)=O)COCC2)=O)c[nH]c2cnc(Cl)cc12 94076,c1(SCC)cc(CC(N2CC(C(=O)OC)C2)=O)cs1 94077,c1(C(=O)NCC2(OC)CCN(C(=O)CC3CCCO3)C2)cnc2ncccn12 94078,C(=O)(C(CCC(C)(C)C)ON)OC.c1(C=O)cc(O)ccc1Br 94079,N1(C(c2ccc(COC)[nH]2)=O)CC(C)CCC1CNC(c1nccc(C)n1)=O 94080,C1(CNC(c2ccc(C(C)(C)C)s2)=O)CN(C(=O)C2CC2)CC1C(F)(F)F 94081,C1(COC)CN(C(=O)CCCC2CC2)CCN1C(=O)CC(=O)Nc1nccs1 94082,C(=O)(C(O)CCCNC(c1c(C)ccnc1O)=O)N1CC(CC)OCC1 94083,N1(C(c2c(CC)cc(N)cc2)=O)CCCC2(NC(C3CCN3CC)=O)CC2C1 94084,c1(OCC(=O)OC)ccc(CCNC(=O)NCC2C(F)(F)C23CC3)cc1 94085,C1(CCNC(C2CCN(C)C2)=O)CCN(C(C2(c3cccnc3Cl)CC2)=O)CC1 94086,CCCC(O)CNC(=O)C(=O)NCc1cn(C2CCCNC2)nn1 94087,C1(NC(C2(C)CC(F)C2)=O)CCCCC1NC(=O)CSc1ccccc1Cl 94088,C1(C(=O)NCCC(C)NC(C(C)Cc2cccc(F)c2)=O)CC(C(C)(C)C)=NO1 94089,c1(C(=O)NC2CN(C(C3CCCOC3)=O)C2)ccc(O)cc1F 94090,N1(C(c2cc(OC)ncn2)=O)CCOC(C)(CNC(=O)Cc2cccnc2C)C1 94091,CN1CCC(CC(=O)N(C(=O)Cc2ccccc2)Cc2ccccc2)C1 94092,CC1(C)CC(NC(=O)CCNC(C)(C)C2CC2)CCN1 94093,c1(CC)cc(N)ccc1C(=O)NCC1CCCCN1C(=O)CCc1cnc(O)[nH]1 94094,c1(NC(=O)NC(CSC)C(C)(C)C)cc2cccc(F)c2cn1 94095,S(=O)(=O)(c1ccc(NC(c2ccc(C)cc2)=O)cc1)NC 94096,c1(C(=O)OC)cnc(C)[nH]c1=NCCC(C)NC(=O)C1CCCc2n[nH]cc21 94097,CCCC(CNC(=O)C(=O)C(C)(C)C)C(=O)N1CC(N2CCCC2=O)C1 94098,C1(NC(C2N(C(C)=O)CCOC2)=O)CC2(C1)CN(C(=O)C(=O)NC1CC1)C2 94099,C1(NC(C2CCS(=O)CC2)=O)CCCN(C(=O)CCC2CCCCC2)CC1 94100,N1(C(C)C)CC(C(=O)OC(C)C)C1.C1(=O)CNC(=O)C2(CC2)CN1 94101,Cc1cc(F)c(C(N2CCCC2CN(C)C(C2CC=CC2)=O)=O)cc1F 94102,n1(CC)cc(CNC(C2CN(C(C3CC3c3ccccc3)=O)CCO2)=O)c(C)n1 94103,c1(OC)ccc(NC(=O)C2CC2)cc1NC(=O)NCc1ccccc1C(C)C 94104,c1(OC)ccc(C(N2CC3CC2CN3C(=O)C(CSC)OC)=O)c(N)c1F 94105,N1(Cc2cc(COC)no2)CCC(=O)N(CCC(C(F)(F)F)OC)C1=O 94106,C1(NC(=O)C=Cc2cscn2)CC2CCC1(CNC(c1cc(Cl)c[nH]1)=O)C2 94107,c1(C(=O)NC(CNC(C2(COC)CCCO2)=O)C)ccc(Cl)c(N)c1 94108,N1(C(c2nc(CC)sc2)=O)C2CCC1C(NC(c1cnc(C(F)(F)F)nc1)=O)C2 94109,C(CCNC(=O)CSC)(C(N)=O)NC(COC(CC)CC)=O 94110,c1(SC)ncc(F)c(NC(CCCCC2CCN(C(=O)OC(C)(C)C)CC2)=O)n1 94111,Cc1oc(C#N)cc1C(N1CCCC(n2cc(C3(F)CCOCC3)nn2)CC1)=O 94112,Cc1nc2ccc(NC(N3CCCN(C(C45CC6CC4C5C6)=O)CC3C)=O)cc2[nH]1 94113,CC1CSc2ccc(Br)cc2C1NC(c1c(N)sc2ccccc12)=O 94114,c1(C(N(C)CC2N(C(C3CCC(CC)O3)=O)CCCC2)=O)cccn2cnnc12 94115,N(C(=NCc1ccccc1)NCC12CC(C(=O)OC)(C1)C2)Cc1cnc(CC)o1 94116,CC(CCc1ccccc1)CC(=O)N(C1CCN(C(C2(F)CC2)=O)CC1)CCO 94117,n1(CC)nccc1C(=O)N(C)CC1CCCN1C(C1(Br)CC1(F)F)=O 94118,C(=O)(CN=c1cc[nH]cc1)NCC1CCN(C(c2c(CC)noc2)=O)C1(C)C 94119,c1(C(N2CC(CNC(C(CC=C)OC)=O)C(C)C2)=O)cc2ccccc2o1 94120,c1(C(N(C2CCC(NC(CCOCCOC)=O)C2)C)=O)csc2cccnc12 94121,C1(C(N2CC3C(CNC(c4c(C)ccs4)=O)(C3)C2)=O)C(O)C(=O)N(C)C1C 94122,N1(C(C(C=C)C)=O)CC2CC2C1C(=O)NCCN1CC(CF)C1 94123,CC(C)(O)CC(=O)NC1CC1NC(C1(c2ccc(O)nc2)CCC1)=O 94124,c1(C(C)C)ccc(C(=O)NCC2CCCCCN2C(C2C=CCCC2)=O)cc1Cl 94125,Cc1snnc1C(N1CC(c2ccccc2)(NC(c2cc(CO)on2)=O)C1)=O 94126,C(=O)(CS(=O)(=O)c1ccccc1Cl)NC(CNC(C1N2CC(C)N(CC2)C1)=O)C 94127,CCC(CCC(=O)NCCCC(C)NC(=O)CNS(N)(=O)=O)OC 94128,N1(CCC(=O)OC(CN(C(C)=O)CC)OC)c2ccccc2Sc2ccccc21 94129,Cc1nc(O)[nH]c1C(=O)NCC(C)(O)CNC(=O)CN1CCOCC1 94130,C1(C(=O)NC2CCC(NCc3c(C)c(Cl)ncc3)C2)CCc2cc(Br)ccc2O1 94131,Nc1ccc(NC2CN(C(CN3C(C(=O)NC4CCOCC4)CCC3)=O)C2)cc1 94132,C1(CNC(CSCC=C)=O)CC2CCC1N(C(c1cc(C)nc(N(C)C)n1)=O)C2 94133,N1(C(C(C)OC)=O)C2CCC1CC(NC(=O)Cc1ccc(O)c(C)c1)C2 94134,c1(C(=O)NCC2C(NC(CCNC(=O)NC)=O)C2)ccc2c(ccn2C)c1 94135,N1(C(c2cc(C)cc(F)c2)=O)CC(NC(c2cccc(C)n2)=O)C2CCCC12 94136,C1(NC(C2CC(OC)C2)=O)C2CC(NC(=O)CC3NC(=O)NC3=O)CC12 94137,c1(C(=O)NC2(CNC(C(C(C)C)F)=O)CC(F)(F)C2)nccc2n[nH]cc12 94138,c1(C2(C(C)(C)O)CC2)cn(CC(N2CCC(N3CCC3)C2)=O)nn1 94139,N1(C(c2ccn(CCC)n2)=O)CC2CC1(C(=O)N(CC(C)CO)C)C2 94140,CCC(C)(C)C(=O)N1CCCC(CC(=O)NCCCNC(=O)OC)C1 94141,c1(C(=O)NC2CCCN(C(C(C)N(C(C)=O)C)=O)CC2)cc2ccc(F)cc2[nH]1 94142,CN1CC(C)(C(=O)NCC2CC(NC(c3cccc(OC(F)F)n3)=O)C2)CC1=O 94143,C1(CNC(C=C2CCC(C)C2)=O)CN(C(=O)CC2(C)CC(F)(F)C2)CC1O 94144,c1(SC)cccc(C(=O)NC(C)(C)CCCNC(=O)Cn2cnnn2)n1 94145,c1(C(=O)NCC2N(C(c3c(CC)nccn3)=O)CC2)c(F)ccc(Cl)c1F 94146,c1(C(N2CC(c3cn(C)nc3)OCC2)=O)ccc(F)c(N)c1 94147,C(=O)(C(CC)NC(C1CC(n2cc(C3OCCO3)nn2)C1)=O)NCCC 94148,C1(C)(C(=O)NC)CCN(C(C2(NC(=O)CN3CCOCC3=O)CC2C)=O)C1 94149,C1(=O)C(C)(O)C(C)N1.Cc1c(-n2cc(C3CC3)nn2)cnn1-c1cccc(Cl)c1 94150,C1(=O)C(C)(C)C(=O)N2CC(C2)N1C.c1(NC(=O)NCCCCl)cccc(F)c1C 94151,C#Cc1cccc(CC(=O)NC2CCOCC2C(N2CCOCC2CO)=O)c1 94152,CC(C)C(C)C(CNC(=O)Cc1cnn(C)c1)NC(=O)C=Cc1cncn1C 94153,N1(C(CCc2cccc(C)c2)=O)CCN(C(=O)COC2CC=CC2)C(C(F)F)C1 94154,N1(C(c2c(F)ccc(C)n2)=O)CC2CCN(C(c3cnc(C4CC4)[nH]3)=O)C(C2)C1 94155,C(CC(=O)NCC(C)CNC(=O)CCNC(C1CCCO1)=O)NC(C)=O 94156,c1(-c2scc(C(=O)NCC(C3CN(C(=O)CN(C)C)C3)C)n2)cccc(Cl)c1 94157,c1(C(=O)NC(CCCNC(C(CC)C(C)O)=O)C)ncn2ccccc12 94158,C1(F)(C(=O)NCCCOCCNC(=O)CNC(c2ccco2)=O)CCOCC1 94159,Cc1cncnc1C(=O)NCCC1(C)CCN(C(c2conc2C2CC2)=O)C1 94160,C1(N(C(C(C2CCOCC2)C)=O)C)CN(C(=O)CCC(=O)N(C)C)CC1(C)C 94161,C1(CC)CN(c2nnc(-c3ccccn3)n2C2CCS(=O)(=O)C2)CCO1 94162,CC(CC(=O)NC(CNC(C1CC1F)=O)CO)n1ccnc1 94163,C=CCC(C(=O)N1CCC(CNC(=O)CN(S(C)(=O)=O)C)CC1)C(C)C 94164,C1(CCNC(CCOCC)=O)CCCN(C(C2CC(C)(C)C2)=O)CC1 94165,C1(C(=O)NCc2onc(C(N)=O)n2)CC(=O)CN1C(=O)C=Cc1cncs1 94166,C1(C(C)(C)C)CC(N=c2[nH]c(=NCC=CC3CC3)[nH]c3cccnc23)CCO1 94167,C1(O)(C(N2CC3(C(=O)OCC)C(C2)CCO3)=O)CCc2ccccc2C1 94168,N1(C(c2cc(C(C)C)nc(O)c2)=O)CC2CCC1CN2C(=O)C=CC1CCOC1 94169,C1(NC(Cn2c(CCC)ncc2)=O)CC2CC1CN(C(c1nc(O)sc1C)=O)C2 94170,C1(NC(C2CC(=O)OC2)=O)CCOCC1NC(c1cocc1C(N)=O)=O 94171,Cc1ccccc1NC(C1CCCC(NC(=O)Cc2c(C)n[nH]c2C)C1)=O 94172,c1(OCCC)ccc(CNc2ccc(OCCOC)cc2)nn1 94173,Cc1cccc(CNC(=O)C(CNC(C2(C)CCC3CC3C2)=O)C(C)C)c1C 94174,C1(NC(c2c(OC)cccc2)=O)CN(C(C2CC(F)C2)=O)CC2(CCC2)C1 94175,C(C(CC(C)C)C(=O)N1CCC1CNC(c1cc(Cl)cc(Cl)c1OC)=O)OC 94176,C1(NC(C2CCN(C(C=NOC)=O)C2C)=O)CCCN2CCCC12 94177,N(C)(C1CCc2c(Cl)cccc21)C(c1scc(C)c1)C(=O)NC(C)(C)C 94178,C1(CNC(C2C(=C)C2)=O)CC2CCC1N2C(C1(c2ccccc2)CCOCC1)=O 94179,CCC1CNC(C)C2(CC2)SCC(=O)N1C.C(CC#N)SC 94180,c1(C(=O)NCC2C=CC(NC(=O)CCSC(F)(F)F)C2)sc([N+](=O)[O-])cc1Cl 94181,N1(C(C(CCCCC)C)=O)CCC2(CC1)CC(C(=O)N(C)CC#N)CO2 94182,CC1CN(C(=O)C(=O)N(C)C)CCCN1C(=O)CCC(=O)c1ccc[nH]1 94183,N1(C(CCc2n(C)ncc2)=O)CCC(C(C)(C)NC(=O)CC2CS(=O)(=O)C2)CC1 94184,c1(C(=O)NCCN(C(c2ccc(OC)c(Cl)n2)=O)C2CC2)c[nH]nc1S(N)(=O)=O 94185,O=C1NCCn2nc(C(=O)NC3CCN(C(C45CCC(CC4O)C5)=O)CC3)cc21 94186,CC1(C)OC2C3CC(C2O1)N(C(c1ccc(OC(F)(F)F)cc1O)=O)C3 94187,N1(C(c2c(OC)cc(C)s2)=O)CCCOC(CCNC(C2CC2[N+](=O)[O-])=O)C1 94188,C1(CNC(=O)CN2CC3CCC2C3)(NC(c2cc(F)n[nH]2)=O)CC2CCC1CC2 94189,C(=O)(C(CC)CC(C)C)NCCCOCCN(C(CCCC(=C)Br)=O)C 94190,C1(NC(C2CC(=C)C2)=O)CCC2CCN(C(c3ccc(C4CC4)c(N)c3)=O)C1C2 94191,c1(C(=O)NC(CC)CNC(=O)CC(=O)OC(C)(C)C)cc(C)c(C)c2ncsc12 94192,N1(C(C(CCC)C#N)=O)CCC(C)(C)CC1C(=O)NC(c1ncc(C)cn1)C 94193,N1(C(c2cc3ccccn3c2)=O)CCC2OCCN(C(C3CC4CC4C3)=O)C2C1 94194,C1(COC)CN(C(c2ccsc2)=O)CCN1C(=O)C#CC1(C)CC1 94195,C1(CNC(C2(SC)CCC2)=O)CCN(C(c2c(Br)ncn2C)=O)CC1 94196,CC1CN(C(c2cc(Cl)c[nH]2)=O)CC1NC(c1ccnc(CO)c1)=O 94197,C1(O)(C(N(CCNC(c2ccccc2O)=O)C2CC2)=O)CCSCC1 94198,N1(C(CN(C(C(C)C)=O)C)=O)CCOC(CNC(=O)CCC2CCCCN2C)C1 94199,N1(C(=O)CCN2CCC(O)CC2)CC2OCC(NC(C34CC(CO3)C4)=O)C2C1 94200,C1(NC(Cc2ccc(C)o2)=O)CN(C(c2snnc2C(C)C)=O)CC1C(F)F 94201,C(C(=O)NC1CCCCC1NC(=O)CCOC1CCC1)(C(C)C)OCC 94202,C1(C(=O)OC)C(C(=O)OC)C2CCC1N2Cc1ccccc1Br 94203,C(=O)(C(C)CC(F)(F)F)NC1COCCN(C(CCCCOC)=O)C1 94204,N1(C(C(C)C(C)(C)C)=O)CC(NC(c2nccc(Cl)c2O)=O)CC12CCCCC2 94205,C12(C(=O)NCC(CNC(c3coc(C4CC4)n3)=O)F)CCC(CO)(CC1)C2 94206,Cc1c(NC2C=C(C#N)CC2)ccc(C(F)(F)F)c1F 94207,C(=O)(CCCCC(C)=O)NCC1CCN(C(c2ncc(CC)cn2)=O)CC1C 94208,c1(C(N2C(C)CC(CNC(C(C3CCOCC3)C)=O)C2)=O)cc(Cl)ncc1F 94209,c1(C(N2CC(C)(C)C2CO)=O)cc(C(=O)O)ccc1O 94210,c1(OC)c(F)ccc(C(=O)NCC2CCC2NC(c2ccsn2)=O)c1F 94211,c1(CCC(=O)NCCC(CNC(C2(COC)CCC2)=O)O)cc2ccccc2o1 94212,C1(C(=O)NC(C=C)C)OCCC1CNC(C1(OC)CCC1)=O 94213,Cc1c(CNC(C2COCCN(C(c3cnsn3)=O)C2)=O)cccc1O 94214,C1(C#N)(C(N(CCCCN(C(c2cc(CCC)on2)=O)C)C)=O)CC=CC1 94215,C1(C(N2CC(O)C(O)C2)=O)(CC)CCCN(C(c2ncccc2N)=O)C1 94216,CNS(=O)(=O)N1CCC(C(N2CC(CNC(=O)CC(C)COC)C2)=O)CC1 94217,c1(N(C)C(=O)NCC2CCCN2C(c2cnn(C)c2)=O)cc(F)cc(F)c1 94218,Cc1[nH]c(C#N)cc1C(=O)NC1CN(C(=O)C2=CC(C)(C)C2)CC1C(F)F 94219,CCCCC(C(=O)NC1CC(=O)N(C2CN(c3ccc(Br)cc3F)C2)C1)NC(N)=O 94220,c1(OCCC(=O)NCCC(F)Cn2cc(C3CCCCO3)nn2)ccccc1Cl 94221,C1(NC(c2nn(CC)c(O)c2)=O)CN(C(=O)Cc2cnccc2C)CC2(CC2)C1 94222,c1(OC)ccn2cc(C(=O)NC3(C)CN(C(=O)C4=CCCCC4)C3)nc2c1 94223,n1(CCC)cccc1C(N1CC(CC)(NC(=O)C(CSC)OC)C1)=O 94224,C12(C(=O)NC3CCN(CC)C3)C(NC(c3cnc(S)nc3)=O)C3CC1C2C3 94225,C1(CC(=O)NCC#CCNC(C2CCN(CC(C)C)C2)=O)COC(C)(C)CO1 94226,C(C)(c1ccccc1F)=CC(=O)NC1CCN(C(c2nccc(CC)c2)=O)C1C 94227,c1(OC(c2ccc(N(C(=O)CC3C(=O)ON=C3C)CC)cn2)=O)ccc(Br)cc1C 94228,C1(CC)(CNC(CN2CC(CNC(=O)CSC(C)C)C2)=O)CCCC1 94229,C1(NC(CSC(C)C)=O)CCCCN(C(C2(Cl)CC2(F)F)=O)CC1 94230,c1(CC(=O)NCCN(C)C2CC2)n[nH]c2cc(Cl)ccc12 94231,N1(C(C(C)(C2CC2)OC)=O)CCC2(CCCCC2NC(=O)C(C)C2CC2)C1 94232,C12(CC(=O)N(C)CCNC(=O)C=CC3COC(C)(C)O3)CCCCC1C2(F)F 94233,N1(C(C=CCC(C)(C)NC(c2n(C)cnc2)=O)=O)CCOCC(C(N)=O)C1 94234,c1(CN(c2ccnc(Br)n2)C(=O)CSC2CCCN2)ccc(Cl)cc1 94235,C(c1ccc(Br)o1)=CC(=O)NCC(C)(C)NC(c1ccc(=N)[nH]n1)=O 94236,N1(C(c2cc(OC)no2)=O)CCN(C(c2ccccc2)=O)C2CCCC12 94237,C(C)(C)(C(C)NC(C1(C(=O)OC(C)(C)C)CC1)=O)NC(C1N(CC)CC1)=O 94238,C1(CC)CN(C(=O)C(C)C)CCC1NC(=O)C(Cc1cccc(C)c1)N(C)C 94239,CCC(C(=O)NC1CC(CO)N(C(C2CNC(=O)O2)=O)C1)C(C)C 94240,N#CC1(NS(=O)(=O)Cc2cccc(Br)c2)CCN(Cc2cc(I)ccc2Cl)C1 94241,c1(-c2n3c(nn2)C3)cn2ccccc2n1.c1(CN(CCOC)C)cccc(O)c1 94242,CC(C)CC(CNC(c1cnn(C(C)C)c1)=O)C(=O)NC1CCSCC1 94243,N1(CC)C2CCC1CN(C(C1(NC(C3CCC(C)=C(C)C3)=O)CCOCC1)=O)C2 94244,Cc1cccc(C2(F)CCN(C3CCN(c4cccc(F)c4)C3=O)C2)c1 94245,C1(OC)CC(CNC(c2cncc(C(C)C)c2)=O)N(C(=O)COCC(F)(F)F)C1 94246,Cc1cc(Cl)c(C(N2CC(CNC(c3ncnc(C)c3C)=O)C(F)(F)C2)=O)cn1 94247,c1(C(=O)NC(C(C)NC(C2CCCS2(=O)=O)=O)(C)C)cccc2c1nc(O)n2C 94248,C1(C(=O)NC(C)(C)C(N2CCOCC(O)C2)=O)CC(=O)CC12CCC2 94249,c1(C(N2CC(O)(CNC(CC3C(C)(C)C3)=O)C2)=O)nc(F)ccc1Cl 94250,CC1C(C)N(C(C2CCC2)=O)CCN1C(c1cc(C2CCOCC2)[nH]n1)=O 94251,c1(N(CC(C)C)CCN(c2ccccc2)C)cn(C)nc1O.Cc1n[nH]cc1C 94252,C(=O)(C(CCC1CC1)NC(=O)C(C)SCCCC)NC(C=C)CO 94253,CC(C(=O)N1CCC(OC2CCCCC2)C1)S(C)(=O)=O 94254,C1(F)(CNC(CC)=O)CCC(CNC(C2CCC(C3CC3)C2)=O)CC1 94255,CC1CN(C(=O)C=Cc2cc(Br)cs2)CC1NC(C1(Cl)CC1)=O 94256,CCCCCCCCCC(=O)N1CCN(C(=O)C(C)C2CCCO2)CC1 94257,N1(Cc2cccc(C(N)=O)c2)CCCC2(C1)CN(c1ncnc3n[nH]c(Br)c13)C2 94258,c1(C(N2CCC3(C(C(=O)NCCCCCO)C3)C2)=O)cccc2[nH]ccc12 94259,C1(=O)C(C2CC2)CNC(=O)CN1.C(COCCOC)(C1CC1)COCC 94260,c1(C(=O)NCC23CC(COC)(N(C(=O)C4=NOCC4)C2)C3)coc2ccccc12 94261,c1(C(=O)OC)ccc(C)cc1Cn1cc(SCCN(C)CC2CC2CO)nn1 94262,Cc1ncc(N)cc1C(=O)NC12CC(NC(=O)CNC(c3cccnc3)=O)(C1)C2 94263,c1(C(N2CCCC2C)C(=O)NCCCSC)cc(C(F)(F)F)ccc1C 94264,N1(C(C(C(CC)C)C)=O)CC2CC(NC(c3sc(O)nc3C)=O)C(C2)C1 94265,c1(C(CNC(C(c2ccccc2)OC)=O)NC(=O)C=CC2CCC2)cnn(C)c1 94266,c1(C(c2nc(-c3cccnc3C)no2)OC)ccc(C)c(F)c1 94267,c1(C2C(C(=O)OCC)C2C(C)C)ccc([N+](=O)[O-])c(N)c1 94268,Cc1cnccc1C(C)C(=O)NC1CC(F)(NC(=O)CN2C(C)CCC2C)C1 94269,C1(C(N2CCC(CC(C)NC(=O)C3CC3)CC2)=O)CCCCC1(C)C 94270,Fc1ccc(N2CCN(CCCC3CC3)CC2)cc1 94271,Oc1ncccc1NCCCN(c1ccccc1)CCC1CC1C1CC1 94272,Cc1cc(C(=O)NC(C)CNC(C2(c3c(C)cccc3C)CC2)=O)c(N)c(Cl)c1 94273,Cc1cccc(CC(=O)NCCC2(NC(C3CCCC3C(C)C)=O)CCC2)c1 94274,c1(NC(C)=O)cccc(C(N2CC(C(C)NC(=O)C(C)c3ccsn3)C2)=O)n1 94275,Cc1cc(N2CCC(NCCCCCN(C)C(C3CC3C)=O)C2=O)ccc1F 94276,c1(NCC)ncc(C(=O)NC2(CCNC(C3CNC(=O)C3)=O)CC2)cc1Cl 94277,C(=O)(CC(O)CNC)N(CC)CC1CCS(=O)(=O)C1 94278,N1(C(CC2(OCC)CCC2)=O)CCCCC1CCNC(C1CC(N=[N+]=[N-])C1)=O 94279,Cc1oc(C(=O)NC2C3CN(C(c4cnc(O)n4C)=O)CC23)cc1S(C)(=O)=O 94280,N1(C(C(CC=CC)NC(c2ccn(C)c2)=O)=O)Cc2nc(C)sc2C1 94281,n1(CC)ncc([N+](=O)[O-])c1C(=O)NC1C2CN(C(=O)C(C3CCCC3)OC)CC12 94282,c1(C(N(C2CN(C(C3CC(CF)C3)=O)C2)C)=O)sc(Cl)cc1Br 94283,S(=O)(=O)(c1ccc(N2CCC(CC3CC(NC)C3)C2)c(Cl)c1)NC(CC)CCO 94284,C=C1CCN(C(c2ccc(F)cn2)=O)C(C(=O)NCCN(C(C)C)C2CC2)C1 94285,c1(C(=O)NC2(CCC)CCC2)cnc(CNC(C2CCN2CC)=O)nc1 94286,C1(NC(c2cc(C)[nH]c2C)=O)CC(O)CN(C(C2CCC(C)O2)=O)C1 94287,n1(C(CC)CC)nc(C(=O)N(C(CCC(=O)OC)C(=O)OC)C)ccc1=O 94288,N1(Cc2ccc(N(C)C(c3csc(Br)c3)=O)cc2)CCCN(CC(N)=O)CC1 94289,C1(C2CN(C(c3ccsc3)=O)C2)(NC(c2cnc(C(F)F)cn2)=O)CC1 94290,c1(C(C)(C)C)ccc(C(=O)NCC(C)(CO)NC(C23CCC2C3)=O)nc1 94291,N1(C(COc2ccc(C#C)cc2)=O)CC(C)CN(C(C2(C)CC=CC2)=O)CC1C 94292,C1(OC)CC(CNC(c2cc(F)n(C)n2)=O)N(C(c2ccc(C#N)o2)=O)C1 94293,C(=O)(CCS(=O)(=O)C(F)(F)F)NC(C(C)(C)C)CNC(C1CCCCN1N=O)=O 94294,C1(C(=O)NCCCN(CC)CC)(CC)CCCN1C(c1n[nH]cc1C)=O 94295,CC1(C(=O)NCC2(NC(C3CCS3(=O)=O)=O)CCCC2)CCC(O)CC1 94296,C1(NC(C(COCC)C)=O)CN(C(c2cc(C)c(Br)o2)=O)CC1SC 94297,CC1(C)CC(C(=O)NCC2CN(C(=O)CCC3CCC3)C(C)(C)C2)CNC1=O 94298,N1(C(C(C)SCC)=O)CC(NC(C2Cc3nnc(C)n3C2)=O)CC12CCOCC2 94299,C1(NC(c2ncc(OC)cc2F)=O)CN(C(C2CC3CCC3C2)=O)CC2(CC2)C1 94300,C1(OC)CC(CNC(c2cccnn2)=O)N(C(C2CC2OC(C)(C)C)=O)C1 94301,N1(C(Cc2c(OC)cccc2Cl)=O)CCCC2(CCc3ccccc32)C1 94302,C1(CNC(C(CCC)NC(C)=O)=O)CCN(C(c2ccn(CC#N)n2)=O)C12CC2 94303,C(N1C(C)CCCN1C)c1c(C(=O)OC)c(C)[nH]n1 94304,Cc1ccc(C(C)CC(=O)NCC2CCN2C(=O)C(C)(C)c2cc[nH]n2)cc1 94305,c1(C(N2C3(CNC(CNc4c(C)n[nH]c4C)=O)CC(C2)C3)=O)c(Cl)cccc1Cl 94306,N1(C(C(=O)N(CCCSCC)C2CC2)c2ccns2)CCOCC(C(N)=O)C1 94307,c1(OC)cncc(Oc2ccnc(COC(c3ccnc(Cl)c3)=O)c2)n1 94308,c1(C(N2CCCCC2C2CCCCC2)C(=O)NCCC)nn(CC)cc1Cl 94309,N1(C(c2c(C(C)C)cco2)=O)CC(CNC(C2CC2C)=O)OC(C)(C)C1 94310,C(=O)(CC(C)CCC=C(C)C)N1CC2(CN(CCC)C2)C1.c12ccc(c(O)c1)CN2 94311,c1(OC)ccc(CCC(=O)NC23CC(NC(C4CC45CCOC5)=O)(C2)C3)cc1O 94312,C1(N(C(CCOCCN(C)C(c2cnccn2)=O)=O)C)CCN(C(=O)CO)CC1 94313,c1(C(N(C2CCN(C(=O)C(C)CSC)C2)C(CSCC)=O)=O)ccccc1NC 94314,C[Si]1(C)CCN(C(C2CCCCC2CNC(C2CCC(O)C2)=O)=O)CC1 94315,c1(CC)cccc(NC(=O)COCCOCc2ocnc2CC)c1 94316,c1(C(N(CC(C)NC(C2OCCC2C)=O)C)=O)cc(C2CC2)oc1C1CC1 94317,CCCCC(CC)CC(=O)NC1CCC(C(=O)NCC2(OC)CC2)C1 94318,N1(C(CC(=O)NC)=O)CCN(C(=O)CCc2c(C)nn(CCC#N)c2C)CC1C 94319,c1(C(N2CCC(CNC(C(C)SCC)=O)(OC)C2)=O)ccc2c(c1)CCC2 94320,C1(OC)(CNC(=O)Cc2c[nH]ccc2=O)CCN(C(=O)CC2CCCSC2)C1 94321,c1(CN(C2CCOC2C)C(C)C)ccc(C(F)Cl)cc1 94322,C(=O)(C(C)(CC)CC)NC(C(=O)N1CCC(CCCC)C1)CCF 94323,C1(CC(=O)N(CCN=[N+]=[N-])C)C=CC(NC(=O)CCc2cccs2)C1 94324,C1(CNC(CC(C)NC(c2cc[nH]n2)=O)=O)CC(C)(C)CN1C(c1ccncc1)=O 94325,N1(C(C2N(C(c3c[nH]nc3Cl)=O)CC23CCCC3)=O)CCCC(C2CC2)CC1 94326,c1(C(N2C(C)(CNC(C3=C(C)CCC3)=O)CCC2)=O)cc(Cl)c2ccccc2n1 94327,C(CS(=O)c1ccccc1)NC(CC1(OCC)CCC1)C 94328,n1(CCC)ncc(C(N2CCCC(CNC(=O)CC=CC3CC3)C2)=O)c1C(C)C 94329,c1(C(=O)NCCCN(C(C2(COC)CCCO2)=O)CC)ccc2n[nH]cc2c1 94330,C1(NC(COCC)=O)CCN(c2ncc(O)c(C)n2)CC1OC 94331,c1(C(=O)NC2C(NC(CCCCC(C)C)=O)COC2)cc(F)cc2cnccc12 94332,CCC(CC(C)C)C(=O)NC1CCC1NC(C1(N(C)C)CCCC1)=O 94333,N1(C(C2C(OC)C2)=O)CCN(C(=O)Cc2csc(Br)n2)CC(O)C1 94334,N1(C(c2cnc(C(C)O)s2)=O)Cc2c[nH]nc2C(C)(C)C1 94335,Cc1cc(C(=O)NC2CCCC(C(=O)NOCC3CCCCC3)C2)nc(C)c1 94336,CCC(C)(CCC(C)C)C(=O)N1CC2OCCN(C(=O)C=CC(C)(C)C)C2C1 94337,c1(COC(C2CCN(C(C3CCC(OC)C3)=O)CC2)=O)cc(=O)n2ncsc2n1 94338,c1(OC)cc(N(C)C)ccc1C(=O)NCC1CC(NC(C2(CO)CC2(F)F)=O)C1 94339,C1(CCNC(c2c(CC)non2)=O)CCCN(C(c2cnc(OC)nc2)=O)C1 94340,N1(C(CCN(CC)CC)=O)CCC2(NC(=O)CCOCC(C)(C)C)CCCCC12 94341,C1(COC)(NC(=O)CCC(C)(C)F)CCN(Cc2cc(OC)ccn2)CC1 94342,c1(-n2c(Cc3nc(C)sc3C)nc(C(C3CC3)OC)n2)cc(CO)ccc1C 94343,CC(C)(CCCC(=O)N1CC2(CCCCC2)C1)NC(=O)Cn1cccn1 94344,C1(n2cc(C(=O)OCC)nn2)CCCN(c2ncccn2)C1.c1ccc(Br)cc1 94345,c1(C(N(C)CC2N(C(C(C)C3CC3)=O)CCOC2)=O)cnn2c1CCC2 94346,CCC(C#N)(CC)C(=O)NCC(N1CCN(C(c2cc(C)ncc2C)=O)CC1)C 94347,c1(CCCC(=O)NCCNC(C2COCCO2)=O)c[nH]c2ccccc12 94348,C1(C(=O)NCc2cc(OC)ns2)CN(C(=O)C=CC2CCCC2)CCN1C 94349,N1(CC)CC(C(N2CCC(CCNC(=O)CC(C)F)CC2)=O)CCC1=O 94350,c1(C(N(C)CC2(O)CCN(C(c3cnn(C)c3)=O)C2)=O)ccc(F)c(O)c1F 94351,c1(-n2ncc(C(=O)NCC(CNC(CNC=O)=O)CO)c2)ccc(F)cc1 94352,c1(NC(C(=O)NC2(CN(C(CC(C)C)=O)C)CC2)=O)ccc(C#N)c(Cl)c1 94353,N1(C(c2cc(C)oc2)=O)CCC(NC(c2cnn(C)c2)C)C(C)C1 94354,c1(C(N2CCN(S(c3ccc(C)s3)(=O)=O)CC2)=O)ccc2c(c1)CCC2N 94355,n1(CC#C)cccc1C(=O)NCC1(NC(=O)C=CC2CCC2)CCC1 94356,C1(N(C(c2c(C)occ2)=O)C)CCCC2CN(C(c3ccc(=O)n(C)c3)=O)CC12 94357,C1(NC(CSCC#C)=O)CC2CN(C(=O)C(C)CC3CCCC3)CC2C1 94358,C1(C(=O)OC)CCN(C(=O)CSc2cc(Cl)ncc2OC)CCC1(F)F 94359,c1(CN2CC(CNC(c3cocn3)=O)C2)cccnc1O 94360,O=C1C=C2CN(CN=c3ccnc(C4COc5ccccc5C4)[nH]3)CCC2S1 94361,c1(C(N(C(C)CNC(c2cccc(Cl)c2OC)=O)CC)=O)cc(Cl)cc(C)c1N 94362,c1(C(=O)NCC(=O)NC(C(=O)OC)Cc2cn(C)cn2)cccc(Br)c1 94363,N1(C(c2cc(C3(C)CC3)on2)=O)CC2CN(C(C3CCCN3N=O)=O)CCC12 94364,Cc1ncsc1CCC(=O)NC1CC(CCNC(C2(CO)CCC2)=O)C1 94365,C(CCC(O)C(=O)NCCOc1ccccc1)NC(Cn1nc(C)oc1=O)=O 94366,CC(C)S(=O)(=O)CC(=O)NC1CC(CNC(c2ccc(N(C)C)cc2Cl)=O)C1 94367,C1(C(=O)NCCC(CC)C)CC2(CC(NC(c3c(C)cccc3C)=O)C2)C1 94368,C(C)(C(=O)NC(C(=O)NCCCCOCCN(C)C)C1CCC1)OCC#C 94369,O=C(CCC(F)(F)F)NC1CC(NC(C2(N3CCOCC3)CC2)=O)C12CCC2 94370,N1(C(c2cc(C)on2)=O)CCN(C(C2COC3COCC3O2)=O)CC(O)C1 94371,N1(C(c2ccc(C(C)=O)cc2)=O)C2CCC1CC(NC(c1cc(Cl)cnn1)=O)C2 94372,C1(NC(C2CC(OC)C2)=O)CCCC2CN(C(=O)CCn3c(C)csc3=O)CC12 94373,c1(C(=O)NCC2(O)CN(C(=O)CC3CCC(O)C3)C2)cnc2c(c1)COCC2 94374,C(=O)(CCCCC(C)(C)OC)NCCC(C)NC(C(CC(=C)C)OC)=O 94375,C1(NC(C2C(CC)C2)=O)CC2(CCCCN2C(c2cn3cccc(Cl)c3n2)=O)C1 94376,C1(C(=O)NCc2cscn2)CC2(C1)CN(C(=O)C(c1ccccc1)O)C2 94377,Cn1ncc2c(NCC3COCC4(CCC4)O3)[nH]c(=NCCCC(F)(F)F)nc12 94378,C12(c3cc(CN(CCCCCCCC)CCC(N)=O)[nH]n3)CC3CC(CC(C3)C1)C2 94379,c1(C(=O)NC2C(NC(C3C(=C)C3)=O)CCC2)cn(C)[nH]c1=N 94380,N1(C(c2ccn(C)c(=O)c2)=O)CC2CCC(CNC(C34CC3CNC4=O)=O)C2C1 94381,c1(SC)ncc(C)c(N2CCCC(C(N3C(CO)CCC3C)=O)C2)n1 94382,C1(C(=O)NCC2(CCNC(c3cc(-c4ccoc4)[nH]n3)=O)CC2)CCCCS1 94383,c1(CNc2cc(CO)c(Cl)cc2)cccc2sccc12 94384,c1(C(=O)NC(CCCC)CNC(C2C(C)C2C)=O)cccn2ncnc12 94385,CCCCCCCC(=O)N1CCC1CNC(c1ccc(C(F)(F)F)nc1)=O 94386,c1(N2CCC(C(C(=O)OC)F)CC2)nnc(C2CCc3c[nH]nc32)n1CC(C)C 94387,c1(CNC(C(c2cnn(C)c2)NC(CCCCNC(C)=O)=O)=O)cc(C)cnc1F 94388,C(CC(O)C(F)(F)F)NC(C=CCN(C(CCCOCC=C)=O)C)=O 94389,C1(C)(CNC(C(C)SC)=O)CCN(C(c2cncc(CO)c2)=O)C1.C(N)=O 94390,CC(c1ccco1)=CC(=O)N(C1(CC(=O)NC(c2nc(C)no2)CO)CC1)C 94391,C1(C2(OC(C)=O)CCC2)(N(C2CCC2)C(C2(C#N)CCN(C)CC2)=O)CCC1 94392,N1(C(C)C(=O)NCC(c2ccccc2)NC(=O)CC2CCC2)CCC(O)CC1 94393,c1(NC(=O)NC2CCN(C(=O)C=Cc3ccccc3)C2)ccc2cccnc2n1 94394,N1(C(=O)OC(C)(C)C)CCCC1CNC(C1CC(N2CCCC2)C1)=O 94395,c1(C(N(CC(C)NC(=O)CCc2ccc(F)c(F)c2)C)=O)ccc(Cl)c(F)c1 94396,c1(CNc2ccc(C(CC)C)cc2)cnc2[nH]ccc2c1 94397,N1(C(COC)=O)CC(NC(c2sc3ccsc3c2C)=O)CC12CCOCC2 94398,c1(OC)ccc(C(C)(C)C)cc1NC(=O)C(=O)NCC1CC(=O)C12CCC2 94399,c1(OC)cc(NC2CCC(NC(=O)C(C)CN(C)C)CC2)ncn1 94400,C1(C(N(CCF)CC)=O)CC(NC(C2CC(F)(CF)C2)=O)CCO1 94401,n1(CC)ncc(C(=O)NC23CC(C(N4CC(n5ccnc5)C4)=O)(C2)C3)c1C 94402,C(C(O)CC(C)(C)C)NC(c1c(CNC(c2n(CC#C)cnn2)=O)cc[nH]1)=O 94403,c1(C(=O)NCC(N(C(c2c(C)snc2)=O)C)C2CC2)cnn(C)c1Cl 94404,C(=O)(CC(C)C(C)C(C)C)NC(CC)(CC)CCNC(c1cn(C)ccc1=O)=O 94405,C=CCCC(O)CNC(C12CC1CN(C(=O)COC)C2)=O 94406,C(CCCCC(=O)NC1(CF)CCN(C(=O)CC(=O)OCCC(C)C)C1)SC 94407,c1(OC(CC)C#N)cc(NC(=O)C(N2CCC(CN(C)C)CC2)=O)ccc1OC 94408,Cc1ccc(S(=O)(=O)CC(=O)N2CCCC(O)CC2)cc1C 94409,CC1CCN(c2ncc(C(=O)NCC(C3CC3)NC(=O)C=CCF)s2)CC1 94410,Cc1cncc(OCC(=O)NC(CNC(=O)C2=CCSC2)Cc2ccccc2)n1 94411,N1(C(C2CN(C(CCOCC#C)=O)CC2C(C)C)=O)CCCC(C)(F)C1 94412,C(C(COC)C(=O)N(CC(C)(C)CNC(=O)CC1C=CCCC1)C)OC 94413,CC(C)C#CC(=O)NC1CCC(NC(C2CCCOC2c2ccnn2C)=O)CC1 94414,C(=O)(C(C)(C)C(=O)N1CCC(C)C(NC(=O)C=CCOC2CCOCC2)C1)NC 94415,N1(C(C)CNC(c2cnccn2)=O)CCN(C(=O)CN2CCC(C)(C)C2)CC1 94416,C1(CCC)(CNC(=O)CCCN(C)C)CCN(C(C2(CCOC)CCC2)=O)CC1 94417,C=CC(C)CC(=O)NC(C)CN(C(=O)CNC(=O)C(C)CC)C 94418,N1(C(C23C(CCN(C(C(C(=C)C)(C)C)=O)CC2)C3)=O)CC(C)(C)OC(C)(C)C1 94419,C(=O)(CCC1=NNC(=O)CC1)N1CC2(OCC(NC(C(CCC#C)O)=O)C2)C1 94420,c1(OC)cccc(C(=O)NC(C)CCN(C(=O)C(C)(C)C2CCCC2)C)n1 94421,CCCC(CC)C(=O)NCC1CCCN(C(c2cncc(CO)c2)=O)CC1 94422,C#Cc1ccc(C(=O)NCC2CCCN2C(=O)C(C)CN2CCOCC2)cc1F 94423,CC1CNC(=O)CC(NCCCc2cn(C(C)C(=O)O)nn2)C1 94424,c1(C(N2CCCC(CCNC(CNC(C)=O)=O)C2)=O)cccc2c1CCN2 94425,C1(NC(C(CO)OC)=O)CCCC(C(=O)NCC2(c3ccon3)CC2)C1 94426,Cc1cc(C(=O)NC2CC3(C2)CN(C(c2cc(C)sn2)=O)C3)c(O)c(C)n1 94427,C1(NC(C2(C)C=CCC2)=O)C=CCN(C(=O)Cc2ccnc(Br)c2)C1 94428,Cc1ccc(CN(CC(N2CC(NC(C3CCCC3(C)C)=O)C(C)C2)=O)C)cc1 94429,C1(OC)CCC2(C(N3CC(NC(=O)C(C)OC4CCCC4)C(C)C3)=O)CC12 94430,C12(NC(c3cncc(OC)c3)=O)CCCN(C(=O)Cc3ccsc3)CC1C2 94431,c1(C(=O)NCCN(CC(C)O)C(=O)CC2CC=CCC2)ccc(Cl)c(N)c1 94432,N1(C(c2ccc(SC)cc2)=O)CC2CC1CCN2C(=O)C=Cc1nc(C)cs1 94433,C#Cc1cncc(C(=O)NC(C)C(c2c(F)cccc2F)O)c1 94434,C(c1ccc(F)cc1)=CC(N1CC2CN(C(C3CCCS3)=O)C2C1)=O 94435,N1(C(C2N(C(c3cc(OCC)n[nH]3)=O)CCC2)=O)CC2CCOC2C1 94436,C(=O)(C1=C(C#N)CCC1)N1CCC(C=C)(C(=O)NCC(C)N(C)C)C1 94437,C(=O)(C(C)(C)CC(F)(F)F)NC1C(NC(CCCc2n(C)cnn2)=O)COC1 94438,c1(C(N2C(C(=O)NCC(=O)OCC)CC2)=O)cc2cc(Cl)ccc2[nH]1 94439,Cc1cc(F)cc(C(=O)NC2CCC(NC(=O)C(C)c3cc[nH]n3)CC2)c1C 94440,Cc1cc(F)c(NC(=O)NCCC2CCCN(C)C2)cc1Cl 94441,CC(C)(O)CCN(CCC#N)C(=O)NC1CCN(Cc2ccccc2)C1 94442,N1(C(c2cc(C)on2)=O)CCCC(C)(C(=O)Nc2c(Cl)cnnc2Cl)C1 94443,N1(C(C=C(C)C(C)(C)C)=O)CC2CC1C2C(=O)N(C1CCCC(O)C1)C 94444,C1(C)(CNC(C=NOC)=O)CN(C(=O)COCC2CCOC2)C(C)(C)C1 94445,C1(C(=O)NC2CCC(CNC(CC(C)(C)OC)=O)C2)Cc2ccccc2C1 94446,N1(C(C2(OC)CS(=O)(=O)C2)=O)CC(NC(C2CCCC2C(C)C)=O)CCC1C 94447,C1(C)(C(=O)NC(C2N(C(c3c(C)snn3)=O)CCC2)C)CCN(C)C1=O 94448,C#Cc1ccc(NC(=O)CC2(C)CCN2C(=O)Cc2ccc(OC)cc2)cn1 94449,C(C(C)(C)C(=O)NC(c1ccccc1F)CNC(C1CCCO1)=O)N(C)C 94450,S(=O)(=O)(c1ccccc1-c1cnc(F)nc1)NCc1nccc(C)n1 94451,C1(NC(c2c(C)cc(F)s2)=O)CC2CCC(C1C)N2C(c1ccc(CF)cc1)=O 94452,C1(C(=O)NCCOCCNC(CC)=O)COc2cc(OC)ccc2C1 94453,C1(NC(CCC(C)=O)=O)CCN(C(c2ccc(C(F)(F)F)nn2)=O)C(C)C1 94454,c1(SC)cc(F)ccc1C(=O)NC(C)CCCCNC(C12CCC(C)(CO1)C2)=O 94455,C12(CNC(C(COC)(F)F)=O)CCCC1N(C(c1c[nH]c(=N)s1)=O)CC2 94456,C#CCC(CC(F)F)C(=O)NCc1ccc(CNC(C2(C)CCCO2)=O)cc1 94457,c1(C(=O)NCC(CC(C)C)NC(=O)C(F)CC2CC2)cccc([N+](=O)[O-])c1 94458,C1(OCCCCC)CCCC(OC(=O)Cn2nnnc2C)C1 94459,c1(CC(=O)N(CC(C)(C)Nc2ccnc(COC)n2)C)c[nH]c2ccccc12 94460,CC1CCCN(Cc2ccccc2F)C1NC1CCN(C(c2ccccc2)=O)CC1 94461,c1(NC(C2(CC#C)CCCO2)=O)nc2ccccc2c2nc(C)nn12 94462,c1(C(N(CCC(C)NC(c2cnc(OC)s2)=O)C)=O)cccc2c1CCO2 94463,c1(CSc2ccc(OC)cc2)c(C)o[nH]c1=NC(=O)c1nnn2c1C(=O)NCC2 94464,c1(C(=O)NCC2C(C)CN(C(=O)Cc3cccc(Cl)c3)C2)ccnc2[nH]cnc12 94465,N1(C(CCCC)=O)CC(NC(=O)CNC(c2ccc(C)s2)=O)C(C)C1 94466,C1(CC2CCN(C(c3ccc(COC)cc3)=O)CC2)(NC)CC(O)C12CCC2 94467,N1(C(Cn2c(C)cc(C)n2)=O)CCCN(C(c2cn(C(F)F)cn2)=O)C(CO)C1 94468,C1(NC(C2C(COC)C2)=O)CCN(CCNC(c2ccc(Br)o2)=O)CC1 94469,c1(C(=O)NCC2(F)COCCN(C(=O)C=CCO)C2)cccc2c1CCCC2=O 94470,c1(C(C)NC(C2(F)CN(C(C(C)SC)=O)C2)=O)cncc(F)c1 94471,C(=O)(C1=COCCC1)NC(CC(=O)NCC(CC(C)O)C)(C)C 94472,C1(CCC)CC(C(=O)NCC2CCCCN2C(=O)Cc2cccs2)CCO1 94473,c1(N(CCCF)C)nc(=N)[nH]c(=NC2CC2C(C)(C)C)[nH]1 94474,CC1(C)CCOC1CC(N1C(CNC(C2CNC(=O)N2)=O)CC2CC12)=O 94475,C(=O)(C1=CC2CCCCC12)NC(c1ccccc1)CNC(C(=C(C)C1CC1)F)=O 94476,c1(C(=O)NCC(C2CCCN2C(c2cc[nH]n2)=O)(C)C)cnc(Cl)[nH]1 94477,C1(NC(c2nc(C(C)OC)oc2)=O)CCC(NC(C2CC2F)=O)CC1 94478,c1(C(=O)NC2CC2NC(C2CC(=O)N(C3CCCC3)C2)=O)csc2c1CCCC2 94479,c1(N2CC(C(=O)NC)OCC2)nc2c(c(=NCCC3CC3)[nH]1)CCC2 94480,N1(C(CC(CC)CN(C)C)=O)CCC(N=c2nc(C(F)(F)F)[nH]s2)C2(CCC2)C1 94481,CC#CCC(C(=O)NCCC(C)CC)NC(=O)C(=O)N(C)C 94482,N1(C(CNS(CC)(=O)=O)=O)CCCC(CCNC(C2CCCO2)=O)CC1 94483,c1(OC)ccc2cc(C(N3CCC4CN(S(=O)(=O)CC(C)C)CC34)=O)ccc2c1 94484,c1(OC)nc(C)ccc1C(N1CC(NC(=O)Cc2nnc(C)o2)C(C#N)C1)=O 94485,Cn1cnc2c[nH]c(=NCCC3CCCN3C(c3ccc(NC(N)=O)nc3)=O)nc12 94486,N12CC3CN(CC3C1)CC2=O.C1(CCC(=O)NC2CC3(CC3)C2)CCCCC1 94487,C(=O)(CCCCCCCC1CC1)NCC(C)NC(c1c(C)ccs1)=O 94488,N1(C(C2C(=C)C2)=O)CCCC2(C1)C(NC(=O)C(C(F)(F)F)C(F)(F)F)CCN2C 94489,C1(CC)CCCN(C(=O)Cc2ccoc2C)C1C(=O)NC1CN(C)NC1=O 94490,CC1CCCC=C1C(=O)N1CC2(CCCC2NC(c2cnc3nccn3c2)=O)C1 94491,CC(C)(C(=O)NCC1CC(F)(F)CN1C(c1ccoc1Br)=O)C(F)F 94492,CCC1=C(C(=O)NCC2CN(C(=O)C(C)c3ccco3)CCO2)CCCO1 94493,Cc1cc(SCC(=O)NCC(C)(CO)NC(C2CC(C)CCO2)=O)cc(C)c1 94494,CCC(CC(=O)NC1CC1CNC(=O)CN(C)C(N)=O)C(C)C 94495,c1(C(N2CC(Cn3cc(-c4c(C)nn(C)c4Cl)nn3)C2)=O)cc(S(N)(=O)=O)co1 94496,C(=O)(C(C)CCCOC)NC(CCCCNC(C(C)N(CCCCCC)C)=O)C 94497,c1(C(=O)NCC(CNC(CCC(CC)OC)=O)CO)c(C)cc(C#N)cc1C 94498,n1(CC)nc(C)c(C(=O)NC(CNC(c2sccc2C)=O)CO)c1C(F)F 94499,N1(C(C(=O)NCc2ccc(C(C)=O)nc2)=O)CCN(C(=O)CNC2CC2)CC1 94500,c1(NC(=O)C(=O)NCc2cscc2Br)ccc(CCOCC(=O)N(C)C)cc1 94501,C1(C(=O)NC2(C(N3C(C(C)O)COCC3)=O)CC2(C)C)Cc2ccccc2C1 94502,[N-]=[N+]=NC1CC(C(=O)NCCc2cscn2)N(C(=O)C#CC2CCOC2)C1 94503,N1(C(=O)NC(C)Cc2c(Cl)cccc2Cl)CC(=O)N(C)CC1C(=O)O 94504,CC1CN(C(C2CN(C(=O)CCC3(C#N)CCC3)CCO2)=O)Cc2c[nH]nc21 94505,c1(C(=O)NC(C(C)C)Cc2ccc(F)cc2)ccc(N2CCCC2=O)c(Cl)c1 94506,Cc1ccc(-n2nc(CCSc3ccccc3)nc2-c2ccccc2F)c(C)c1 94507,CC1(C(=O)NCC2OCCC2C(=O)NCCOCC2CCC2)CC(C#N)C1 94508,Cc1cccc(Br)c1C(C(=O)NCC(C)C(C)(C)C)NC(C1CCCSC1)=O 94509,C=CC(CC)CC(=O)NCC12CC(CO1)N(c1nc(Cl)c(C#N)s1)C2 94510,C=CCCCCCC(C)(c1nnnn1CCCOC)NC(C)CCCC(C)C 94511,C(C)(C)(CN=c1[nH]cnc(NCCN2CCCCC2C)c1C)c1ccc(C)cc1 94512,C1(C(=O)NC(C)CNC(=O)CCc2cncc(F)c2)Cc2nn(C)cc2C(=O)N1 94513,C12(C(N3C4(CNC(c5c(C)snn5)=O)CC(C3)C4)=O)CC(C)(C1)OC21CCC1 94514,CCC1=NOC(C(=O)NC(CNC(c2cnn(CC)c2C2CC2)=O)CC)C1 94515,C1(C(=O)NC2CC(NC(c3c[nH]c(=NC)s3)=O)C2)CCc2c[nH]nc2C1 94516,Cc1cc(CO)oc1C(N1CC2CC2(NC(c2cocc2Br)=O)C1)=O 94517,CN1CCOC(C(=O)N(C)CC2COCCN2C(c2csc(Cl)c2)=O)C1=O 94518,C1(CC(N2C(C(CNC(COC(CC)(C)C)=O)O)CCC2)=O)COCCN1CC 94519,Cc1csc(C(N2CCCC(C(C)NC(C34CC(CCO3)C4)=O)C2)=O)c1C 94520,C1(C(=O)NCCCCC(=O)NC(CC)CCCO)CCOC(=O)CC1 94521,c1(OC)ccc(C(C)(C)C(=O)N(CC(O)CO)C(C)C)cc1OC 94522,C1(C(N(CC(C2CC2)OC)C)=O)CC2(CC2)CN1C(c1n[nH]c(O)n1)=O 94523,C1(CCC)CN(C(=O)CC(C)CC)CCN1C(=O)CN1CCC(C)CC1 94524,C1(CCC)(NC(=O)CCC2CC2C)CCN(C(C2CC3CCC3C2)=O)CC1 94525,c1(C(=O)C2CC2)cc(C2CC2)nn1NCC1C(NC(C(C)Oc2ccccn2)=O)C1 94526,N1(C(C2CC(CF)C2)=O)CCC(Cn2cc(C3COCC3O)nn2)C(F)(F)C1 94527,CCCC(CC)C(=O)NC1(CO)CCCN(C(c2cc(C(CC)CC)no2)=O)C1 94528,N1(C(CC2CC(=C)C2)=O)CCCC2(CC(NC(=O)CC3(C)CCCC3)CO2)C1 94529,C(=O)(CCC(F)(F)F)N(CC(C)NC(=O)C(C)CC1CC1)CC 94530,C1(C(N2CC(C)C(NC(=O)CS(N)(=O)=O)CC2)=O)CC12CCc1ccccc12 94531,C(=O)(CCCC(=O)OC(C)C)N(CCCNC(C(COC)OC)=O)C 94532,c1(CN)ccccc1-c1cn(CCC(=O)NC2CC3CC3C2)nn1 94533,C1(NC(c2cnc(C)nc2O)=O)CC2CC(C1)N(C(C1CN(C(N)=O)C1)=O)C2 94534,n1(CC(=O)OC(C)(C)C)cccc(Nc2cccc(CC(=O)O)c2)c1=O 94535,c1(C(N2CC3CC2CCC3NC(=O)C(F)(F)CC2CC2)=O)cccn2ccnc12 94536,N1(C(C(C)(C)NC(=O)OC)=O)CCC(C2CC2)(CNC(=O)C=CC2CC2)C1 94537,C1(C)(CNC(C(C)OCCC=C)=O)CCCN(C(c2cn(C(F)F)cn2)=O)C1 94538,O=C(C1CCCOc2ccccc21)NC1COCC1n1cc(-c2ccsc2)nn1 94539,c1(CNC(c2c(C)cnn2C)=O)ccc2c(c1)CCC2NC(=O)CSC(F)(F)F 94540,c1(C(=O)NC(C2(CNC(C3CC(SC)C3)=O)CC2)C)cc2ccncc2c(O)n1 94541,N1(C(CCSCCCC)=O)CC2CC2(NC(c2oncc2C)=O)C1 94542,C1(C)CCN(C(c2ccc(CN)[nH]2)=O)CC1.C1(C(=O)OC(C)C)(COCC=C)CC1 94543,N1(C(c2nn(C)c(F)c2)=O)CCCCCC1CNC(C1C2CCCCC12)=O 94544,c1(C(N2C3(CNC(C(CC)F)=O)CC(C2)C3)=O)nc(C(C)C)ncc1Br 94545,C1(C(F)(F)F)CCC(F)(CNC23CC4CC2C3C4)C1 94546,c1(C(=O)NC2(c3ccccc3)CN(C(C3C4COCC34)=O)C2)n[nH]c(O)n1 94547,c1(C(=O)NC2CC3(C(NC(CN4C(C)CCC4)=O)C3)C2)ccnc2[nH]c(O)nc12 94548,n1(CC(N2CCCCCC(NC(C(C=C=C)C)=O)C2)=O)[nH]cc2c(=O)ncnc1-2 94549,C1(C(=O)NCC(CNC(CC(C)OC)=O)O)CC(=O)N(C(C)C2CC2)C1 94550,CCCCC(CC)C(=O)NC(C)CCNC(c1sccc1SC)=O 94551,Cc1cc(C(N2CCNC(C(=O)NC3CC(O)C3)C2)=O)cc(C#N)c1 94552,c1(C(=O)NCCC2(O)CN(C(CSCC)=O)C2)sc2cncn2c1C 94553,c1(CNC(C2CCN(CC(C)(C)C(=O)O)CC2)=O)ccc(F)c2[nH]ncc12 94554,N1(C(C(CCF)NC(c2cc(C)ns2)=O)=O)CCCC(C)(O)C1 94555,C1(NC(CC)=O)CCCC12CCN(C(=O)COc1ccc(F)c(F)c1)CC2 94556,c1(C(=O)NC)cccc(F)c1-c1cnc(F)c(C(N2CCC(F)(CO)CC2)=O)c1 94557,c1(C(=O)NC(c2cccc(N)n2)C)cnc2n1CCOCC2 94558,C(=O)(C(C)(C)CC(F)(F)F)N(CC(CNC(c1c(OC)n(C)nc1)=O)C)C 94559,CCC(C)(O)C(=O)NC1C=CCN(C(c2cn(C)nc2C)=O)C1 94560,c1(CC(=O)NCC(C(=O)NCCCC2CCC2)N(C)C)ccc(O)cc1 94561,CCC(CC)C(F)C(=O)NC(CC1CCCC1)C(=O)N(C1CCC(F)(F)C1)C 94562,C1(C(=O)NC(CN(C(=O)CCCCSC)CC)C)COCCN1C 94563,C12(C(=O)NCC3(CNC(Cc4c(C)ncs4)=O)CCCC3)CC(C)(CO1)C2 94564,C(CN=c1[nH]c2c(c(=NC3CC(n4cccn4)C3)[nH]1)CCC2)N(C1CC1)CC 94565,Cc1cc2ncc(C(=O)NCC(C)NC(=O)CN3CCCC3C)cc2[nH]1 94566,N1(C(CCC=C)=O)CCC(CO)(NC(=O)Cc2csc(-c3cnccn3)n2)C1 94567,c1(CN2C(CC(=O)OC)CS(=O)CC2)cc(Br)c(C(F)(F)F)cc1F 94568,C1(CNC(=O)C(O)CN2CCCC2)CCN(C(c2cc(CF)on2)=O)CC1 94569,N1(C(C(C)NC(CC)=O)=O)CCC(C(=O)NC2CC(O)(CO)C2)(CF)C1 94570,c1(CNc2ccc(OC)c(Br)c2F)cnc2c(c1)c(C)nn2C 94571,C1(=O)C(C2CN(C(=O)OC(C)(C)C)C2)OCCN1C.CCCN(C)CCOC.SCC 94572,C1(CNC(CC(CC)OC)=O)CC2COCC2N1c1nnc(C(F)F)s1 94573,c1(C(C)NCCCN(C(=O)OCC)C)cccn1Cc1ccccc1 94574,c1(NC)cccc(C(N2CC(CN3CCN(C(=O)C(C)CO)CC3)C2)=O)n1 94575,C1(NC(CN2C(C)CC2)=O)COC2(C1)CN(C(c1cnc(C3CC3)[nH]c1=N)=O)C2 94576,N1(C(C2CN(C)C2)=O)CCCC1C(=O)N(C)Cc1nnc(O)o1 94577,c1(C(=O)NCC2(O)CN(C(C(C)Sc3nncn3C)=O)C2)nn(C)cc1N 94578,c1(OC)ncc(C(=O)NCCOC2CN(C(=O)C(c3cccnc3)=O)C2)s1 94579,c1(Nc2c(C)c(Br)cnc2)ccc(F)cc1[N+](=O)[O-].C12C=CC(C1)NN(CC)C2=O 94580,c1(NC(C)CC(C)NC(C2CCC3CC3CC2)=O)c([N+](=O)[O-])cnn1C 94581,c1(C2(N(CC(=O)O)Cc3cnc(CCCC)[nH]3)CC2)ccc(F)c(F)c1 94582,n1(CCCSC)nnnc1C(NCc1ccccc1)CNCCO.C1(C)CC1 94583,C1(CCNC(C(COC)C)=O)CN(C(=O)C(F)=C(C)C)CCCO1 94584,c1(OC)cccn2ncc(C(=O)N(C3CN(C(=O)CN4CCC4C)CC3O)C)c12 94585,c1(OC)cc(CC(=O)N(CCNC(=O)CC(C)(F)F)CCC2CC2)cc(F)c1 94586,c1(C(N2CC3CN(C(C4CCN(C)C4=O)=O)C3CC2)=O)ccc2c(c1)OCCC2 94587,c1(C(=O)NCCN(C(=O)C(c2ccc(F)cc2)C)CC)ccc(F)c2c1OCC2 94588,C12(CNC(c3cn(CCC)nc3)=O)CC1CN(C(=O)CC1CCC1(F)F)C2 94589,C1(C(N2CCN(C(CNC(=O)CC(F)(F)F)=O)CC2)=O)CCc2nc(O)[nH]c2C1 94590,Cc1c(C(=O)NCC2(CC(N3CCCC3C(N)=O)=O)CC2)[nH]ccc1=O 94591,Cc1noc(C)c1C(=O)Nc1ccsc1C(=O)NC1CC1(F)F 94592,c1(N(c2ccccc2)C(c2c(C)nc(C)[nH]2)=O)ncc(Br)c(C)n1 94593,CC1(C(N2CC(CO)C(c3ccccc3)C2)=O)Oc2ccccc2NC1=O 94594,N1(Cc2ncn(C)n2)CC2C3CCC(C2C1)N(C(c1cc(O)cc(=O)o1)=O)C3 94595,c1(NC(C2COCCN2C(C2CC2C2CC2)=O)=O)cc(F)ccc1Br 94596,N(C(=NCCc1cnccn1)NCCN1CCCC1)CC1(C)CCCCO1 94597,C1(O)(CNC(CC(CC)C)=O)CC2CCC(C1)N2C(c1cc(C)nc(O)c1)=O 94598,C1(CCNC(C(C2CCCN(C(C3C4CN(C)CC34)=O)C2)C)=O)CCCC2CC12 94599,C1(C(=O)NC2C(NC(Cc3c(C)cco3)=O)CCCC2)CN2CCN1C(C)C2 94600,C1(CCC)CN(C(c2nc(C)oc2OCC)=O)CCN1C(c1cc(=O)cc[nH]1)=O 94601,c1(C(=O)NC(C)(CNC(c2cn[nH]c2)=O)Cn2cccn2)cccc2scnc12 94602,c1(CC(C(=O)NC(c2nccn2C)C)N)cc2cc(Br)ccc2o1 94603,c1(C(=O)NCC(CC(=O)N(C)Cc2c(C)nco2)C)ccc(F)c(F)c1 94604,c1(C(=O)NCC(=C)CCNC(=O)Cc2occc2C)ccccc1SCC 94605,C1(C(=O)NCCC2CSCCN2C(=O)C(C)N=[N+]=[N-])(CC)CC(C)(C)C1 94606,N1(C(CC(CC)(C)C)=O)CCCC12CCN(C(=O)CCc1cc(C)n(C)n1)C2 94607,C(=O)(C(C)(C)C(=O)N1CC2C(OC)C2C1)NCCOc1c(OC)cccc1 94608,c1(CNC(CC(C2CC2)NC(c2cnc(C)o2)=O)=O)ncc(Cl)cn1 94609,c1(COC)ccc(C(=O)NC2CN(C(=O)CCCN(C)C(=O)OC)CC2O)cn1 94610,c1(C(=O)NC(CC)(CNC(=O)C(F)(F)COC)CC)ccc2cccnc2n1 94611,C12(NC(C3CC34CCC4)=O)CC(C(=O)OCc3snnc3C3CC3)(C1)C2 94612,C(C)(C)(CCNC(=O)Cc1cc(C(C)C)no1)NC(COCC(=O)NC)=O 94613,CCCC1=C(C(=O)OC)C(c2cc(CN)nn2C)NC(=O)N1CCOC 94614,CC(=O)CCC(=O)N1CCC(C(C)C(=O)N2CC(N(C)C)C2)C1 94615,C1(NC(CN2CC(C)(C)C2)=O)CN(C(c2cc(C3CC3)oc2C2CC2)=O)C2CC12 94616,c1(C(=O)NCCN(C(=O)CCOCC2CCCO2)C)cc2cccc(F)c2s1 94617,C(C(C(=O)NOCCCCF)NC(c1ccc(C)nn1)=O)SCC 94618,c1(OC)c(Cl)ccc(C(=O)NCC2CC(C)CCN2C(C23CC(OC)C2C3)=O)c1F 94619,N1(C(C(CCC)(C)CC)=O)CC2(C1)CN(C(c1csc(C)c1C)=O)CC2CO 94620,Cc1cc(C(N2CC3CCC2C(NC(=O)C(F)C2CCOC2)C3)=O)c(Cl)cc1F 94621,c1(CC)ccc(C2(C(N3CCC(N(C(=O)COCCF)C)C3)=O)CCCC2)cc1 94622,Cc1cc(F)ccc1OCCCNCCOCCN(C)CCN(C)C(=O)C1CC1 94623,c1(C(N2CCC(c3ccco3)C2)C(=O)NCCSC)cccc(C(F)(F)F)n1 94624,Cc1ccc(C(=O)NCCNC(N2CC(CO)CC2C)=O)cn1 94625,c1(COC)cc(NCC2(CC3CC3)CCOC2)cc(Cl)c1C#N 94626,c1(OC(c2nccn2C)C)ccc(NC(C2CCC(C)(C)CO2)=O)cc1Cl 94627,CCCCC(O)CC(=O)N(C(CC)CC(N1CCC2(CCCO2)C1)=O)C 94628,c1(C(=O)OC)ccc(NC(C2CC(O)CN2Cc2ccsc2Br)=O)cc1Cl 94629,c1(C(=O)NC23CCN(C(c4c(C)cc(C)o4)=O)CC2C3)ccc2occ(C)c2c1 94630,N1(C(COCC)=O)CCCC2C1CCN2c1ncc(Br)c(OC)n1 94631,C(=O)(C1=CCSC1)N(CC)CC1CCCCN1 94632,C1(C(=O)NCCCn2cc(CC3CCNC3=O)nn2)C2Cc3cc(Cl)ccc3C12 94633,c1(C(N(C)CC2CCCN(C(c3c(C)cn(C)n3)=O)C2)=O)cc2cccnc2s1 94634,N1(C(c2cncc(OC)c2)=O)CCCC(C)(C(N2C(C)CCC2(C)C)=O)C1 94635,C1(NC(C2C(OC)CC2)=O)CCCC(NC(c2nc(OC)c(C)s2)=O)C1 94636,C=CC(C)(O)C(=O)N1CC(NC(=O)CCOCC)C(C(F)(F)F)C1 94637,CN1CCN(C(=O)C(C)(C)n2cnnn2)CC1CNC(=O)C(C)(C)C1(O)CCC1 94638,C=C(C)CC(C(=O)NC(c1cccc(F)c1)C)NC(=O)C(=O)NCC(F)F 94639,c1(C(=O)NC2C(NC(c3ccn(CCOCCOC)n3)=O)C2)ccc(C)nc1 94640,c1(CCC)nc(=NC2(CNC(C3CCC4(CCOCC4)O3)=O)COC2)s[nH]1 94641,c1(N2CCC(C(C)(C)C)CC2)nc(N2CCC3C(C2)C3(F)F)c2[nH]ccc2n1 94642,C1(OC)(CNC(C2CC2C)=O)CCN(C(c2sccc2CC#N)=O)C1 94643,c1(C(N(C(CNC(C2CCN(C(CC)=O)C2)=O)C)C)=O)cc([N+](=O)[O-])cc(C)n1 94644,C1(NC(C2CC(C(F)F)C2)=O)CN(C(c2ccc(N3CCC3)nc2)=O)CC1CO 94645,c1(N2CC(CN(C)C(c3c[nH]cc3Br)=O)C2)nc(Cl)nc2c1ncn2C 94646,c1(C(N2C(NCc3onc(C)n3)COCC2)=O)ccc(S(N)(=O)=O)o1 94647,c1(C(=O)Nc2c(C)n(-c3ccc(OC(F)F)cc3)nn2)cn2cc(F)ccc2n1 94648,CC1SCCN(C(=O)C(C)(C)C2CCN(C(=O)C#CC3CC3)C2)C1C 94649,CC1=C(C(=O)NCC(C)(F)CNC(C2(C(C)C)CNC(=O)C2)=O)C(C)(C)CCC1 94650,c1(C(N2CCN(C(C(CC)CC)=O)C(C(C)(C)C)C2)=O)ccc2c(c1)COCO2 94651,C(=O)(CCC(=O)NCCSCC(N1CCC(C2(C)N=N2)C1)=O)NC 94652,Cc1cc(N)c(C)nc1C(=O)NC1CCN(C(=O)Cc2ccc(F)cn2)C1 94653,CN1CCN(C(=O)CC2CCCCO2)C(CNC(C2C(C)(C)C2(C)C)=O)C1 94654,c1(C(=O)NCC=C2CCN(C(c3cnc(C)n3C)=O)CC2)cnn2c1N(C)CC2 94655,n1(CC(=O)NCC(CNC(CN(C2CCSC2)C)=O)F)nnc2ccccc12 94656,N1(C(c2scc(C)c2Cl)=O)CC2(CCCC2NC(c2cccc3nonc23)=O)C1 94657,c1(C(=O)NC(C(=O)OC)Cc2cn(-c3cnn(C)c3)nn2)cccc2nccn12 94658,C1(CNC(C(=Cc2ccccn2)C)=O)CN(C(=O)Cc2csc(Cl)c2)CCCO1 94659,C1CCCCCN1.c1(C(C(=O)OCCO)(F)F)cccc(C(F)(F)F)n1 94660,c1(C(=O)NCc2c(C)c(Cl)ncc2)n[nH]c2c1CN(C(C1CC1C)=O)CC2 94661,c1(C(=O)NC2(CCCNC(C(CCCOC)C)=O)CC2)cc(O)c2ccsc2c1 94662,c1(N(CCCC)C)ncnc2c1ncn2CC(C)(Cc1ccccc1)CO 94663,C1(CNC(c2ccc(C(F)(F)F)o2)=O)CC2CC2N1C(=O)CC12CCC(CC1)C2 94664,C(=O)(CCS(C)(=O)=O)N1C(C)(C(=O)NC2(COCC)CC2)C=CC1 94665,N1(C(C(OC)OC)=O)CCN(C(=O)CCCSC)CC(CO)C1 94666,C(=O)(C(CN(C)C)C(C)C)N1CCC(N(C(C2(C)CCCN2)=O)OCC)C1 94667,C=C1CC(C(=O)NC2CCCSC2)(CNC(=O)C(C)n2cccc2)C1 94668,O=C1CCOC(C(=O)NCC2CC(F)(CNC(=O)C(F)n3ccnc3)C2)C1 94669,C1(C(=O)NCCCCC2(NC(C3CCCN(CC)C3)=O)CC2)CC(=O)NC(=O)C1 94670,N1(C(C(=O)NCCC2(C)CC2)CC2(C)CC2)CCC2(CCCCO2)C1 94671,CCC(CCC(=O)N(C)CC1(CO)CC1)NC(c1cn(CC)nc1C)=O 94672,C1(NC(c2csc3nccn23)=O)CC(C(=O)O)C12CCOCC2 94673,c1(C(=O)NCCCCN(C)C(C2CCC(=O)N2)=O)ccc2scnc2c1 94674,N1(CC(=O)NCC2(O)CC(NC(c3ccc(CC)o3)=O)C2)CCCCCC1=O 94675,Cc1nc(N(C2(CN)COC2)Cc2ccnc(C)n2)cc(O)n1 94676,N1(C(Cn2c(CCC)nnc2S)=O)CC(C(N)=O)CC(C)C1 94677,Cc1nccc(C(=O)NC(CCC2CC2)C(=O)NCC2(CO)CCCO2)c1C 94678,c1(OCC(=O)NC2(CC=C)CCOC2)cc(C)cc(C)c1 94679,CC1CCN(C(C2CCCOC2C)=O)CC1CNC(=O)C(c1ccccc1Cl)O 94680,N1(C(CC=CC=C)=O)CCC(OCC(=O)N(CC(C)OC)C(C)C)C1 94681,c1(OC)n[nH]c(NC(C2CC23CCN(Cc2cnc(O)c(Cl)c2)C3)=O)c1C#N 94682,CN1CCN(C(C2CC2C)=O)C(C(=O)NOC2CCCC2)C1.C1(=O)CN1 94683,c1(C(N2CC(NC(C(C)C3CCOC3)=O)(CO)C2)=O)coc2c1CS(=O)(=O)C2 94684,N1(c2ncc(C(=O)OC)s2)CCOC(C)(CNC(=O)CSCc2cccnc2)C1 94685,N1(C2CN(C(C=C(C)Cl)=O)C2)CCN(C(c2ccc(CCC#N)cc2)=O)CC1 94686,C(=O)(C1CCCn2cnnc21)N1C(CNC(c2c(Cl)cncc2Cl)=O)CC1 94687,c1(C(=O)NC2C(CNC(=O)CCCF)C2)ccc([N+](=O)[O-])c(C(N)=O)c1 94688,c1(C(c2n(CCOC)nnn2)NCC2(Br)CC2)nc(Br)cn1C 94689,c1(C(=O)NCC2C(CNC(C3CC(CC)OCC3)=O)C2)nc(N(C)C)nc(=N)[nH]1 94690,c1(C(=O)NC(COCC)C(=O)N2CCC(O)C2)ccc([N+](=O)[O-])[nH]1 94691,N1(C(C(C)(C2CC2)OC)=O)CCC2(CC1)CC(NC(=O)C=CC1CC1)CCO2 94692,C1(F)(C(N2CCC(CC(C)O)CC2)=O)CCN(C(c2ccsc2C#N)=O)CC1 94693,C(=O)(CCCCCF)NC(CC)CNC(=O)C=Cc1nnc(C(C)C)o1 94694,c1(C(=O)NCC(C)(C2CC2)NC(CC(CC)C)=O)cccc(-c2ccccc2)c1O 94695,C1(NC(C2=CC(C)C2)=O)CCC12CCN(C(=O)Cc1cnnn1C)CC2 94696,N1(C(C2(C)CCC(C)C2)=O)CC(C2CN(C(c3nn[nH]c3C(F)(F)F)=O)C2)C1 94697,C1(C(=O)O)(NC(Cn2cc(C(=O)OC)nn2)=O)CC2CCC12 94698,c1(OCC)cccc(CC(=O)NC(C)CNC(=O)CC2COC3CC2C3)n1 94699,C(CCC(C)(C)NC(=O)C(c1ccc(C)s1)C)NC(C(C)NC(COC)=O)=O 94700,C(=O)(C1=C(Cl)CCC1)NCC(C)(C(=O)O)OC 94701,N1(C(=O)CC(F)(F)F)CC2(C1)CN(C(C1C(C3CC3)C1(F)F)=O)CCO2 94702,c1(C(=O)NCC(CC)(CC)NC(=O)CCCC#N)sc2nccc(C)c2c1C 94703,C1(C(N2CC=CC(NC(C3N(C)C(=O)CC3)=O)C2)=O)CC2(C1)OCCO2 94704,N1(C(=O)OC(C)(C)C)CC2(C(F)F)CC1(C(=O)N1CC(O)CO1)C2 94705,CCC1CN=C2C=CN=C(N2)N1.C(CS(=O)(=O)N(C)C)NC(=O)OC 94706,c1(OC)cc([N+](=O)[O-])ccc1C(=O)NC1CC1C(=O)Nc1c(C)cc(Cl)nc1Cl 94707,C1(C(=O)Nc2cn[nH]c2)CCN(Cc2cnn(-c3ccccc3)c2)C1 94708,C(=O)(C(C)C(F)(F)F)N1CC(NC(C(c2c(OC)cccc2)O)=O)C(SC)C1 94709,CC1CC(NC(=O)C#CC(=O)N(C)C)CN(C(=O)C(n2cc(Cl)cn2)C)C1 94710,CC1(C#N)CN(C(C2NCC3CCCC23)=O)CCO1 94711,C(=O)(C#CC1CCCCO1)NC(CNC(C(CCCC)O)=O)(CC)CC 94712,C1(C(N(CCN(C)C(C2CCS(=O)(=O)C2)=O)C)=O)CC(=O)CC12CCC2 94713,C(=O)(C(C)(CC)CC)N1CCCC(N(C(C2CC(CC(F)F)C2)=O)CC)C1 94714,c1(OC)ccnc(CNC(C2(CNC(=O)CC3CCOC3=O)CCCCC2)=O)c1 94715,C1(C(N2CC(F)(CNC(c3nc[nH]c4ncnc3-4)=O)C2)=O)CN=C2N=CNN2C1 94716,N1(C(c2c[nH]c(=NC)o2)=O)CCCCC(CNC(C2CCC23CCC3)=O)C1 94717,CC(CF)CC(=O)N1CCCC(N(C(=O)C(C#N)=CC2CC2)C)C1 94718,N1(NC(C2(CCO)CCCC2)=O)CC(F)(F)C(F)(F)C1.C12CC(C1)C(=O)NC2 94719,CC1(C)CC2(CC(C(=O)NCC3CCCN3C(=O)Cc3cccc(F)c3F)C2)C1 94720,c1(OCC)nc(C)ccc1C(N1CC(NC(c2cnc(SC)s2)=O)C(O)C1)=O 94721,N1(C(c2ncnn2-c2ccccc2)=O)CCC2C(C1)C2(F)F 94722,c1(C(=O)Nc2c(C)nc(C(F)(F)F)cc2)cnn2ccc(CN)cc12 94723,CS(=O)(=O)CCCC(=O)NCC1(F)CCC(NC(C2CN(S(C)(=O)=O)C2)=O)C1 94724,C1(C(=O)NCC2C(C)(C)CN(C(=O)CSCC(N)=O)C2)COc2ccccc2O1 94725,C1(NC(C(C)OCOC)=O)CCN(C(c2cnn(CC(C)C)c2C)=O)CC1 94726,c1(C2(C(=O)NC(C3CN(C(C(=O)NC(C)C)=O)C3)C)CCC2)ccccc1 94727,c1(C(=O)NCC(C2CCCCN2C(C2CC2(F)F)=O)(C)C)cccc(N)c1 94728,C1(C(=O)NC2CC(C)OC2=O)CN(C(=O)C2=CCCSC2)CC1(F)F 94729,C(=O)(C1=C(C)CCC1)N1C(CC=C)(C(N2CC(c3nncs3)C2)=O)CCC1 94730,C1(CNC(C(N2CCSCC2)C)=O)CCC(CNC(=O)Cc2cn[nH]c2)CC1 94731,C1(NC(c2cc(C(F)F)no2)=O)CC2CN(C(=O)Cn3nccn3)CCN2C1=O 94732,CCCCCCC(F)C(=O)NCC#CCNC(=O)Cc1nc(C)sc1C 94733,CC(CC(C)(C)C)C(=O)N(CCCN(C)C(c1cc(C(N)=O)no1)=O)C 94734,N1(c2snc(COC)n2)CCC2(CCOC2)C(CNC(C2CC3(C2)CC3F)=O)C1 94735,N1(C(CCNC(=O)NC)=O)CC2(COC(CNC(c3cc(Br)no3)=O)C2)C1 94736,c1(OC)ncc(NCc2ccc(-c3ccccc3OC(F)F)s2)cc1Br 94737,O=C1CCCCC(C(=O)NC2CC(c3ncc[nH]3)C2)C1 94738,N1(C(C(C)OCC(F)(F)F)=O)C2CCC1C(CNC(c1ccccc1)=O)C2 94739,c1(C(=O)NCCC2(OC)CN(C(c3scc(OC)c3)=O)C2)cc(C)cc(O)n1 94740,C1(C)(C(=O)NCCCCC)CCCN(C(c2cccc(OC)c2O)=O)C1 94741,C12(CNC(C3C(C)(C)CC3)=O)CCCC1CN(C(C1CCC(CC#N)CC1)=O)C2 94742,c1(NC(C2C(=C)C2)=O)cccc(CNC(c2ccccc2-n2cccc2)=O)c1 94743,c1(C(=O)NC2CC(CNC(C3CN(C)C(=O)C3)=O)C2)ccc2nc[nH]c2n1 94744,N1(C(C(C)OCC)=O)CCC2(CC1)COC(CNC(=O)Cc1cncc(C)c1)C2 94745,C1(N(C(COCCC#C)=O)C)CC2CC1N(C(=O)CNC(=O)NC)C2 94746,C1(CC)CCN(C(C2CCS(=O)(=O)C2)=O)C1CNC(c1cscn1)=O 94747,O=C(CC1OCc2ccccc21)NC1CCCN(C(c2ccns2)=O)CC1 94748,c1(OC)ccc(S(=O)(=O)N2CCC2C(=O)Nc2ccc(-n3nccn3)cc2)cc1 94749,c1(CC)ccccc1C(=O)N(CCC(C(C)C)NC(=O)CC1CCCC1)C 94750,c12nnc3c(ccc(CCC(=O)O)n13)CN2C.N1(CC)CCCC1C.C(F)(F)F 94751,c1(C(=O)NCCC(=C)CNC(c2cc(O)n(CC)n2)=O)cc[nH]c(=NCC)c1 94752,C1(NC(C(C)OCC(C)C)=O)COC2C(NC(c3cnn(C(C)C)n3)=O)COC12 94753,c1(C(=O)NC2CCN(C(C(n3ncc(C)c3)C)=O)C2)ccccc1CO 94754,N1(C(CN2CC(=O)NCC2)=O)CCC2(CCCC2NC(c2ccccc2)=O)CC1 94755,Cc1nc(O)c(Br)cc1C(=O)NC1(CO)CN(C(=O)C(Cl)=CCl)C1 94756,c1(OCC(=O)NC(CCNC(c2nc(CCC)oc2)=O)(C)C)cc(Cl)cc(Cl)c1 94757,c1(C(C)=O)ccccc1C(=O)N(C)CC1CCCN1C(=O)CC12COCC(C1)C2 94758,C(CCCC)(CC(=O)NC(CO)C(C)(C)CO)NC(CCCC#C)=O 94759,C1(N(C(=O)C2CC2)SCC(=O)Nc2cocn2)CCCC12CCNCC2 94760,c1(C(N2CCC(C3CC3)C2CNC(C2(CF)CC2)=O)=O)ccc([N+](=O)[O-])cc1Cl 94761,CN1CCN(C)C(C(=O)NC(C2(O)CCCCC2)C(=O)NCCn2cnnn2)C1 94762,C12(C(N(C3CCN(C(=O)Cc4cc(Cl)cs4)C3)C)=O)CC3CC(C1)CC(O)(C3)C2 94763,Cc1nc2c(C(N3CC(NC(c4cc(CO)[nH]n4)=O)CC3C)=O)ccnc2[nH]1 94764,c1(OC)cnc(F)cc1C(N1CC(NC(=O)Cc2cc(C)no2)C(C)(C)C1)=O 94765,N1(C(C(CCC#C)O)=O)CC2CCN(C(c3cccc(CC)c3)=O)CC2C1 94766,c1(C(N2CCC(COC)C2)=O)cnc(CNC(=O)C=CC2CCCN2C)nc1 94767,C1(C)(COC(c2sc(Cc3ccc(C)cc3)c(Br)c2)=O)CCCCC1C 94768,CC(C)C(CNC(=O)C(c1cncnc1)C)C(=O)NCc1ccc(C#N)cc1 94769,c1(C(=O)NCCN(C(C2COC3(C)CC2C3)=O)CC)c(C)cccc1C 94770,C1(NC(c2n(C(C)C)ncc2F)=O)CC(O)CN(C(C2CCN(C)CC2)=O)C1 94771,c1(C(N2CC(OC)C(NC(c3occc3C)=O)C2)=O)ccnc2cc(F)cnc12 94772,CN1CCCC2CN(Cc3cc(N4CCCC4)nc(F)c3)CCC12 94773,c1(C(N2CC(n3cc(C(CC(C)C)O)nn3)C2)=O)ccc(Cl)c(F)c1 94774,N1(C(c2c(C)cns2)=O)CCC2CCC(NC(c3cc4ncccc4s3)=O)C1C2 94775,CC(C)C(F)C(=O)NCC1(F)CC(Nc2ncccc2C(=O)C(F)(F)F)C1 94776,c1(C(N(C2CCN(C(C34CC(C)(CCO3)C4)=O)CC2)CC)=O)cc(=O)cc(C)[nH]1 94777,c1(CN(C(=O)Cc2cc[nH]n2)C)cnn2c1CN(C(C1CCC(C)(C)C1)=O)CC2 94778,C1(NC(CC2CN(C(C)=O)C2)=O)CC2(CCN(C(c3ccc(C)c(Cl)c3F)=O)C2)C1 94779,N1(CCN(CC)CC)CC(O)CC1c1ccc(Br)cc1 94780,c1(CC)cc(C(=O)NCC(O)CNC(c2cnc(C)n2C(F)F)=O)cc(Cl)c1 94781,C1(C(N(C)CC2COCCN2C(C2CCC(=O)O2)=O)=O)CC2CCC1C21CC1 94782,c1(C(=O)NC(C2CCN(C(=O)CC3CCC3)C2)C)cscc1S(C)(=O)=O 94783,Cc1onc(C(=O)NC(CNC(C2CC(O)C2)=O)C(C)C(C)C)c1[N+](=O)[O-] 94784,N(C(=NCCc1ccc(Cl)cc1)N1CCC(CSC)C1)C(CC)CC 94785,C(=O)(C(C(C)(C)C)NS(C)(=O)=O)NCC1(C)N(C(Cc2c(C)ncs2)=O)CCC1 94786,N1(C(C=CC)=O)CCC(NC(c2ccc(N3CCCC3)nn2)=O)C(CC)C1 94787,C1(CCNC(C2(CC)COC2)=O)CN(C(c2ccc(-c3cccs3)o2)=O)CCO1 94788,c1(C(=O)NCC2(C(C)NC(C3N(CC)CCOC3)=O)CC2)ccc([N+](=O)[O-])cc1 94789,CN1CC(CNC(C2CCCC2CNC(=O)C=Cc2cocn2)=O)CC1=O 94790,c1(NC(CCN(C(=O)C(F)C2CCOC2)C)=O)cccc2ccccc12 94791,c1(C(NOCC(=O)N(C)Cc2cccnc2O)=O)cccc2[nH]ccc12 94792,C1(CC(=O)N(C2CCCC2)CC#CC)CC(NC(=O)CNC(=O)NC)C1(C)C 94793,c1(C(N(CCC(C(C)C)NC(COC(C)C)=O)C)=O)cc2n(n1)CCCC2 94794,c1(C(=O)NC2C(CNC(C3(CC=C)CC3)=O)C2)c[nH]c2ccc(Cl)cc12 94795,CC1CC(O)CN1C(=O)NC(C1CC(F)(F)C1)C(F)F 94796,N1(C(CCC=C=C)=O)CC2(CO)CC1(C(=O)NCCc1ccccc1F)C2 94797,c1(CNC(C(Cc2cc(C)c(O)cc2)N)=O)cnn2c1CCCC2 94798,Cc1ccc2cccc(C(=O)N(C3CN(C(c4cnc(Cl)cn4)=O)C3)C)c2n1 94799,Cc1sc2ncc(C(=O)NCC3(NC(c4cc(Br)co4)=O)CCC3)n2c1C 94800,CS(=O)(=O)c1ccnc(NC2C3CN(C(c4cc(Cl)on4)=O)CC23)n1 94801,C(=O)(C1=CCC(C)(C)CC1)N1CCC(CC)C1C(=O)NOC(CC)CC 94802,N1(C(c2c(C)ncn2C)=O)CC=C(CNC(=O)C(C)OCCC(C)C)CC1 94803,C(=O)(C(C(=O)NC1(CN(C(=O)C(C)n2cncn2)CC)CC1)C(C)C)OCC 94804,C(=O)(C1=C(C)OCC1)Nn1c(N2CCN(CC(=O)NC)CC2)nnc1C1CCC1 94805,CC1CCCC1N(C)C(C1(CCNC(=O)Cc2ccsc2)CCC1)=O 94806,C1(NC(C(COC)(C)OC)=O)CCCCCN(C(c2ccccc2Cl)=O)C1 94807,C(CCC(C)C)(C(=O)Nc1ccc(N(C)C)cc1)NC(C(CCC)CC)=O 94808,N12CCC3(CC1)CC(C)N(C3)CCN(C)C(=O)C2.CCS(=O)(=O)NC1CC(O)C1 94809,N1(C(c2nc(SC)sc2)=O)CCC2(CCC2)C(NC(=O)C(C)n2cccn2)C1 94810,C(C(C)C(=O)NCC1C=CCCC1)N(C(C1(OC(C)=O)CC1)=O)C 94811,N1(C(C(CCCNC(c2n(C=C)ncc2)=O)(C)C)=O)CC(C)OCC(C)(C)C1 94812,N1(C(c2c(C)nns2)=O)C2CCC1C(c1cn(CC(c3ccccc3)O)nn1)C2 94813,Cc1cc(CNC(C2C3CCC2(c2ccnn2C2CCC2)C3)=O)c(C)s1 94814,c1(CC)ccc(C(=O)NC(C)(C)CN(C(=O)COCC2CC2)C)cc1 94815,c1(C(=O)NC(CN(C(=O)C(C(C)C)n2cc(C)cn2)CC)C)cn(C)nc1Cl 94816,c1(CN(C(=O)Cn2cc(C3(C)CCCC3)nn2)C)cc(OCC(F)F)ccn1 94817,N1(C(C2(F)CCN(C(c3scc(OC)c3)=O)CC2)=O)CCCC2(CCC2)C1 94818,C(=O)(C(C)CC(C)(F)F)NCC1(F)CN(C(c2c(OC)c(Cl)ccc2)=O)C1 94819,C1(NC(CSC)=O)CCC2(CC1)CN(C(=O)C=Cc1ccncc1)CCO2 94820,c1(N(C)C)nc(F)ccc1CNc1ccc(C(=O)Nc2ncc(Br)cc2Cl)nc1 94821,C1(C(=O)NC(C(C)(C)O)C2CC2)CCN(C(c2csc(Cl)c2)=O)CCO1 94822,C=Cn1nccc1C(=O)NCC(CC(=O)NCCN(CCCF)C)C1CCC1 94823,c1(C(=O)NCCC(CNC(CC2N(CC)CCC2)=O)O)cc(O)n(CC)n1 94824,c1(C(=O)NC(CC=C)CNC(c2c(C)cccc2C)=O)n[nH]c2c1CC1CC21 94825,C(=O)(C(C)Cc1ccoc1)NC1(CCC(=O)NCC#CC)CCC1 94826,c1(C(=O)NC)cc(=NC2CCCN(CCS(C)(=O)=O)C2)[nH]c2ccccc12 94827,CCC(C)(C#N)C(=O)NCC12CC(NC(=O)CCc3cnccn3)(CO1)C2 94828,c1(C(=O)NCCC(C)N(C)C(c2ncc(Cl)cc2Cl)=O)cnn2c1OCC2 94829,N1(C(C(C)=CC2CC2)=O)CC2CC(C1)CN(C(=O)C(O)(C1CC1)C1CC1)C2 94830,CC1CN2CCN1CC2C(=O)NC1CC(C)(NC(c2ccncc2N)=O)C1 94831,c1(-c2ccc(N3C(=O)OCCC3)cc2)cccc2c1CCN(S(=O)(=O)CCCCCl)C2 94832,C1(C(=O)NCC(C)(C)NC(C(C)SC)=O)CCC(=O)N(C)C1 94833,CC1CCC(CNC(C2CC(CC(F)F)C2)=O)N(C(=O)Cn2ncnn2)C1 94834,CC1CN(C(C2C3CCC(C3)N2C(c2cc(Cl)cs2)=O)=O)CC(=O)N1C 94835,C(=O)(CC(C(C)(C)C)NC(=O)CC1CC2CC2C1)NCC12N(C)CC(C1)C2 94836,c1(CCNC(C(C)NC(c2ccc(Cl)cc2)=O)=O)c[nH]c2cnc(Cl)cc12 94837,C(c1ccccc1)=CC(=O)NCCCOCCNC(C(OC)OC)=O 94838,C1(C(=O)NCCCN(C(C=C(C)Cl)=O)CC2CCCC2)CCC2(CC2)C1 94839,C(=O)(C(C)CC(=O)N1CCC(n2cc(-c3cc(CO)ccc3C)nn2)C1)OC 94840,C(=O)(C(C#N)C(C)(C)C)NC(CC)CN(C)C(C1CCCC1F)=O 94841,C1(C(=O)NCC2(C(N(C)Cc3cc(C)n(C)n3)=O)CCCO2)CCCC1C1CC1 94842,CC(C)(C#CC(=O)NC1CCC12CCCC2)CNC(=O)CCn1cncn1 94843,C1(C2CC2)(CNC(CCCCCC)=O)CCN(C(=O)C(C)(C)C(O)CC)C1 94844,c1(CCC(=O)NC(C)C(CO)NC(C2(C)CCCCC2)=O)c[nH]c2ccccc12 94845,Cc1cccc(C(N2CCC(NC(C3CCC(C)(C)CO3)=O)C2)=O)c1C(F)(F)F 94846,CC1(NC(=O)C(O)CC(F)F)CCN(C(=O)Cn2ccc(C3CC3)n2)CC1 94847,O=C(CCc1ccccc1)C(=O)NCC1CCCN1C(=O)Cc1nccs1 94848,c1(OC(C)C)nc(NC(c2ccccc2CN(CCC(F)(F)F)C)=O)ncc1Br 94849,CCCC(C)(C)C(=O)NC(Cc1ccccc1)CCNC(c1ccc(Cl)nc1O)=O 94850,C(=O)(CCCCC1CC1)NC1(C(N2CC(CC)(CO)C2)=O)CSC1 94851,C1(CCC(=O)NCC(=O)NC(C)(C)C)C2CN(C(C3(C#N)CC3)=O)CC12 94852,CC(C)(C)C(C)(C)C(=O)NC1CCN(C(c2cnc[nH]2)=O)C(C2CC2)C1 94853,N1(Cc2c(S(=O)(=O)NC)ccs2)CCCC(C2CCC2)C1 94854,c1(OC(C(N2CC(C)(NC(c3c(NC)cncc3)=O)C2)=O)C)ccc(C#N)cc1 94855,C1(C(F)(F)F)(C(=O)NC)CCN(Cc2ccn(C)n2)C1 94856,C#Cc1nccnc1NC(C1CC12CCN(Cc1ccc(OC)c(I)c1)C2)=O 94857,c1(C(N(C2CN(C(C(CCC)N(C)C)=O)CC23CC3)C)=O)nnn2c1CCCC2 94858,C1(CNC(C(N2CCS(=O)CC2)(C)C)=O)CN(C(=O)C2=COCC2)C2(CCC2)C1 94859,N1(C(C2C(C(C)(F)F)C2)=O)CC2CC(C1)N(C(c1nn(CO)c(C3CC3)c1)=O)C2 94860,C1(CCC)CN(C(=O)Cc2c(C)noc2C)CC1C(=O)NCC1CCC=CCC1 94861,N1(C(c2c(OC)nn(C)c2)=O)CCc2onc(C(=O)N=c3cc[nH]cc3I)c2C1 94862,N1(C(c2c(C)nncc2)=O)CCC(C(=O)NCC2CCN(C(N)=O)C2)C12CC2 94863,N1(C(C2C(OCC)C2)=O)CCCCC(CNC(=O)C(c2cc(Cl)cc(Cl)c2)O)C1 94864,C(=O)(C1CSc2ccccc21)NC1CCN(C(c2c(N)cc(F)c(Cl)c2)=O)C1 94865,C(=O)(C1CC(=O)Nc2ncccc21)N(CC(C)CNC(=O)C(O)C1CCCC1)C 94866,N(C(=NCC(C)(C)C1(O)CCC1)N1CCC(NC(=O)CC(F)(F)F)C1)C(CC)C 94867,O=C(C1=CC2CCCCCCC12)NC1(CNC(c2cc[nH]n2)=O)CCCC1 94868,c1(C(N2C(C(=O)NCC(CC)C)CC3CC32)=O)cc(C)cc(O)n1 94869,N1(C(CC2CC(C)N(C(=O)CCCC(C)(C)C)C2)=O)CCOCC(C)(C)C1 94870,c1(CCC(=O)NC2(CC=C)CN(C(=O)C(C)(O)C3CC3)C2)cc(Br)ccc1F 94871,C(=O)(C(CC(C)C)ONC(c1ccnc(C)n1)=O)NCc1ccc(C)cc1 94872,N1(C(CCCCC=C)=O)CC2CCN(C(c3ccc(=O)n(C)n3)=O)C(C2)C1 94873,CCC(CN=c1ccc(Br)c(S(=O)(=O)N(C)CCN(C)C)[nH]1)OC 94874,C1(C(=O)NC(COCC)C(=O)N2CC(N3CCCOCC3)C2)CCC(F)(F)C1 94875,c1(C(N(c2ccc(OC)cc2)C)=O)cc(N2CCOCC2)cc(F)c1 94876,C1(C(C)C)C(C(=O)NCC(C)(C)C)CCN1C(=O)CCC1CCC(=O)C1 94877,N1(C(C(C(=C)Cl)(C)C)=O)C2CCCC1CC(NC(c1cscc1C(F)(F)F)=O)C2 94878,c1(C(=O)NC(C)(C)CNC(=O)COCCCF)cc2c(s1)COCC2 94879,C1(N=[N+]=[N-])(C(N(C)CC2(C#N)CCC2)=O)CCN(C(=O)CC(F)(F)C(F)F)C1 94880,C1(NC(=O)CCCn2cncn2)CC2CC1N(C(=O)CCCc1ncco1)C2 94881,c1(C(N(CCNC(Cc2cn(C)nn2)=O)C2CC2)=O)noc2c1COCC2 94882,c1(C(N(C2CCN(C(C3CCC4(CC4)C3)=O)C2)CCO)=O)ccc(F)cc1O 94883,c1(C(=O)NCC2CC3CC3N2C(c2cccc(C(F)F)c2)=O)occ2c1CCC2 94884,C(=O)(N1Cc2ccccc2CO1)c1nn(C)c(C(=O)O)c1Br 94885,N1(C(CCN(C)CC)=O)CCC2(CC1)CC(NC(c1csc(Cl)c1OC)=O)C2 94886,N(C(=NCC1CCSCC1)NCC1CCOC1)Cc1c(COC)noc1 94887,N1(CCOC(C)C)CCCC(N(CCCNc2csc(CCN)n2)C)C1 94888,N1(C(c2cnc(OC)nc2)=O)CCN(C(=O)CC(C)C)CC1C(C)C 94889,c1(CC)cccc(F)c1C(=O)NC1CN(C(=O)CNC(=O)CCC(C)C)CC1C 94890,c1(C(=O)NC2CCN(C(C=Cc3ccc(OC)cn3)=O)C2)cc(C#N)c(C)cn1 94891,N1(C(c2cc(CC)[nH]n2)=O)CCN(C(=O)Cc2nc(=N)[nH][nH]2)C(C2CCC2)C1 94892,CN1CC=C(c2ccc(NC(c3cc4ccccc4[nH]3)=O)nc2)CC1 94893,C(=O)(CCCCC(=O)NC(c1cccnc1)C(=O)NC1CC(C(F)(F)F)C1)OC 94894,CC1CCN(C(c2ccc(CNCc3cccc(C(F)F)c3)cc2)=O)CC1(C)O 94895,Cc1c(Br)cnn1CC(=O)NC(CNC(c1cc(Cl)ns1)=O)C1CC1 94896,C1(C(=O)NCC2(CO)C(C=C)C2)N(C(=O)C2=C(Cl)CCOC2)CC12CCCC2 94897,C12(NC(=O)NC3C(OC(C)(C)C)CC(F)(F)C3)CCC(O)(CC1)CC2 94898,C12(C(=O)NC3CN(C(CS(=O)(=O)NC)=O)CC3C)CC(C)(C1)OC2C 94899,C1(C)(CNC(CNC(CC)=O)=O)CN(C(=O)CC(C)NC(N)=O)C(C)(C)C1 94900,N1(C(COCCOC)=O)CCCC1(C)CNC(=O)CCc1n[nH]c(=N)s1 94901,CCCC(C)(O)CC(=O)NC1C2CC(NC(c3cc(OC)nn3C)=O)CC12 94902,c1(C(=O)NCC(F)CNC(=O)C(F)F)ncnc2c1CCC2 94903,C1(C(=O)NC2C(CC)N(C(c3cc[nH]n3)=O)CC2)CCCC2(CCOCC2)O1 94904,c1(OC)ccc2nc(C)c(C(=O)NC(C)CN(C)C(c3c(C)ccn3C)=O)n2n1 94905,CC1CN(N2Cc3ccc([N+](=O)[O-])cc3C2)CC(C)N1C1CC1 94906,N1(C(c2cnc(CC)o2)=O)CCN(C(C2CCCN2C(C)C)=O)CC(C)C1 94907,C1(NC(=O)CC2CCCCO2)CCCC(C(N2C3COCC2C3)=O)C1 94908,C(=O)(C(C)(C)CS(N)(=O)=O)NCC(C)NC(c1c(Cl)ccc(Cl)c1F)=O 94909,CC1(C(=O)OCC2CCS(=O)(=O)C2)CC2(C1)CC(F)(F)C2 94910,N1(C(C=CCN(C)C)=O)CCC(C2CCCN(C(c3ccn(O)c(=O)c3)=O)C2)C1 94911,c1(C(C(CC)NC(=O)C(F)CC2CN(C(=O)OC(C)(C)C)C2)=O)ccc(F)cc1F 94912,c1(C(N(CCNC(COC(CC)C)=O)CC)=O)oc(-c2cnn(C)c2)nc1C 94913,c1(C(=O)NCC(CN(C(C2C(=C)CC2)=O)CC)(C)C)c(C)nc(C)nc1C 94914,C1(O)(CC(=O)NC(CC)CNC(=O)CC23CCC(CC2)C3)CCCN(C)C1 94915,CCC(CNC(=O)CC1CCN(C(=O)COC2CC=CC2)CC1)C(C)C 94916,N1(C(C(=O)Nc2c(C(C)C)n(C)nc2)=O)c2ccc(Cl)cc2OCC1C 94917,CC(C(=O)N(C1CCN(C(=O)COC2CCCOC2)CC1)C)S(C)(=O)=O 94918,c1(C(C)=O)ccc(NC(C2C=CCN2Cc2ccc(F)nc2)=O)c(Cl)c1 94919,CC1CCc2c(sc3ncnc(N4CCCCC(NC(=O)CC=C(Cl)Cl)C4)c23)C1 94920,N1(C(C(C)NC(C2CCC2)=O)=O)CCCCC(NC(C2CCC3CC3CC2)=O)C1 94921,C1(OC)CC(CNC(C2CC(F)C2)=O)(NC(=O)C=C2CCCCC2)C1 94922,n1(CC)ccnc1C=CC(=O)NCCCCCCNC(C1(F)CCC1)=O 94923,c1(OC)nc(C)ccc1C(=O)NC(CNC(=O)CC1C(=O)NN=C1C)CO 94924,N1(C(C2C(CNC(C(SC)SC)=O)C2(C)C)=O)CCC(C)C(O)C1 94925,N(C1c2ccc(Br)cc2CC1(F)F)CCc1ccc(OC)cc1Cl 94926,c1(C(=O)NCC(CNC(C(C=C)(C)O)=O)CO)cc(OC)cnc1F 94927,N1(C(C2(C(C)C)C(C(=O)OCC)C2)=O)CCN(c2ccc(OC(F)F)cc2)CC1 94928,CCC(C)(CO)C(=O)NC(c1ccc(N(C)C)cc1)CNC(=O)COCCOC 94929,CC1CCN(C(C2CCCO2)=O)CC1CNC(c1ocnc1C1CC1)=O 94930,c1(C(=O)NC2CC(NC(C(CC)Sc3ccccc3)=O)C2)oc(COC)cc1C 94931,C1(NC(C=CC(CC)=CC)=O)CC2CC1N(C(=O)C(CC)Oc1ccccc1)C2 94932,C(=O)(C(CC(=C)C)NC(=O)C(F)F)NC(CC#C)(C)C 94933,O=C(O)CC(CC1CCCCC1)NC(C1CC(F)C(=O)N1)=O 94934,C1(c2cn(C3COC(=O)O3)nn2)(C(N2CC(c3ccc(F)nc3)C2)=O)CCOCC1 94935,C1(O)(CC(=O)NCCN(CCC)C(C2(c3ccn(C)n3)CC2)=O)CCCCC1 94936,C12(C(=O)NCC3CCCN(CC)C3)CCCC1CCN2C(=O)C(O)CCC(C)C 94937,C(=O)(C1=NOC2(CCC2)C1)NC1CCCC(C(N(C)CC2CN(C)C2)=O)CC1 94938,c1(OC)cccc(OCC(=O)N(CCCCCNC(C2(C)COC(=O)C2)=O)C)c1 94939,C1(NC(CCn2ccc(C)n2)=O)CC2CC(NC(C3CCCC34CCC4)=O)C2C1 94940,N1(C(=O)Nc2ccc(C(F)(F)F)cc2Cl)CC(C2CCOCC2)C1 94941,C#Cc1cc(C(=O)N(CCC(N2CC(C)(C)CCC2CO)=O)CC)ccc1C 94942,C1(NC(COC(C)C)=O)CCCC(NC(C2CN(C(=O)N(C)C)C2)=O)C1 94943,CCC(CC(=O)NCCOCCNC(c1cc(Br)n(C)n1)=O)C(C)(C)C 94944,CCC(COC)(CC)C(=O)N1CC(C(=O)N(C(C)CO)C)CCC1(C)C 94945,C(=O)(CCC1=CCCCC1)NCC1CN(C(CC(CC)(C)C)=O)C2(C1)CCC2 94946,C1(C2(O)CCN(C(c3ccc4c(n3)OCC(=O)N4)=O)CC2)(OC)CC1 94947,CC1CC(C(=O)NCc2nocc2C(N2CC(C)(CCO)C2)=O)CC(=O)N1 94948,N1(C(c2c(C#N)ccnc2)=O)CCC2(CC1)OCCC2NC(=O)Cn1nccn1 94949,CN1N=C(CC(=O)N2CCCC(n3cc(-c4cnn(CCF)c4)nn3)CC2)CC1=O 94950,C(=O)(C1CCc2ccc(Cl)nc21)NC12C(NC(c3ccc[nH]3)=O)CC(CC1)C2 94951,N1(C(CNC(C)=O)=O)CC(NC(=O)C2=NOC(C)(C)C2)C2(CCCC2)C1 94952,C1(CNC(CCC(C)OC)=O)(NC(C2CC(N(C)C)C2)=O)CCC(F)(F)CC1 94953,C1(C(N(CC)Cc2ccoc2)=O)(CC)CN(C(C2CCCC2F)=O)C1 94954,c1(COC)ncc(C(=O)NCCC2CCN(C(=O)CC3CCCCC3)C2)s1 94955,Cc1cc(=NCC=C(Cl)Cl)[nH]c(NC(CCO)C(F)F)n1 94956,C12(C(=O)NCCC(C)N(C)C(c3ncoc3C3CC3)=O)CCC(C)(CO1)C2 94957,N1(C(C(COC)(C)O)=O)CCC(NC(c2cccc(COC(F)F)c2)=O)C(C)C1 94958,c1(CNC2CCCC(C(=O)OCC)C2)c[nH]c2ccncc12 94959,C1(C(=O)Nc2ccc(Br)nc2Br)CCC2(CN(Cc3csc(Br)n3)C2)O1 94960,C(CC(C(=O)NCCN1CCC(O)CC1)NC(=O)CCC(=O)C1CC1)SC 94961,C1(C(N2CC(C(C)NC(=O)C(C)n3cncn3)C2)=O)(COC)CCCO1 94962,C1(CNC(c2cc(C(C)C)[nH]n2)=O)CN(C(c2cc(Cl)c[nH]2)=O)CC1C 94963,N1(C(C(COC(C)C)NC(C2CN(C)CCN2C)=O)=O)CCCC(C)(C#N)C1 94964,C1(NC(c2cc[nH]n2)=O)(CO)CCN(Cc2cccc(Br)c2F)CC1 94965,C(=O)(C1=CC2(CCOC2)C1)NCCC1CCCN(C(C(n2ncc(C)c2)C)=O)C1 94966,N1(C(C2(C(N)=O)CC2)=O)CCC(CNC(C2C3CC4C(C3)C24)=O)CC1 94967,N1(CCOC)CC(C(=O)NC(C)(CNC(c2cc[nH]c2)=O)C(C)C)CC1=O 94968,Cc1cc([N+](=O)[O-])c2nonc2c1NC(C)CCN1CCCC1 94969,CC1CN(CS(=O)(=O)CCc2ccccc2)CCN1C(=O)Cc1ccccn1 94970,C1(CNC(Cc2cncc(C)c2)=O)CCC(C)(C)CN1C(=O)C(C)NS(C)(=O)=O 94971,CN1CCC(O)C(NC(c2occc2CNC(C2(C)CCCC2O)=O)=O)C1 94972,C1(C(N2CC(N(C)C(c3cnc(S)[nH]3)=O)C3(C2)CC3)=O)Cc2n[nH]cc2C(=O)N1 94973,N1(C(=O)C(O)c2cnc[nH]2)CC2CCCC(C1)N2C(=O)C(O)c1ccsc1 94974,C1(C)(C(=O)NCc2onc(N(C)C)n2)C=CCN1C(C1CC(O)C(F)C1)=O 94975,CC1CCN(C(=O)Cn2cc(C(F)(F)F)nn2)CCN1C(C1OCCC1C)=O 94976,N1(CCN(C(C(=O)NCc2ccccc2)=O)CC2CC2)CCCOC1=O 94977,C1(F)(CNC(CCCC)=O)CCC(NC(c2ccc(N(CC(C)C)C)nc2)=O)C1 94978,c1(CCC)ccc(CN(C2COCCC2CO)CC)cc1C 94979,C(c1ccc(O)cc1)=CC(N1CCCC(C(C)NC(c2cc(Br)cs2)=O)C1)=O 94980,C1(NC(c2c(CNC(C(C)CC3CC3)=O)n[nH]c2)=O)CC(=O)N(C)C1 94981,C1(C(N(CC(COCC)O)C)=O)CC2(CC2)CN1C(=O)CSC 94982,C12(C(N(CC)CC3CCN(C(C4CCCN4C=O)=O)CC3)=O)CC1COC2(C)C 94983,c1(OC)c(Cl)cc(C(=O)NCC(C)(C2CC2)NC(=O)C=CC(C)(C)C)nc1Cl 94984,N1(C(C(C)NS(C)(=O)=O)=O)CCN(C(c2cccc(F)c2)=O)CC12CCC2 94985,c1(C(C)C)cccc(C(=O)NC(C)(C)CCCNC(C2CNC(=O)C2)=O)c1N 94986,C(C(C)(C)C(=O)N1CCCC(C(N)=O)C1)NC(CC(OCC)OCC)=O 94987,C1(CCN(C)C(c2ncccc2F)=O)CCN(C(c2ccn(CC#N)n2)=O)CC1 94988,c1(OC)ccc2c(c1)OCC(N=c1[nH]c(=NCC=CCl)[nH]c3c1CSC3)C2 94989,N1(C(c2cc(C)[nH]c2)=O)CCCC1(C)C(N1CCC1CF)=O 94990,C1(n2cc(C3(C)COC3)nn2)CC2CC1N(C(=O)COc1cccc(I)n1)C2 94991,C1(CN(C2(C)CNC2)C)CN(C(=O)OC(C)(C)C)CC1CN(C)C 94992,c1(C(N2CC(F)(CNC(C3C(C=C)C3)=O)C2)=O)oc(C2CCC2)nc1C 94993,c1(OC)ncc(C(N2CCCCC2CCNC(=O)C(O)C2CC2)=O)cc1F 94994,c1(C(N(CC(C)NC(=O)CCSCC(N)=O)CC)=O)cc(C(F)(F)F)ncc1F 94995,c1(CC(=O)NC2CCN(C(=O)CCCc3cccs3)C2)ccc(O)nc1 94996,c1(CC(C)Nc2nccc(N3CCN(C(C)=O)CC3)n2)sc2ccccc2c1C 94997,c1(C(N(C2CC(NC(C3C(C)CCC3)=O)C2)C)=O)ccnc2c1ccn2C 94998,c1(OC)ccc(C(=O)NCC2CN(C(=O)C(C)OC3COC3)CC2C)cc1O 94999,N1(C(C(C)OCC)=O)CCN(C(=O)CCc2nc3ncccn3n2)CCC1C 95000,c1(COCC)nc(C(=O)NC(C)CC(C)NC(c2cc(CSC)on2)=O)cs1 95001,Cn1cc(C(O)C(=O)NCC2CCC2C(=O)NCCCc2ccncc2)cn1 95002,C(=O)(C(O)C(F)(F)F)N(C)CCOCCN(C)C(C1CCC1C(C)(C)C)=O 95003,N1(C(C)C)CCN(C(=O)CCn2cc(CCN3CCOCC3C)nn2)CC1C 95004,c1(C(=O)NCCCOCCNC(C(C)(C)C2CC2)=O)ccc(Br)nc1N 95005,C1(CC=C)(NC(C2(OC)CCC2)=O)CCN(C(=O)CC(C)F)CC1 95006,N1(Cc2ccc(OC)cc2)C2CCC(C2)C1C(N1CCOC(CN(C)C)C1)=O 95007,CCCC(O)CC(=O)NC1(COC)CCN(C(=O)CC(F)(F)Br)C1 95008,c1(CC(C)NC(=O)CCn2cc(Cl)cn2)ccc(F)cc1 95009,C1(CC(=O)N(CCCNC(=O)CC(C)c2ccncc2)CC)CCC(=O)N1C 95010,c1(C(=O)NC2CC(NC(=O)CCC34CCC(CC3)C4)C2)nccc2nn[nH]c12 95011,C(=O)(CS(C)(=O)=O)NC1CCN(CCCNC(C(C)NC(=O)NC)=O)C1 95012,N1(C(C(F)=CCC)=O)CCC(C2CC2)C1C(N1CC(C)C(C)C1C)=O 95013,N(C1CCCn2ccnc21)C(N1CCC(Cc2ccc(C)nc2)C1)=O 95014,c1(OC)c(Cl)ccc(C(=O)NCC2(O)CN(Cc3cc(C#N)ccn3)C2)c1F 95015,N1(C(C=C(CC)C)=O)CC2(CCCC2NC(c2cc(F)c(C(F)F)c(F)c2)=O)C1 95016,CC1CC2(CCN(C(C3(CF)CC3)=O)CC2)CN1C(C1CC12CCCC2)=O 95017,c1(-n2c(-c3sccc3Br)nc(CC(C)OC)n2)cccc2c1CCCC2 95018,C1(CNC(C2CC(=O)NC(=O)C2)=O)CN(C(c2csnn2)=O)C2(CCOCC2)C1 95019,Cc1ncc(CCC(N2CCCC2C(C)NC(C2CCC3CC23)=O)=O)o1 95020,N1(C(C2C(C)(C)C2)C(=O)Nc2ccccc2)CCOC2(CC2)C1 95021,CC(C(=O)NCC1(N2CCOCC2)CCCC1)S(C)(=O)=O.C123CC(CN1C2=O)C3 95022,N1(C(C(CCCC=C)NC(C2C=CC2C(=O)OC)=O)=O)CCC(C2=NOCC2)C1 95023,N1(C(c2cc(Cl)c[nH]2)=O)CC2CC(NC(c3ccc(C4CC4)o3)=O)C2C1 95024,C(=O)(CS(=O)(=O)CCC(F)(F)F)N1C(C)CN(C(=O)CN2CSCC2=O)CCC1 95025,c1(C(N(CCCCCNC(c2c(SC)cnn2C)=O)C)=O)c(Cl)ccnc1C 95026,C1(NC(C2CCCC(c3ccccc3)O2)=O)CCCN(C(C2(C3CC3)CC2)=O)C1 95027,C12(CCN(CC(C)(C)CC3CC3)C(c3cc(C(C)C)[nH]n3)=O)CC1COC2(C)C 95028,c1(C(=O)NCCC(C)NC(C2OCC2(C)C)=O)cnncc1O 95029,CC1(C)OC(=O)NC1C(N1CCN(C(=O)C(O)CC2CCCCC2)CC1)=O 95030,C1(C#N)(C(=O)NCC(CC)NC(=O)C(C)OCCN(C)C)CCC1 95031,Cc1ccc(C(N2CCC(C(C)NC(C3CC(=O)N(C4CC4)C3)=O)C2)=O)cn1 95032,CCCCC(CNC(C1OCCO1)=O)NC(=O)Cc1cc(=O)n(CC(C)C)[nH]1 95033,N1(C(c2c(CC)c[nH]c2)=O)CC(C)(C)CC1CC(=O)N(C)Cc1n[nH]c(C)n1 95034,c1(C(N2CCCC(NC(=O)C3CC3)CC2)=O)cc2sccc2n1CC(F)(F)F 95035,c12cncc(c1)C(=O)NCCCC(C)NC2=O.C1CCN(S(C)(=O)=O)C1.CCN 95036,c1(C(=O)NC(CNC(CNC(C(CC)C)=O)=O)(C)C2CC2)cc(S(N)(=O)=O)co1 95037,c1(SC)c(C(=O)NC(C)CNC(=O)COCc2nc(C)no2)cccc1F 95038,N1(C(C(CC)n2cccn2)=O)CC(NC(C2(C(C)C)CC2)=O)C(CC2CC2)C1 95039,c1(CNC(C2(NC(=O)Cn3ccnn3)CSC2)=O)ncccn1 95040,c1(CCC(=O)N(CC(C)NC(C(C2CC2)OCC)=O)C)ccncc1 95041,Cc1csc(=O)n1CCC(=O)NCC1COC(CNC(C2(CO)CCCO2)=O)C1 95042,Cc1cc(C(N2CCCC2CN(C)C(C2CC(F)C2)=O)=O)c2scnc2c1C 95043,c1(CC(=O)N(C)CCOC2CCCCC2)ccc(S(C)(=O)=O)cc1 95044,c1(C(=O)NCCC(=O)NC(c2nccs2)CC)cocc1C 95045,C1(CC(N2CCC(CC(C)NC(C3C(CCC)C3)=O)CC2)=O)CC2(CCC2)CO1 95046,N1(C(C(CC)OCC)=O)CCCN(C(=O)Cc2cccc(OC)c2)C(CO)C1 95047,C(CC(=O)N1CC(NC(N)=O)C1)(C(F)(F)F)NC(c1c(CC)ocn1)=O 95048,C1(NC(C2(CC=C)CCCC2)=O)CCN(C(=O)COCC(=C)C)CC1CO 95049,c1(C(=O)NC2CC(NCc3ncccc3O)C2)cc(O)c(O)c(Cl)c1 95050,C1(CNC(C2C(C)=CCS2)=O)CN(C(C2(C)CCCCCC2)=O)CCCO1 95051,c1(C(=O)NC2C(NC(CNC(=O)OC(C)(C)C)=O)CCC2)c[nH]nc1S(N)(=O)=O 95052,C1(C(=O)NC2C(NC(c3c(CC)scc3)=O)COCC2)CCCCC(=O)N1 95053,CC(C)(CC(F)C(=O)NC1C2CCCC12)NC(=O)Cc1ccsn1 95054,N1(C(CC2CN(C(C)=O)C2)=O)CCC2(C=C(C(=O)NCCN=S(C)(C)=O)C2)C1 95055,Cc1cc(O)c(Cl)cc1C(=O)N(C)CC1CCCN1C(c1cccc(F)c1F)=O 95056,CC1CC2CN(C(=O)CC(C)(C)N(C)C(C3COCC3(C)C)=O)CCN2C1 95057,N1(C(C2N(C(C(N3CCNC3=O)C)=O)C(C)CC2)=O)CCc2c[nH]nc2C1 95058,N1(C(C(=Cc2cnc[nH]2)C)=O)CCCC(NC(=O)Cn2cc(Br)c(C)n2)C1 95059,C1(N(C(C(F)=CCC)=O)CCNC(=O)C(c2ccccn2)C)CCCCCC1 95060,O=C(CCCn1cccc1)N1CCC(N(C(C2CC3(CC3)C2)=O)CC2CC2)C1 95061,N1(C(C(F)OC)=O)CCC2(CC1)COCC(CNC(c1ncc[nH]c1=O)=O)O2 95062,N1(C(c2cc(-c3cccc(F)c3)on2)=O)CC2CC2(CNCc2ccsc2)C1 95063,C1(NC(C(=O)NC(C)C)=O)COCCN(C(=O)CC=C(Cl)Cl)C1 95064,C1(C(=O)NC2CC(c3c(F)cccc3F)C2)CN(C(=O)C(=O)C2CC2)CCC1O 95065,Cc1ccc(N2CCC2CN(C)CC2CCC(NC(=O)CN3CC(C)C3)O2)cc1 95066,N1(C(C2OCCC(C)(C)C2)=O)CC(NC(c2cn[nH]c2)=O)C2(CCC2)C1 95067,C1(OC)COc2c(C(N3CCCC3CNC(c3nnsc3C)=O)=O)cnn2C1 95068,CC1CN(C(=O)NCCc2c(F)cccc2Cl)CC1(F)F 95069,n1(CC)ncc(NC(C2CC(NC(c3cccnc3O)=O)C2(C)C)=O)c1C 95070,C1(CN(C(=O)Cc2csc(-c3ccccn3)n2)C)CCCN(C(=O)CCF)C1 95071,C(C(=O)NCC1(C(=O)NC2CC(N(C)C)C2)CCC1)(C(C)C)OCC(C)C 95072,CN1CCCC(F)(C(=O)NC(C2CCCC2)CNC(c2cscc2Cl)=O)C1 95073,C(CCCCC(=O)NCCc1cnc(C)[nH]1)N(C(CNC(=O)OCC=C)=O)C 95074,C1(C(=O)NCC2(C(=O)N(C(C)C(=O)OC)CC)CC(=C)C2)CCS(=O)CC1 95075,C1(C(=O)NCC2(NC(C(c3c(C)cccc3)C)=O)CCC2)CC12CCOCC2 95076,N1(C(=O)Nc2ccc(NC3(OC)CCCCC3)cc2)CCC2(CCOC2)CC1 95077,S(=O)(=O)(c1ccc(NCC(C)O)c(F)c1)N(CC(C)N(C)C)C 95078,c1(C(=O)NC2CCC(NC(c3n(C)cc(Cl)c3)=O)CC2)cc(F)ccc1F 95079,N1(C(C(C)(C)OC)=O)CC2OCC(C(=O)Nc3cnccn3)C2C1 95080,c1(C(N2CC(C(C(=O)NC(C)CC3(O)CCC3)O)C2)=O)cnnn1C1CC1 95081,C(=O)(C(O)CC(C)(C)C)N1CCN(CCN(C(CC(C(=C)C)O)=O)C)CC1 95082,N1(C(=O)OC(C)(C)C)CC(O)CC1CNC(=O)NCc1conc1C(C)(C)C 95083,N1(C(CC(C)O)=O)CC(C(=O)NCCCCC(C)(C)C)CC1(C)C 95084,c1(C(=O)NC2CCN(C(c3n(CC)c(O)nc3)=O)CC2)cccc(C(F)F)c1F 95085,C1(C2CCN(C(c3cc(C)n(C)n3)=O)CC2)(NC(C(CC)CN(C)C)=O)CC1 95086,Cc1nc(O)ccc1C(=O)NCC1CN(C(=O)CC2CCC(=O)N2C)CC1(F)F 95087,c1(C(=O)NCc2c(C(=O)NC(C(=O)OC)C)nco2)ccncc1O 95088,c1(OC)cc2cc(c1)-c1csc(c1)C(=O)N2.C(C(C)OC(C)C)NC(C)=O 95089,C1(CNC(C2(C(F)F)CCCO2)=O)CCCCC1C(=O)NCc1cc(Cl)ccn1 95090,c1(C(N2CCC(C(=O)NCCC3(OCC)CC3)C2)=O)cnc2ccccn2c1=O 95091,CC1CN(C(=O)CC2CC=CC2)C1C(=O)NC1(CCCCO)CC1 95092,C1(CC(=O)OC)CCN(C(=O)N(CC(c2ncccn2)(C)C)CC2CC2)CC1 95093,N1(C(c2c(CC)ocn2)=O)CCCC1C=CC(=O)NCc1cncn1C1CC1 95094,c1(C(C)C)ccc(C(=O)NCC2CCC(C)N(C(c3ncn(C)n3)=O)C2)c(F)c1 95095,c1(OCCC(=O)NCC(C(C)C)NC(=O)C2=COCC2)cccc(Br)c1 95096,C1(CC)C(NC(=O)CN2CCCNC2=O)CCCN1C(C1CCC(=O)NC1)=O 95097,C1(CCC)CCCN(C(=O)CCN(C(c2cc(CO)oc2C)=O)CC2CC2)CC1 95098,C(C(C)C)(C(O)C(=O)NCCN(C(=O)COc1ccc(C(C)C)nc1)CC)OC 95099,n1(CCC(=O)NC2CN(C(C(C)O)=O)C3(C2)CCC3)c(=O)n(C)c2ccccc12 95100,C1(C(N(CCNC(C(CC)F)=O)C)=O)(NC(C)=O)COc2ccccc2C1 95101,CC1CN(C(C2(Cl)CCC2)=O)CC(C(=O)NCCN=S(C)(C)=O)O1 95102,C=CC1(C(=O)NOCC(=O)NCC(=O)NCC(C)C)CCC1 95103,c1(C(=O)NC(C2CCCN(C(C3CCCCCC3)=O)C2)C)cnn2c1OCCC2 95104,c1(N(CC)CC)ccc(C(=O)NCC(CO)NC(c2nnc(S)n2C)=O)c(O)c1 95105,CS(=O)(=O)CCC(=O)N1CC(CCCCNC(=O)Cc2ccccc2F)C1 95106,C(C(C)(C)CC(=O)NCCCOC1CCN(C(=O)C(O)C(C)C)CC1)OC 95107,c12cccc(c1)CCCO2.C1(CCC(=O)NCCC2CN(CC)C2)CCC(C)O1 95108,c1(C(=O)NC(C)CC(=O)c2ccco2)cc(P(C)(C)=O)cs1 95109,c1(-c2cn(CC(C)NC(=O)CC34CCCC3C4)nn2)ccc2nc[nH]c2c1 95110,Cc1cc(F)c(C(=O)NCC2CCCN2C(c2cc3c(o2)CCCC3)=O)cc1F 95111,N1(C(C2CCN(C(C)=O)C2)=O)C2CCC1C(CO)N(C(c1ccc(C)s1)=O)C2 95112,Cc1[nH]c2ncccc2c1C(=O)NC12CC1CN(C(=O)CNc1ncccn1)C2 95113,C1(NC(C=C(C)Cl)=O)CC2CC(NC(c3nc(-c4cnn(C)c4)oc3C)=O)CC12 95114,CC1CN(C(c2nc(Cl)sc2Cl)C(=O)NC2COC2)CC1O 95115,C1(C)(C(N(CCCN(C(c2cccc(C)c2)=O)C)C)=O)CCCC(F)(F)C1 95116,C1(C)(NC(C2OCCC(NC(Cn3ncn(C)c3=O)=O)C2)=O)CCCCCC1 95117,Cc1ccc(NC(C2(F)CCN(c3cc(C)nc(C)n3)C2)=O)c(C#N)c1 95118,C12(C(=O)NCC(C)C)CC1CN(C(c1ccc(SC(F)(F)F)cc1)=O)C2 95119,c1(OCC)cccc(C(C(=O)NCC2CN(C(c3ccsn3)=O)CCO2)OC)c1 95120,CN1CCC(C)(NN2CC3CC2CS3)C1 95121,c1(C(=O)NC2CC(NC(C3=C(C)CCC3)=O)C2)cccc2c1OCCCO2 95122,N1(C(C(C)n2cccn2)=O)CC2(CCC(CNC(C3(CCF)CC3)=O)O2)C1 95123,C1(NC(C2(CCCC)CC2)=O)CN(C(c2csc(NCC)c2)=O)C2(CCOC2)C1 95124,N1(C(c2cc(C(C)C)no2)=O)CC2(C1)CN(C(C1CC3CCC1O3)=O)C2 95125,C1(CC=C)(NC(=O)CNC=O)CC2CCC(C1)N2C(=O)CCC#N 95126,C1(F)(CNC(=O)CCC2CCCC2)CCN(C(c2cc(Cl)c[nH]2)=O)CC1 95127,c1(COC)nn[nH]c1C(N1CCC(C(N2CCCC2CC2CC2)=O)C1)=O 95128,C1(CNC(CCOCC)=O)(CO)CCN(C(c2ccoc2Cl)=O)C1 95129,c1(C(=O)NCc2c(C(N(C(C)COC)CC)=O)[nH]cc2)cc2ccccn2c1 95130,Cc1ccc2c(C(=O)N(C3CN(C(c4cc(O)nc(Cl)c4)=O)C3)C)cnn2c1C 95131,C1(NC(=O)C(F)(F)C2CCCC2)CCCN(c2ccc(F)cc2F)C1=O 95132,S(=O)(=O)(c1cncc(Br)c1Cl)NCCCCCCC(=O)O 95133,C1(C(N(CCCNC(C2C(OC(C)=O)C2)=O)C)=O)CCCN1c1ncccn1 95134,C1(CNC(CNC(=O)OC)=O)CC(NC(=O)C(N2CCCCC2=O)C)CCO1 95135,N1(C(C)=O)CC2CC(O)C1C2NC(=O)CCCc1ccc(C)cc1 95136,c1(C(N(CCCNC(c2cc(C3CC3)ns2)=O)CC)=O)cccc(N(C)C)c1 95137,C1(C2CCC2)(C(=O)NC(C)CCCNC(=O)CNC(c2cccnc2)=O)CC1 95138,N1(C(CCC#N)=O)CC2(CCOCC2)CC1CNC(C1(C(N)=O)CCC1)=O 95139,N1(C(c2c(C)ncn2O)=O)CCC(N(C(=O)C=CC=C(Cl)Cl)C)C(C)C1 95140,CC(O)CC(C)(C)CNC(c1cnn(CCNC(=O)CC2C=NN(C)C2=O)c1)=O 95141,Cn1cnc2c(C(=O)Nc3cccc(NC(C4CC(C(N)=O)C4)=O)c3)ccnc12 95142,Cc1ccc(C(C)C(=O)N(C2CCCN(C(c3nc(O)c(C)s3)=O)C2)CCO)cc1 95143,C1(NC(c2c(OC)nsc2)=O)CC2CC1CC2C(=O)NCCC1CC1C 95144,N1(C(C(CC)(F)F)=O)CCC(NC(=O)Cc2ccc3n[nH]cc3c2)CC(C)(C)C1 95145,C(C(C)C(=O)N1C(C(=O)NCCOCCN(C)C)CC1C)SC 95146,C12(NC(CN(C)CCc3ccccc3)=O)CCCC1CN(C(=O)Cn1cnnn1)C2 95147,Cc1cc(C(N2CCC(C(N3CCC(N(C)C)CC3)=O)C2)=O)cc(C)c1C#N 95148,c1(C(CNC(=O)NC(C#C)CCC)N(C)C)ccc(CC)c(F)c1 95149,C12(NC(C=CC(C)C)=O)CCC(NC(c3cccc(C(N)=O)c3)=O)(CC1)C2 95150,N1(C(Cc2ccc(C)o2)=O)CCC2CCC(NC(=O)Cc3ccc(Cl)s3)C1C2 95151,C#CC1(O)CCCCC1.C(=O)(CC(C)C(=O)OCC)N1C(CNC=O)(COC)C1 95152,C1(C)(NC(c2ccc(Cn3cc(C(C)NC)nn3)cc2)=O)CCCC1(F)F 95153,C=CCCCC(=O)N1CCCC1C=CC(=O)NCCN(C)C1CC1 95154,N1(C(CNC(CC)=O)=O)CCC2(CCOCC2)C1.C1C(=O)N1C(C)C 95155,C1(NC(Cn2ccc(C)c2)=O)CCC(CC(=O)NC2CC2c2ccn(C)n2)CC1 95156,n1(CC)cnc(C(=O)NCCN(CCOCCO)C(c2cc[nH]c2C)=O)c1 95157,N1(C(c2c(CC)con2)=O)CC2CCN(C(c3coc(Br)n3)=O)CCC2C1 95158,c1(CC)c(C(N2CCC(CNC(c3cccc(CO)c3)=O)CC2)=O)cnn1CC 95159,CN(Cc1ccc(S(=O)(=O)N2CCCCC2)cc1)N1CCC2(CNC(=O)OC2)C1 95160,C1(CC)CN(C(=O)CSc2nnc(S)s2)CCC1NC(C1(O)CC(C)(C)C1)=O 95161,c1(C(N(CC(=O)NCC(C)C)CC(C)C)=O)ccn2ccnc2c1 95162,C1(CNC(C(COC)(C)O)=O)CC(F)(F)CN1c1nccc(C#N)n1 95163,c1(NC(c2c(NC(c3c(C)ccc(O)c3)=O)c[nH]n2)=O)ncnc2sccc12 95164,CCCCCC(O)CC(=O)NC1CN(C(c2ccc(OC(F)F)cc2)=O)CC1F 95165,c1(CSCC(=O)N(CC)CC)ccc2c(c1)OCCO2.C1CC(C)N1 95166,c1(C(C)N(C2CCCC2)C(=O)CC2CCOC2)ccc(NC(c2cccs2)=O)cc1 95167,C1(COC)(NC(c2nnn(C)c2C)=O)CCN(C(c2cnoc2C)=O)C1 95168,c1(C(=O)NCCCNC(CN2CCC(C)C2)=O)cnc([N+](=O)[O-])n1C 95169,C(=O)(CC1=CCOCC1)NCCn1cc(C(N2CCN(CCCC)CC2)=O)nn1 95170,C#CCCCC(C)C(=O)N1CCC(CCC(=O)NCC(C)(C)OC(C)C)C1 95171,N#Cc1cccc(CNc2ncc(C)s2)c1.C1(C=O)C2CN(CC(F)(F)F)CC12 95172,c1(C(N2CCC(N(C(=O)CC3CCCO3)CCO)C2)=O)ncc(Br)cc1O 95173,c1(C(C(=O)N(CCCCCNC(c2c(C)n[nH]c2)=O)C)(F)F)ccc(F)cc1F 95174,c1(C(=O)NCC(CO)NC(C2CCS(=O)(=O)C2)=O)cccc(O)c1F 95175,Cc1sc(O)nc1C(=O)N(C(CNC(C1(O)CCOC1)=O)Cc1ccccc1)C 95176,c1(CC)nn(C)c(C(N2CCOC(C(=O)NCC(C)(C)C)CC2)=O)c1Cl 95177,c1(C(=O)NCCC2CC(NC(C3(CC=C)CCOC3)=O)C2)cc2occc2n1C 95178,c1(OC(C)C(=O)N(C2CCS(=O)(=O)C2)C)cc(Cl)ccn1 95179,C1(n2cc(C(C3CCCC3)C)nn2)CCN(C(=O)CCCC2CCCCC2)CC1O 95180,C1(CNC(c2cncc(C)n2)=O)CC2(CC2)CN1C(=O)C(CO)c1ccccc1 95181,Cc1ccc(NCC2C(C)CCCN2C(C)C)c(C)n1 95182,C1(F)(C(=O)NC(CC2CCN(c3ncnc(C)c3F)CC2)C)CCC(F)(F)CC1 95183,Cc1ccc(CC(N2CC(NC(=O)CCN3CCOC3=O)CC2(C)C)=O)c(F)c1 95184,CC1(C)CN(C(c2cc[nH]c2)=O)C(CNC(=O)CCN2CCCS2(=O)=O)CO1 95185,Cn1ncc(C(F)(F)F)c1C(=O)NCCC1(O)CCN(C(C2CC23CCC3)=O)C1 95186,c1(C(N2CCCC(Cn3cc(CCC#N)nn3)C2)=O)ccc2nc[nH]c2n1 95187,Cc1cc(Br)sc1Cn1cc(COCC2CCOC2)nn1 95188,C1(NC(COCCC)=O)CC2CCC1(CNC(c1ccc(COC)[nH]1)=O)C2 95189,N1(C(c2noc(CC)c2C)=O)CCCCCC1C(=O)NCC1CSC1 95190,c1(C(N2CCC(CCC)C2)C(=O)NCc2ccc(OC)cc2)ccc(C)cc1C 95191,CC(C)C(C(=O)NCC1(O)CN(C(C2CCOC2C)=O)C1)Nc1ccccc1 95192,C1(COC)(NC(c2cc(C)oc2C)=O)CCN(C(=O)Cc2conc2C)CC1 95193,CCC(C)CC(=O)C(=O)N1CCC(C(C)C(=O)N(C2CC3CC3C2)C)CC1 95194,C1(NC(N(CCC(C)C)CC)=O)CC(CF)C1 95195,C(=O)(C(CO)OC)N(CCOCCCNC(C1C(=C)C1)=O)C 95196,c1(C2C(F)(C(=O)NC(c3nnc(O)o3)C)C2)ccccc1 95197,c1(C(N2CCC(N(CC)CC)C2)C(=O)NCC=C)ccnc(Br)c1 95198,c1(C(=O)NCC=CCNC(=O)CCN2CCC2)cccc2c3c([nH]c12)CCC3 95199,N1(C(c2c(Br)cnn2C)C(=O)NC(c2ccccc2)C)C2CCCC1COC2 95200,n1(CC(N2C(C)C(NC(=O)CC(C)C(F)F)CC2)=O)sc(=O)c2ccccc12 95201,Cc1cccc(CN2CCCC(C(=O)N(C3CCCC3)CCO)CC2)c1C 95202,C1(C(=O)NCC(CO)NC(CC2(CSC)CC2)=O)Cc2cccc(C)c2O1 95203,S(=O)(=O)(c1cccnc1N1CC=CCC1)NCCNC(=O)C1CC1 95204,c1(C(=O)NC2(CCCNC(CS(=O)(=O)NC)=O)CC2)ccc2n[nH]cc2c1 95205,N1(C(C2CCCOC2)=O)CCOC(CNC(C23CC(CC(F)F)(C2)C3)=O)C1 95206,CCCC(C(=O)OC)C(=O)NCCCOCCC(=O)Nc1csc(C)c1 95207,c1(C(c2nnnn2C2CCOC2)NCC(=C)Br)cccnc1-c1ccccc1 95208,c1(C(=O)NCC2N(C(C(C)n3cccc3)=O)CCN(C)C2)cc2c(s1)CCCC2 95209,C(=O)(C(CC(C)C)NC(c1cnn(N2CCNCC2)c1)=O)NC 95210,CC(C)(O)C(F)C(=O)N1CC(NC(c2cccc(C(F)(F)F)c2)=O)C(C(F)F)C1 95211,C1(C(N(c2cccc(Br)c2)CC#C)=O)CCNC2C1C2(F)F 95212,c1(CN(C)C)ccc(CN2CCCC2(C)C(N2CC(N3CC(F)C3)C2)=O)cc1 95213,CC(CC(=O)NC1CCN(C(=O)C(N2CCCC(C)C2)=O)CC1F)C(F)(F)F 95214,Cc1ccc(Br)c(C)c1C(=O)NC(C)(C)CNC(C1CCC(C(F)(F)F)C1)=O 95215,c1(OC)cc(OC)c(C(N2CCC3CN(C)CC23)=O)cc1OC 95216,C(=O)(CC1CNc2ccccc21)N1CCC2CCN(C(CC(C)C)=O)CC2C1 95217,c1(CCC)nc(C)c(C(=O)NC2CC(CNC(=O)Cn3nnc(C)n3)CC2O)s1 95218,C1(C)(NC(C=CC(C)NC(C2C(C#N)C2(C)C)=O)=O)CN2CCC1CC2 95219,N1(Cc2nnc(CC)s2)CCC2(CN(C(c3cc(C)[nH]n3)=O)CC(C)O2)C1 95220,c1(C(=O)NC2CCN(C(c3on(C)c(=O)c3)=O)C2)nccc2nn[nH]c12 95221,N(C1CN(C(=O)C2=CCCOC2)CCc2ccccc21)C(c1cccc(N)n1)=O 95222,N1(C(C(CC)COC)=O)CCC2(CCN(C(c3cc(C(C)(C)C)oc3C)=O)C2)C1 95223,CC1(C)OCCC1NC(c1coc(CNC(C23C=CC(CC2)C3)=O)c1)=O 95224,c1(C(N(CC(C)NC(c2cnc(C(C)C)[nH]2)=O)C)=O)cc(S(C)(=O)=O)ccc1Cl 95225,N#Cc1cc2c([nH]c1=NCCNC(C1CC3C=CC1C3)=O)CCOC2C1CC1 95226,C1(C(=O)NC2CCCC2NC(c2cnc(C)[nH]2)=O)(OC)CCCCC1 95227,c1(CCC(=O)NC2C(NCC3CCN(C)CC3)COC2)n[nH]c2ccccc12 95228,C1(NC(C(=O)Nc2ccc(OC(C)C)cc2)=O)CCC2CCCC2C1 95229,c1(CN(C(=O)Cn2nnc(C(=O)O)c2C)Cc2cc(C)no2)c(F)cccc1Cl 95230,C1(CC(N2CCC(O)(CC)C2)=O)CCN(C(c2ncc(F)cc2F)=O)C1(C)C 95231,c1(C(=O)NC(CC)CNC(C2CC3OC2C2CC32)=O)ccc2nnnn2c1 95232,c1(OC)nc(N2CC(C(C)NC(c3csc(CSC)n3)=O)C2)nc(C)c1F 95233,C1(N(C(C2(C)CCCS2)=O)CC)CCCN(C(c2c[nH]nc2OC(C)C)=O)CC1 95234,c1(C(=O)NC2CN(C(C3(C)CC(=C)C3)=O)CC2F)csc2c1CCCC2 95235,c1(NC)ccc(C(=O)NCC(C)(C(C)C)NC(=O)Cc2ccc(O)nc2)cc1F 95236,C1(C(=O)NCc2cc(CC)[nH]n2)CCCCCN1C(C1C2CCC(C2)C1C)=O 95237,C1(N(C(C(C)OCCOC)=O)C)CCCN(C(c2ccc(C#N)o2)=O)CC1 95238,N1(C(c2c(Cl)cc(C)nc2)=O)CCC2CCN(C(=O)CC3CC3(C)C)C2C1 95239,c1(NC(c2cccc(Cl)c2I)=O)ccc2c(c1)CN(c1nccc(C(F)F)n1)C2 95240,c1(C(N2CCCC2)=O)ccc(C(F)F)cc1F.c12ccc(nc1)Cn1cc-2nn1 95241,c1(C(N2CCC(C)(CNC(C(C)N3CCC3)=O)CC2)=O)c2c(nn1C)CCOC2 95242,CCC(F)(F)C(=O)NC(C1CC(NC(=O)CC2CCC(=O)NC2)C1)C 95243,N1(C(c2cc(OC)ncn2)=O)CCCC(CO)(NC(=O)CN(C)C(=O)C2CC2)C1 95244,c1(C(=O)NCCCCCC(=O)N(C2CCCC2C#N)C)cc2ccccc2[nH]1 95245,c1(C(N2C(C(=O)NC(CC)C(C)O)CC(F)C2)=O)ccc2cc[nH]c2c1Br 95246,n1(CC(=O)NCC(=O)N(C)C2CC2)cc(CNC(=O)Cc2cnsc2)nn1 95247,C1(C(N2CCOCC2)=O)(N(C(C(F)=CCC)=O)C2CC2)CCSC1 95248,Cc1nn(C)c(Cl)c1CN(C1CCCN(CCN(C)C(c2ccccn2)=O)C1)C 95249,N1(C(CC(C(=O)OC)(C)C)=O)CCCC2C1CCCN2C(c1ncn(C)c1C)=O 95250,C12(C(=O)NC3C(OCC)CC3)C(NC(=O)CN3CC(C)(C)C3)C3CC1C2C3 95251,N1(C(C2CCCC(C)C2)=O)CC(CNC(C2OCCCC2(C)C)=O)CC(C)C1 95252,C1(NC(CCC)C(=O)OC(C)(C)C)CCC2(CC2)CN1C(=O)OCC 95253,N1(C(CC2CC(=O)C2)=O)CCCC2(CNC(=O)C=CC3CCCO3)CCCC12 95254,N1(C(C(COC)C)=O)C(C(=O)Nc2c(-c3ccccc3)nnn2C)CCC1C 95255,C1(NC(c2n[nH]c3c2COC3)=O)CN(C(c2cc(O)ncc2F)=O)C2CCCC12 95256,c1(C(C)S(N)(=O)=O)ccc(C(=O)OCCP(C)(C)=O)cc1 95257,N1(C(C2(CN(C)C)CC2)=O)CCN(C(=O)C(C)(O)CC(F)(F)F)CC12CCC2 95258,c1(C(N2CCC(C(C)NC(=O)CC#N)CC2)=O)cc2cc(Cl)sc2[nH]1 95259,c1(CC)ncc(C(=O)NC2CC(C)(NC(=O)Cc3ccc(SCC)cc3)C2)cn1 95260,C1(NC(CCCOC)=O)CCCC(CNC(=O)CSc2cccc[n+]2[O-])C1 95261,c1(CS(CC(=O)N2CCOCC2)(=O)=O)cc2oc(-c3ccccc3)nc2cn1 95262,c1(C(=O)NCC2C(NC(C3C(C)N(C)CC3)=O)C2)cnc(N)c(Cl)c1 95263,C(=O)(C(C)C(C)(C)O)NCC(N(C(c1nn(CC)c(C(C)C)c1)=O)C)C1CC1 95264,N1(C(C(=O)NCC(C)O)=O)CCCC1c1ncc(-c2ccccc2)[nH]1 95265,Cc1cnn(CC(N2CCC3(CC3NC(=O)CC3COCC(C)O3)C2)=O)c(=O)c1 95266,c1(CC(=O)N(C2C(NC(CC=CC)=O)CCCC2)C)ccc(C)c(Cl)c1 95267,C1(C(N(C(C)C(=O)N(C)CC2CC2)C)=O)CCCN(C(n2cncn2)=O)C1 95268,c1(-c2nnc(C)o2)ccc(C(=O)NC2CCC2NC(=O)CCC=CC(C)C)cc1 95269,c1(NC)ccc(Cl)c(CNC(=O)C(=O)NCCN2CCCC2)c1 95270,O=C1NCCOCC1Nc1ccc(Oc2ccncc2)cc1 95271,c1(OC)cccc(Cl)c1CC(=O)N(C(C)CN(C)C(C1COC(C)(C)CO1)=O)C 95272,n1(CCCOC)nnnc1C(c1nncn1C(C)C)NC(COC)C(C)C 95273,C1(CC(=O)NCC(CCNC(C(CC)=CCCC)=O)O)CCCOCC1 95274,C1(NC(=O)C=Cc2cncs2)COC2(CCN(C(=O)Cc3cnns3)C2)C1 95275,Cc1cc(C(=O)NC(CNC(=O)C(C)Cc2ccc(F)cc2)C(C)C)nc(O)c1 95276,c1(NCc2ccc(C)nc2Cl)ccc(S(=O)(=O)NC2COC(C3CC3)C2)cc1Cl 95277,c1(C(=O)NC2C(NC(C(C3CCC3)OC)=O)C2)sccc1Cl 95278,C1(CNC(C(C=CC)O)=O)CCN(C(c2csnc2Cl)=O)CC1O 95279,Cc1coc(C(N2CCC(C3CCCN3C(=O)C(F)OC(F)(F)F)C2)=O)c1C 95280,n1(C(c2cccc(Br)c2)C#C)c(-c2cn(C)nn2)csc1=Nc1ccc(O)cc1 95281,C(c1cncnc1O)=CC(=O)NC1CCCC1CNC(=O)Cc1ccon1 95282,C(CCCCCO)c1cn(CCOCCNC(CC2C(C)C2)=O)nn1 95283,N1(C(c2cc(C)oc2)=O)CCCC(NC(=O)CC(C2CC2)C2CC2)C1C 95284,C1(CC(=O)N(C2CCCCC2)C)C2CN(C(=O)CC(F)F)CC12 95285,O=C(C1CCCn2nccc21)NC1(CO)CN(C(c2cc(F)c(F)cc2Cl)=O)C1 95286,c1(C(=O)NCCC2CCN(C(C=CC(=O)OC)=O)C2)cc(C)ccc1OC(F)F 95287,c1(NC2C(C(N)=O)CCC2)nc2ccccc2nc1NCCCO 95288,c1(C(=O)NCC(C)N(C(C2C(C=C)CC2)=O)C)ccc(Br)c(OC)c1 95289,c1(C(N(CCC(=O)N(CCCO)C)CC=C)=O)nn(C)cc1Cl 95290,C1(CNC(c2c(OC)csc2)=O)CN(C(=O)CCc2c[nH]c(=N)[nH]2)CC1C 95291,C(=O)(C1=C(F)CN(C(c2ccc3occc3c2)=O)CC1)N(C(C)C(C)(C)O)C 95292,N1(C(C(CCSC)NC(N)=O)=O)CCCC(CCNC(=O)C=C(C)C)CC1 95293,Cn1ncc(C(=O)NC(C2CCN(C(C3CCC3(C)C)=O)CC2)(C)C)c1Cl 95294,N1(C(c2c(C)cc(SC)o2)=O)CC(C2CN(C(=O)C(CN(C)C)N(C)C)C2)C1 95295,N1(C(CCc2nc(C)c(C)o2)=O)CC(CO)C2(C1)CN(C(C1CC(F)(F)C1)=O)C2 95296,c1(CC(N2CCCC(N(C(COCC(=O)NC)=O)CC)C2)=O)ccc(C#N)cc1 95297,c1(C(N(CCNC(=O)C(C)(CC)OC)CC)=O)ccc([N+](=O)[O-])cc1Br 95298,Cc1ccc(CC(C)C(=O)NC(C)C(CO)NC(=O)CCC2CCCCC2)cc1 95299,C(=O)(C(=O)N1CCC(C(N2CCCC(C#N)C2)=O)O1)N(C)C 95300,c1(OC)ccc(CN2CC3CC3(C(=O)Nc3c[nH]nc3C)C2)nc1Br 95301,C1(C(=O)NCCCNC(c2[nH]n(C)c(=O)n2)=O)CCCC12NC(=O)NC2=O 95302,N1(C(C2CCC(COC)C2)=O)CC2(CCN(C(c3cc(C)sn3)=O)C2)C1 95303,C1(C(=O)NCCN2CCC(NC(C3C4CCCC34)=O)CC2)CCCCC1(F)F 95304,C1(CNC(C(C(C)C)F)=O)CC(C)CN(C(c2ccnn2C2CCCC2)=O)C1 95305,C1(C(N2CCC(C(C)NC(=O)Cn3cnnc3)CC2)=O)Cc2nccnc2C1 95306,N1(C(=O)Cc2ccn(C(F)F)n2)CCCC(C2CN(S(=O)(=O)C3CC3)C2)C1 95307,C(C)(CCC(=O)NCCN1CCC(NC(C2(C)CC2Br)=O)CC1)SC 95308,N1(C(C(C(C)OC)NC(c2c[nH]c(C#N)c2)=O)=O)CC2(C1)CC2(F)F 95309,C1(NC(CCSC)=O)CN(C(=O)COCC=Cc2ccccc2)CC12CC2 95310,Cc1ccc(F)c(C(N2CCC(O)(C(C)NC(=O)C=C3CCOCC3)C2)=O)c1Cl 95311,c1(CNC(C2(CNC(C3(C)CCCS3)=O)CCCC2)=O)cccc(CO)c1 95312,C(=O)(C1CCc2snnc21)NCCN(C(=O)CC1OCCOC1(C)C)C(C)C 95313,C1(NC(C(C2CCCC2)NC(C(COC)C)=O)=O)CC2CCC1O2 95314,C=CCN=C(NCC=CC1CC1)NCC1C(C)(C)C1(F)F 95315,C1(NC(CN(CCC)C)=O)CCSC12CN(C(=O)C(C(C)C)n1cncn1)C2 95316,C(=O)(CC1=CCCCC1)NC1CN(C(C2CC3(CC(C)C3)C2)=O)CC12CC2 95317,C1(C(=O)NCC2N(C(c3c(SC)ccs3)=O)CCC2C)CC2(CCCO2)C1 95318,c1(C(=O)NCCC2N(C(CSCCC)=O)CCOC2)c(C)nc(O)nc1C 95319,C=CCC(C)C(=O)NC1COCCC1C(=O)NCC(F)C1CCC1 95320,Cc1ccc(C(=O)NC2CC(C)CN(C(=O)CCSc3ccccn3)C2)c(N)c1 95321,C1(C)(CNC(C2(COC)CC2)=O)CC(NC(N)=O)CN1C(c1cncn1C)=O 95322,CC1(C)CCC(NC(=O)CCSC2CC2)C(CNC(=O)C=CC2(C)COC2)C1 95323,N1(C(C2(OC)CC2)=O)CC2(C1)C(NC(=O)C(C)c1ccsc1)CCS2(=O)=O 95324,Nc1ccc(Cl)cc1C(=O)NCC1(F)CC(NC(=O)CC2CCC(O)C2)C1 95325,C1(NC(=O)C(=C2CCCCC2)F)COC2(CCN(C(C3CC4(CC4)C3)=O)C2)C1 95326,CC1(C)CCN(C(C2OCCC2(C)C)=O)CC1C(=O)NC1(CC(N)=O)CC1 95327,CN=C(NCCCn1cccn1)NC1CC(OC(C)(C)C)C1 95328,c1(CC(=O)NCC(C2CC2)NC(c2c(C(N)=O)coc2)=O)cnc2cccnn12 95329,C1(C(N2CC(N(C(=O)C(CO)NC(=O)C(F)(F)F)C)C2)=O)CC2(C1)CC2F 95330,CC1(C)CCN(CCNC(C2C=CCCN2C(C2CCCC(=O)C2)=O)=O)C1 95331,Cc1c(CC(=O)NCC=C2CCN(C(=O)CCCCN(C)C)CC2)cnn1C 95332,CC1CCC(C(=O)NC2CC2CNC(c2ccnnc2O)=O)CC1 95333,c1(CNC(C2(C(=O)NC3CCN(C)C3)CCCO2)=O)c[nH]c2ccncc12 95334,Cc1cc(N2CC(CN(C(=O)CC(C)c3cnn(C)c3)C)C2)c(Br)cc1[N+](=O)[O-] 95335,Nc1cc(C(N2CCN(C(=O)C3=COCCC3)CC(O)C2)=O)c(F)c(F)c1F 95336,c1(C(N2CCCC(C)(NC(=O)CCC3CC3(F)F)C2)=O)ccc([N+](=O)[O-])cc1 95337,N1(C(c2c(CC)cc(F)cc2)=O)CC2CCN(C(c3cnc(N)c(N)c3)=O)C2C1 95338,c1(C(=O)NCc2nc(C(=O)NCC3CC3)co2)cnc(O)c(F)c1 95339,C(=O)(C(F)C(CC)CC)N1C(CNC(CN(C2CC2)CC)=O)CCCCC1 95340,Cc1cnc(C(=O)NC2CCN(C(=O)C=CC3COC(C)(C)O3)C2)cc1Br 95341,c1(CCC(=O)NCC2N(C(c3occ(C)c3C)=O)CC2)c(Cl)cncc1Cl 95342,C1(NC(CSCC#C)=O)C2CC3CN(C(=O)CC(n4nc(C)cc4C)C)C1C3C2 95343,c1(C(=O)NCC(CNC(CCNS(CC)(=O)=O)=O)(C)C)cc(Cl)nnc1O 95344,c1(C(=O)NCCCOCCN(C)C(C2CC23CCOC3)=O)cn2cccnc2n1 95345,c1(C(N(C(C(=O)NC(C(=O)OCCC)(C)C)C)CCC)=O)ccc(CC)c(F)c1 95346,CCCC(C(O)C(=O)N1CCC(N(C)CC)C1)NC(=O)CCn1cnc(=N)[nH]1 95347,CC(C)(F)C(C)(F)C(=O)N1CCCN(C(C2CCCCN2C2CCCC2)=O)CC1 95348,C(=O)(C1=CCCN(C(C2C=CC=CC=C2)=O)C1)NCC=CCCC 95349,CC1CCCc2c(C(=O)NC3CC(CCNC(=O)CN4CCCC4=O)C3)cnn21 95350,CC1C(C(F)(F)F)NCCN1C(C1(c2cccc(F)c2)CC(N)C1)=O 95351,C12(C(N3C4C(NC(CC5(OCC)CC5)=O)CC(C4)C3)=O)CCC(CO)(CC1)CC2 95352,n1(CC)c(O)nc2cc(C(=O)NCC(C)NC(c3ccc(Cl)c(N)c3)=O)ccc12 95353,C1(CC)COC(C)CN1C(c1nc(F)ccc1Br)C(=O)NC1CC(F)(F)C1 95354,C12(NC(C=CC(=O)N(C)C)=O)CCCCC1N(C(=O)Cc1csc(=N)[nH]1)CC2 95355,N1(CC(=O)NCC(CNC(CCOC(C)=O)=O)C)CCCCC1C 95356,CC1OC2(C)CC1(C(N1CC3CC3(CNC(c3ccc(C#N)cn3)=O)C1)=O)C2 95357,C1(CC(=O)NCCC)CN(C(c2cc[nH]c(=N)n2)=O)CCO1 95358,C(=O)(C(O)C(F)(F)F)N1CC(C(C)(C)O)(CNC(=O)Cc2ccccc2)C1 95359,c1(OC)ccc2c(ccn2CC(=O)N(CC(C)NC(=O)CCCF)C)c1 95360,c1(C(=O)NCC2N(C(C3CCC3)=O)CCN(C)C2)nnc(O)c(Br)c1O 95361,C1(C(=O)NC2C(C)(C)C(Nc3ncc(Br)cn3)C2)CC2CCCCCCC12 95362,CC1CC(C(N2CC(NC(C3(C)CC3(F)Cl)=O)C2)=O)CCS1 95363,O=C1CC(c2ccc(C(=O)NCc3ccc(Cl)cn3)cc2)NC(=O)N1 95364,C(=O)(C(=O)N=S(C)(C)=O)N1CC(C)(c2cn(C3CC4OC(=O)CC34)nn2)C1 95365,C1(CC)CCN(C(=O)C(O)C(F)(F)F)C(C(N2CCCN(C(N)=O)CC2)=O)C1 95366,c1(C(CNC(c2c(C(C)C)n[nH]c2)=O)C(F)F)c[nH]c2ccccc12 95367,C1(CC)CCCC1C(=O)NCC1(NC(=O)C(C)NC2(CO)CCCC2)CCOC1 95368,C1(NC(C2CC(NC(C3CNC(=O)N3)=O)C2)=O)CC2CC(O)C1C2 95369,C1(C(=O)NC2CC(C3CCC3)C2)(CC)CCCN(C(=O)CC2CC2)C1 95370,N1(C(C(n2nnnc2C(C)(C)C)C)=O)CC(NC(=O)C(C)C(C)(F)F)C(C)(C)C1 95371,CC(C)CCC(C(=O)NCC1(O)CC1)NC(=O)C(C)CC(F)F 95372,C(CC(N)=O)(C(=O)NC(c1ccccc1O)C)NC(CC(C)OC)=O 95373,CC1(C)Cc2ccc(C(N3CC(F)(CNC(C4CC45CCCC5)=O)C3)=O)cc2C1 95374,C1(OC)CN(C(=O)CN2CSCC2=O)CC1NC(C12CC1CNC2=O)=O 95375,c1(OC(C)C)cccc(C(=O)NC2CC(NC(=O)Cc3cnsc3)C2)n1 95376,c1(C(=O)NCCC2CC(NC(C3N(CCC)CCC3)=O)C2)cccc2sccc12 95377,C(C)(CCC(=O)NC1CCCC1NC(C1(NC(N)=O)CC1)=O)OCC 95378,c1(C(=O)NC2CN(C(c3cc(CC)no3)=O)CC(C)C2)sc2cncn2c1C 95379,c1(-c2ccc(C)cc2)cn2cnc(C(=O)Nc3nc(C)ccc3C#N)c2s1 95380,N1(C(CCNC(C)=O)=O)CCCCC1CCCNC(C1CC2CCC1C2)=O 95381,C1(C(N2CCC(c3ccccc3)C2)C(=O)NC(C)(C)C)CCOC2(CCC2)C1 95382,c1(SCC)cccnc1C(=O)NC(C1CCCN(C(c2cc(C)co2)=O)C1)C 95383,FC1(F)CCCC(CN=C(NCC2CCCCO2)NCCOCF)C1 95384,c1(C(=O)NCCC2CN(C(c3cc(C(C)(C)C)n[nH]3)=O)C2)cccc2c1CCC2 95385,C1(NC(CCCSC)=O)CC2CCC(C1)N2C(=O)C=Cc1ccc[nH]1 95386,N1(C(CCCOCC)=O)CC2(CC(NC(=O)C(F)(F)c3ccccn3)C2)C1 95387,C1(CC(=O)NC(C)CCOC)(OC)CN(C(C2(N(C)C)CC2)=O)C1 95388,C1(C(=O)NC(CNC(C(CC)CO)=O)CC)CCn2c(O)nnc2C1 95389,N1(C(c2cnc(COC)s2)=O)CC2C(CNC(=O)C(n3ccnc3C)C)C2C1 95390,CCCC(C(F)(F)F)NC(=O)C=C(C)CNC(c1ccc(OC)s1)=O 95391,C=C(C)CCCC(=O)NC1CCC1NC(=O)CC1CCCCN1C(C)=O 95392,N1(C(c2ccc(CC#N)cc2)=O)CCCC2(CCN(C(=O)CNS(N)(=O)=O)C2)C1 95393,c1(NC(C(C)OCc2cccc(C)c2)=O)cccc2c1CC(=O)N2 95394,C1(NC(C2CC(C(F)(F)F)(OC)C2)=O)CN(C(=O)CC(C)(C)O)CCC1F 95395,c1(OCC)cc(C)nc(N2CCOC(c3cc(C)cc(C)c3)C2)n1 95396,C(=O)(C1CCc2ccccc21)N(CCCN(C(CCc1cc(C)on1)=O)C)C 95397,C12(C(N3CC(O)(C(C(=O)N(C(C)C)C)F)C3)=O)CCC(CC1=O)C2 95398,N1(C(C(C(=O)OCC)F)=O)CC2(CCN(C(c3ccc(F)cc3O)=O)C2)C1 95399,c1(NC(C(C)OC(C2C3CCC23c2ccccc2)=O)=O)cnc2[nH]cc(C#N)c2c1 95400,N1(C(c2cc(C(C)=O)[nH]n2)=O)CCC2(CCN(C(=O)CN3CCCCC3C)C2)C1 95401,C#CCC(O)C(=O)N(C)CC1CCCN(C(=O)C(O)C2CC2)C1 95402,c1(C(=O)NC2CN(C(c3cccn3Cc3ccccc3)=O)C2)ccc(OC)nc1 95403,C1(C)CCN(C)C1.c1(N(NS(=O)(=O)NCc2cnn(C)c2)C)nnnn1C 95404,C(=O)(C(O)CCCCC)N1C(C2(NC(CC=CCC)=O)CC2)CCC1 95405,CC(C)(C)S(=O)(=O)CC(=O)N1CCN(C(=O)CCN2CCCC2=O)C(C(F)F)C1 95406,C1(CNC(=O)CC2(O)CCC2)CN(C(c2ccc3[nH]ccc3c2)=O)CC12CCC2 95407,c1(OC)ccc(C(=O)NCc2csc(CNC(=O)CCF)n2)c2ccccc12 95408,N1(C(C(c2ccc(F)cc2)CC)=O)CC(CC(N)=O)OC(C)(C)C1 95409,C(=O)(NNC(=O)CCN1CCCCC1)NC1CCN(CCC)C1 95410,C1(CNC(C2CC(N3CCCC3)C2)=O)CCC2CN(C(c3ccsn3)=O)CC12 95411,C1(CNC(CCOCCCOC)=O)CN(C(=O)C(c2ccc(Cl)cc2)=O)CCO1 95412,C1(CCNC(CN(CC)CC)=O)CCC(NC(c2ccc(C)o2)=O)C1 95413,C(=O)(C1CCc2c[nH]nc21)N(C(CC)CC(=O)N1CC(CO)C1(C)C)C 95414,c1(OCC)ccc(F)c(C(=O)NC(C2CN(C(=O)C3=CCCS3)CCO2)C)c1F 95415,Cc1ccc(C(=O)NCC2(CNC(=O)CC3CC4(CCC4)C3)CC2)nn1 95416,c1(CCCC(=O)NC2CCCC(CNC(C=CCOC)=O)C2)c(F)cccc1F 95417,CC1(C)CC(CNC(c2ccc(F)c(F)c2F)=O)CN(C(C2COC(=O)O2)=O)C1 95418,c1(C(=O)NC2C(CNC(C(N3CCC(C)C3)=O)=O)C2)ccn2nccc2n1 95419,N1(C(CCCOC(C)=O)=O)CCN(C)CC1C(N1CC(CCO)C1)=O 95420,N1(C(Cc2c(C)nc(Cl)cc2)=O)CCC2(CC1)CCN(C(c1ccc(Br)o1)=O)C2 95421,C1(CCSC)C(=O)N1.[N-]=[N+]=NC1(C(=O)O)CC1.C1CC1 95422,N1(C(c2nc(CC)sc2Br)C(=O)NCCCF)CCCN(c2nc(C)cs2)CC1 95423,C1(OC)CN(C(=O)C(C)Oc2cccc(Br)c2)C(C)(C)C1 95424,c1(-n2cnc(C(=O)OC(C(c3ccc(C(C)C)o3)=O)C)n2)ncc(Cl)cn1 95425,N1(C(c2c(C)nc(CO)s2)=O)CC=C(CNC(C23CCC2C3)=O)CC1 95426,c1(C(=O)NCC2N(C(C3C(COC)C3)=O)CC2)cnn(CC(F)F)c1C 95427,N1(C(C(C)n2cccc2)=O)CCCC(CC(=O)NCCCc2cc[nH]n2)CC1 95428,C1(F)(CNC(C2(CC#C)CC=CCC2)=O)CCN(C(=O)C=CC)CC1 95429,C(C(=O)N1CC(c2ccccc2)(NC(=O)Cc2cnns2)C1)(C(C)(C)C)SC 95430,c1(CC)nc2n(n1)CC(NC(=O)NCC1CCCN(C)C1=O)CC2 95431,C1(C(=O)OC)C(C)CCN1CC(O)CNC(N)=O 95432,C(=O)(C(CNC(C12CCCC(CO1)C2)=O)C(C)C)N(CCC(C)C)C 95433,N1(C(CCCN2CCN(C(C)C)CC2)=O)CCC2CCN(C(=O)CO)CC12 95434,C1(CN(C(c2cc(C)oc2)=O)C)CCN(C(C2CCOC(=O)N2)=O)CC1 95435,C(N=c1cc(C)[nH]c(=NCc2cc(C)co2)[nH]1)C1(OC)CC(C)(C)CC(C)(C)C1 95436,N1(C(C2(SC)CN(C(=O)CCN3CCCCC3)C2)=O)CC2(C1)CN(C)CCO2 95437,CC1CCN(C(=O)C(C)SCc2cccc(Cl)c2)CCS1(=O)=O 95438,CN1C(=O)OCC1C(N1CCC(CCNC(C23CC(C)(CO2)C3)=O)C1)=O 95439,c1(C2N(C(C3COCC4(CCC4)O3)=O)CCC2)c(F)cc(Br)cc1F 95440,c1(C(=O)NC2CC(CCNC(C(COC)(C)OC)=O)C2)cc(C)c(C)cc1N 95441,c1(C(N2CC(COC)C2)=O)ccc(Br)c2ccncc12.c12cnc(cn1)o2 95442,C1(NC(CC(=O)OCC)=O)(CNC(=O)C(=O)Nc2cnn(C)c2)CCOCC1 95443,CCC(CC)C(C(=O)N1CCC(N(C(=O)CCn2ccnc2C)CCO)C1)OC 95444,c1(C(N2CCC(NC(CNC(=O)CCCCO)=O)C2)=O)cccc(C=C(F)F)c1 95445,C1(CCOC)(OC)CCN(Cc2cnc(F)cc2C)CC1 95446,C12(C(=O)NC(CC)CN3CCNCC3)CCCCC(CNC1)C2(F)F 95447,N1(C(c2cc(CNC(=O)CC3CCCC3)on2)=O)CCn2cnnc2C1 95448,N1(C(c2cc(OC)c(Br)s2)=O)CCCC12CCCN(C(=O)C(C)O)C2 95449,N1(C(C(CC(=O)OCC)C)=O)CCC(C)N(C(=O)CCc2cn[nH]c2)CC1 95450,c1(OC)noc(C)c1CNC(c1ccccc1OC(F)F)C 95451,Cc1ccc(C=CC(=O)NC2CN(C(=O)OC(C)(C)C)CC2C)nc1 95452,C(C1=C(C(=O)OC)C(c2cc(OC)c(O)c([N+](=O)[O-])c2)NC(=O)N1CCF)SC 95453,C(=O)(C1=CC(O)C(NC(=O)CCC2CCCC2)C1)N1CC(C#N)(SC)C1 95454,C(=O)(CC(O)C(C)C)N1C(C(N2C(CC)(CC)CC2)=O)CC(=O)C1 95455,c1(OC)cc(C(=O)NCCn2cc(SC(C)Cn3ccnc3)nn2)nc(C)c1 95456,c1(COC(c2cc3ccccc3[nH]2)=O)c(F)c(F)cc(Br)c1F 95457,N1(C(C2(OC)CCC(C)C2)=O)CCC(O)(CNC(C2CCOC2)=O)CC1 95458,c1(CNCC2(OC)CCN(C)CC2)cccc2c1NC(=O)CO2 95459,C1(CNC(c2noc(CC)c2C)=O)CC(C)(C)CN1C(=O)CC(O)CN(C)C 95460,CCC(C(=O)NC(C)(CO)C(=O)Nc1cnn(C2CC2)c1C)C(C)C 95461,C(C(C)(C)CN(C)C(C1CC1(Cl)Cl)=O)NC(C(C1CC(F)(F)C1)OC)=O 95462,CC(C)CC(F)(F)C(=O)N1CCC(CC(C)NC(=O)C=CC2CCOC2)CC1 95463,C(=O)(CCCC(=O)N1CCCCC1CCC(=O)NCc1ccc(C)cc1)OC 95464,c1(OC)ccc(C(=O)NC(C2(CNCC3(C)CC=CC3)CC2)C)c(OC)c1OC 95465,c1(NCCC2CC=CCC2)cc(N2CCC(c3cc[nH]n3)C2)ncn1 95466,C1(NC(C(CCC)NC(C2CC(C3CC3)C2)=O)=O)CCn2nnnc2C1 95467,N1(C(Cc2cccc(CC)c2)=O)C2CCCC1CN(C(c1coc(SC)c1)=O)C2 95468,C1(CNC(C(C2CCOC2)OC)=O)CCN(C(c2cc(Cl)on2)=O)C1 95469,C(=O)(CS(=O)(=O)CC(C)C)N1CCC(NC(Cc2c(C)noc2)=O)C(C(C)C)C1 95470,C1(NC(c2nc(NC(C)=O)sc2)=O)CCSC12CN(C(C13CCCC1C3(F)F)=O)C2 95471,N1(C(C=C(C)C)=O)CCC2(CC1)CN(C(C1(O)CC3CCC1C3)=O)CC2CO 95472,C1(O)(CC(=O)NCC(C)(C2CC2)NC(c2n(CC)ccc2)=O)CCOCC1 95473,c1(NC2(C(=O)OC)CCCOC2)ccc(C#N)c(C)n1 95474,C(c1ccccc1Br)=CC(=O)NC1CN(C(c2ccc(C(N)=O)[nH]2)=O)C1 95475,c1(C(N(CC(CNC(CCCOCCOCC)=O)O)C)=O)nn(C)nc1C 95476,c1(CC)c(C(N2CCC(NCc3nc(C)no3)C(C)C2)=O)cccc1F 95477,CC1CC(C(=O)NCC(F)C2CCC2)CCN1C(c1occ2c1CCC2)=O 95478,C1(CC(=O)NCCCC2CCCCN2C(=O)CSC2CCCC2)CCCOCC1 95479,C(=O)(CC(C(F)F)NC(C1OCCO1)=O)N(CC=C)CC 95480,C1(CC(=O)N(C2CNCCC2O)C)CCC(F)(F)CO1 95481,C(N=c1nc2c(cnn2C(C)C)c(NC2CC3CC(O)C2C3)[nH]1)c1c(C)occ1 95482,C(CC(=O)NCCCCN(C(=O)CCSCCC)C)OCC#C 95483,C1(NC(c2ccn(CCCC)n2)=O)CN(C(C2C(F)(F)C23CCC3)=O)CCC1O 95484,CC(C)CC(CNC(=O)COCCc1cccc(F)c1)NC(C1CC1(C)C)=O 95485,Cn1cnc2cccc(C(N3CCC(CNC(C4CC4(F)F)=O)C3)=O)c12 95486,c1(CNCc2c(C)sc(Br)n2)c(Cl)sc(Cl)c1Cl 95487,C(C1=CCN(C(C2CC3C=CC2C3)=O)CC1)NC(C(c1cnn(C)c1)OC)=O 95488,O=C(C1CCCc2ncnn21)NC1CN(C(C2CC(Cl)(Cl)C2)=O)C1 95489,O=C(CCCCCF)NC12CCC(CC1NC(=O)C(c1ccc(F)cc1F)=O)C2 95490,Cn1nc(C(=O)NCCC2(NC(c3cc[nH]n3)=O)CCC2)cc1C(F)(F)F 95491,C(=O)(C1=C(C#N)CCC1)NC(CC)C(N1CCC2(C=CCO2)C1)=O 95492,C1(C(=O)NCC(=C)CCNC(c2cscc2C(N)=O)=O)(CC)CCC(C)(C)CC1 95493,CC1CN(C(C2CCC(C)(O)CC2)=O)CCC1NC(C1SC2C=CC1CC2)=O 95494,C(=O)(CC(O)C(C)(C)C)N(CCN(C(c1ccnc(OC)c1F)=O)C)C 95495,Cn1cnnc1CCC(=O)N1CC(c2ocnc2Cn2cc(C3(C)CC3)nn2)C1 95496,CC1Oc2ccccc2N(CC(=O)N2CCN(Cc3ccc(N)cn3)CC2)C1=O 95497,N1(C(C2(CC)CCN(C(C3CC3Cl)=O)CC2)=O)CCC2CN(C)CC2C1 95498,C(CCC(C)(C)NC(=O)Cc1cnc(C2CC2)[nH]1)NC(C(C)OCCCC)=O 95499,CCC(CCC(=O)NCc1cccc(C#N)n1)NC(=O)CC1CCCN1C 95500,C(C)(C)(CCNC(C1CC(C)(C)C1)=O)NC(C1N(C)CC1)=O 95501,Cc1cnc2c(CN3CC4CC3CC4N3CCC(OC(C)C)CC3)cnn2c1 95502,c1(C(=O)NC(CNC(c2cc(C)c(N)cn2)=O)C2CC2)ccc2sc(C)nc2c1 95503,C(CCCCC(=O)NC(C1CCC1)C)N(C(C1(C(=O)OC)CC1)=O)C 95504,c1(OC)coc(C(=O)N(C(C)CNC(c2csc(C)c2C)=O)C)cc1=O 95505,c1(C(N2CC(CC#N)N(C(c3ccc(O)nn3)=O)CC2)=O)ccc2ocnc2c1 95506,N1(C(c2ncn(C(C)(C)C)c2)=O)CC(NC(c2ocnc2C(F)F)=O)C(CO)C1 95507,C#CCCCCCCC(=O)N1CCC(C(C)C(=O)N(C(C)C(=O)OC)C)CC1 95508,N1(C(C2CN(C)C2)=O)CCCC2(C1)CN(C(=O)Cc1ncn3c1CCC3)CCO2 95509,C1(C(N2C(CN(C)Cn3cc(C(=O)N)nn3)CCC2)=O)CC2CCC2C1.C1CC1 95510,c1(C(=O)NCC(CC(C)C)NC(=O)CN(CC(C)(C)C)C)nc2ncccn2n1 95511,Cc1ncc(C(N2CC(C3CCCCN3C(=O)C=Cc3ccsc3)C2)=O)n1C 95512,C(CNC(C1CN(C(C)=O)C1)=O)(C(C)(C)C)NC(C(CC1CCC1)OC)=O 95513,C#CC1(NC(c2cnn(CCNC(C3CCSC(C)C3)=O)c2)=O)CCCCC1 95514,c1(OC)cc(C(C(=O)NC2(C)CC2)N(C(C)C)C)c(Br)cn1 95515,c1(CC)c(Cl)nc(C2CCC2)[nH]c1=NCC(C)NC(c1cccc2nsnc12)=O 95516,C1(C(=O)NCC(CCC)O)CCN(C(=O)C(C(=O)OC)OC)C12CC2 95517,c1(C(N2CC(NC(c3scc(C)c3C)=O)C(F)C2)=O)ccc2c(c1)CCC=C2 95518,CCC(O)C(C)C(=O)NC1CC(c2ccccc2)(NC(c2cc[nH]c(=N)c2)=O)C1 95519,C1(C2CCN(C(C3CCNC3=O)=O)CC2)(NC(C2=NOC(C)C2)=O)CC1 95520,n1(CC(=O)NCCOCCNC(=O)CC2CC(F)(F)C2)cnc(Br)c1 95521,c1(OC)cc(CCC(=O)N(C2CCC(NC(=O)C(C)(C)C)C2)C)ccc1F 95522,Cc1ccccc1CN1CCC(N(C(=O)C(CO)c2ccccc2)C)C1 95523,c1(C(=O)NC(CNC(c2c(OC)cc(Cl)c(C)c2)=O)C)ccc2c(C)noc2c1 95524,Cc1ccc(C(N2C(C(=O)NCC3(C)CC(O)C3)CC2C)=O)cc1 95525,N1(C(C(C)C2CCC2)=O)CCC2C(C1)NC(=O)CN2C(=O)C(=O)N1CCCC1 95526,N1(C(C(C)N(C(C)=O)C)=O)CCC(O)(CNC(=O)CN2CCCC2CO)CC1 95527,c1(C(=O)NCC2(C(F)F)CCN(C(C(CCC)O)=O)C2)cc2ccc(C)cc2[nH]1 95528,C(CCCCCNC(=O)C1CC1)NC(C(n1cc(Br)cn1)C)=O 95529,C1(c2c(C)cccc2C)CCN1N1CC2CCC(CO)(CC2)C1 95530,CC12CCC1CN(C(C1CCC(CNC(c3cnn[nH]3)=O)C1)=O)C2 95531,C1(C(=O)NCC(C)N(C(CCC=CC)=O)C)CCCC(OC)C1 95532,c1(C(N2CCC(O)(C(C)NC(=O)CNS(N)(=O)=O)C2)=O)cc(Cl)cc(Cl)c1 95533,c1(C(N(CCCCN(C(=O)Cn2ncc(Br)n2)C)C)=O)cnc(Cl)n1C 95534,C(=O)(C1=NN(C)C(=O)CC1)NC1CC(N(C(C(c2ccc(Cl)cc2)C)=O)C)C1 95535,C(=O)(CC(F)(F)C(C)C)N(CC)CC1CCCN1C(=O)C=Cc1c(C)noc1C 95536,N1(C(c2ccc(OC)nc2)=O)CC2CC(NC(c3cc(C)nc(C)n3)=O)C(C2)C1 95537,c1(OC)cc(O)c(CNC2CC2C(=O)Nc2ccc(Br)nc2F)c(Br)c1 95538,N1(C(C=CC=CC)=O)CCC(NC(c2cnn3ccnc(N)c23)=O)C12CCCC2 95539,CCC(C(C)(F)F)NC(=O)CN(C1CC(C#N)C1)C(c1cc(C)c(C)[nH]1)=O 95540,c1(OC)cc(C(N2CC=CC2CNC(=O)C(C)C(C)C)=O)cc(Br)c1 95541,Cc1c(-n2cc(CC3CCN(C(c4ccc(CO)cc4)=O)C3)nn2)cccc1Cl 95542,O=C(N=c1[nH][nH]cc1I)C1CC(F)CN(S(=O)(=O)c2ccc(Cl)s2)C1 95543,c1(CNC(C(CC)C)c2nnnn2CC(F)F)ccc(F)c(F)c1C 95544,CC1(CN(C(C2(C)CN(C(=O)CC34CC(C3)C4)C2)=O)C2CC2)CCOCC1 95545,C1(NC(c2coc(Cl)n2)=O)CCC2CCN(C(C3CCC(=O)N(C4CC4)C3)=O)C12 95546,c1(CC)nn(C)c(CC(=O)NC2CCN(C(=O)COC3CCC3)C2C(C)C)c1Cl 95547,n1(CC(=O)NCCC(C)N(C(c2c(C)n[nH]c2)=O)C)cc(Cl)c(O)nc1=O 95548,c1(C(=O)NC2C(CNC(Cc3scc(C)n3)=O)CCCC2)cc2ccccc2o1 95549,N1(C(CCC=C=C)=O)CC(NC(=O)Cn2ccccc2=O)C2(CCC2)C1 95550,C1(C(=O)NC(CCNC(c2c(C)snc2)=O)C(C)C)CC2(CCOC2)C1 95551,C(=O)(CC(C)(O)CC(=O)O)NC1CCCN(C(c2ccc(C)cc2C(C)C)=O)C1 95552,c1(CC)cc(C(=O)N(CC(C)NC(=O)C(F)(F)c2cncs2)C)cc(O)n1 95553,c1(C(=O)NCC(CNC(c2nc(CCCC)sc2)=O)C)c(C(C)C)cnn1C 95554,Fc1ccc(C2CCCCC2)cc1Cl.c1(CNC2CC2)nnnn1C1CCOC1 95555,c1(C(N2CC(C)C(CNC(=O)C3=CC4C=CC3C4)CC2)=O)cccn2nccc12 95556,C(=O)(C1OCC(C)c2ccccc21)N(CCNC(c1cc(CS(C)(=O)=O)on1)=O)CC 95557,N1(CCC(N2C(CO)CC(NC(C(C=C)(C)CC)=O)C2)=O)Cc2ccccc2C1 95558,N1(C(C(C=C=C)C)=O)CC2N(C(C3CC4(CC4)CO3)=O)CCC2(C)C1 95559,C1(C(=O)NCCNC(C2CC3(C2)CC32CCC2)=O)CCCC12OCCO2 95560,C1(C(N(C2CCC(NC(C=Cc3ccc(C)o3)=O)CC2)C)=O)CCCC(C#N)C1 95561,N1(C(c2cc(C)c(C)nn2)=O)CC(C)CN(C(c2ccn(C)c(=O)c2)=O)C(C)C1 95562,C1(NC(C(C)OCCOC)=O)CC(O)CN(C(=O)CCS(=O)(=O)N(C)C)C1 95563,N1(C(c2ccc(C)n2C)=O)CCN(C(C2(C)CCCNS2(=O)=O)=O)CC12CCC2 95564,CCCC(C)(O)C(=O)N1C2CCC1C(NC(c1ccccc1OCCF)=O)C2 95565,C(=O)(C1CCCn2ncnc21)NC(CNC(c1cccc(C)c1Cl)=O)C 95566,C(=O)(C1=CCCCC1P(C)(C)=O)N1C(C(C)NC(CCOC)=O)CCC1 95567,N1(C(C2C3(CC(NC(c4cnc(CC)o4)=O)C3)C2)=O)CC2CC(C)C2C1 95568,C#Cc1ccc(C(c2nnnn2C(C)C)NCc2ccc(F)nc2F)cc1 95569,Cc1cc(C(=O)NC2C=CCC(C(=O)N(C3CCSC3)C)C2)ncc1F 95570,C1(CC(=O)OCC(C(C)C)(C)C)Sc2ccccc2NC1=O 95571,C1(COC)(NC(C2CCCCS2)=O)CCCN(C(c2cn(C)nn2)=O)C1 95572,Cc1cc(C#N)cc(C)c1C(=O)NC(CNC(=O)C=Cc1cncn1C)C1CC1 95573,CCCCCC(O)C(=O)N1CC(C(=O)NCC2(C)CC(C)=NO2)(CC)C1 95574,CC1=C(C(=O)NCCCCCN(C(=O)C(n2ccnc2C)C)C(C)C)CCC1 95575,c1(C(=O)NC(CC)CN(C(=O)CC(C)c2cccnc2)C)ccsc1S(N)(=O)=O 95576,c1(SC)ccc(NC(=O)NCCc2cncc(C)n2)c(Br)c1 95577,N1(C(C2(C)CCN(S(=O)(=O)C3CC3)CC2)=O)CCC2(CCNC(=O)O2)CC1 95578,O=C1CCCCC(C(N2CC(O)CC2CNC(C2CC3CC2CC3O)=O)=O)N1 95579,CCC(O)C(C)C(=O)NCc1cc[nH]c1C(=O)NC(C)CCO 95580,C1(C(N2CC(C#C)(N(C)C)C2)=O)CC(F)(F)CN1C(c1cc(C)on1)=O 95581,C1(COC)(CNC(=O)CC=CCc2ccccc2)CCN(C(c2cnns2)=O)C1 95582,C12(C(=O)NC(CCOC)CNC(c3ncc(C)cn3)=O)COCC1C2(F)F 95583,C12(N(C)C)CCC(NC(=O)CCCc3cnc[nH]3)(CC1)OC2 95584,c1(C(N2CCC(C(=O)NCC3(C)CCOCC3)C(O)C2)=O)ccc(C#N)c(F)c1 95585,c1(C(C)=O)ccc(O)c(NC(=O)C=CC2CCCN2C(=O)COCC(C)C)c1 95586,N1(C(C(N2C(c3nc(C)[nH]n3)COCC2)=O)=O)CCC2CC1C(=O)N2C 95587,Cc1ccc(C#N)cc1C(N1CCC(NC(C2(C)CC(C)(C)C2)=O)C(C)C1)=O 95588,N1(C(C(C=C)O)=O)CC(NC(=O)C(C)Cc2ccc(OC)cc2)C(C)(C)C1 95589,C(=O)(CC(C)(C)C(C)(F)F)NC(CNC(C1(C)CCN(C)C1)=O)(C)C 95590,N1(C(c2cc(COC)no2)=O)CCOC2(C1)CN(C(c1ccnn1COC)=O)C2 95591,N1(C(C(C)(C)O)=O)Cc2ccccc2CC1CNC(=O)Cc1c[nH]nc1O 95592,CCCCCC(C)(C)CNC(c1sc(-c2ccc(OC)cc2)nc1C)=O 95593,c1(C(N2CC(CNC(CC(=O)NCC#C)=O)C2)=O)cncc2sccc12 95594,N1(C(c2ccsn2)=O)CCc2sc(CNC(C3(c4cc[nH]n4)CC3)=O)nc2C1 95595,CCCCC(O)C(=O)N(CC(=O)NCc1cnc(C)n1CC)CCC 95596,CN1CCCC(O)(CC(N2CCC2CNC(C2CC(=O)CO2)=O)=O)C1 95597,C(=O)(CC(C(C)(C)C)NC(=O)CC1=CCOCC1)NCc1c(C)non1 95598,c1(C(N2CC(N(C(CC(n3ccc(C)n3)C)=O)C)C2)=O)n[nH]c2c1CN(C)CC2 95599,c1(CC(=O)NCC(C2CCOC2)NC(CCC#C)=O)cccnc1OC 95600,n1(CC(CC)O)cc(C(=O)NCC(C)NC(C2(CC)CCOC2)=O)nn1 95601,C1(C(=O)NCC2(CO)C(C)(C)C2)CC2CC1CC2NC(=O)CCCC#N 95602,C1(C)(CC)CC(NC(C2CC(=O)NC(=O)C2)=O)CN1C(c1cnco1)=O 95603,C1(NC(c2cnc(C3CC3)[nH]2)=O)(CF)CCN(C(=O)Cn2cnc(C(F)(F)F)c2)C1 95604,N(S(=O)(=O)N1Cc2ccccc2C1)Cc1cccc(N=[N+]=[N-])c1 95605,c1(C(=O)NC23CCN(C(CC(=O)NCC)=O)C2CCC3)cnc2c(c1)nnn2C 95606,N1(C(C(C)OCCC(C)C)=O)CCN(C(=O)C=CS(C)(=O)=O)C(C(C)C)C1 95607,S(=O)(=O)(c1cc(Br)c(OC)cc1Br)NC(C(C)C)C(F)(F)F 95608,N#CC1CCC(C(=O)NCC2(CNC(=O)CCC3CCOCC3)CC2)CC1 95609,C1(NC(=O)CCCC(F)(F)F)CCC2CN(C(c3ccc(O)nn3)=O)CCC2C1 95610,C1(CNC(c2cccc(Cl)n2)c2n(CC)ncn2)CC12CCC(F)(F)CC2 95611,N1(C(CC)=O)C(C)C2CC1C2NC(=O)CCCc1ccc(Cl)c(C)c1 95612,c1(NC(C2CCN(C(=O)C=C3CC3)CC2)C)ncnc(Cl)c1C 95613,c1(OC)ccc(CNC(=O)N(C)CCOc2c(C)cccc2C)cc1OC 95614,c1(C(C)C)ccc(C(N2CC(C)CC2C(=O)NC2C3COCC23)=O)cc1 95615,Cc1cccc(C(=O)NC2(C)CC(NC(=O)C(C3CC(F)(F)C3)O)C2)c1 95616,C1(C(=O)NC2CCN(C)CC2)CN(C(C2CC2C)=O)CC12C(=O)Nc1ccccc12 95617,N1(C(C2CC3(CC(NC(c4ccc(NC)cn4)=O)C3)C2)=O)CC2OCCOC2C1 95618,c1(C(N(CC(CN(C(C2(CSC)CC2)=O)C)O)C)=O)cn(C)cc1C(F)(F)F 95619,c1(CC(=O)NCCC(C)N(C(C(COC)C)=O)C)c(C)cccc1F 95620,N(C1CCC(NC(=O)Cc2cccs2)c2ccccc21)C(CC=C(C)C)=O 95621,N1(C(C=CCC2(NC(C(CC)CC)=O)CCC2)=O)CCN(CCOC)CC1C 95622,c1(N(CCCCN(C)C(c2cnn(C3CCCC3)c2)=O)C)ncnc(Cl)c1CO 95623,N1(CC(=O)NCC2CN(C(C(OC)OC)=O)C(C)CC2)C(=O)CC(C)(C)C1=O 95624,c1(CC)cc(C(=O)NC(c2ncc(C(=O)OC)s2)C)sc1CC 95625,N1(C(CNC(=O)OCC)=O)CCOCC(C)(CNC(=O)C(C)C2CCCO2)C1 95626,C1(C(=O)NC2(CNC(C3(C4CCC4)CC3)=O)CCC2)CC(c2ccccn2)=NO1 95627,C=CCC(C)(C)C(=O)NC.c1(C(=O)NCCC2(OC)CCC2)cnc(CC)s1 95628,CCC(C(=O)NCC(C)NC(c1ccc2nccn2c1)=O)C(C)(F)F 95629,c1(CC(=O)NC2C(NC(C(C)OC(C)(C)C)=O)C(O)C2)cncnc1O 95630,c1(C(=O)NCCCC(=O)NC2(CC=C)CC2)cncc(OCC)c1 95631,C1(C(=O)Nc2cccc(C3(C)CC3)c2)CC2CCCCN2C1=O 95632,c1(C(N2CC(NC(C34CCCC3C4(F)F)=O)CC(C)C2)=O)ccc2c(c1)OCO2 95633,c1(OC(C)C)ccccc1-c1cn(C(N2C(C)CCC2)=O)nn1.C1(O)CC1 95634,C(=O)(C(F)(F)c1ccccn1)NCC(C)(C1CC1)NC(=O)C(O)CN1CCCC1 95635,CCCC(C)CC(=O)N1CC(NC(c2ccnc(Cl)c2O)=O)C(C)C1 95636,Nc1ccccc1-c1cn(CCCC(=O)NCCc2csc(O)n2)nn1 95637,c1(-c2ccc(OCC)s2)cccc(CNC(c2cc(C)no2)=O)c1 95638,C(CCSC)(C(=O)N1CCC1C(=O)NOC(C)C)OC.c1(N)cnn(C(F)F)c1 95639,c1(C(=O)NCC(C)NC(=O)C(C2CC2)N(C)C)cc(-c2cccnc2)on1 95640,O=S(=O)(c1ccc(N2CCC3(CCC3)C2)cc1Br)NCC1C2CCCCC12 95641,N1(C(=O)CC2CCCN2c2ncc(F)c(N3CCC3)n2)CCc2c(O)ncnc2C1 95642,c1(C(C(=O)Nc2ccccc2Cl)N(CCOCC)CC)ccc(F)c(OC)c1 95643,C1(NC(N2CC(=O)NCCC2)=O)C2Cc3ccccc3C12 95644,C1(CC(=O)NCCN(C)C(C2CC2C(N)=O)=O)CCCCO1 95645,C1(C(N2C(CC(=O)N(C)Cc3cccc(O)c3)COCC2)=O)OCCN(C)C1=O 95646,N1(CC(CNc2ccc(CN(C3CCOCC3)CC)cc2)O)CCC(F)(F)C(C)C1 95647,c1(OC(c2ccc(C)cc2)CCCC2CCC(C)CC2)cc(C)cc(C)c1.C1CCNS1 95648,CCC(CC(=O)N1CCC(C2CC2)(CNC(c2cnsc2)=O)C1)C(F)F 95649,Cc1ncc2n1CCC(C(N1CC(C)(C)OCC1CNC(=O)C(C)(C)C#N)=O)C2 95650,C1(C(N2CC(C(=O)NC(C=C)(C)CC)C(OC)C2)=O)OCCCC1(C)C 95651,N1(C(c2cnc(CNC(C(CCCC)N(C)C)=O)nc2)=O)CCN(C)C(=O)C1C 95652,c1(C(C)OC)nn(C)c(C(N2CCN(C(=O)CN(C)C)C(CS(C)(=O)=O)C2)=O)c1Cl 95653,C(=O)(C(O)CCNC(c1ccc(N)cn1)=O)NC(COC(C)=O)CO 95654,Cc1cc(C)c(C(N2CCC(C)(NC(=O)CC3NC(=O)NC3=O)C2)=O)[nH]1 95655,Cc1nc(N2CC3CC2CN(C(=O)CCC(C)N(C)C)C3)ccc1[N+](=O)[O-] 95656,CC(CCN=c1nc(-c2ccccc2)c(F)c[nH]1)NC(=O)CC1CCN(C)C1 95657,N1(C(C2(C)CC2)=O)CCCC2C1CCN2C(C1CCc2ccccc2O1)=O 95658,Cc1cn2ccc(C(=O)NCC(C)(C(C)C)NC(c3cnnc(O)c3)=O)cc2n1 95659,C1(C(N2CC(CCNC(c3n[nH]cc3C3CCC3)=O)C2)=O)CCc2nncn2C1 95660,N1(C(C(C)NC(C=C)=O)=O)CC2C(C(=O)NC3CC(C(F)(F)F)C3)C2C1 95661,N1(C(c2ccc(C(F)F)cc2Cl)C(=O)NC)CC2(CCC2)CCC1C 95662,c1(C(N2C(CC)CN(C(C3CC(O)C3)=O)CC2)=O)c(F)cc(OC(F)F)cc1F 95663,c1(SC)ncc(C(N2CC(NC(c3cccn3C)=O)C3CC23)=O)n1C 95664,c1(C(=O)NCC23CC(NC(C4(C(C)(C)OC)CC4)=O)(C2)C3)cccc(CO)n1 95665,C12(C(=O)OCc3cc(C4CCCC4)no3)CC1CCN2C(=O)Nc1ccc(Br)o1 95666,C1(C(=O)NCCN(C(C=CC=CC)=O)CCOCCO)CCCC2(CCC2)O1 95667,c1(OC)ccc(CNC(=O)CNc2ccn(CCF)n2)cc1OC 95668,c1(OC)ccc(-n2nc(CC(C)C)nc2C(c2ccccc2)F)cc1F 95669,c1(C(=O)NCC(CNC(C(C=CC)O)=O)C(F)(F)F)cncc(P(C)(C)=O)c1 95670,c1(NC(N2C3(C)CC(C(F)F)(C2)C3)=O)ccc2c(c1)CCO2 95671,C#CCCCCC(=O)N1CCN(CC2COCCN2C(=O)CCNC(C)=O)CC1 95672,Cc1nn(C)c(Cl)c1C(N1CCN(C(C2(COC(C)C)CC2)=O)CC1C)=O 95673,Cc1nn(C)c(C)c1CC(=O)NCC1CC(F)(CNC(=O)CC2(C)CC2(F)Cl)C1 95674,Cc1nn(C)c(C)c1OCC(=O)NCCC1CCC(NC(c2scnc2Cl)=O)C1 95675,Cc1ccc(C)c(OCC(N2CC3CC2C3NC(=O)C(C)(C)C(F)F)=O)c1 95676,C(=O)(CC(C(C)(C)C)NC(=O)C(C)CC#N)NCC1CCN(CC)C1 95677,N1(C(C(CC=C)C)=O)CC(C(=O)NC2CCC3(CC2)N=N3)CCC1(C)C 95678,C(=O)(CC(C)(C)C1CC1)NCCC1CCN(C(C(C)N(c2ccccc2)C)=O)C1 95679,C1(CCC(=O)NCCC(=C)CNC(=O)CN2CCCCC2)C(=O)NN=C1C 95680,CCC(C)C(CNC(C1CSCN1C(C1(CC)CCC1)=O)=O)CO 95681,C1(NC(C(CC)Oc2ccccc2)=O)CCCC(CNC(=O)C(F)=CCCF)C1 95682,c1(C(=O)NC(C(C)NC(=O)C(C2(O)CCCC2)F)C)cnn2ccn(C)c12 95683,CCCC(C(=O)N1CCC(CCNC(c2[nH]cc3c2CCC3)=O)CC1)C(C)C 95684,c1(CCC)c(C(=O)NCC2(F)CN(C(C34COCC3C4)=O)C2)nnn1CC 95685,C1(CNC(c2ccc(C#C)o2)=O)CC(C)(C)CCC1NC(c1occ(C)c1C)=O 95686,C1(CNC(COc2cc(C)on2)=O)CN(c2nc(C)nc(C)c2C)CCC1(F)F 95687,CC1(CNC(C2CN3CCN2CC3)=O)CCN(C(C23COCC(C2)C3)=O)CC1 95688,Cc1cnc2nccc(C(=O)NCC(C)NC(=O)C(C(C)C)n3cccc3)c2c1 95689,N1(C(c2cccc(-n3ccc(C)n3)n2)=O)CCc2c(C)cccc2C1C(=O)O 95690,c1(C(=O)NCC(CCOC)NC(c2ccc(C)c(F)c2)=O)ncc(Cl)cc1F 95691,C(=O)(C(C)CC(C)(F)F)N1CC(CNC(C(C(CC)C)O)=O)(OC)C1 95692,c1(C(=O)NCCC(C)N(C(C(C2CC2)OCC)=O)C)c(C)ccc(Cl)c1O 95693,N1(C(c2csc(-c3ccccc3)n2)C(=O)NCCC(=O)OCC)CC(C)C(C)C1 95694,N1(C(CSc2n(C)nnn2)=O)CCN(C(=O)C(C)(C)NS(C)(=O)=O)CC12CCC2 95695,C1(C(=O)NC2C=CC(C(N3CC(C)(CC)C3)=O)C2)CCCCNC1=O 95696,N#Cc1cccc(CCN=C(NC2CCC2)NC2CC2C(F)F)c1 95697,CC1CCC(O)(C(=O)NCC2CC(C(=O)NCc3noc(C(N)=O)n3)=NO2)CC1 95698,C(CC)(C(=O)NCCN(C1CCCC1)C(=O)COCC(C)(C)C)OCC 95699,c1(C(N2CC(NC(C(CC)(CC)CO)=O)C(O)C2)=O)n[nH]c2c1CC(C)(C)CC2 95700,C1(CNC(C2CN(CC)C(=O)C2)=O)CN(C(c2cnc(S)[nH]2)=O)C(C)(C)C1 95701,C1(CCCNC(CC2(OC)CCCC2)=O)CCCCN1C(c1ccccc1O)=O 95702,c1(CC=O)c[nH]c2c(Br)cccc12.N1(C(C)C)CCN(C(C)C(N)=O)CC1 95703,c1(OC)cnc(C(N2CCC3(NC(c4ccnc(C)c4)=O)CC3C2)=O)c(F)c1 95704,C1(C(N2C(C(=O)N(C3CC3)CC3CCOC3)CCC2)=O)C2(CC2)C12CC2 95705,C1(c2nnc(N3CCC(OC)C3)n2CCc2ccccc2)CC2CCCCN2C1 95706,C(CCCCNC(=O)CN(C(=O)C(c1ccn(C)c1)C)CC1CC1)SC 95707,Cc1nc(O)ccc1C(N1CCC(CCNC(=O)CC2(C(F)F)CC2)C1)=O 95708,C1(C(N(CCNC(=O)COCC2CCCCO2)CC2CC2)=O)CCn2nccc2C1 95709,C=CC1COCCN1C(C1(NC(=O)CCC(C)CN(C)C)CCCC1C)=O 95710,N=c1[nH]nc(CCCC(=O)NCCC(O)CNC(C2C=CCC2)=O)s1 95711,c1(C(=O)NCC(CO)NC(C(C(CC)O)C)=O)ccc2sccc2c1 95712,N1(C(CC(=C)C)=O)CCC2C1CCCN2C(c1cc2c(Cl)cncc2o1)=O 95713,N1(C(CC=C)=O)CC2(CCC(CNC(=O)C(c3ccc(F)c(F)c3)(C)C)O2)C1 95714,CCCCCC(=O)NC1CCN(C(=O)C(C)Cc2ccncc2)C1C(C)(C)C 95715,CN1CCC(CO)(NC(C2CCCCN2C(=O)CNc2cncnc2)=O)C1 95716,C1(C(=O)NC(C)CNC(c2cnc(S)n2C2CC2)=O)COC2(CO)CC1C2 95717,c1(C(=O)NCCC2N(C(CSC(C)C)=O)CCC2)ccc(OCC(F)F)cc1 95718,C1(NC(c2ncc(CC)nc2)=O)CCN(C(C2CCOC2)=O)CC1C 95719,C(=O)(C1CCc2ccccc21)N1C(C(=O)NCc2c(C)ocn2)C(C)CC1 95720,C(=O)(CC1OCCc2ccsc21)NC1CCN(C(C2C(=C)CC2)=O)CC1(C)C 95721,Cc1c(C(=O)NCCC2CCCN(C(=O)CC(C)CN(C)C)C2)ccn1CCO 95722,C1(OC)CC(NC(=O)CCOC2CCCCC2)C12CCN(C(=O)C(C)=C(C)C)CC2 95723,CCCC(CC(C)C)C(=O)NC1CC(F)(CNC(c2ccnc(OC)c2)=O)C1 95724,C1(NC(COCC=C)=O)CC2CCC1CC2NC(c1n[nH]c2c1CSCC2)=O 95725,C1(NC(C(C)OC2CCCCC2)=O)CC2CC1CN(C(c1cscc1F)=O)C2 95726,C1(OCC)CCC(C(N2CC(CC(F)(F)F)C2)=O)CC1.C12(CCC1)CC(=O)N2 95727,CC1CC(C(=O)NCCOC2CCN(C(c3ccc(O)nn3)=O)CC2)C1(C)C 95728,CC1=C2CC(CNC(=O)Oc3ccccc3OC3CCC3)CN=C2NN1 95729,C12(NC(C(CCCC)Nc3cccc(Cl)c3)=O)CCC(CC1)N(C(=O)OCC)C2 95730,C1(NC(COCCN(C)C)=O)CCN(C(C2COC3(CCC3)C2)=O)CC(C)(C)C1 95731,C1(C(N(C(CC)C(=O)N2CCC(SC)C2)C)=O)CCCN(C(C)=O)C1 95732,C1(C(=O)NCc2c(COC)nn(C)c2)CCN(C(C)=O)C1(C)C 95733,C1(CNC(=NCC)NC2COC3CC2C3)CCCC2CCCCC12 95734,C1(NC(C=CCOCCOC)=O)CC(O)CN(C(c2cnc(-n3cccn3)s2)=O)C1 95735,C(=O)(C1=NN(C)C(=O)CC1)N1C(C)CN(C(c2ncon2)=O)CC1 95736,c1(C(=O)OC)cc(OC)cc(C(=O)N(CCCNC(C2(C3CC3)CCC2)=O)C)n1 95737,C1(C)(CNC(C2C(C)(CC)C2)=O)CCN(C(=O)CCc2nccn2C)CC1 95738,C12(NC(c3ccc(=N)[nH]c3)=O)COCCC1CN(C(C1(CF)CCOCC1)=O)C2 95739,N1(C(CCN(CC=C)C(c2scnc2C)=O)=O)CCCC(OC(C)C)C1 95740,Nc1ccc(C(=O)NCC2CCN2C(c2cccnc2S)=O)c(F)c1F 95741,C1(CNC(CSCCCC)=O)CC(F)CN1C(=O)COC1CCC1 95742,C(=O)(CCCC(C)(C)NC(c1ncn(C(C)C)n1)=O)Nc1cc(C)sc1 95743,N1(C(C(C#C)(C)C)=O)CC2CCOC2(CNC(=O)C(C)CC(N)=O)C1 95744,C(CCC(=O)N(Cc1ccccc1)OC)N(C(c1cc[n+]([O-])cc1)=O)CC 95745,c1(C(=O)NCCC(C)NC(c2coc(C(F)F)c2)=O)cn2ccnc2s1 95746,N1(C(C(C(C)C)OCC)=O)CCOCC(CNC(C2CC(C)(CC)C2)=O)C1 95747,N1(c2cc3ccsc3cc2)CCCCC(C2CCOCC2)C1 95748,C(C(CC(F)(F)F)NC(C1CCCOC1)=O)NC(=O)CCc1ncc[nH]1 95749,C(=O)(C#CC1(C)COC1)N1CCCC(C)(CNC(CNC(C2C(C)C2)=O)=O)C1 95750,c1(C(=O)NCCC2(O)CN(C(C(C)NC(N)=O)=O)C2)cnc(O)c(C(F)(F)F)c1 95751,C(=O)(C1=NOC(C(N2CCC(NC(=O)CCc3ccc(C)s3)C2C)=O)C1)OC 95752,Cc1cn2c(n1)CC(C(=O)NCC1(F)CCC(NC(=O)C=Cc3ccco3)C1)C2 95753,N1(C(C(C(C)C)c2cnc(C)s2)=O)CCOC(C)(CNC(c2ccncc2)=O)C1 95754,c1(C(=O)NCCNC(C(=O)NC(CC)C)=O)cc(S(=O)(=O)NC)ccc1C 95755,c1(C(=O)NC2CCCC(N(C(c3c(C)snc3)=O)C)C2)cccc(C(F)F)c1Cl 95756,Cc1cc(C(N2CC(CO)C(CO)C2)C(=O)NC2CC(C(=O)OC)C2)ccc1I 95757,c1(C(=O)NCC(CNC(c2cc(C)nc(C)c2)=O)OC)cnn2ccn(C)c12 95758,C1(NC(c2cc(CC)oc2C)=O)CC2CCC1N2C(=O)C(C)C 95759,n1(CC(=O)OCC)cc(CNC(=O)CSCC2CCCCO2)nn1 95760,CCCS(=O)(=O)CC(=O)N1CC(CNC(c2ncsc2C)=O)C(C)C1 95761,CCC(C(=O)N1CC(N(C(=O)Cc2ccc(Cl)nc2C)C)C2(CC2)C1)C(F)(F)F 95762,c1(NC)ncccc1C(=O)NCC(C)CNC(C1CCC=CCC1)=O 95763,N1(C(c2ccn(CCC)n2)=O)CCC2(NC(=O)CCSc3nnnn3C)CC2C1 95764,c1(C(=O)NC(CC=C)CNC(=O)COCCSC)cc(O)nn1C 95765,n1(-c2ccn(C)n2)nc(C2CCOCC2)nc1-c1ccc(OC2CC2(F)F)cc1 95766,c1(C(=O)NCC(CNC(c2n(CC)ncc2)=O)F)ccc(N2CCC(C)C2)cc1 95767,c1(NC(=O)CC2CCN(CCc3ccncc3)C2)cccc(COC2CC2)c1 95768,C1(C(=O)NC2C(CN(C)C)CCC2)CCOCC1NC(=O)CCn1cccn1 95769,Cc1cc(N)ccc1C(=O)NCC1CC2CN(C(c3cccc(Cl)c3F)=O)CC12 95770,C1(C(=O)NC(CC#CC)C)CC2(CCN1C(c1ccn3ccccc13)=O)CC2 95771,c1(C(N(CC(CC)NC(C2CCC2)=O)C)=O)cccc(Cl)c1Cl 95772,C(=O)(C1CCCc2nn[nH]c21)NC1C(NC(=O)COc2cccnc2)CCCC1 95773,Cc1ccc(C)c(C(N2CCC2C(=O)N(C)CC#N)=O)c1 95774,N1(C(CCOCCC)=O)CC(OC)CC1CN(C(=O)Cc1cnc[nH]1)CC 95775,C1(C(N(CCNC(=O)Cc2cncn2C)CC)=O)CCCCC1(C)C 95776,C=CCCCCCCNC(C12CC1CN(C(=O)CCC(=O)CC)C2)=O 95777,N1(C(CCC=CC(C)C)=O)CCCC(C)(C)C1CNC(c1cc(N)ccc1O)=O 95778,C(=O)(CC(C)C=C)NC(C(=O)NCC(=O)OCC#C)CC1CCC1 95779,CCCCC(C(=O)NC(C1CCCC1)CNC(c1ccc(Cl)cc1C)=O)C(C)C 95780,C1(CC(C)OC)CCN(C(=O)CN2CCCC2CN2CCCCC2)CC1 95781,N1(C(Cc2nnc(C)o2)=O)CCC(NC(=O)CCCCN(C)C)C(F)(F)CC1 95782,CC(C)(C)C(CO)C(=O)NCC1CC(C(=O)N2CCC2(C)C)=NO1 95783,c1(OCCC(=O)NC2CCSC2)cccc(N(C)C)c1.C123CC(C1)(C2)C(=O)N3C 95784,N1(C(C2C(CC)CCO2)=O)CCN(C(c2cnc(C)o2)=O)C(CCO)C1 95785,N1(C(C(C(C)(C)C)=O)=O)C2CCC1CC(C(=O)N(CC)CC1CC1c1ccoc1)C2 95786,C1(C(=O)NC2CC(CC(NOCC(=O)N(C)C)=O)C2)CC(=O)CC(=O)N1 95787,C(=O)(C(F)(F)C(F)(F)C(F)F)N1CCN(C(c2cc(OC)c(O)c(Cl)c2)=O)CC1 95788,c1(C(=O)NC23CCN(C(c4cccc(C)n4)=O)CC2C3)cnc2ccnn2c1C 95789,N1(C(c2c(C)nn(C(C)(C)C)c2)=O)CC(NC(=O)CCCCCF)CC(O)C1 95790,C1(C)(C(=O)NC2CC=C(C)CC2)CC(=O)C12CCC2 95791,C1(C(=O)NCCCOC(=O)NC)CCOCC1NC(c1n[nH]c(C)c1O)=O 95792,Cc1noc2nc(C(=O)NCC(CNC(C3CN(C4COC4)C3)=O)CO)ccc12 95793,N1(C(CCN(CC#C)C(C2CC(O)(C#C)C2)=O)=O)CCOC2C(O)CC12 95794,C1(C(N(C)Cc2ncc[nH]2)=O)CN2CCC1CC2 95795,c1(C(N(CCCN(C(C(C2CCC2)OC)=O)C)C)=O)ccccc1C#CC1CC1 95796,C1(C(N2C(C(=O)NC(c3cn(C)nn3)C)C=CC2)=O)C2CCC(F)C12 95797,c1(-c2cccc(C(=O)Nc3ncc(CC)cn3)c2)cc(NC(C)=O)ccc1F 95798,C1(NC(=O)NCCN(C(CC)C)C)CSC(C(F)(F)F)C1 95799,CCCC(C)CC(C(=O)NCC)N(CCN(C)C)Cc1ccc(F)cc1 95800,c1(C(N2CC(C)(NC(C3CC(C)N(C)CC3)=O)C2)=O)ccc2ccncc2c1 95801,C(CCCC(=O)NC(C1CCCN1C(C1CSCCS1)=O)C)SC 95802,Cc1cccc(-c2noc(CCC(=O)Nc3cccc(-n4ccnn4)c3)n2)c1 95803,C1(NC(CC(CC)O)=O)CC(C(=O)N2CCC(n3ccnc3)C2)=CC1O 95804,C1(C(N(C(C)C(N2CCC(N3CC=CC3)C2)=O)CC)=O)CCCSC1C 95805,CCC(C)CCC(=O)NC1C2CC(NC(=O)CCC3CC3C)CC12 95806,CC(F)(C(=O)N1C2CCC1CC(NC(=O)C(=O)NCC(F)(F)F)C2)C(F)(F)F 95807,N1(C(C(CC)C)=O)CC2=C(C1)CN(C(=O)C(=CC1CCCC1)C)C2 95808,C1(CNC(C(C)Oc2ccc(C=O)cc2)=O)CC2(CCC2)C(=O)O1 95809,c1(NC)snc(C)c1C(=O)NCC1(C)CCN(C(=O)Cc2ccoc2)C1 95810,C1(C(COC2CN(C(=O)OC(C)(C)C)C2)=O)C2CCC(=O)C12 95811,C#CC(C)(C1CCCC1)NC(C1(NC(=O)C(C)=C(C)CC)CC1)=O 95812,c1(NC(C2CCCC(C(=O)NC)C2)=O)cc(O)nc(NCC2(CCOC)CC2)n1 95813,c1(C(=O)NCC2(C)CCN(C(C(C3CCC3)OC)=O)C2)ccc(Cl)cc1F 95814,C1(C(=O)OC)(CO)CCN(C(C2CCC(n3cc(-c4c[nH]nc4F)nn3)C2)=O)C1 95815,C1(NC(Cn2c(C)ncc2)=O)CC2CC1N(C(c1csc(C)c1N)=O)C2 95816,C1(CC(=O)NCCC(C)NC(=O)Cn2ccccc2=O)CC2(CC2)CO1 95817,C(=O)(CC(C(F)F)C(C)(C)C)NCC1(OC)CCN(C(=O)Cc2cc(C)[nH]n2)C1 95818,C=CCC(CC(C)C)C(=O)NC1CCC1CNC(=O)CN1CCCOC1=O 95819,N1(C(CC(C)CN(C)C)=O)CC(CNC(c2ccc(CO)cc2)=O)OC(C)(C)C1 95820,CC1(C)CN(C(=O)C(=Cc2c[nH]cn2)F)C(CNC(=O)CCC(N)=O)CO1 95821,C(=O)(CCCc1ccccn1)NCC(C)(C1CCC1)NC(C(C1CC1)OCC)=O 95822,CC1c2ncc(C(=O)NC3C4COCC34)n2CCN1C(c1cnoc1)=O 95823,Cc1cc(C(=O)NC2CCCC2NC(=O)Cc2cnsc2)cn1C(C)C 95824,c1(C(=O)NC(C(=O)N(CCCOCC)C)C(C)(C)C)cn2ccccc2n1 95825,C=C=CC(C)C(=O)NCC1CN(C(=O)C(=Cc2ccncc2)C)CC1C(F)(F)F 95826,N1(C(CN(C)CC)=O)CCC2(NC(c3ncoc3-c3cccs3)=O)CC2C1 95827,c1(C(N2CC3(CCN(C(C4(C#N)C(C)(C)C4)=O)C3)C2)=O)cncc2nc(O)[nH]c12 95828,N1(C(c2scc(CNC(C3C(C)CCO3)=O)c2)=O)CCC(F)(F)C1 95829,C(C(F)(C(=O)NC1CC(OC(C)C)C1)C(C)C)NC(C1CN(CC)C(=O)C1)=O 95830,N1(C(CNS(N)(=O)=O)=O)CCC2CN(C(c3ccc4cncn4c3)=O)C2C1 95831,c1(C(N2CC3CN(C(CCCC)=O)CC3CC2)=O)cc(=O)c2cc(O)ccc2o1 95832,Cc1nc2cc(CC(=O)NCCN(C(=O)CC(C)CC(C)(C)C)C)ccc2o1 95833,CC(=O)CCCCC(=O)N1CCC(NC(=O)C(C)CC(F)(F)F)C1 95834,C12(C(N3C(CNC(CCC4(C)N=N4)=O)CC3)=O)CC(C)(C1)OC2C 95835,N1(C(c2c(OC)csc2)=O)CCC(NC(=O)C(C)P(C)(C)=O)C2(CCC2)C1 95836,Cc1cc2cc(NC(c3cccc([N+](=O)[O-])c3)c3ccccc3C)ccc2[nH]1 95837,C1(CNC(CCc2nnc(C(C)C)o2)=O)CC2(CC2)CN1C(=O)C(F)C1CCC1 95838,C(CCC(C)CC(=O)NC1CCN(C(C2CCN2S(C)(=O)=O)=O)CC1)=C(C)C 95839,C#CC1CCCC(NC(C2CCCC(NC(=O)CCOCCCOC)CC2)=O)C1 95840,c1(OCC)ccc(CC(=O)NCC(O)CN(C)C(C2(C)CNC(=O)C2)=O)cc1 95841,c1(C(N2CC(=C(CNC(c3ccn(CCC)n3)=O)F)C2)=O)ccnc2[nH]ncc12 95842,N1(C(C(C(=O)OC)C)=O)CCN(C(=O)CC2CC(C)(C)C2)C(C2CC2)C1 95843,C1(C(=O)Nc2cncc(SC)c2)CCOCCN1C(C1CCC(N(C)C)C1)=O 95844,N1(C(C2COCCN(C(C(C3CCCCC3)C)=O)C2)=O)CCC2(C=CCO2)CC1 95845,c1(NC(C2CCCN(Cc3ccc(O)cn3)CC2)=O)cnc(Br)c(Br)c1 95846,c1(C(N2CC3C(NC(c4ccc(C(OC)OC)o4)=O)C3C2)=O)cc(C)ccc1C 95847,C1(C(=O)NCC=CCSC)CC12CC(NC(=O)C=Cc1cc[nH]n1)C2 95848,N1(C(C2CCC(C)CC2)=O)CC(NC(=O)CCF)CC(O)C1 95849,S(=O)(=O)(c1ccc(NC(C)C)nc1)NCC(=O)N(CC(C)C#N)CC 95850,c1(C(N2CCC(OCCNC(C(C)SC)=O)C2)=O)c(F)ccc(O)c1F 95851,c1(C(N(CC(C)(C)NC(CC(C)C2CCCC2)=O)C)=O)cc(C2CC2)n(C)n1 95852,c1(C(=O)NCC2N(C(c3c(C#N)scc3)=O)CCC2)cc(O)cnc1Cl 95853,c1(C(=O)NC(CC(C)NC(c2ccn(CC)n2)=O)C)cnn2cc(OC)ccc12 95854,C1(CNC(C=CC(=O)OCC)=O)CN(C(C2CC2C(F)(F)F)=O)CCO1 95855,C1(C(=O)NCC(=C)CCNC(=O)C(C)NS(=O)(=O)CCC)CC2CCC2C1 95856,c1(CC(N)=O)ccc(C(=O)NCC2C3CN(C(=O)CN4CSCC4=O)CC23)cc1 95857,c1(C(=O)NCc2c(C(N(CC(CC)(F)F)C)=O)nco2)cc(C)nc(O)c1 95858,c1(OC)nccc(=NC(=O)C2CN(C(c3c[nH]c4ncccc34)=O)CCC2O)[nH]1 95859,C(CC(C)(C)C)(C(=O)NC1CN(C(=O)CCOCC(F)F)C1)OC 95860,c1(C(=O)NC2(CC=C)CCN(C(C3(Br)CC3)=O)CC2)ccc2scnc2c1 95861,C(=O)(C(C(C)C)C(C)C)NCC(F)(F)F.N12CCC(C1)C(OC)CNCC2=O 95862,c1(C(=O)NCC2C(CNC(=O)CC3CC34CC4)C2)ccc2c(c1)NC(=O)C2 95863,C1(NC(C(CSC)OC)=O)CCN(C(=O)CCc2cnn(C)c2)C1C(C)C 95864,C(C1CCN(C(=O)CCC2CCCCO2)CC1)=CC(N1CC(O)(CCC)C1)=O 95865,C=C(C)CC(C(=O)NCCC1(C)CCCC1)NC(c1cncc(C)n1)=O 95866,N#Cc1ccc(C(N2CCC(NC(=O)CCc3cccc(F)c3F)C2)=O)c(Br)c1 95867,N1(C(C(N2CCC(C)(OC)CC2)=O)C(C)C)CCc2ccccc2C1 95868,c1(NC(c2scc(C(=O)NCCc3ccc(OC)nc3)n2)=O)cncc(C#N)c1 95869,Cc1ccc2cc(C(N3CC(C)C(C)C3)C(=O)NC(C)C)ccc2n1 95870,C(=O)(N1OC2CCC1CC2)C1(C)N(C(c2ccc(CC)cc2)=O)CC(O)C1 95871,c1(CC(N2CCC(O)(C(CNC(C(C)=C(C)C)=O)C)C2)=O)cc(C)cc(F)c1 95872,c1(CC(=O)NCC2CC(NC(C3C4CCC3CC4)=O)CC2O)cc(Cl)ccc1Cl 95873,N1(C(c2c(CC)nc(C)[nH]2)=O)CC2CCC(CNC(=O)CC3CCSC3)(C2)C1 95874,CC1C=C(C(=O)NC2(C(=O)NC3(c4nc[nH]n4)CC3)CCCCC2)C1 95875,N(C(=NCCCCl)NC1CCCCC1)Cc1nnn(C)n1 95876,C1(C)(CC(=O)NC2CC(NC(c3ccc(COC(C)(C)C)s3)=O)C2)COCCO1 95877,N=C1NC(=O)C(CC(N2CCCC2CCNC(c2ccco2)=O)=O)S1 95878,CCC(C)CC(C)C(=O)NCC1(O)CCN(C(c2cccc3ccnn23)=O)CC1 95879,C(=O)(C1c2c[nH]nc2CN1C(c1snc(C)c1N)=O)N(CC#C)CC1CC1 95880,CC1CC(NC(c2cc(Cl)ccc2F)=O)CCN1C(c1csc(C(F)(F)F)c1)=O 95881,C1(CC=C)(C(=O)NCCCOc2cccc(O)c2)CCCN1C(=O)CC1(C)CC1 95882,c1(CNC(C(=O)NC23CCC(CC)(OC2)C3)=O)cc(OC)c(F)c(C)c1 95883,C#CCC(C)(C(=O)N(CCSC)CC)NC(c1ccc(C)c(C)c1)=O 95884,C1(C)(C(=O)NCCC2(O)CN(C(C(C)c3cccs3)=O)C2)CCC(=O)N(C)C1 95885,Cc1cccc(C(N2CC(C(C)NC(c3cccc(Cl)c3)=O)C2)=O)c1N 95886,N1(C(c2cc(CC)no2)=O)CCCC2C(CCCN2C(=O)Cc2nnc(C)s2)C1 95887,C1(C(N(CC(C)(C)O)CC)=O)COCCC1NC(=O)CCCOC(C)(C)C 95888,N1(C(C(C2CCOCC2)OCC)=O)CCCC(NC(=O)C(C)OCCOC)CC1 95889,c1(C(=O)NCCC2CCN(C(=O)Cc3ccoc3)C2)cnc(-n2cccn2)cn1 95890,C1(CNC(C(C(C)C)C)=O)C2CCC(C2)N1C(=O)CN(C)Cc1ccccc1 95891,C=C(Cl)C(C)(C)C(=O)NCC1(F)CC(CNC(C2OCC2(C)C)=O)C1 95892,c1(C(CNC(C2CC(OC)C2)=O)NC(=O)CCOC)ccc(F)cc1 95893,C#CCC(C)(C)C(=O)NCC1(O)CC(CNC(=O)C=Cc2ccc(O)cc2)C1 95894,Fc1cc(-n2nc(-c3ccc(Br)cn3)nc2-c2cnn(C3CC3)c2)ccn1 95895,C1(COC)CN(C(C2(NC(c3coc(C)n3)=O)CC2(C)C)=O)CCO1 95896,Cc1nn(C(C)(C)C)cc1C(=O)NC1CCC(C)(CNC(=O)CC(F)(F)F)C1 95897,Cc1cc(=NC(=O)CNC(CSCC23CCCN(C(=O)CC4CC4)C2C3)=O)[nH]o1 95898,c1(C(N(C2CCCC(NC(C(C=C)(F)F)=O)C2)C)=O)ccc2ccc(Cl)cc2n1 95899,C(=O)(C1=CC2C=CC1C2)NC1C2CC(C(=O)NCCC(C(=O)OC)C)C(C2)C1 95900,c1(C(N2CCC(N(C(=O)CN3CCNC3=O)CCC)C2)=O)oc(COC)nc1C 95901,c1(C(N2C3C(NC(CN(C4CCSC4)C)=O)C(C3)C2)=O)sc2ncccc2c1N 95902,CC1(C(=O)NCC#CCNC(=O)Cc2cccc(C(N)=O)c2)CC2CCC1C2 95903,C1(N(C(C(CC)CN(C)C)=O)C)CN(C(=O)CC2CC2)CCC1C 95904,C(C)(C)(CC(F)C(=O)NCC(=O)N(C)C)NC(CN(C(C(C)C)=O)C)=O 95905,n1(CC(=O)NCCC(C)NC(CC2CC(=C)C2)=O)c(=O)nc(O)c2ccccc12 95906,C1(CNC(C2(C)CCN(C(CSCC(C)C)=O)C2)=O)CCC2(CCC2)O1 95907,Cc1ccnc(O)c1C(=O)NC1CCCCCC1NC(=O)Cc1sc(O)nc1O 95908,C1(NC(c2sccc2I)=O)CN(C(c2c[nH]nc2F)=O)CC1O 95909,C1(NC(C2ON=C(CC)C2)=O)CCCCCC1C(N1CC(C(=O)NC)(SC)C1)=O 95910,C(=O)(C(C(C)(C)C)C1CCCCC1)NCCN(C(C1(C)CCN(C)C1)=O)C 95911,c1(C(=O)NC2CCC(NC(C3CC4(CCC4)CO3)=O)CC2)ccn2ccccc12 95912,CC1(C)CC(C)(C(N2CC3CC3(CO)C2)=O)CN1C(=O)CS(C)(=O)=O 95913,CC(CC(=O)NC(CNC(=O)CN1CC2CC2C1)CO)NC(C1CCCC1)=O 95914,C1(C(C)NC(=O)C(C)(C)c2ncco2)CCCN(C(=O)CCCCNC(N)=O)C1 95915,C(=O)(CCCC(F)(F)Br)N(C1CCN(C(C2CC(C)(C)CO2)=O)C1)C 95916,N1(C(C(CC2CC2)OC)=O)CC2CCC1CN2C(c1ccc(C)s1)=O 95917,N1(C(COC(C)=O)=O)CCN(C)C(C(=O)NC(c2cccnc2C)C)C1 95918,C1(C(=O)NCC2CC(NC(C3(C#N)CC(C)C3)=O)C2)CCOC(C)(C)C1 95919,N1(C(C(C)=NOCC#N)=O)CCN(C(c2n[nH]c3ccccc23)=O)CC(O)C1 95920,CCCCCCC(O)CCC(=O)NCC1(OC)CN(C(=O)C=CS(=O)(=O)CC)C1 95921,CC1CC(C(=O)NCC2CC(n3cnnc3)C2)N(C(=O)OC(C)(C)C)C1 95922,C(Cn1cc(CNC2CCC2)nn1)(CC(C)C)NC(C1C(C=C)C1)=O 95923,N1(C(C2CC(=C)C2)=O)CC(NC(=O)CCOCC(F)(F)C(F)(F)F)CC(O)C1 95924,CC1CN2CCN1C(C(N1CCC(C)(NC(c3nccn4nccc34)=O)C1)=O)C2 95925,N1(C(=O)Nc2ncnc(O)c2Br)CCC2(C(=O)O)C(C1)C2(F)F 95926,c1(C(C(=O)NC2(C)CC2)N(CCC#C)C2CC2)ccc([N+](=O)[O-])c(O)c1 95927,N1(C(C2(CC)CC2)=O)CC2CCC(NC(=O)CCc3c(C)noc3Cl)CC2C1 95928,C=C(C)c1cccc(NC(C2C=CCCN2C(C2CCC(=O)N(C)C2)=O)=O)c1 95929,C(C(C)(O)C(F)(F)F)NC(=O)Nc1ccc(NC(=O)OC(C)(C)C)nc1 95930,C1(NC(C(C)N=CC=C(Cl)Cl)=O)COCCN(C(C2(Nc3ccccc3)CC2)=O)C1 95931,CC1(C)OCCCC1CNC(=O)CC1CCN(C(c2cccc(CO)c2)=O)CC1 95932,N1(C(C)=O)CCC(N(C(=O)CC2(N(C(=O)C(C)n3cncn3)C)CC2)C)C1 95933,c1(CCCC(=O)NCC(CNC(CN(C2CCC2)C)=O)F)csc2ccccc12 95934,C1(C(C(=O)NCC(CCC)C)C)CCCN(C(=O)CCCn2cccn2)C1 95935,CC1CN(C(=O)CN(C)C(N)=O)CC(CCNC(=O)C(c2ccccc2F)O)O1 95936,c1(C(N2CC(N3CCN(C(C(CCSC)O)=O)CC3)C2)=O)cc2n(n1)CCO2 95937,c1(CCCC(=O)NC2C=CCN(C(CSCC(=O)OC)=O)C2)ccc(C)c(C)c1 95938,Cn1cc(C(N2CCC(C)(CC(=O)Nc3cc(CO)cc(F)c3)C2)=O)n(C)c1=O 95939,N1(C(C2(F)C(C)OCC2)=O)CCCC2(CCN(C(=O)CC3CCC=CCC3)C2)C1 95940,c1(C(=O)NCCCCNC(C2COC(=O)O2)=O)ccc2cncnc2c1 95941,c1(C(=O)NCC(C)NC(=O)C2=CCSC2)c[nH]c2cccc(C#N)c12 95942,N1(C(c2cc(C(F)(F)F)ccc2I)=O)CCC2(CCN(Cc3cccnn3)C2)C1 95943,N1(C(c2ccc(C(=O)OCC)cc2)=O)CCN(C(=O)C(C)C(C)(C)C)CC(O)C1 95944,C1(C(=O)NCC(c2ccc(F)cc2)NC(=O)C(F)C2CCC2)CCCCS1(=O)=O 95945,c1(C(C)(C)CNC(=O)OCc2nc[nH]n2)ccc(F)cn1 95946,C(=O)(C(CC(F)F)C1CCC1)NCCN(C(C1(C)ON=C(C)C1)=O)C 95947,CC(C)(C(=O)NCC(CO)NC(C1CCOC1)=O)C1CCC1 95948,C1(NC(C2(C(=O)OC)CC23CCC3)=O)C2CC3CC1CC(O)(C3)C2 95949,CNS(=O)(=O)N1CCC(C(=O)NCCNC(C2CN3CCCN2CC3)=O)CC1 95950,C1(c2ccccc2)(NC(C2C(C=C)C2)=O)CCN(C(=O)C=Cc2nccs2)C1 95951,CC1CCC(Cl)=C(C(=O)N2CCCCC2CNC(=O)CC2CCCOC2)C1 95952,N1(C(c2c(C)csc2)=O)CC2CC(C1)CN(C(C1CC(C)(C)C(C)(C)C1)=O)C2 95953,c1(C(N2CCOCC(NC(C(COC)(F)F)=O)C2)=O)cc2ccc(F)cc2cn1 95954,c1(C(=O)Nc2ccc(C(=O)NC3CCCCC3)cn2)ccc(F)c2ccsc12 95955,C1(N(C(c2cc(C(C)C)no2)=O)C)CCCC(NC(C2(CCN(C)C)CC2)=O)C1 95956,c1(CC(=O)NC(CC)(C)CNC(C2CNC(=O)C2)=O)nc2ncccn2n1 95957,Cc1cccc(F)c1C(=O)NCC1CN(C(C2CC(=O)NC(=O)C2)=O)C1 95958,N=c1cc[nH]cc1CNCC1CCN(c2ccc(-c3cn[nH]c3)cc2)CC1 95959,C1(CNC(Cc2cccc(OCC)c2)=O)CN(C(c2scnc2C)=O)CC12CC2 95960,CN(CCCC(=O)N1CCC(c2n[nH]cc2CNC(=O)C(O)C(F)(F)F)C1)N=O 95961,c1(CC)cccc(C(=O)NC2CN(C(=O)CC3CCCN3C)C(C)(C)C2)c1O 95962,O=C1CCC(C(=O)N2CC3(NC(C4CCCCS4(=O)=O)=O)CCC2CC3)=NN1 95963,Cc1onc(C(N2CCCC(NC(c3cc(Br)no3)=O)C2)=O)c1[N+](=O)[O-] 95964,c1(C(C)(C)C)ccnc(C(=O)NC2CC(NC(C3(n4cccn4)CCC3)=O)C2)c1 95965,c1(N(C)CC23CCC(CC2)C3)nc2cccnc2c(=NC2CCCS(=O)(=O)C2)[nH]1 95966,N1(C(C(CC#C)(C)C)=O)CC(CNC(=O)C(C)n2cccn2)C2(CCOCC2)C1 95967,C1(OCC)(CC2CCN(C(c3cccnc3OC)=O)C2)CCCCC1.C1(=O)CN1 95968,C12(C(N(C)Cc3ccnn3C)=O)CCCC1CN(C(C1(C#N)CCCCC1)=O)C2 95969,c1(CSC)cccc(-c2nnc(N(CCCC(C)C)C)n2CC2CCCCO2)c1 95970,N1(C(C(CC(C)C)ONC(C2CCOCC2(C)C)=O)=O)CCc2c(nnn2C)C1 95971,c1(C(=O)Oc2cccc(CN=c3nnn(C)[nH]3)c2)oc2ccccc2c1CO 95972,C1(C(N2CC3C(NC(C(C)N(C(C)=O)C)=O)C3C2)=O)CCC([N+](=O)[O-])CC1 95973,c1(CNC(=O)CCc2ncc[nH]2)ccc(CNC(c2cc(Cl)ns2)=O)cc1 95974,C(CC(=O)N1CC2CCC(C1)N2C(=O)C=Cc1ncc[nH]1)(C(F)(F)F)OC 95975,C1(C(=O)NC(C(=O)NC)CC2CC2)CCC(C2CC2)N1C(C1CC(F)CN1C)=O 95976,N1(C(c2cnc(COC)s2)=O)CC2(CCC2NC(=O)C(C)=C(C)C)C1 95977,c1(CC(=O)NCC(C)(C)NC(C2C(C)C2)=O)ccc(O)c(Cl)c1 95978,N1(C(C2(C)COC2)=O)CCCC2(CCCCC2NC(C2CC3CC3C2)=O)C1 95979,Cc1cc(C(=O)N(C2CC(C#N)C2)CC(N2CCC(CCO)CC2)=O)cc(C)n1 95980,N1(C(C(C)NC(COC)=O)=O)CC2C(NC(=O)CCN3CCC(O)CC3)C2C1 95981,N1(C(CCC(C)(C)NC(CCCOCCOC)=O)=O)CC2CCCCCC2C1 95982,CN1C(=O)Cc2c(C(N3CC(O)(c4ccsc4)C3)=O)cccc21 95983,C(=O)(CC(C)(C)C)N(CCC)CCNC(C1CCC(OC(F)(F)F)C1)=O 95984,CC(C)(C)CC(O)C(=O)N1CC=CC1CNC(c1ncc2[nH]ncc2n1)=O 95985,N1(C(C2(C3CCCO3)CC2)=O)CCCCC1C(=O)N(C)CC1(CC)CC1 95986,C(CC(C(=O)N(CC(N1CCCC(N(C)C)C1)=O)CC(C)C)OC)OC 95987,c1(C(N(C2(C(N3CCCC(C)(C)C3)=O)CCOCC2)C)=O)ccc2[nH]ccc2c1 95988,CCC(CC(F)(F)F)C(=O)N(CCC(C)NC(c1cnc(Cl)s1)=O)C 95989,c1(C(N2C3(CNC(CC4(C)CC4(Cl)Cl)=O)CC(C2)C3)=O)cccc2c[nH]nc12 95990,N1(C(c2c(COC)ccs2)=O)CCN(C(=O)C=Cc2cscn2)C(CC(F)F)C1 95991,c1(C(N2CCC(C(C)(C)NC(CS(=O)(=O)NC)=O)C2)=O)cc(C)ccc1N 95992,Cc1nc(NC2CC2)sc1C(=O)NC(C)CN(C)C(C1CC2CC2C1)=O 95993,C(CC(C)(C)C)(C(=O)NOCc1ccc(F)cc1)NC(CC=C(C)C)=O 95994,c1(-c2ccc(C)cc2)ccc2c(c1)C(C(=O)O)OCC2 95995,c1(CC)cc(NC(=O)C=CC(C)NC(c2cc(F)n(C)n2)=O)ccc1C 95996,c1(C(=O)NC2C(C)CN(C(=O)CCCN(C)N=O)C2)noc2c1CC(C)(C)CC2 95997,C#CCC(C)(C)C(=O)NC1CC(N(C(=O)CCC=CC(C)C)C)C1 95998,c1(OC)cnnc(C(=O)NC2CCC(N3CCN(C(c4cncs4)=O)CC3)C2)c1 95999,O=C(CN1C(=O)Cc2ccccc21)NC1C2CCCN(C(=O)CSC)C2C1(C)C 96000,C1(C(=O)NCCN(C(c2ccn(C)n2)=O)CC)CCN(S(=O)(=O)NC)CC1 96001,CC(CC(N)=O)C(=O)N1CCCC(C(CC2CC2)N=c2[nH]ncs2)C1 96002,C1(CNC(C2CC(F)(CO)C2)=O)C2CN(C(=O)CSc3ccc(F)cc3)CC12 96003,C(=O)(NNc1cc(Cl)cc(Cl)c1)Nc1ccc(-c2ccc(C)cc2)cn1 96004,n1(CCCOC)nc(-c2ccc(N)cn2)nc1-c1cc(C(F)(F)F)no1 96005,C1(C2C(OCCC(=O)NC3CC3)C2)CCCN(C(c2cncc(C3CC3)c2)=O)C1 96006,N1(C(C=NOC)=O)CCCC(C)C1CNC(=O)CCc1ccccc1O 96007,C1(NC(CC(C)F)=O)CN(C(=O)CCNC(c2ccccc2)=O)C2(CCCC2)C1 96008,C(CCC(O)CO)NC(C1CC(CNC(C2(CO)CCCO2)=O)OC1)=O 96009,C1(NC(c2cc(OC)c(Cl)cc2)=O)CCC2CN(C(c3nncn3C)C)CC2C1 96010,c1(C(=O)NC2CCC(C)(CNC(c3c(C)nn(C)c3)=O)C2)cccc([N+](=O)[O-])c1 96011,c1(SC)ccc(Cl)c(C(N2CCN(Cc3cn(CCF)nn3)CC2)=O)c1 96012,CC(C)C(C)CC(=O)N1CC(O)CC1CNC(=O)COc1ccon1 96013,N1(C(CC2CCCC(C)(C)O2)=O)CCN(C(=O)CC(F)(F)F)CC12CCC2 96014,N1(CC(=O)Nc2cccc(C(C)C)c2)CC2CN(S(=O)(=O)C(F)(F)F)CC12 96015,C1(NC(C2CC(CC)(CC)C2)=O)C=CCN(C(=O)C(N2CCOCC2)C)C1 96016,c1(C(N2C(CC(=O)Nc3c(OC)cccc3)CCC2)=O)ccc(S(C)(=O)=O)c(F)c1 96017,Cc1c(C(N)=O)cccc1C(=O)N(C)CC1(NC(c2ccc(C(N)=O)o2)=O)CC1 96018,N1(C(C(C)(C)OC(C)C)=O)CCCC(N(CCF)C(c2coc(Br)c2)=O)C1 96019,C(C)(CNC(c1ccc(-c2cccs2)o1)=O)(CO)NC(C=C(CCC)C)=O 96020,c1(OC)ccc(C(=O)NCC2(C)CN(C(c3cccc(Cl)c3)=O)C2)c(Br)n1 96021,c1(C(c2nnnn2CC2CC2)NC2(CCCC)CC2)ccc(-c2csc(C)n2)s1 96022,c1(C(=O)NCCn2cc(C(=O)NC(COC)C3CCC3)nn2)cncc(C)n1 96023,c1(NC(C(C)=C2CC2)=O)cccc(CNC(c2ccoc2Br)=O)c1 96024,c1(OC)c(F)c(CNc2ncnc(NC(C)CF)c2C)cc(F)c1F 96025,C1(CC(=O)NC2CC(OCC(C(=O)CCc3ccoc3)=O)C2)CC1(Cl)Cl 96026,N1(C(C=CCNC(c2c(NC)cccc2)=O)=O)CCOCC(C(=O)O)C1 96027,C1(CC(=O)N(C2CCCN(C(CN(C(=O)OCC)C)=O)C2)C)CCC(C)(C)CO1 96028,C(=O)(CC(C)(C)CC(F)F)NC1CC(C)N(C(C2CCN2C2CCCC2)=O)C1 96029,Cc1cccc(CC(=O)NCCOCCN(C)C(c2cncnc2)=O)c1 96030,C1(C#N)(C(=O)NCC2CC(OC)CN2C(C2CCC2(C)C)=O)CCOCC1 96031,C1(C(=O)NCCSCCC=C)CCC(O)CN1C(c1cccc(NC)n1)=O 96032,C12(NC(CN(CCC)C)=O)CC(CNC(=O)CCC(C)(C)OC)(C1)OC21CCC1 96033,c1(C(N(C(CCC)C)C)=O)ccn(CCNC(=O)CC2(C)CCCO2)c1 96034,N#Cc1cc(Br)ccc1CN1CC2CN(c3ncc(C4CC4)cn3)CC2C1 96035,N1(C(C2(C)C(C)C2)=O)CCOCC(CNC(c2ccc(Cl)c(Cl)c2)=O)C1 96036,n1(CC(C)C)ccc(N(CC(C)Cl)C)n1 96037,N1(CC(=O)NCC(CC)NC(=O)C(C2CC2)N(C)C)C(=O)NC2(CCCC2)C1=O 96038,N1(C(CCCC(=O)NCC)=O)CC2C3CCC(C2C1)N(C(c1cn(C)nn1)=O)C3 96039,C(C(=O)N=c1ccn(C(C)C)[nH]1)(c1cccs1)NC(c1c(C)cns1)=O 96040,c1(-c2cccc(C3C(=O)CCC3)c2)ccc2nccn2n1 96041,CN=c1[nH]c(=NCCCN2CCN(C)CC2)[nH]c(=NC2CCSCC2)[nH]1 96042,C#CC(C(C)(C)C)NC(=O)COCCNC(c1cccc(CC)n1)=O 96043,C(=O)(C(C)Cc1cnc[nH]1)N(CC(C)NC(=O)COCCCOC)CC 96044,C(CC1C(=O)Nc2ccccc21)NC(=NCCCC)NC(C)CCC(C)C 96045,C1(NC(C2(NC(C)C)CC2)=O)COC2(C1)CN(C(=O)C(N1CCCCC1)C)C2 96046,C1(CNC(C2C(C)CCO2)=O)CN(C(=O)CCc2ccc[nH]2)CC(C)(C)O1 96047,C(=O)(C(C)S(=O)(=O)CCC)N1CCCC(N2CCN(C(CCC)=O)CC2)C1 96048,c1(N2C3C(CNC(C4(C)CC4Br)=O)C(CCC3)C2)nc(O)c2ccc(Cl)cc2n1 96049,c1(OC(C)C)cnccc1C(N1CCC(CNC(C2(CO)CCCCC2)=O)C1)=O 96050,c1(C(C(C)NC(=O)CCc2cnc[nH]2)NC(=O)CSc2nncs2)ccccc1 96051,C1(CNC(CCC(CC)C)=O)CC2(CO1)CN(C(=O)CC1CCCCC1)C2 96052,N1(C(C(COC)Cl)=O)CC(NC(=O)Cc2cc(Br)cs2)C2(COC2)C1 96053,C=CCN(OC)C(=O)C(C)N(C(=O)CCC(CC)N(C)C)C1CC1 96054,c1(-c2n(CCC=C)c(N(C)CCc3ccc(Cl)cc3)nn2)cnc(OC)c(F)c1 96055,C(=O)(C#Cc1ccccc1)NC1CCCN(Cc2c(C)c[nH]n2)CC1 96056,C1(N(C(C2N(C(c3cccc(C)c3)=O)CCC2)=O)CCO)CC2CC1CC2CO 96057,CCN=c1ccc(C(=O)NCC(C)(C(C)C)NC(C2CC(S(C)(=O)=O)C2)=O)c[nH]1 96058,C#CCCCCC(=O)NCC12CC(NC(C3CCCC3(F)F)=O)(C1)C2 96059,C1(C2CCOC2)(C(N(CCN(C(C(C2CC2)OC)=O)C)C)=O)CCOCC1 96060,c1(C(=O)NC2CCN(CCCNC(C(C=C)OC)=O)C2)cc(O)cc(=O)o1 96061,C(=O)(CC(CCCC)NC(C1CC=C(C)CC1)=O)NC(CC#C)(C)C 96062,c1(C2(C(=O)NC(C3CN(C(C4(F)CCOC4C)=O)CCO3)C)CC2)ccc(F)cc1 96063,CC1CCN(C(C2OCC2(C)C)=O)CCN1C(C1CCCC(=O)CC1)=O 96064,N1(C(C2(C(F)F)CCCC2)=O)CC(Nc2ncnc3scnc23)CC2(CCC2)C1 96065,C(=O)(CCC(=O)NN(C)C)N1C(CNC(c2nc(OC)nc(O)c2)=O)CC2CC21 96066,CC(=O)CCCC(=O)N1CCCC1CNC(=O)C(c1cccc(Br)c1)(C)C 96067,C1(C(N2CC(CNC(=O)CCCCCO)C(C(F)(F)F)C2)=O)Cc2ccncc2C1 96068,Cc1nc2c(s1)CCCC2CNC(c1nc(Br)n2c1CCNCC2)=O 96069,c1(C(N2CCCC(CNC(c3cncs3)=O)CC2)=O)c(F)ccc2c1OCO2 96070,N1(C(C(c2ccc(Cl)cc2)N(C)C)=O)CCC2C(NC(c3ccccc3F)=O)C12 96071,c1(C(=O)NCCC(C)NC(c2ccc(CC)o2)=O)c(Cl)ccc(Br)c1N 96072,C1(C(=O)NCC(C)(CNC(c2ncc(C)cc2F)=O)OC)CC(=O)CC(=O)N1 96073,c1(C(=O)OC)ccc(C(=O)NC(CNC(c2ccn(CCOC)n2)=O)CO)s1 96074,N1(C(C2(NC(c3c(C)c[nH]c3)=O)CC(CO)C2)=O)CCN(C(C)(C)C)CC1 96075,C1(O)(C(C)NC(=O)CC2CCOC2)CCN(C(C2COC3COCC23)=O)CC1 96076,c1(C(=O)NC2(CCOC)CCN(C(CC(=C)C)=O)C2)cn2cnnc2cn1 96077,C1(C(N(OC)C)=O)CC(O)CN1C(C)=O.C(C)(C)C 96078,CC(C(C)(C)CO)NC(c1n[nH]c(CO)n1)C 96079,N1(C(C(C)CC(N)=O)=O)C2CCC1CC(N(C)C(c1cccc(C(N)=O)c1)=O)C2 96080,c1(-n2cc(-c3ccc(NC(C)CC(=O)O)cc3)nn2)ccc2c(c1)C(=O)OC2 96081,N1(C(C(CC)O)=O)CCN(C(=O)CCN2CCCS2(=O)=O)C(CC(=O)NC)C1 96082,C1(NC(CCC2(C)CN(C(c3cc(COC)no3)=O)C2)=O)CCSC(C)C1 96083,N1(C(=O)Cn2cc(C(F)(F)F)cn2)CCC2CN(C(=O)CC3CC3)CC2C1 96084,C1(C(C)Cc2cc[nH]c2)CCN(NC(c2cc(C(C)(C)C)n[nH]2)=O)CCC1(F)F 96085,c1(CNC(c2cccc(NC(c3cc(CC)n(C)n3)=O)c2)=O)nc(Cl)ccc1F 96086,c1(OCc2ccc(C(=O)NC)o2)ccc(OC)cc1.C1(C)(C)CC(=O)OCCO1 96087,c1(C(=O)NCCN(C)C(C2CCCC2)=O)cc(-c2ccoc2)on1 96088,Cc1cnc(C(=O)NC2CN(C(c3c(O)cccc3F)=O)CC2CO)c(C)c1 96089,c1(C(=O)NC(C(CO)NC(CN(CC)CC)=O)C)ccc(F)cn1 96090,CC(C)C(C(C)NC(c1cscc1Br)=O)NC(c1ccc(CO)o1)=O 96091,C=CCCC(C)NC(=O)C(C)CN(C)C(c1csnc1OC)=O 96092,c1(NC)ccc(Cl)c(C(=O)NCC(C(C)(C)C)NC(=O)C=Cc2ccoc2)c1 96093,C1(NC(C2CC(=O)NC2)=O)CN(C(c2cnc(Cl)c(Cl)c2)=O)CCC1(F)F 96094,CCCS(=O)(=O)CC(=O)N1CCC(NC(=O)CCC(F)F)C1 96095,C1(CC(=O)NCCCC2CCC2)C2CCC(C2)N1C(C1CCOC1)=O 96096,C1(N(C)C(C2CCCS2)=O)CCCC2CN(C(=O)CC3CCS(=O)(=O)CC3)CC12 96097,C=CCC(CC(=O)Nc1cccc(C#N)n1)NC(=O)NCc1ccccc1 96098,N#Cc1cc(NC(C2COCCN2C(C2CC2C2CC2)=O)=O)cc(Cl)c1 96099,C=CCC(C)(C)CC(=O)NCC(CC)(CC)NC(=O)CCC(C)C#N 96100,c1(OC)cc(OC)c(C(N2CC(NC(=O)C(C)O)CC3(CC3)C2)=O)c(N)c1 96101,c1(C(=O)NC2C(C)CCN(C(=O)CCOC3COC3)C2)cc2cccc(Cl)c2[nH]1 96102,c1(C(N(CC(C)O)CCNC(=O)Cc2cc(C3CC3)no2)=O)cnc2c[nH]nc2c1 96103,N1(Cc2c(C)n[nH]c2C)CC2(CN(C(=O)COc3ccccc3)CCO2)C1 96104,C1(CC)(CO)CCN(C(=O)C(CO)NC(c2cc(Cl)no2)=O)C1 96105,C1(CC#C)(C(=O)NC(C)CC(C)NC(C2(O)CC2)=O)CCCC1 96106,Cc1cc(CCNC(C2(c3cn(CCC(F)(F)CO)nn3)CCC2)=O)ccc1Cl 96107,c1(OC)ccc2[nH]nc(C(=O)NC(C)CNC(c3c(F)cc(C)cc3F)=O)c2c1 96108,C=Cc1cccc(CN2CCN(CC(N3CCC(C)CC3)=O)CC2)c1 96109,CC1CN(C(c2cccn3ncnc23)=O)C(C)CN1C(c1ccc(O)nc1Cl)=O 96110,CCCC(CCC)CC(=O)NCC1(F)CC(CNC(=O)CC(CC)OC)C1 96111,C(CO)(CCCCNC(C1(CC(F)F)CCC1)=O)NC(=O)COc1ccccc1 96112,c1(C(N2C3CC(C(N4CC(C)OCC4)=O)C2CC3)=O)cccc2nc[nH]c12 96113,C(=O)(C(C)CS(C)=O)N(CCNC(c1cc(-c2cccc(C)c2)no1)=O)C1CC1 96114,c1(C(=O)NCC#CCNC(c2nncc(OC)c2)=O)cc2ccc(Cl)c(F)c2o1 96115,c1(C(N(C)CC2C3CN(C(COC)=O)CC32)=O)ccc2ncccc2c1F 96116,c1(C(NC(=S)NNC(=Nn2ccc3cc(Cl)ccc23)N)C)cc(S(C)(=O)=O)ccc1F 96117,C12COCCC1CC(=O)N2.CS(=O)(=O)SC1CC1c1ccco1 96118,C1(NC(C(CCC)O)=O)CCCN(C(=O)CCc2ccc(F)nc2)CC1 96119,C1(CC(=O)NCC(CNC(C=CC2C(C)C2(Cl)Cl)=O)O)C2CC3CC(C2)CC1C3 96120,C(CC(=O)NC1CCn2ccnc2C1)(C(C)(C)C)NC(C=Cc1n(C)ncc1)=O 96121,c1(-c2c(C)occ2)nc(CC2CCC(O)C2)n(C2CS(=O)(=O)C2)n1 96122,c1(C(=O)NC(CC=CC)C(=O)NCC=CC2CC2)cnc2ccccn12 96123,C(=O)(C1=CCOCC1)NCC1(C)CCN(C(=O)CC2C=CCCC2)C1 96124,N1(C(C(=Cc2ccco2)C)=O)CC2CCC(C1CO)N2C(=O)C(C)N1CCC1 96125,CC1COCC(C(N2CCC(C(=O)NCC(C)(O)C(F)F)C2)=O)O1 96126,c1(NC(CC)CNc2ccccc2)nccc(=NC(C)c2cccnc2)[nH]1 96127,c1(N(C)C)ccc(C(N2CC(NC(C3CC3(F)F)=O)C3CC3C2)=O)cc1[N+](=O)[O-] 96128,c1(CCC(=O)NC2CC3CCC2N3C(c2ccnnc2)=O)ccc(O)c(F)c1 96129,CC(C)C(C(=O)NC1(C(N)=O)CC1)n1cc(C(C)(C)O)nn1 96130,C1(NC(CCc2cc(C)sc2C)=O)CCCCN(C(C2(CF)CCC2)=O)C1 96131,c1(C(N2CCC(CCCc3cn(CC)nn3)CC2)=O)ccc(C)cc1C(C)C 96132,N1(C(C2CCN(C(c3cscc3Br)=O)C2)=O)CCC(O)(CO)CC1 96133,CCC(CN(C)C)CC(=O)NC1CC(CNC(=O)C(=O)Nc2ccccc2)C1 96134,c1(C(=O)NCc2cccc3c2CCN3)ccc2c(F)cc(F)cc2n1 96135,C(=O)(CC(C)P(C)(C)=O)NCC(C(C)(C)C)NC(c1scc(OC)c1)=O 96136,C1(C(=O)NC(CCNC(=O)CNC(=O)NC2CC2)c2cccs2)(SC)CC(F)C1 96137,C1(C(N2CCN(c3nnc(SC(C)C)n3C)CC2)=O)CCC(C2CCCO2)O1 96138,N1(C(C(CC=C)C)=O)Cc2ccccc2CC1CNC(c1c(C)ncn1C)=O 96139,c1(C(=O)NCCC2CCN(C(CS(CC)=O)=O)C2)cc(F)cc(C)c1C 96140,C12CN(C(=O)OC(C)(C)C)CCC1C2.c1(NC2C(OC)C2)cnc(C)s1 96141,N1(C(c2n[nH]c(C)c2O)=O)CC(=O)NCC1C(=O)NC1CCOC1(C)C 96142,C1(CCNC(=O)C=CC2CC2)CN(C(c2ccc(N3CCCC3)nc2)=O)CCO1 96143,CC(C)(C#N)CC(=O)NCC1CCN(C(=O)CCOCC2CC2)CC1O 96144,C(=O)(CC(C)c1ccco1)NCCN(C1CCCCC1)C(CSCC#C)=O 96145,Cc1sc(Cl)c(C(=O)N2C3CC(C3)NC(=O)C2)c1C.C(C)(CCCC(C)C)N.CC 96146,C(=O)(C(C(C)C)C(C)C)N1CC2C(CN(C(COCc3cc(C)on3)=O)C)C2C1 96147,C1(C(N(CCCCC2CC2)C)=O)CCCN1C(=O)C(=O)NC1CCCCO1 96148,N1(C(COCC(=O)NC)=O)CCCC(NC(c2cc(N)cc(F)c2)=O)CC1 96149,C1(NC(c2c(SCC)cccn2)=O)CC2CC1CN(C(=O)CC1CC3CC3C1)C2 96150,C1(CCCNC(c2scc(C)c2)=O)CN(C(c2sccc2C#N)=O)CCO1 96151,c1(C(=O)NC2C(CNC(c3c(OC)nn(C)c3)=O)C2)cccc2c1OCCC2 96152,c1(OC(C(=O)NCC=CCNC(CCC)=O)(C)C)ccc([N+](=O)[O-])cc1 96153,c1(CCN(C(c2c(C)cc(CC)o2)=O)Cc2cccnc2)ccc(Cl)c(Cl)c1 96154,C1(NC(C(C)c2cccs2)=O)CCN(C(c2c[nH]c(C(F)(F)F)c2)=O)CC1F 96155,c1(C(=O)NCCC2OCCN(C(CC(=C)C)=O)C2)ccc(O)cc1[N+](=O)[O-] 96156,C1(CCC(=O)NC(C2(C(N(CCCOC)C)=O)CC2)C)CCC(=O)C1 96157,c1(C(=O)NCCC2(NC(COC(CC)(C)C)=O)CC2)cc2ccc(OC)nc2[nH]1 96158,N1(C(C(c2ccc(C)cc2)C)=O)CCC(F)(F)C(NC(=O)C(F)F)C1 96159,C1(NC(C2(CC#C)CCCCC2)=O)COC2(C1)CN(C(=O)C(C)N1CC(C)C1)C2 96160,N1(C(CN(C)C)=O)CCC(N=c2ccc3nnc(-c4cccc(Br)c4)n3[nH]2)CC1 96161,N1(C(COCCC#C)=O)CC(CNC(=O)C(CCC)N(C)CC)C(C)C1 96162,C1(C)(C(=O)NC2(CCCC(=O)NCC(c3ccsc3)C)CCC2)CC(=O)N(C)C1 96163,C1(C(N(CC(O)CNC(c2coc(CO)c2)=O)C)=O)CC12CC(C)(C)C2 96164,N1(C(C2(CNC(c3c(C)snn3)=O)CC3(CC3)C2)=O)CC2CCC(C1)C2C#N 96165,c1(C(=O)NC2(C)CC(C)(C)C2)cnc2ccccc2c1 96166,C1(C)(CC)CC(NC(C23CC(CO)(C2)OC3C)=O)CN1C(=O)CSC(F)F 96167,C1(NC(c2ncccc2O)=O)CN(C(c2cnc(S)nc2)=O)CC2(CCC2)C1 96168,C1(n2cc(C3(O)CN(C(=O)CC4CC45CCC5)C3)nn2)CCOCC1O 96169,c1(C(=O)NC2CC(NC(CCCOCCC)=O)C2)ccc(C(C)C)cc1O 96170,C1(C)(C(=O)NCC(CC)NC(C)=O)CCCN(C(c2cccc(C)c2)=O)C1 96171,N1(C(Cc2c(C)scc2)=O)CCCC2(CC(NC(c3ncccc3F)=O)CO2)C1 96172,c1(C(=O)OC)nc(C)n2c1N(C(C1CCC1c1ccccc1)=O)CCC2 96173,C(C(CCO)C(C)(C)C)N(C(=O)NC1C(C)CCC1)CC1CC1 96174,N1(C(=O)Nc2c(C)c(O)c(Br)cn2)CC2(COC(C)(C)C2)C1 96175,c1(NCC2(CCOC)CC2)nc[nH]c(=NCC2Cc3ccccc3C2)c1C 96176,Cn1cc(Cl)c(C(=O)NCC2CC2NC(c2cnc(-c3ccc(Cl)s3)s2)=O)n1 96177,C1(N(C)C(C2(C(=O)C3CC3)CC2)=O)CCN(C(=O)C=C(C2CC2)C2CC2)CC1 96178,C1(CCC(=O)N(C(C(C)SC)C)C)CCN(C(c2cnc(O)o2)=O)CC1 96179,c1(OC)nccc(C(N2CCCCC2CNC(c2ncccc2C2CC2)=O)=O)n1 96180,N1(C(CC(CCCC)O)=O)CC2(CCN(C(c3cc(C)nc(Cl)c3N)=O)CC2)C1 96181,C1(C)(CC(=O)NCC2(CSC)CC2)CCN(C(C2C3CCC(=O)C23)=O)C1 96182,C1(F)(C(N(C)CC2N(C(c3c(CC)ncs3)=O)CCC2)=O)CCCN(C)C1 96183,c1(-c2nc(C(C3CC3)OC)nn2-c2ccn(C)n2)cnn2c(C)ccnc12 96184,Cn1cc(C(N2CCSCC2CCNC(c2ccnnc2O)=O)=O)c(Cl)n1 96185,N1(C(C2C(NC(C(C)n3cccn3)=O)CCC2)=O)CCC(C)(CO)C(O)C1 96186,C#CCCC(O)CCNC(c1cccnc1CNC(=O)C(C)C1(O)CCC1)=O 96187,C1(C(N2CC(SC)C(n3cc(C(C)(C)CO)nn3)C2)=O)CCCCN1N=O 96188,Cc1cnc2nccc(C(=O)NC3(CN(C)C(c4cnn(C)c4C)=O)CC3)c2c1 96189,c1(NC(C2C(NCc3ccc(OCC)c(C#N)c3)C2)=O)nccc2scc(Br)c12 96190,N1(C(Cc2cc(CC)no2)=O)CCC2CN(C(C3CCc4c[nH]nc4C3)=O)C2C1 96191,N1(C(C)C)CCN(C(=NC2CC2)NC2CC(c3ccccc3F)C2)CC1 96192,C(=O)(C(O)P(C)(C)=O)N1CC2C(C(N3C(C)(C(=O)NC)CC3)=O)C2C1 96193,C1(NC(c2c(NC)snc2C)=O)CCCN(C(=O)C(C)CC(C)C)CC1 96194,c1(C(N2CCC(C(=O)NCCCOC)(CO)C2)=O)cc(C#N)[nH]c1C 96195,C1(C(=O)NC(c2cnn[nH]2)C)CC(O)CN1C(C1CN(C(N)=O)C1)=O 96196,c1(CC(=O)NC(CNC(c2ncn(C)c2)=O)C2CC2)cccc(Br)c1 96197,c1(CC)ccc(CC(=O)NC2CCC(C)N(C(c3[nH]c(C)cc3C)=O)C2)cc1F 96198,C(=O)(C1=NOCC1)N(C1CCCC(N(C)C(c2cncc(N)n2)=O)C1)C 96199,C(=O)(C#CC1CCCOC1)N1CC(C(C)NC(CC(C)C)=O)OCC1 96200,Cc1ccc(CN(CCO)C(c2c[nH]cc2Br)=O)cc1 96201,c1(C(=O)OCC)cc(C(N2CCCC2CCNC(=O)C(C)C2CCC2)=O)[nH]c1C 96202,C1(NC(CCCCCSC)=O)CN(C(C2(F)CCOC2)=O)CC1N=[N+]=[N-] 96203,c1(C(=O)NC2C(CNC(C3(C(C)C)CCOCC3)=O)CC2)cc(C#N)ccc1F 96204,c1(CN2CC(C(C)NC(=O)Cc3nnco3)C2)ccc(-c2ccccn2)cc1 96205,N1(C(C(C2CC2)OC)=O)CC2CCC(NC(c3sccc3S(C)(=O)=O)=O)(C2)C1 96206,Cc1ccc(C(=O)N(C2CCN(C(c3cc(Cl)no3)=O)CC2C)C)nc1O 96207,CCC(F)(C(=O)OC)C(=O)N1CC(O)(C(C)NC(C2CN(S(C)(=O)=O)C2)=O)C1 96208,CC1CN(C(=O)C=Cc2cn[nH]c2)CC(C)CN1C(c1cc(O)cs1)=O 96209,Cn1ccc(CNC2CC2C(=O)Nc2ccc(C(F)(F)F)cc2F)cc1=O 96210,C1(CCC)CCCN(C(=O)C(CNC(=O)C(C)(C)C2CC2)CCC)CC1 96211,C12(CNC(C3CC(CC)(CC)C3)=O)CCCC(CN1C(c1cncc(C)c1)=O)C2 96212,c1(NC(C2CCCC(C(=O)OC)C2)=O)nn(C)c2ccccc12 96213,c1(OC)ccc(NC(=O)NC2CN3CCC2(C(F)(F)F)C3)c(OC(F)F)c1 96214,C1(CNC(c2cc(Br)no2)=O)CCN(C(C23CCCC2C3(F)F)=O)C12CC2 96215,C1(CC=C)(C(=O)NCCN2CCOCC2)CN(C(C2CCCO2)=O)C1 96216,C1(CC(=O)NCC(C(C)C)NC(C2CCC(C(=O)OC)C2)=O)CCCC(C)(C)O1 96217,C(CC(C)C)(C(=O)NCC(O)C(C)(C)O)NC(C1C(COC)CC1)=O 96218,C=CCC(F)(F)C(=O)NC1CN(C(c2cc(CC)ccn2)=O)CC1OC 96219,N1(C(c2ccn(CC)n2)=O)CCCCC(NC(c2c(NC(C)=O)c[nH]c2C)=O)C1 96220,CC1CN(C(c2ccnn2CCF)=O)CCC1CNC(C1CC2(CCOC2)C1)=O 96221,CC1CN(CC(=O)NCC2(O)CC2)CCC1NC(c1cn(CCC2CC2)nn1)=O 96222,Cn1ccc2ccc(C(=O)NC(C)(CNC(=O)CCN3CCCCC3)CO)cc12 96223,c1(C(C(=O)NCCC)N(CCC(C)OCC)C)ccc(C)c(OC)n1 96224,N1(CC(c2cccc(C)c2)=O)CC(S(=O)(=O)C2CCCCC2)C1 96225,N1(C(C2N(CC)CCOC2)=O)CCCC(O)(CCNC(=O)Cc2ncoc2C)C1 96226,Cc1nn(-c2ccccc2)nc1CNC(=O)Cn1cc(C2CC2CO)nn1 96227,C(C(C)C(F)C(=O)NC(CCO)C(C)C)NC(c1c(C)n(C)cn1)=O 96228,c1(CN2CCC(CC(N3CCC(CC(=O)NC)CC3)=O)C2)ccc(C#N)c(Cl)c1 96229,C(CCC(C)CC(=O)NC1(CF)CCN(C(=O)CN(C)CCO)C1)=C(C)C 96230,n1(CC(=O)NC2C(CNC(CCSCCC)=O)C2)nc2n(c(=O)c1=O)CCC2 96231,CC(C)CCC(=O)N(CC(O)CN(CC(=O)NS(=O)(=O)Cc1ccon1)C)C 96232,C1(NCCC2CC=CCC2)COC2(CCC2)C1 96233,N=c1c(C(=O)OC2CCCC2(F)F)c[nH]n1-c1ccc(Cl)cc1 96234,N1(C(C(c2cncnc2)C)=O)C2CCC1C1CC1(NC(=O)CCc1cncs1)C2 96235,C(=O)(C(C)(C)C(=O)N1CCCCC1C(=O)NCC1C2CCCOC12)OCC 96236,Cc1ccc(CC(N2CCC(C(F)F)(CNC(C3CCC3(C)C)=O)C2)=O)c(C)c1 96237,C(=O)(CC(F)(F)F)NCC1CN(c2ncccn2)C1.CC1CNC(=O)NC1 96238,c1(C(N2CCCCC(CNC(C3C(C)C3)=O)C2)=O)ccc2nn[nH]c2c1 96239,Cc1ncc(Br)c(Nc2coc(C)n2)n1.N1(C(C)=O)CC2CNCC2C1 96240,CC(C)(CCNC(c1csc(-c2ccccc2)c1)=O)C1CC1 96241,C(=O)(C1=CCCN(C(=O)CC2CC(O)C2(C)C)C1)NC(CSC)(C)C 96242,CC1SCCCN1C(N1CCCC1c1cccnc1)=O 96243,C1(C(N(CCC(=O)NCC2C3COCC23)C)=O)OC2CCC1C2 96244,CC1CC(NC(=O)CCc2ccon2)CN1C(c1ncccc1C(F)(F)F)=O 96245,N1(C(COC(C)C)=O)CCCC(NC(c2ccn(C)c(=O)c2)=O)C(F)C1 96246,N1(C(CC2(C=C)CN(C(c3cc(OC)no3)=O)C2)=O)CC2(C1)CC2(F)F 96247,c1(OCC)ccc(C(=O)NC(C)(C)C(C)NC(=O)CCNC(=O)C=CCl)cc1 96248,C1(C(=O)OC)(NC(c2cc(C3CCCN3C)[nH]n2)=O)CCCNC1 96249,N1(C(c2c(C)cno2)=O)CCN(c2nc(C(C)C)ns2)C(CCO)C1 96250,c1(CN=C(NC(COC)C)NCCc2c(C)cccc2C)cc(F)c(C)cc1F 96251,C1(C)(C(=O)NCCCN(C(C)=O)C)CCN(C(C2CC(=C3CC3)C2)=O)CC1 96252,C1(C(N(C(C(N)=O)C2CCCC2)C)=O)CCC1NC(C1CC12CC2)=O 96253,N1(CC)CCC(NC(C2(CCNC(=O)Cc3ccc(C)o3)CC2)=O)C(C)C1 96254,N1(C(c2ncn(C)n2)=O)CCCC(C2(NC(c3cnc(Cl)c(F)c3N)=O)CC2)C1 96255,c1(NC2CCN(C(=O)NC)CC2)nc(C(F)(F)F)ccc1I 96256,c1(OC)ccncc1C(=O)NCc1nocc1C(N1CCC1C(N)=O)=O 96257,CC(C)CC(C)(O)C(=O)N1C2CCC(C(=O)NCc3cnns3)C1CC2 96258,N1(C(C2CN(C)C2)=O)CCC2(NC(=O)Cc3cc(O)nnc3O)CCCCC12 96259,c1(OC)cc(C=CC(=O)NCCCC(C)NC(=O)C(C)SC)ccc1O 96260,N1(C(CC(COC)(C)O)=O)CCC(N=[N+]=[N-])(C(=O)NOCC(N)=O)C1 96261,Cn1ccc2[nH]c(C(N3CCC(NC(C4(C5CCC5)CC4)=O)C3(C)C)=O)cc12 96262,c1(CNC(CCC2N(C)CCC2)=O)ccc(C(=O)NCC(N2CCCC2)C)nc1 96263,C(C(O)C(=O)NCCC1(NC(=O)C(C)n2ccnc2)CCC1)=CCCC 96264,N1(C(COC)=O)CCC2(CCCN2C(=O)CCc2ccc(OC(F)F)cc2)C1 96265,Cc1cccnc1CC(N1CCC(C(F)F)(CNC(c2cc(CF)on2)=O)C1)=O 96266,c1(C(N2C3(CNC(C(CCOC)C)=O)CCC2CC3)=O)cc(Cl)cc(Cl)c1OC 96267,CC1(C(N2CCCC2c2cn(-c3ccc(CN(C)C)cc3)nn2)=O)CCCC1(F)F 96268,c1(C(=O)NC(CNC(=O)C=CCn2cncn2)CO)ccc(-n2ccnc2)nc1 96269,CN1CCC(C(c2nnnn2-c2ccccc2)NCCC(C)(C)CCCC)C1=O 96270,c1(NC(C(C)NC(=O)NC)=O)cc(NC2CCCC2)c(F)cc1F 96271,Cc1ccc2c(Cl)c(C(=O)NCCC(C)CCNC(c3nocc3C)=O)sc2c1 96272,c1(NC(C2CC2NCc2cscn2)=O)cccc(Cl)c1I 96273,c1(C(=O)OCC)nc2c(s1)C(NC1CC1C1CCNCC1)CCC2 96274,N1(C(COCCOC)=O)CCC2(CNC(=O)C3=NNC(=O)CC3)CCCCC12 96275,c1(NCC(C)CNC(=O)CC2CC(O)C23CCC3)ncnc(N(C)C)c1[N+](=O)[O-] 96276,c1(CN2CCCC(C(N3CCOC4CC34)=O)C2)cnc(Cl)cc1Cl 96277,c1(C(=O)NC2(CN(C)C(c3ccc(CO)cc3)=O)CC2)cccc(N(C)C)n1 96278,Cc1c(C(N2CC(CCNC(C3OC4CCC3C4)=O)C2)=O)[nH]c2c(Cl)cccc12 96279,c1(C(=O)NCC2CN(C(C(C)NC(c3ccoc3)=O)=O)CC2C)cccc(Cl)c1F 96280,N1(C(CCCCC=CC)=O)CCC(C2(NC(=O)Cc3sccc3C)CC2)C1 96281,c1(OC)cc(-c2ccc(Cl)c(C(C)=O)c2)ccc1O 96282,c1(SC)nn(C)cc1C(N1CCC(C)C1CNC(C1(C(F)F)CCC1)=O)=O 96283,N1(C(c2cnn(C)c2C2CC2)=O)CCC2(CCN(C(=O)CC3(C)CC3(Cl)Cl)C2)C1 96284,c1(C(=O)NCC(CN(C(c2c(O)ccc(CC)c2)=O)C)C)cc(S(N)(=O)=O)co1 96285,c1(OC)cc(C(=O)CN2CCC(S(N)(=O)=O)C2)cc(Br)c1OC 96286,C1(OC)CCC(C(=O)NCC2CCCCC2NC(=O)CSC2CC2)CC1 96287,Cc1ccc(Cl)c(N)c1C(N1CCC(CNC(=O)C(C)(F)F)C(F)(F)C1)=O 96288,C=CCCC(C(=O)N(CCNC(=O)CC(=O)NC1CCC1)CC)c1ccccc1 96289,C1(CNC(C(C)(C)C#N)=O)CCCCN(C(=O)CC2SC(=N)NC2=O)C1 96290,c1(C(=O)OC(c2ccc(F)cc2F)C(=O)OC)cccc2nsnc12 96291,C1(CNC(=O)OC(C)(C)C)(CNc2cc([N+](=O)[O-])cs2)CC2CCC1CC2 96292,CCC(C)(C#N)C(=O)NC1CCCN(C(=O)C(F)=C(C)C2CC2)C1 96293,C1(NC(c2cnn(C)c2F)=O)CCC2CC1CN2C(c1cc([N+](=O)[O-])c[nH]1)=O 96294,c1(CSCC(=O)NCCNC(C2ON=C(CC)C2)=O)n[nH]c2ccc(Cl)cc12 96295,Cc1csc(CC(=O)NCC(=O)NCCn2ccnc2C)c1 96296,CCCCCCCCN(C(=O)C(CC1CC1)N(C(=O)C(C)OC)CC)CC 96297,C1(C(N(C)CC2(O)CN(C(C(C)n3cnnn3)=O)C2)=O)CCC2(CCC2)C1 96298,N1(C(c2c(OC)c(Br)ccc2)=O)CCn2cnc(C3=CCSCC3)c2C1 96299,Cc1cc(C(=O)NCCN2CCN(C(C3CCNC3=O)=O)CC2)cnc1O 96300,N1(C(C(C=CC)O)=O)CCCC2(CCN(C(=O)C=CSc3ccccc3)CC2)C1 96301,CCC(C)(CC)C(=O)NCCCCCNC(C1CCCC(C)CC1)=O 96302,C(=O)(C(F)(F)C(F)(F)F)NCC(CC=C)NC(c1coc(Cl)n1)=O 96303,C#Cc1cccc(CC(=O)NCC2CC(F)(F)CN2C(=O)CSC2CC2)c1 96304,CC(C)CN=C(NCC1(COC)COC1)N1CC(C)N(CCO)C(C)C1 96305,CCC(CC(C)C)C(=O)NCC1CC2(CC2)CN1C(=O)CCC(=O)N(CC)CC 96306,CS(=O)(=O)c1ccc(C(N2CCC(N(CCO)C(C3CCNC3=O)=O)C2)=O)cc1 96307,C1(CNC(CC(C)N(C)C)=O)CN(C(c2n[nH]c3c2COCC3)=O)CC(C)(C)O1 96308,CCCC(C(C(=O)NC)N1CC(O)C2(CCC2)C1)OC 96309,c1(CC(N2CC(=C(CNC(C(CC)SC)=O)F)C2)=O)ccc(F)cc1C 96310,C(=O)(C(F)(F)C(F)(F)F)NC1CCC(CNC(C2CC(OC)CN2C(C)=O)=O)C1 96311,N1(C(C2CC(CNC(=O)CCn3ccnn3)C2)=O)CC(O)(C(F)F)C1 96312,N1(C(C2(C)CCCCO2)=O)CC2(CCCC2NC(C2(C3CCC3)CC2(F)F)=O)C1 96313,c1(C(N2CCC(=CC(N3CCC34CCCCC4)=O)CC2)=O)c(F)cc(F)cc1Cl 96314,C1(CNC(C(c2ccccc2)OCC)=O)CCN(C(=O)CNS(=O)(=O)CC)CC1 96315,N1(C(C2(C)CC(=C)C2)=O)CCN(C(c2ccnn2C)=O)C(CCCC)C1 96316,CC(C(=O)N1CCC(n2cc(-c3ccc(Br)cc3)nn2)CC1)C(F)F 96317,N1(C(=O)Cn2nnc(=O)[nH]2)CC2(CCN(C(c3ccc(Br)cc3F)=O)CC2)C1 96318,N1(C(C(Cn2ccc(C)n2)C)=O)CC2CN(C(c3ccc(C)c(O)c3)=O)CCC12 96319,N1(C(CC(COC)(C)C)=O)CCCC2(NC(C3CC3F)=O)CCCC12 96320,c1(C(N2CC=CC(NC(C(C)Oc3ccccc3)=O)C2)=O)cn2ccncc2n1 96321,N1(C(Cn2cnc(=N)[nH]2)=O)CCC2(NC(c3ccc4nc[nH]c4n3)=O)CCCC12 96322,c1(OCC(=O)N(CC(C)O)CCNC(=O)CNC=O)ccc(Cl)cc1 96323,c1(C(N2C(CNC(CCOC(CC(C)C)C)=O)CC2)=O)ccc([N+](=O)[O-])s1 96324,c1(C(=O)NC(CC=C)CNC(=O)CC2CCC2(F)F)nc(Cl)sc1C(C)C 96325,c1(C(N2CCC(CCOC)C2)=O)n[nH]c2c1CN(C(=O)CCc1cccnc1)C2 96326,N#Cc1ccc(F)cc1CNC1CCN(c2ncccn2)C1 96327,CC1C(NC(=O)CC2=CCN(C)CC2)CC2CCC1N2C(C1CCCOC1C)=O 96328,C12(CNC(c3cccc(C)n3)=O)CCCCC1N(C(c1ccc(O)cc1)=O)CC2 96329,c1(C(=O)OC)cc(Cl)ccc1S(=O)(=O)Nc1ccc(CC(C)O)cc1 96330,C(N=c1[nH]c(=N)[nH]c(=NCC(CSC)N2CCN(CC)CC2)[nH]1)C1(OC)CCC1 96331,c1(OC)ccccc1C(F)(F)C(=O)N(C)CCNC(c1cc(Cl)ncn1)=O 96332,CCCS(=O)(=O)CC(=O)NC1CC2(C1)CN(C(=O)C(C)(C)C1CCOCC1)C2 96333,C1(N(C)C(c2cc(C(C)(C)C)on2)=O)CCC(NC(=O)CCCC#N)CC1 96334,c1(C(=O)NC(CNC(c2c(C(C)C)c[nH]n2)=O)(C)C)ccc2c(c1)C(C)C(C)O2 96335,C1(CNC(CC2(CSC)CC2)=O)CC12CCN(C(c1c(C)nsc1Cl)=O)CC2 96336,CN1CCOCC1CNC(C1(NC(C2CCCOCC2)=O)CCCCC1)=O 96337,C1(C(=O)NCC(C)NC(c2cnoc2CC(C)(C)C)=O)CCCCC1O 96338,N(C(=NCCOC(F)F)NCC(Cc1ccccc1)C(C)C)CC(CC)(C)C 96339,c1(N2C(=O)C3CC3C2=O)cc(F)cnc1Br.c1(NC)cc(C)nc(Br)c1 96340,C1(C(=O)NCC(C)NC(c2c(CCC)n[nH]c2)=O)CC12CCC1(CC1)CC2 96341,Cc1cc(C(=O)NC2(c3cc(Br)ccc3Cl)CC2)cc(C)c1N 96342,c1(C(C(N2CCC(C)(C(=O)NCC3CC3CF)C2)=O)(F)F)ccc([N+](=O)[O-])cc1 96343,CC(F)(CC1CCCC1)C(=O)NCC1CCN1C(c1cc(Cl)cs1)=O 96344,N(C(=NCC(C)C)N1CCN(Cc2nc(C3CC3)n[nH]2)CC1)CC(=C)C 96345,C1(CNC(CCC2CCN(C(C=CCOC)=O)C2)=O)C2CCCCCC12 96346,C1(NC(COCCNC(C(n2c(C)ccn2)C)=O)=O)CCC(C(C)C)CC1 96347,CC(CC(N)=O)C(=O)NC(CC(N)=O)C(=O)NC(C)CCO 96348,N1(C(CC=C=C)=O)CCN(C(=O)C=Cc2ccc(-c3ccccc3)s2)C(CO)C1 96349,c1(N2C(C(CNC(C=Cc3n(C)ncc3)=O)(C)C)CCC2)nccc(C#N)n1 96350,C1(c2cn(CC3N(C(C(c4cn(C)nc4)O)=O)CC3)nn2)CC2C=CC1C2 96351,C1(C(=O)Nc2c(COC)nn(C)c2)N(C(C2CC=C(C)CC2)=O)CCC1(C)C 96352,N1(C(c2c(CNC(CC(C)c3ccco3)=O)noc2)=O)CCC2(CCN(C)C2)C1 96353,c1(NCCc2ccc(OC)nc2)ccc(S(=O)(=O)N2CCCC(C)C2C)c(Cl)c1 96354,c1(C(=O)Nc2ccc(-c3nc(C)c(C)[nH]3)cc2)cc(Br)cc(Cl)c1C 96355,C1(C)(C(N2CC=CC(C(=O)NC(CCC(C)C)C)C2)=O)CCC2CC2C1 96356,c1(NC(C(C)SCC2CONC2=O)=O)cccc(Br)c1 96357,N1(C(C2CCCN(C)C2)=O)CC(CNC(c2c[nH]c(=O)cn2)=O)C(C)(C)C1 96358,c1(CONC(c2cn(C)nc2CCC(F)(F)F)=O)c(F)cccc1I 96359,C1(C(N2C(C(=O)NC3(C)CC(O)(CO)C3)C=CC2)=O)CN2CCN1CC2 96360,N1(C(CCC(=O)NC)=O)CC(C)CN(C(c2cnccn2)=O)C(C)C1 96361,C(c1csc(C)n1)=CC(=O)NC(CCNC(c1n(CC)cnn1)=O)C 96362,c1(OC)cncc(CCC(=O)NCC(C2CCC2)NC(=O)C=C(C)C(F)F)c1 96363,c1(C(C(=O)NC2(CNC(C(C)OCCOCC)=O)CC2)(F)F)cc(Cl)sc1Cl 96364,c1(C(N)=O)ccc(CCC(N2CC3C(CNC(=O)COCCCF)C3C2)=O)cc1 96365,N1(C(=O)OC(C)(C)C)CC(N=[N+]=[N-])CC1C(=O)NCC1(C(C)(C)O)CCC1 96366,C1(NC(CCCOCCOC)=O)CN(C(C2(C(F)(F)F)CCC2)=O)CC1C.C1(C)CC1 96367,c1(C(=O)NC2CCCN(C(c3ccc(CC)o3)=O)C2)c(C)ccc(C)c1N 96368,c1(C(=O)NC(CNC(CSCC#C)=O)CCOC)cnc2c(C)cccc2c1 96369,CC(CCNCCc1ccnc(Cl)c1F)P(C)(C)=O 96370,N1(C(COC(C)(C)C)=O)CC(C)(C)OC2(C1)CN(C(C1C3CS(=O)(=O)CC13)=O)C2 96371,C1(C)(C(N(CC(C)O)CCNC(=O)Cc2ccno2)=O)CCC(=O)N1 96372,c1(CC)nc(CCNC(C2CC(C)N2C(c2ccnn2CCF)=O)=O)n[nH]1 96373,N1(C(=O)CCOc2ccccc2C(F)F)CC2(CCN2C(C2CC2Cl)=O)C1 96374,C(c1scnc1C)=CC(=O)N(CC(C)(C)NC(c1c(CC)occ1)=O)C 96375,c1(C(=O)NC2C(NC(c3cc(Cl)cs3)=O)COCC2)ccc(F)c2c1CCC2 96376,C(=O)(CC1=CCOCC1)N1CCC(O)(C(C)NC(=O)Cc2c[nH]nc2O)C1 96377,Nc1ccc(C(=O)NCC2CCN(C(C3CC(F)C(=O)N3)=O)C2)cc1F 96378,C1(CC(=O)NC2C(NC(c3c(OC)nsc3)=O)CCOC2)SC2=NCCN2C1=O 96379,n1(CC(=O)NC(C)CC(C)NC(=O)CSCC(F)(F)F)nc2n(c1=O)CCOC2 96380,CC1CC=C(C(=O)NC(C2CCCC2)CNC(=O)CSC(C)(C)C)CC1 96381,Cc1ncc2cc(C(N3CCC(c4nc(C5CC5)no4)CC3)=O)c(O)nc2n1 96382,c1(COC)nn[nH]c1C(=O)N(C1(C(=O)NCCC(C)SC)CC1)C 96383,CCC(C)CCCCC(=O)N1CCC(NC(c2cnc(N(C)C)cn2)=O)CC1C 96384,N1(c2snc(C(C)(C)OC)n2)CCOC(C(C)NC(C2CC(=O)N2)=O)C1 96385,c1(CC(N2C(CNC(C3OC4CCC3C4)=O)CC(F)C2)=O)nc([N+](=O)[O-])n[nH]1 96386,C1(C(=O)NC(CC)(CNC(=O)CCSCC(=O)OC)CC)OCC2COCCC12 96387,Cc1nc(C2CC2)nc(O)c1C(=O)NC1CCC(N(C(=O)Cc2cscn2)C)C1 96388,C1(CCNC(COCCN(C)C)=O)CN(C(=O)Cc2cncnc2)CCO1 96389,C1(NC(CCCN(C(=O)CCC(F)(F)F)C)=O)CC2CCC(C1)N2C 96390,C1(C2CCOCC2)(C(N2CC3(CN(C(C4CC4F)=O)C3)OCC2)=O)CCOCC1 96391,CC1CCc2onc(C(=O)N(CC(C)NC(c3ccc(Cl)cn3)=O)C)c2C1 96392,C(C(N=c1ccnc(COCCOCCO)[nH]1)C(C)C)NC(C(C)OCCNC)=O 96393,c1(CN(CCC)CCO)cncc(-c2ccc(CNC)cc2)c1 96394,C=CCCC(C(=O)NCC=Cc1ccccc1)NC(C1CC2(CC2)C1)=O 96395,C#CCC(C)(C)C(=O)N1CC(C(N2CC(C(F)(F)F)C2)=O)C2(CC2)C1 96396,C1(CC=C)(NC(COCCC=C)=O)CN(C(c2cc(Br)cs2)=O)C1 96397,C(C(C)N(C)N1CCCC1C1CCCCN1C)c1cccc(C)c1 96398,O(N=c1cc[nH]c2ccncc12)CCC(N1CC(C)OCC1)=O 96399,c1(C(N2C(CNC(CCC)=O)C(C)CC2)=O)ccc(F)c(OC)c1F 96400,c1(NCCC(C)NC(C2CC2(C)C)=O)nnccc1C#N 96401,N1(C(C(C)OCC)=O)CC(C)C(C)(CNC(c2ccnn2CC(F)F)=O)C1 96402,c1(C(=O)NC2CC(NC(CCc3c(OC)cccc3)=O)C2)nc(Cl)ccc1N 96403,N1(C(C(c2cccc(Cl)c2)(C)C)=O)CC2CC(C1)N(C(=O)C(O)CCN(C)C)C2 96404,N1(C(C(=O)NC(C)C)C)CCC(NC(c2ccsc2C(F)F)=O)C(C)C1 96405,C1(C(=O)NC2CC(C(C)C)OC2)CN(C(C2(C)CC(=O)C2)=O)CC1F 96406,C1(C(=O)NC23CC(NC(C(C)c4ccco4)=O)(C2)C3)CN2CCN1CC2.C12CC1C2 96407,Cc1nc2ccc(C(=O)NC(C)C(C(C)C)NC(=O)CC(C)C)cc2c(=O)n1C 96408,C1(C(N2CC(C(C)NC(C3(C)CC3)=O)OCC2)=O)CC2CC(=O)C1O2 96409,O=C(NNC(=S)NC1CC1)C1CSCN1S(=O)(=O)Cc1ccon1 96410,CC(C)CCCC(C)C(=O)NCC1CN(C(c2ccc(CO)o2)=O)CCCO1 96411,N1(C(C(C)S(C)(=O)=O)=O)CC2CN(C(C3(C)CCC(F)(F)CC3)=O)CC2(C)C1 96412,c1(C(N2CCCC(C)(NC(c3cc(C(N)=O)[nH]n3)=O)C2)=O)cc(F)c(F)c(F)c1 96413,C12(NC(C3CCS3(=O)=O)=O)CCCN(C(c3cc4ccsc4s3)=O)CC1C2 96414,c1(N2CC(CC=C)(NC(c3cc(C4(C)CC4)on3)=O)C2)nc2ccc(Br)cc2o1 96415,C1(NC(C2(COC)CC2)=O)CC(O)CN(C(c2c(OC)ccnc2O)=O)C1 96416,CCCC(C(=O)N(C)CCNC(=O)C=CC1CCCO1)S(N)(=O)=O 96417,C(=O)(CC(C)C(C)C)N1CC(CCCCNC(CCc2cnc(C)o2)=O)C1 96418,C(CC(C)C)(C(N)=O)NC(c1n(CC=C)nnn1)c1cnc(-c2ccccc2)s1 96419,CC(C)CC(CC(=O)NC(C(N)=O)C1CC1)NC(C1COCCC1C)=O 96420,C(=O)(CCC(=O)c1cccs1)NCC(C)(C)CNC(c1ccsc1)=O 96421,CC(C)(C#N)C(=O)NCCCOCCCNC(C1CC(O)(c2ccccc2)C1)=O 96422,N1(C(CCCC(=C)C)=O)CC2(CCN(C(=O)C(C(C)(C)C)N(C)C)CC2)CC1C 96423,C12(F)CCN(C1)C2=O.c1(N(CC(=O)NC)CC)ccc(Oc2cccnc2)cc1 96424,C1(CNC(CCCN(C)C)=O)CCCCN(C(=O)CC2(C3CC3)CC2)C1 96425,N1(C(COCc2onc(CC)n2)=O)CCOC(CNC(C2COCCN2C)=O)C1 96426,C1(N(C(CCC(C)C)=O)C)CN(C(C2CCCN(C(N)=O)C2)=O)CCC1C 96427,c1(C(=O)NCC2(NC(C(C)CF)=O)CCCCC2C)ccc2nc(O)[nH]c2c1 96428,c1(C(N2CCC(N(CC#C)C(c3ccc(C)nc3)=O)CC2)=O)ccc(N)c(O)c1 96429,C1(NC(CCCOCC)=O)CCCC(CNC(=O)C(C)NC(c2cccs2)=O)C1 96430,C(=O)(C1CCCc2nn[nH]c21)NCCC1CC(NC(=O)C=CCF)C1 96431,C(=O)(NNC(=O)C1CC(=O)N(c2ccccc2)C1)NCCCCN(C)C 96432,N1(C(C(CC)(C)F)=O)CC(CNC(=O)CNC(=O)CNC(C)=O)OC(C)(C)C1 96433,C1(N(C)C(C2CCC(=O)C2)=O)CCCN(C(=O)CCCN2C(=O)CNC2=O)CC1 96434,C1(CNC(CCCC#C)=O)CCCCN(C(c2ccc(O)nc2C)=O)C1 96435,C1(C2CCC2)(C(=O)NCC2C(NC(c3cccc(C(F)F)n3)=O)CC2)CC1 96436,c1(C(=O)NC2C(CNC(C(C=C)O)=O)CC2)sc2ccc(C(=O)OC)cc2c1C 96437,C1(CCNC(CC2(CC)CCC2)=O)(NC(c2cnc(OC)s2)=O)CCCC1 96438,c1(OC)ccc(F)cc1CC(=O)NC1CC(C)N(C(c2ncccc2OC)=O)C1 96439,Cc1cccc2[nH]c(C(=O)NCC3CCCCN3C(C3(C)CCCS3)=O)cc12 96440,C1(NC(C2C=CCC2)=O)CC2CC(C1)N(c1nccc(CO)n1)C2 96441,C(c1nc2ccccc2s1)=CC(=O)OCC(c1c(C(=O)OC)scc1)=O 96442,C1(NC(Cc2c(C)cccc2)=O)CCN(C(C2CN(S(C)(=O)=O)C2)=O)C12CCC2 96443,N1(C(C2CCCC(C)(C)C2)C(=O)NCC)CCOc2ccccc2C1C(=O)OC 96444,Cc1nn2c(c1CNC(C1(n3nccn3)CC1)=O)CN(C(=O)Cc1ccco1)CC2 96445,N1(C(c2ccc(OC)c(C)c2)C(=O)NC2CCCC2)CCC2(CC(=O)N(C)C2)C1 96446,c1(OC)ccc(CC(N2CCCC2CC(N2CCC(F)C2)=O)=O)c(OC)c1 96447,Cc1cc(C(=O)NC2CCN(Cc3cncc(C(F)(F)F)c3)C2)c(F)c(Br)c1 96448,N1(C(c2c(C)c[nH]n2)=O)CC(NC(C2CC23CC3)=O)CC1(C)C 96449,CC1CCC(C(C)(O)CNC(=O)NCCNC(c2cnnn2C)=O)CC1 96450,c1(C(N2CCC(NC(c3cc(Cl)cc(F)c3F)=O)C2)=O)cccc2cc[nH]c12 96451,CC1=C(C(=O)NC(C)CN(C(=O)C(C)N(CC(F)(F)F)C)C)S(=O)(=O)CCO1 96452,C1(CN(C)C(N)=O)CCCN(C(C2CCCN2C(C2C3(CC3)C23CC3)=O)=O)C1 96453,C1(NC(C(C2CCOC2)OC)=O)CCC2CC1CN2c1ncnc2[nH]cnc12 96454,C(=O)(C1Cc2ccccc21)N1CCC(C)(CNC(c2c(C)nsc2)=O)C1 96455,c1(C(=O)NC(c2cccc3cc[nH]c23)c2ccccc2)nc2c(s1)CCCCC2 96456,S(=O)(=O)(c1cccnc1NCC1CCC(C2CC2)O1)N1CCCC(C=C)C1 96457,c1(C(N(C2CN(C(C3(C)CCCCO3)=O)C2)C)=O)coc(S(C)(=O)=O)c1 96458,N1(C(c2c(OC)nsc2)=O)CCN(C(=O)CC(C)N(C)C)C(c2cccnc2)C1 96459,c1(C(=O)NCCC(C)NC(C(Br)=C(C)C)=O)cccc2cccc(C)c12 96460,c1(C(C(=O)NCC2CC(NC(=O)COC3CC3)C2)=O)ccc(Cl)cc1Cl 96461,C1(CC(=O)NCCOC(C)=O)C=CC(NC(=O)C=Cc2ccsc2)C1 96462,c1(C(=O)NC)cc(OC)ccc1C(=O)NC1CCN(C(=O)C(C)C(C)C)C1 96463,C#Cc1cccc(C(=O)NCC(N2CCN(C(C3CC3C(F)F)=O)CC2)=O)c1C 96464,c1(OC)nccnc1-c1cccs1.c12csc(n1)C(=O)N1CC(C1)N2S(C)(=O)=O 96465,Cc1ccc(C)c(CC(=O)NC2CN(C(C34CC(CO)(C3)OC4C)=O)C2)c1 96466,C#CCC(C(=O)NCCOC1CCN(C(=O)CC(=O)NCC(F)(F)F)C1)C1CC1 96467,C1(CC)(NC(=O)CCCCN(C)C)CCN(C(=O)CSCCOC)CC1 96468,C1(COC)(CNC(=O)CC(C)N(C)C)CCN(C(=O)C(C)CC(C)C)CC1 96469,CC1(C)CC(C(=O)NC2CCN(CCF)C2)CN1C(=O)CCC(=O)c1ccc[nH]1 96470,c1(NCC2(c3ccccn3)CN(C(=O)OC(C)(C)C)C2)ccc2cccnn12 96471,c1(OC)ccc(C(N2CCCC(CNC(=O)CCc3ccoc3)C2)=O)c(Br)c1 96472,c1(C(=O)OCC2OCC(C)(C)C2)ccn2ncnc2c1 96473,N1(C(c2c(C)cccn2)=O)CCCN(C(c2c(F)ccc(Cl)c2F)=O)C(C)C1 96474,c1(C(C)C)cnn(C)c1C(=O)NCC1(O)CC(NC(=O)CC2CCS(=O)(=O)C2)C1 96475,CC1(C)OC(=O)CC1C(N1CCC12CN(C(=O)Cc1ccc(Br)cc1)C2)=O 96476,C1(N(CC)CC)CCN(C(C2CC(C(=O)Nc3ccnnc3)CN2)=O)CC1 96477,c1(CC)oc(C)cc1C(N1CC2CC2(CNC(c2sc(C)cc2OC)=O)C1)=O 96478,C1(NC(c2cccn2CC(F)F)=O)CCCC1n1cc(CCn2cncn2)nn1 96479,C1(CNCC(COC(C)=O)C)C2CC3CC(C2)CC1C3 96480,c1(C(=O)NC2(C)CC(NC(c3ccc(CO)o3)=O)C2)cnc2scnc2c1 96481,CC(CC(F)F)C(=O)NCCCOCCN(C(=O)Cc1sc(O)nc1O)C 96482,C(=O)(CCCCC(N)=O)NCC(S(C)(=O)=O)CNC(C1CC1C#N)=O 96483,Cc1cccc2ncc(C(N3CCC(C)CC3CNC(c3c[nH]c(=N)o3)=O)=O)n12 96484,C1(CNC(CC(=C)C)=O)CCC2(CO1)CC(NC(=O)C=CC1CCC1)C2 96485,N1(C(=O)OC(C)(C)C)CC(C(=O)Nc2ccc(Cc3cncs3)cc2)C2CC12 96486,CCCC(C)(CC)NC(C1(C(C)C)CCN(C(=O)CCc2cnco2)C1)=O 96487,C(C(CNC(=O)CCc1cncc(OC)c1)S(C)(=O)=O)NC(CCCC=C)=O 96488,C(=O)(C1CCCc2c[nH]nc21)NC1(CC=C)CN(C(=O)C(C)C(C)(C)C)C1 96489,Cn1nc(C(=O)NC2CC3(CCCN(c4nnn(C)n4)C3)C2)c2cc(F)ccc12 96490,C1(NC(C(c2cccs2)SC)=O)CC2(C1)CC(NC(=O)CC1CCC(F)(F)C1)C2 96491,c1(C(=O)NCC(CNC(c2c(CC)nc(C)[nH]2)=O)F)cc(O)cc(F)c1 96492,c1(C(=O)NCCNC(C2CCCN2CCN2CCCCC2=O)=O)cnc(S)nc1 96493,N1(C(CC2CCN(C(C(C)Oc3ccccc3)=O)C2)=O)CC2COC(=O)C2C1 96494,N1(C(C2(CNC(c3ccc(O)cc3)=O)CCCC2)=O)CCC(F)(F)C(O)C1 96495,N1(C(c2noc(CC)c2C)=O)Cc2occ(C(=O)NCCC3CC(F)(F)C3)c2C1 96496,Cc1cc(F)c2nc(O)cc(C(=O)NC3CCCN(CC(F)F)C3)c2c1 96497,c1(C(=O)NC2C(F)CCN(C(CCC(C)=O)=O)C2)ccc(Cl)c(C)c1F 96498,c1(C(=O)NC2CC(C)N(C(=O)CNC(C3CCCC3)=O)C2)csc2nccn12 96499,c1(C(=O)NC2CC(NC(C3CC3(F)F)=O)C(O)C2)cnc2c(F)cccn12 96500,N1(C(Cc2cc(CC)no2)=O)CCC(C2CC2)C1CNC(=O)C(=O)NCC(F)F 96501,c1(C(N2CCCCC(C(N3CC(CC)N(C)CC3)=O)C2)=O)cccc2[nH]ncc12 96502,C1(C(N2CCCC(CO)C2)=O)C2CCCC2CN1C(c1cn(CCO)nn1)=O 96503,C1(NC(CCc2n(C)ccc2)=O)CC2C(NC(C3CC(F)C(=O)N3)=O)C2C1 96504,C(C(C)(C)C(=O)N1CCC(C)C1)N(C(C1(CC(=O)OCC)CC1)=O)C 96505,c1(C(=O)NCC(=C)CCNC(=O)C(C)CCC)cccc([N+](=O)[O-])c1O 96506,c1(C(=O)NCC2CN(C(CC(C)NC(N)=O)=O)CC2O)onc2c1CCCC2 96507,c1(NC(C2C(NC(c3ccccn3)=O)C2)=O)ncc(F)cc1Br 96508,N1(C(CCC=C)=O)CCn2cc(C(N3CCCC4(CCO4)C3)=O)nc2C1 96509,N1(C(=O)NCc2nc(C3OCCO3)cs2)CCOc2c(F)cccc21 96510,N1(C(CN(C(C(C)Cc2ccccc2)=O)CO)=O)CCN(C2CCNC2=O)CC1 96511,C1(O)(CCNC(C(=O)NC(C)C)=O)CN(C(=O)C(C)CC2CCCCC2)C1 96512,N1(C(c2c(Cl)cnc(C)n2)=O)CC2(CCC2)CC1CNC(=O)CCc1cnco1 96513,C1(NC(c2cncs2)=O)CCC2(CC1)CN(C(c1ccoc1Cl)=O)CCO2 96514,c1(CNC(Cn2cc(C3(C)CC(OC)(OC)C3)nn2)=O)ccc2nsnc2c1 96515,n1(CC(N2CC(C(N)=O)(CNC(CC(C)CF)=O)C2)=O)nnc2c1CCCC2 96516,C1(SC)CN(C(=O)Cn2cnc(=N)[nH]2)CC1NC(C1(C)CCCO1)=O 96517,C12(CNC(C3N(C(C)C)CCC3)=O)CC1CN(C(c1cc(C3CC3)nn1C)=O)C2 96518,N1(CC2CCN(C(=O)COC3CCCCC3)C2)CC2C3C=CC(CC3)C2C1 96519,C#CCCCC(=O)N(CCCN(C(=O)C(C)(CN)NC(=O)NCCC)C)C 96520,C1(NC(C2N(CC)C(=O)CC2)=O)CCC2CC1CN2C(C1(C)CCN(C)C1=O)=O 96521,c1(C(N2C(CNC(=O)C=C(Cl)Cl)CC3(CC3)C2)=O)cc(O)nc2cnccc12 96522,C(=O)(CC(O)C(Cl)(Cl)Cl)N1CCC(OCC(=O)N(c2ccn(C)n2)CC)C1 96523,C1(CC(=O)NCCCCCCN(C(=O)C=Cc2cnccn2)C)CCC(=O)NC1=O 96524,O=C1CN(C(=O)CCc2nc(O)n[nH]2)C(C(=O)NC2CCC3(CC3)C2)CN1 96525,C(=O)(C1CSc2ccccc21)NC1C(NC(c2cccc(S(C)=O)c2)=O)CCC1 96526,C1(C(=O)OC)(OC)CN(S(=O)(=O)CCc2ccsc2)C1 96527,c1(OC)ccc(F)c(C(=O)NC2CC2CNC(=O)CCOC(C)CC(C)C)c1Cl 96528,C1(C(=O)OC)CCC(CC(=O)N(C)CCN(C)C(c2cccn2C)=O)CC1 96529,CC1(C(=O)NCCC2(O)CCN(C(=O)CC3CSC3)C2)CCC(F)(F)CC1 96530,C1(C)(CC(=O)NC2(CC(=O)NC3CC(OC)C3)CCC2)CCCCC1 96531,C1(C(=O)NC2C(CNC(C3(C(N)=O)CCC3)=O)C2)CCC2(CC1)CC2 96532,c1(-n2cc(C(C)N(C)C)nn2)ccccc1C(=O)N(C(C)CCO)C 96533,CCC(COC)(CC)CN=c1ccc(Br)c(S(=O)(=O)NCC)[nH]1 96534,C(C)(c1ccc(F)cc1F)=CC(=O)N(CC)CC1CCN(C(=O)C=CCF)CC1 96535,C#CCCCCC(=O)NCc1ccc(C(=O)NC(CCC)C(F)(F)F)nc1 96536,C12(C(=O)NCC3C(C)CN(C(C4CCC5(CC5)C4)=O)C3)CCC(CC1)OC2 96537,C1(OC)CC(C(=O)NCCn2ncn(C)c2=O)N(C(=O)CC2CC3(CCC3)C2)C1 96538,c1(OC)cc(F)c(Br)cc1S(=O)(=O)N1CCOCC1C 96539,N1(C(C2CC(C)=C(C)CC2)=O)CCC(C)(C)CC1C(=O)NCc1ccnc(O)c1 96540,C1(OC(C)C)CC(NC(c2ccc(OC(F)F)cn2)=O)C1(C)C 96541,c1(C(=O)NC2C(NC(C3(C#N)CCCO3)=O)COC2)cc2ccncc2s1 96542,S(=O)(=O)(CCCCF)N1CCN(C(C2(c3ccc(F)cc3)CC2)=O)CC1 96543,CC#CCC(C(=O)N(C(C)(C)CCCO)C1CC1)NC(=O)OC(C)(C)C 96544,c1(NC(=O)NCCCC(C)c2ccccc2)cc2cccnc2c(Br)n1 96545,N1(C(C2CC3CC2C2CC32)=O)CC2CCC1CN2C(C1CCCS1)=O 96546,C1(C(N(CCO)CC)=O)C2CCCC2CN1C(c1cnn2cccc2c1)=O 96547,N1(CCC(=O)NC(CC(C)NC(Cc2ccn(CC)n2)=O)C)CCN(C)CC1 96548,N1(C(c2n(CC)ncc2Cl)=O)CCC(C2CCN(C(=O)C(C)=C3CC3)C2)C1 96549,Cc1coc(C(C)C)c1C(=O)NCC1CN(C(=O)C(C)OCCC(C)C)CCO1 96550,N1(C(C2C(OC)CC2)=O)C2CCC1C(F)C(NC(=O)Cc1cnccn1)C2 96551,CC1C(=O)CCC(C(=O)NC2(CF)CCN(C(c3cscn3)=O)C2)C1(C)C 96552,c1(-c2ccc(C(=O)OC)c(F)c2)ccc2c(c1)OC(=O)CC2C 96553,CC1(C)C(NC(=O)C2=CCCC2)CCN1C(c1csc(Br)n1)=O 96554,Cc1ccc(C(=O)NCC(c2ccccc2)NC(=O)C(F)C2CCC2)c(F)c1F 96555,c1(C(C)CNC(=O)NCc2sncc2Br)cccc(C(F)(F)F)c1 96556,C(c1cnc[nH]1)=CC(=O)NCC(c1ccccc1)CNC(C12CC(CO1)C2)=O 96557,C(C(C)C(=O)NC1CCC1NC(=O)C(C)(C)C)OCC 96558,N1(C(C2CN(C(N)=O)C2)=O)CC(O)(CNC(=O)COC2CCOC2)C1 96559,Cc1ccc(C)n1CCC(N1CCC(N(C)C(c2ccc(F)cc2)=O)C1)=O 96560,c1(C(=O)NC(CC(C)C)CNC(C2CC2C#N)=O)c[nH]c2c(F)cccc12 96561,N1(C(CC=CCNC(=O)Cc2cccc(O)c2)=O)Cc2cccnc2C1 96562,N1(CCC(C(Cc2cn(CC(C)CC(=O)NC)nn2)(C)C)=O)CCn2nccc21 96563,C#CCCCC(=O)NC1CCC(CCNC(c2ccc(Cl)cc2)=O)C1 96564,c1(OCC)cc(C(=O)N(C2CCN(C(=O)C=C(C)C)C2)CCO)ncn1 96565,C1(NC(C(C(C)C)SC)=O)CN(C(c2nc(C)c(C)nc2C)=O)CC(F)(F)C1 96566,C1(OC)CC(NC(=O)CN2CC=CC2)CN(C(C2(CC(C)C)CC2)=O)C1 96567,C(=O)(C1CCc2cc(Cl)ccc21)NC1C2CN(C(COC(CC)C)=O)C1C2 96568,CS(=O)(=O)C(CNC(=O)Cc1cc[nH]c1)CNC(C1(F)CCOC1)=O 96569,O=C(CCCOc1cccnc1)NCC1CN(C(c2csc(CO)n2)=O)C1.CCO 96570,c1(C(=O)NCC(CNC(c2c(C)ccn2C)=O)C)cccc2[nH]cc(Cl)c12 96571,CC1(C)CC(CC(=O)NCC(=C2CN(C(C3(C4CC4)CC3)=O)C2)F)CO1 96572,Cc1cc(C(=O)NCCC2CCC(NC(c3ccc(Cl)c(F)c3)=O)C2)cc(O)n1 96573,N1(C(Cn2c(C)cnc2)=O)CCN(C(=O)CCCCC#N)CC1C 96574,C1(CNC(C2C(C)(C(C)C)C2)=O)C2CN(C(=O)CCc3c(N)cnn3C)CC12 96575,c1(C(=O)NCCCN(C(C2CC(C(C)C)OCC2)=O)C)c(F)cc(O)cc1F 96576,C(=O)(C(C)(C)CN(C)C)NC(CC)(C)CNC(=O)CC1COCC1O 96577,N1(C(c2csnn2)C)CCC(C2(NC(=O)CCC(C)(C)C)CC2)CC1 96578,C1(C(N(CCCOCCNC(c2ccc(C)cc2)=O)C)=O)CCC2(CCC2)C1 96579,n1(Cc2cc(C)no2)[nH]cc(C(=O)NC(CNC(=O)OC(C)(C)C)C2CC2)c1=O 96580,C1(CCNC(c2cccs2)=O)CN(C(=O)CC2C=CS(=O)(=O)C2)CCS1(=O)=O 96581,C12(CC)CC1CN(C(=O)CN(C(=O)Cn1cc(C3(O)CCCC3)nn1)C1CC1)C2 96582,Cn1c(C(N2CC(C)(C)C2c2ccncc2)=O)cnc1Cl 96583,C(=O)(C(C)CC(F)(F)F)N1CC(C)(C(=O)NCCCc2cc(C)no2)C(C)C1 96584,CC1(C)CC(C(N2CC3CCC3(CNC(=O)CSc3cn[nH]c3)C2)=O)C(C)(C)O1 96585,CCCC(C)CC(=O)NC(C)(C)CNC(C1SCCS1)=O 96586,N1(C(C(C(CC)CC)C)=O)CC(CNC(c2csc(CO)n2)=O)OC2(CCC2)C1 96587,C1(C(=O)NC(C(C)C)CNC(C2(S(N)(=O)=O)CCC2)=O)CC2(CCCCC2)CO1 96588,n1(CC)cnc(C(N2CC(O)(CCNC(=O)C=CC3CC3)C2)=O)c1 96589,c1(-c2nc(Cc3cc(C)nc(C)n3)nn2C(C)CN(C)C)nc2nc(C)ccn2n1 96590,N1(C(CN(CCCCC)C)=O)CC(NC(=O)COCCCCC)CCC1C 96591,C1(CNC(CCCC2C(C)C2)=O)CCCN(C(c2cn(C)nc2C(C)(C)C)=O)C1 96592,N1(C(c2cc(COC)sc2)=O)CC2CC1CN2C(=O)CC1CC2(CC2)C1 96593,CC1CCc2[nH]c(C(=O)NCCNC(C3(CCO)CC3)=O)cc2C1 96594,C(C(=O)N(OC)C(C)CC)C1CC(NC(CC2ON=C(CC)C2)=O)C1 96595,C1(NC(C2(CC#C)CC2)=O)(COC)CCN(C(c2ccc(CC)cc2O)=O)CC1 96596,c1(C(CC)NC(=O)COC(C)(C)CNC(c2cc(C)no2)=O)ccccn1 96597,c1(OCC(=O)NCCCNC(C(C)(C)CF)=O)ccc(Cl)c2ccccc12 96598,C(=O)(C(C(C)C)c1cc(C)no1)NC(CC(C)NC(C(C)=C(C)C)=O)C 96599,Cc1c[nH]cc(C(=O)NCCC2(O)CCN(C(c3ccc(Cl)cc3N)=O)C2)c1=O 96600,c1(SC)c(C(=O)N(C)CCN(C(C2CC2C2CCC2)=O)C(C)C)cccc1F 96601,CC1(C)C(CO)CN1C(=O)NCCC1OCCO1 96602,CCCCC(C(=O)NC1(C(=O)OC)CCC1)NC(C1CC1C(N)=O)=O 96603,N1(C(CCCC(C)=O)=O)CCCC2(C1)C(NC(c1cccs1)=O)CCN2C 96604,CCCCN=C(NCC(CC1CC1)CO)N1CCC(NC(c2ccccc2)=O)C1 96605,c1(C(=O)NC2CC(F)(CNC(c3cc(CC)nn3C)=O)C2)cc2ccccc2o1 96606,CC(C)CC(C)(CNC(C1CC(CF)C1)=O)NC(=O)CN1CCCCCC1 96607,C1(C(N(CC(=C)C)CC)=O)CC(CNC(=O)CCc2cn[nH]c2)C1 96608,N1(C(c2ncc(OC)cn2)=O)CCN(C(=O)C2=CCCSC2)C(CS(C)(=O)=O)C1 96609,c1(C(=O)NC(CNc2nccc(OCC)n2)C2CC2)[nH]c2ccc(F)cc2c1C 96610,c1(CCC(=O)NCCNC(=O)C(F)C2CC2)ccccc1O 96611,C1(C(N2CC(CCOC)C2)=O)CCC2CCC1N2C(=O)CCc1cn(C)cn1 96612,C#CCC(CC#C)C(=O)NC(C)(CC)CCNC(c1ccc(Br)c(C)n1)=O 96613,C(CCC(=O)NC(C)(CNC(C1(c2ccccc2)CC1)=O)C1CC1)OCCOC 96614,CCCC(C)(C)C(=O)NCC1CCCN1C(c1cnn(C2CCOCC2)c1)=O 96615,C(=O)(C(O)C(C(C)C)OC)N1C(C(=O)NC2CCN(C(CC)=O)C2)CC(F)(F)C1 96616,C(CO)(C(C)(C)CO)NC(C(C)CNC(=O)CCn1cccc1)=O 96617,N1(C(C=C(C)C)=O)CCCC(C(=O)NC(c2nncs2)C)CC1 96618,C1(C(=O)NCCCC(CCC)NC(=O)C(=O)NCC)COC2COCC2O1 96619,c1(C(=O)NC(CO)C(=O)Nc2ccc(OC(F)(F)F)cc2)c(F)ccc(Cl)c1F 96620,C1(C(=O)Nc2ccc(C)c(C)c2)(COC)CCN(C(=O)CC2CNC(=O)O2)CC1 96621,C1(CC(=O)NC2C(NC(c3c(C#N)ccs3)=O)COCC2)CCn2cncc2C1 96622,C1(F)(C(=O)NCC2C(NC(CC3(CSC)CC3)=O)CC2)CCN(C)CC1 96623,c1(C(=O)NCC2N(C(CC(C=C)C)=O)CC(F)C2)c[nH]c2cc(C)ccc12 96624,N1(C(CC2CC(=O)NC2=O)=O)CC(NC(=O)COCCCN(C)C)C2CCCC12 96625,c1(CC(=O)NCC(C)NC(C(c2ccc(Cl)s2)C)=O)cc2ccccc2c(=O)o1 96626,c1(OC)ncc(Br)cc1C(=O)NCC1(C)CN(Cc2csc(C)c2)C1 96627,Cc1ccccc1C(C)C(=O)NC1CCC1CNC(=O)CC1CC2CC2C1 96628,C1(NC(C(CC)Sc2ccccc2)=O)CCN(CC=C(C)C)CC1O 96629,c1(COC)nc(N2CCCC(C(C)NC(=O)C(=O)NCC(F)F)C2)cc(O)n1 96630,c1(C(N(CC(C)NC(=O)C(C)Cc2cnco2)C)=O)ncccc1N 96631,C12(NC(CS(=O)(=O)NC)=O)CCCCCC1N(C(=O)CCc1ccc(C)o1)CC2 96632,C1(C(=O)NCc2cc(C(N(C)CC3C(C)C3)=O)n(C)n2)CNC(=O)CC1C 96633,C1(COC(c2ccc(CNC3CCOC3=O)cc2)=O)CCN(C2CC2)CC1 96634,c1(NCC(c2ccccc2)(C)OC)ccc(S(=O)(=O)NCCS(C)(=O)=O)cc1Br 96635,C(C(C)(F)C(C)(C)F)NC(C(CNC(CN1C(C)CCC1)=O)O)=O 96636,CC1CC(NC(C2CC(F)(F)C2)=O)CCN1C(c1cc(CO)ccn1)=O 96637,N1(C(C2(SC)CC2)=O)CC2CN(C(C34C5CC(CC35)C4(F)F)=O)CC2C1CO 96638,N1(C(C(=O)NC2C(C)NCCC2)=O)CCOC2(CCS(=O)(=O)C2)C1 96639,CCC(CC)CC(=O)NC1CCCCC1NC(=O)C(C1CCCC1)OC 96640,c1(C(N(CCCC=C)Cc2ccccc2)=O)cn(CC2CCCO2)nn1 96641,C1(C(=O)NCc2cc(C)sc2)(NC(C2CCCN(C)C2)=O)CCN(C)C1 96642,c1(C(N(C(CCNC(C(C)NC(CC)=O)=O)C)C)=O)cnc(-c2ccccc2)[nH]1 96643,C1(C(=O)NCCOCCCNC(COCC(=O)NC)=O)CCCCN1C 96644,c1(C(=O)NCCC(C)N(C(CC(CC)O)=O)C)[nH]nc2ncnc(O)c12 96645,N1(C(C(CSC)C)=O)CCCCC1CC(=O)N(C(C)C(=O)NC1CC1)C 96646,N1(C(Cc2ncn(C)c2)=O)CC=C(C(=O)NCCC2CCCC3CC23)C1 96647,CC(CC(=O)N1CCCCC1C1(NC(=O)C(=Cc2c[nH]cn2)F)CC1)C(C)(C)C 96648,c1(N2CCC(C)C(F)(F)CC2)nc(=NCC2COCC2(C)C)[nH]c2c1CCCC2 96649,C(C(=O)N(C)Cc1ccncn1)(C(C)O)NC(c1c(CC)cco1)=O 96650,CC(C)CC(=O)NC(c1ccnn1C)C(=O)NC(C)CC(N)=O 96651,NC(=O)CC(O)C(=O)NCCC1(NC(=O)COC2CCCCC2)CCC1 96652,CC1CCn2ncc(C(N3CCC(C)C(NC(=O)C(F)C(C)(C)O)C3C)=O)c2C1 96653,C(=O)(C(F)(F)C1(O)CCC1)N(CCCCN(C(C(N1CC(C)C1)C)=O)C)C 96654,c1(C(=O)NCC(=C2CN(C(C3COCCO3)=O)C2)F)cnc2[nH]cnc2c1 96655,CCCCC(O)C(C)C(=O)NC1CC(N(C)C(c2c[nH]nc2Cl)=O)C1 96656,N1(C(CC(CC)C)=O)CC2CC(NC(C3CC(C)C3)=O)CC2C1 96657,c1(C(N2CC(C(C)NC(CCC(=O)NCC)=O)OCC2)=O)cc(Cl)c(N)c(Cl)c1 96658,C(N=c1nc2c(cnn2C)c(NCC2CCC2)[nH]1)C1(OC)CCCOC1.C1CCC1 96659,N1(C(C2(F)C(C)OCC2)=O)CC2(CCCCN(C(c3c[nH]nc3C3CC3)=O)C2)C1 96660,c1(N2CC3(C(CO)CN(C(C(CC)OCC)=O)C3)C2)cc(C)c([N+](=O)[O-])cc1F 96661,CC(CN=c1[nH]c(N2CCC(Cn3cccn3)C2)nc2ccc(Cl)cc12)N(C)C 96662,c1(C(N(CC(CNC(C2(CC)CCNC2=O)=O)O)C)=O)ccc2ncncc2c1 96663,c1(CN(CCC)C(=O)NC2(CC(F)F)CCCO2)c(C)noc1C 96664,c1(CCC)c(C(N2CC(NC(C3CN(C(C)=O)CCO3)=O)C(C)C2)=O)cnn1C 96665,Cc1cnc2ccc(C(N3CCC(C)C(CNC(C4(CCF)CC4)=O)C3)=O)cn12 96666,C1(NC(CCOCC)=O)CN(C(=O)CCC=CC(C)C)C2(CCOC2)C1 96667,N1(C(c2c(C)nccn2)=O)CCC2(CC1)CC(NC(=O)C1CCc3nccn31)C2 96668,C(=O)(C#CC1CCOCC1)N1CC(OCC)C(CNC(c2cc(SC)on2)=O)C1 96669,C1(NC(CC(C)=C(C)C)=O)CC2CN(C(=O)CCn3cnc(=N)[nH]3)CC2C1 96670,N#Cc1ccc(Cl)c(C(N2CCC(OCCNC(C3CCCS3)=O)CC2)=O)c1 96671,Cc1[nH]cc(C(=O)NCC2CC2NC(=O)CCC23CCC(CC2)C3)c(=O)c1Cl 96672,C12(c3nc(CCCOC)nn3-c3ccc(C)cc3)CSCC1C2(F)F 96673,Cc1ccc(C(C)(C)C(=O)NCC2(c3ccc(Cl)cc3)CC2(C)C)cn1 96674,CC1CCCCN1CC(=O)NC(CC1CCCC1)C(=O)N1CC(C)(C(F)(F)F)C1 96675,C(CN=c1nc(Cl)[nH]c(C)c1C#N)N(C(c1ccc(OC)cn1)=O)C 96676,N1(C(c2c(C)cn(C)c2)=O)CCCCC12CC(NC(C1CCCCS1)=O)C2 96677,Cc1cn2cc(C(=O)NCC3CN(C(C4OCCC4C(C)C)=O)C3)sc2n1 96678,C(=O)(C(C)(C)CC(=O)NC1CCCC1(C)CN(C(=O)C(C(C)C)SC)C)OC 96679,CCC(CC)(CO)C(=O)NCCOCCCN(C)C(c1cn(C)ccc1=O)=O 96680,C1(CC)COC(C)CN1C(=O)Nc1cccc(NC2CCS(=O)(=O)CC2)c1 96681,c1(Cc2scc(C(=O)NC(CN(C)C(C3CCS3(=O)=O)=O)(C)C)n2)ccccc1F 96682,N1(C(C(=O)NCCOCC)C2CCSC2)CCCC(C(=O)OC)C1C 96683,c1(C(=O)NC(CN(C(=O)CCC2CCCCO2)CC)C)cnc2[nH]nc(O)c2c1 96684,N1(C(C=C(CC)CC)=O)CC2CCCN(C(=O)CCc3c(C)nn(C)c3C)C2C1 96685,N1(C(C2(C=C)CCN(C(=O)CC(=O)OC)C2)=O)CCc2nc(O)[nH]c2C1 96686,C(=O)(C1=CCCOC1)N1C(CCNC(C2CC2(Cl)Cl)=O)CSCC1 96687,C1(C(=O)OCC(c2ccccc2)=O)CCCCC12CCC2 96688,c1(C(N2CCCC(NC(=O)CN3CCSCC3)CC2)=O)cc(F)cc2[nH]cnc12 96689,N1(C(C2=C(C)CC2)=O)CCN(C(=O)COC2CCCCCC2)C2COCC12 96690,Cc1cc(=NCC2(C)CC2(F)F)[nH]c(=NCCN2CCCC2)[nH]1 96691,c1(-c2cn(C3CCN(C(C4CCN(CC(C)C)C4)=O)C3)nn2)cc(F)ccc1F 96692,CN1CCC(C(=O)NC(C)(C)CN2CCN(C(C3(C)CC3(F)F)=O)CC2)C1=O 96693,C1(NC(Cc2ccc(OCC)cc2)=O)CC(C)CN(C(c2cscc2C#N)=O)C1 96694,N1(C(CCOCC#C)=O)CC2CCCC(N(C(=O)CN(C)C(=O)C3CC3)C)C2C1 96695,N1(C(CCNC(=O)NC)=O)CCC(CNC(c2ccc(C(N)=O)cc2)=O)C(C)C1 96696,C1(C(C)NC(C(F)(F)C2(OC)CCC2)=O)CCCN(C(=O)CC2CCCC2)C1 96697,c1(CC(=O)NC(CC)CN(C(=O)CN(S(=O)(=O)CC)C)C)cccc2c1OCO2 96698,C(=O)(C1=CCCC1C)NC1CCC(C(=O)NCC2CC(C(=O)OC)C2)C1 96699,c1(C(N2CCC(CCNC(C=COCC)=O)CC2)=O)oc2c(c1C)C(=O)CCC2 96700,n1(CCOCC=C)c(N2CCC(C)(C(=O)OC)C2)nnc1CO 96701,C1(C(=O)NC(c2ccccc2)CNC(C2C(=C)C2)=O)(CC)CCOCC1 96702,c1(C(N(C)CC2(NC(CSC)=O)CC2)=O)cnn(C2CCC2)c1 96703,c1(C(=O)NC2CC(CNC(C3CC34CCC4)=O)C2)cc(Br)cc2c1OCC2 96704,C1(CNC(CC(C)C2CC2)=O)CCCCN(C(C2CCCC(O)C2)=O)C1 96705,N1(C(CCCN(C(C)C)C)=O)CC(C)(C)CC1CNC(c1[nH]nnc1C1CC1)=O 96706,N1(C(c2cc(OC)ns2)=O)CCCCC1CCNC(=O)C=Cc1c(C)coc1C 96707,N1(N2CCCC(CNC(=O)COC3(C)CCC3)C2)CCC(C)CC1.CCC=O 96708,c1(-c2cccn(C)c2=O)ccc2[nH]cc(C(N3CCc4ccsc4C3)=O)c2c1 96709,c1(CC(=O)NC2CCCCC2NC(C2CC3C=CC2C3)=O)cccnc1Br 96710,C1(OC)CC2CC(C(=O)Nc3cccc(CNC(=O)C=CCF)c3)CC12 96711,c1(NC(c2ccncn2)=O)n[nH]c2cc(C(=O)NCCNC(C)=O)ccc12 96712,c1(-c2ccc(C(=O)NCC(C3CN(C(C=NOC)=O)C3)OC)s2)cccc(F)c1 96713,Cc1ccc2c(CC(N3CCC(O)(c4ccc(Br)cc4)C3)=O)c[nH]c2c1 96714,C(c1ccc(=N)[nH]c1)=CC(N1CC(C)(NC(c2ccn(CC)n2)=O)C1)=O 96715,C(=O)(C1=CC2CCC1C2)NC1C(CNC(CN2CCN(C)C(=O)C2)=O)CCCC1 96716,c1(-n2c(Cc3onc(C)n3)nc(C3CCC(C)CC3)n2)cccc2ccccc12 96717,c1(CNC(C(=O)NCc2cc(C(F)F)cc(F)c2)=O)cccc2c1OC(F)(F)O2 96718,n1(CCCC)cc(C(=O)N(CCN(C(=O)C(C)n2cccc2)CC)CC)c(C)n1 96719,C1(C(=O)NCCC2CCCC(C)C2)(NC(C2CC(CC)C2)=O)CC(F)(F)C1 96720,CCCC(CCC)CC(=O)NC(C)(CO)C(=O)NCC(O)C1(Cl)CC1 96721,CP(C)(=O)CCC(=O)N1CCCCC(CCC(=O)NC2CC3C=CC2C3)C1 96722,CCC(C)(F)C(=O)N(CCNC(=O)COC)CCOCCOc1ccncc1 96723,N1(C(CN(CCC)C)=O)CCC(CNC(=O)C(c2ccc(C)s2)C)C1 96724,c1(CCC(=O)NC2C(CNC(Cc3cc(C)sc3)=O)C2)cnc2ccccc2c1 96725,N1(C(CC2(C=C)CC2)=O)CCOCC(CNC(c2c(CC)cccc2C)=O)C1 96726,C(=O)(C1CC(=O)Nc2ncn(C)c21)N1C(C)CN(C(C2CCSCC2)=O)CC1 96727,c1(C(=O)NC2C(C)N(C(c3cnc(C4CC4)nc3O)=O)CC2)cc(Cl)cc(Cl)c1 96728,C1(CC(=O)NCCOC2CCN(C(=O)C(F)(F)c3nccs3)C2)CCNC(=O)C1 96729,c1(SC)ncc(C(=O)NC2(C)CCN(C(=O)C=CC3CC3)C2)c(O)n1 96730,c1(CC)ccc(C(N2CCC(C(=O)NCC3CCC(F)(F)C3)C2)=O)cc1 96731,N1(C(CN(C(C)=O)C)=O)CCCCC(CNc2ncc(C)c(C)n2)C1 96732,C(=O)(C1OCCn2ccnc21)NCCCN(C(C(CC)(C)O)=O)C 96733,C=CCCC(C(=O)NC1CC(CO)(CO)C1)NC(c1ccc(C)nn1)=O 96734,c1(C(C(=O)NCC2CCCO2)N(c2cnn(CC)c2)CC)cc2cc(Cl)ccc2s1 96735,CS(=O)(=O)c1cc(C(N2CCN(C(=O)C=CC3CCCO3)C(CCO)C2)=O)cs1 96736,c1(C(=O)NCC2(CCCNC(C=COC)=O)CCCC2)ccc(P(C)(C)=O)nc1 96737,N1(C(CCC(C)=O)=O)CC2CC(C1)N(C(c1cccc(C3CC3)c1)=O)C2 96738,c1(C(=O)NC2C(C)CN(C(c3ccc(C4CC4)s3)=O)C2)coc2c1CSC2 96739,N1(CC)CCCCC1C(=O)OC(C)C(=O)NCCNC(=O)N(C)C 96740,C=CC(C)(CCOC)C(=O)N(CC(C)C(=O)NC1C(C)C1(C)C)C 96741,c12ncsc1C(=O)N2CC(C)(C)C.C(=O)(C)OCC 96742,c1(N2CC=CC(NC(COC(CC)(C)C)=O)C2)cc(C)ncc1C#N 96743,C12(C(=O)NC(CNC(c3cc(C4CC4)no3)=O)C3CC3)CC(C1)C(C(F)(F)F)O2 96744,c1(C(N2CC(NC(CC=CCC)=O)CC2(C)C)=O)cnn2c1CC(C)CC2 96745,C#CCCCC(=O)NC1(CCNC(c2cc(C(F)(F)F)n[nH]2)=O)CC1 96746,CCC(C(=O)N(C(C)CCNC(c1cn(C)cn1)=O)C)NC(C)=O 96747,C1(CCNC(Cc2cc(CC)no2)=O)CCN(C(C23CC(O)C2C3)=O)CC1 96748,c1(OC)cc(C(=O)NC2CN(C(C3CCC4CC34)=O)CC2OC)ccc1C 96749,c1(C(=O)NC2C(NC(C(C)O)=O)C2)cc2ncccc2[nH]1 96750,C(=O)(C(CSC)c1ccccc1)NCCN(C(=O)C(C)(C)N(C)C)CCC 96751,C(=O)(CC1OCc2ccccc21)NCC(CNC(CCC=CC)=O)(C)O 96752,C1(C(=O)NCC2(C)CCN(C(C)=O)C2)CC2(CCOCC2)CN1 96753,N1(C(=O)C=C2CCOCC2)CCC2CN(C(C3(C4CCCO4)CC3)=O)CC2C1 96754,CC(C)CCCCC(=O)N1CCN(C(=O)CCCCc2cnn[nH]2)C2CC12 96755,C(=O)(C1CCc2nnc(C)n21)NCc1scc(CNC(C(CC=C)(C)C)=O)n1 96756,C1(NC(C2CCN(C(CNC(CC)=O)=O)C2)=O)CC12CCCCC2 96757,Cc1ccc(C=CC(N2CCC(O)(C(C)CNC(=O)CCc3ccco3)C2)=O)s1 96758,N1(C(CC2(N(C(C(c3cncnc3)C)=O)C)CC2)=O)CC(F)(CO)C1 96759,CCCCCC(O)CC(=O)NC(CCC)CC(N1Cc2ccccc2C1)=O 96760,C1(CCC)CN(C(=O)Cn2ccc(O)nc2=O)CCN1C(C1CCN(C)C1=O)=O 96761,C(=O)(C(O)CC(F)(F)F)NC(c1ccnn1C)C(=O)N(CC(C1CCCC1)O)C 96762,C(=O)(CCCCC(C)(C)OC)N1CCCCC(CNC(CS(CC)(=O)=O)=O)C1 96763,c1(-c2cc(C(=O)NC3CN(Cc4cccc(Cl)n4)C3)n[nH]2)ccc2c(c1)OCO2 96764,C(=O)(C1CCCc2nncn21)NC(CC)(CC)CCNC(C1CCCO1)=O 96765,CC1(C)CCCC(C(N2CCCC2CNC(C2(C(N)=O)CC2)=O)=O)C1 96766,CON(C(=O)C(C)=CCNC(C1CC1C1CCC1)=O)C1CCCC1 96767,C(=O)(C(C)(CC)C(=O)NCC1(CNC(C2CNC(=O)N2)=O)CC1(F)F)OCC 96768,C(=O)(C(CCc1ccc(F)cc1)C(C)(C)C)NCC1N(C(CC=C)=O)CC(O)C1 96769,n1(CC)cc(Cl)c(=NC(=O)N2CCCC2C2=CC=CC2)[nH]1 96770,C(=O)(CCC(C(C)C)NC(=O)C1=C(C)OCC1)N1CC=C(COC)CC1 96771,CCS(=O)(=O)CC(C)NC(=O)C(N1CCCC(C(F)(F)F)CC1)=O 96772,C1(CC(=O)N(C(C)C)CCN(C(=O)C=Cc2ccco2)C)CC2(CCC2)CCO1 96773,c1(C(=O)NCC2(NC(CC(CCC)O)=O)CCOC2)c2c(c[nH]c1=N)CCC2 96774,c1(C(N(CC(CNC(CC2C(CC)C2)=O)(C)C)CC)=O)cc(=O)cc[nH]1 96775,c1(OC)cccc(C(=O)NC(c2ccccc2)C(=O)NCCC(O)C(C)C)n1 96776,Cc1noc(C(=O)NCCC(C)N(C(=O)C(C)Cc2c(C)noc2C)C)c1C 96777,c1(NC(CC2CCN(C(C(N)=O)=O)C2)=O)cccnc1OC(F)F 96778,N1(C(CC2(OCC)CCC2)=O)CCOC(CNC(c2nnc(S)n2C)=O)C1 96779,C12(C(N3CC(Cn4cc(C(CC)O)nn4)OCC3)=O)CCCCC(=O)N1CCC2 96780,c1(OC)cc(C(=O)O)ccc1CNc1ccc(-c2nncs2)cc1 96781,C1(C(=O)NC(C(=O)NCCSC(F)F)C2CCCC2)CCC(O)C1 96782,C1(COC)(CNC(c2sccc2Cl)c2nnnn2Cc2ccccc2)CCCO1 96783,C1(Cn2cc(-c3ncc(C)s3)nn2)CCCN(C(C2CCC(=O)N2)=O)C1 96784,c1(CCNC(C(c2csnc2C)N(CCC)CCN(C)CC)=O)ccccc1Br 96785,CCCCCC(C)(CC)C(=O)N1CC2(CCC2NC(=O)CSC(F)(F)F)C1 96786,n1(-c2ccc(OC)cc2)[nH]nnc1=NCC(CN(C)C)C1CC1 96787,N1(C(CC)C(=O)NCCC(C)NC(=O)Cn2nnc(=N)[nH]2)CCN(CCO)CC1 96788,C1(C(=O)NC2C=CCN(C(c3cc(F)ccc3Cl)=O)C2)CCn2c(O)nnc2C1 96789,c1(CNC)cccc(N)c1.c1ccc(OC2CCCC2)nc1 96790,Cc1cc([N+](=O)[O-])c(S(=O)(=O)N2CCC(CCC3CCCCN3)C2)cc1F 96791,C1(CNC(c2c(OC)ccs2)=O)C(C)CCCN1C(c1cn(CCO)nc1C)=O 96792,c1(C(=O)NCC2(NC(=O)CCCN3CCCC3)CCC2)c[nH]c2nc(Cl)ccc12 96793,N1(C(C2(C)CN(C(CC(C)C)=O)C2)=O)CCOC(CN(C)C)C1 96794,N1(C(c2cc(CC)on2)=O)CCC(NC(C2(C)CCCOC2)=O)C(C(N)=O)C1 96795,C(=O)(CC(C(F)(F)F)N1CCOCC1)N(CC(C)NC(c1cc(Cl)ns1)=O)C 96796,CC1CCN(CC(=O)N(CCC(C)(C)NC(=O)C(F)CC2CCOC2)C)C1 96797,C=CC(C)(C)CC(=O)NC(C)CCN(C)C(c1cc(Cl)ncc1NC)=O 96798,C(CCC(=O)NCC1CC1C1CC(=C2CCC2)C1)OC(C)C.C12CCCN1C2.C1(=C)CCC1 96799,N1(C(CCc2cc(C)[nH]n2)=O)CCOCC1CN(C(=O)CSCC(F)(F)F)C 96800,Cn1ccnc1C(=O)NC(C(=O)NCC1(O)CCSC1)C1(C)CC1 96801,C(CCCC(=O)NCC#CCNC(=O)CSc1ccccc1)SC 96802,CC(O)C(C(=O)NCC=CBr)NC(C1CC(=O)C1(C)C)=O 96803,Cc1nc(N(C)CC2CCCN2C(=O)C(C)NC(=O)CC(C)(C)C)c(C)c(C)n1 96804,N1(C(c2ccc(C)c(F)c2)=O)CCC2(CC1)CC2(C)C(=O)N(C)CCN(C)C 96805,CC(C)(C(=O)NCC1CC(NC(=O)CN2CCCCS2(=O)=O)C1(C)C)C(F)F 96806,C1(CNC(CCC(C)(F)F)=O)CN(C(c2cnc3c[nH]nc3c2)=O)CCC1(C)C 96807,C1(OC)=NC=C1C(=O)N(CCn1cc(C(=O)O)cn1)CC1CCCO1 96808,c1(CC)ccc(C=CC(=O)NC2CCCN(C(=O)CN3CCCCC3)C2)cc1 96809,c1(C(N2C(CNC(N)=O)CCCC2)=O)ccc(OC)c(OCc2ccccc2)c1 96810,C(=O)(CC(C)(C)C(=O)N1CC(C(=O)NCC2(O)CN(C)C2)C(CC)C1)OCC 96811,C1(CNC(C(C)OCCOC)=O)CCC(C)(C)CN1Cc1cccc(C)c1 96812,CCCCN=C(NCCCc1cc2ccccc2[nH]1)NCC1CC(O)C1(C)C 96813,C1(c2cn(CC(COC)O)nn2)CCCN(C(C2CC3(CO)CC2C3)=O)CC1 96814,C(C)(C)(CCC(=O)N1CCCC(C(N2CCC(C)(C(N)=O)C2)=O)C1)OC 96815,N1(C(c2c(C#C)c[nH]n2)=O)CCC(F)CC1C(N1CCC(C)CC1)=O 96816,C(=O)(C(C)CC(F)(F)F)NC1(CC=C)CN(C(=O)C(COCC)N=[N+]=[N-])C1 96817,C=C(C)CCCC(=O)NCC(CCOC)NC(c1coc(C(C)OC)n1)=O 96818,CC1CN(CC(C)(C)O)CCN1C(=O)NCC1(C)CC=CCO1 96819,C(=O)(CC(C)CC(F)(F)F)NCC1N(C(c2cnc(SC)s2)=O)CC(O)C1O 96820,N1(C(C2C(CC)OCC2)=O)CC(C)(C)CCC1CNC(c1cc(C)nc(O)n1)=O 96821,C1(C)(C(N2CC(C)(NC(=O)CN3CCSCC3)C2)=O)C2Cc3ccccc3C12 96822,N1(C(c2cc(CC)on2)=O)CCC(NC(C2CCC(OC(C)=O)CC2)=O)C(CC)C1 96823,N1(C(c2cccc(C)c2C)=O)CC2CCC1(CNC(c1[nH]c(O)nc1C)=O)CC2 96824,c1(CC(N2CC(NC(CCOC)=O)C(C(F)F)C2)=O)ccc(OC(F)F)c(F)c1 96825,CC1(C)C2CC(C(=O)NC3(C)CCCC3NC(c3ncncc3Cl)=O)CC12 96826,c1(NCC2(C(C)(C)C)CCN(C(C(CC)OC(C)C)=O)C2)nc(CC)cc(C)n1 96827,N1(C(c2nccc(N)c2Cl)=O)CCC(NC(c2ncc(F)cn2)=O)C(CO)CC1 96828,C1(NC(C=C(COC)C)=O)COC2(C1)CN(C(c1cc3sc(C)nc3[nH]1)=O)C2 96829,C1(OC)(CNC(C23CC(F)(C2)C3)=O)CCN(C(c2c(Cl)sc(Cl)c2C)=O)CC1 96830,N1(C(c2cc(OC)ncn2)=O)CCN(C(=O)C(O)CC(C)C)C(C(F)F)C1 96831,c1(N2CCN(CCCC)CC2)nc(NCCC(C)F)nc2c1CCC2 96832,CCC(C)(C)C(C(=O)N(C)CC1(CNC(c2ncc3ccccn23)=O)CC1)OC 96833,Cc1ccc2nc(C)c(C(=O)NC3CCN(C(c4ncccc4Cl)=O)C3)cc2c1 96834,c1(NC)c(C(=O)NCCCNC(c2cc(F)c(F)c(F)c2)=O)sc2nccnc12 96835,N1(C(C(C)N(C)C(c2ccc(=O)n(C)n2)=O)=O)CCC(C2CCC2)C1 96836,C1(C(=O)NCC(CC(=O)NC(C)COC(F)(F)F)OC)CCCCCN1C 96837,C1(C)(CNC(C(C)NC(N)=O)=O)CCCN1C(C1CCOC(=O)N1)=O 96838,C1(NC(C=C(CCC)C)=O)CC2CC1N(C(=O)CC1(O)CCCCC1)C2 96839,c1(CC(C(N2C(CNC(c3cnc(C)[nH]3)=O)C=CC2)=O)C)cccc(Br)c1 96840,c1(NC(CC)COCC2CC2)ncc(S(=O)(=O)NC2CS(=O)(=O)CC2O)cc1Cl 96841,C#CC1(O)CC(C(N2CC(NC(c3scnc3C(C)C)=O)C(O)C2)=O)C1 96842,C(=O)(C1=COCCC1)N1C(CN(C(c2ccc(OC)nn2)=O)C)CCCC1 96843,CCC1=NOC(C(=O)NC23CC2CN(C(=O)CCOC2CCCC2)C3)C1 96844,Cc1cc(C(=O)NCCN2CCC(NC(C3(C4CC4)CCCO3)=O)CC2)ncn1 96845,CC1(C(N2CCN(C3CCCN(C(C4(C(N)=O)CC4)=O)C3)CC2)=O)CCNC1=O 96846,c1(C(=O)NCC(C2CCOC2)NC(c2n(C(C)C)nnc2)=O)cnc2n1CCC2 96847,N1(C(COc2ccc(C(C)=O)cc2)=O)CC(C2(NC(=O)CC#N)CC2)C1 96848,C1(NC(c2c(C)ccc(Cl)c2)=O)CCN(C)C12CCCN(C(C1(C)CC1Br)=O)C2 96849,c1(C(=O)NC2CC(CNC(c3c(CC)n(CC)nn3)=O)C2)cnc(O)n(C)c1=O 96850,C1(C)(NC(c2n(C(C)C)nnn2)C(C2CCOCC2)C)CCC(=O)N(C)C1 96851,CC1(C(=O)NCc2ccoc2C(=O)NC2CC(O)C2)CCC2CC2C1 96852,c1(CC(=O)NCC2(NC(=O)CNc3ccccc3)CC(F)(F)C2)ccc(O)cc1 96853,c1(C(=O)NCC(=C)CCNC(C23CCCCC2C3)=O)cc2c(cc1Cl)NC(=O)C2 96854,O(NC(=O)N(CCOc1nn[nH]n1)C)CC(=O)OCC(=O)N(C)C 96855,C1(C(=O)NC2C(NC(CC(C(C)C)O)=O)CC2)CC12C1CC3CC(C1)CC2C3 96856,C(=O)(C(C)(O)CCN(C)C)NCC(CCC)NC(c1cccc(C(F)F)c1)=O 96857,c1(OC(c2ccc(CC)o2)=O)cccc(C)c1C 96858,N1(C(Cc2c(C)noc2C)=O)C2CCC1(CNC(c1ccco1)=O)CC2 96859,c1(C(N2C(CNC(CC(=O)NCC)=O)CC(OC)C2)=O)cc2c(=O)[nH]ccn2n1 96860,c1(C(C(=O)N(CCNC(C(C)CO)=O)C)C)nc(F)ccc1Cl 96861,C1(C(=O)NCCCOC=C)C2CCCC2CN1C(=O)CN1CCCCC1=O 96862,N1(CC(=O)NC(C2CCCC2)CNC(C=CCOC)=O)CCC(C)C1 96863,c1(OC(C2C3CC(N)C(C3)C2)=O)c(Br)cc(Br)c2cccnc12 96864,Cc1cc(C(F)(F)F)nn1CC(=O)NC1CCCCC1N(C)C(c1ccc[nH]1)=O 96865,N1(C(CCCOCC)=O)CC2(CCN(C(=O)C(C)CCO)CC2)C1C(C)C 96866,CC1=C(C(=O)N2CC(NC(c3ccsc3CN)=O)C(C)C2)CCO1 96867,CCC(C(=O)NC1CC(C)(CNC(=O)C=CCOC(C)(C)C)C1)C1CC1 96868,N1(C(C2N(C)CCCC2)=O)CCC(C(F)(F)F)(NC(=O)C2=COCCC2)CC1 96869,c1(OC2(C(=O)OC3CCCCCC3)CC2)ccc(Br)cc1Br 96870,N1(C(CC(CCC)C)=O)CC(CNC(c2ccnnc2C)=O)OC(C)(C)C1 96871,Cc1ccc(C(N2CC(C(F)C(=O)N=c3ccn(CC)[nH]3)C2)=O)c2c1CCCC2 96872,c1(CC(=O)NCCCC2(NC(=O)Cc3ccncc3Cl)CC2)ccc(Cl)cn1 96873,CC(C)C(CCN(C(=O)CC1CCSC1)C)NC(=O)CC1CCC(=O)N1 96874,Cc1cc(=NCC2CCSC2(C)C)[nH]cc1S(=O)(=O)N1CCOC(CCO)C1 96875,Cc1c(NC(=O)N(C)CC2CCN(CC(F)F)CC2)cnn1C1CC1 96876,c1(CC(N2CC3(CNC(CC)=O)C(C(F)(F)F)(C2)C3)=O)ccc(S(C)(=O)=O)cc1 96877,CC1CCC(CCNC(=O)C(C2(C)CC2)NC(C2CNC(=O)O2)=O)O1 96878,Cc1nn(C)c2nc(C(=O)NCCN(C(=O)C(=O)NCC(F)F)C(C)C)ccc12 96879,C1(C(N(C2CNC(=O)C23CC3)C)=O)CCN(C(=O)CCC2(C)N=N2)O1 96880,CCC(CCC(=O)NC(CC(=O)NC)C1CC1)NC(=O)C(C)(C)n1cnnn1 96881,C12(C(N(CCNC(c3c(CC)nns3)=O)CC3CC3)=O)CC3CC(C(=O)N1)C2C3 96882,N1(C(C23CC(C)C2C3)=O)CCC2(CCC(NC(=O)C=C(Cl)Cl)CC2)C1 96883,CCCCCC(CC)C(=O)NC(C)C(C)(C)NC(c1ccc(CC)[nH]1)=O 96884,c1(CCC(=O)NC(C2N(C(c3cnc(SC)s3)=O)CCC2)C)ccnc(Cl)c1 96885,N1(CCCCNC(c2c(C)ccnn2)=O)CCCN(C(C2CCOC2C)=O)CC1 96886,N1(C(C(F)=CC)=O)CC(NC(=O)CC2COCCO2)CC2(CCC2)C1 96887,N1(C(C=C(CC)CC)=O)CCN(C(c2cnn(C)c2COC)=O)C(C)C1C 96888,c1(NC(c2n(CC(=C)C)nnn2)c2cc(CC)on2)cc(F)cc(F)c1 96889,N1(C(C2C3CN(C(C4C(C5(C)COC5)C4)=O)CC32)=O)CCCc2occc2C1 96890,c1(CC(=O)OC)ccc(C(=O)NCC(Cc2ccc(Cl)cc2)C(=O)O)cc1 96891,Cc1ccc(COONC(C2C=CCCN2C(c2ccn(C(C)C)n2)=O)=O)cn1 96892,C1(NC(c2c(Cl)cn(CC)n2)=O)(CC)CCN(C(=O)CSc2nccn2C)CC1 96893,C1(NC(c2cn[nH]c2)=O)CCOCC1NC(c1cc(-c2ccncc2)on1)=O 96894,C(=O)(CCC(CC)NC(=O)C1=C(Cl)CCC1)Nc1ccc(CC)nc1 96895,c1(OC)ccc(CCCC(=O)N2CC(C(C)NC(=O)CC3CC3)C2)cc1OC 96896,c1(OC(C)C(F)(F)F)ccccc1-n1cc(C2CCSCC2)nn1 96897,C(S(=O)(=O)CC(=O)NCCCNC(C1CC1C(C)(C)O)=O)c1cn(C)nc1 96898,c1(NCC(N2CCN(Cc3c(OC)c(Br)ccc3)CC2)=O)c(F)ccc(F)c1Cl 96899,C1(C)(C(=O)NC(c2nn[nH]n2)CC)CC(NC(=O)CC(C)=C(C)C)C1 96900,c1(C(=O)NCC=Cc2c(OC)cc(Br)cc2)c(Cl)ccc2c1OCO2 96901,N1(C(CCSC)=O)CC(NC(c2cc(-c3ccncc3)no2)=O)CC12CCOC2 96902,C1(NC(C2CCC(C)(C)O2)=O)CC2CN(C(c3ccnn3CC(F)F)=O)CC2C1 96903,c1(CC)cc2c(N3CCC(CF)(NC(c4cnsn4)=O)C3)nc(C)nc2s1 96904,c1(OC)nsc(C(C(=O)NC2CCCC2)N(c2ccccc2)C)c1Cl 96905,c1(CNC(c2n(C)nnn2)(C)CC2CCCOC2)cc(SC)n(C)n1 96906,c1(C(N2CCN(C(Cc3cncc(OC)c3)=O)C3C2C3)=O)cncc2sccc12 96907,C(=O)(C1CCCc2ncnn21)N1C2CC(CNC(C(C)N(CC)CC)=O)(OC2)C1 96908,C1(NC(C(CC)C)=O)CCN(C(=O)C(C2CCNCC2)F)CC1 96909,C(CO)(CCF)NC(CC=CCNC(=O)Cn1cncn1)=O 96910,C(=O)(C1CCOc2ccccc21)N(CCCN(C(C(CC(C)C)=O)=O)C)C 96911,c1(C(=O)NCC(CC)NC(c2ccccc2S(C)=O)=O)cccc(C#CCO)c1 96912,CC1(C)OC2(C(=O)NCC(C3CCCC3)NC(=O)CC3CCOCC3)CCC1C2 96913,N1(C(c2c(CC)nc[nH]2)=O)CC2(CCC2NC(c2cn3ccnc3s2)=O)C1 96914,S(=O)(=O)(C1CN(C(=O)OC(C)(C)C)C1)NC(C)CC1CCC(C)(C)CC1 96915,N#Cc1[nH]c(=NCCC2CCN(C(=O)C=Cc3ccco3)CC2)sc1Cl 96916,c1(N(C)CCOc2ccccn2)ccncc1S(=O)(=O)NCC1CC1(F)F 96917,C1(CNC(c2c(C)cnn2C)=O)CN(C(c2c(C)ncn2O)=O)CCC1C 96918,C1(NC(C2CCC(=C)CC2)=O)CCCN(C(=O)CCn2cnc(C)cc2=O)C1C 96919,c1(C(N(CC(C)NC(COCCCC)=O)C(C)C)=O)cnc(SCC)s1 96920,N1(C(CCC(CC)C)=O)CC2CC(C1)CN(C(=O)CCC1CNC(=O)N1)C2 96921,CC(C)C(C(=O)NC1CC(NC(=O)C(C)N(C)C)C1)N1CCCCC1 96922,C(CCN=C(NCC(c1ccc(C)cc1)(C)C)N1CC(C)C(C)C1)OCCOC 96923,C=C1CCN(C(=O)C(C2CCCO2)NC(c2cnn(CCO)c2)=O)C1 96924,O=C(C#CC1CCOC1)NC1CCOCC1NC(=O)Cc1nc2ncccn2n1 96925,c1(C(N2CCCC(C(C)NC(=O)CSc3ccncc3)C2)=O)cnc(Cl)cc1Cl 96926,c1(OC)cc(C(N2CCC(CC(=O)NC3CCCNC3=O)C2)=O)cc(C)c1 96927,c1(C(=O)NCC2(NC(c3ccc(F)s3)=O)CC2)cccc2cccnc12 96928,N1(C(CCC(c2cc(C)nnc2O)=O)=O)CC(C2CCCC2)C1.C123CC(C1)(C2)N3 96929,C1(O)(C(=O)NCC2C(NC(C(CCC)O)=O)CCCC2)CCc2ccccc2C1 96930,CC1CCN(C(=O)CCc2ccc(Cl)cc2F)CC1CNC(=O)CN(C)C(N)=O 96931,C1(CC(=O)NC2CC2c2ccccc2)CCN(Cc2ccccc2Br)CC1 96932,C(=O)(CS(=O)(=O)CCO)NC1C(C)CN(C(=O)CCc2cccc(Cl)c2)C1 96933,C(CC(C)(C)CC(=O)NC1CC(=C2CCC2)C1)OC 96934,C(N=c1[nH]c(=N)[nH]c(=NC2CCCCC2C(N)=O)[nH]1)c1ccc(SC)s1 96935,CC(CC(=O)N1CC(O)(CCNC(=O)CCCn2cccc2)C1)CC(F)(F)F 96936,CC1OCCCC1C(=O)N(C)CC=CC(=O)NC1(C2CC2)CC1 96937,c1(C(=O)NC2CC(CCNC(C=CC(C)C)=O)C2)cc2c(s1)CCS(=O)(=O)C2 96938,C(COCC(N1CC(NC(N)=O)C1)=O)(C(=O)N1CC(O)(C(F)(F)F)C1)N(C)C 96939,C1(C(=O)NC(c2nncs2)C)CN(C(C2CC2Cl)=O)CC12CCC2 96940,c1(CN(C(C2CCCN(CCCN(C)C)C2)=O)C2CC2)nnc2ccccn12 96941,c1(C(CC)C)ccc(C(C(=O)NCCC2(C)CC2)N(C2CCCCCC2)C)cc1 96942,N1(C(C(C)(C)OCC)=O)CCC(N(C(c2sccc2F)=O)CC)CC1 96943,Cc1cc([N+](=O)[O-])c(Cl)c(S(=O)(=O)NCC(O)COc2cccc(I)c2)c1 96944,C1(CC(N2CCCC2Cc2ccccn2)=O)CCc2ccccc2N1 96945,c1(C(N2CC(C(C)NC(C(CC)(C)C)=O)OCC2)=O)cc2sccc2[nH]1 96946,C1(CC(NOC(C=C)C)=O)CN(C(c2ccn(C3CC3)n2)=O)CC1C 96947,Cc1ccc(O)c(C(=O)N(C)CC2CC(F)CN2C(C2CN3CCC2CC3)=O)c1 96948,N1(C(c2n(CC)ncn2)=O)C2CCC1CC(N(C(=O)CN1CCCCCC1)C)C2 96949,C1(CC)CN(c2nnc(C(N(C)S(N)(=O)=O)(C)C)n2C)CC(C)O1 96950,C1(NC(CCC(=C)C)=O)CCN(C(c2coc(C(F)F)n2)=O)CCC1CO 96951,c1(C(=O)NCCN(C(C(C)=C2CCC2)=O)C(C)C)cccc2c(C)ccnc12 96952,C(CC(=O)NCC1CN(C(C)C)C1)(C(F)(F)F)NC(C=C(C)C)=O 96953,C(=O)(C1=Cc2ccccc2C1)N(CC(C)NC(CC(C)c1ccccc1)=O)C 96954,N1(C(C(CN(C)C)O)=O)CCC2C(C1)CN2C(c1cnn2cccnc12)=O 96955,C1(NC(C(CC)C)=O)CCCN(C(C2CC(O)(C#N)C2)=O)C1C 96956,C=CC(CCC)CC(=O)NC1(CF)CCN(C(c2nc(C)sc2C)=O)C1 96957,c1(C(=O)NC2CN(C(=O)C(O)Cc3ccccn3)CC2F)c(F)cc(F)cc1F 96958,N1(C(=O)CCc2nc(O)n[nH]2)CCC2CCN(C(C3CCCC(F)C3)=O)C2C1 96959,N1(C(c2n(CC#N)ncc2)=O)CCOC(CNC(c2ccnnc2)=O)C1 96960,O=C(C1=CCCC1)NCCc1ccc(Oc2cccnc2)cc1 96961,C1(CC)CN(C(C2CC2[N+](=O)[O-])=O)CCN1C(=O)C#CC1(C)CC1 96962,CCCS(=O)(=O)CC(=O)NCC1(CCNC(c2cncc(NCC)c2)=O)CC1 96963,N1(C(c2ccc(C)nn2)=O)CCC2CCN(C(=O)C(C)CCO)CC2C1 96964,C1(C(C)C)CN(C(=O)C(C(C)C)OC(N)=O)CCN1C(c1cccc(Cl)c1)=O 96965,c1(SCCC)cc(C(=O)NCCCCCNC(C2CCC(CN(C)C)C2)=O)no1 96966,Cc1ccnc(C(O)CNC(C2CCCN2C(=O)OC(C)(C)C)(C)C)c1 96967,N1(C(C(COC)O)=O)CCCC(NC(=O)C(O)CCc2ccccc2)C1C 96968,Cc1cc(Br)cc2c1C(NC(C1COC(C)CN1)=O)CC2 96969,C1(C(N2CC(=C(CNC(=O)Cc3ncc(Cl)s3)F)C2)=O)C2CCCCCCC12 96970,c1(C(N(C2CCCN(C(C3CC4(CCC4)CO3)=O)C2)CC)=O)cc2sccc2s1 96971,O=C1CSc2cc(C(N3CC4CCNCC(C4)C3)=O)ccc2N1 96972,Cc1cccc([N+](=O)[O-])c1NC(C1CC1C(=O)N=c1cc(C2CC2)[nH][nH]1)=O 96973,CCC(C)C(O)CC(=O)NC(C(=O)NC1CCCC1(C)N(C)C)C1CCOC1 96974,C1(C(=O)NC(CCCNC(C(C)SC(C)C)=O)C)Cc2ccncc2N1 96975,N1(C(C=CCOC)=O)CC2CCC(C1)N2C(=O)NCCCCl 96976,N1(c2ncnc(NC3CCN(CC)CC3C)c2C)Cc2c(n(C)[nH]c2=N)C1 96977,Cc1c(CNC23CCC(C(=O)NCc4cccnc4)(CC2)C3)ccnc1Cl 96978,C(C)(C)(CN(C)C)OCC(=O)N(C)CC1C(C)C1 96979,C1(C(N)=O)CC(F)CN1C(=O)CC1CCCC(NC(c2cnn[nH]2)=O)C1 96980,c1(CC)nc(-c2cnc(CCN(C)C(=O)OC(C)(C)C)[nH]2)n(CC)n1 96981,C1(OCC)CC2(C1)CC2C(=O)N(C(C)CN(C(=O)CCc1cccn1C)C)C 96982,c1(C(=O)Nc2cccc(CNC(c3cscn3)=O)c2)ncc2ccccn12 96983,CCC(C)(COC)CNC(c1ccsc1Cl)c1nnnn1-c1ccccc1 96984,C(=O)(C(F)CC(C)(C)NC(=O)CC(C)Oc1ccccc1)NC(C)CN1CCCC1 96985,Cc1ccc(O)c(C(=O)NCC2CC(NC(=O)CC3(O)CCC3)C23CCC3)c1 96986,C(=O)(CC(F)(F)CC(F)(F)F)N1CCC(n2cc(C(C)OCC)nn2)C1 96987,c1(C2(NC(CC3(C)CN(Cc4cnc(C(C)C)[nH]4)C3)=O)CC2)ccc(F)cc1 96988,N1(C(c2n(C)ncn2)=O)CC(NC(=O)Cc2ccc(Br)cc2Cl)CC(F)(F)C1 96989,C1(CCC(=O)NC2(C)CC(NC(c3ocnc3C(F)(F)F)=O)C2)NC(=O)NC1=O 96990,C=CC(C)CC(=O)NCCC1CCN(C(=O)CCCc2cc(C)no2)C1 96991,C1(CCC(C)C)CCCCN1C(=O)NCC1(N(C)C)COC1 96992,C#Cc1ccc(C(=O)NCC2(C)CN(C(=O)COCC=C)CC2C)cn1 96993,N1(C(C=CC(C)NC(c2ccc(CC)s2)=O)=O)CCCC1(C)CO 96994,c1(C(=O)NCC2(C(F)F)CCN(C(C(C)(C)C(N)=O)=O)C2)ccc2ccsc2c1 96995,CC(C)(C)CCC(F)C(=O)N1CC(C)(OCC(N2CCC3(CNC(=O)O3)C2)=O)C1 96996,CN(C)S(=O)(=O)N(C)CC(N1CC(NC(C2CC3CCCC23)=O)C1)=O 96997,C1(NC(c2ccc(C(F)F)nc2)=O)CCCC(CNC(C2CCCC23CC3)=O)C1 96998,CC1CCN(C(=O)C(F)(F)F)CC1C(=O)Oc1c(C(=O)OC(C)(C)C)cccc1 96999,c1(C(=O)NCCCC(C)NC(C2CCC(=O)N2)=O)ccnc(C(F)(F)F)c1F 97000,CCCCCC(O)C(=O)N1CCCC(CC(=O)NC(C)C(=O)OC)C1 97001,C1(NC(c2c(C)nc[nH]2)=O)C2CN(C(c3ccc(OCCF)cn3)=O)CC12 97002,N1(C(CCSCC(C)C)=O)CC(CNC(=O)CCNC(=O)NC2CC2)C2CC12 97003,C12(C(NOCC)=O)CCN(C(=O)CCc3ccccn3)CCC1C2 97004,c1(-n2ccc(C(=O)NC(C(C)NC(C3(O)CCC3)=O)CO)n2)cccc(C#N)c1 97005,C12CC3OCCC3N(C1)C2.C1(c2ncn(C)c2)CN(C(=O)NC(C)(C)C)CCO1 97006,c1(C(N2CCCC(C(N3CCCC34CC4)=O)C2)=O)cccc2c(O)ncnc12 97007,C=C(C)CC(C(=O)NCc1cn(CC(=O)N(c2cnn(C)c2)CC)nn1)OC 97008,C(=O)(C(C)(C)CCC(=O)NC1CCCCCC1NC(=O)C(O)CC(C)(C)C)OC 97009,c1(CNC(CCOCC)=O)ccc2c(c1)CCN(C(c1c[nH]c(=NC)o1)=O)C2 97010,O=C1CCCc2ccc(CNC(N3CC4(CCSCC4)C3CCO)=O)cc2N1 97011,c1(C(N(C2CN(C(c3cnn(-c4ccncc4)c3)=O)C2)C)=O)nscc1Br 97012,C1(C(N)=O)C2CCN(C(=O)C3=CCC(NC(=O)CC4CC4C4CC4)C3)CC12 97013,S(=O)(=O)(c1ccc(NCc2nc(Cl)ccc2Br)cc1Br)NC(CC)C(C)O 97014,Cc1[nH]ccc(=NC(=O)C2OCCC2Cn2cccn2)c1Cl 97015,c1(C(CNC(c2ccnc(Cl)c2)=O)NC(c2c(C)cco2)=O)ccc(F)cc1F 97016,Cn1cnnc1C(CO)NC(=O)CC1(NC(=O)CN2CCOC2=O)CC1 97017,c12ccc(C(F)(F)F)cc1[nH]c(=O)[nH]2.C12CCCC(C1)S2.CCOC 97018,C(CN=c1nc(-c2cc(Cl)cc(Cl)c2)[nH]o1)C1CN(C(C2(C)CCCS2)=O)C1 97019,c1(CC)cc(C(=O)N(C(CNC(c2nnc(COC)s2)=O)C2CC2)C)no1 97020,S(=O)(=O)(c1cccs1)NC(C(N1CCC(NC(c2cc(CC)no2)=O)C1)=O)C 97021,c1(CNC(=O)CC2CC(F)C2)n[nH]cc1C(=O)NCC#CC1CC1 97022,C(C(C(=O)NCC1(CO)CCC1)NC(=O)C(C)CC1CCC1)OCC 97023,c1(C(=O)NCCC2N(C(C(C)C(F)F)=O)CCC2)csc2ccc(F)cc12 97024,N1(C(c2c(CC)noc2)=O)CC(C2CCN(C(c3ccnn3C3CC3)=O)CC2)C1 97025,N1(C(CCSC)=O)CCC(OCCNC(C2CC(C)(F)C2)=O)C1 97026,Cn1cnnc1SCC(=O)NCC1(F)CC(NC(C2(CO)CC2)=O)C1 97027,C(=O)(C(=O)NNC(=O)C(C)(C)C)NCCCOCCC(C)C 97028,C1(C)(C(N(CC(C)O)CCNC(C2(CCCC)CCC2)=O)=O)CCOC1 97029,N1(C(C(CC)N(C)C(c2ccc(O)cc2)=O)=O)CC2(CCC(=O)O2)C1 97030,c1(OC)ncccc1C(=O)NC(C)CNC(c1[nH]c(C2CC2)nc1C)=O 97031,CCC(CC(=O)NCC(C)(F)CNC(=O)CCc1csnn1)C(F)F 97032,C1(C(N2CC(CC(CNC(C(C)C)=O)(C)C)C2)=O)CCCN(c2cn[nH]c2)C1 97033,Nc1cccc(C(=O)NCCC2CCC(NC(=O)CC(C3CC3)C3CC3)C2)c1F 97034,n1(CC=C)cccc1C(=O)NC1CC(N(C)C(c2ccc(C(F)(F)F)s2)=O)C1 97035,N1(C(CSCC(C)C)=O)CCCCC(NC(C2COC2)=O)C1 97036,c1(C(C(=O)NC(c2cn(-c3cccc(F)c3)nn2)C)(F)F)cccc(F)c1F 97037,c1(C(=O)NCC(c2cccs2)C)cc(CCNC(=O)CC2CCCC2C)on1 97038,Cc1ccc(=O)n(CC(=O)NC2CC(C)(NC(C3CC(CF)C3)=O)C2)n1 97039,c1(C(=O)NC2CN(C(CC(C(C)C)O)=O)C(CO)C2)cc2ccccc2o1 97040,C=CCC(CC=C)C(=O)N1CCN(C(=O)CC2CC(=O)NC2=O)CC1CF 97041,Cc1cc(Br)cnc1CNC1CCN(C(c2cncnc2C2CC2)=O)C1 97042,C1(CNC(C(C2CC2)OC)=O)CN(C(=O)C(C(C)C)NC(=O)CC(C)C)CC1C 97043,C1(C)(SCc2nc(C34CC(C)(C3)OC43CCC3)on2)CCc2ccccc2O1 97044,CC(C#N)CCC(=O)N1CCC(CNC(=O)CCC2CCCCC2)CC1 97045,C(=O)(C1=CCCCC1)NCCCCC1CN(C(C2(OC(C)C)CCC2)=O)C1 97046,C(=O)(C(CC)C(F)(F)F)NCC(CC(=O)NC(C#C)(CC)CC)C 97047,N1(C(CC(CCC)NC(=O)C2CC2)=O)CCCC12CCOCC2 97048,N1(C(CCc2cnc(C)o2)=O)CC2C(CN(C(=O)C(C3CCOCC3)O)C)C2C1 97049,C12(NC(C(C3CCC3)OC)=O)CC(CNC(C3CCN(C)C3C)=O)(C1)OC2(C)C 97050,C1(NC(c2cnc(OCCO)cn2)=O)CCCN(C(=O)COCCO)C1 97051,C(C(O)CC(F)(F)F)NC(CC1CN(C(CCOC)=O)C(C)C1)=O 97052,C1(NC(COC(C)C)=O)CCC(N(C(=O)CCNC(=O)OC(C)(C)C)C)CC1 97053,c1(C(=O)NC(CC(C)NC(C=C(C)C(F)F)=O)C)cc(Br)c2[nH]c(C)nc2c1 97054,C(CCC(O)C(=O)N1CCOC(C2CC2)CC1)NC(C1(C)CCSCC1)=O 97055,Cc1c(C(=O)NCCCNC(=O)C(C)c2ccco2)c(C)n2ccncc12 97056,c1(SCCC)ccc(C(N2CC3(NC(=O)C(C(=O)OC)OC)CC2C3)=O)cc1 97057,c1(C(=O)NCC2CCCC(NC(c3c(OC)nsc3)=O)C2)cccc2sccc12 97058,C1(N(CC(=O)N(C)CC2CC(C)C2)CC2(CC(C)C)CC2)CC2CC2C1 97059,C1(CC(=O)N(CCCNC(C2CCN2S(C)(=O)=O)=O)CC)CC(C2CC2)C1 97060,c1(C(N2CCCC(C(F)F)C2)C(=O)NCc2nccs2)cc2cc(Br)ccc2o1 97061,c1(NC2CC(C)N(C(=O)C3=CCC3)C2)c(C#N)nnc2ccccc12 97062,C(CC(C)(C)C(=O)N1CC(CC(=O)N(C)CC2CC(F)(F)C2)C2(CC2)C1)OC 97063,C1(N(C(c2c(C)nsc2)=O)C)CN(C(c2cn(C3CC3)nc2C)=O)CC12CC2 97064,N1(C(c2c(C)ccs2)=O)CCC(C)C(NC(=O)CCOc2ccc(F)cc2)C1 97065,C1(CNC(c2c(CC)onc2)=O)CCCC2(CN(C(c3cnnn3C)=O)C2)O1 97066,C1(C(=O)NCCOC)CCN(C(=O)Nc2cn(C)nc2C(F)(F)F)CC1 97067,N1(C(C2(CCOCC)CCC2)=O)CCC12CN(C(c1c[nH]c(C(N)=O)c1)=O)C2 97068,c1(C(=O)NC2(c3cnccn3)CCC2)nccc2nc[nH]c12.C12CC1CNC2=O 97069,CC1CC(=O)NCCN1C(C1C2CCC(C2)N1C(=O)C=Cc1ccsc1)=O 97070,c1(NC(=O)NCCNC(N2C(C)(CC(=O)O)CC2)=O)ccc(Cl)nc1 97071,O=C1CCNc2cc(C(N3CC4C(NC(=O)C(F)(F)C(F)F)C4C3)=O)ccc2N1 97072,N1(C(C2C(C3CN(C(C(CC)OC)=O)C3)C2)=O)CCC2(CNC(=O)N2)C1 97073,C1(CC)CN(C(C2CN(C)C2)=O)CCN1Cc1c(C)cccc1O 97074,N1(C(CCC=CCC=C)=O)CC(NC(=O)CC(C)c2cnn(C)c2)C(CO)C1 97075,c1(C(N2CCN(C(CN(CC)CC)=O)CC2C(C)C)=O)onc2cc(C)ccc12 97076,N#CCCCC(=O)NCC(O)CNC(c1cnc(C(c2ccccc2)=O)cn1)=O 97077,C1(C)(OC)CCN(C(C(C)NC2CCCCC2)=O)C1.C12CCCN(C1)C2=O 97078,c1(C(=O)NC2CC=C(C(=O)NC(=O)C=Cc3ccco3)C2)cc2cccnc2[nH]1 97079,C1(C(N(C2CC2)CC)=O)CCN(C(C2(CSC)CCOC2)=O)C1 97080,Cn1cc(NC(=O)C(CNC(=O)CCC(N)=O)N(C)C)c(C(N)=O)n1 97081,CCCCC(O)CC(=O)NC1CN(C(c2c(F)cc(N)cc2F)=O)CC2(CC2)C1 97082,N1(C(C=CC)=O)CC2CCC(C1)N(C(c1cnn(-c3cccc(F)c3)c1N)=O)C2 97083,NC12CCC1CN(CC(=O)NCc1ccn(-c3ccc(Br)cc3)n1)C2 97084,C1(CNC(C2CC(=O)N(C3CC3)C2)=O)CC(O)CN1C(=O)Cc1csc(S)n1 97085,C(=O)(CC(C)(C)C=C)NC(CC=C)CNC(=O)C(c1cccc(F)c1)O 97086,c1(C(N(C2CCN(C(c3nccnc3N)=O)C2)C)=O)n[nH]c2c1COCC2 97087,O=C1Nc2cccc(-c3ccc(F)c4c3CCC4)c2CO1 97088,C(=O)(C1=CCC(NC(C2CC3CC2CC3O)=O)C1)NCCCC1(C)CC1 97089,N1(C(c2ccc(CNC(CC(C=C)C)=O)nc2)=O)CCC(N(C)C)C(C)C1 97090,c1(C(N(CCN(C(C=C(C)c2ccsc2)=O)C)C)=O)cc(C)n(C)c1C 97091,C(CC)(CC)(CCNC(c1[nH]cnc1C)=O)NC(c1c(CC)cco1)=O 97092,Cc1cc(C(=O)NCCCNC(C2CCCOC2C)=O)cnc1C(F)(F)F 97093,c1(OC)cc(OC)c(C(N2CCC(NC(C3CCC3(F)F)=O)C2C)=O)cn1 97094,C(CCCCC(=O)Nc1cnc(NCc2cncc(Cl)c2)cn1)N(C)C 97095,c1(C(=O)NCCC(CNC(C=CS(C)=O)=O)O)cc(F)c(N)c(F)c1 97096,C(C)(CC(C)(C)CO)NC(C(CCOC)NC(C(CC)C#N)=O)=O 97097,c1(-c2cccc(OC)c2)[nH]c(=NCC2COCCN2C(C)=O)sc1C 97098,N1(C(C2C(CC)CCCC2)=O)CCC(NC(=O)C2=CCCC2)C(C)(C)C1 97099,c1(C(=O)NC2(C)CC(NC(C(CO)N(C)C)=O)C2)cccc(F)c1Br 97100,CC1(NC(c2coc(CNC(=O)CCn3cncn3)c2)=O)CCOC1C1CC1 97101,N1(C(C(COC)OC)=O)CCOC(CN(C)C(c2ccccc2)c2cc(C)on2)C1 97102,c1(OC)cc(C(=O)O)ccc1OCC1CCCC(N(C)C)C1 97103,c1(C(N2CCC(C)(NC(CCSC)=O)CC2)=O)ccc2cn(C(F)F)nc2c1 97104,C=CC1CCCN(C(C)=O)C1.c12ccc(cc1Cl)NC(=O)CCCn1cc-2nn1 97105,N1(C(CCCC#N)=O)CCN(C(C2CC(c3cccc(F)c3)C2)=O)CC1C(F)F 97106,c1(CC)sc(C(=O)NCC(C)(C)CNC(c2ccc(C(=O)OC)nc2)=O)cc1C 97107,N1(C(C(C)CN(C)C)=O)CCC2(CCC(NC(c3cnc4sccn34)=O)CC2)C1 97108,CCC(C)CCC(=O)NCCC1CC(NC(c2sccc2OC)=O)C1 97109,C12(CNC(c3c(C)nc(O)[nH]3)=O)CCCCC1N(C(=O)Cn1ccnc1C)CC2 97110,c1(OC)cc(N2CCN(CC3CCC(NN4CCCCC4C)C3)CC2)nc(C)n1 97111,C1(NC(=O)C(c2ccccc2)F)COC2(C1)CN(C(c1scnc1Cl)=O)C2 97112,N1(C(CC2(C)CN(Cc3ccc(OC)nc3)C2)=O)Cc2cccc(F)c2C1 97113,N1(C(C2(SC)CCC2)=O)CC(CNC(c2cc3nc(C)sc3[nH]2)=O)OC(C)(C)C1 97114,C(=O)(C1CCCc2nncn21)NC(C1(O)CN(C(c2csc(C3CC3)n2)=O)C1)C 97115,C(=O)(CCC(=O)NN(C)C)N1C(CN(C(C2C(CN(C)C)C2)=O)C)CCC1 97116,N1(C(c2cc(C(C)(C)O)on2)=O)CCN(C(C2CSCCS2)=O)C2COCC12 97117,c1(C(=O)NC2CC3(CC(NC(=O)COCCF)C3)C2)cncc2ccc(F)cc12 97118,C1(C)(CNC(C2CCN(CC)C2)=O)CCCC1NC(=O)C(F)=C(C)C1CC1 97119,C1(NCc2cn(C(C)(C)C(=O)O)nn2)CN(C(c2cnncc2O)=O)CCO1 97120,C1(NC(c2cnc(C)[nH]2)=O)CCCCC1NC(=O)COCCc1cccc(F)c1 97121,CC1CN(C(=O)C=Cc2ccccc2Cl)CC(=O)N1 97122,c1(C(=O)NC(CC(C)NC(C=CC=CC)=O)C)cc(O)n(C)n1 97123,C(=O)(Nn1cnn(C)c1=S)C1N(C(CCNC(=O)NC)=O)CCC1 97124,c1(C(N2CC(C(C)NC(C=C(C)C(C)(C)C)=O)OCC2)=O)c(C)nn(C)c1C 97125,N1(C(c2c(C)nn(C)c2)=O)CCOC2CN(C(=O)CC3CC3C(F)(F)F)CC12 97126,C=CC1(C(=O)NCC(C2CC2)N(C)C(c2cccc(F)c2)=O)CCCCC1 97127,c1(CC(=O)NCC2C(NC(c3n(C)ncc3)=O)CCC2)ccc(Cl)cn1 97128,N1(C(C=C(CCC)C)=O)CC(CNC(c2cnc3cc[nH]c3c2)=O)C2(CCC2)C1 97129,C1(C(=O)NCCCN(C(=O)C(c2ccc(F)cc2)(F)F)C)CCCC(F)C1 97130,C=CC(C)(C)CC(=O)NCC(O)CC(=O)NC(C1CCCC1O)C 97131,c1(C(=O)NCCNC(c2cnnn2-c2ccccc2)=O)snc(O)c1Cl 97132,c1(C(N2CCC(C)(CCNC(C(CSC)C)=O)C2)=O)ccnc2ccsc12 97133,c1(CNCC(C(C)C)NC)c(F)ccc(Br)c1OCc1ccccc1 97134,C1(NC(CCCC(C)=O)=O)CCC2(CCCN(C(C3(S(N)(=O)=O)CC3)=O)C2)C1 97135,Cc1nc(C(=O)NCC(=O)NC(C(=O)O)C(C)C)[nH]c1C 97136,C1(C(=O)NCC(C#C)OC)CC(NC(=O)CCCC=CC)CCO1 97137,C12(C(=O)NC3(C4N(C(c5cnc(Cl)s5)=O)CCCC4)CC3)COCC1C2(F)F 97138,c1(CCCC(=O)NCCCN(C(C(C)OC)=O)C)nc2ccccc2s1 97139,CC1=C(C(=O)N2CC(NC(=O)C(C)S(C)(=O)=O)C3(CCC3)C2)COCC1 97140,CC1=NS(=O)(=O)N(C)C=C1C(=O)NCC1C=CC(NC(=O)C(C)CC2CC2)C1 97141,C1(C(N)=O)CCC2CCC1N2C(=O)CSCC(=O)NC1COC(C2CC2)C1 97142,C1(CNC(CS(=O)(=O)NCC)=O)CN(C(C2CC(=C3CC3)C2)=O)C(C)(C)C1 97143,c1(CC(n2cc(-c3n(CCOC)ncc3)nn2)C)ccc(C(C)C)cc1 97144,N1(C(C(CC)CC)=O)CC(C)(C)C(NC(=O)CC2CCOC(CC)C2)C(C)(C)C1 97145,CCCCCCC(O)CNc1cccc(C(F)(F)C(F)(F)F)c1 97146,N1(C(c2c(C)cc(SC)o2)=O)CC2CCC1CC2NC(=O)C(C)C 97147,c1(C(CCOC)NC(C2(c3ccccc3)CC2(Cl)Cl)=O)ccc(C)cc1 97148,C1(CNC(CN(C(C)C)C)=O)CN(C(=O)C(C)Oc2ccccc2Cl)C(C)(C)C1 97149,c1(C(=O)NC(C2CCOC2)CNC(c2ccc[nH]2)=O)cc2c(s1)CCCC2 97150,c1(C(N2CC3C(CCNC(CCC(N)=O)=O)(CC3)C2)=O)cc2c(s1)CCCC2 97151,C(C(CC(C)(C)C(=O)OC)NC(=O)NCCC1(n2nccn2)CC1)OC 97152,N1(C(C(CCC)OC)=O)CCCN(C(c2nc(C)ccc2OCC)=O)C(C)C1 97153,c1(C(C(=O)NCC(C)N(C(C2CCCO2)=O)CC)(C)C)cccc2ccccc12 97154,c1(C(N2C(C)C(NC(C3CC3F)=O)CC2)=O)cc2c(cc1[N+](=O)[O-])OCCCO2 97155,Cc1cc(N)cnc1C(=O)NC1CC2CC(NC(=O)CC3CCCCO3)C1C2 97156,N1(C(C(C2CCCC2)OCC)=O)CC2CCC1CN2C(=O)C(c1ccccc1)O 97157,c1(C(=O)NC2C=CCN(C(C(CC(C)C)C)=O)C2)cc2cccc(F)c2s1 97158,c1(CC(=O)NCCN(C(=O)OC)C)ccc(C)c(Br)c1 97159,C1(C(=O)NCC(=C)C)(CNC(=O)CCc2conc2C)CCCCC1 97160,c1(C(N2CC(F)CC(NC(C3(C)CC3)=O)C2)=O)ccc2c(c1)OCO2 97161,C1(C(N2CC(NC(N)=O)C2)=O)(OC)CCN(C(=O)C(Cl)Cl)C1 97162,c1(OC)cccc2c1CN(C(C1CN(C(c3ncccn3)=O)CCC1O)=O)C2 97163,C(=O)(C1Cc2ccc(Cl)cc21)NC1(CO)CCCN(C(c2c(CC)cno2)=O)C1 97164,CC1(C)CCC(C(=O)NCC2=CCCC2)OC1 97165,Cc1cc2ccc(C(N3CCC(NC(=O)C(C)C4CC4)C(F)C3)=O)cn2c1 97166,C1(C(C)NC(=O)CCc2cncn2C)CCN(C(c2ccccc2F)=O)CC1 97167,c1(C(C(=O)NC(C)C(=O)OC)N(CC(CC)C)CC)ccc2c(c1)oc(=O)n2C 97168,Cc1nc(CC(=O)NC2CCN(C(C3CC(C)(F)C3)=O)C2C2CC2)[nH]c1C 97169,Cc1ccn2ncc(C(=O)NC3(C)CCCN(C(C4CCS(=O)CC4)=O)C3)c2n1 97170,c1(C(=O)NC2C(CNC(C(C)OCCCC)=O)CC2)cccc2nccnc12 97171,C1(CNC(=O)CC2CCCCC2)CCN(C(C2C3CCCC23)=O)CC1O 97172,N1(C(C=CC(CC)=CC)=O)CCC(NC(c2cc(C)[nH]n2)=O)CC1C 97173,c1(C(N2CCC(C3N(C(=O)OC(C)(C)C)CCC3)C2)=O)ccc(F)c(Cl)c1 97174,Cc1cccc(C(n2cc(-c3cncc(F)c3)nn2)CCO)c1.C(=O)CC1CC1F 97175,C1(CCNC(CC=C=C)=O)CCCN(C(c2cncc(N)n2)=O)CC1 97176,C12(C(=O)NC3(CC#C)CCC3)CCC(CN(C(=O)C(C)(O)C3CCC3)C1)C2 97177,Cc1cc(Cl)c(C(=O)NC2CC(C)N(C(C3CC(CF)C3)=O)C2)s1 97178,c1(C(=O)NCCN(C(=O)COC2CCCC(C)C2)CC)cncc2[nH]ccc12 97179,C1(CC(=O)NC2CC2)CCC(C2CC2)O1.C12CCN(C1)C(=O)N2 97180,CC1CN(C(=O)CSc2ccc(Cl)cc2)CCCN1C(c1cnn(C(F)F)c1)=O 97181,c12ccccc1OC2.C(C)(C(=O)N(C)CCOCCCN(C)C)OC.C1(=O)CO1 97182,c1(CNC(=O)NC2CC(C)SC2)ccccc1C(F)F 97183,N1(C(CNC(c2cccnc2)=O)=O)CCn2ncc(C(N3CC(F)C(F)C3)=O)c2C1 97184,N1(C(C2C(CC)CC2)=O)CCC2CCC(C1)N2C(c1cc(OC)c(N)c(N)c1)=O 97185,C1(NC(C(CCOC)C)=O)C2CCN(C(=O)C(C)(C)COC(C)C)CC12 97186,C1(C(=O)NCC2(CN(C)C(c3cc(C#N)cs3)=O)CC2)CCc2ccccc2C1 97187,C1(NC(c2ccoc2)=O)CN(C(=O)Cc2ccns2)CCC12CCOCC2 97188,C1(C(CNC(C(CC)n2ccnc2)=O)C)CCN(C(=O)Cn2nnc(C)n2)CC1 97189,N1(C(c2[nH]ccc2CNC(C2(O)CCOC2)=O)=O)CCC2CCC(C2)C1 97190,c1(NC(=O)NC(C(=O)OCC)CSC)cc(C(F)(F)F)cc(S(N)(=O)=O)c1 97191,C12(C(N(CCO)CC)=O)CC(CO)(CN1C(C1CCCCCCC1)=O)C2 97192,c1(C(=O)NC2C(=O)N(c3cccc(Br)c3)CC2)cc(I)c(Cl)cc1Cl 97193,c1(C(=O)NC2C(NC(C(C)OCC#C)=O)CC2)cc(N)ccc1O 97194,CC(CN(C)C(=O)OC(C)(C)C)C(=O)NCC1CCC1NC(c1coc(O)n1)=O 97195,Cc1cc2c(cc1C)C(NC(c1ccc(N3CCN(C)C3=O)cc1)=O)CCS2 97196,C(=O)(C1=C(C)N(C)c2nnnn2C1C)NCCN(C(C(CC)OCC)=O)CC 97197,N1(C(C(C)C2CC2)=O)CCOC2(CCN(C(c3csc(C(C)(C)C)n3)=O)C2)C1 97198,c1(C(=O)NCC(CC(=O)Nc2c(OC)nn(C)c2)OC)cc(C)cc(O)n1 97199,c1(CC(=O)NCC2N(C(C34CC(OC)C3C4)=O)CCC(C)C2)c[nH]c2cccnc12 97200,c1(CC(=O)N(CCC(C)NC(C(CC)N(C)C)=O)C)coc2c(C)c(Cl)ccc12 97201,CC1NC(=O)OC12CN(C(C13CCC1CN(C(=O)CC1(C)CCOCC1)C3)=O)C2 97202,C(CCC(CCC)NC(c1c[nH]nc1-c1ccncc1)=O)NC(COCC#C)=O 97203,C(=O)(C1CCc2nccn21)NC(C(C)C)CNC(c1ccc(C(=O)N(C)C)cc1)=O 97204,C1(NC(c2cncc(NC)c2)=O)CCCN(C(C2C=CCS2)=O)C1C 97205,Cc1cn2c(n1)C(C)N(C(CC1CCCCC1)C(=O)NC(C)C)CC2 97206,CCC(C)(O)C(=O)NCCC1CN(C(C2(c3nccs3)CC2)=O)CCO1 97207,N1(CC(CC)C(C)C)C(=O)CN(CCCc2nccs2)C1=O 97208,c1(C(N(C)CCNC(C2(CF)CCOCC2)=O)=O)ccc2c(c1)N(C)C(=O)CO2 97209,c1(CCN=C(NC(COC)C)NCc2cc(C)cc(Cl)c2)ccc2[nH]ccc2c1 97210,C(=O)(C(CC(C)C)C(C)C)NCC1C(NC(c2c(OC)ccnc2)=O)C1 97211,C(=O)(CC(C)(C)C)N1CC(NC(C2CCN(C(C)=O)C2)=O)(CO)C1.C1(=O)C(C)N1 97212,C12(C(=O)NCC3(F)CCC(CNC(Cc4ccn(C)n4)=O)C3)CC1COC2(C)C 97213,c1(C(=O)NCC2(C(C)NC(C3C(CC)C3)=O)CC2)cnc(C)o1 97214,c1(CC(=O)NC(C)CNC(C2COC2)=O)ccc2ccncc2c1 97215,N1(C(c2cc(C)cc(Cl)c2)=O)C2CCC1CC(CNC(C1CCC(C)C1)=O)C2 97216,O=C(CC(C(F)F)NC(C1CCOCC1)=O)NCCC1CC(F)(F)C1 97217,Cc1cc(O)ncc1C(=O)NC(c1ccccc1)CNC(c1ccc(CO)s1)=O 97218,c1(NC(C2C(NC(C=CC=CC)=O)CCCC2)=O)cc(Cl)ccc1I 97219,O=C1CN(CCN(C(=O)CC(O)C2CCCC2)CC)CCN1.C12CCC1C(=O)NC2 97220,N1(C(CN2CCC(C)C2)=O)CCC(N(C)Cc2ncccc2OC(F)F)CC1 97221,CC(C)(C)CC(C)(C)C(=O)NC1CN(C(=O)C(C)(C)Cc2ccccc2)CC1O 97222,N1(C(C(c2cn(C)nc2)O)=O)CCC2CN(c3ccc(Cl)cc3[N+](=O)[O-])CC2C1 97223,Cc1cc(N2CCCC2)nc(=NCCc2ccc(CC(C)C)cc2)[nH]1 97224,c1(C(=O)NC(C(=O)NC2C(OC)C3(C2)CCC3)CC(C)C)cccc2cncn12 97225,C(=O)(C1=CCN(C(=O)C(C)(C)C2CCCO2)C1)N(C)CC1CCCO1 97226,Cc1nsc(N)c1C(=O)NCC1(O)CCN(C(c2ccoc2Cl)=O)C1 97227,CC1C(NC(=O)C(F)C(C)(C)O)CC2CCC1N2C(c1ccsc1Cl)=O 97228,C1(C)(CC)CC(C(=O)NCCCC(CO)NC(=O)Cc2ccoc2)CCO1 97229,CN1CCN(CCN2CCOCC2CN2CCCC2)CC1 97230,C(=O)(CC(F)(F)C(F)(F)F)NCC(C)(C1CC1)NC(CCOCCC)=O 97231,C1(NC(C(N2CCN(C)CC2)C)=O)CC2C(NC(=O)C(C)(C)O)C2C1 97232,N1(C(c2c(C)cncc2)=O)C2CCC(C2)C1CNC(=O)CSCC1CCCCO1 97233,C1(C)(CC(=O)N(C)CCNC(c2csc(C3CC3)n2)=O)CCS(=O)(=O)N1 97234,C(CO)(CO)(CO)NC(C1(CCNC(C(C)C2CCCO2)=O)CC1)=O 97235,N1(C(C(N2CCN(C(=O)OC)CC(C)C2)=O)=O)CCC2(CC1)CNC(=O)C2O 97236,N1(C(C(C)c2cc[nH]n2)=O)C2CCC1CC(CNC(C1(CF)CCC1)=O)C2 97237,N1(C(C(=O)NCc2ccc(OC)cc2)c2ccon2)CCC(C)C(C)(C)C1 97238,C(=O)(CC(F)(F)C(F)F)NC1CCN(C(c2ccc(OCC(F)F)cc2Cl)=O)C1 97239,c1(SC)ccc(O)c(C(=O)NCC2CCCC2NC(C2CC2C(F)F)=O)c1 97240,N1(C(c2ccc(CNC(c3c(C(C)C)cco3)=O)cc2)=O)CCC(O)CC(C)C1 97241,C1(CC(=O)NCC2(COC)CN(C(=O)CCn3ccnc3C)C2)CCCCC1O 97242,C1(CNC(C=C(CCC)C)=O)C(C)CCCN1C(C1CN2CCC1CC2)=O 97243,C12(C(=O)NCC3(CNC(C=CC(CC)C)=O)CCC3)CCCC1(C(N)=O)C2 97244,C(=O)(C1=CCCN(C(c2ccncc2CO)=O)C1)N(C1CCOC1=O)C 97245,CCN=c1[nH]c(C(N2CCN(C)CC2CNC(c2c(C)ccn2C)=O)=O)cs1 97246,N1(C(c2c(COC)scc2)=O)CC(OC)CC1CNC(=O)CCc1ccn(C)c1 97247,c1(C(N2CC3CC3(C(=O)Nc3cnn(CCO)c3)C2)=O)ccc(I)cc1 97248,N1(C(C2(CNC(=O)CC3CC=CCC3)CC(=C)C2)=O)CCOCC(F)(F)C1 97249,C1(NC(c2csc(C)c2N)=O)CC2CCCC(C1)N2C(=O)C(C)(C)CC1CC1 97250,C1(C(N2C(C(N3C(CC(C)C)COCC3)=O)CSC2)=O)CCC(C)(O)CC1 97251,C(CCCCN(c1ccc(F)cc1)CCC#N)(C(=O)OC)N1CC(CC)OCC1 97252,C1(C)(CNC(c2ccc(C)cc2)CCO)CCC2CC2C1 97253,C12(NC(C(=O)NCC)=O)CCC(CC1NC(=O)C(c1ccc(F)cc1)=O)C2 97254,C(=O)(C1=CC(O)C(NC(=O)C(C(=O)OCC)OC)C1)N(C1CCCCC1)CC#C 97255,C1(n2c(CCOCCC(C)C)nc(-c3c(C)cccn3)n2)CCCCC1(C)C 97256,c1(CC(C)C)ccc(C(=O)NCC(C2CCCCO2)O)c(F)c1 97257,CC1(C)C(CC(=O)NCC2(O)CCSC2)CCN1C(c1cn[nH]c1)=O 97258,CC12CN(C(c3ccc[nH]3)=O)CC1CN(C(C1(C3CCCO3)CCC1)=O)C2 97259,N1(C(CCN(CC)CC)=O)CCCC(C)(C(N2CCCC(F)(F)C2)=O)C1 97260,c1(NCC2(C(=O)NC(c3cnn(C)c3)C(=O)OC)CC23CCC3)ncncc1I 97261,CC1(C)NC(=O)N(CC(=O)NCC2CCC(NC(=O)CCSC(F)(F)F)C2)C1=O 97262,Cc1cc(N2CCC(C)(N(C)C)C2)ncc1S(=O)(=O)NC1CCCOC12CCC2 97263,c1(OCC)cccc(CC(=O)NCC2(OC)CCN(C(c3cc[nH]c3)=O)C2)n1 97264,N1(C(CCC(=C)Br)=O)CC(NC(c2cscc2CC)=O)CCC(O)C1 97265,c1(C(N2CCN(C(C3(COC)CC=CC3)=O)CC2C)=O)cc(N)c(C)cc1Cl 97266,N1(C(C(=O)N(C(C)C2CC2)C2CC2)=O)CCc2c([nH]c3c(Br)cccc23)C1 97267,c1(OC)c(Cl)cc(C(=O)NC2CC(NC(c3nccc(C)n3)=O)CC2O)nc1Cl 97268,N1(C(CC(C)F)=O)CCN(C(=O)CC2CCC(F)(F)CC2)CC12CCC2 97269,C(=O)(C(CC1CC1)NC(=O)C=CCO)NC1(COCC)CC1 97270,C1(NC(C2CCC(C)C2)=O)CN(CCCC(C)(C)C)CCC1C 97271,CC1(C(=O)NCC2CCC(F)(CNC(c3ccc(C(N)=O)o3)=O)C2)CCC(=O)N1 97272,Cc1cc(C)c(C(N2CC(C(=O)NCC(O)C(F)(F)F)C(C)C2)=O)cn1 97273,c1(C(=O)NC2CCN(C(c3cnc(CCC)s3)=O)C(C)C2)cc(F)c(C)cc1Cl 97274,C=C=C(C)CC(=O)NCCN(CC(C)O)C(=O)CN(C)C1CC1 97275,c1(NC(c2n(CC=CC)ncc2)=O)cnc2c(c1)CN(S(=O)(=O)CC(C)C)CC2 97276,C1(NC(CCc2cc(OC)no2)=O)(CO)CCN(C(C2COCCO2)=O)C1 97277,N1(C(CC#N)=O)CC2CCCCN2CC1CNC(=O)CC1(O)CCC1 97278,N1(C(c2cnc(C)s2)=O)CCC(C)(C(=O)NCCC2CCCC2(C)C)C1 97279,C1(OC)(CNC(=O)C(F)F)CCN(C(=O)C(C)Cc2ccc(F)cc2F)CC1 97280,N1(C(CC2ON=C(CC)C2)=O)CC(F)(F)CC1CCNC(c1cc(OC)n[nH]1)=O 97281,C1(CNC(C(C)C(F)F)=O)CCCN(C(=O)Cc2cc(F)ccc2F)CC1 97282,CC1(C)CC1(C)C(=O)NC(c1csnc1C1CC1)=O.C12CN(C1)C2.C1C=CC1 97283,CC(C)C(O)CC(=O)NCCC1(NC(c2cccn(C3CC3)c2=O)=O)CCC1 97284,N1(C(C=CCOC)=O)CCCC(C)(NC(c2cn3ccsc3n2)=O)C1 97285,c1(C(=O)NCC2CC(NC(c3c(OC)cccc3)=O)C2)cnnc2ccccc12 97286,c1(OC)cccc(C(N2CCN(C(c3cnc(C)[nH]3)=O)C3CC23)=O)c1[N+](=O)[O-] 97287,c1(OCC)ccc(C(=O)NCCC2CN(C(=O)CCC(N)=O)CC2C)cc1OC 97288,C#Cc1ccc(C(=O)N(C2CC(NC(C3(CC(C)C)CCNC3=O)=O)C2)C)cc1 97289,CCC(C)(COC)C(=O)NCC(N1CCN(C(=O)CCC=C(C)C)CC1)C 97290,Cc1cccnc1C(=O)NC1CCCC1n1cc(CCC(C)C)nn1.N 97291,C1(n2cc(NS(C)(=O)=O)nn2)CCCN(C(C2CC(n3ccnn3)C2)=O)C1 97292,N1(C(Cc2c(C)nn(C)c2C)=O)C2CCC1CN(C(C1CC(=C3CC3)C1)=O)C2 97293,c1(CNC(COC(CC)C)=O)ncccc1CNC(C1CN(C)C(=O)N1)=O 97294,C1(NC(C(Cc2ccoc2)NC(c2c(C)n(C)cn2)=O)=O)CCNC(=O)CC1 97295,C1(CNC(C=CCN(CC)CC)=O)CN(C(=O)CS(N)(=O)=O)CCCO1 97296,c1(N(C(c2ccnn2CC)C(=O)NC(CC)C)C)ccc(C)c(F)c1 97297,C1(C2CCN(C(=O)CN(C)C(=O)OC(C)(C)C)CC2)(NC(C=CCCC)=O)CC1 97298,CC1(C)CCC(F)(F)CC1C(=O)NC1CCN(C(=O)CC2CC=CC2)CC1F 97299,C1(CC(=O)NC2CCCC(NC(=O)C=C3CCCCC3)C2)(OC)CCCCC1 97300,C(=O)(C1=COCCO1)NCC1C(NC(c2n[nH]c(C)c2Cl)=O)CCCC1 97301,N1(C(c2c(CC)ccs2)=O)CCCC2CN(C(c3cccc(C)c3N)=O)CCC12 97302,CS(=O)(=O)c1ccc(OCC(=O)NC2(CNC(C34CCCCC3C4)=O)CC2)cc1 97303,c1(Cc2n(C(C)(C)C)cnc2)ccc(NC(CC(N)=O)c2ccccc2)cc1 97304,CON(C(=O)C=C(C)CNC(c1sccc1CO)=O)C(C)C 97305,C1(c2cn(C3CN(C(C(C)(C)OC(C)=O)=O)C3)nn2)C(C)(C)C1(C)C 97306,N#CC1CCC(CC(=O)NCCCCC(=O)NCCN2CCC(O)CC2)C1 97307,C1(NC(c2scc(C(C)=O)c2)=O)CC(NC(c2cncc(C(F)F)c2)=O)CC1O 97308,C1(C)(CN(C(=O)CC2C=CCC2)C)CCCC1NC(c1sccc1Cl)=O 97309,C(CC(C(=O)N1CC(N2CCCC2=O)C1)NC(=O)Cn1cnnc1)OC 97310,N1(CCC(N2CCCC(NC(C=C(CC)CC)=O)C2)=O)Cc2ccccc2C1=O 97311,c1(NC)ccc(C(N2CC(NC(=O)CCc3ccc(O)nc3)C(F)C2)=O)cc1F 97312,c1(CNC2CCN(C(C(C)OC(C)(C)C)=O)C2)c(I)ccnc1F 97313,N1(C(C=C2CCC(C)CC2)=O)CC2CCC(CNC(C3CC3(Cl)Cl)=O)C2C1 97314,N(C(=S)N1CCC(N2CCOCC2)(C(N)=O)CC1)C1CCCC(C)C1 97315,c1(OCCC)ccccc1C(=O)NCC(O)CNC(=O)C(=O)NCCC(F)(F)F 97316,c1(C(N2CCCC(C)(NC(C(C)n3cccn3)=O)C2)=O)ccc2[nH]ccc2c1 97317,N1(C(CCCN(C(C)=O)C)=O)CCC(C(=O)NCCC(O)C(F)F)CC1 97318,C1(C(=O)NC2CC3(CN(C(COCC)=O)C3)OC2)CCC2(CC1)CC2(F)F 97319,c1(-c2ccc(CC)cc2)cc(NC2CCCCC2C#N)cc(=O)o1 97320,C(c1cn[nH]c1)=C(C)C(=O)N1CC(n2cc(CNC(c3cocn3)=O)nn2)C1 97321,C(=O)(C(F)(F)C1=CCOCC1)NC.O=C1C(=O)NCC2(CC2)CN1.C(C(F)F)N 97322,N1(C(C)=O)CCCC1C(=O)NCC1(F)CC(NC(C2CC(C)=NO2)=O)C1 97323,C(=O)(C(C)(C)n1cc(NC(N2CCC2(C)c2ccccc2)=O)cn1)OCC 97324,c1(C(=O)NCCC2CCN(C(C(COC)O)=O)C2)ccc(OC)c(SC(C)C)c1 97325,c1(C(=O)NCC2C(NC(c3c(C)c[nH]c3)=O)CCCC2)cc(Cl)ncc1Cl 97326,C1(CC(=O)OC)CC2(CCN(C(c3cc(C)[nH]n3)C(=O)NCC3CC3)C2)CO1 97327,C1(C(N(CCOC)C2CC2)=O)CCCN(C(c2cc(OCC)cnn2)=O)C1 97328,Cc1cnsc1C(N1CCCC1CCCNC(=O)Cc1cnn(C)c1)=O 97329,c1(CNC(=O)NC(c2ccccc2)COC)ccnc(S(C)(=O)=O)c1 97330,c1(CC)ccccc1CC(N1CCCC1(C)CNC(=O)C=Cc1cnn(C)c1)=O 97331,C(=O)(CC(C1CC1)NC(C1CCCN1C(C1CCCO1)=O)=O)NC 97332,c1(OC)ccc(C(=O)NCCC2CN(C(C3C(C)(C)C3(C)C)=O)CCO2)nc1N 97333,N1(C(c2c(CC)nn[nH]2)=O)CCOCC1CC(=O)N(C1CCN(C)C1=O)C 97334,c1(C(=O)NCC(C2CC2)NC(c2n(CCC)ncc2)=O)cc(OC)ccc1OC 97335,C1(OC)CN(C(=O)CC(C)SC)CC1NC(=O)CCC1CCCCCC1 97336,N1(C(C(C)OCC=C)=O)CCN(C(C2CCCSC2)=O)C(c2ccncc2)C1 97337,n1(CC)ncnc1C(C)NC(=O)C(C)(C1CC1)N(C)C(C1CCC(N(C)C)C1)=O 97338,N1(C(C2(C)CC2(Cl)Cl)=O)CC2CCC1C1CN(C(=O)CCN3CCCC3)CC21 97339,N1(C(=O)CCc2cccc(N3CCCS3(=O)=O)c2)CCC(O)C12CCSC2 97340,C(=O)(C1CCCc2cccnc21)NCC1CN(C(C2C(C)C2C)=O)CC(C)(C)O1 97341,N1(C(C2(CC=C)CC2)=O)CC(C(=O)NCC2CC(C(C)(C)C)C2)C(F)(F)C1 97342,N1(C(C(CC(CC)C)C)=O)CCC2(CC1)CCN(C(=O)C(C)(C)OC(C)=O)C2 97343,C1(C(N2CCCC(CN(C(=O)CCF)CC)C2)=O)CCC2(CCC2)CO1 97344,c1(C(=O)NC2C(NC(c3cc(OC)ncc3)=O)C2)cc2cc(Cl)ccc2s1 97345,C(=O)(CC1=NN(C)C(=O)C1)NC12CC(CNC(C(CC=C)(C)C)=O)(OC1)C2 97346,S(=O)(=O)(c1ccc(N2CCC(n3cc(Cl)cn3)C2)c(Br)c1)NC(COC)(C1CC1)OC 97347,N1(C(C2C(=C)C2)=O)CC2CCCC(CNC(c3c(CC)noc3C)=O)C2C1 97348,Cc1cccc(C(C(C)C)NC(=O)NCCc2nc(C(C)(C)C)no2)c1 97349,C1(CNC(Cc2nc(C)sc2)=O)CCC(C)CN1C(=O)C=Cc1cnn(C)c1 97350,CCC(CC(C)C)C(=O)NCC1CCCC1C(=O)NC1(C(=O)OC)CC1 97351,N1(C(c2cc(C)no2)=O)CCCC(C(=O)NCC23CCCC2C3)C1 97352,C1(CNC(C(CC)OC)=O)CN(C)CCN1C(=O)CCOCC(C)C 97353,c1(OC)ccc(C(N2CCC(NC(c3cnc(C)nc3C)=O)C2)=O)cc1OC 97354,Cc1ccc(F)c(OCC(N2CC3CCC2C3NC(C2CC3CC3C2)=O)=O)c1 97355,Nc1cc(C(N2CCN(C(=O)Cc3cncnc3)C3CC23)=O)c(F)c(F)c1F 97356,C1(C(=O)NCCCNC(=O)Cc2cncnc2O)CCC12CCOCC2 97357,C1(CNC(c2cc(CO)[nH]n2)=O)C2CN(C(=O)C=CC3CCC3)CC12 97358,N1(C(C=NOC)=O)CCC2CN(C(=O)CSCC(F)F)C(C)C12 97359,C1(CC#C)(C(N2CC(O)C(O)C2)=O)CCN(C(c2cc(CC)oc2C)=O)C1 97360,N1(C(C(C)NC(N)=O)=O)CC(NC(=O)C(F)(F)c2nccs2)C(C)C1 97361,C1(OC)(CNC(C2CC(O)C2)=O)CN(C(C2(c3ccccc3)CC2(Cl)Cl)=O)C1 97362,CCC(CC)C(=O)NCCN(C(c1c[nH]nc1Br)=O)C1CC1 97363,c1(N2CCc3c(cc(C)s3)C2)nc(NCc2scnc2C)c2c(n1)c(C)nn2C 97364,c1(C(=O)NCC(CC)(C)NC(=O)CCCSC)cnc2ncccn12 97365,C1(CNC(c2ccc(CC)cc2)=O)CCCCN(C(C2(C)CCC(=O)N2)=O)CC1 97366,C(C(N)CC(F)(F)F)NC(C1CCCN(Cc2nc(CC)sc2)C1)=O 97367,c1(C(N(C)CC2CN(C(C3CC(N=[N+]=[N-])C3)=O)CCO2)=O)ccn2nccc2n1 97368,c12ccc(c(F)c1)[nH]2.C1(C(=O)NCCC#C)C2CN(C(=O)OC)CC12 97369,c1(C(=O)NC2(CCCC(=O)N(CC(=O)NC3CC3)C)CCC2)ccc(F)cc1F 97370,CCCCC(CC)CC1C(=O)NC2CCN1C2.C1(C(=O)OC)(COC)CCOCC1 97371,CC(CC(C)(C)C)C(=O)N1CC(NC(=O)C(C)(C)CC2CC2)C(C)C1 97372,c1(C(=O)NC(c2nc(C)on2)C=Cc2ccccc2)ccc(N2CCOCC2)cc1O 97373,c1(C(N(CCCOCCNC(=O)COCC2CC2)C)=O)c(F)cccc1F 97374,C1(N(C(C(CSCC)NC(=O)CC=CC(C)(C)C)=O)C)CCCC(C)C1C 97375,c1(NCC(=O)NC(CN(C(=O)CC(C)(C)C)CC)C)c(F)c(F)cc(F)c1F 97376,CC(C)P(=O)(CC(=O)NCC(CNC(=O)CCCN(C)C)CO)C(C)C 97377,C1(C(N2C(CCNC(c3c(CC)nc[nH]3)=O)CCCC2)=O)CNC(=O)CC1(C)C 97378,C1(CC(=O)N(CCN(C)C)C)COCCN1C(c1ccc(C(F)(F)F)nn1)=O 97379,C1(O)(CNC(c2cnc(OC3CC3)s2)=O)CCCN(C(=O)COc2ccccc2)C1 97380,Cc1ccccc1OCCCC(=O)NCCC(O)CNC(C1CN(C(C)C)C1)=O 97381,N1(CCCCOCC)CC(c2ccccc2)C1CNC 97382,N1(C(C2(CC#C)CCCC2)=O)CC(C)C(N=c2[nH]n(C(C)C)cc2[N+](=O)[O-])C1 97383,C(C(C)(C)C(=O)N(CCCN(C(=O)C(=C1CCCCC1)F)C)C)OC(C)C 97384,Cc1cccc(O)c1C(=O)NCC1(CNC(=O)CC2CCN(C)C2)CC12CCC2 97385,c1(C(N2CCC(N(C(C(CC=C)OC)=O)CCOC)C2)=O)cc2n(n1)CCCN2 97386,CCCC(CNC(c1cc(Cl)n(C)n1)=O)C(=O)NCC1(CCOC)CC1 97387,Cc1ccc(C(C)C(=O)N(CC(=O)O)C(c2cn(C(C)(C)C)nn2)C)cc1 97388,N1(C(C2C(C)=C2)=O)CCCC1C(C)(C)CNC(C1CC(=O)N1)=O 97389,C#CCC(C(=O)NC)NC(c1coc(CNC(=O)CSC2CC2)c1)=O 97390,c1(C(N(C2CCN(C(c3ncc(F)cc3Cl)=O)C2)C)=O)cc(Cl)cc(Cl)c1 97391,N1(C(CC=C(C)C)=O)CC2(CCN(C(c3sccc3Cl)=O)CC2)CC1C 97392,C1(CNC(=O)CCOC2COC2)(NC(c2cc[n+]([O-])cc2)=O)CCOCC1 97393,Cc1cn(C)nc1C(N1CC(n2cc(Cn3cncn3)nn2)C(O)C1)=O 97394,C1(CC)CN(C(c2cnnn2C)=O)CCC1NC(=O)CCCCNC(N)=O 97395,c1(CC)ccc(C(N2CCOCC2CNC(=O)CC(C)COC)=O)nc1 97396,C1(CC(=O)NC(C)C(C)(C)NC(c2cccc(C(F)(F)F)c2)=O)CCC(=O)N1C 97397,N1(C(c2nccc(C)c2)=O)CCN(C(c2cnc3[nH]cncc2-3)=O)C2CCC12 97398,Cc1nccn2ncc(C(=O)NCCC(C)NC(c3cc4c(s3)CCCC4)=O)c12 97399,c1(C(N(C(CNC(c2c(C)nc(OC)s2)=O)C)C)=O)cnc(O)c(C(F)(F)F)c1 97400,c1(C(=O)OC)cnc(N2CCN(C(c3ccnn3C)=O)CC2C)nc1C 97401,c1(C(c2nc(Cc3sccc3Cl)no2)(C2CCCO2)C)ccncc1 97402,C1(CC(=O)NCCOC2CCN(C(c3c(C)cno3)=O)C2)CCC(C)(C)CC1 97403,c1(C(=O)NC(C)CN(C(=O)C(CO)NC(N)=O)C)cccc2cnnn12 97404,c1(C(N2C(C(=O)O)C3CC3C2)=O)cnn2ccsc12 97405,O=C(C1CCCc2nn[nH]c21)N1CCC2(CNCCO2)C1 97406,N1(C(C(C=C)C)=O)CC2CCCC(N(C)C(c3nnsc3CC)=O)C2C1 97407,N1(C(C(CC)COC)=O)CCCC(F)(CNC(=O)Cc2ccccc2OCC)C1 97408,CC1CN(C(C2CC2(Cl)Cl)=O)CC1CCNC(C1CCCCCC1)=O 97409,c1(OC)ncc(C(=O)NCC(C2CC2)NC(=O)CCNC(C2CCCCC2)=O)s1 97410,c1(C(C)C)nccn1CC(=O)N(CCNC(=O)CN1CCC1C)C(C)C 97411,C1(CC(N2CCC(C)(CCC)C2)=O)CC2(C1)CN(C(C1(C)COCCO1)=O)C2 97412,C(=O)(CCCCCF)NCC(C)(C)NC(C(C(=O)N(C)C)C1CC1)=O 97413,c1(OCC(C)(C)NCCS(N)(=O)=O)ccccn1 97414,CC(C(=O)OC)C(=O)N(CCCNC(C1CCC(C(=O)OC(C)(C)C)CC1)=O)C 97415,C(CC(C)C(=O)N1CC(NC(=O)C(c2ccc(O)cc2)=O)C(C)C1)OC 97416,c1(CNC(C(N2CCC(CN(C)Cc3cccc(Cl)c3)C2)=O)=O)ncccc1F 97417,c1(C(C(=O)N(C2CCCC2)CC2CC(NC(=O)C=CCF)C2)O)ccc([N+](=O)[O-])cc1 97418,c1(NC(C(CC)n2cnc(-c3nn[nH]n3)n2)=O)ccc(Br)c2c1CCO2 97419,C=C(C)C1OCCCC1C(=O)NCC1CN(C(C2CN(C)C2)=O)CC12CCC2 97420,c1(OC)cc(OC)nc(N2CCCC2CN(C(=O)C(O)C(C)C)C)n1 97421,C(CC(C)C)(C(=O)NCC(n1ccnn1)C)ONC(c1c(CC)ncs1)=O 97422,c1(ON)ccc(C=NOC(C=COCN)=O)cc1 97423,CC1CCCC1(C)C(N1CCOC(CNC(=O)Cn2cc(N)cn2)C1)=O 97424,CC1(C)CCCC(CCN(C(c2ncc(Cl)s2)C(=O)NCCCOC2CC2)C)C1 97425,C1(CNC(CCn2c(C)ncc2)=O)CCN(C(=O)CCc2cncnc2)CC1O 97426,CCCCC(O)C(=O)N1CCN(C(c2cc(OC)cc(F)c2)=O)C(CCC)C1 97427,C1(NC(COCc2nnc(C)s2)=O)CCN(CCc2ccc(F)c(F)c2)CC1C 97428,CC(CN=c1[nH]c2c(c(=NCc3ccccc3-n3ccnn3)[nH]1)CCC2)C(F)F 97429,C1(N(C(c2c(OC)csc2)=O)C)CCCCC1NC(c1cncc(C(F)F)c1)=O 97430,C1(NC(c2ccc(O)cc2)=O)COCCN(C(C2CCN(C3CC3)C2=O)=O)C1 97431,C(CCO)(C(F)F)N(C(=O)CP(C)(C)=O)C(C1(C(CC=C)(C)CC)N=N1)=O 97432,C#Cc1cc(NC(=O)C(C2CCCO2)NC(=O)Cc2csnn2)cc(F)c1 97433,c1(OC)ncc(C(=O)NC(C)C(CO)NC(c2ccc(F)cc2SC)=O)cc1C 97434,c1(CCC(=O)N(CCNC(C(C)(C)OC(C)=O)=O)C)ccc(Br)nc1 97435,c1(N2CC3(CN(C(=O)C=Cc4ccc(Cl)nc4)C3)C2)ncnc2ccc(Cl)cc12 97436,c1(OC)cccc(NC(C(c2c(C)noc2C)NC)=O)c1.C1CCN1.C1(OC)CC1 97437,C1(C(=O)NCCNC(c2ccc(CC)cc2F)=O)CC(=O)N(C)C(=O)N1 97438,Cc1ccc(C(N2CCN(Cc3ccc(N4CCCC4)nc3)C3CC23)=O)cc1Cl 97439,Cc1cc(CC(=O)NC(C)(CNC(=O)C(C)CO)C2CC2)n[nH]1 97440,CCC(C)CC(=O)NC(c1ccc(CO)s1)C(=O)N(C)C(c1cccc(C)c1)C 97441,C1(C(N2CCN(C(C(=O)NCC3CC3)=O)CC(CO)C2)=O)CCc2nnnn2C1 97442,c1(OC)cc(CC(N2CCC(NC(C3CC3C)=O)C2(C)C)=O)ccc1Cl 97443,C(=O)(C(CCc1ccccc1)N1CCOC(C(=O)NCCSC)C1)NCCOC 97444,N1(C(C)C(=O)Nc2cc3nccnc3cc2Cl)Cc2cc(Br)ccc2CC1C 97445,N12CC(CC1=O)NC(=O)N(C(C)(C)C)CC2.C(c1cn(C(C)C)cn1)=CCN.CO 97446,c1(C(N2CC(CC)C(NC(=O)COC3CC=CC3)CC2)=O)cc2cccnc2s1 97447,c1(C(=O)NC2(C)CC(N(C)C)C2)cccc(S(=O)(=O)N(C)CC2CCCCC2)c1 97448,Cc1ncn(C)c1C(=O)NC1(CO)CN(C(=O)CSc2ccc(Cl)cc2)C1 97449,C1(C(=O)NCCCC2(CO)CCC2)CCN(Cc2c(F)cccc2Cl)CC1O 97450,C12(CC(=O)NC3CC(CNC(=O)Cc4cnc(C5CC5)o4)C3)CCCN1CCC2 97451,N1(C(c2cnc(C3CC3)nc2)C(=O)NCC)CCC(O)CC(C)(C)C1 97452,Cc1nc(NCCC2=CCCC2)cc(N2CCCN(S(C)(=O)=O)CC2)n1 97453,c1(NCC(C2(O)CN(C(CCCSCCC)=O)C2)(C)C)ncc(C)cc1[N+](=O)[O-] 97454,C=C(CNC(=O)CSCCNC(=O)CC(CC)C1CC1)C(F)(F)F 97455,C(C(=O)Nc1noc(C2(C)CC2)n1)(C(C)C)OC 97456,C=C=C(C)CC(=O)NCCN(CC(C)O)C(=O)CC1CC(OC)C1 97457,C(Cc1ccoc1)(C(=O)NCCCn1ccnc1)NC(C1C(CC(C)C)C1)=O 97458,Cc1cc(Br)ccc1CC(=O)NC1CC1NC(C1(C)CC(C)(C)C1)=O 97459,CCCC(C)(O)CC(=O)NCCNC(=O)Cc1ccc(CC(C)C)cc1 97460,Cc1cc([N+](=O)[O-])cc([N+](=O)[O-])c1NC(C)CNC(c1n[nH]cc1Cl)=O 97461,CC(C)C(C)CC(=O)N1CCC(N2CCN(C(c3cc(Br)no3)=O)CC2)C1 97462,c1(C(=O)NC2CCCC2C(=O)Nc2ncccc2Br)c(Br)cccc1Br 97463,c1(C(N2C(CNC(CC)=O)CC(C(F)(F)F)C2)=O)cc2c(cc1F)NC(=O)CC2 97464,c1(C(C)CC(=O)Nc2cn[nH]c2)cccc(I)c1 97465,CCC(C)CC(C(=O)N(CC(C1CCC1)OC)C)NC(c1cnn(C2CC2)c1)=O 97466,c1(C(=O)Nc2cnccc2[N+](=O)[O-])cc(-c2ccc(CO)o2)cc2c[nH]nc12 97467,CC(C)C(C)CC(=O)N(C1CC(C(=O)NCC(O)(C2CC2)C2CC2)C1)C 97468,c1(C(N2CC(CNC(C3CCc4nn[nH]c4C3)=O)C2)=O)cc2n(n1)CC1(CC1)C2 97469,Cc1ccc(CN2CC(C)(CC(N3CCOC(C#N)C3)=O)C2)cc1Cl 97470,CC(CN(C)C)CCC(=O)NCCN(C)C(C1CCC(F)(F)C1O)=O 97471,C(CC(C)(C)C)(C(=O)NCC1CCC=CCCC1)NC(C=CC(C)(C)SC)=O 97472,C1(C)(CNC(C(C=C)O)=O)CCCN(C(=O)Cc2ccc(Cl)cc2F)C1 97473,C(C)(CC(C)(C)C)(c1nnnn1C1COC1)NC1CCC(CC)CC1 97474,c1(C(=O)NCCN(C)C(c2ccc(Cl)c(Cl)c2)=O)cc2sccc2[nH]1 97475,c1(-c2cccc(OC(C)=O)c2)nc2c(s1)CCN(C(C1C3COCC13)=O)C2 97476,C1(C(N2CCC(OCCNC(C3(C4CC4)CCCO3)=O)C2)=O)(CC)CCOCC1 97477,Cc1cc(=NC2CCCn3ccnc32)[nH]c(N2CC3C(C(F)(F)F)C3C2)n1 97478,N1(C(C2C(c3c(C)cccc3)C2)=O)CCN(C(c2nc(O)c(C)s2)=O)CCC1C 97479,C1(C(=O)NC(CNC(Cn2cnc(C(C)=O)n2)=O)C(C)(C)C)CCCC2(CC2)C1 97480,C#Cc1cccc(C(N2CC=CCC2C(N2CCCC(C(C)(C)C)C2)=O)=O)c1C 97481,Cc1cnn(C)c1C(=O)NCC(CC(=O)NC(C)(C)CC(C)C)C1CCC1 97482,c1(C(N2C(C(=O)NCC3CC(F)(F)C3)(CC)CCC2)=O)cc(C)cc(C#N)c1 97483,c1(C(=O)NC(C)C(C)NC(=O)CCNC(C2CCC2)=O)ccc2ncccc2c1 97484,c1(C(N2CC(NC(C(CCC)C)=O)C(O)C2)=O)sc2ncccc2c1Cl 97485,c1(CC(=O)NCCC(C(C)C)NC(c2c[nH][nH]c2=N)=O)ccc2c(c1)CCOC2 97486,C1(NC(c2cc(OC)ns2)=O)CCCCCN(C(=O)C(C)(C)c2ccsc2)C1 97487,C(=O)(C1=C2CCN=C2NC=C1)NCC(CNC(C1N(C)CC(C)(C)C1)=O)O 97488,C(=O)(C1=COCCC1)N1C(C)CC(NC(=O)Cc2nnn(C(C)(C)C)n2)C1 97489,C(=O)(C1OCCn2ccnc21)N(CCCCNC(C1(C(=O)NC)CCC1)=O)C 97490,C1(CNC(Cn2c(C)ccn2)=O)CCC2CN(C(=O)CCc3nncs3)CC12 97491,c1(-c2onc(-c3cccc(OC)c3)n2)cccc2cc(OC)ccc12 97492,C12(NC(Cc3cccc(COC)c3)=O)CCC(C1)N(C(=O)C(C)NS(C)(=O)=O)C2 97493,CC(F)(F)CCCC(=O)NC1CC(NC(=O)Cc2cnsc2)C12CCC2 97494,CC1=C(C(=O)NCCCN(CCCCNC(=O)CCN2CCNC(=O)C2)C)CCO1 97495,C1(C(N2C3C(CNC(C(C(C)O)C)=O)CC(CC3)C2)=O)CCc2cnn(C)c2C1 97496,N1(C(C(C)(C)O)=O)CC2CCC1CN2C(C1(C#N)CCC1)=O 97497,C1(C(=O)NC(CCCNC(c2c(Cl)cc(C)s2)=O)C)CCCC2(CCC2)O1 97498,C1(C)(C(=O)NCC(=C)CCNC(=O)CCOCCOC)C2CCC(C2)C1(C)C 97499,N(C1C(=O)Nc2ccc(F)cc21)C(C1=C(C)OCC1)=O 97500,N1(C(C(N2C(C)CN(c3ccncc3)CC2)=O)=O)CCC(C2(O)CCC2)CC1 97501,CN1CCC1C(N1CC(CNC(=O)C=CC(C)(C)C)C1)=O 97502,CCC(C(=O)OC)C(=O)N(CCCCNC(C1(c2ncco2)CCC1)=O)C 97503,c1(C(N(CCNC(c2cccc(C(=O)OC)n2)=O)CC)=O)sccc1S(N)(=O)=O 97504,C(=O)(C1CC(C)(C)Oc2ccccc21)N1CCC(NC(c2n(C)cnc2)=O)C1 97505,N1(C(C(=O)NCC(c2cn(C)nc2)(F)F)=O)CCc2c(ncn(C)c2=O)C1 97506,O=C(C1CCCc2nn[nH]c21)NCC1CCN1C(C1(c2noc(C(=O)O)n2)CC1)=O 97507,C(CCCCCNC(C1(C)CC1F)=O)NC(C1CC(O)(CC#C)C1)=O 97508,N1(C(C2(COC(C)C)CC2)=O)CC(N(C(=O)C(C)CN2CCOCC2)C)C(O)C1 97509,Cc1ccc(C(=O)NC23CC2CN(C(c2ncn(C)n2)=O)C3)c2ccccc12 97510,c1(C(=O)NC(c2ccc(F)cc2)CNC(CC(C)CF)=O)cnn2ccccc12 97511,c1(C(=O)NCC2COCCN2C(c2ccnnc2O)=O)c[nH]c2ncnc(O)c12 97512,Cc1ccc([N+](=O)[O-])cc1C(N1CC(O)CC1C(=O)Nc1cnc(Br)c(Cl)c1)=O 97513,C1(C(=O)NCC2CC(NC(CSC(C)(C)C)=O)C2)CCC(c2ncc[nH]2)CC1 97514,c1(C(=O)NCC(CC)(C)NC(C2CCC23CCC3)=O)nsc2ccccc12 97515,Cc1[nH]nc(C(=O)NC2CN(C(=O)C=CCF)CC2C(F)F)c1C 97516,N1(C(C(C(=O)OCC)(C)C)=O)CCc2ccccc2C(NC(=O)CCC2CC2)C1 97517,CON(C(=O)C=CC(C)NC(=O)C(C(C)C)NC=O)C1CCC1 97518,CC1(C)CCOC1CC(N1CCCCC1C1CCN(C(=O)C(O)C2CCC2)C1)=O 97519,C(=O)(CC(O)CC(C)C)NCC(C1CCCCC1)NC(C(CC)(CO)OC)=O 97520,N1(C(CC(C=C)C)=O)CCC2CCCC12C(=O)NCCCC(=C)Cl 97521,C(=O)(C1=NOC(C)(C)C1)N1C(C(C)(C)NC(COCCCCC)=O)CCC1 97522,Cc1cc(C(N2CCCN(C(=O)CCN3CCC3)CC2C)=O)cc2c1CCC2 97523,CCC(C)(C(=O)NC(C1CCN(C(=O)C(C)=CC2CC2)CC1)C)C(N)=O 97524,Cc1noc(C)c1C(C)C(=O)NCC#CCNC(=O)Cc1ccccc1F 97525,c1(C(=O)NC(CCCC)CNC(=O)CC(C)n2cccn2)cc(C)c(C)c(Br)c1 97526,c1(NCC(C)N(C(=O)CC2CCS(=O)(=O)C2)C)cc2nn[nH]c2cc1[N+](=O)[O-] 97527,N1(CC(=O)N(C2CC2)CC)CCN(C(=O)C(C2CCC(=O)N2)C)CC1 97528,C1(C(=O)OCC)CCCC(NCCc2ccc(Cl)s2)CC1 97529,c1(OC)cc(C(N2CCC(CO)(NC(=O)CN(C)C)C2)=O)cc(F)c1F 97530,C1(NC(C(C(CC)C)OC)=O)CC2CCC(C1)N2C(C1(C)CCOCC1)=O 97531,c1(CC)ccc(C(=O)NCC2CC(NC(=O)CCCc3nccs3)C2)c(O)c1 97532,c1(C(C(=O)NC(CC(C)NC(C(C)(C)OCC)=O)C)CC)c(C)noc1C 97533,C(C)(CO)(CC(C)C)NC(C1C(CNC(C(COCC)C)=O)C1(C)C)=O 97534,Cc1cc(Cl)cc(Br)c1NC(C1CC(C)CN1C(c1cnc(O)cc1O)=O)=O 97535,C(=O)(CS(=O)CCC(F)(F)F)NC12C(CN(C(C(C)NC(C)=O)=O)C1)C2 97536,N1(C(c2ccc(OC(F)(F)F)c(F)c2)=O)CCC2CN(C(C3CC34CC4)=O)CC12 97537,N1(C(C2(C)CC2(Cl)Cl)=O)CCC(C)(NC(=O)CN2CCS(=O)CC2)C1 97538,N1(C(c2occ(C)c2)=O)CC2(NC(c3c(-c4ccsc4)noc3C)=O)CCC1C2 97539,CCC(C)(O)C(=O)NCCCN(C(=O)CC1CCCS1(=O)=O)CCO 97540,C12(C(=O)NCCC(C=C)C)CC(CN1C(=O)CC1COCC1O)C2 97541,C(=O)(C1CCCc2nncn21)N1C(CNC(C(C)S(N)(=O)=O)=O)CCC1 97542,n1(CCC)cc(C(=O)NCC2CCCC2NC(=O)C(C)SC(F)(F)F)cn1 97543,c1(NC(c2ccc(O)cn2)=O)c(Cl)cc(F)cc1Cl.N12CCC(O)C(C1)C2=O 97544,c1(C(N2CCC(C)C2c2cccc(NC(=O)OC(C)(C)C)c2)=O)cc(O)nc(O)n1 97545,c1(C(=O)NCCC2CC(NC(C3ON=C(C)C3)=O)C2)ccccc1-n1ccnn1 97546,c1(C(=O)Sc2ccccc2)ncn(Cc2cc(C(F)F)no2)n1 97547,C1(C(=O)NCC(C)(C2CCC2)NC(C=COCC)=O)CC2(C1)CC(O)C2 97548,CCCCC(CNC(C1OC(C)CC1C)=O)NC(=O)C(C)CSC 97549,CC1=C(C(=O)NC2(C)CN(C(c3c(F)ccc4nc[nH]c34)=O)C2)C(=O)OC1(C)C 97550,N=c1[nH]c(=NCC2CCOCC23CCCC3)[nH]c(=NCCn2ccnc2)[nH]1 97551,c1(C(=O)NC(CC=C)CNC(=O)CC(C)P(C)(C)=O)ccc2c(O)ncnc2c1 97552,CC(C(=O)NCC1(F)CN(C(=O)C(c2ccc(Cl)cc2O)=O)C1)C1=CCCC1 97553,c1(C(N2C(C(N3CCCC(C)CC3)=O)CC2)=O)ccc(C#N)cc1Cl 97554,Cc1cc(CC(=O)N(CC(O)CN(C)C(C2(O)CCCC2)=O)C)ccn1 97555,CCC(CCC(=O)NCCF)NC(C1CCC(=O)NC1)=O 97556,Cc1nc(C(C)NC(=O)CC2CCN(C(c3c[nH]c(C(N)=O)c3)=O)CC2)c(C)o1 97557,S(=O)(=O)(c1ccc(C(N2CCCC2C(N2CCCC(F)C2)=O)=O)cc1)NC 97558,CCCCCC(F)C(=O)N(C(C)C(N1CCOC2(CC2)C1)=O)C 97559,N1(C(c2nn(CC)nc2C)=O)CC(C)OC2(CCN(CC3CCC3)C2)C1 97560,N1(C(C2(C)CC(=C)C2)=O)CC2CC(C1)CN(C(=O)CCOC1CCC1)C2 97561,C1(C(=O)NC(CCO)C2CCC2)C2CCC(C2)N1C(=O)CC1CSCCO1 97562,N1(C(C(=O)N(c2ccccc2C)C(CC)C2CC2)=O)CCCC(C)(CC#N)C1 97563,N1(C(C2CCN(C(C(C)CC3CCCC3)=O)C2)=O)CCC2(CCCCC2)C1 97564,c1(C(N2CCN(C(=O)C(O)C3CCCC3)CC2C(F)F)=O)cnc2n1CCOC2 97565,C(CC(C(=O)N=c1cc(C2CC2)n(C)[nH]1)NC(C1(n2nccn2)CC1)=O)N(C)C 97566,c12cc3c(s1)CCC3CN2.C1(N(C)C)CN(C(=O)OC(C)(C)C)CC1F 97567,C(=O)(C1=CCN(C(=O)C(c2ccccc2)F)C1)NC(C#C)CC 97568,c1(N2CCN(C(=O)NCCC(CC)CO)CC2)cc(OC)c(OC)c(F)c1 97569,C(=O)(CCCCC(F)(F)F)N(C)CC1CCCC(NC(COCCSC)=O)C1 97570,C1(N(C(C(CC)CC(C)C)=O)C)CCCC2CN(C(c3csc(=N)[nH]3)=O)CC12 97571,c1(-c2nc(CCC)nn2Cc2cccc3ccccc23)ccc2nnc(C)n2c1 97572,C(=O)(C(C)C(C)C(C)(C)C)N1CC(CCNC(c2c(OC)cc(F)cc2)=O)C1 97573,CC1(C)CC(CNC(=O)C=CSCCO)CN1C(=O)CNC(=O)Nc1ccco1 97574,CC(C)(Cc1ccccc1)CN=c1[nH]c(N2CCC(CF)CC2)nc2c1CSC2 97575,N1(C(c2cn(CC(C)O)c(=O)cc2)=O)CCC2CN(C(C3(O)CCOC3)=O)CC12 97576,N1(C(CSc2ccc(C)cc2)=O)CCC(NC(=O)CN2CC(C)C2)CC1C 97577,c1(CC(=O)N(CCCNC(CC(C)OC)=O)C)cccc(OC(F)F)n1 97578,c1(CNC2(c3ccc(C)cc3)CCOCC2)ccc2c(c1)NC(=O)NC2 97579,C1(C(N2C(CNC(C(C(C)C)NC=O)=O)CCCC2)=O)CCCCNC1=O 97580,c1(N(CCCN(C(=O)COC(F)(F)F)C)C)cc2c(cn1)C(=O)CCC2 97581,C1(NC(C2(OCC)CCC2)=O)CCN(C(c2cc(Cl)ccc2OCC)=O)CC1C 97582,CC1CN(C(c2cncs2)=O)CC2(CCN(C(=O)CNC(c3ccoc3)=O)C2)O1 97583,Cc1cc(C(=O)NCCN(C(C2CCC(=O)NC2)=O)C(C)C)cc(C)c1O 97584,C1(C(=O)NCC(C)(O)CO)C2CN(C(=O)Cn3nccn3)CC12 97585,C1(C(N(C2CCN(C(c3c[nH]cc(Cl)c3=O)=O)C2)C)=O)OC2CCC1CC2 97586,N1(C(C(C)OCC=C)=O)CC2(CNC(=O)CN3CCC(C)C3)CC1(COC)C2 97587,c1(N(C(CC(CC)C)=O)C2CNCC2C#N)nc(-c2ccccc2)cc(C)n1 97588,C=C(C)CCCC(=O)N1CC(C(=O)NC(C)(C)CCCF)OC(C)C1 97589,C1(CNC(c2cc(C)no2)=O)CCC2(CN(Cc3csc(C(=O)O)n3)C2)O1 97590,CC(C)(CCNC(c1ccc(NC=O)cc1)=O)CN=c1[nH]c2cc(Br)cnc2s1 97591,C1(NC(CC2N(CC)CCC2)=O)CN(C(c2ccc(N)cc2O)=O)CC12CCC2 97592,C1(C(N2C(CN(C(CCC3C(C)C3)=O)C3CC3)CCC2)=O)CCCC1C1CC1 97593,N1(C(c2[nH]cc(CC)c2)=O)CC2(C1)CN(c1nc(SC)ns1)C2 97594,Cn1cnc(CC(O)C(=O)NCC(C)(C)NC(=O)CCc2cnco2)c1 97595,C(CN=c1[nH]c(N2CCC(COC)C(F)(F)C2)nc(=N)[nH]1)C1(CSC)CC1 97596,c1(C(=O)NCc2cc(C(N(C(CO)C3CC3)C)=O)sc2)cnn(C)c1Cl 97597,C(=O)(CCCC(=O)N1CCOCC1C(=O)NCC1(C)CC(O)C1)OCC 97598,c1(C(N2CCC(NC(C3CCN(C)C3)=O)C2)=O)cc2n(n1)CCCCO2 97599,C(=O)(C(O)CC(C)C)N1C(CNC(CC(CC)OC)=O)CC(c2ccccc2)C1 97600,CC(=O)C(C(C)C)NC(=O)CN(C(=O)C(C)Oc1cccnc1)C(C)C 97601,c1(C(N2CC(C(C)NC(c3cccn3C)=O)C2)=O)ccc(Br)cc1O 97602,c1(C(C)C)nnc(C=CC(=O)NCCC2(CNC(C3CC4(C3)CC4F)=O)CC2)o1 97603,O=C1COc2cc(C(N3CCN(Cc4ccc(F)cn4)CC3)=O)ccc2N1 97604,c1(CN(C=O)Cc2ccccc2)cc(=NCCC2CC2)[nH]cc1Br 97605,C#CCC(C(=O)NCC(C)CNC(c1ccn(CC(F)(F)F)n1)=O)C1CC1 97606,C1(C(N)=O)(CN)CC2CCCC2C1.c1(NC(=O)C(N)=O)ccc(NC(=O)CO)cc1 97607,C1(C(=O)NCC2(C#C)CCCC2)CCC2(CC2)N1C(c1ccc(C)n1C)=O 97608,C1(CNC(c2cn(C(C)C)c(=O)cc2)=O)CC12CCN(C(C1CCC1)=O)CC2 97609,C1(C(N(CC(=O)OCC)C)=O)(CNC(=O)CN2CCCC2=O)CC12CCC2 97610,C(=O)(N=c1[nH]oc2c1COCC2)n1cc(C(=O)OC)c(O)nc1=O 97611,c1(C(N2CCN(C(c3cncc(C(N)=O)c3)=O)CC2)=O)cc(Cl)nc(Cl)c1 97612,c1(C(=O)NC(C2CCN(C(c3ccc(F)nc3)=O)C2)C)cc2cc[nH]c(=O)c2s1 97613,C1C(CC)(CC)N1.C1(CC)COCC1NC(c1ccccc1)C 97614,C(=O)(C(C)(C)C(N)=O)NCC1C(NC(C2N(C(=O)NC)CCC2)=O)CCCC1 97615,N1(C(C(C(=O)OCC)OC)=O)CCC(CC)CC1C(=O)NC(C)C(O)C(F)F 97616,C1(NC(C(C2CN(C(CC)=O)C2)OC)=O)CCN(Cc2coc(C)c2)C1 97617,C(=O)(CC1CCNc2ccccc21)NC1CCCN(C(c2ncn(C)c2)=O)CC1 97618,C1(NC(CCOCC)=O)CCC(C(=O)N(C(CC2CC2)CO)C)CC1 97619,c1(C(=O)NCC2C(C)CN(C(=O)C(F)(F)CO)CC2)cnc2ncc(Cl)cn12 97620,CCC(CC(=O)N1CC(SC(C)(C)C)C1)C1CC1.n12cc(nn1)CCN(C)CC2 97621,N1(C(CCN(C)CC)=O)CCN(C(c2ccncc2C)=O)C2CC12 97622,N1(C(CC=CC(C)(C)C)=O)CCC=C(C(=O)NCc2ncccn2)C1 97623,C1(C)(NC(C2C(CCC)C2)=O)CCN(C(c2ncoc2-c2ccccc2C)=O)C1 97624,c1(OC)cc(C)c2cc(C(=O)NCCc3nnc(C(F)F)o3)[nH]c2c1 97625,C1(C(N2C(CCNC(C(N3CCNC3=O)C)=O)CCCC2)=O)CC2(CC2)CN1C 97626,C(=O)(C1=CCOC1)NC(C1CN(C(=O)Cn2nccn2)CCO1)C 97627,c1(C(=O)NCC23CN(C(CC(CC)O)=O)C(C2)CO3)ncn2c(C)cc(C)nc12 97628,N1(C(c2nc(CC)sc2)=O)CC2(CC2)CC1C(=O)NCC1(O)CCCOC1 97629,C1(C(=O)NC(C2CCN(C(c3cnco3)=O)C2)C)CCCC(=O)N1C 97630,Cc1cnc(F)cc1-c1c[nH]nc1C(=O)Nc1nccc(C(F)(F)F)n1 97631,N1(C(c2ccc(S(C)(=O)=O)s2)C(=O)NCC=C)CCCC2CCNC(=O)C12 97632,CN1CCC(N(C)C(C2COCCC2NC(c2cncc(Cl)c2)=O)=O)CC1 97633,C(C(C)(C)C#CC(=O)NCc1ccc(F)cc1)NC(c1n(CC)ncc1)=O 97634,N1(C(CCOCCOCC)=O)CC(CNC(C2CCCC2(C)C)=O)CC1(C)C 97635,N#Cc1ccc(NC(=O)C(=O)NC(c2ccccn2)CC2CCCCC2)cc1F 97636,C(=O)(C#CC1CCC1)N1CCC(C(C)(C)NC(c2ccc(OC)nn2)=O)C1 97637,c1(C(N2CCCN(C(c3cccnc3)=O)CCC2)=O)cc(Br)c2occc2c1 97638,C1(NC(Cn2cccc(C)c2=O)=O)CC(N=c2[nH]cnc3cnccc23)C1 97639,C1(NC(c2c(C)c[nH]n2)=O)C(C)(C)CN(C(=O)CC2CCNC(=O)C2)CC1(C)C 97640,C1(C)(CNC(c2c(CC)nc(C)[nH]2)=O)COCCN(C(C2(C#N)CCCO2)=O)C1 97641,CC1(C)CC(C(F)F)CN1CC(C1CCOC1)F 97642,c1(OC)cc(CNC(C2CC2C(N2CCCC(CO)C2)=O)=O)cc(Cl)c1 97643,C12(CNC(C(CCC(C)C)O)=O)CCCC(CN(C(=O)C=C3CCC3)C1)C2 97644,c1(CCCNC(c2csc(Nc3ncc(F)cn3)n2)=O)cc(Cl)cnc1F 97645,c1(C(N2C(C)CC(CNC(=O)CC3CCC(=O)N3)C2)=O)cnc2c(c1)CCC2 97646,C1(C(N(CCCCNC(C(C2CC(F)(F)C2)OC)=O)C)=O)CCC2CC1CO2 97647,C12(C(=O)NCC(=O)NCC)CCCC1CCN2C(c1c[nH]c(=S)cn1)=O 97648,N1(C2C(OCC)NC2=O)CC(c2cccc(C(F)(F)F)c2)OC(C)C1.C1(OC)CC1 97649,c1(C(=O)NCC(CCNC(c2ccc(F)c(F)c2F)=O)O)cccc2c[nH]nc12 97650,c1(Nc2scc(CC(=O)NC(c3n(CC)ncn3)C)n2)ccc(Cl)cc1 97651,CCCC(C(=O)NC(C1CN(C(c2cc([N+](=O)[O-])c(C)s2)=O)C1)C)C(C)C 97652,c1(CCCC)cc(NCC2CN(C(C3CC4CCC3C4)=O)C2)n2ncnc2n1 97653,c1(C(N2CC(CNC(C(C(C)O)N(C)C)=O)C(O)C2)=O)ccc2c(n1)CCCN2 97654,N1(C(CCCc2onc(CC)n2)=O)CCC2CCN(C(=O)CC(O)CC)CC2C1 97655,C(=O)(CC(C)C(C)(C)C)N1C(C(=O)NC2(C(=O)OC)CCCCC2)CC1C 97656,c1(C(C(=O)NCCC2CC2)N(C2CC(OC)C2)C)ccncc1 97657,c1(C(N2C(CNC(c3cn(CC(CC)O)nn3)=O)C=CC2)=O)cc(N)cc(N)c1 97658,C12(CCNC(CCc3c(C)cccc3)=O)CCC1CN(C(=O)C(C)(C)CF)C2 97659,C1(CNC(=O)C=CCF)CC2CCC1N2C(C1CC2CCC(C1)S2)=O 97660,CC1CCCC(C(=O)NC2CCCC2CN=c2[nH]nc(C3CC3)s2)CC1 97661,N1(C(C(CC)NC(c2cc(S(C)(=O)=O)ccc2F)C)=O)CCc2ccccc2C1C 97662,c1(C(=O)NCC(CC=C)NC(c2ccc([N+](=O)[O-])[nH]2)=O)cccn2cc(C)nc12 97663,C#CC1C(C(=O)NC2CCC(CNC(=O)Cc3csc(NC=O)n3)C2)C1(C)C 97664,C(=O)(CS(=O)(=O)CC(=O)NC(C)(C)C)NC1C(=C)CC1 97665,C#CCCCC(=O)NC(C)CCN(C)C(c1ccncc1Cl)=O 97666,Cc1cn(C)nc1COC(C1(NC(=O)NCc2ccccc2)CCOC1)=O 97667,C1(CNC(C)C)CN(c2ccnc(NCCC3CCCC(C)C3)n2)CCO1 97668,N1(CCNC(C2CCCCC2F)=O)CCCN(C(c2cc(CF)on2)=O)CC1 97669,C=C(Cl)CC(C(=O)NC1C(N)CC1O)NC(c1cnc(Cl)n1C)=O.OC 97670,N1(C(CCC(C)N(C)C)=O)CCCC2(CCN(Cc3nnc(C4CC4)o3)C2)C1 97671,C(=O)(C(C(C)NC(=O)CCCn1cccn1)C(C)C)NCc1cc(C)oc1 97672,c1(C(=O)NCCN(CC(C)O)C(C2CCOC2(C)C)=O)ccc(C(F)(F)F)cn1 97673,n1(CC)ccc(C(=O)NC(c2ncc(C)[nH]2)C2CC2)c1C 97674,C1(NC(C(C2CCC(O)CC2)(C)C)=O)CCC(NC(C23COCC2C3)=O)CC1 97675,C1(C(=O)NC)C2CCC(C2)N1C(C1CCC(NC(=O)NC2CCCC2)CC1)=O 97676,c1(C(=O)NCC(CO)NC(C2CS(=O)(=O)C2)=O)cc(C2CCC2)ccc1F 97677,CCCC(CC)C(=O)NCc1cn(C2CN(C(=O)C(C)(C(C)C)OC)C2)nn1 97678,N1(C(C2C3(CCN(C(=O)CCN4CCCC4)C3)C2)=O)CCc2ncncc2C1 97679,C1(CCC(=O)NC2(CNC(Cc3c(C)ocn3)=O)CC2)CCC(C2OCCO2)O1 97680,CN1CCC(NCCN2CCN(CCOC(=O)CCC3CC3)CC2)CC1 97681,N1(C(c2ccc(S(C)=O)cc2)C(=O)NCCOCC)CCC2(CCN(C)CC2)C1 97682,C1(O)(CNC(C(CN(C(c2c(C)snc2)=O)C)C)=O)CCCCCC1 97683,CC1COC2CN(C(=O)C(N3CCOCC3c3ccc(C(F)(F)F)n3C)=O)CC12 97684,N1(C(c2c(CCC)n(C)nc2)=O)CCC(C)(NC(C2CC2C(C)O)=O)CC1 97685,C1(CN(C(c2cc(CN(C)C)on2)=O)C)CN(C(=O)Cc2cnns2)CCO1 97686,O=S(=O)(C(F)(F)F)NCC(C)NC(c1ccccc1)Cc1ccccc1 97687,CCC(CC(=O)NC1CN(C(=O)Cn2nc(C)oc2=O)CC1(C)C)C(F)F 97688,C1(CC(=O)NC2COC(C3CC3)C2)CC2(C1)CN(C(C13CCC(CC1F)C3)=O)C2 97689,N1(C(C(COC)NC(CCCCC=C)=O)=O)CCC(N=[N+]=[N-])C(O)C1 97690,C1(C)(NC(c2ccc(CNC(C)=O)s2)=O)CCN(C(=O)CC2CCNC2=O)C1 97691,c1(CC(=O)NC(C)(C)CNC(C2COC(=O)O2)=O)ncn2c1CCC2 97692,N1(C(C2C(C(C)(C)C)C2)=O)CC2(CCCN(C(c3cccn3C3CC3)=O)C2)C1 97693,C(=O)(CC(CC)C1CCC1)NCc1cc(OCC)n[nH]1.c1(O)ccccc1 97694,C1(C(C(=O)NCC=C=C)C)CCN(C(c2ccc(C3CC3)cc2)=O)CC1 97695,Cc1ccc(C(=O)NCC2CC(NC(c3cccc(F)c3N)=O)C2)nc1C 97696,N1(C(CNC(CC)=O)=O)CCC(CF)(NC(c2ccc(CO)s2)=O)C1 97697,CC1CCC(N(C(=O)CNC(=O)OC(C)(C)C)N2CCN(CCCO)CC2)C1 97698,C(=O)(CCC(=O)NC1CCCC1)NC(CNC(CC(=C)Br)=O)C1CCC1 97699,C(=O)(C1=CCC(C(F)(F)F)OC1)NC1CN(C(c2c(C)ncn2O)=O)CC1CO 97700,C(=O)(CCCC(=O)N1CC(NC(=O)CCC2OCCO2)CC(F)C1)OC(C)(C)C 97701,N1(C(C(N2CCN(c3ccc(C)cc3)CC2)=O)=O)CCCC(CN(C)C)CC1 97702,C1(CNC(CCOCC(C)(C)C)=O)CC(CNC(=O)C=Cc2cn[nH]c2)CO1 97703,c1(CCC)ccc2ccc(-c3nc(-c4sc5nccc(C)c5c4C)no3)cc2c1 97704,n1(CCCC)cc(C(=O)NCCN(C(=O)C2=CCC2)CCC)c(C)n1 97705,Cc1cc2[nH]c(C(=O)NC3CN(C(C4CC4C(C)O)=O)CC3(C)C)cc2s1 97706,O=C1NCCN(C(=O)NC2CCN(Cc3ccccc3)CC2)C1CC(F)(F)F 97707,N1(C(=O)Cc2nc(Cl)cs2)CCC(F)(F)C(NCc2ccc(OC(F)F)s2)C1 97708,C(=O)(N(CC1CC1)OC)C1C(NC(C2C(CC)OCC2)=O)CCC1 97709,C1(CNC(C2OCCN(C(CN(CC)CC)=O)C2)=O)CCC=CCCC1 97710,c1(CNC(=O)Nc2ccc(N3CCOC3=O)cc2)ccc(-n2cncn2)cc1 97711,CC(C)CC(CNC(=O)CN1CCCC1CO)NC(c1cn(C)nc1C(F)F)=O 97712,c1(OCC)ccc(CN(c2nc(C(C)NC3CNC3)cs2)CC)c2cccnc12 97713,N1(C(C(C)OCC2CC2)=O)CC2CCC1C(CNC(C1C(C)OC(C)C1C)=O)C2 97714,C(C(C(=O)NC1CCC(NC(=O)CC2OCCCO2)C1)C(C)(C)C)OCC=C 97715,CCCC(C)(C)CC(=O)NCC1CN(C(=O)CC2CC23CC3)CCN1C 97716,N1(C(CCC(C)C)=O)C2CCCC1CN(C(=O)CSc1ccccc1[N+](=O)[O-])C2 97717,C1(C(=O)NC2(CCNC(c3cc(F)c[nH]3)=O)CCC2)CC1C1CCCCC1 97718,C#Cc1ccc(OC)c(C(N2CC(OC)C(NC(C3CCCS3(=O)=O)=O)C2)=O)c1 97719,N1(C(c2c(O)ccc(C)n2)=O)CCC2(CCCN(C(C34CCC3C4)=O)C2)CC1 97720,C1(C(N(CC(c2ccccc2)O)C)=O)C2CCC(C2)N1C(c1cncn1C)=O 97721,C1(N(c2c(F)ccc(C)c2)C(=O)C(C)n2cnnn2)CCC12CCNCC2 97722,c1(OC)cc(Cl)ccc1C(=O)NCCCOCCNC(=O)C(C)SC 97723,Cc1c(NC(C2CCN(C(c3cncn3C)=O)CC2)=O)ccc(C#N)c1Cl 97724,Cc1cc(F)ccc1C(=O)NC(C)CNC(=O)C(c1cccn1C)=O 97725,C1(CNC(c2c(C)scn2)=O)C(C)CCCN1C(=O)Cn1cc[n+](C)c1 97726,c1(C(=O)NCCCN(C)C(c2nc(O)nc(O)c2F)=O)nnn2c1C(=O)NCC2 97727,Cc1ccc(Cl)cc1C(=O)NC1CN(C(=O)COC2CCN(C)CC2)CC1C 97728,CCC1=C(C(=O)N2CC(CNC(=O)C(F)(F)c3cnn(C)c3)C2)SCCO1 97729,N1(C(C(CCCC)O)=O)CCC2(CCC(CNC(c3ncoc3C)=O)OC2)CC1 97730,C(=O)(CCCC(=O)N1CC(CCNC(C2CCCOC2)=O)C(C)C1)OC 97731,CCCCC(O)CC(=O)NC(C)(CC)CCNC(c1cc(OC)nc(C)c1)=O 97732,C(=O)(C(F)CC(C)(C)NC(=O)C(CCSC)OC)NCC(C(CC)C)CO 97733,C(C)(C(=O)NN1C(=O)c2ccccc2C1=O)(c1ccc(Br)cc1)OC 97734,N1(CCNC(C2N(C(c3c(C)onc3)=O)CCC2)=O)CCS(=O)(=O)CC1 97735,CC1CCC=C1C(=O)NC1(CCC(=O)NCCCc2cn[nH]c2)CCC1 97736,CC1CCN(C(C2CC(N=[N+]=[N-])C2)=O)C1CNC(=O)CCS(C)=O 97737,c1(C(CSCC(=O)NCc2c(C)cno2)=O)c(C)nn(C)c1C.C12(CC1)C(=O)N2 97738,c1(C(=O)NCC(C2CCCCC2)NC(C(CCOC)C)=O)ccc(C)nc1C 97739,n1(CC)cc(C(=O)NCC2CN(C(=O)CCC3CCC(=O)N3)C2)nn1 97740,CC(C)C(C(=O)N1CC(CC(C)(C)CNC(c2coc(CO)c2)=O)C1)n1cnnn1 97741,c1(C(N2CC(NC(c3cc(C(C)C)[nH]n3)=O)(CO)C2)=O)ccc(Cl)c(Cl)c1 97742,N1(C(C(C)CC(N)=O)=O)Cc2ccc(C(=O)Nc3nccn4ccnc34)cc2C1 97743,c1(N(CC)CC)ccc(NC(C2CCCN(C(C3CCCN3)=O)C2)=O)cc1 97744,N1(C(c2ccc(C)nc2C)=O)CC2CCN(C(=O)C(C)N(C)C)CC2C1 97745,Cn1c(Cn2ccnc2-c2cnc(Cc3ccccc3)nc2)nc2ccccc12 97746,C1(CC)(CC)CC(NC(c2ccc(C#N)[nH]2)=O)CN1C(c1cn(C)nc1SC)=O 97747,c1(CC(N2C(CNC(=O)CC3CC3)CC(O)C2)=O)c[nH]c2ccc(F)cc12 97748,N1(C(c2cn(C(C)C)nn2)C(=O)NC2CCCC2)CCCC(C)(C#N)C1 97749,C(CC(=O)N1CC=C(CCNC(=O)C(C)(C)C)CC1)(C(F)(F)F)OC 97750,CC(O)(C(=O)N1CC2CN(C(C3CNC(=O)C3)=O)CC2C1)C(F)(F)F 97751,c1(OC)ccc(OC)c(C(=O)NCc2ccc(-n3cncn3)cn2)n1 97752,C1(CNC(=O)COCC2CC2)CN(C(c2cnn3c2CCC3)=O)CC12CC2 97753,C(CN=c1[nH]ccnc1F)C1CCC(NC(c2nc(CC)sc2)=O)C1 97754,Cc1ccc(C(C(=O)NCCC2CC2)N2CCC2C(=O)OC(C)(C)C)cc1.N(C)(C)C 97755,N1(C(N(CC(=O)NC2CC(OC(C)(C)C)C2)C)=O)CCCC1c1ccccc1 97756,c1(OC)ccc(C(=O)Nc2nc(C(=O)Nc3ccccc3N(C)C)cs2)c(Cl)n1 97757,N1(C(CCC(=C)C)=O)CC2(CC(NC(C3CCCC3OC)=O)CO2)C1 97758,C(C(C)(CNC(c1cccc(C(F)(F)F)c1)=O)CO)OC 97759,C(CC1=CCN(C(=O)Cc2cnccn2)CC1)NC(CN(C)C1CC1)=O 97760,C1(NC(Cc2c(OC)cccc2)=O)CC2CCC(C1)N2CC1CCS(=O)(=O)C1 97761,C1(NC(=O)C=CSc2nc[nH]n2)CC2CCC(C1F)N2C(C1CCCCCC1)=O 97762,C(=O)(C(C(C)(C)C)N(C)C)NCCSCC(=O)N(C1CN(C)CC1O)C 97763,N1(C(COCCCCC)=O)CCC2CCN(C(=O)Cc3c(Cl)cnn3C)C2C1 97764,C(c1c(Cl)cccc1Cl)=CC(N1CCN(C(C2CC2F)=O)C(CO)C1)=O 97765,N1(C(C(C)OCc2ccccc2)=O)CCc2c(-c3cncc(O)c3)cccc2C1 97766,c1(C(C)=O)c(NCCCCC(C)NC(=O)C(c2ccc(C)s2)C)ncnc1Cl 97767,c1(C(N(CC(N2CC(CC3CC3)C2)=O)C)=O)ccnn1C(F)F 97768,c1(C(=O)NCC(CNC(CC2(C)CC(F)(F)C2)=O)F)cnc2c(c1)NCC(=O)N2 97769,c1(OCC)c(C(=O)NC2CCN(C(C3(C(F)F)CC(F)(F)C3)=O)C2)cccc1F 97770,C12(C(=O)NCCCC(C)(C)NC(CC(CC)C)=O)CCC(=O)N1CCS2 97771,CN1CCCCC1CC(=O)Nc1cc(C(C)(C)C)ncn1.C12CC(C1)C2 97772,Cc1ccc(C(N2CC(NC(=O)Cc3n[nH]cc3Br)C(C)(C)C2)=O)cc1C#N 97773,C1(CC(=O)NCC23C(CN(C(Cc4ccc(C)cc4)=O)C2)C3)CCOCC1(C)C 97774,C12(NC(c3n(CC)ccn3)=O)CCC1CN(C(=O)C(C1CC1)N(C)C)C2 97775,C1(C(C)C)N(C(c2nc(N(C)C(C)C)ncc2Cl)=O)CC12CCS(=O)(=O)CC2 97776,c1(CCC(=O)N(CCCNC(C2OCCCO2)=O)C)ccc(Cl)nc1 97777,C(=O)(CC(F)(F)CC)N(CC(=O)NC(CCSCC)C)C 97778,c1(C(=O)NCC2CCN(Cc3cnc(CCC)s3)CC2)cc(Br)cnc1O 97779,c1(CC(=O)NC2(CC(=O)NC(c3cnn(C)c3)C)CC2)cncnc1 97780,C12(CC3(CCC3)C1)C(=O)OC(=O)N2.c1(C(=O)CNC(C2CC2)C2CC2)c[nH]c(=O)cn1 97781,c1(C(=O)NC2C(CN(C(C(CCOC)OC)=O)C)CCC2)cnc(O)cc1OC 97782,C(=O)(CCCC(C)(C)C)N1CC(C)C(CNC(C2C3CC2(c2cccs2)CO3)=O)C1 97783,N1(C(C2C(C)OCCO2)=O)CC2CCC1CN(C(=O)CC(C)(C)C)C2 97784,Cc1ccccc1-c1cnc(CNC(=O)NCCN2CCSCC2)o1 97785,c1(C(=O)NCC(C)N(C(c2cc(C)ns2)=O)C)ccccc1SC(C)C 97786,C1(CNC(C2(C)CC=CC2)=O)CC2(CCC2)CN1C(=O)COCC1CCCO1 97787,CC1(NC(=O)Cn2cc(Br)cn2)CC(NC(C2(CC3CCC3)CC2)=O)C1 97788,N1(C(c2ccc(CC)[nH]2)=O)CCC(N(C(=O)C(C)COCC)CC)CC1 97789,Cc1cc(Cl)c(Cl)cc1C(N1CCC(C)CC1C(=O)OC(C)(C)C)=O 97790,c1(C(=O)OC)cccn(CC(=O)NCCc2cc(C)[nH]n2)c1=O 97791,N1(C(CCC#CC)=O)CCc2ccccc2C1CNC(=O)CCN(C)C(C)=O 97792,N1(C(CN(CCOC)C)=O)CCCC(C(C)C(N2CC(CO)CC2CO)=O)C1 97793,c1(C(N2CCC(C(C(=O)NC3CC(C)(C(=O)OC)C3)F)C2)=O)ccc(C)nn1 97794,C1(C(N2CCC(CNC(C3(CC(C)C)CCC3)=O)C2)=O)C2CCCCC12 97795,C1(CC)C(C(N2CC(F)(F)C2C2CC2)=O)CCN1C(c1cc(C)n(C)n1)=O 97796,C1(CNC(CCOCCN(C)C)=O)(NC(C2(CO)CCOC2)=O)CCCC1 97797,C(=O)(C(CC)C(F)(F)F)NC1CC(CCNC(C2(CC=C)CC2)=O)C1 97798,c1(CC)cc(C(=O)NC2C=CC(CNC(=O)C(C)=C3CCC3)C2)ccn1 97799,c1(C(N(CCCNC(C2CCCC23CC3)=O)CC)=O)ccc(F)c(CO)c1 97800,Cc1coc(C)c1C(=O)NCC1CCN1C(C1(c2ccc(Cl)cc2)CCCCC1)=O 97801,c1(C(=O)NCC(C)(CO)NC(C(CC(=C)C)C)=O)cccc2[nH]ncc12 97802,C1(NCCOC)Cc2ccc(C)cc2S1.c12cccnc1C(=O)N(C)CCNC2=O 97803,Cc1cncc(CCNC(C2(NC(=O)C=CC3CCOC3)CSC2)=O)n1 97804,c1(NCCOC)ccc(C(=O)NC2CCCCC2NC(c2cocc2C)=O)cc1 97805,c1(C(=O)Nc2cncc(C(=O)NCc3c(C)cccn3)c2)ccc2c[nH]nc2c1 97806,N1(C(C(COC)(C)OC)=O)CC2CC(NC(c3c(Br)nnn3C)=O)C1C2 97807,c1(NC(c2n(CCCSCC)nnn2)CCc2ccsc2)cc(OC)ccc1C 97808,C=CCC(CNC(=O)C(C#N)C(C)C)C(=O)NC(c1cncn1C)CO 97809,Nc1cncc(C(N2CC(CO)(NC(C3CC3c3ccc(Cl)s3)=O)C2)=O)c1 97810,C1(NC(C(c2ccccc2)C)=O)CCN(Cc2c(O)cccc2F)CC1O 97811,C(=O)(CC(C)CN(C)C)NCC(=CC(N1CC(F)(CC)C1)=O)C 97812,CCCCC(C(=O)N1C2CCCC1CN(C(C1CCN(C3CC3)C1)=O)C2)C(C)C 97813,Cc1ccc(C2CC2C(=O)N(CCS)CCN(C)C)o1 97814,C1(C(=O)NCC(C)(O)C2CC2)CCN(C(=O)C2=CCCC2)CCO1 97815,N#Cc1cccc(CN2CC(F)(F)CC2C(=O)Nc2cnc(Br)nc2)n1 97816,C(c1cccc(F)c1F)=CC(=O)N(C1CC(NC(C(C2CC2)OC)=O)C1)C 97817,CCC(CNC(c1cc(COC)[nH]n1)=O)(CC)NC(=O)CC1CC(C(=O)OC)C1 97818,C#CC1CCC(C(N2CCCC(N(C(=O)CCOCC(F)(F)F)C)C2)=O)CC1 97819,C1(NC(c2cc(C)n(C)n2)=O)CC2CC(NC(c3ccncc3O)=O)CC2C1 97820,N1(C(C(CCC)=CC)=O)CCC2CN(C(=O)C(CC#N)c3ccccc3)CC2C1 97821,CC(C(=O)NC(CCN(C)C(c1ccc(C(N)=O)c(Cl)c1)=O)C(N)=O)P(C)(C)=O 97822,C1(C(C)C)CC(NC(=O)C(N)Cc2cccc(Cl)c2)CN1C 97823,CC1CCCC1(C)C(=O)NCc1cccc(CN(C(=O)Cn2cnc(=N)[nH]2)C)c1 97824,c1(C(N2CCC(NC(c3cc(C(N)=O)oc3)=O)C23CC3)=O)occ2c1CCOC2 97825,CC1CN(C)CCN1C(=O)CC1CCCN1C(c1ccc(F)cc1I)=O 97826,c1(OC)ccc(CC(N2CCC(CNC(C3CC4CCC3C4)=O)(OC)C2)=O)cc1 97827,c1(OC)cc(-c2cnc(Cl)c(C(=O)NC(C)C3CC3)c2)c(F)cn1 97828,O=c1c2ccccc2ncn1C1CCN(S(=O)(=O)c2ncc(F)cn2)C1 97829,C1(c2cn(C)nc2)CC1C1CC1C(=O)OCc1ccccc1CF 97830,n1(CC(=O)NCC2CN(C(C(COC)NC(C)=O)=O)CC2O)nc(O)ccc1=O 97831,C(=O)(C(C)(C)C(N)=O)NCC(C(=O)NCC(=O)N(C)O)OC 97832,CN1CCOC(CNC2CCC(CNC(c3cnccc3Cl)=O)CC2)C1 97833,C1(NC(CCC)=O)CC=CCC1C(=O)NCC(=O)NCCCC 97834,c1(C(=O)NC(C)CNC(c2c[nH]c(Br)c2)=O)ccc(F)cc1OC(F)F 97835,Cc1c(C(=O)NCC(C2CC2)NC(=O)C(O)C(F)F)cccc1CO 97836,Cc1ccc(C(=O)NCCn2ccc(C(=O)N(C3COCC3(C)C)C)c2)n1C 97837,C1(c2cccnc2)(C(=O)NCC(CCNC(c2c(C)scn2)=O)O)CC(F)(F)C1 97838,c1(OC)cnc(Cl)[nH]c1=NC1CC2CN(C(=O)CCc3ccc(F)cc3F)CC12 97839,Cc1cnc2n1C(C(=O)N1CCC(C)(NC(c3csnc3Cl)=O)CC1)CCC2 97840,C#CCC(C)(C)C(=O)NCC(CNC(c1ccnn1C1CCC1)=O)C(F)(F)F 97841,S(=O)(=O)(c1cccc(Cl)c1)NCC(=O)NC1C2CN(C(CC(C)OC)=O)C1CC2 97842,C12(NC(c3nccc(OC)c3F)=O)CCCN(C(=O)C(C)SC)CC1C2 97843,C1(NC(c2ncn(CC)n2)=O)CC2CC1N(C(=O)Cc1cccc(C)c1Cl)C2 97844,N1(C(C(C)SC)=O)CC(C2CN(C(=O)COc3ccsc3)C2)C1 97845,N1(C(c2cc(OC)cc(C)n2)=O)CC2CC(C)N(C(=O)CC3CNC(=O)C3)C2C1 97846,O(NC(=O)CCN(C(=O)CC1CCC(C#N)C1)CCO)CC(C)C 97847,C1(CCC)CN(C(=O)C(C)C=Cc2ccccc2)CCN1C(=O)CC 97848,N1(C(c2c(CC(C)C)onc2)=O)CC(NC(c2cn(CCO)nn2)=O)CC(O)C1 97849,Cc1cc(Cl)ccc1NC(=O)C(C)(C1CCC1)NC(C1CC(CF)C1)=O 97850,N1(C(c2c(C)nc(Br)s2)=O)CCC(C)(NC(C2CC(CF)C2)=O)CC1 97851,c1(C(C(=O)NC2CCOC2)N(CC)Cc2cccnc2)nc(C2CC2)cs1 97852,N1(C(C=CCCC)=O)CCN(C(c2cncc(C3CC3)c2)=O)C(CCO)C1 97853,N1(C(CCOC(C)=O)=O)C(CNC(=O)Cn2cc(C3CC3)nn2)CC2COCC12 97854,N1(C(C2CCCC(C)(C)C2)=O)CCC2(CCCCC2NC(=O)Cc2cn[nH]c2)C1 97855,Cc1cc(=NC(C)c2snnc2C)[nH]c(=NCC(C)C)[nH]1 97856,c1(C(N(CC(C)NC(CCOCC)=O)C)=O)cc2cc(Cl)ccc2o1 97857,c1(C(N2C(C(N3CC(C#C)C(O)C3)=O)COCC2)=O)cccc2c[nH]nc12 97858,C(=O)(C1CCc2cc(C)ccc21)NCCC(C)NC(COCCOCC#C)=O 97859,n1(CC)nc(C)c(C(=O)NC2CC(NC(C3(OC)CCCSC3)=O)C(O)C2)c1C 97860,C(CCC(C)(C)C(=O)NCC(O)CC(C)C)NC(C(C)=CC(C)(C)C)=O 97861,CCCCCCCCC(=O)NC(CC)CCCC(=O)N1CCOC2CCC12 97862,C1(CNC(CC(C=C)C)=O)CC2CCC1N2C(c1ccc(CO)s1)=O 97863,Cc1cccc(Cl)c1C(N1CCC(C)C1CNC(=O)CCOCCN(C)C)=O 97864,C(=O)(C#CC1CCCCC1)N(C)CC1CCCCN1C(C1CC(O)CN1C)=O 97865,CCC(C)C(C(=O)NCCCCn1ccnc1)N(C(=O)CC(F)(F)F)C 97866,C1(C(N(CC(C)NC(=O)CCc2ccc[nH]2)CC)=O)CCCN1C1CC1 97867,n1(CC(=O)NCC2(F)CC(NC(Cc3cn(CC)nc3)=O)C2)nc(O)ccc1=O 97868,C1(C(=O)NCC2(O)CN(C(C(C)Cc3ccc(N)cc3)=O)C2)CCC2(CCC2)O1 97869,c1(C(=O)NCC(C2N(C(C(COCC)C)=O)CCC2)(C)C)c(OC)cccc1Cl 97870,c1(Nc2cn(CC)nc2)ccc(NC(=O)C(=O)NC2(N(C)C)CCC2)cc1 97871,CCCCCC(=O)NC(Cc1ccco1)C(=O)NCc1cc(C(N)=O)no1 97872,c1(OC)cc(N)c(Cl)cc1C(=O)NC1(C)CC(NC(=O)C(C)CC2CCC2)C1 97873,C=C1CON(C(=O)C23CC2CCN3C(=O)Cc2ccncc2C)C1 97874,C(N=c1nc2sccc2c(NCC2CC(=O)NC(C)C2)[nH]1)c1nc(C)c(C)s1 97875,N1(C(=O)Cc2ccccc2)CCC(C(C)C(=O)NC2(CC(=O)OC)CC2)C1 97876,CCS(=O)(=O)CC(C)N=c1[nH]c(N(CC(F)(F)C(F)(F)F)C)nc2c1CSC2 97877,CON(CCC(=O)N(C)C)C(=O)NC(CO)CC(C)(C)C 97878,Cn1cc(C(=O)NC2CCC2CNC(c2ccc(C#N)[nH]2)=O)c(C2CCCO2)n1 97879,C1(NC(C=C(C)C2CC2)=O)CC(CNC(c2cc(CO)c(C)o2)=O)C1(C)C 97880,N1(C(CC=C=C)=O)CC2CC(NC(=O)CS(=O)(=O)CCC)C(C2)C1 97881,CCCC(C(O)C(=O)NCCC1CCC(C)(C)C1)NC(c1cc(C)nnc1C)=O 97882,CCC(C)(C(=O)NCC1(C)CC(F)(F)CN1C(c1ccc(F)c(O)c1)=O)C(N)=O 97883,C12(C(N3CC(O)(CNC(CSc4ccc(C)cc4)=O)C3)=O)CCC(C)(CC1)OC2 97884,N1(C(C(C)CCO)=O)CCCC(C2CN(C(=O)C(F)(F)C(C)O)C2)C1 97885,O=C(NN1CCOC1=O)c1cccc(NC(N2CCCC2)=O)c1 97886,c1(COC(c2ccc(-c3ccc(OC)nc3)nc2)=O)ccc(OC)cc1F 97887,C(=O)(CC(CC)C(F)F)N(CC(=O)NCc1cccnc1)CCC 97888,N1(C(C(CO)OC)=O)CC2(CNC(c3sccc3NS(C)(=O)=O)=O)CCC1CC2 97889,C1(CC(=O)N(CC(COCC)O)C)CN(C(c2nnsc2C)=O)C(C)(C)C1 97890,c1(C(C(=O)N2CC(CNC(c3cc(C(F)(F)F)sn3)=O)C2)(F)F)cc(Cl)ccc1Cl 97891,C1(NC(C2N(CCC)CCC2)=O)CCCN(C(C2(CC)COC2)=O)C1 97892,c1(CN(CC(=O)Nc2n(C(C)C)ncc2)C)cccc(Cl)c1 97893,Cc1cc(=NCCCCC2(C)OCCO2)[nH]cc1S(=O)(=O)N(C)C(C1CCC1)C 97894,CCS(=O)(=O)c1ccc(C(=O)NCC2CN(C(=O)C(C)CO)CCCO2)cc1 97895,C1(C(=O)NC(C(=O)N(CC)CC)C)CN(C(=O)Cc2scnc2C)CC1C1CC1 97896,C(=O)(CC(C)(C)C#N)NCC1CN(C(c2ccc(C(C)C)cc2)=O)CC1C 97897,Cc1ncc(C(N2CC(NC(c3cccc(Cl)n3)=O)C(C)C2)=O)n1C 97898,N1(Cc2ncc(CC)o2)CC(C)(C)CCC1CNC(c1nc(C)ccc1C)=O 97899,C1(C2CCC2)(C(=O)NCCCC(C)NC(C2CCCN2C)=O)CCC1 97900,CC(C)CC(C(=O)N1CCCC(N2CCN(C(=O)CC(C)F)CC2=O)C1)N(C)C 97901,C1(COC(C)C(N2CC(C)(CNC(C3(C)CC3C)=O)C2)=O)CCCCO1 97902,C(=O)(CCCCC(=O)NCC1CCN1CC1(O)CC1)OC 97903,C1(C(=O)ONC(C2CCN(CC#C)CC2)=O)CN(C(=O)CSC(F)F)C2CCCCC12 97904,c1(C(N(CC(=O)NC(CCCC=C)C2CC2)C)=O)cc(C)cc(O)n1 97905,c1(NC(C(c2ccc(SC)cc2)N(C(COC)C)C)=O)ccc(F)cc1 97906,c1(C(=O)NCC=CC)n[nH]cc1CNC(=O)C(C)n1cccn1 97907,c1(C(C)CC(=O)NC2(CO)CN(C(=O)CCN3CCCC3)C2)cccc(F)c1 97908,CC1CN(C(c2coc(C(F)(F)F)c2)=O)CCN1C(C1CC1c1cnc[nH]1)=O 97909,c1(CC(=O)NCC(CC)(C)NC(=O)C(C)CC(N)=O)sc2ccccc2c1C 97910,c1(CC(=O)Nc2ncc(-c3ccc(OCCCC)cc3)s2)cc(F)cc(Cl)c1 97911,CC1(C)CC(C(=O)Nc2cnc(F)nc2)(CNC(C2C(C)(C)C2(F)F)=O)C1 97912,N1(C(C=CC(C)NC(C(C)(C)NC(C)=O)=O)=O)CCC(O)(CO)C1 97913,N1(C(CCNC(C(C)(C)C)=O)=O)CCCC(O)(CNC(=O)CSCC(F)(F)F)CC1 97914,C1(CC(=O)NC2(CCOC)CCN(C(=O)C=CI)C2)OCCCC1(C)C 97915,c1(CC(=O)NCC(C2CCCC2)NC(CC=C)=O)ccc(Br)cc1 97916,C1(COC)(NC(=O)CCCc2cccs2)CCN(C(=O)C(C)CF)C1 97917,N1(c2nnn(C)n2)CCCCC1CNC(C1COC(=O)N1C)=O 97918,Cc1cccnc1C(=O)N(CCCNC(=O)CCC1CCCC1)C(C)C 97919,Cc1cc(C(=O)NC2(CNC(c3ccccc3Br)=O)CCOC2)cc(O)c1 97920,c1(C(N(C(C)CNC(=O)Cc2ccc(OC(C)C)cc2)CC)=O)cn(C)c(O)n1 97921,C1(C(=O)NCC2CN(C(CC(=C)C)=O)CC2C(F)(F)F)Cc2nnc(C)n2C1 97922,C1(NC(C2(OC)CC2)=O)CCCCN(C(=O)CC2(O)CCCOC2)C1 97923,N1(c2ncc(CC)cn2)CCC(F)(F)C(CNC)C1.c1(C=O)cnc2n1CCS2 97924,n1(CC(=O)NCC(CNC(C(CC)c2cccnc2)=O)F)c([N+](=O)[O-])cnc1C 97925,c1(OC)cccc(CC(N2CC3CC2C3C(=O)NCc2cccc(F)n2)=O)c1 97926,C1(c2nc(C)[nH]n2)COCCN1C(c1ccc(Br)cn1)C(=O)NCC(C)C 97927,Cc1ccc(F)c(C(=O)NC(Cc2cn[nH]c2)C(=O)NC2CC3CCC2O3)n1 97928,c1(C(=O)NC)ccc(C(=O)NC2CCC2NC(c2cc(O)ccc2Cl)=O)cc1F 97929,C1(CNC(=O)CC2CN(CC)C2)CCN(C(=O)C(CCC2CC2)N(C)C)CC1 97930,n1(CC(=O)NCCCOCCNC(=O)Cc2cc[nH]n2)cc(CO)nn1 97931,C1(NC(c2c(C)nc(C)o2)=O)CCC(C)N(C(C2CCN2C)=O)C1 97932,CCCCCC(O)C(=O)NCCCCCCNC(=O)C(C)OCC 97933,c1(C2CC(C(N3CCC(OCCNC(CC)=O)C3)=O)C2)cccc(F)c1 97934,O=C(C1=CSCCO1)NCC1(CNC(c2ccc([N+](=O)[O-])o2)=O)CC1 97935,N1(C(CC2(OC)CCC2)=O)CCCCC1C(=O)N(C1CCC1C)C1CC1 97936,CCC(C(=O)N(CCCNC(=O)CC1CC(F)C1)C)NC(N)=O 97937,N1(C(c2cnn(-c3ccccn3)c2)=O)CC2CCCC(C1)C2(F)F 97938,C1(CC)C(=O)NCCN1C(=O)C(F)C(C)CNC(=O)COc1cnn(C)c1 97939,c1(Cn2c(CC3CC(C(F)F)C3)nc(-c3cn(C)nc3)n2)c[nH]c2ccccc12 97940,C(=O)(C1=NOC2COCC12)NC1CCC(C(N(C(C)C(C)(C)C)C)=O)C1 97941,N1(C(CC=CCCCCC)=O)CCC(C)(C(=O)N(C2CC3(CCC3)C2)C)C1 97942,c1(C(=O)NCc2c(C(N3C(COC)CCC3)=O)c[nH]n2)cncc(C)c1 97943,N1(C(C(C)C(F)F)=O)CC(NC(=O)CC2CC(C)(C)C(=O)N2)CC12CCCCC2 97944,N1(C(C2CCN(C)C2=O)=O)CC(C2CCN(C(c3ncn4c3CCC4)=O)CC2)C1 97945,Cc1cccc(C2(C(=O)NC(C3CCN(C(C4(O)CCSC4)=O)C3)C)CC2)c1 97946,C1(CC)CN(C(=O)CCOCC(C)(C)C)CCN1C(c1cnn(C)c1OC)=O 97947,CN1CCC2C(CCCN2C(c2cn(C)nn2)C(=O)NC2COC2)C1 97948,Cc1noc(C2CN(C(=O)CC(C)N(C(=O)C(C)OCCN(C)C)C)C2)n1 97949,Cc1cc[nH]c(=N)c1C(=O)NCC1(C)CCN(C(c2c(C)ncn2C)=O)CC1 97950,C1(NC(C2CC(=C)C2)=O)CC2CC(NC(=O)C(C)CC3CCCCC3)CC2C1 97951,C1(C(N(C2CCN(C(c3n[nH]c(O)n3)=O)C2)CCO)=O)CCC2CC2C1 97952,C(=O)(CCS(=O)(=O)c1ccc(F)cc1)N1CCN(C(CC=CC)=O)C(C2CC2)C1 97953,c1(C(N2C(C)(CC(=O)OCC)CC2)=O)cncc(-c2cc[nH]n2)c1 97954,N1(C(CSCC(C)C)=O)CCC(C)C(CNC(=O)C(C)(C)C#N)C1 97955,c1(OC)cccc(C(F)F)c1C(N1CCC(NC(=O)C(C)(C)CF)C(CO)C1)=O 97956,n1(CC)nccc1C(=O)NCC1CC1CNC(=O)CNC(c1cnn(C)c1)=O 97957,c1(C(C(=O)NCC=C)N(C)Cc2cnn(C3CC3)c2)cccc(O)n1 97958,C=C=CC(C)C(=O)NCC(C)(C)OCC(=O)Nc1ccc(O)nc1 97959,CN1CCC2(CCN(C(C3C4CCC(C4)N3C(=O)CCC(F)(F)F)=O)CC2)CC1 97960,CC(C)C(O)C(F)(F)C(=O)NCC1CC(F)CN1C(C1CC2CCC1CC2)=O 97961,C1(NC(CNC(=O)OC)=O)CC2CCC1N2C(c1ccn2ccsc12)=O 97962,n1(CC(=O)NCC(CO)NC(c2n(CC#N)ncc2)=O)nc(C(F)(F)F)cc1Cl 97963,c1(CC)cnc(C(N2CC(NC(c3ccc(NC(C)=O)cn3)=O)CC2C)=O)cn1 97964,c1(CNC(=O)NC23COC(COC)(C2)C3)ccccc1NS(CC)(=O)=O 97965,CC(C)C(C(C)NC(c1ccc(C(F)F)s1)=O)NC(c1cnc(S)[nH]1)=O 97966,C1(COC)CCN(C(=O)C(CC2CCC2)NC(c2ccns2)=O)C1 97967,c1(C(N(C2CCN(C(C(C(=O)OC)OC)=O)C2)C)=O)cnn2c(C)ccnc12 97968,C1(C)(C(=O)NC(c2cccnc2O)C)C=CCN1C(c1cc(C2CC2)[nH]n1)=O 97969,C(=O)(CCC(N)=O)N(C1CCN(C(=O)C(CCSC)N(C)C)C1)CC 97970,c1(C(=O)NC(C2CCN(C(=O)CSc3ccccc3)C2)C)ccc2scnc2c1 97971,c1(C(=O)OC)ccc2cnn(CC(N3C4CSCC3C4)=O)c(=O)c2c1 97972,CC1CC=CCC1C(=O)NC(c1cnn(C)c1)C(=O)NC1CCC(F)CC1 97973,N1(C(C(CC)C)=O)CCCC12CCN(C(c1ccccc1[N+](=O)[O-])=O)C2 97974,N#CC1(C(N2CC3(C2)CN(C(=O)COCCN(C)C)C3)=O)CC2CC2C1 97975,c1(C(N2CCC(c3cnc(C)o3)C2)C(=O)NC)ccc(F)cc1.c1(C2CC2)ccccc1 97976,N1(C(C=C)=O)CCC2(CCC2)C(NC(C2CCc3cncn3C2)=O)C1 97977,Cc1noc(CCOCC(=O)Nc2ccc(CN3CCOCC3)cc2)c1C 97978,c1(N2C(C(N3CC(NC(C=CC(=O)OCC)=O)C3)=O)CCC2)ccc(Cl)cc1 97979,N1(C(C(C)O)=O)CCc2nc[nH]c2C12CCN(C(=O)C(F)Cl)C2 97980,C=CCC(Cc1ccccc1)N=c1nc2c(ncn2C)c(NC2C=CCCC2)[nH]1 97981,C(=O)(C#CC1CCCCC1)NCCCC(=O)NC1(CC(=O)OCC)CCC1 97982,N1(C(C2(CC#C)CCOC2)=O)CC(C)N(C(=O)CC2CC(C)(C)C2)C(C)C1 97983,c1(C(=O)NCCn2cc(CCCC(O)c3cccs3)nn2)ccc2nccn2c1 97984,N1(C(C=Cc2ccc(C)o2)=O)CCOCC(CNC(c2ccoc2C2CC2)=O)C1 97985,N1(C(Cn2c(CCC)ncc2)=O)CCN(C(=O)CC2(CO)CC2)C2(CCC2)C1 97986,CC(C)(C(=O)NCC(C1CCCC1)NC(=O)Cc1cnc[nH]1)Oc1ccccc1 97987,C12(C(=O)NC3C(CNC(C(C)OCCCC)=O)C3)CC3CC1C2C3O 97988,C1(C2CCOCC2)(C(N2CC(CNC(=O)CCc3ccccn3)C2)=O)CC1(F)F 97989,S(=O)(=O)(c1cc(C(N)=O)co1)N1C(CC)CCCC1 97990,c1(OC)cc(C(=O)NC(C2CCN(C(=O)Cc3sccc3C)CC2)C)ccc1F 97991,C1(C(=O)NC(c2cccnc2O)C)CCCC(NC(=O)CCOC2CCC2)CC1 97992,C1(NC(c2nc(Cl)sc2Cl)=O)CCCCN(C(C2CN3CCC2CC3)=O)CC1 97993,N1(C(c2nc(COC)sc2)=O)CC2CC1C2CNC(c1n[nH]cc1Br)=O 97994,Cc1ccc(F)c(CNC(C2(C)CCCN2C(=O)CCN2CCCC2=O)=O)c1 97995,c1(NC(C2CCN(C(C=C(C)c3ccco3)=O)CC2)=O)c(O)cccc1O 97996,c1(OCC)cccc(CC(N2CCC(CCNC(C3(C)CC(O)CN3)=O)C2)=O)c1 97997,c1(OC)c(C(=O)NCC(C)(C)CNC(=O)CCCc2ncc(C)o2)cccc1F 97998,n1(CC)cnc2c(NC3CC(NC(=O)COCC4CC4)C3)ncnc12 97999,C1(NC(c2ccc(C)cc2)=O)CN(C(=O)C(C2CCCCC2)N(C)C)CC1(C)C 98000,C1(C(C)C)CN(C(=O)CC(F)(F)F)CCN1C(=O)C(C)OCC(F)(F)F 98001,c1(CC(=O)NC(CC)(C)CNC(c2n[nH]cc2Br)=O)ccc(F)c(F)c1 98002,c1(C(=O)NCCCN(C(C(C)OCC2CCCO2)=O)C2CC2)ccc(=O)n(C)n1 98003,C1(C(N2CCC(Cc3ccc(-c4cccc(C)c4)s3)C2)=O)Cc2c[nH]nc2CN1 98004,Cc1cc(C2CCCN2C(=O)NC(c2cccc(Cl)c2)(C)C)c(C)o1 98005,C(=O)(CCP(C)(C)=O)NCC(CC)(CC)NC(C1CC12CCOC2)=O 98006,N1(C2CCC(NC(C3(C(N)=O)CC3)=O)C2)CCN(C(=O)C=Cc2cnc[nH]2)CC1 98007,C#CC1(NC(=O)C(CC(C)CC)NC(c2coc(C)n2)=O)CCCCCC1 98008,N12CC3C(C3C1)C2=O.C(=O)(CCCCN1CCCC1)NC1C(c2ccn(C)n2)C1 98009,c1(SC)c(C(=O)NC2CC(N(C(=O)CC3CC(C)=NO3)C)C2)cccc1F 98010,C1(NC(c2ccc(C)nc2)=O)C2CC3CN(C(=O)CN4CCC(C)(O)C4)C1C3C2 98011,c1(C(=O)NC(c2cn(CCOCCO)nn2)CCC)cc2cccc(Br)c2o1 98012,c1(COC(C)(C)C)cc(C(=O)NC2CCC2NC(c2csnn2)=O)no1 98013,C(=O)(C(C)C(C)NC(c1ccnc(CO)c1)=O)N1CC(CC(=O)OC)C1 98014,c1(CC(=O)NC2C(NC(Cc3cc(C)ns3)=O)COC2)cccc(C(C)C)c1 98015,C1(NC(c2c(OC)cc(C)cc2)=O)C(C)CCN(C(=O)C(C)C2CCOC2)C1C 98016,C1(C(CNC(COCC)=O)F)CCN(C(c2nnsc2-c2ccccc2)=O)CC1 98017,c1(C(=O)NC2CC(CNC(C3(n4nccn4)CC3)=O)C2)ccc2c(n1)OCCO2 98018,C1(C(N(CC(CC)NC(c2cscc2C2CC2)=O)CC)=O)CCC(C)(C)C1 98019,Cc1cccc(F)c1CNC(C1CCCN(C(C2CC2C)=O)C1)=O 98020,CCC(C)(CO)C(=O)NCc1cccc(CNC(C2CC3(C2)CC3(F)F)=O)c1 98021,c1(C(N2C(Cn3cc(CNC=O)nn3)CCC2)=O)ccc(S(F)(F)(F)(F)F)cc1 98022,CC1CC2(CCN(CC3CCCS(=O)(=O)C3)CC2)CN1C(=O)CCS(N)(=O)=O 98023,N1(C(C(C)CF)=O)CC2CC(NC(=O)CSCc3ccccc3Cl)C1C2 98024,N1(C(C(=C(C)C2CC2)F)=O)CCCN(C(=O)CC2(C)CCS(=O)(=O)N2)C(CO)C1 98025,C(=O)(C(=O)N(O)C(C)C)NCCN(C(c1c(C)ccc(C)n1)=O)C1CC1 98026,CC(c1ccccc1)=CC(=O)NCCNC(C1CC(C(F)(F)F)C1)=O 98027,c1(COC)csc(C(=O)NCC2(CO)CN(C(=O)C(F)=C(C)C)C2)c1 98028,C(=O)(CCC(=O)CCC(=O)c1cccs1)OC(c1ccc(OC)c(OC)c1C)=O 98029,C12(CNC(C3CC(C)(O)C3)=O)CCC1CCN2C(=O)CCc1ccccc1Cl 98030,C1(NC(=O)CCN2C(=O)C(=Cc3cccc(Br)c3)SC2=S)CCCCC(F)(F)C1 98031,CC1CN(C(C2(CNC(=O)CCC3CCCN3C)CCC2)=O)CCN(C)C1 98032,S(=O)(=O)(c1ccc(NCC2(C)CCN(C)C2)c(Cl)c1)N1CCC2(CC(OC)C2)C1 98033,C1(N(C(c2c(CC)ncs2)=O)C)CCC(NC(C2CC23CC3)=O)CC1 98034,c1(C(N2C(C(=O)NC3CC(C(=O)OC)C3)CC2)=O)cnc(C2CC2)nc1 98035,C12(NC(C(c3ccc(C)cc3)C)=O)CCC1CN(C(=O)CN(C)C(C)C)C2 98036,CC(=O)CCCC(=O)NC1(C(=O)NCCc2noc(=O)n2C)CC(F)C1 98037,c1(C(=O)NCCN(C(=O)C(C)(CC)CO)CCC)ccc(Cl)nc1OCC 98038,N1(C(C2N(C)CCCC2)=O)CCC2(CC(NC(c3cc4n(c3)CCOC4)=O)C2)C1 98039,c1(OC)cc(N(C)CC2CCN(C(=O)CC3CC=CCC3)C2)nc(OC)n1 98040,c1(C(N(C)CCNC(c2ccc(=N)[nH]n2)=O)=O)ccc2oc(O)nc2n1 98041,C1(C(N2CC(CC)(CC)C2)=O)(CF)CCN(C(=O)CC2CC2COC)C1 98042,C1(CC=C)(NC(=O)CCCNC(C)=O)CC2CCC(C1)N2C(c1c[nH]c(=N)o1)=O 98043,CC(C)C(F)(F)CC(=O)N1CCN(C(C2CC(CC(F)(F)F)C2)=O)C(C)C1 98044,N1(C(=O)CCc2nc[nH]n2)CCN2C(=O)NCCC2C1 98045,C(=O)(CCN=C(NCc1cccc(C)c1C)NCC12CCC(C)(CO1)C2)NC 98046,CC1CN2CCCC2CN1C(C1CC(C)(C)CCN1C(=O)CCC(N)=O)=O 98047,C(=O)(CCC(CC)OC)NC(CCCNC(C1(COCC)CCC1)=O)C 98048,c1(CC)ccc(OC)cc1C(N1CCC(CO)(NC(c2cnc(O)s2)=O)CC1)=O 98049,N1(C(C2=C(C)OCC2)=O)CC2CCC(C1)C(NC(C1CC3(C1)CC1(CC1)C3)=O)C2 98050,Cc1ccc(SCC(=O)NCC(C)NC(c2cc(C)nn2C2CCC2)=O)cc1 98051,c1(C(C)C)ncncc1C(N1CCN(CC(C)NC(=O)CC2(C#N)CC2)CC1)=O 98052,C1(CN(C(c2cn(CCC(C)C)nn2)=O)C)C2CN(C(=O)C(CO)N(C)C)CC12 98053,C1(NC(CC(C)C)=O)CC(NC(c2ccc(O)c(C(C)C)c2)=O)C12CCOCC2 98054,C1(NC(=O)CCN2CCOC2=O)CN(C(C2CC3(C2)CC32CC2)=O)CC12CC2 98055,c1(C(=O)NC2CN(C(c3c(C)cc(N)cc3)=O)CC2F)cccc2c[nH]nc12 98056,C1(NC(CCOC(C)=O)=O)CCN(C(=O)C(C)Sc2nncn2C)CC1C 98057,c1(C(=O)NC(C)COC2CNC2)ccc(N=NC(N)=O)cc1.C1(C)CC1 98058,CC(C)C(C(=O)NCCOC1CC1)C(C)NC(C1CC(F)(CF)C1)=O 98059,C=CCC(C)(C)CC(=O)NCC1(O)CC(CNC(C2CCCC23CC3)=O)C1 98060,N1(C(C2(CC)CC2)=O)CCOC2(CCS(=O)(=NC(=O)C3(C)CCCC3C)CC2)C1 98061,C1(C(N(C(C)C(=O)NCCCC(C)CO)C2CC2)=O)CCC(=O)N(C)C1 98062,C(C)(C)(CCC(=O)N1CSCC1C(=O)NCc1snnc1C)OC 98063,CC(C)C(F)(CNC(c1cccc(O)c1F)=O)C(=O)Nc1ccc(F)cc1F 98064,N1(C(CC(C(C)C)C)=O)CCC(CNC(=O)CCCc2ncco2)C(F)(F)CC1 98065,C1(C(=O)NC2(C(=O)NC3C(C#N)CCC3)CC(CO)C2)Cc2ccccc2C1 98066,CC(=O)CCCCC(=O)NC(CC(=O)NC1C=CCC1)C(C)C 98067,c1(C(=O)NC2CC(C)(C(=O)OC)C2)cncc(-c2ccc(Cl)cc2)c1 98068,C1(C(=O)NCC2N(C(C(C)(C)C(N)=O)=O)CCC2)CN2CCCC2CO1 98069,C1(CNC(Cc2c(C)cc(F)cc2)=O)CCC2CN(C(=O)Cn3cnnn3)CC12 98070,N1(C(C(CC)NC(N)=O)=O)CCC(OCCCNC(=O)C=CC(C)(C)C)CC1 98071,C(=O)(C1CCCn2nccc21)NC(C1CN(C(c2ccc(=O)n(CCO)c2)=O)C1)C 98072,N1(C(C=C(C)C)=O)CC(CCO)(NC(C2(C3CCCCO3)CC2)=O)C1 98073,C1(NC(N(C)Cc2nnc(O)o2)=O)CNC(=O)C12CC2 98074,N1(C(c2c(CC)ncs2)=O)CCC(C(N2CC(NC(N)=O)C2)=O)CC1C 98075,C(CC)(CCC(=O)N1CC(O)CC(O)C1)NC(C(C=C)OC)=O 98076,c1(COC)cc(N2CCCC(C3CCCCN3C(C3CC3C(C)O)=O)C2)ncn1 98077,N1(C(c2c(C)[nH]nc2Cl)=O)C2CCC1CC(C(N1CCCC(C)(N(C)C)C1)=O)C2 98078,Cc1noc2ncc(C(N3CC(CNC(c4cc(F)cc(Br)c4)=O)C3)=O)cc12 98079,C12(C(=O)NCCC3CN(C(COCC=C)=O)CC3C)CCC(N(C)C)(CC1)CC2 98080,C1(NC(c2cccc(COC)n2)=O)CN(C(C2CC2C)=O)CC(C)(C)C1 98081,C1(C(=O)NCc2c(OC)nsc2)C(C)OCCN1C(=O)CC1CCN(C)C1=O 98082,N1(C(c2c(C)cc(CO)o2)=O)CC2(CNC(=O)C(C3CCOCC3)O)CCC1C2 98083,c1(C(C)NCC2C(C)CN2C(=O)OC(C)(C)C)nc(N(C)C)co1 98084,N1(C(C(C)(C)CO)=O)CCC2(CCOC2)C(CNC(C23CCC(CC2)OC3)=O)C1 98085,N1(C(C23CCCCC2C3)=O)Cc2cc(Cl)ccc2CC1CO 98086,C1(CNC(C=CCC)=O)(CO)CCCN(C(=O)C(C)OCCCCCC)C1 98087,c1(C(=O)NC2(CF)CCN(C(C(C)(C)c3cc[nH]n3)=O)C2)cc2c(s1)CCC2 98088,O=C1OC(CNC(c2cccs2)C2CC2)CC12CCOCC2 98089,c1(C(N2C(CNC(COCC(C)C)=O)C=CC2)=O)cccc(-n2cnnn2)c1 98090,C1(NC(C(C)n2cncn2)=O)(CO)CCN(C(=O)CC2(CN(C)C)CCC2)C1 98091,C(=O)(CCC(F)(F)Cn1cc(CC(O)C2CC2)nn1)NC(c1cc(Cl)sc1Cl)C 98092,C12(CNC(Cc3scc(C)c3)=O)CCCC1N(C(=O)CNc1cn[nH]c1)CCC2 98093,C1(CC(=O)NCCC(=O)NCC#C)CCCN(C(=O)C(C)N(C)CC)CC1 98094,C=CC1(C(N2CCC(O)(CC(C)C)C2)=O)CCN(C(c2ccc(Cl)o2)=O)C1 98095,c1(C(=O)NCCCNC(=O)C=CCN2CCCC2)c(Cl)csc1Cl 98096,CC1(C)CC(CNC(=O)C=CC2CC2)N(C(C2CCC(C)(C)O2)=O)C1 98097,C1(C(N2CCC(NC(C(C)=C3CCC3)=O)C2C)=O)CCOC2(CCC2)C1 98098,C(CCNC(c1ncccn1)=O)(C(=O)NC1COCCC1O)OC 98099,CCCC(CCCNC(=O)Cn1nc(C)n(C)c1=O)NC(c1cc(C)[nH]c1C)=O 98100,c1(C(=O)NCC2(CC(=O)N(CC(C)(C)O)C)CC2)cc(=N)[nH][nH]1 98101,C(=O)(C(C)C(F)(F)C(F)F)NCC(CNC(c1ccc(C(C)C)nc1)=O)(C)O 98102,c1(C(N(C2CN(C(c3c(CC)nc[nH]3)=O)C2)C)=O)ccc(O)c2c1CCCC2 98103,c1(NCC(C)N(C)C)ccc(S(=O)(=O)N2CCOC(C3CCOCC3)C2)cc1Br 98104,N1(C(c2cc(CNC(=O)Cc3cnoc3)no2)=O)CC2CCC(CC2)C1 98105,N1(Cc2cn(C(C)C(=O)N3CCC3CC3CCOCC3)nn2)CCCCCC1 98106,C1(NC(C(N2CCC(C)CC2)=O)=O)CC2CCC1N(C(=O)C(C)C(C)O)C2 98107,CCC(C)(C)C(C)CC(=O)N1CC(NC(c2cc(Br)n(C)n2)=O)C(F)C1 98108,C(=O)(CCCN(C)N=O)N1C(C(C)NC(C2CC3C(C2)C3(F)F)=O)CCC1 98109,CC(C)(CN=c1ccnc(C(C)(C)C)[nH]1)NCCCOCCNC1CC1 98110,c1(OCC(=O)NCC2(F)CCN(C(C3C(CC)C3)=O)C2)ccc(Cl)c(Cl)c1 98111,O(S(=O)(=O)c1cc(Br)ccc1Br)c1ccc(-c2ccc(COC)cc2)cc1CO 98112,N1(C(c2csc(CO)n2)=O)CC2CCCCC2(C2CCCN2C(=O)C2CC2)C1 98113,N1(C(C(C2CC2)OC)=O)CCCC1C1CCN(C(C2CC(C(F)(F)F)C2)=O)C1 98114,Cc1c(Br)noc1C(N1CCC(O)(CN(C(=O)C2=C(Cl)CC2)C)C1)=O 98115,S(=O)(=O)(c1c[nH]ccc1=NCC1CCS(=O)(=O)N1C)NC(C)Cn1ccnc1 98116,C1(C(=O)NC(C)CF)C2CCC(C2)N1C(c1ncccc1Cl)=O 98117,c1(C(N2CCC(N(C(C3CC3C)=O)CC)C2)=O)ccc2oncc2c1 98118,C1(C(=O)Nc2cnc(I)cn2)CN(C(c2cccc(CO)c2)=O)CCC1O 98119,C1(C(=O)OCCSCC(F)(F)F)CCCN1C(=O)Cc1ccccn1 98120,c1(C(NNC(C2COCCN(C(C)=O)C2)=O)=O)ccc(Cl)c(Cl)c1F 98121,c1(C(=O)NCC(C)CN(C)C(C2CC(F)(CF)C2)=O)c(C#N)ncn1C 98122,C1(NC(c2cc([N+](=O)[O-])c[nH]2)=O)CC2CCC1N(C(=O)Cc1ccno1)C2 98123,c1(C(N(CCC(C)NC(c2ccc(C3CC3)o2)=O)C)=O)ncccc1Br 98124,C(C(C)NC(=O)Cn1nc(C)cc1C)(C(C)C)NC(CCC#C)=O 98125,c1(OCC(=O)NC2CC(NC(C3CS(=O)(=O)C3)=O)C(O)C2)cccc(F)c1 98126,C1(CC(N2CCC(CCNC(=O)CN3CCCNC3=O)C2)=O)CC2C=CC1CC2 98127,N1(C(CCOCC#C)=O)CCCC(CCNC(c2cc(CC)[nH]n2)=O)C1 98128,Cc1nc(NCc2n[nH]c3c2CCC3)cc(=NCCc2nccn2C2CC2)[nH]1 98129,C=CC1(CC(N2CC(CO)(CF)C2)=O)CN(C(C2CCC(C)C2)=O)C1 98130,C1(CN(C(=O)Cn2cccn2)C)CCCN1C(C1(CF)CC1)=O 98131,Cn1ncc2c(NC3CC3(F)F)nc(N3CC4C5CCC(C5)C4C3)nc12 98132,C#CCCCC(=O)N1CCCC1C(C)NC(C1CC=C(C)CC1)=O 98133,N1(CC)CC(CNC(C2(CC)CCN(C(=O)C(C)NC=O)C2)=O)OC1=O 98134,c1(C(=O)NCC(CC=C)NC(=O)COC(C)(C)CC)ccc(C(F)F)c(F)c1 98135,Cc1cc(C(=O)NC2CC3(C2)CC(Nc2cc(Cl)nc(C)n2)C3)cc(O)n1 98136,CC1CC=C(C(=O)N2CC(C)(C)CC2CNC(c2sccc2C(C)(C)C)=O)CC1 98137,C1(CNC(c2c(OC)cccc2)=O)CCC2(CN(CCC(=O)NC(C)C)C2)O1 98138,N(C(=NCCC1(O)CCC1)NCC1C2(CC2)C12CC2)C(c1ccccc1)C 98139,C1(CNC(CC2(C)CC2(F)Cl)=O)CC2(CO1)CN(C(=O)COCC(F)(F)F)C2 98140,N1(CC(=O)NC(CC)CN(C(C2(OC)CCC2)=O)CC)CCC(C)C1 98141,N1(C(C2CCC(C)C2)=O)CC(C)CN(c2ncncc2Cl)C(C)C1 98142,C1(CNC(C2C(C)(C)C2)=O)CCCCCN1C(=O)C=Cc1cc(Cl)sc1Cl 98143,C1(C(=O)NC(C)C(C)(C)NC(c2cnc3occc3c2)=O)CCc2nnnn2C1 98144,c1(NC(c2ncccc2Br)c2n(CCSC)nnn2)ccc(C)c(C)c1 98145,CC1CC2(CO1)CN(C(=O)CCN(CCO)C(c1coc3c1COC3)=O)C2 98146,c1(C(N2CCC(NC(C3CCCN(C)C3)=O)(CO)CC2)=O)cc2ccncc2s1 98147,c1(C(=O)NCC2COCCN(C(C(CCCC)O)=O)C2)c(C)nn2cccnc12 98148,c1(NC(=O)NC2CCc3c[nH]nc3C2)nc2ccccc2cc1[N+](=O)[O-] 98149,C=CCCC(C)(C)C(=O)N1CC2CC2(CNC(c2ccnc3[nH]nnc23)=O)C1 98150,c1(CC(=O)OC(c2ccc(OC)cc2)CC)c(F)cccc1F 98151,c1(C(=O)NCC2C(CNC(c3ccc(SC)cc3)=O)C2)cc(C2CC2)nc(Cl)c1 98152,C1(NC(C(C)O)=O)CCCCC12CCCN(C(=O)CC1(O)CCC1)C2 98153,C(=O)(CC(C)C(C)(C)C)NC(C1CCCC1)CNC(c1nc(CC)sc1N)=O 98154,c1(OC)cc(C(=O)NCCC2(O)CN(C(c3cc(Cl)ccc3O)=O)C2)cc(Cl)n1 98155,C1(C(N(CC(Cl)Cl)C)=O)C(NC(c2ccccc2)=O)C1(C)C 98156,CC1CC(C(=O)N(C2CCCCCC2)CCNC(c2cncc(F)c2)=O)C(=O)O1 98157,N(C1CC(C)n2ncnc21)C(C1CCCN(CCCOC(C)C)C1)=O 98158,C1(NC(Cc2nc(C(C)C)on2)=O)CC(F)CN(Cc2ncccc2C(F)F)C1 98159,c1(-c2ccc(C(C)O)cc2)cnc2ccc(C(=O)Nc3ncccc3Br)cn12 98160,N1(C(C(C(C)C)OCC(C)C)=O)CC(NC(=O)C=CS(C)(=O)=O)CCC1C 98161,CC(CN(C)C)CC(=O)NC1(CNC(c2cnc(C3CCC3)s2)=O)CCC1 98162,N1(C(CCC#CC)=O)CCC(NC(=O)C(C)NS(=O)(=O)CCCC)C(F)(F)CC1 98163,N1(C(c2cnc(CC)s2)=O)C2CCC1CC(CC(C)NC(C1CC13CC3)=O)C2 98164,C(C(C)(C(=O)N(CC(C)CNC(c1cn(-c2cccnc2)nn1)=O)C)OC)OC 98165,c1(CC)ncncc1C(N1CCN(C(CNC(C2CC(O)C2)=O)C(F)F)CC1)=O 98166,c1(CN(C(=O)CCCNC(c2cncn2CC2CC2)=O)C)ccc(Cl)cc1 98167,C(CCCC(=O)N(C(C)CNC(c1cccc(OC)c1)=O)C)OC 98168,C(C(=O)Nn1cnn(C)c1=S)C1(C)N(C(CCCC#CC)=O)CC1 98169,N1(C(c2c(C)c(O)ccc2)=O)Cc2ccccc2C1C(=O)NC1CNC(=O)C1 98170,CC1CN(C(C2(O)CC3CCC2C3)=O)CCC1CNC(=O)CC1CCCCC1O 98171,C1(C(=O)NCCCN(C(C2N(CCC)C(=O)CC2)=O)C)CC2(CCCCC2)CO1 98172,C1(C(=O)Nc2nocc2C(=O)NCC(CC)OCC)NC(=O)NC1=O 98173,c1(CC)nnc(N2CCC(OCCNC(=O)Cn3cnnn3)C2)o1 98174,N1(C(C(CCC2CCC2)NC(C(C(CC)C)N(C)C)=O)=O)CCOC(C)(C)CC1 98175,C(C)(CO)(C(=O)NC1CCN(CCNC(=O)CC2CCCCC2C)CC1)OC 98176,C1(O)(C(N2CC(NC(c3cnc(SC)s3)=O)C2)=O)CCCCCC1 98177,CC1(C#N)CC2(CC(c3nnnn3C3CCC3)(NCCC3C=CCC3)C2)C1 98178,C1(CC(=O)NC(CN(C(=O)CCc2cnn(C)c2)CC)C)CCNC1=O 98179,CCOC(C)(C(=O)Oc1ccc(C(=O)OCC)c(C(=O)O)n1)c1ccccc1 98180,N1(C(C(C)Cn2cccn2)=O)CCOC2(CCN(C(=O)C(=O)NC3CC3)C2)C1 98181,C=CCCC(C)(C)C(=O)NC1CCCC1NC(=O)C(CC)NC(N)=O 98182,c1(C(=O)NCCNC(CCc2ccn(C)n2)=O)cc(N2CCCCC2)ncn1 98183,N1(C(C(CNC(C2C(OCC)CC2)=O)CC2CC2)=O)CCC12CCC(O)CC2 98184,C1(N(C(=O)CCC2CCC2)C)CCCN(C(C2(CSC3CC3)CCC2)=O)CC1 98185,C(=O)(CCC(C)(C)NC(=O)C1CC1)N1CC(c2nc(C)[nH]n2)C1 98186,C(=O)(C1CCc2c[nH]nc21)N1CC(OCC)(CNC(c2cnn[nH]2)=O)C1 98187,CC(c1ccccc1F)=CC(=O)OC.C1(=O)CCC(C)SCC(=O)CCN1CC(C)O 98188,N1(C(c2cccc(CC=C)c2)=O)CC2(C(=O)N(CC(C)C(F)(F)F)C)CC1CO2 98189,Cc1cc(CN2CCCC(C)(C(=O)NCCc3nn[nH]n3)C2)cc(Br)c1 98190,CC1=C(C(=O)NC2CCC2NC(c2cnoc2C)=O)CCCC1 98191,c1(N(CC(CNC(CN(C)CC)=O)C)C)c(C#N)cnc2c(C)cc(F)cc12 98192,C1(C(C)NC(C2(NC(C)=O)CCC2)=O)CCCN(C(c2nocc2C(C)C)=O)C1 98193,C1(C(=O)NCC2C(NC(C(C#C)(C)C)=O)CCC2)CCc2nncn2C1 98194,Cc1csc2cc(C(=O)NC3CC3NC(c3cc(F)cc(F)c3)=O)[nH]c12 98195,Cc1cc(Cl)c(C(=O)NC2CCN(c3ccc(Cl)cc3)C2=O)cc1C 98196,c1(C(=O)NCC(=O)NC(C)CN(C)C(c2csnc2C2CC2)=O)ccc(N)cc1 98197,N(C1CCCc2n[nH]cc21)C(C(c1ccoc1)NC(CC(C(CC)C)O)=O)=O 98198,c1(C(=O)NC2CCC(NC(c3n(CC)nnc3)=O)CC2)ccc(SC)cc1Cl 98199,N1(C(C(C)=C(C)C)=O)CCN(C)CC1CNC(=O)C(O)C(F)(F)F 98200,c1(C2(C(=O)OCC3CCN(S(C)(=O)=O)C3)CCCC2)cc(F)ccc1F 98201,C12(C(N3CC(C(=O)N(C)Cc4cc[nH]n4)(CC)C3)=O)CCCC1C2(F)F 98202,c1(C(=O)NC2CCCN(C(c3n(CC)c(O)nc3)=O)C2)cc(F)cc(F)c1 98203,N1(C(CCCC#N)=O)CCCCCC1CNC(=O)CCCn1ccnn1 98204,C(c1ccc(Cl)cc1)(C(F)(F)F)=CC(N1CCN(C(C(C)O)=O)C2(C1)CCC2)=O 98205,C1(=CC(=O)N(CCOCCN(C(Cc2ncc(C)s2)=O)C)C)CCC(C)(C)CC1 98206,CCC(CNC(c1cccnc1CNC(C1(C)CCCN(C)C1)=O)=O)(CC)CO 98207,N1(C(C2OCCN(CC)C2)=O)CC2CN(C(c3cncc(C)n3)=O)CC2(C)C1 98208,C1(C(=O)N(C2CCCCC2O)C)(CNC(c2n(CC)nnc2)=O)CC(C)(C)C1 98209,c1(C(=O)NCCC(C)NC(=O)CC2COC(=O)C2)cncc(C(F)F)c1 98210,C1(C(N2CCC(CNC(C34OCC(C)(C3)C4)=O)C2(C)C)=O)Cc2cccnc2C1 98211,c1(NC2(CNC(C(CC)CC(F)F)=O)CCCCC2)nc(O)c2c(ncn2C)n1 98212,Cc1csc2c(C(=O)NC3CCC(CCNC(c4cnc(O)o4)=O)C3)ncnc12 98213,CC1CN(C(=O)CC2COC(=O)C2)CC(C)CN1C(=O)CCNc1cncnc1 98214,c1(C(N(CCC(C)NC(Cn2c(C)ncc2)=O)C)=O)cc(F)cc([N+](=O)[O-])c1 98215,Cc1ccc(N)c(C(=O)NCC(C)(C)CN(C(=O)Cc2c(F)cncc2Cl)C)c1 98216,Cc1ccc(C(=O)NC2CCC(C(=O)Nc3nccs3)OC2)cc1F 98217,C1(NC(C(=Cc2cccs2)C)=O)CCCN(C(=O)C(n2ccc(C)n2)C)C1C 98218,Cc1nccnc1CNC(=O)CCCN(C(=O)C(C)CC#N)C 98219,c1(C(=O)NCC2(CN(C(C3CC(C)OC3)=O)C)CC2)cccc2[nH]c(=N)oc12 98220,C(CCC(C)CC(C(=O)NC1CC1)N(CC(C)C(F)(F)F)C)=C(C)C 98221,CC(CN(C)C)CC(=O)NC1(C(N2C3CCC2CC3)=O)CCOCC1 98222,CCC(C(=O)NCC(C1CCC1)NC(=O)CCCNC(N)=O)N(C)C 98223,C1(C(=O)NC2C(CC)N(C(=O)CN3CCC(F)CC3)CC2)CC2CC(=O)C1C2 98224,CCC(CO)(C(=O)N1CC(C)C(C)(COC)C1)OC.C1(C=O)C2CC3C(C2)C13 98225,C1(NC(C2C3CCC(C3)N2C(c2ccccc2)=O)=O)CCCC1C1CCCC1 98226,C(C(=O)N1CCCC(CNC(C2(C(F)(F)F)CC2)=O)C1)(C(C)O)NC(C)=O 98227,C1(CC(=O)NCC2C(NC(CC(=O)NCC)=O)CCC2)CC2(CCC2)CCO1 98228,C1(NC(c2c(C)ncnc2)=O)C2CCCN(C(c3ncc[nH]c3=O)=O)C2C1(C)C 98229,Cc1cc(NC(C2CN(C(=O)CCc3cc(F)cc(F)c3)CCN2)=O)cc(F)n1 98230,c1(CC)ccnc(C(N2CC(N(C)C(c3cc(Cl)c(Cl)s3)=O)C2)=O)c1 98231,C12(NC(c3c(C)ccs3)=O)CCN(C(c3cccc(C(F)F)n3)=O)CC1C2 98232,C1(NC(C(c2ccccc2Cl)C)=O)CC(F)(F)CC1NC(c1cc(C#N)c[nH]1)=O 98233,N1(C(CCC2CCN(C(C3(C)CC(F)(F)C3)=O)C2)=O)Cc2n[nH]cc2C1CO 98234,C=CCC(C(=O)NC1CC2(CCN(C(=O)CN3CCSCC3)C2)C1)C(C)(C)C 98235,N1(C(c2c(Cl)cc(C)s2)=O)CCC(NC(C2SC3C=CC2CC3)=O)C(CO)CC1 98236,C1(C(=O)O)(OC)CC(OC(=O)CC2CN(C(=O)NC(C)(C)C)C2)C1 98237,c1(C(=O)NC2(C)CN(C(C3CCCCC3C3CC3)=O)C2)cccc2[nH]ccc12 98238,N1(C(C(=O)NCCCC)C(C)C2CCCCC2)CC(C)NC(=O)C12CC2 98239,N1(C(c2ccc(C(C)C)cc2)=O)CC=C(C(=O)N2CC(N(C)C)C(C)C2)C1 98240,c1(CCC(=O)NCC(C)(C)OCC(=O)N(CCCC)C)cccn1C 98241,C1(C(F)(F)F)CCCC(Cc2nc(C3CCCNCC3)no2)C1 98242,N1(C(c2c(CC)ccc(F)c2)=O)CC2CCC(C1)N2C(c1cc(Cl)c(Cl)s1)=O 98243,Cc1nn(CC(C)C)c(Cl)c1C(=O)NCC(C1CC1)NC(C1CCC(O)CC1)=O 98244,c1(C(N2CCC(CC(=O)OCC)CC2)=O)nc(C2=CCCCC2)cs1 98245,C1(NC(CCCSC)=O)CC(C)CN(C(c2cccc(Br)c2F)=O)C1 98246,c1(NC(C2C(C)(C)C2CN=[N+]=[N-])=O)ccc(O)cc1.C12(F)CC(C1)NC(=O)NC2 98247,C(=O)(C(C)CS(C)(=O)=O)NCCCN(c1ccccc1)CCCC 98248,n1(C(C)C)cnc2cc(NCC3CCC4(CCOCC4)O3)ccc12 98249,N1(C(c2cc(C)c(O)cc2)=O)CCC2(CCCCC2NC(=O)C2=CCCSC2)C1 98250,c1(C(=O)NC2CCC(CNC(C3(C=C)CCC3)=O)CC2)c(C)ccc(Br)c1F 98251,c1(CC(=O)NC(CC=C)CNC(=O)C(c2cncn2C)O)ccc(Cl)c(C)c1 98252,Cc1cccc(CN(c2nnc(CNS(C)(=O)=O)n2CCCCl)C)c1 98253,c1(C(N2CCN(C(C#CC3(C)CC3)=O)C3C2C3)=O)cccc2c1OC(F)(F)O2 98254,C1(CC=C)(C(=O)NC2CCC(CNC(C3(O)COC3)=O)C2)CCOCC1 98255,C=CC1CCCN(N2CCC(c3ccc(OC)c(F)c3)C2)C1 98256,N1(C(C2CC(O)(CC#C)C2)=O)CCOCC1CNC(c1c[nH]nc1F)=O 98257,CN1CC=CCC1CC(=O)NC1CCCCC1NC(c1ccsc1C(F)(F)F)=O 98258,c1(C(N2CCC(C)CC2C(=O)NOCCC2CC2)=O)c[nH]c2ccccc12 98259,c1(C(=O)NC2CC(NCc3cc(C)[nH]c3C)C2)c(F)c(F)c(O)c(F)c1F 98260,c1(NC(c2ccc(CCC(=O)Nc3nn[nH]n3)[nH]2)=O)ncc(F)cc1O 98261,NC1COC2(C(=O)NCC3C4CCCC34)CC1C2 98262,C1(C(N2C(C)CN(C(c3cnc(O)s3)=O)CC2)=O)CCn2ncnc2C1 98263,C=C(C)C(CC(=O)N1CCCC1CN(C(=O)CC1(O)CCC1)C)OCC 98264,c1(CC)nc[nH]c1C(=O)NC(C)CCN(C(=O)CNS(N)(=O)=O)C 98265,C12(C(=O)NCC3OCCN(C(c4ncn(C(C)(C)C)n4)=O)C3)CC(C1)S(=O)(=O)C2 98266,C1(NC(=O)Cc2cccnc2)CCN(C(=O)CSC(F)F)CC1O 98267,C(=O)(CS(=O)(=O)CCC(F)(F)F)NCC(C)(C1CC1)NC(C1ON=C(CC)C1)=O 98268,N1(C(C(C=C)O)=O)CC2CCC(C1)N2C(C1CC1C(c1ccccc1)=O)=O 98269,C(=O)(CC(C)(C)CNC(=O)C=CC1CCCCC1)N(CC)Cc1ccn(C)n1 98270,CC(CN(C)C)C(=O)NC(C1CCCN1C(=O)C=CCO)C 98271,N1(C(c2cc(C)oc2)=O)CC2CCCC2(Nc2ncncc2I)C1 98272,c1(CC(=O)N(C(C(=O)NC2CC(SC)C2)C)C2CC2)c(C)n[nH]c1C 98273,CC1(C)C(NC(=O)CCCCCNC(=O)CCC(=O)NC2CC2)CC1(F)F 98274,C1(NC(c2cncc(C)n2)=O)CCSC12CN(C(c1cc(C(F)F)ccn1)=O)C2 98275,C12(C(=O)OC)CC(C(N3CCC(CNCC4(C)CCC(=O)N4)C3)=O)(CO1)C2 98276,C1(C(=O)NCCC(CCC)C2CC2)CN(C(=O)C(C)(C)C(C)O)CC1(F)F 98277,C(C(C)(C)CN=c1cccc(S(=O)(=O)NC2CCCN(CC(F)(F)F)C2)[nH]1)OC 98278,N1(C(C2(c3cnccn3)CC2)=O)CCCC2(CCN2C(c2cc(I)ccc2Cl)=O)C1 98279,C(=O)(C(C)(C)C)NCCC(=O)NCCN(C(CSCC=C)=O)C1CC1C 98280,c1(C(=O)NCCCNC(c2nc(CCC)oc2)=O)cncc(C(C)=O)c1 98281,c1(C(N2C(CN(C)C(c3cc(Cl)no3)=O)CCC2)=O)cnc(Cl)cc1N 98282,c1(C(=O)NC(CSCC)C(N2CCC(NC(N)=O)CC2)=O)cnc(F)cc1C 98283,C(C(C)CN=c1[nH]c(=NCCS(=O)(=O)CCO)[nH]c2cccnc12)OCC 98284,Cc1ccc(CNC(=O)N(CC(C)O)CC2CCCO2)nc1 98285,S(=O)(=O)(c1ccc(N2CCCC(CC3CC3)C2)c(Cl)c1)NC1(CCCC)CC1 98286,CN1CCN(C(=O)CC2CCCN2C(=O)CCc2csnn2)CC1C1CC1 98287,c1(N(C(CCNC(c2ccc(C(C)C)cc2)=O)C)C)ccnc(C#N)n1 98288,C1(O)(C(N2CCC(N(C(=O)C(C)O)CCOC)CC2)=O)CCC(C)CC1 98289,N1(C(CC2(OC)CCC2)=O)CCOC2CCN(C(C3CC3(Cl)Cl)=O)CC12 98290,Cc1ccc(C(N2CC(CNC(=O)C(C)NC(C)(C)C)C2)=O)c2cccnc12 98291,c1(C(N2CCN(C(C3C(C)(C)C(=O)C3)=O)CC2CCO)=O)cnn2cccnc12 98292,N1(C(C=C(C)C)=O)CC2(C=C(C(=O)N3CC(C(F)(F)F)C3)CO2)C1 98293,C1(CNC(c2ccnc(S)c2)=O)CC12CCN(C(=O)CS(=O)(=O)C1CC1)CC2 98294,C(=O)(CC(C)C(C)(C)NC(=O)Cc1cc(C)[nH]n1)N(CCCN(CC)CC)C 98295,Cc1cc(NC(C2CC(C)CN2Cc2ccc(I)c(F)c2)=O)ccc1O 98296,C1(CCNC(CC=C=C)=O)CCCN(C(=O)CC2(C#N)CCOCC2)CC1 98297,C(=O)(CC(C)(C)C(C)(F)F)N1CCC(N(C(CCC(C)C#N)=O)C)CC1 98298,C1(CNC(C2(C3CC3)CC2)=O)CCCC1(C)C.C12(CCC1)CC(=O)N2C 98299,C1(NC(c2c(OCC)ccc(Br)c2)=O)CN(C(C2CCCCO2)=O)CC(F)(F)C1 98300,C1(CC(=O)NCCN(C(C(C2CCCCC2)OC)=O)C(C)C)COCCN1C 98301,C#Cc1ccc(OCC(=O)NCC2(CNC(=O)C(C)CC)CCC2)cc1 98302,C1(C(N(CCNC(COCC)=O)C)=O)(NC(=O)OC(C)(C)C)CCN(C)CC1 98303,C(C1CCCCC1)=CC(=O)NCc1cc(C(=O)NCc2c[nH]nc2C2CC2)no1 98304,CCCCC(F)(F)C(=O)N1CCC(C(F)C(=O)N(CC(C)(C)O)C)C1 98305,CC(CN=c1[nH]c(=NCC2CC(F)C2)c2[nH]ccc2[nH]1)S(N)(=O)=O 98306,c1(C(=O)NC(CCCNC(C=CCCC(C)C)=O)C)cc2scnc2[nH]1 98307,C1(C(N(CCC)CCNC(C2(c3cc(C)no3)CC2)=O)=O)CC2CC1CC2O 98308,c1(C(C(=O)NCC)N(C(C#N)C2(SC)CC2)C)ccc2nc(C)oc2c1 98309,c1(C(=O)NCCN(C(C(C=C)(C)C)=O)CC)cc(=O)n2nccc2[nH]1 98310,C1(C(N(C)CCOCCNC(c2cc(C(F)(F)F)n(C)n2)=O)=O)CCC12CCCO2 98311,CCCC(C(=O)NCCCCCN(C(=O)C(C)OC(C)(C)C)C)OC 98312,C1(N(C(c2cc(CC(C)C)[nH]n2)=O)C)CCCC(N(C(=O)CC2(O)CC2)C)C1 98313,C(C(CCO)N=c1[nH]c2c(c(=NCCCn3ccnc3)[nH]1)CCCCC2)N(C)C 98314,c1(C(N(CC(N2CCC(N(CC)CC)C2)=O)C)=O)ccc(Cl)nc1OC 98315,C=Cc1cnn(C)c1C(N1CC(N(C(=O)CC2CC(=O)NC2=O)C)C2(CC2)C1)=O 98316,C1(CNC(C2(C#C)CC2)=O)CN(C(c2cc[nH]c2CC)=O)CC12CCC2 98317,c1(CC(=O)NCCC(C)NC(=O)C(c2ccccc2)O)cccc2c1OCO2 98318,Cn1cc(Br)cc1C(=O)NCC1(CNC(=O)CSCC(N)=O)CC12CCC2 98319,c1(C(N2C(CNC(c3n(C)ccn3)=O)COCC2)=O)cc2c(Cl)c(F)ccc2[nH]1 98320,c1(C(=O)NCC(C)N(C)C(C2CCS(=O)(=O)N2)=O)ccc(F)c2c1OCC2 98321,C1(C(N(C2CCN(C(=O)C(C)(O)C3CCOCC3)CC2)CC)=O)CCC12CCC2 98322,C(=O)(CS(=O)(=O)C1CCCC1)NC1C(NC(C(C(CC)CC)OC)=O)C1 98323,C1(NC(CC(C)(C)SC)=O)CC(O)CN(C(c2cccc(O)c2Cl)=O)C1 98324,C1(NC(c2c(C)cccc2O)=O)CC2CCC1N(C(C1CSC1)=O)C2 98325,c1(C(=O)NC2CCOC2C(N2CC(CO)C2)=O)cncc(O)c1 98326,Cc1nc2cc(C(=O)NC3CN(C(=O)CC4CC5CC5C4)CCC3O)cnc2[nH]1 98327,c1(C(=O)NCCN(C(=O)C(F)(F)C2CC2)CCOC)c[nH]cc(C)c1=O 98328,C=C=CC(C)C(=O)NC1(C(N2CC(N3CCCCC3)C2)=O)CC1(C)C 98329,c1(C(N2C(CNC(Cc3c(C)n(C)cn3)=O)C(C)CC2)=O)cnc(Cl)cc1N 98330,c1(C(=O)NCCC2(CNC(CC(C)c3ccco3)=O)CC2)nccc2ccsc12 98331,Cc1cc(=O)c(NC(=O)C(C(C)NC(c2csc(Cl)c2)=O)C(C)C)c(C)[nH]1 98332,C1(CC=C)(C(=O)NCc2nc(C(N3CCCC3C(=O)NCC)=O)co2)CCOC1 98333,c1(CC)noc2ncc(C(=O)NCC(F)CNC(C3CC3CC)=O)cc12 98334,c1(N(C2CC23CCNCC3)C(COC(C)C)=O)ccc(O)cc1O 98335,c1(NC(C(Cc2cc[nH]n2)NC(C(C)=C2CC2)=O)=O)ccc2c[nH]nc2c1 98336,N1(C(C(C2CN(C(CCc3cc(C)[nH]n3)=O)C2)O)=O)CC2C(C1)C2(F)F 98337,c1(C(=O)NC2CC(NC(=O)CC3CCOC3)CC2O)cc2sc(Cl)cc2[nH]1 98338,Cc1cc(O)ccc1C(N1CCC(NC(=O)C(=O)Nc2c(F)cccc2F)C1)=O 98339,C(=O)(CCCCCCNC(=O)Cn1ccccc1=O)NC(C)C(C)(C)O 98340,N1(C(C=CC)=O)CC(NC(c2ncsc2CC)=O)C(CC2CCCCC2)C1 98341,N1(C(CCN(C(C(C)OCC=C)=O)CC2CC2)=O)CCC(O)(CN(C)C)C1 98342,C1(OC)CC(C(N2CCCCC2CNC(=O)CC2CCCSC2)=O)CC1OC 98343,c1(CN(c2ccccc2)CC(N2CCC(N(C)CCO)C2)=O)ccccc1 98344,c1(NC(C(C)NC(c2c(C(N(C(C)(C)C)CC)=O)occ2)C)=O)ccc(Cl)cc1 98345,C1(C(N2CCCC(NC(C3CC3(F)F)=O)CC2)=O)CCC2(CCOCC2)O1 98346,C(=O)(C1=NOC(CNC(=O)C(O)CN(C)C)C1)NCC1ON=C(C)C1 98347,N1(C(C2N(C=O)CCC2)=O)CCN(C(=O)Cc2c[nH]nc2O)CC(O)C1 98348,C1(C(=O)NCC(c2ccccc2)CNC(CCSC)=O)CC(=O)C12CCCC2 98349,c1(N(C(c2scc(C)c2)C(=O)NC2CCOCC2)C)cccc(F)c1 98350,O(NC(=O)CC(CNC(=O)CC1CC1)OC)CC#C 98351,c1(CC(=O)N(CCN(C(C)C)C(c2ncccn2)=O)C)cn(C)nc1Cl 98352,O=C(CS(=O)(=O)N1CCOCC1)NCC1CC(O)CN1C(=O)C=CC1CCCO1 98353,C(=O)(CCC(C)(C)F)N1CC(C2N(C(c3cc(C)n(C)c3)=O)CCC2)(O)C1 98354,N1(C(c2n(CC)ncn2)=O)CC(NC(c2ccccn2)=O)C(C(F)(F)F)C1 98355,Cc1cc(=NCC2CC=CCC2)[nH]cc1S(=O)(=O)N(CCCN(C)C)C 98356,C=CCC(CNC(=O)CNC(N)=O)NC(C1CCN1C)=O 98357,N1(CCOC)CC(C(=O)NCC2CCC2NC(c2cc(C)ns2)=O)CC1=O 98358,c1(C(N(CCN(C(Cc2cc(C)[nH]n2)=O)C(C)C)C)=O)cc(C)c(N)cc1F 98359,N1(C(C=CC(C)C)=O)CCC2(CCC2)C(CNC(C2(C)COC(C)(C)CO2)=O)C1 98360,CC1(C)CC(CNC(C2CCCCC2)=O)CN(C(=O)CC2NC(=O)NC2=O)C1 98361,n1(CC(=O)NC23C(C)OC(CNC(=O)CC#N)(C2)C3)nc2ccccn2c1=O 98362,C(=O)(C(C(C)CC)N(C)C(c1ccccc1Br)C)NCC(=C)C 98363,N1(C(C2CC3OC2C2CC32)=O)CCC2CN(C(c3ccnc(C(F)F)c3)=O)C2C1 98364,C(CC(C)(C)C(=O)NC1CCC1NC(=O)Cc1ccc(C)cc1)OC 98365,C1(C#N)(C(=O)NC2CCN(C(c3c(Cl)nc(OC)s3)=O)C2)CC12CCC2 98366,N1(C(c2c(OC)nccc2)=O)CCN(C(=O)CN(C2CCSC2)C)CC2(CC2)C1 98367,C1(NC(C2N(CCCC)CCOC2)=O)CCN(C(C2(COC)CC2)=O)C(C)C1 98368,C1(C(C)C)C2CCN(C(=O)C(C3CCN(C(c4nc(=N)cc[nH]4)=O)CC3)C)CC12 98369,c1(C(=O)NCC2(CN(C(=O)C3=CC(C)(C)C3)C)CC2)ccc2[nH]c(=N)[nH]c2c1 98370,c1(C(=O)NC2CCC3(CN(C(C=C(C)C(=O)O)=O)C3)C2)c(O)cccc1[N+](=O)[O-] 98371,c1(C(C)NC(C(CC)O)=O)ccc(CNC(=O)Cc2csc(S)n2)cc1 98372,C1(CNC(c2c(C(C)C)nns2)=O)C2CN(C(C3CCCN3S(C)(=O)=O)=O)CC12 98373,C(=O)(C(CC)C(C)O)NC1(CC=C)CCN(C(=O)CCc2ccc(O)nn2)C1 98374,CCCC(C(=O)N1CC(C)(CCC(=O)NC(c2nccnc2C)C)C1)NC(C)=O 98375,C1(NC(C(CC)C)=O)CCCCCC1C(=O)NCc1ccc(Cl)cc1 98376,N1(C(=O)CCF)CCC2CN(C(=O)CCCOc3ccccc3Cl)CC2C1 98377,C1(C(N2CC3CC3(C(=O)NC3CCC3)C2)=O)CCC(C(F)(F)F)CC1 98378,C(=O)(C1CCCc2nc[nH]c21)N1CCC(C)(NC(c2cccc(N)c2N)=O)C1 98379,C1(C)(C(=O)NCCC2(O)CN(C(C3CCCC(C)(C)C3)=O)C2)CCCCNC1=O 98380,N1(C(Cc2c(C)ocn2)=O)CC(NC(C2CC3CC3C2)=O)CC(C)C1 98381,C(=O)(C#CC(C)(C)CNC(C1COCCN1C)=O)NCC1(C)ON=C(C)C1 98382,c1(-n2c(-c3ccc(-c4[nH]cc(C#N)c4)cc3)ncc2)ccc(F)cc1F 98383,C1(CNC(C=CC=CC)=O)CCN(C(c2ncc(C)cc2F)=O)C1(C)C 98384,N1(C(COCCCC)=O)CCN(C(=O)CC2COC(C)(C)CO2)C(C2CCC2)C1 98385,C1(C2CCC2)(C(N(CCCNC(C(C(C)C)CO)=O)C)=O)CC1(F)F 98386,c1(C(N2C(C(N3CC(C)OCC3C)=O)C3CCC2C3)=O)cc2cc(Cl)ccc2[nH]1 98387,c1(NCC2(C)CN(C(=O)CCNC3COC3)C2)ncc(C(F)(F)F)cc1Cl 98388,c1(C(=O)NCC(CC)NC(C2C(C#C)C2)=O)ocnc1C1CC1 98389,c1(CN2CCC(N(C(=O)COCC3CCOC3)C)C2)c(F)cccc1F 98390,C1(C(=O)Nc2c(CC)n(CC(C)C)nc2)CCC2(CC1)CCC2N 98391,c1(C(N2C(CNC(c3cncc(C)c3)=O)CC(C)(C)C2)=O)cncc2nc[nH]c12 98392,CCC1=C(C(=O)NC2C=CC(CC(=O)NCCC(C)(O)C3CC3)C2)CCCO1 98393,c1(C(=O)NC(CC)CNC(=O)CCCc2n[nH]c(=N)s2)ccc2oc(O)nc2n1 98394,N1(C(c2ccc(CC)o2)=O)CCCN(C(c2cscc2CC)=O)CC1CO 98395,C1(CCC2CC2)CN(C(c2cn(CCC(C)C)nn2)=O)CCN1C(=O)C(=O)OC 98396,c1(N(CCN(C2CCN(C)CC2)C)C)c(C#N)ccc2ccccc12 98397,Cc1nc(C(=O)NCc2csc(C(=O)NC3CCC(N(C)C)C3)c2)cn1C 98398,CC1(NC(c2cn(Cc3ccccc3)nn2)=O)CN(C(C2(C)CCCC2)=O)C1 98399,C(=O)(C1CCCc2c[nH]nc21)N1CC(CCNC(C2CCCC(C)(C)CC2)=O)C1 98400,C1(CNC(COC2(C)CN(C(c3c[nH]c(C#N)c3)=O)C2)=O)CCCC(F)C1 98401,CCCN=C(NCCN(C1CCCCC1)CC)NCC.C12CCN1C2 98402,c1(OC)cc(CCC(=O)NC2CCCN(C(C3CCOC3C)=O)C2)ccc1Cl 98403,Cc1cc(C(c2nnnn2C2COC2)NCCc2c[nH]nc2C2CCC2)sc1Cl 98404,c1(C(N(C2CN(C(CC(=C)C)=O)CC2F)C)=O)cnc(O)c(Cl)c1 98405,c1(C(=O)NCC(C(C)C)NC(C(CC)N(C)C)=O)cc2ccccc2n1C 98406,CCC(CC)C(=O)NCC1CN(C(=O)C(n2ccc(C)n2)C)CC1O 98407,C=CC(C)CC(=O)NCC(CC1CCCC1)C(=O)NCCOCC(=O)OC 98408,c1(C(N(C2(C(=O)Nc3ccc(CC)cc3)CCC2)CC)=O)cccc(C)c1C#N 98409,C1(NC(CC2(C#N)CCC2)=O)CCN(C(c2ccns2)=O)CC1CO 98410,c1(N2CCC(C)C2CNC(c2cccc(F)c2F)=O)nc(Cl)nc2nc(Cl)n(C)c12 98411,N1(Cc2c(Br)ccc(C)c2)CC2CC(NC(=O)Cc3c(C)noc3C)CC2C1 98412,C1(CNC(CC2CC(SC)C2)=O)C(C2CC2)CCN1C(=O)Cc1cscn1 98413,C1(C(=O)NCC(CC)N(C(=O)CCC2CCC(C)O2)C)CC(F)(CF)C1 98414,C1(NC(c2c(C(C)(C)OC)cccc2)=O)CC(O)CN(C(=O)C(C)=C2CCC2)C1 98415,Cc1c(Br)ccc(F)c1C(=O)NCCN(C(=O)CC1CNC(=O)C1)C 98416,Cc1[nH]c(C#N)cc1C(=O)NCc1cccc(C(N2CC(C)(C)C2)=O)n1 98417,CCC(CC)CC(=O)N1CC(NC(c2nnsc2SC)=O)C(C(F)F)C1 98418,C1(CNC(C(N2CC3(CN(C(C)=O)C3)C2)=O)=O)CC2CC1CC21CC1 98419,C12(NC(=O)COC3CCC3)CCCN(C(=O)CCCC(F)(F)F)CC1C2 98420,Cc1cc(=NC2CC3CN(C(=O)CC4(C)CCCC4)CC23)[nH]c(Cl)n1 98421,C(c1cnc(O)nc1O)=CC(=O)NC(C)(CNC(c1ccccc1Cl)=O)C1CC1 98422,c1(N(CCn2c(C)ncc2)C)nc(=NCC(C)CCO)[nH]c2ccccc12 98423,C1(C(N(CCOC)CC)=O)(CNC(=O)C(C)n2cccc2)CCCC1 98424,c1(CCCC(=O)NCC(CNC(CNC(CNC(C)=O)=O)=O)O)ccc(O)cc1 98425,C1(CCOCC)(C(=O)NCC2CCC2NC(c2cc(Br)c[nH]2)=O)CCCC1 98426,C(=O)(C(C)(C)CS(N)(=O)=O)N(CCN(C)C(c1ccc(F)cc1C(F)(F)F)=O)C 98427,Cc1cc(C)c(C(=O)NCCCCC(C)NC(=O)C(C)(C)C2CCCCO2)cn1 98428,N1(C(C(CC=C)CN)=O)CCc2sccc2C1CC 98429,c1(C(=O)NC(C2CCCCC2)CNC(C(C)CF)=O)cncc(F)c1 98430,C1(C(=O)NCCC)CCN1C(=O)CSc1nc[nH]n1 98431,C1(C)(NC(C2N(C(CS(CC)(=O)=O)=O)CCOCC2)=O)CCCCC1(C)C 98432,c1(OC)cc(C(N2CCCCC2CNC(C2CCS(=O)(=O)N2C)=O)=O)cc(C)n1 98433,n1(CC)cc(Cl)c(C(N2CCC(N(C(=O)CC3CCS(=O)(=O)C3)CCO)C2)=O)n1 98434,C1(C)(CC(=O)NCCOC2CCN(C(C3(C(C)C)CC3)=O)C2)CCS(=O)(=O)N1 98435,N=c1[nH]c2c(s1)CN(CC1CCN1C(=O)C1=NOC(c3ccccc3)C1)CC2 98436,CCCC(C(=O)N1CC2CC1C2NC(C1CCC1c1nc(S)n[nH]1)=O)S(N)(=O)=O 98437,C1(CNC(C(C)NC(=O)Cn2cnnn2)=O)CCCCN1C(C1CCCC1)=O 98438,C(C(C)CN=c1nc(N2CCCC3(CCSCC3)C2)c2sccc2[nH]1)OC 98439,CCCCC(C(=O)NCC(C)(C)NC(c1cnnc(O)c1)=O)C(C)C 98440,C(=O)(C1=NOC(C)(C)C1)NC(C(C)C)CC(=O)NC(c1nccc(O)n1)C 98441,c1(SC)cc(C(=O)NCC2CC(NC(C3CC=CCO3)=O)C2)nn1C 98442,c1(C(=O)NCC2CC(NC(c3cc[nH]n3)=O)C23CCC3)c[nH]c2cnccc12 98443,N1(C(C(C(=O)OCC)F)=O)CC2CCC1C1CN(C(=O)C(C)(F)C(C)(C)F)CC21 98444,C(C(C(C)C(C)C)NC(=O)CSC)NC(CCc1cncc(OC)c1)=O 98445,C1(c2n(CCOC)nnn2)(NCC2COC2)CC2CC1CC21CC1 98446,n1(CC(=O)NCC2(F)CC(NC(C(C(C)C)SC)=O)C2)cnc2ccccc12 98447,c1(N2CC(C)(CCO)OCC2)ccncc1S(=O)(=O)NCC(C)(C)c1cccs1 98448,c1(C(NOCC(=O)NC(CC#C)C)=O)ccc(O)nn1 98449,N1(C(c2cc(OC)cc(=O)o2)C(=O)NCC(=C)C)CC2COCC(CO)(C1)C2O 98450,CC(O)(Cn1ccccc1=O)C(=O)NC1CC(F)(CNC(=O)Cn2cncn2)C1 98451,Cc1ccc2c(=NCc3ncc(F)cc3F)[nH]c(=NC3CCCC3C)[nH]c2c1 98452,c1(NCC(COC)(C)CO)[nH]c(=NCCc2ncccc2C)nc2scnc12 98453,N1(C(C2(C(C)NC(=O)CC3C=CCCC3)CC2)=O)CCC(C)(CCO)CC1 98454,O=C1CNc2cc(C(N3CC4CC3CN(C(=O)C3=CCOCC3)C4)=O)cnc2N1 98455,N1(C(C(COC)NC(C)=O)=O)CCN(C(=O)C(O)CC(N)=O)C(C)C1 98456,N1(C(C(CC)OC)=O)CC2(C1)CN(C(=O)C(CC(C)C)OC(C)C)CC2CO 98457,N1(C(N(C)C)=O)CCC2C1CCN2C(C1C2C=CSC12)=O 98458,C12(CCCCC1)C(=O)N2.C1(CNC(N)=O)CCCC(NC(=O)CN(C)C2CC2)C1 98459,CC(C)C(C)C(=O)N(CCn1cc(-c2ccc(OC(F)(F)F)cc2)nn1)C1CC1 98460,C(C(=O)NCC(C)NC(=O)C(c1cscn1)N(C)C)(OCC)OCC 98461,c1(C(N2CC(NC(=O)CC3CCCCS3)C(O)C2)=O)ncc(Cl)cc1O 98462,N1(C(CCN(C(CCC)C)C)=O)CCN(C(C2CC3(C2)CC(O)C3)=O)C2(CC2)C1 98463,Cc1cc(C(F)(F)F)sc1CNC(=O)C(=O)NC(c1ccccc1)C 98464,C1(C(N(C2(CC(=O)NCCC3(C)CCOC3)CC2)C)=O)CCCC(=O)N1 98465,C1(CC)CCCN(CC(=O)NC2CN(C(=O)CC3(C#N)CC3)CC2O)C1 98466,n1(CC)ncc(C(=O)NC2CC(NC(=O)CCC3CCCCN3C)C(O)C2)c1C 98467,C1(NC(COCC(=O)NC)=O)CN(C(c2cc(OC)cnc2F)=O)CC12CCC2 98468,N1(C(c2cn(CCOC)nc2)=O)CCC(CCNC(=O)C(C)SC(C)C)CC1 98469,C(C(=O)NC1CC(CO)N(C(=O)C(C(C)C)n2cc(C)cn2)C1)(C(C)(C)C)SC 98470,C#Cc1ccc(F)c(C(=O)NC2CCN(C(=O)C(C)(CO)OC)CC2)c1 98471,c1(C(N2CC(CCCNC(C(CC)OC)=O)OCC2)=O)cc(F)ccc1C1CC1 98472,CCC(CNCC1CCN(C2CC2)C1)(CC)C(=O)Nc1ccc2cc[nH]c2n1 98473,CC1CN(C(=O)CC2COC(=O)N2)CCN1C(c1csnc1Br)=O 98474,C1(NC(c2c(OC)csc2)=O)CCN(Cc2c(C)noc2C)CC1(C)C 98475,CCC(CC(=O)N(CC(O)CNC(c1ccn(CC)c(=O)c1)=O)C)C(F)F 98476,c1(C(C(=O)NCC2N(C(C=CC=CC)=O)CC=C2)C)ccc(SCC)cc1 98477,c1(C(c2nnnn2CCOCC2CC2)NCCC=C=C)cc2nc(Cl)ccc2s1 98478,c1(C(N(C(C(N2CCC(n3cncn3)C2)=O)C2CC2)C)=O)nnn(C)c1N 98479,C1(C(N2CC(CCCCNC(C(C)=C(C)C)=O)C2)=O)C2Cc3cc(Cl)ccc3C12 98480,N1(C(C(C)SCC)=O)CCOC(CCNC(C2(c3cccnc3)CCCC2)=O)C1 98481,C1(C(=O)Nc2ccc(OCC(=O)NCC)cc2)CCCCC1(OC)OC 98482,N1(C(Cn2c(C)nc(C)n2)=O)CCC(C(=O)NCCc2nncn2C)CC1(C)C 98483,N1(C(C2OCCC(C)C2)=O)CC2CN(C(c3cc4cnccc4o3)=O)CC2(C)C1 98484,C1(NC(CC=C)=O)CCN(C(c2occc2C)=O)C1C(C)(C)C 98485,C1(C(=O)NC2C(CNC(c3nc(C)c(C)s3)=O)COC2)CCC(=O)N(C(C)C)C1 98486,c1(N(C(C)=O)C)cccc(C(=O)NC2CCC(NC(c3cncs3)=O)CC2)c1 98487,CC(CC(=O)N1OCC(F)(F)C(=O)NCC(C)C1)C(C)(C)C 98488,CC(CC(=O)N1CC(NC(c2cccc(Cl)c2)=O)C1)C(=O)c1ccccc1 98489,c1(NC(CC(CCC)NC(c2cn3ccccc3n2)=O)=O)cnc(C)c(C#N)c1 98490,CCCCCCCCCCCC(=O)NCC1CCCN(C(C2CCSC2)=O)C1 98491,c1(C(=O)NC2CC(CCC(=O)NCCC(C)(C)OC)C2)c(C)nsc1N 98492,c1(C(N(CCNC(C(CC)SC)=O)CCOC)=O)nc(C)ncc1Br 98493,C1(NC(c2n[nH]c(C)c2O)=O)CN(C(=O)C2=C(Cl)CCOC2)C2(CCOC2)C1 98494,C1(NC(C(C)SCC)=O)CCCC12CCN(C(c1cc(Cl)cc(F)c1F)=O)CC2 98495,c1(N2C(C)CC(Nc3ncnc(Cl)c3CO)C2)ccn2nccc2n1.C=O 98496,N1(C(C(C2(O)CCC2)NC(=O)CCN2CCOCC2)=O)CC(F)(C2CC2)C1 98497,N1(C(CCCNC(C)=O)=O)CCOCC1Cc1cn(CC)nn1.C(=O)CS(N)(=O)=O 98498,C1(C(=O)NCCN(C(c2ccc(C)c(C)n2)=O)CC)CC2(CCOC2)C1 98499,N1(C(C2(COC)CC2)=O)CCC2(CCC(NC(C3CC(C4CCCC4)C3)=O)C2)C1 98500,c1(C(=O)NCC(CC=C)NC(=O)C(F)n2ccnc2)cnc(C(F)(F)F)nc1 98501,C(=O)(N=c1ccn(C(F)F)[nH]1)C1(C)CCCN1C(c1csc(Cl)c1)=O 98502,Cc1cc(=NCc2n[nH]cc2C(C)C)[nH]c(N2CCCC(NS(C)(=O)=O)C2)n1 98503,c1(OC)c(NC(C2(C)CN(Cc3c(F)ccc(C)c3F)C2)=O)ccc(F)c1F 98504,N1(C(c2c(CC)n(CC)nc2)=O)CC2(C=C(C(=O)NCC(O)CC(C)C)CO2)C1 98505,N1C(C(=O)OC(CC2(N)CCC2)=O)CCOCC1=O.c1(CC(=O)NC(C)(C)C)nn[nH]n1 98506,C1(C)(NC(c2n(C)nnn2)c2ncoc2C(C)(C)C)CN2CCC1CC2 98507,c1(N(C2CNC2)C(c2n(C)nnc2)=O)ccn2ncc(Br)c2n1 98508,C1(CNC(c2ccc(OC)s2)=O)CC(C)(C)CCC1NC(=O)C(C)(C)CC(C)C 98509,C(=O)(C1=CCCCC1P(C)(C)=O)NC1(CNC(C(C)(C)c2ccccc2)=O)CC1 98510,c1(C(=O)NC2C(CNC(c3ccnc(C(F)F)c3)=O)C2)cncc2cnccc12 98511,N1(C(c2c(C)cco2)=O)CCC(C(=O)NOCCN(C)C)C12CC2 98512,C1(NC(=O)COCC2CCCO2)CCCC(NC(=O)Cc2nccc(O)n2)C1 98513,N12CCC3CCCC13C(=O)OCC(O)CC2=O.N1(C(=O)OC(C)(C)C)CCCC1 98514,N1(C(CCCCOC)=O)C2CCC1CC(NC(=O)C(C(C)(C)C)NC(C)=O)C2 98515,CCC(CC)CC(=O)N1CC=CC(C(=O)NCC=CC(=O)OC(C)C)C1 98516,N1(C(C=Cc2n(C)ncc2)=O)CCC(NC(=O)CC2CCC(=O)NC2)C12CCC2 98517,N1(C(CCCC(=C)C)=O)CCCC(C2CCN(C(C3CN4CCN3CC4)=O)C2)C1 98518,c1(C(N2CCN(Cc3nc(Cl)ccc3F)C3CC23)=O)cnn2cccc(F)c12 98519,c1(N(C(=O)OCC)C)ccc(NC(C2(c3ccccc3Cl)CCOCC2)=O)cc1 98520,c1(C(N2C(C(=O)OC)CC(n3cc(C(C)(C)CO)nn3)C2)=O)c(C)sc(C)c1Br 98521,CC1CCCN(C(c2cnc(C(N)=O)s2)=O)C1CNC(C1CC(O)C1)=O 98522,C(C(C)CC(F)(F)F)NC(C(c1ccnn1C)NC(C(C)SCCOC)=O)=O 98523,c1(CCC(=O)NC2(C)CC(NC(C(C)=CC)=O)C2)ccc(F)cc1Cl 98524,Cc1cc(Br)cc(C(N2CCC(O)(C(=O)N(C)C)CC2)C(=O)NC2CCCCC2)n1 98525,c1(C(=O)OC)ccc([N+](=O)[O-])c(N2CC3CC(NC(c4ccc(C)[nH]4)=O)C3C2)n1 98526,c1(NCC)cccnc1C(=O)NCC1CCC1NC(C1(n2cccn2)CC1)=O 98527,O(N1CCC(CC(=O)N(C(C)CN(C(=O)CC(C)COC)C)C)CC1)CC 98528,C1(NC(c2ncn(C(C)C)c2)=O)CCOCC1NC(=O)CC(=O)NC1CC1 98529,C1(C(C(=O)N(C(C)C2CC2)C)C)CCN(C(c2ccnnc2)=O)CC1 98530,c1(CC)ccc(F)cc1C(N1CCC(NC(=O)C(F)(F)c2cncs2)C(O)C1)=O 98531,C#Cc1cccc(CC(=O)NCC2(NC(c3ncccn3)=O)CCCCC2C)c1 98532,C1(C(=O)NCc2c(C3CN(C(C(CC)C)=O)C3)ocn2)CCn2c(cnc2C)C1 98533,O=C1c2ccccc2NC2=NC3CCC(CC3c3ccccc3)N12 98534,c1(OC)ccc2c(c1)OCC(C(=O)N1CCN(C)C3(CC3)C1)=C2 98535,N1(C(c2cnc(-c3sccc3C)s2)C(=O)NCCC)CCN(C(C)=O)CC1C 98536,c1(C(N(C2CCN(C(c3cc(C)on3)=O)C2)CCO)=O)cc(N)cnc1C 98537,O=C1NC(=O)C2(CCN(C(=O)C(=O)NC(c3ccc4ccccc4c3)CF)C2)N1 98538,O=C(C1=CCCC1)NC1CN(c2cc(-n3cncn3)ncn2)CC1F 98539,C(c1c(F)cccc1F)=CC(N1CC(OCCNC(C(C(C)OC)O)=O)C1)=O 98540,N1(C(c2ccn(CCCC)n2)=O)CC(NC(=O)CCn2cccn2)CC(O)C1 98541,Cc1cc(C(N2CCCC(C(C)NC(=O)CCF)C2)=O)cc(I)c1 98542,c1(N2C(C)CCC2)ncc(F)cc1[N+](=O)[O-].c1cncc(OC(F)F)c1 98543,N1(C(C(CC)Oc2ccccc2)=O)CCC2CN(C(c3ccn(C)c3)=O)C2C1 98544,C1(C(N(CCCCCNC(C(COC)N(C)C)=O)C)=O)OCCOC1(C)C 98545,c1(C(=O)NC2CCC(NC(c3c(N)cc(Cl)nc3)=O)CC2)n[nH]c2c1CCSC2 98546,C1(C(=O)NCc2cccc(CNC(CCCC#C)=O)c2)CCn2c(C)cnc2C1 98547,c1(C(=O)NCC(CC=C)NC(C2CCC(CO)CC2)=O)cc(C#N)ccc1F 98548,C(CCCCCC(=O)N1CCC(O)C(F)(F)C1)NC(C1CC2CCC1CC2)=O 98549,CCCCC(C)CCC(=O)NCC1(NC(c2ccc(O)cn2)=O)CCOCC1 98550,n12c(N(C)CC)nnc1N1CCOC(C1)C2.C(C(=O)NCC(=O)OCC)=CC 98551,C(N=C(NC1CC1)NC1CC(C)(C)Oc2cc(F)ccc21)c1c(C)ncs1 98552,C1(CNC(COCC(C)(C)C)=O)CC(CNC(c2cc(C3CC3)cs2)=O)CO1 98553,n1(CC(N2CCC(CN(C(c3c(OC)scc3)=O)C)C2)=O)nc(C)c(Cl)c1C 98554,C(=O)(CCC(C)(C)[N+](=O)[O-])NCC1C(C(=O)NC(CC=C)C2CC2)CCO1 98555,CC1(C)CN(C(=O)COc2ccccc2F)CC1NC(=O)CCCCO 98556,CC(C)(C)CC(C)(C)C(=O)NCCN(C1CCCCCC1)C(=O)Cn1[nH]cnc1=N 98557,Cc1ccc(NC(C)CNC(c2sccc2C(F)F)=O)c([N+](=O)[O-])c1 98558,Cc1cccc(COC(C)C(=O)NC2COCC2NC(=O)C#CC2CC2)c1 98559,CCC(C)CCC(=O)NC1CCCCC1NC(=O)Cn1ccc(C(=O)OC)n1 98560,C1(C(=O)NC(CCSC)Cc2ccccc2)CCCCC(C)(C)C1 98561,c1(C(=O)NC(CC)CNC(=O)C(C(C)C)OC)c(Cl)nc2ccccn12 98562,c1(C(=O)N(C2CC2)CC2CCCN2C(c2csnn2)=O)coc2c1CS(=O)(=O)C2 98563,C1(CNC(CC2CCC(NC(=O)OC(C)(C)C)CC2)=O)CCCC2(CCOC2)O1 98564,N(C(=NCCN1CCOCC1(C)C)NCC1(c2cccc(C)c2)CC1)CC(=C)C 98565,C(=O)(C#CC1CCCC1)NC(CC=CC)C(=O)N(C)CCC1CCCO1 98566,N1(C(c2cc(SC)oc2C)=O)CCC2(CCC2NC(c2occc2C)=O)CC1 98567,C=CCC(C)C(=O)N(C1(C(=O)N(C)CCn2ccnc2)CC1)C 98568,Cc1nn(CCO)c(C)c1C(=O)NCCCNC(=O)Cc1ccccc1Cl 98569,C1(COC)(NC(=O)Cc2nnc(C)s2)CCCN(C(c2ccc(OC)cn2)=O)C1 98570,c1(C(N2C(CNC(C(CCC)C)=O)CCCC2)=O)c(C)cccc1C 98571,C(=O)(C(O)CC(C)C)NCCN(C(c1csc(-c2nc(C)cc(C)n2)n1)=O)CC 98572,C12(NC(c3nc(COC)oc3)=O)CCN(C(=O)CN(C)C(N)=O)CCC1C2 98573,c1(NC(=O)NC2C(C(C)(C)C)OCCC2)nccc(Br)c1F 98574,C1(NC(C2CC(C)(CC)C2)=O)CN(C(C2C3CCC(=O)C23)=O)CCC12CCC2 98575,C=CCCC(C(=O)NCCCC(CC)CC)NC(c1cncc(CC)c1)=O 98576,N1(C(CCC2C(C)(C)C2)=O)CC2CC(C1)N(C(c1occc1Br)=O)C2 98577,C(C)(C)(C(C)CC(=O)NCC1CC12CC2)NC(CNC(=O)NC)=O 98578,N1(C(C(CCC#C)O)=O)CCN(C(c2ccc(CC)c(F)c2)=O)CC2(CC2)C1 98579,C(C1=CCN(C(=O)CC(F)(F)F)CC1)NC(Cn1c(C(C)C)nnn1)=O 98580,C(=O)(CCCC(F)(F)C(F)(F)F)NCC1(NC(c2nc(C#C)sc2)=O)CC1 98581,C1(C(C)(C)C)CCC(NC(=NCc2cnccn2)NCC(F)F)CC1 98582,N1(CCC)CCCCC1CN=C(NC(CC)CC)NC1CCS(=O)(=O)C1 98583,C1(NC(c2ccc(CCC)s2)=O)CC2CCC1N2C(C1CC2(CCO1)CC2)=O 98584,c1(C(=O)NC2CC3CN(C(c4c(CC)nccc4)=O)C2C3)cc2cccnn2c1 98585,C1(SC)CN(C(C2(O)CC(F)(F)C2)=O)CC1NC(C1(C)CC1(F)F)=O 98586,C1(NCc2cccc(-c3nnc(C)o3)c2)CCC(C)(C)CC1C(=O)O 98587,Cc1oc(C)c(CN2CCC(NCCN3CCCCC3)CC2)c1C 98588,C(c1cccc2cccnc12)=CC(=O)NC1CN(C(C2CC(C)(O)C2)=O)CC1O 98589,Cc1ccc2oc(C(=O)N(C(C)CN(C)C(c3cn(C)c(O)n3)=O)C)cc2n1 98590,c1(C(N2CCC(Cc3cn(C(C(=O)OC)C)nn3)C2)=O)cc(CO)ncc1OC 98591,c1(NC(=O)NC)cccc(C(=O)NCC(C)CN(C(=O)COC(C)CC)C)c1 98592,CCCC(C)(O)C(=O)NC1CC(CC(N2CCC2CC2CC2)=O)C1 98593,N1(C(c2cnc(C(C)C)o2)=O)CCOCC1CC(=O)NCC1(C)CCCC1O 98594,N1(C(C(C2CCCO2)NC(CCCCOC)=O)=O)CCC2(C1)CN(C)C2 98595,CC(F)(F)CCCC(=O)N1CCC(CNC(=O)CC(=O)NC2CC2)C1 98596,C1(C(=O)NCC2(CCC)CCC2)CCC(n2cc(-c3csc(C)c3)nn2)C1 98597,c1(C(=O)NC2COCCN(C(C3CC4(CCC4)CO3)=O)C2)ccc2ccnn2c1 98598,N1(C(=O)CNS(=O)(=O)C2CC2)CCCC(CCNC(C2(C3CCC3)CC2)=O)C1 98599,c1(C(N(C2CCN(CC)C2)C)=O)cnc(CNC(=O)C=Cc2cncs2)nc1 98600,CC(C)C(CCNC(c1cnn(CC2CC2)c1)=O)NC(=O)Cc1cn(C)nn1 98601,c1(OC)cc(OC)cc(C(c2n[nH]cc2Br)NC(c2nnnn2C2(C)CC2)C)c1 98602,c1(NC(C2CC23CC(NC(C2CCC2)=O)C3)=O)ccccc1CCO 98603,N1(CC)CC(C(=O)NCC(c2ccccc2)NC(c2ncn(CC)n2)=O)NC1=O 98604,CN1CCN(C(C2(C)CC2(C)C)=O)CC1C(=O)NCc1ccc(F)cc1 98605,N1(C(C2C(C=C)OCC2)=O)CCCN(C(c2nc(C)n(C)c2C)=O)C(C)C1 98606,c1(C(=O)NCC(CC)NC(=O)C2=CCCCO2)ccnc2ccncc12 98607,c1(C(=O)NC2CN(C(=O)C=Cc3cscn3)C3CC23)ccc(COCCO)cn1 98608,CS(=O)(=O)c1cccc(S(=O)(=O)N2CCC3C(CCN3C(=O)CNC(N)=O)C2)c1 98609,C1(OC)CCn2cc(C(=O)N(C)CCN(C(=O)C(C)C#N)C)nc2C1 98610,N1(C(COC)=O)C(C)CN(C(=NCCCc2cccs2)NCCCF)CC1C 98611,O=C(C1CC(O)c2ccccc21)NCC1CCN1C(c1n[nH]cc1Cl)=O 98612,CC(C)CC(O)C(=O)N(C(CNC(=O)CCC(=O)c1ccc(Cl)cc1)C1CC1)C 98613,N1(CC2CCC(OC)CC2)CCCC(C)C1c1cn(-c2cc(C)cc(F)c2)nn1 98614,N1(C(CS(CC)=O)=O)CCC2(CCCCN(C(C3(c4ccccc4)CC3)=O)C2)C1 98615,C(=O)(C(C)CS(C)=O)NCc1cn(C2CN(C(C=C(C)C(C)(C)C)=O)C2)nn1 98616,c1(OC)ccc(CCC(=O)NCC(C)N(C)C(c2ccc[nH]2)=O)cn1 98617,C(CC(=O)N(C(C)CNC(=O)C=C(C)C(C)C)C)N(CCC)C 98618,Cc1nc(C(=O)NCCOC(C)(C)CNC(=O)CC2(C)CCCO2)co1 98619,C1(CC)(CC)CC(NC(=O)Cn2nccc2C)CN1C(=O)CSC1CC1 98620,C(=O)(C(O)CC(C)(C)C)NCCCCNC(C(c1c(C)n[nH]c1C)C)=O 98621,Cn1ncc2c(C(N3CC4CN(C(c5cc(O)n[nH]5)=O)CC4C3)=O)cc(Br)cc12 98622,CC12CC(NC(c3csc(O)n3)=O)(C1)C1(CN(C(=O)CC3=NNC(=O)C3)C1)O2 98623,Cc1cc(CCC(c2nnnn2C(C)C)NCc2cc(C(=O)N(C)C)no2)no1 98624,C(C)(CNC(=O)C(=O)NCC(C)OC(F)F)(CO)OC 98625,C1(C(C)C)CCCC(C(N(CC(F)F)CCO)=O)C1 98626,c1(C(=O)NC2C3(CC(NC(C(CC=C)CC)=O)C3)C2)ccc(S(=O)(=O)NC)nc1 98627,C(CC(C(=O)N1CC(SC)C1)NC(=O)CC1CC=CCC1)OCC 98628,c1(NC(COc2cc(C)on2)=O)cccc(NC(=O)CC2CCNC(=O)C2)c1 98629,c1(C(=O)NCC(C)NC(=O)CN(C)C(N)=O)ccn2ncc(Br)c2n1 98630,N1(C(=O)C=CC2CCCO2)CCC2(NC(=O)C(F)(F)c3cscn3)CCCC12 98631,N1(C(c2ncc(C)nc2)=O)CCC(O)CC1C(=O)NOCC1CCC1 98632,N1(C(C(CC)O)=O)CC2CCCC(CNC(c3ncccc3F)=O)(C2)C1 98633,c1(NC(=O)NCCCNC(C(C)C)=O)cc(CN(C)C)nn1C 98634,c1(-c2cc(C(=O)NCCC(C)N(C)C(C3CC4CC4C3)=O)no2)cccc(Cl)c1 98635,c1(OCC)cncc(C(=O)NCC(C2CCC2)NC(=O)CC2CCN(C)C2=O)c1 98636,c1(-n2cc(CN(CC(=O)OC)C(=O)Cc3cscc3C3CC3)nn2)ncccc1C 98637,CC1CC(NC(c2ccn(CCNC(c3cc(C(N)=O)[nH]n3)=O)c2)=O)CCS1 98638,c1(CC)cc(N2CC3C(CNC(c4n[nH]cc4Cl)=O)C3C2)nc(CC)n1 98639,CCC(O)CC(=O)NCC(C)(F)CNC(c1c(C)nsc1C)=O 98640,N1(C(CN2CCC(OC)CC2)=O)CC2CN(C(=O)CSC)CCC2(CO)C1 98641,N1(C(c2c[nH]c(=NC)s2)=O)CCC(NC(=O)CN2CCCNS2(=O)=O)C(F)C1 98642,Cc1ccn(CCC(=O)NCC2CC(O)(CNC(=O)Cc3csc(C)n3)C2)n1 98643,C1(CNC(C(C)NS(C)(=O)=O)=O)CC2(CCC2)CN1C(c1cc(=O)cc(Cl)[nH]1)=O 98644,CCCCS(=O)(=O)NC(C)C(=O)NC1(CNC(c2nnn(C(C)C)c2C)=O)CC1 98645,N1(C(CC=CC=C)=O)CCN(C(c2ccc(Cl)c(CCC)c2)=O)C2(CC2)C1 98646,C1(C(=O)NCC(CC(N2C(C3(C)CC3)CCCC2)=O)O)CC(C)(C)CN1C 98647,C1(C(=O)NC2(CO)CN(C(=O)CC3OCCCO3)C2)CCC2(CCOC2)O1 98648,N1(C(c2cnc(CC)s2)=O)CC(C)CCC1CNC(=O)CNS(N)(=O)=O 98649,C1(CNC(=O)C(F)Cc2ccccc2)CN(C(C2SCCS2)=O)CCCO1 98650,C(CN=c1[nH]cnc(Cl)c1CO)N(C(C1Cc2ccccc2O1)=O)CC 98651,N1(C(c2c(SC)snn2)=O)CCCCC1CCCNC(C1CCS1(=O)=O)=O 98652,c1(C(=O)NCC2(C)CCCN2C(c2cccc[n+]2[O-])=O)ccc2scnc2c1 98653,C1(C(N2CC(CC(C#C)C)C2)=O)COC(CNC(=O)CCc2ccco2)C1 98654,CCCCCCC(C)(CC)C(=O)NCC(C1(O)CN(C(=O)C(C)(C)CC)C1)(C)C 98655,C(=O)(C(CC(C)(C)C)OC)NCC(CNC(C1CCC(=C)CC1)=O)OC 98656,c1(C(N2CCC(O)(C(N3CCOC(CO)C3)=O)C2)=O)c(F)cncc1F 98657,C#CCC(CC#C)C(=O)N(C)CC1(O)CCN(C(C2(C)CCN(C)CC2)=O)C1 98658,CC1CN(CC(=O)CCc2c(F)cccc2F)CC2(CCCOC2)O1 98659,CCC(O)CC(=O)N1CC(CC(C)NC(c2cc(-c3cccs3)on2)=O)C1 98660,C1(C(=O)NCCC(C)N(C(=O)CCCN2CCCC2)C)CCC2(CCC2)OC1 98661,C1(C(=O)NCC(C(C)C)NC(CC(C(F)(F)F)OC)=O)COc2ccccc2O1 98662,N1(C(c2ccc(N(CCC)C)cc2)=O)CCN(C(=O)CSCCO)C2CC12 98663,CN1CCOc2ncc(C(=O)NCC3(NC(C4CCCOC4)=O)CCCC3)cc21 98664,CC1CC(C(=O)NC2C=CCC2)N(C(C2CCOC2(C)C)=O)C1 98665,C(CC(F)F)(C(=O)NCCC1(C)CCCO1)N(C)C(C1CC(C2CC2)=NO1)=O 98666,N1(C(C2CN(CC)C(=O)C2)=O)CCC(NC(C2CN(S(=O)(=O)C(F)F)C2)=O)C1(C)C 98667,C1(c2cn(CC3CC(F)(F)C3)nn2)(NC(=O)CC2CCCO2)CCCOC1 98668,C(=O)(CCCC(C)(C)NC(=O)C=Cc1cccnc1)N1CCC(CC)C1 98669,C1(NC(c2coc(C(F)F)n2)=O)CN(C(=O)CN2CCCNC2=O)CCC1O 98670,N1(C(C2(CNC(C3CCSC(C)C3)=O)CC(=C)C2)=O)CCOC(C)(C)CC1 98671,C(=O)(C(CNC(c1csc(F)c1)=O)CC1CCCC1)N(C)CC1(CO)CCC1 98672,C1(NC(C(C)NC(=O)C(C)(C)C)=O)CN(C(=O)CSCCN(C)C)CC1COC 98673,c1(CNC2CCCN(c3cc(COC)ncn3)C2)cc(Br)ccc1OCC 98674,C1(NC(Cc2cn(CC)nn2)=O)CCC(C)N(C(=O)CC2(C)OCCO2)C1 98675,N1(C(C(C=C)(C)C)=O)C(CNC(=O)CCOC)CC2COCC12 98676,N1(C(c2c(C#N)ccs2)=O)C2CC1CN(C(=O)CC1CCCC13CC3)C2 98677,O=C(CCCCCCNC(C1CCOC(=O)CC1)=O)NC1CCC=CCC1 98678,C(CCN=c1[nH]c(N2CCN3CCOCC3C2)nc2c1SCC2)SCC(C)C 98679,CCCC(C)(CC)C(=O)NCc1ncccc1CNC(=O)Cc1ccsc1C 98680,c1(OC)ccc2c(c1)C(C)CN(C(=O)C(N1CC(=O)N3CCCC3C1)=O)CC2 98681,C1(C(N(C2CCN(C(c3cc(C(C)(C)C)on3)=O)C2)C)=O)CCCS(=O)(=O)N1 98682,C1(C(=O)NC(CC)C(=O)N(C)C)CC(NC(C2(C)CC(C)=NO2)=O)C(O)C1 98683,c1(C(N2CC(CNC(CN(C(C)C)C)=O)C(C)CC2)=O)cn2cc(Cl)cnc2n1 98684,c1(CNC(c2cc(CNC(C(CC)(C)O)=O)no2)=O)cc(C)cc(F)c1 98685,Cc1cc(C(F)F)n(CC(=O)NC(CNC(=O)C(C)CC2CCC2)C2CCC2)n1 98686,N1(C(C2(C)CC2)=O)CCOC2(CCN(C(c3cc(C)nc4c3c(C)nn4C)=O)C2)C1 98687,CC1CN(c2nnc(-c3cc(C4CC4)[nH]n3)n2C)CC(c2ccsc2)O1 98688,c1(CNC2CCN(C(Cc3ccc(OC)cc3)=O)C2)c[nH]c2cccnc12 98689,CCCCCC(C)CC(=O)NCCN(C(=O)C(F)CC1CCCC1)C 98690,N1(C(c2cccc(C(C)C)n2)=O)CC(CNC(=O)COC2CC2)N2CCC1C2 98691,C(CC(F)F)(C(=O)NCc1cc(O)cc(F)c1)N(C)C(c1ccnc(CO)c1)=O 98692,C12CCC(CC1)C(=O)NC(C(C)O)C(=O)N2.C(CC(=O)N1CCCC1)NC(C)=O 98693,n1(CC(=O)NC2C3N(C(c4c(C)cn(C)c4)=O)C(CC3)C2)cc2ccccc2n1 98694,N1(C(CC(CC(C)C)C)=O)CCC2CN(C(C3CC34CC4)=O)C(C)C12 98695,C1(CNC(C2N(C(N)=O)CC(O)C2)=O)CC2(CC2)CN1C(=O)CCC1CC1 98696,C1(C(C)NC(C2CCNC2=O)=O)CN(C(=O)C(c2cccc(Cl)c2)(C)C)CCO1 98697,c1(C(C(=O)NC2CCC2)N(C(C)C)Cc2ccccc2)ccc2ncccc2n1 98698,N1(C(C(C)(C)CF)=O)CCN(C(c2cc(F)c(CO)c(F)c2)=O)CC(O)C1 98699,c1(C(=O)NC(C2(O)CN(C(Cn3ncc(C)c3)=O)C2)C)nc(C2CC2)ncc1Cl 98700,N1(C(C(C=CCCC)O)=O)CCN(C(=O)CNC(=O)OCc2ccccc2)CC1 98701,Cc1cc(C(N2CCCC2CCCNC(C2CC23CCSCC3)=O)=O)nc(C)c1 98702,CC(C)CC(C(=O)NC(CCF)C(=O)NCCCOC1CCC1)C(N)=O 98703,c1(C(=O)NCCN(C)C(c2ccc(C(F)C(F)(F)F)cc2)=O)ccnc(Cl)c1N 98704,c1(C(=O)NCC#CC(=O)NCC2CN(C(C)=O)C2)c[nH]c(=S)cn1 98705,c1(C(=O)NCC2(O)CCN(C(C3N(C)C(=O)OC3)=O)C2)cncc2c1CCCC2 98706,C(=O)(NNC(=O)c1ccc(I)cc1)NCC(C)C#N 98707,Cc1c(Cl)ccnc1C(N1CCC(C)(NC(C23CCC(CC2)OC3)=O)C1)=O 98708,C(=O)(CC(C)CC(=O)NC1(CCNC(C2CCN(C(=O)C3CC3)CC2)=O)CC1)OC 98709,c1(COC)csc(C(=O)N(CCNC(C2CCCC2O)=O)C2CC2)c1 98710,N1(C(C(CC#C)C)=O)C2CCC1CN(C(=O)Cc1ccc(Cl)nc1F)C2 98711,C12(C(N3CC(O)CC(NC(c4ccncn4)=O)C3)=O)CCCC(CCC1)C2O 98712,C(C)(CCC(F)(F)F)(C(F)(F)F)NC(CNc1ccc(OC)cc1)=O 98713,C(=O)(CCC(C)(C)F)N(CC(Cc1ccccc1)NC(C1CCSC1)=O)C 98714,CC1CCC(NC(c2c(C(F)F)cccc2F)=O)CN1C(c1cccc(N)n1)=O 98715,C1(C(N2C(CNC(=O)Cc3cnns3)CC2)=O)CC12CCCCCC2 98716,c1(C(N2CCC(N(C(C(C)=C3CCCC3)=O)C)C2)=O)c(C)c[nH]c1CC(N)=O 98717,C1(C#N)(C(=O)NCCn2cc(CNC(CN3CC(C)C3)=O)nn2)CC12CCC2 98718,C(=O)(CCS(C)(=O)=O)NCC(C)(CO)NC(=O)CSCCCc1ccccc1 98719,N1(C(C(CN(C)C)N(C)C)=O)CC(O)(C2(CNC(C3(C)COCCO3)=O)CC2)C1 98720,C1(CCNC(=NCCC)NC2CCNC(=O)C2)CCC2(CC1)OCCO2 98721,c1(CNC(C2C(CNC(C3(C)C(C)(C)C3)=O)C2)=O)ccncc1F 98722,c1(C(N(CC(C)NC(=O)C(c2ccc(C(F)F)cc2)C)C)=O)cc(Cl)cn1C 98723,C1(CNC(Cc2c(C)nc[nH]2)=O)CN(C(=O)CC2CCC(C)C(C)C2)CCCO1 98724,Cc1nc2c([nH]1)C(C(=O)N1CCC(N(C)C(C3CC3C)=O)C1)CCC2 98725,CC(C)CC(CNC(c1cnn[nH]1)=O)C(=O)N(C)CCc1ncon1 98726,N1(C(c2cc(SC)oc2)=O)CC(CNC(c2sccc2C(F)F)=O)C(C)C1 98727,C12(CNC(c3cccc(OC)n3)=O)CCC(CC1)N(C(=O)CC1CCC3CC13)C2 98728,C1(C(N(CCCNC(C2CC(n3cnnc3)C2)=O)CC)=O)CCC(=O)NC1 98729,C1(CNC(C2(NC(C(CC3CCC3)OC)=O)CCSC2)=O)CCCCC1(C)C 98730,c1(C(=O)NCCCCN(C(Cc2cc(C)sc2C)=O)C)cc(O)nc(O)n1 98731,c1(C(=O)OC)cc(C)nc(N(C(C)CNC(=O)Cc2cc(C)ns2)C)n1 98732,C1(NC(C=C(C)C(C)(C)C)=O)CCC(NC(=O)CC(O)c2ccccc2)CC1 98733,Cc1c(C(=O)NCC2(CNC(C3CC4C(C3)C4(C)C)=O)CCCC2)cccc1N 98734,Cc1cc(C(=O)NC2CC2NC(c2nccnc2C)=O)cc(C)c1Cl 98735,C1(NC(=O)CC2COCCO2)CCOC12CCN(c1ncc(O)cn1)CC2 98736,C(=O)(C1=CC(C)(C)C1)N1CCC(CC(C)NC(=O)CCC2CCCCO2)CC1 98737,c1(OC)c(NC(C2CC(F)CN(C(=O)CCC3CC3)C2)=O)cccc1Cl 98738,CC1(C)Cc2c(cnn2-c2ccccc2)CN(C(c2cc(I)cs2)=O)C1 98739,C1(CCNC(CCCNC(N)=O)=O)CCN(C(=O)Cc2ccsn2)CC1 98740,O=S(=O)(c1cccc2ccc(Cl)cc12)NCCCCC(F)(F)F 98741,CCCCS(=O)(=O)CC(=O)N1CC2C(CN(C(=O)CCc3cn(C)cn3)C)C2C1 98742,n1(CCC(=O)NC2CN(C(C3CC3C(F)(F)F)=O)CC2O)ncc2c1CCCC2 98743,N1(C(C=CC)=O)CCC(C(C)NC(C2(CCS(N)(=O)=O)CCC2)=O)CC1 98744,C1(NC(CCCc2onc(C)n2)=O)CC2CCC1N2C(C1CC(C(C)C)=NO1)=O 98745,N1(C(C2C(NC(CNC(C3C(C)C3)=O)=O)CCO2)=O)CCC(CCN(C)C)CC1 98746,C1(CC)CN(C(=O)Cc2ccnc(Br)c2)CCN1C(c1nc(O)c(C)s1)=O 98747,C1(CNC(CCCOCC)=O)CCC(C)(C)CN1C(=O)C(C1CCCCC1)OC 98748,N1(C(CC2C(C)CCCC2)=O)CC2CN(C(=O)CCNC(=O)CO)CC(C1)O2 98749,N1(C(C2C(C=C)C2)=O)CC2CCC1C(NC(=O)C(C)Oc1cccc(F)c1)C2 98750,C(=O)(C(CC)(CC)C(C)C)N1C(C(N2CCC(=CCC)C2)=O)CC1C 98751,c1(C(N2CCC(CC)(NC(=O)CCCCF)CC2)=O)cccc2c1C(=O)NC2=O 98752,c1(N2CCCC(C)CC2)nc(=NCCCc2ccccc2Br)[nH]c2ccccc12 98753,C(c1cccnc1)=C(C(=O)NCCCCCNC(c1[nH]cc(C(=O)OC)c1)=O)F 98754,N1(C(C2(SC)CCC2)=O)CCC(C=CC(=O)Nc2ccn(CCO)n2)CC1 98755,C1(C(N2C(C(=O)NCC(COC)(C)O)COCC2)=O)CC2(C1)CC2(F)F 98756,c1(C(=O)NCC(C)NC(c2c(CC)nc[nH]2)=O)ccc(F)c(Cl)c1N 98757,N1(C(C2(C)CC(F)(F)C2)=O)CCC(O)C(NC(C2CC23CCC3)=O)C1 98758,c1(C(=O)OC)ccnc2c1CCC2NC(c1cc(F)cc(F)c1)=O 98759,CC1(C)SCC=C1C(C(=O)NCCc1cccc(F)c1)N1CCc2nn[nH]c2C1 98760,c1(C(=O)NC2CC(CNC(C(Cc3ccccc3)OC)=O)C2)cccc(C)c1F 98761,C12(CNC(C3N(CC)CC3)=O)COCCN1C(=O)CN(C(c1cnc(S)[nH]1)=O)C2 98762,c1(CC)ocnc1C(=O)NC(C)C(CO)NC(c1cc(F)n[nH]1)=O 98763,C12(NC(C(CC)CC)=O)CC3CCC(C1C2)N3C(=O)Cc1cn(C)nn1 98764,c1(N2CC(C(=O)Nc3c(CC)cc(Br)cc3)SCC2)ncnc2cc(I)sc12 98765,N1(C(Cc2c(C)ncnc2C)=O)CCC2CN(C(=O)CC3NC(=O)NC3=O)C2C1 98766,c1(N2CCCC(C#N)C2)nc2c(c(=NC3CCc4nn[nH]c4C3)[nH]1)COC2 98767,C(=O)(C(C)(C)C(C)O)NCC1(C(C)NC(c2nc(CC)sc2)=O)CC1 98768,c1(OC)cc(OC)cc(C(=O)OCCSCc2cc(Br)oc2Br)c1 98769,C(C)(C)(CC(=O)N1CC(C)(CCC(N2CCOCC2C(C)C)=O)C1)OC 98770,N1(CC)CCOC(C(N2CCC(CNC(C3(COC)CC3)=O)C2)=O)C1 98771,Cc1cc(C(N2CC(NC(c3c(C4CC4)cccc3F)=O)C(F)C2)=O)c(C)n1C 98772,C1(C(C(=O)NC2COC2)N(C(C2(O)CCC2)C)C)CCOC(C)(C)C1 98773,C1(NC(C2C(C(=O)OC)C2)=O)CCN(C)C12CCCN(C(c1sccc1Cl)=O)C2 98774,c1(C(c2nnnn2CSc2ccccc2)NC(CCC)C)cc(Cl)n(C)n1 98775,c1(C(N(CC(CC)NC(=O)CCCn2cncn2)C)=O)cnn2cccc(Cl)c12 98776,C1(CNC(c2c(Cl)ncc(C)c2)=O)CCC2CN(C(C3CC3F)=O)CCC2C1 98777,C1(C(N(CCC)CCNC(=O)CC2CC2)=O)CC12CCc1ccccc12 98778,c1(C(=O)OC)cc(C(N2CC(CNC(=O)CCC3CCCO3)(OC)C2)=O)nn1C 98779,n1(CCC)ncc(C(=O)NC(CNC(C2CCCN2CC(C)C)=O)C2CC2)c1C 98780,CC(CCN(C)C)C(=O)NC1CC(C)N(C(=O)CCC(=O)N(C)C)C1 98781,C1(CN(C(c2n(CC)nnc2)=O)C)COCCN1C(c1nncs1)=O 98782,C#CCC(CCOC)NC(=O)C(C)N(C(C1CNC(=O)C1)=O)CC 98783,C(=O)(CC(CC)NC(=O)C(O)C1CC1)NCC(=O)OCC=C 98784,C1(NC(C2C(C(C)(C)C)C2)=O)CC2CC1N(C(C1CN3CCC1CC3)=O)C2 98785,c1(CC)nc(C(=O)NC(C)C(=O)NCC2CCN(C(C)=O)C2)co1 98786,N1(C(COCCCOC)=O)CCCC(C2CCN(C(=O)COCCF)CC2)C1 98787,C=CCCCC(=O)NCC1CCCC(CNC(=O)CCc2cnc(C3CC3)o2)C1 98788,C1(C)(NC(CC2(C)CCC2)=O)CCCN(C(C2CC(C)(F)C2)=O)C1 98789,C=CC1(NC(=O)C(F)CC2CN(C(c3cccc(CO)c3)=O)C2)CCOCC1 98790,c1(NCCCNS(NC)(=O)=O)cc(S(=O)(=O)N(C(C)C)CC2CC2)ccc1C#N 98791,CC#CCC(C)NC(=O)CN(CCC)C(c1cccnc1)=O 98792,C1(CNC(c2nc(CC)sc2)=O)CCC(C)N(C(c2cnc(C3CC3)o2)=O)C1 98793,C(=O)(C(CN=[N+]=[N-])NC(c1n[nH]c2c1CCC2)=O)NCC1CCCN(C)C1 98794,N1(C2CN(C(C(=O)OC)C)C2)CC(O)CCC1=O.Cc1ccc(C2(C)CC2)cc1 98795,CN=c1ncc(-c2cnc(NCc3ncc(C)cc3F)nc2)c[nH]1 98796,CCC1=C(C(=O)N(C)CC2CCCN(C(c3cnncc3NC)=O)C2)CCCO1 98797,N1(CCC(=O)NC23CC(C2)N(C(c2cnoc2C2CCC2)=O)C3)C(=O)CCC1=O 98798,c1(C(=O)NCCN(C(=O)CC2C(=O)NN=C2C)CC)ccc(P(C)(C)=O)s1 98799,CC1CN(C(=O)C=Cc2nccs2)CCN(C(C2CC=CC2)=O)C1 98800,c1(C(=O)NC2CCCCN(C(C3N(CC)CCC3)=O)C2)c(C)c(C)nn(C)c1=O 98801,c1(CCNC(c2cnn(C)c2OC)c2n(CCOCC)nnn2)ccccc1C 98802,c1(C(C(=O)NC)N(C)CC2(C)CCCO2)cn(C)c(=O)n(C)c1=O 98803,C(=O)(C#CC1CCOC1)NCCN(C(c1cnc(C(C)C)s1)=O)CCOCCO 98804,N1(C(C2(C)N(C)CCC2)=O)CCCC(CO)(CNC(=O)CCc2cnccn2)C1 98805,c1(CCCCC)cc(C(=O)NC2(CO)CN(C(c3cc(C(N)=O)co3)=O)C2)n[nH]1 98806,c1(C(C(=O)NC(C(C)NC(C(C)Cn2ccnc2)=O)CO)(C)C)ccccc1Cl 98807,C1(C(C)(C)C)CCCC1C(=O)NCC1(NC(=O)Cc2cscn2)CCC1 98808,c1(COC)ncc(C(=O)NC(C)(CNC(C2CNC(=O)N2)=O)C2CCC2)s1 98809,CC(N=c1nc(N2CCC(CCF)CC2)c2c([nH]1)CSC2)C1CCCO1 98810,N1(C(c2cc(Cl)ccn2)=O)CC2(CCCN2C(=O)N(CCCl)CCO)C1 98811,c1(NC(C(=O)NCCC2CCCS(=O)(=O)C2)=O)cccc2c1OCCC(=O)N2 98812,N1(C(C2CN(C)C(=O)C2)=O)CC2(CCCC(CNC(=O)C(F)=CCCF)O2)C1 98813,c1(NC(=O)NCc2cc(Br)nn2C2CCCCO2)cc(-c2ccccc2)ccn1 98814,c1(NC(C2(F)CN(CCO)CC2c2ccccc2)=O)cccc(F)c1Cl 98815,C(=O)(CS(=O)(=O)C1CCCC1)NCC1CN(C(C(CSC)OC)=O)C2(C1)CCC2 98816,N1(C(C(C=C)OC)=O)CC2CC2(NC(C2C3CCC(=O)C23)=O)C1 98817,C#CCC(C)(C(=O)NC1CC1(C)CCC)NC(=O)CCOC1CCCC1 98818,C1(C(N2CCCC(CC3CC3)C2)C(=O)NCC(=C)C)C2CCOCC12 98819,C(c1c(C)cccc1C)=CC(=O)NCC(CCC)NC(C1(n2cccn2)CC1)=O 98820,c1(C(=O)NC(CC=C)CNC(C2CCCCCN2C)=O)cc2cc(C)ccc2o1 98821,C1(C)(CCNC(C2N(CC)CCC2)=O)CCN(C(=O)CCc2cccn2C)C1 98822,c1(C(N2CC(C(C(=O)N(CC(C3CCC3)OC)C)O)C2)=O)sccc1Cl 98823,C(CC(F)F)(C(=O)N(C12CCC(CC1)CC2)C)n1cc(-c2cccc(C)c2)nn1 98824,Cc1nc2cc(C(N3CC(NC(=O)CC(C)P(C)(C)=O)C(O)C3)=O)cc(O)c2[nH]1 98825,C1(C(=O)NCCN(C(C2(COC)CCCCO2)=O)C)CC(=O)N(OC)C1 98826,c1(CC(=O)NC2CC(C)(NC(C3N(C)CCC3)=O)C2)cc(F)ccc1O 98827,c1(C(N2C(C)(C(=O)OCC)CCC2)=O)ccc2c(Br)cnn2c1 98828,c1(C(=O)NCC(CNC(CCCNC(N)=O)=O)F)sc([N+](=O)[O-])cc1Cl 98829,c1(C(N(c2c(O)nc(=O)n(Cc3ccco3)c2N)CC)=O)ccn2nccc2c1 98830,C(C(CC(C)C)C(=O)N(C1CCCCC1NC(c1cccc(F)c1C)=O)C)OC 98831,c1(C(N(C)CCN2CCN(C(C3CC3C(F)F)=O)CC2)=O)cnc2[nH]ccnc1-2 98832,c1(NC(c2cccc(Br)c2)=O)ccc2[nH]cc(-c3ccc(C(=O)O)c(F)c3)c2c1 98833,c1(C(=O)NCCOCCNC(C(C(C)SC)O)=O)c(C)oc2ccccc12 98834,CC(CC(=O)N1CCOC(CC(=O)NCC(F)Cl)C1)C(C)(C)C 98835,CC1(C)CC(C(=O)NC(C)(CO)C2CC2)CN(C(C2(C3CCCC3)CC2)=O)C1 98836,Cn1nc(C2CC2)c(Br)c1C(N1C(CO)CSCC1c1ccccc1)=O 98837,Cc1nc(C(C)(C)C)nc(O)c1C(N1CCCC(C)(NC(C2CC2CF)=O)C1)=O 98838,C(=O)(C(C(C)(C)C)N1CCCC1=O)NC1CCN(C(c2ccc(OC)cn2)=O)C1 98839,N1(C(COCC=C)=O)CC(CNC(C2CCCN2CC(C)C)=O)C(C)C1 98840,N1(C(C(C)(C)C2CCCCC2)=O)CCC(O)(CCNC(=O)CSC(F)F)C1 98841,Cc1ccc(C(N2CC(NC(c3ncoc3C(C)C)=O)CC(C)C2)=O)c(N)c1C 98842,N1(C(C2C=C(C)CS2)=O)C(C)CN(C(=O)CC2CCC(C)(C)O2)CC1C 98843,C(=O)(C#CC1CCOCC1)NC1C(NC(c2c(C)noc2C)=O)CCCC1 98844,C1(N(C(=O)CSCCN(C)C)CCC)CCN(C(=O)C(COC(C)(C)C)NC)C1 98845,C#Cc1cccc(C(=O)NC(CNC(c2ccc[nH]2)=O)CCOC)c1F 98846,C=CCCN=C(NCc1ccc(O)cc1Cl)N1CCCC(C(O)C(F)(F)F)C1 98847,C(=O)(C(C)(C)CC(C)(C)C)N(C)CC1N(C(C(C)S(C)(=O)=O)=O)CCC1 98848,c1(CN2CCC3(C(C(=O)Nc4ncc(C#N)cn4)C3)C2)ccc([N+](=O)[O-])c(Br)c1 98849,c1(C(=O)NCC2N(C(c3cc(CC)c(Cl)cc3)=O)CC2)ccc(N)c(C)c1C 98850,c1(CC)cccc(CNC2CCCCN(C(=O)CCCCCBr)C2)c1O 98851,c1(C(=O)NC2CCN(C(C(CC)(C)O)=O)CC2CO)cccc2c1CCO2 98852,N1(C(c2ccc(OC)cc2)=O)CCN(C(=O)Nc2cc(Br)ccc2OC)CC1C 98853,c1(C(N(C)CC2(O)CCN(C(Cc3nc(CC)sc3)=O)C2)=O)cccc(N)c1C 98854,N1(CCC=C)CCC2(CC1)OCCc1cc(C(=O)NCC3(C(C)C)CC3)sc12 98855,c1(C(=O)NCCN(C(=O)C(F)n2ccnc2)CCC)cc(F)c(Cl)cc1Cl 98856,c1(C(=O)N(C(C(CCCC)CC)=O)C2(C)CC2)ccc2c(=O)n(C)c(C)cc2n1 98857,c1(NC(c2c(C)n(C)nc2)c2nnnn2C)cc(NS(C)(=O)=O)cc(Br)c1 98858,C1(C(N(C)CC2CCN(C(CCC=CCC=C)=O)CC2)=O)Cc2ccccc2C1 98859,N1(C(C=C(C)C(C)(C)C)=O)CC(O)CC1CNC(=O)C(O)C1CC1 98860,c1(C(=O)NCC(C(=O)NC(CCC)C(=O)N(C)C)O)cc(C)c(C)nn1 98861,N1(C(c2cccc(SC)c2)=O)CC2(C1)OC1(C)CC2(NC(C2CCC(C)O2)=O)C1 98862,Cc1cnn(C)c1CNC(C1C(C)CCN1C(=O)CC(C)(C)C)=O 98863,C1(C(N(C2CCOC2)C)=O)(CF)CCN(C(c2ccn(C(F)F)n2)=O)C1 98864,N1(C(C(CN(C)C)NC(c2cc(C)nnc2)=O)=O)Cc2ccc(O)cc2C1 98865,CCCC(C)CCCC(=O)N(CC(O)CNC(=O)Cc1csc(CC)n1)C 98866,C1(C(C)NC(C(=O)NCC2N(S(CC)(=O)=O)CCC2)=O)Cc2ccccc2CO1 98867,C(C)(C(=O)NCC1CN(C(=O)C(F)C(F)(F)F)CCCO1)(C(C)C)NC(C)=O 98868,C1(C(=O)NCCN(C(c2nc(OCC)oc2)=O)C2CC2)CCCC12CC2 98869,C1(NC(=O)NCCCNc2ccc(C)cc2Br)CC(C)c2ccccc2N1 98870,N#Cc1cnc(N2CCC(F)(F)C(CNC(c3cccc(Cl)c3Cl)=O)C2)c(Cl)c1 98871,N1(C(c2sc(C)c(Br)c2)=O)CCC2CN(C(c3c(F)cccc3Br)=O)CC12 98872,C1(C(=O)NCC(C)OCC=C)(OC)CCN(C(C2COCC(C)O2)=O)C1 98873,Cc1cn2ccnc(C(=O)NC3CCCC3CNC(c3cn(C)nn3)=O)c2n1 98874,CC(=O)CCCCC(=O)NCC(CNC(=O)C(c1ccnn1C)C)CO 98875,CONC(=O)C(=O)N1CCC(C(F)C(=O)NCC2C3CCCCC23)C1 98876,C1(C(N(CCC(C)NC(=O)Cn2cnc(C(N)=O)n2)C)=O)C(C)(C)C1(F)F 98877,c1(CC)cc(C(N2CCCC(NC(=O)Cc3cc(C)sc3C)CC2)=O)ccc1O 98878,C(=O)(CN1C(=O)Cc2ccccc21)N1C(CCN(C(C(CC)F)=O)C)CCCC1 98879,C1(NC(c2c(OC)cccc2)=O)COC2(CCN(C(c3coc(CO)c3)=O)C2)C1 98880,c1(CN2CC(OC)C(NC(=O)C(C)(C)CN(C)C)CC2)c[nH]c2cc(Br)ccc12 98881,c1(CC(N2CCC(NC(Cc3c(C)cccn3)=O)C2)=O)ccc2oc(O)nc2c1 98882,C1(C(N(C(C)C(=O)N(C)CCc2cc[nH]n2)CCC)=O)CCC(CC)O1 98883,N1(C(C(C)CO)=O)CCC2(CCCC2NC(=O)C=CC2CCOCC2)CC1 98884,C1(C(N(CCn2c(C)ncc2)C)=O)CCC(O)CN1C(c1cccc(F)c1O)=O 98885,c1(NC(=O)NC)cccc(C(=O)NCC(C)(C)NC(C2CCC(O)C2)=O)c1 98886,C1(CC#C)(C(=O)N(C2CCCCC2O)C)CCN(C(C2CCOC2C(C)C)=O)C1 98887,C12(NC(=O)CCC3CCCO3)CC3CCC(C1C2)N3C(=O)CC1(C(F)(F)F)CC1 98888,N1(C(C2(OCC)CCSCC2)=O)CCCC(NC(=O)CC2(C)CC2(F)F)CC1 98889,c1(C(=O)NCCOC2CN(C(c3cc(C(N)=O)[nH]n3)=O)C2)noc2c1CCCC2 98890,c1(C(=O)NC(CN(C(=O)CCC(C)SC)CC)C)cccc2c1NCCC2 98891,c1(C(=O)NC2CC(CNC(C(CC)OCC)=O)C2)ccc(OC)cc1F 98892,C(=O)(CCS(C)(=O)=O)N(C1CCN(C(c2c(C)onc2)=O)CC1)CCN(C)C 98893,c1(C(=O)NC(CN(C(=O)C(F)CC2CCC2)CC)C)cc(OC(C)C)cc(F)c1 98894,n1(CC(N2CCn3nc(Br)nc3C2)=O)ncc2c(c1=O)CCCC2 98895,C1(C(=O)NCc2n(CC)ncn2)CC2CC1CC2NC(c1cc(C)nnc1C)=O 98896,C1(CC(C)NC(C(=C(C)C2CC2)F)=O)CCN(C(=O)CNC(N)=O)CC1 98897,C(=O)(C(C)C(=O)NC1(CO)CN(C(C2(CO)CCC2)=O)C1)OC 98898,C(=O)(C1c2c[nH]nc2CN1C(=O)CCNC(C)=O)NCCOCCC 98899,C1(CNC(CC2CCCN(C)C2)=O)CN(C(=O)Cc2cccnc2)C(C)(C)C1 98900,c1(C(N(CCC)CCNC(C2(F)CCC2)=O)=O)cc(C)c2c(c1)CCC2 98901,C1(CC)CN(C(c2cnns2)=O)CC1NC(c1ccc(C(C)(C)CC)cc1)=O 98902,CC1Cn2nccc2CN1C(C12CC(C)(CN1C(=O)C1=CCCOC1)C2)=O 98903,C#Cc1cnn(C)c1C(=O)N(CC(N1C(C(=O)OC)CC1C)=O)C1CC1 98904,c1(SC)cccc(C(N2CCC(NC(c3cncc(C)n3)=O)C2)=O)c1O 98905,N1(C(c2ccc(SC)o2)=O)CCC2(COC(CNC(C3(C)CCSCC3)=O)C2)C1 98906,c1(C(=O)NC(CNC(c2cc(CC)n(C)n2)=O)C)c[nH]cc(Br)c1=N 98907,c1(C(N(CCNC(C2CCC(COC)O2)=O)CC)=O)c(Cl)ccc(OC)c1N 98908,c1(CN2CC(F)CC(C(N3CC(CC)OCC3)=O)C2)c(Cl)ccc(Br)c1F 98909,C1(CCN)CCNCC1(F)F.c1(C(C(C)C)NC(=O)C(=O)N)ccccc1F 98910,C1(C(C(=O)NCCOCC=C)C)CCNCC1 98911,C(=O)(C1=C(C)CCOC1)N1CC2C(C(=O)NC(c3ccncc3)CC)(COC2)C1 98912,c1(C(N2CC(CCNC(C3CC(C)(CC)C3)=O)C2)=O)cc(C)ccc1[N+](=O)[O-] 98913,CC(C)C(F)(F)CC(=O)NC1CCC(C)N(C(c2cc(=O)c(Br)c[nH]2)=O)C1 98914,C1(C(=O)NCC(CCNC(C2OCCC2C(C)C)=O)OC)CCCN(C)C1 98915,c1(C(=O)O)cc(CNC2CC(NC(=O)Cc3ccc(Cl)s3)C2)cc(Br)c1 98916,c1(CC(=O)NCC(CNC(C(CC(C)C)O)=O)C)coc2c(Cl)c(Cl)ccc12 98917,C1(NC(c2c(C(C)C)cnn2C)=O)CN(C(=O)C(F)C(C)(C)O)CCC1O 98918,c1(CC)cccc(C(N2CCC(CCNC(C3(C)C=CCC3)=O)C2)=O)c1N 98919,c1ccc(C)cc1.C#CCCCN(CC(=O)NCC(=O)NCCC(=O)OC)C 98920,C1(C(=O)NCC(CCNC(C2(C)CC(F)(F)C2)=O)O)COC2(CCC2)CO1 98921,c1(CC)cc(C(=O)NCCCNC(=O)C(c2ccc(C)cc2)C)cn(C)c1=O 98922,c1(C(=O)NC2(C#N)CCC(C)C2)ccc(S(=O)(=O)N2CCOCC2)cc1 98923,N1(C(C(Cc2cc(C)c(Br)cc2)(C)C)=O)CC2CCN(C)C2C1 98924,C(S(=O)(=O)C(C)C(=O)NC(C)CCSC)c1cncc(OC)c1 98925,Cc1c(C(N2CC3C(N(C(=O)C(F)CC4CC4)C)C3C2)=O)oc2c(Cl)cccc12 98926,c1(C(N(C(C)CNC(c2conc2C)=O)CC)=O)cc(F)ccc1N 98927,c1(C(C)=O)cc(=NCC2CN(C(C3CC(C)CO3)=O)CCO2)[nH]cn1 98928,N1(C(C2CC=C(C)CC2)=O)CCCC(C2CC2NC(=O)C(C)(C)C(F)F)C1 98929,CC1C(=O)N(C)CN1C(=O)Nc1cnn[nH]1 98930,c1(NC(C(C(C)NC(C(C2CCOCC2)C)=O)(C)C)=O)cccc([N+](=O)[O-])c1 98931,C12(C(C)C)CCC(NC(=O)C(Cn3cccn3)NC(=O)CN3CC=CC3)C1C2 98932,c1(C(N2C(CNC(=O)Cn3cncn3)CCC2)=O)ccc2nn[nH]c2c1 98933,C(C)(C)(CC(F)C(=O)NC(C1CCOC1)CO)NC(C1CCN(C)C1=O)=O 98934,c1(C(N2CC3C(CNC(C(C)CC(F)F)=O)C3C2)=O)nnc2ccccc2c1N 98935,CN=c1[nH]cc(C(N2CCCC(C3CCCCN3C(=O)CNC(N)=O)C2)=O)s1 98936,C1(C(C)C)COCCN(C(c2ccn(C(F)F)n2)C(=O)NCCCC2CC2)C1 98937,Cc1cc(C(N2CC(NC(c3cncc(Cl)c3)=O)C3(CC3)C2)=O)nc(N(C)C)n1 98938,C1(S(C)(=O)=O)(C(=O)NC2C(CNC(C3C(C)C3C)=O)C2)CC1 98939,N1(C(Cc2c(C)ocn2)=O)CCC(C)(C)C1C(=O)NCCCN1CCC(O)C1 98940,c1(C(=O)NCC(CC)NC(CSCC=C)=O)cn2c(Br)cnc2s1 98941,c1(N(C)C)ccnc(C(=O)NCCC2CCCN2C(=O)C=Cc2ccco2)c1 98942,C1(NC(=O)CC2CC=CC2)CCC(O)CN(C(C2(c3ccc(Cl)cc3F)CC2)=O)C1 98943,c1(OC)ccc(C=CC(=O)NC(C)(C)CN(C)C(C2CCCC(O)C2)=O)cc1F 98944,c1(C(N2CCC(N(C(=O)CN(C)C3CC3)CC)C2)=O)cccc2nsnc12 98945,Cc1cc(-c2cn(Cc3csc(C(F)(F)F)n3)nn2)ccc1N(C)C 98946,N1(C(C(Cc2cccc(OC)c2)N)=O)CC(C)(C)CCC1CC(=O)O 98947,C1(CNC(c2c(C)snn2)=O)CCN(C(c2cnn3ccn(C)c23)=O)CC1(F)F 98948,Cc1sc(C(=O)Nc2ccc(-n3ccnc3)cc2)c(C)c1Br 98949,c1(NC(=O)NC2CCCN(CCC(=O)OC)C2)ccc(F)cc1C 98950,C(C(C(=O)N1CCC(n2cncn2)C1)n1cc(-c2csc(OC)c2)nn1)OCC 98951,CC(C(=O)NCc1cccc(COC2CCOCC2)c1)C(C)(C)C 98952,C(=O)(CCCCNC(C)C)N(CC(=O)OCC)CC(c1ccccc1)C 98953,C1(C)(CNC(CCSC)=O)CC(NC(C2CSCC2c2ccccc2)=O)C1 98954,C1(NC(=O)C(O)C2CCCC2)CCC2CN(C(c3cc4c(s3)CCC4)=O)CC2C1 98955,C1(CCC#C)CCCN(C(=O)CCC(C)NC(=O)C(C)C(C)C)C1 98956,Cc1c(C(=O)NCCCCNC(c2csc(C)c2C)=O)cc(F)cc1Br 98957,N1(C(C(C)OCC=C)=O)CC(NC(c2nc(O)c(C)s2)=O)C(n2ccnn2)C1 98958,C1(COC)CCCC1NC(=O)CC1(C)CCN1C(C)=O 98959,CCC(CC)(CC)C(=O)NC(CC1CC1)CC(=O)NCC1(F)CC1 98960,c1(-c2onc(CN(C(=O)OC(C)(C)C)CC)n2)cc(CO)cc(C)c1 98961,C1(CNC(c2c(C(C)C)csc2)=O)CCCCN(C(=O)COc2ccsn2)C1 98962,C(C(C)CC(C)C)NC(c1n(CCCSCC)nnn1)c1ncnn1C 98963,N1(c2cc(NCC3(CO)CC=CC3)nc(C)n2)CCC(C)C2(CCC2)C1 98964,C1(C)(CNC(c2[nH]cc(C)c2)=O)CN(C(=O)CCNc2ccccn2)CCO1 98965,C1(NC(c2c(C)n(C)nc2)=O)CC12CCN(C(C1CC3CCC3C1)=O)CC2 98966,n1(CC)nc(C)c(C(=O)N(C)CC2(NC(=O)C(C)S(C)(=O)=O)CC2)c1C 98967,C1(C)(C(=O)Nc2c(CC)noc2)CCCN1C(=O)CCCn1ccnn1 98968,c1(OC)cc(C(=O)NC2CCCC2CNC(C2(CC)CCCC2O)=O)cnc1C 98969,C1(CNC(c2cc(OC)no2)=O)N(C(=O)Cc2cc(C)cc(F)c2)CCC1(C)C 98970,N1(C(C(C=C)O)=O)CC(F)CC1CC(=O)NCc1cncc(F)c1 98971,c1(OC)ncccc1C(=O)NCC(C)(C1CC1)NC(c1ccoc1Cl)=O 98972,CCCCCC(O)CC(=O)NCCN(C(=O)CC(C)C)Cc1ccccc1 98973,c1(CC(=O)NCCCCOCCCC#C)coc2cc(F)ccc12 98974,C12(CO)COCC(Nc3ncc(Br)cc3C(F)(F)F)(C1)C2 98975,C(=O)(C(C(C)C)n1ccnc1)NC1(C)CC(NC(C2(CC)CCCC2)=O)C1 98976,c1(CNC(C(CC)n2ccnc2)=O)cnn2c1CN(c1nnc(C3CC3)o1)CC2 98977,Cc1ccc(NC(=O)C(=O)NCC(C)CNC(=O)CSC(F)F)cc1 98978,C1(NC(CCC#CC)=O)CN(C(C2CSCCS2)=O)CC1(C)C 98979,N1(C(C)C)CCCC(CN2CCCC2c2cc(Br)cs2)C1 98980,S(=O)(=O)(c1c(C)noc1C)NCC(=O)NC1CN(C(CCCC=C)=O)C1 98981,c1(NC(C2CC3(CCN(C(=O)CCC4CC4)CC3)C2)=O)cc2c(Cl)cccc2s1 98982,c1(C(=O)NCC2C(NC(CCC#CC)=O)COC2)ccc(Cl)c2c1OCCO2 98983,N1(C(=O)C2=CCCCC2)CC2OCCN(C(C3CC3C3CC3)=O)C2C1 98984,N1(C(CCC=C(C)C)=O)CC(N=[N+]=[N-])CC1C(=O)NCCN1CC=CCC1 98985,C(=O)(CCC1=NNC(=O)CC1)NC1CN(C(CN(CCC)C)=O)C2(C1)CCOC2 98986,CC(C)(C)C(O)C(=O)NC1CN(C(C23CCC(C2)C3)=O)CC12CC2 98987,N1(C(C(=O)NC(C(=O)NCC(=C)C)C2CC2)C)CCOCC1 98988,C1(CC#C)(C(=O)N(CC(C)CNC(C2(COC)CCOCC2)=O)C)CCCOC1 98989,N1(C(Cc2cc(C)[nH]n2)=O)CCC2CN(C(C34CCC(=O)N3CCS4)=O)CC2C1 98990,C(=O)(CCCCSC)NC(C1CN(C(c2ccc(COC)o2)=O)C1)C 98991,c1(C(=O)OC(C2CCOCC2)C(=O)OC)cccc(S(F)(F)(F)(F)F)c1 98992,CCCC(CCC)=CC(=O)NC(CN(C(=O)C(C)(C)n1cnnn1)C)CC 98993,CC(=O)C(C)CC(C)C(=O)NC1CCC(CNC(C2(F)CCCCC2)=O)CC1 98994,C1(NC(C(CCSC)NC(C)=O)=O)C2CCC1N(C(c1ccsn1)=O)C2 98995,O=C(CC(CC1CC1)NC(c1nc[nH]n1)=O)NCc1conc1C1CC1 98996,N1(C(CC(C)(C)F)=O)CCN(C(=O)C=Cc2nccs2)CC1CO 98997,C1(NC(C2N(C)CC(F)C2)=O)CCC12CCCN(C(C1COCCN1C=O)=O)C2 98998,c1(CC(C(N2CC(c3cn(CC(COC)O)nn3)(F)C2)=O)OC)ccc(C)cc1 98999,C1(NCc2cnc(C(=O)OC)s2)CC(=O)N(OCc2ccccc2)C1 99000,N1(C(C(C)NC(C)(C)C)=O)CC2CC(NC(c3coc(C(F)F)c3)=O)C1C2 99001,c1(N2CCC(SC(F)(F)F)C2)[nH]c(=NCc2cn(C3CC3)nn2)nc2sccc12 99002,C1(CC(N)=O)CN(CC(c2ccc(-c3ccccc3)cc2)O)CCO1 99003,C1(C)(C(N2CCC(C(C)NC(C(F)(F)C3(OC)CCC3)=O)C2)=O)CNC(=O)C1 99004,C(=O)(CCC(=O)C1CC1)N1CC(C(=O)NCc2cc(CC)c(C)o2)(CC)C1 99005,C(=O)(C(C)(C)CC#N)NCC1(C(C)(C)O)CN(C(CSCCC)=O)C1 99006,c12cc(c(Cl)cc1F)NC(=O)C2N(C)Cc1ccon1.C1CS1.CCOC 99007,C1(F)(CNC(c2n(CC)nnc2)=O)COCCN(C(=O)CS(=O)(=O)NC)C1 99008,C=C(C)CCNC(=O)COCCNC(C1CC1(C)C)=O 99009,C(=O)(CC(C)c1cccnc1)NCC1(NC(C(C)C)=O)CCC1 99010,c1(SC)nc(=O)c(NC(=O)NCC2CC2NC(=O)OC(C)(C)C)c[nH]1 99011,C1(CNC(c2cc(C)n(C)n2)=O)(CO)CCCN(C(C2CCN(C)C(C)C2)=O)C1 99012,N1(CCNC(C2OCCN(CC)C2)=O)CCCN(C(=O)CC2(N(C)C)CCC2)CC1 99013,C1(NC(CCC=C)=O)COC2(CCN(C(=O)Cc3cn4c(C)csc4n3)C2)C1 99014,N1(C(C2(OC)CCSCC2)=O)CC2CC1CN2Cc1nc(C)cs1 99015,C(=O)(C1=CC2C=CC(C1)C2)N1CCC(NC(C2(CC)CC2)=O)C(C)C1 99016,c1(Cn2ncc(C)c2)ccc(NC(=O)NCC2CCC(CC(C)(C)C)C2)cc1 99017,N1(C(CCc2c(C)n(C)nc2)=O)CCCC(C)(NC(c2ccn(C)n2)=O)C1 99018,c1(CC)cnn2ccc(C(N3CCC(C)N(C(=O)C(CO)C(C)C)CC3)=O)nc12 99019,c1(CC(=O)NC2CN(C(=O)C3=CCCS3)CCC2CO)cccc2ccccc12 99020,N1(C(C(C)OCC(C)C)=O)CCCC(NC(c2cc(C3(C)CC3)n[nH]2)=O)C1C 99021,C1(C(N2C(C)CC2)=O)CCCC(NC(=O)COCC2CC2)C1 99022,C1(C2(O)CCC2)(CNC(CC2N(C(C=Cc3ccc(C)o3)=O)CCCC2)=O)CC1 99023,CC1=NS(=O)(=O)N(C)C=C1C(=O)N1CCOc2cc(CN)ccc21 99024,N1(C(c2c(CCC)nco2)=O)CC2CC(NC(c3occc3CN(C)C)=O)C2C1 99025,C(=O)(C(O)CC(F)(F)F)N(CCOC)CCNC(C1(N(C)C)CCC1)=O 99026,c1(OC)ccc(CCCNC(c2cccc(C3(C(F)(F)F)CC3)c2)=O)cc1 99027,Cc1nn(C)c(=O)c(C(N2C3CCC2CC(NC(c2cnccn2)=O)C3)=O)c1C 99028,c1(C(N2CC(CNC(C3C(C(N)=O)C3)=O)C(O)C2)=O)cn2c(n1)CCC2 99029,N1(C(C)=O)CCC2(CCCN(Cc3cc([N+](=O)[O-])ccc3O)C2)CC1 99030,S(=O)(=O)(c1ccccc1CNCCCOC(F)F)NCCOC 99031,C(CCCCC(=O)N(C(C)(C(N1CC2C(C1)C2(C)C)=O)C1CC1)C)SC 99032,C=CCCCCCC(=O)NCC=CCNC(C1CNC(=O)N1C)=O 99033,CC1CCCC(C)N1CC(=O)NC1CN(C(=O)CCc2ccn(C)c2)C1 99034,C1(C(N2CC(NC(c3c(C)cc(F)cn3)=O)CC2(C)C)=O)CC2(CCC2)CCO1 99035,C1(C(=O)NC2(C)CN(C(c3ccnn3C(C)(C)C)=O)C2)CCC2C1C2(F)F 99036,c1(C2C(NC(=O)NC(c3ccc(-n4ccnc4)cc3)C)C2)ccccc1Br 99037,C1(C(=O)NCC2(CCNC(C(CN(C)C)N(C)C)=O)CC2)CC(=O)N(O)C1 99038,C=CC(C)(C)CC(=O)NCCC1(C(=O)NC(C(C)(C)O)C2CC2)CCCC1 99039,C=CC(CCC)CC(=O)NC1CN(C(=O)Cn2nc(C)c(C)c2C)CC(F)(F)C1 99040,C(=O)(CS(=O)(=O)C1CC1)N1CCN(C(CNC(c2ncc(OC)nc2)=O)C)CC1 99041,C(=O)(CCCC(=O)OC)N1C(CC=C)(C(=O)Nc2cn(C)nc2O)CCC1 99042,C1(C(N(CCC(C)NC(C2N(CC)CCCC2)=O)C)=O)CCC2(CCCC2)CC1 99043,N1(C(C=C(CCN(C)C)Cl)=O)CC(CNC(c2ccnc(C)c2)=O)N2CCC1C2 99044,c1(CC)cc(C(=O)NCCC2CCN(C(=O)CCC3(C)CC3)C2)c(C)o1 99045,N1(C(CSC(C)C)=O)CCCC2(CNC(=O)Cc3ccns3)CCCC12 99046,n1(CCC)nc(CO)nc1-c1ccn(-c2ccc(C(F)(F)F)cc2)n1 99047,c1(NC(=O)CC2CN(Cc3ccc(Cl)cc3O)CCO2)cc(Br)cc(I)c1 99048,c1(OC)ccc(C(C)C(N2CCCC2C(C)NC(=O)CC2(CO)CC2)=O)cc1F 99049,c1(C(N2CC3CC(NC(C4(COC)CC4)=O)C3C2)=O)ccc2ncnn2c1 99050,c1(C(N(C(CCNC(CCCOC)=O)C)C)=O)sc(Cc2ccccc2)nc1C 99051,c1(CCCC(=O)NCC(O)CNC(c2ccccn2)=O)ccccc1F 99052,C(=O)(C(CC(C)C)OC)NCC(CCCC)NC(C1CCS(=O)(=O)N1)=O 99053,C(=O)(C(C)(C)CCCF)NCCNC(C1CCC(CN(C)C)O1)=O 99054,C(=O)(C1CC(=O)Nc2ncccc21)N(CCCNC(=O)C1CCc2nccn21)C 99055,C(CC(C(C)C)NC(c1cncc(O)c1)=O)NC(C1(c2c(C)cno2)CC1)=O 99056,C(=O)(CCC(C)(C)F)NCC(CC)NC(c1ccc(F)cc1)=O 99057,C1(NC(c2ccn(C3CC3(F)F)n2)=O)CN(C(=O)COC2CC2)CC12CCC2 99058,C1(C#N)(C(=O)NCC(=O)NCC2(CO)C(C=C)C2)CC(=O)C1 99059,c1(-c2ccc3occ(C(=O)NC(COC)C)c3c2)c(F)c(F)c(N)c(F)c1F 99060,c1(C(=O)OC(C)(C)C)ccccc1S(=O)(=O)NCc1ccc(N2CCCC2)cn1 99061,C1(NC(=O)NCC2CC2)(CNC(c2cc(CO)on2)=O)CCCS(=O)(=O)C1 99062,c1(C(=O)NCC(C)N(C(COCCC=C)=O)C)nnn(CC)c1C(F)(F)F 99063,CC1CC(=O)NCC1C(=O)NC1(C2CCCN2C(c2cc(O)cs2)=O)CC1 99064,c1(N(C(C(C)C2CC2)C(=O)OC(C)(C)C(F)F)C)ccc2c(c1)CCC2 99065,N1(C(C2(C=C)CCC2)=O)CCC2CC2(C(=O)Nc2cncnc2O)CC1 99066,C1(C(=O)OCC)CNC(=O)CC12CCN(CCc1ccc(OC)c(OC)c1)CC2 99067,c1(C(C(=O)NCC(CCOC)NC(=O)CCc2cnc[nH]2)(F)F)ccc(Cl)nc1 99068,C1(NC(C2CC23CC3)=O)C2CC(O)C1N(C(c1ccccc1-c1cc[nH]n1)=O)C2 99069,c1(C(=O)NC(C(C)C)CNC(=O)CCC2CCCN2C)cnc(N)c(Cl)c1 99070,C1(CNC(CN(C(C(C=C)OC)=O)CCOC)=O)CCCC12CCC2 99071,C(=O)(C(CCCC)NC(c1ncc(F)cn1)=O)NC(C=C)C 99072,N1(c2n(Cc3cc(C)oc3C)nnn2)CC2COCC2C1 99073,C1(CN(C(CC(C)c2ccccc2)=O)C)CCCN(C(C2(F)CC2)=O)C1 99074,C12(C(=O)NC(c3ccc(C)cc3)CNC(CC(=C=C)C)=O)CCC(C1)C2(C)C 99075,C1(CC(=O)NC2CC(NCc3ccc(C(=O)OC)o3)C2)C(=O)NN=C1C 99076,c1(C(N(CC(C)N(C(c2ccc(C)nc2)=O)C)C)=O)n[nH]c2c1CCOC2 99077,Cc1cnccc1C=CC(=O)NC1CCCC(NC(c2c(C)nn(C)c2Cl)=O)C1 99078,Cc1oc(Br)cc1C(=O)NC1CC2(C1)CC2NC(=O)CN1CCCNC1=O 99079,N1(C(c2ccc(CC)cn2)=O)CC(CNC(=O)CCCc2cccs2)CC1(C)C 99080,CC1C(CN(C2CCCC2)C(=O)NC(=O)CCC2CCCN2)CCCN1C 99081,C(c1c(Cl)nc2sccn12)=CC(=O)NC1C2CCN(C(=O)C(O)CC(F)(F)F)C12 99082,C(C)(CN=c1[nH]c(Cl)ncc1C(F)(F)F)NC(c1c(C(C)C)ocn1)=O 99083,c1(C(=O)NCC2N(C(C(C(C)C)O)=O)CCN(C)C2)cccc2c1COCC2 99084,C1(CNC(c2ccsc2)=O)CCC(NC(c2[nH]nnc2C2CC2)=O)C1 99085,C(CNC(=O)CSc1nnnn1C)(CC(F)(F)F)NC(C(C)CSC(F)(F)F)=O 99086,c1(C(C)NC(c2n(CCCSC)nnn2)c2cscc2C)ccncc1Cl 99087,CC1CCN(C(C2(CO)COC2)=O)CC1NC(=O)CC(F)(F)Br 99088,c1(OC)ccc(C)c(C(=O)N(C2CCN(C(=O)CCC(C)SC)C2)C)c1 99089,c1(NC(CCCCNC(COCC=C)=O)=O)ccc(F)cc1OC 99090,C1(CCC(=O)NCC(N(C(C(C)SCC)=O)C)C2CC2)(N(C)C)CCCCC1 99091,c1(C(N2CCC(C(C)(C)NC(CC3N(CC)CCC3)=O)C2)=O)ccc(CO)cn1 99092,c1(C(C)C)ccc(C=CC(=O)NC2COCCN(C(=O)CCC3CC3)C2)cc1 99093,c1(CC(=O)N(C)CC2N(C(C(C)SC)=O)CCOC2)coc2ccc(F)cc12 99094,CN1CC(O)CC1C(=O)NC1CC(C(N2CC(n3cnnn3)C2)=O)C1 99095,C1(N(C(C=CCCC)=O)C)CCN(C(c2cc(Cl)ncc2OC)=O)CC1C 99096,CC1(C)CC(CC(=O)NC2(C3CCCN3C(C3CC=CCO3)=O)CC2)CCO1 99097,C1(NC(C2(SC)CN(C(C(CCC)CC)=O)C2)=O)CC(C)(C)OC1(C)C 99098,CC(C)(O)C(C(=O)N1CCC1)N(C1CCCC1)C(c1cnn(C2CC2)c1)=O 99099,C(C(C)CC(=O)NCC1(C(N)=O)CN(C(=O)Cn2cnc(C(N)=O)n2)C1)OC 99100,N1(C(CC=CC=C)=O)CC(C2CC2)(C(=O)Nc2ccc(F)c(CO)c2)C1 99101,C=C(C)CC(C(=O)N1CC(OC(=O)NC)C1)NC(c1cn(CC)cn1)=O 99102,N1(C(C(C)OCC(C)C)=O)CC(NC(c2coc(Cl)n2)=O)CC12CCCCC2 99103,C1(OC)(CNC(C2CC3CC3C2)=O)CCN(C(=O)CCc2ccc(O)cc2)CC1 99104,C(=O)(CCCNC(C1CC(CNC(C2CCCN2C(C)=O)=O)C1)=O)NC 99105,c1(COC)ccc(C(=O)NC23CC(NC(=O)CC(=O)Nc4nccs4)(C2)C3)o1 99106,N1(C(C2CCC3CC23)=O)CCOC2(CCCN(C(c3ocnc3C(F)F)=O)C2)C1 99107,c1(C(=O)NC2C3CN(C(CCC(C)SC)=O)C2C3)ncc(Cl)cc1F 99108,C12(CC(=O)N(CCCCN(C)C(C3C4CCC(=O)C34)=O)C)CCCCC1C2(F)F 99109,Cc1n[nH]c(C)c1C(=O)NCC(C)CNC(=O)C(C)Oc1ccc(CO)cc1 99110,C(=O)(CC(O)CC(C)(C)C)N(C(C)CNC(c1ccc(C(C)(C)C)[nH]1)=O)C 99111,c1(C(N(C(C)C)CCNC(C2CCCCO2)=O)=O)c(Cl)c([N+](=O)[O-])nn1C 99112,C12(C(=O)OC)CCC(C(N3CCCCC(CNC(=O)CSC)CC3)=O)(CC1)CC2 99113,N1(C(c2nn(CC)c(C)c2)=O)CCC(N(C)C(c2cc(OC)nn2C)=O)C(C)C1 99114,N1(C(c2cccc(SC)c2)=O)CCN(CC(c2ccccc2)C2CCNC2)CC1C 99115,C1(C(=O)NCC2CNC3CC23)CSC(c2ccccc2O)=N1 99116,N1(C(C=COCC)=O)CCC2(CCCC2NC(=O)CCc2cccc(C#N)c2)C1 99117,Cc1ccc2c(C(=O)NCC3(F)CC(NC(C4(C)CC4)=O)C3)cnn2c1C 99118,c1(C(N(CCCNC(=O)CC(C)C)CC)=O)ccc2oc(N(C)C)nc2c1 99119,c1(C(=O)NCC(CNC(C2CCC(=O)N2)=O)CO)c[nH]c(=O)c2ccncc12 99120,c1(NC(N2CCC(N(C)CC)C2)=O)ccnc(S(C)(=O)=O)c1 99121,C1(NC(COCCCN(C)C)=O)CN(C(c2cc(F)cs2)=O)CC1F 99122,c1(OC(C)C(N2CCCC2CCNC(C2(c3ncco3)CC2)=O)=O)ccccc1 99123,c1(C(=O)NC)ccc(C(=O)N(CC(O)CNC(=O)C(F)n2ccnc2)C)cc1F 99124,c1(C(N(C2CN(C(c3nn(CC)c(C)c3)=O)C2)C)=O)cc(Br)ccc1O 99125,c1(CC)cnc(C(=O)NCC2CC2NC(c2cccnc2C)=O)cn1 99126,c1(C(C)C)ncc(C(=O)NCC2CC2CNC(=O)COCc2nccn2C)s1 99127,N1(CC(N2CC(NC(C(C)NS(C)(=O)=O)=O)(C)C2)=O)CCC(F)CC1.C1CC1 99128,c1(C(N(Cc2cn(CCOC)nn2)O)=O)cccc2scnc12 99129,N1(C(C2(CC#C)CCC2)=O)CCCC(N(C(=O)CC2CCCS(=O)(=O)C2)C)CC1 99130,N1(C(Cc2c(C)ccnc2)=O)CC(F)(F)CC1CCNC(C1CCCOC1C)=O 99131,c1(C(=O)NCC2(F)CCN(C(C(=CC3CCCC3)C)=O)C2)cccn2cncc12 99132,c1(C(=O)N(C2(CCNC(=O)C(c3ccccc3)F)CC2)CCO)cnc2sccn12 99133,C1(F)(C(=O)Nc2nccnc2Br)CCN(C(c2occc2Br)=O)CC1 99134,N1(C(C(F)OC)=O)CC(O)(CCNC(c2ccncn2)=O)C1 99135,C1(C(=O)NCCCN(C)C(C2C(Cl)(Cl)C23CC3)=O)CCc2ccccc2C1 99136,N1(C(=O)Nc2c(CC)ccc(C(F)(F)F)c2)Cc2ccccc2SCC1C 99137,c1(NC(CC(C)F)C)nc2ccccc2nc1NCCN1CCCOCC1 99138,N1(C(c2c(C)n(C)cc2)=O)CCN(C(C2(C)CC(F)C2)=O)C2(CCC2)C1 99139,C(=O)(CC1CCc2ccccc21)NCCN(C(C=CSC)=O)C1CCCCC1 99140,N1(CC)CC2CC(F)(C2)C1.c12noc(n1)CNC(=O)OC2=O 99141,c1(N2CCC(O)(NCCNC(CC)=O)CC2)nc(C(F)(F)F)nc(C)c1Br 99142,C1(C(=O)NCc2cnc(C)s2)CN(C(c2ncn(C(C)C)n2)=O)CCN1 99143,C1(NCCN(CCC2(c3ccccc3)C(C)C2)CC2CC2)CCc2nn[nH]c2C1 99144,C(=O)(CCC(C)(F)F)N1C(C(C)(C)NC(C(C)N(C)C)=O)CCC1 99145,N1(C(c2cncc(N)c2)=O)CCCC(C2(NC(c3ccsc3)=O)CC2)C1 99146,C1(CN2CCC(NC(C3CCC3)=O)CC2)CCC12CCNCC2 99147,c1(C(=O)NCC2(OC)CN(C(C(CC)O)=O)C2)nc2n(c1C(C)C)CCCC2 99148,C(=O)(CCCCN)NCC1(C)CSC1.C12(CC(=O)N)CCCC1C2 99149,C(CCCCC(=O)NCC1CCN1C(c1ncccc1O)=O)=CC 99150,Cc1ccc(F)c(C(=O)NC2CCC(N(C)C(c3cccnc3)=O)CC2)n1 99151,C(=O)(CCCCC1CC1)N(C1(CC(=O)N(C)Cc2cc[nH]n2)CC1)C 99152,c1(C(N2CC3C(CNC(CCCC#N)=O)C3C2)=O)cc2ccccn2n1 99153,S(=O)(=O)(c1cc(C)ccc1C)N1CCC(NC(c2c(OC)nn(C)c2)=O)C(F)C1 99154,N1(C(c2cnc3cn(C)nc3c2)=O)CCS(=O)(=O)Cc2ccccc21 99155,C=CCS(=O)(=O)C(N1CC(CNC(C2CCN(C(=O)OC(C)(C)C)C2)C)C1)=O 99156,C(=O)(CCC(C)(C)C)N1CCC(C2N(C(CCc3c(C)ccs3)=O)CCC2)C1 99157,c1(OC(N2CC(F)(F)C2)=O)c(Br)cncc1Br.C12CCCCN1C2=O 99158,N1(C(C2N(C)CCC2)=O)Cc2ccccc2C1CNC(C1CCCO1)=O 99159,c1(C(=O)NC2CC3(C(C(=O)NC4(C(C)O)CC4)C3)C2)cc(C#N)cn1C 99160,CC1C(NC(=O)C(F)(F)C2CC2)CC2CCC1N2C(c1cc(Br)c[nH]1)=O 99161,Cc1ccc(OCC(N2CCC(C(C)NC(=O)CSCC(C)C)C2)=O)cc1 99162,CCC(C)(CO)C(=O)N1CC(C(=O)NCc2oc(C)nc2C)C(F)C1 99163,Cc1[nH]nc(Cl)c1C(=O)NC(C)CN(C(=O)C(c1cnn(C)c1)C)C 99164,CN1CCCC1CC(=O)NC1CC(NC(C2(C(=O)NC(C)(C)C)CCCC2)=O)C1 99165,C(=O)(CCCC(C)(C)CC)N1CCC(C(F)F)(CNC(C2CCN(CC)C2)=O)C1 99166,N1(C(c2c(OC)ccs2)=O)CC2(CCC(CNC(=O)COC3CC=CC3)O2)C1 99167,C(=O)(C(O)CCC(C)C)NCCN(C(=O)CN1CC2CCC1C2)CCC 99168,CCC(CC(=O)NC1(CCNC(=O)CCSC)CCC1)c1ccccc1 99169,c1(OC)ccc(OC)c(C(N2CCCCC2C(C)NC(=O)C=CBr)=O)n1 99170,CC1CCCN(C(c2ncccc2C2CC2)=O)C1CCNC(c1cnc(Cl)s1)=O 99171,C=CC(C(=O)NCC(CC)NC(=O)C(C)(F)c1ccon1)OC 99172,C(=O)(CC(C)C(=O)NCC1(CNC(=O)Cc2ccsn2)CCOCC1)OC 99173,c1(CNC(C)=O)ccc2c(c1)CN(C(c1cc3c(cc1O)OCO3)=O)C2 99174,c1(C(=O)NC(CC(N)=O)C(N2CCC3C(C2)C3(F)F)=O)ccn2cncc2c1 99175,C1(C(=O)NCCN(C(=O)CCc2cncnc2)CC2CC2)CC12CCOCC2 99176,Cc1ccccc1-n1ccc(C(=O)NC(C)CCNC(=O)CSC2CC2)n1 99177,c1(C(=O)NCC(CNC(C2C(C(N)=O)C2)=O)F)ccsc1Cl 99178,C1(N(C)C)CCc2nc(NC(c3cc(Cl)cc(C#C)c3NC(C)=O)=O)ncc2C1 99179,N1(c2cc(NCc3c(CC)noc3)nc(C)n2)CCn2c(cnc2Br)C1 99180,c1(C(=O)NC(CNC(C(n2ccc(C)n2)(C)C)=O)(C)C)cnc2n1CCCC2C 99181,N1(C(c2cncc(C=C)c2)=O)CC2CCC1CN2C(c1cccc(C)n1)=O 99182,N1(c2[nH]c(=NCc3nccc(C)c3)[nH]c(=N)n2)CC2CCCCCC2(C#N)C1 99183,c1(CC(N2CC(NC(CCN(CCC)C)=O)C2)=O)cc(C(F)(F)F)cc(F)c1 99184,C1(CC)CN(C(=O)CCc2ccncn2)CCC1NC(=O)C=C(C)c1cccs1 99185,N1(C(c2n(C)ncn2)=O)CCCC2(NC(c3cccc4cnnn34)=O)CCCC12 99186,c1(C2(C(=O)Nc3c(SCC#N)cccc3)CCC2)c(F)cccc1F 99187,CCCC(C)(O)CC(=O)NCCOCCOCCNC(C1CCN(OC)CC1)=O 99188,N1(C(C2CCN(C(Cc3cn(C)nc3)=O)C23CCC3)=O)CCC2(CCOC2=O)C1 99189,c1(C(=O)NC(c2nc[nH]n2)C)conc1CNC(=O)CCc1cncn1C 99190,[N-]=[N+]=NC1CC(C(=O)NCC2CCSC2)N(C(c2cnn3ccccc23)=O)C1 99191,C(c1ccc(C)cc1C)=CC(=O)NCC1CC(NC(C2CN(CC)C(=O)C2)=O)C1 99192,c1(NC(=O)NC(c2cccs2)C)c(Br)nnn1C 99193,C(CC(C(=O)NCC1CCN(C(c2ncc(F)cn2)=O)CC1)N(C)C)SC 99194,c1(OCC)cncc(C(=O)N(C(C)CCNC(c2c[nH]cc2Br)=O)C)c1 99195,Cc1cc(NC(=O)C(=O)N(CC(C)C)Cc2ccc(Br)s2)cc(N2CCCC2)c1 99196,N1(C(c2n(C)nnc2)=O)CCCC(C(=O)NC2(C(C)(F)F)CC2)C1 99197,N#Cc1ccc(CN2CC(CNC(c3coc(Cl)n3)=O)C2)nc1 99198,C1(NC(C(CC)F)=O)CC2CCC1N2C(=O)COCC1CCCC1 99199,c1(C(=O)NC2(CO)CCCN(C(C=CC(C)(C)SC)=O)C2)cccc2[nH]ncc12 99200,C1(CNC(CCCOCCC)=O)CN(C(C2CC(C)=NO2)=O)C2(CCOCC2)C1 99201,c1(C(N2CC3C(CN(C(C4(SC)CCC4)=O)C)C3C2)=O)cc(C)c(CO)cn1 99202,n1(CC)nc(C(=O)NCCn2ccc(C(=O)NC3CCC(C)(C)C3)c2)cc1C 99203,CC1(N2CCC2)CCN(C(C(=O)Nc2cccc(-c3cccs3)n2)C2CCOC2)C1 99204,CCCC(C)C(C(=O)NCC)N1CCCC(C)(C(=O)OC)C1 99205,C(=O)(CCC(C)CCN(C(=O)CCc1ccc[nH]1)CC)OCC 99206,CCCC(CNC(C1C(C)C1C)=O)C(=O)NCCC(C)(C)CO 99207,C12CCCCCN1C2=O.c1(COC)c(-c2cn(C(C)C(=O)OC)nn2)cnn1C 99208,N1(C(C(COC)O)=O)CC2(CCCC(CNC(=O)CCNC(=O)C(C)(C)C)O2)C1 99209,C1(OC)CCC(C(=O)NCCCCNC(C2CC(n3ccnn3)C2)=O)C1 99210,c1(CC(N2CC(NC(C(C)N3CCC3)=O)(CO)C2)=O)ccnc(Br)c1 99211,C1(C(=O)NC2CCC(O)C2)CCCC2CN(C(C3(F)CCCC=C3F)=O)CC12 99212,N1(C(C(C2(O)CN(C(c3cnccn3)=O)C2)F)=O)CC(F)C(F)C1.C1(=O)CN1C 99213,N1(C(C2C(=O)NCCC2)=O)CCC(C(=O)NC2CCC3(CCC3)C2)C(O)C1 99214,C1(S(C)(=O)=O)(C(N(C2CCCC(NC(c3ncccc3F)=O)C2)C)=O)CCC1 99215,C1(C(=O)N(C)CCNC(C)(C)C)(NC(=O)NC)CCOC1.c12cocc1NC2=O 99216,Cc1ccc(CN2CCC(C(=O)NC3(C)CCCCC3)CC2)c(Br)c1 99217,C(=O)(CC(C)(C)N(C)C(c1ccn(CO)c1C)=O)NCC1(COC)CCC1 99218,c1(NC)cnncc1C(=O)NCCN(C(=O)CC1CCCCN1C)C1CC1 99219,N1(C(=O)Cc2cnn(C(F)F)c2)CCC(CNC(C2(Br)CCCC2)=O)CC1 99220,c1(OC)cc(O)ncc1C(N1CCCCC(NC(=O)CC(C)C)C1)=O 99221,N1(C(C=CCCC)=O)CC(OC)CC1CCNC(=O)C(Cc1ccsc1)NC=O 99222,c1(C(N2CC(C(=O)NCC)OCC2)=O)cnc2ccccc2c1.C1(=O)C(CO)O1 99223,N1(CCCC)CCCC(CNC(C2COCCC2CN(C)C)=O)C1 99224,Cc1nnc2n1CC(C(=O)NC1CC(NC(=O)CN=S(C)(C)=O)C1)CC2 99225,Cc1csc2c(CNC(=O)NCc3ccc(C#N)cn3)cccc12 99226,CN1CCOC(C(=O)NCC(C(=O)NCCC2CCN(C)C2)N(C)C)C1 99227,C(C(=O)N1CC(C(C)NC(=O)CC2(C)CC2)C1)(C(C)C)OCC 99228,CCCCC(O)CC(=O)N1CC(CC(F)C(=O)NCCC(O)CC)C1 99229,C12CCN(C(C)C1)CCCn1cc2nn1.c1(OCC)ccc(-n2cnnn2)cc1 99230,CCC(C)C(C(=O)N1C(CO)CC1CO)N(C)C(c1cc(OC)ncn1)=O 99231,C(=O)(C(F)C(C)(C)O)N1C(C(N(CC#C)CC2CCCO2)=O)C2CC2C1 99232,C1(NC(c2ccc(C(=O)OC)cc2)=O)CCN(C(c2cc(F)n[nH]2)=O)CC1C 99233,c1(CCC(=O)NC2CCCN(C(C3CC3(F)F)=O)CC2)cncc2ccccc12 99234,C(=O)(C#CC(C)(C)C(F)F)N1CC(OCCNC(Cc2cccc(CC)c2)=O)C1 99235,C1(NC(C(C)NS(C)(=O)=O)=O)COCCN(C(=O)CCc2cnc(C3CC3)o2)C1 99236,c1(C(=O)NCC(C)(O)CNC(C2CC23CCCCCC3)=O)cc(O)c(F)cc1N 99237,C12(CCCCC1)C(=O)N2.C(CCC(=O)NC(c1ccnn1C)CO)OC 99238,c1(OC)ccc2c(C(=O)N(C)CCNC(c3ccn(CCF)n3)=O)ccnc2c1 99239,c1(C(=O)NCC(Cc2cccc(C)c2)CO)ccc2c(c1)CCC(=O)N2C 99240,c1(CNC(COC(CNC(C2(OC)CC2)=O)(C)C)=O)ccc(C)nn1 99241,C(=O)(C(C)C(CC)CC)NC(CC#C)(C)C(=O)NC1(C=C)CCCCC1 99242,c1(C(N2CCC3(NC(C=COCC)=O)C(C2)C3)=O)cc(C)c(Cl)cc1F 99243,c1(C(=O)NCCOC2CCN(C(=O)CCCF)CC2)cnc2n1CCCC2.CCO 99244,c1(C(C)(C(=O)N2CC(OC)C2)OC)cccc(C(=O)N(C)C)c1.C(=O)(CCCCO)N 99245,C1(NC(c2c(C)ccnn2)=O)CC2(C1)CN(C(c1cnc(C(F)F)s1)=O)C2 99246,CC(C)(CC(F)(F)F)C(=O)N1CC(NC(c2ncccc2Cl)=O)CC(F)(F)C1 99247,c1(N(C)CC)ccc(-c2nc(CC3CC4CC4C3)n(CCCCO)n2)cc1 99248,C1(C(=O)NCCn2c(C)nnc2)CCN(C(=O)CC2CCOCC2)CCO1 99249,C1(OC)CCC12CC(C(=O)N(C1CN(C(=O)Cc3ccnn3C)CC13CC3)C)C2 99250,C1(NC(=O)C=CCO)CCN(C(=O)C2=COCCO2)CCC1(F)F 99251,N1(C(Cc2nnc(C)s2)=O)CCC(C)(CNC(c2sccc2SC(F)F)=O)C1 99252,N1(C(C(C)N2CCC2)=O)CCC(O)C(NC(C2(CO)CCCO2)=O)C1 99253,C1(C)(CNC(CC2CC(NC(c3ccc(C)o3)=O)C2)=O)CCCOC1 99254,C(=O)(C(O)CC[S+](C)C)NC1C2CN(C(CN(c3ncccn3)C)=O)C1C2 99255,Cc1cc(F)c(NC(C2CC(NC(=O)CCCCCl)C2)=O)cc1F 99256,c1(CNC(C=CC(C)(C)NC(CN(CC(C)(C)C)C)=O)=O)cncc(C#N)c1 99257,Cc1cc(C(=O)NCC2CN(C(C3CN(S(N)(=O)=O)C3)=O)CC2(C)C)ccc1Cl 99258,C1(OC)CCC12CC(C(=O)NC1CN(C(=O)C(F)(F)c3nccs3)CC1(C)C)C2 99259,N1(C(C=C(CC)CC)=O)CCCCC1C1(NC(c2ccc(COC)cc2)=O)CC1 99260,C(CCC(C)(C)C(=O)N1CC2CCCC2C1)NC(CC1CCCC(C)C1)=O 99261,c1(OC)ncccc1C(=O)N(C)CC1(NC(C2CCOC2C)=O)CC1 99262,C1(O)(C(CNC(CC(=O)NCC#C)=O)C)CCN(C(=O)C(C=C)CC)C1 99263,Cc1ncc(C(=O)NCCCCN(CCCNC(=O)CCn2ccnn2)C)n1C 99264,c1(C(=O)NC2CCCC(C(=O)Nc3cc(C(C)C)no3)C2)ccc(O)cc1Cl 99265,C1(C(=O)NC2(CO)CN(C(C=C(C)CN3CCCC3)=O)C2)CCn2ccnc2C1 99266,c1(Cc2ccc(C)c(F)c2)nc(=NC(=O)N(CC(C)C)CCO)[nH]s1 99267,N1(C(CSCCN(C)C)=O)CC2(CNC(=O)CC3CNC(=O)C3)CCC1CC2 99268,c1(C(=O)NC2(CNC(c3ccc(COC(C)C)cc3)=O)CC2)cc(F)cc(F)c1 99269,Cc1nnc2n1CC(C(N1CCC(C)(CNC(c3cc(F)ccc3O)=O)C1)=O)C2 99270,N1(C(C2(CC)CCCCC2)=O)CCC2(C1)CN(C(c1cccc(F)n1)=O)CCO2 99271,c1(C(=O)OCC(=O)Nc2c(C)ccc(C#C)c2)cc(Cl)cc([N+](=O)[O-])c1O 99272,c1(C(=O)NCCCN(C)C(C2(C(F)F)CC2)=O)cnc(Br)s1 99273,N1(C(Cc2c(SC)cccc2)=O)CC2(CCN(C(c3cnns3)=O)C2)C1 99274,CC1(C)CCC(C(N2CCCCC2CNC(=O)C(=O)NCC(F)F)=O)O1 99275,C1(C(N2CCCC(N(C(c3ccn(C)c3)=O)CC)C2)=O)CCc2nnnn2CC1 99276,N1(C(C=CC(=O)OCC)=O)CCC(CCNC(C2CCC2(C)C)=O)C1 99277,C=CC(CC)C(=O)NCCn1cc(C(=O)NCC(C)(C)CC2CC2)nn1 99278,N1(C(=O)COC2CCCCCCC2)CCCC2(C1)CN(C(C1C3CCC13)=O)C2 99279,O=S(=O)(c1ccc(N2CCC(C3OCCO3)CC2)c(F)c1)NC1CC=CCC1 99280,N1(C(c2c(CC)noc2C)=O)CCn2ncc(-c3ccc(CC)s3)c2C1 99281,c1(C(N2CCC(NC(c3ccc(Br)nc3)=O)C2)=O)ccc(I)c(F)c1F 99282,c1(C(=O)NCC(CNC(=O)CCCn2ccnc2)O)cnc2[nH]nc(O)c2c1 99283,CC1(NC(C2(CNC(=O)C3=COCC3)CCCO2)=O)CCC(O)CC1 99284,C1(NC(c2cn(CCNC(c3c(C#C)c[nH]n3)=O)nc2)=O)CCC(C)(C)CC1C 99285,c1(C(N(CC(CNC(c2ccc(C)n2C)=O)O)C)=O)cc(Cl)ccc1OC(C)C 99286,N(C)(S(=O)(=O)N(C)C)CCNC(CN1CCC(N(C(C(CC)CC)=O)C)C1)=O 99287,c1(C(N(CCC)CCNC(C2CC3CCC2O3)=O)=O)ccc(F)cc1Cl 99288,Cc1nc(CC(=O)NCCNC(C2(NC(=O)OC(C)(C)C)CCCO2)=O)[nH]c1C 99289,N1(C(C(C)NC(c2ccc(CC)[nH]2)=O)=O)CC(O)CC1(C)CO 99290,C(C(O)CC(F)(F)F)N(C)CC1CCC(C)(C)CO1 99291,C1(C(=O)NCc2c(C)cccc2)CC12CCN(C(c1nocc1C)=O)C2 99292,C1(NC(C2CCOC2)=O)CN(C(C2C3CCCC23)=O)CCC12CCOCC2 99293,C12(C(=O)NC3CCN(C(CSSC)=O)CC3)CCC(CO)(CC1)CC2 99294,C1(F)(C(=O)NC2CC(C)N(C(c3coc(C4CCC4)n3)=O)C2)C(C)(C)C1(C)C 99295,c1(C(N(C)CC2CCC(NC(CC3CC(=C)C3)=O)CC2)=O)ccc([N+](=O)[O-])cc1 99296,C1(OC)CC(CC(=O)NC2COCC2C(=O)NCc2ccccc2F)C1(C)C 99297,C1(CNC(c2ccc(OCCCOC)cc2)=O)CN(C(=O)C(C)CF)CC1(C)C 99298,C1(NC(c2c(C)ccc(C)n2)=O)CCCC12CN(C(=O)C(CCO)N(C)C)C2 99299,C1(CNC(=O)NC2CCC(C(N)=O)CC2)(CO)COCC2CCCCN12 99300,C=CCCC(C)(C)CNC(=O)C(CC1CC1)NC(=O)CC#N 99301,N1(c2cc(NC(CCOC)C)nc(C(F)(F)F)n2)CCS(=O)(=O)C(C)(C)C1 99302,CC12CC(C(=O)NC3CC(NC(C4CC45CC5)=O)C34CCC4)(CCO1)C2 99303,CC1(C#N)CCC(c2nnnn2C2(C)CC2)(NC2C=CCC2)CC1 99304,c1(C(=O)NCC2CN(C(Cn3c(C(C)C)nnn3)=O)C2)ccc2cncn2c1 99305,C(C)(CN=c1cc(C2CC2)nc(S(C)(=O)=O)[nH]1)NC(CCCCC)=O 99306,c1(OC)ncnc(OC)c1C(=O)N(C)CCNC(=O)CC1CC(C)(C)CO1 99307,C(=O)(C1c2ccccc2C2CC1C2)NC(C)C(CO)NC(c1ccc(F)cc1)=O 99308,C1(C(N(C(C)C)CC)=O)COC(CNC(=O)Cc2nonc2C)C1 99309,Cc1nn(CC(C)C)c(C)c1CC(=O)NCC1CC1NC(=O)COCC1CC1 99310,C12(NC(c3cccnc3OCCO)=O)CCCN(c3ccnc(Cl)n3)CC1C2 99311,N1(C(Cn2nc(C)oc2=O)=O)CCC2CCCC12C(=O)NC1CC(C(C)C)C1 99312,C(C1C(=O)NC2C(C2)CN1)N(C)C.c1(OCC(=O)Nc2nc[nH]n2)ccccc1 99313,C1(C(N2C(CNC(Cc3n[nH]c(=NC)s3)=O)CCC2)=O)CCc2nnc(O)n2C1 99314,C1(C(N2C3CN(C(C4CCS(=O)(=O)C4)=O)CC2CC3)=O)CCC2(CCOCC2)O1 99315,C1(C(N(c2cccc(-n3cc(CCC(=O)O)nn3)c2)C)=O)CCn2nnnc2C1 99316,CC1(C)CCC2(CC1)CC(C(N1CCC3(CCOCC3)C1)=O)C2 99317,c1(CC(=O)NCC(CNC(Cn2c(=N)[nH]nc2)=O)O)ccc(N2CCCC2)cc1 99318,C1(NC(C2Cc3nccn3C2)=O)CCCN(C(=O)CC2CCC(F)(F)CC2)CC1 99319,c1(C(=O)NCC(CCNC(c2c(OC)ccs2)=O)O)cc(Cl)cc(F)c1F 99320,C1(OC)CN(C(=O)Cc2ccc(Cl)nc2)CC1NC(=O)C(C)OCCC(C)C 99321,N#Cc1ccc2cc(CNC(N3CCc4sc(CN)nc4C3)=O)[nH]c2c1 99322,CCCCCC(O)C(=O)N1CC2(CC(C(=O)NC(CCO)C(C)C)CO2)C1 99323,N1(C(C(C(C)C)SCC)=O)C(C(=O)NCc2cn(C3CC3)nn2)C2CC(O)C1C2 99324,c1(C(C)(C)C)ncnc(N2CC3C(CNC(c4ccc(Cl)o4)=O)C3C2)n1 99325,CCCCCC(O)CC(=O)NCC(C1CC1)N(C(=O)CN(C)S(=O)(=O)N(C)C)C 99326,CC1(NC(C2CCCCC2NC(=O)C=CC2(C)COC2)=O)CC(O)(CO)C1 99327,O=C(CS(=O)(=O)C1CC1)NC1CCCC(NC(=O)CN2CCC(CO)CC2)C1 99328,c1(C(=O)NCc2cncc(C(N3CCOC(CF)C3)=O)c2)cc([N+](=O)[O-])n[nH]1 99329,CC1(C)CC(CNC(c2cc(F)c(F)cc2Cl)=O)CN(C(=O)C(F)F)C1 99330,C(=O)(C1=NOC(CNC(C2CC2(F)Cl)=O)C1)NCC1(C(C)C)CC1 99331,C1(C(=O)NC(C2CCN(C(c3cc(C)c(C)[nH]3)=O)C2)(C)C)CCCC(=O)N1C 99332,C1(CC=C)(NC(=O)CC2C=CS(=O)(=O)C2)CCN(C(=O)CCN2CCC(O)CC2)C1 99333,C12(C(=O)NC(c3ccc(Cl)cn3)C)CCC(CC1NC(c1cc(Cl)n(C)n1)=O)C2 99334,C1(C)(NC(C2OCCN(CCOCC)C2)=O)CCc2ccccc2C1 99335,C(=O)(CCCC(C)(C)NC(c1cc2ncccc2[nH]1)=O)N(CC(CCC)C)C 99336,C1(C(N2CCN(C(CC(=C=C)C)=O)CC2C)=O)CC(C(C)(C)C)=NO1 99337,c1(C(=O)NC(C)(CNC(C2COC2)=O)C2CC2)coc2cc(F)ccc12 99338,c1(CC(C(=O)NCCOCCNC(C2CC3C=CC2C3)=O)O)cc(Cl)cc(Cl)c1 99339,c1(C(=O)NCC(C2CCC2)NC(C(c2cccnc2)OC)=O)ncccn1 99340,n1(CC(N2CCC(C(CNC(C(C=C)(C)O)=O)F)CC2)=O)c(C)cc(C)nc1=O 99341,C(=O)(C1=NN(c2ccc(F)cc2)C(=O)CC1)N1CCC(NC(C2CC2(F)F)=O)C1 99342,c1(C(=O)OC)cccc(OC)c1CNC(c1cncc(-c2ccncc2C)c1)=O 99343,Cc1ncc(C(=O)N(C2CN(C(C3CC3CC(C)C)=O)CC23CC3)C)cc1N 99344,c1(CC(=O)NC2CCCN(C(C3C(CC)C3)=O)C2)ccc(C)c(O)c1 99345,N1(C(C2CN(C)C(=O)C2)=O)CCC(CNC(c2ccc(CCF)cc2)=O)C12CC2 99346,CCC(C(=O)NCC1CC(F)(F)CN1C(C1CCCC(=O)N1)=O)C(C)C 99347,N1(C(C2N(C(CC)=O)CSC2)=O)CCCC(O)(CN(C)C(c2ccoc2Cl)=O)C1 99348,N(C(=NCC(C)(O)c1cccc(Cl)c1)NC1CCCC1)Cc1ccn(CC)n1 99349,Cc1noc2nc(C(=O)NCCOC3CCN(C(C4CCSC4)=O)C3)ccc12 99350,Cc1ccc2c(=NCC3CCCCS3)[nH]c(=NCC3CC4C(C3)C4(F)F)[nH]c2c1 99351,c1(CCNC(C(C2CCCC2)NC)=O)cc(OC)ccc1Br 99352,C=CC1(C(N2CC(NC(=O)CP(C)(C)=O)C(C)C2)=O)CCCCC1 99353,N1(C(CNC(C=CC)=O)=O)CCN(C(C2(OC)CC(C)(C)C2)=O)CC1 99354,C=CCC1C(=O)N1.C1(CC(=O)OC)CC(NC(=O)C(C2CC2)OCC)C1 99355,C1(NC(C(C)Oc2ccc(F)nc2)=O)CCN(C(C2CC(F)(CF)C2)=O)CC1O 99356,C1(C)(C(=O)NCC(C)=CC(=O)NCCn2cncn2)CCC(=O)N1 99357,C1(NC(=O)NCCNS(CC)(=O)=O)CCCC(C(=O)OC)CC1 99358,CCC(CC(=O)N1CCN(C(c2cccc(C)n2)=O)CC1C1CCCC1)C(F)F 99359,Cc1nnc(CNC(c2nnnn2C2CCC2)C2CCC2)n1C1CC1.c1ccccc1 99360,N1(C(C2(OC)CCSC2)=O)C(CNC(c2ccc(F)cc2Cl)=O)CC2COCC12 99361,C(CNC(C1CNC(=O)N1C)=O)(CC(C)C)NC(C(C)SCC)=O 99362,N1(C(N(C)C)=O)CCC(C(=O)NCC2CC2NC(c2cocn2)=O)CC1 99363,C(=O)(C1=NOC(CNC(c2c[nH]c(=N)o2)=O)C1)NCC=CC 99364,C1(F)(C(=O)NC2CCC3(C(C)C)C2C3)CCCN(C(=O)CC(C)n2cccn2)C1 99365,CN1CC2CCCC(C1)N2C(=O)C(CC(C)(C)C)NC(=O)C(C1CCOCC1)O 99366,c1(C(N2CCC(O)C2)C(=O)NCc2ccco2)cn(C2CCOCC2)nn1 99367,C1(NC(C2(C(C)C)COC2)=O)CC2CCCC(C1)N2C(c1cn[nH]c1)=O 99368,O=C(C(O)C(F)F)NCCC1CC(NC(=O)C(c2ccccc2C(F)(F)F)O)C1 99369,N1(C(C)=O)CCC2(CC1)CC2NC(=O)CCNC(=O)OC(C)(C)C.C1CCN1 99370,C1(CNC(CC(CC)O)=O)CC2(CCOCC2)CN1C(=O)CC(F)(F)F 99371,CCC(C)(CO)C(=O)NCC1CC(F)(CNC(c2cnc(S)n2C)=O)C1 99372,C1(CCNC(C2(CN(C)C)CC2)=O)CCN(C(=O)CC2CC3(CC3)C2)CC1 99373,C(=O)(C1=C(F)CN(C(c2cc(F)c[nH]2)=O)CC1)NC1CCCC(C)(C)C1 99374,C(=O)(C(C(F)(F)F)NC(c1cc(-c2cccc(F)c2)no1)=O)OCC 99375,N1(C(C)=O)CCC(C)C(NC(=O)NCC2(NC(=O)OC(C)(C)C)CC(O)C2)C1 99376,C1(COC)CN(C(C2(CCn3cncn3)CC2)=O)CCC1NC(=O)CC1CC1C 99377,N1(C(CSCC=C)=O)CCc2nc(-c3ccc(F)c([N+](=O)[O-])c3)sc2C1 99378,CC1(C)CC(NC(=O)Cc2nc[nH]n2)CN(C(=O)C(F)(F)C(C)(C)O)C1 99379,C1(CN(C(C(C)OCCOC)=O)C)CCC(CNC(C2(C)CCOC2)=O)CC1 99380,c1(-c2ccc(C(N3C(C)CCC3C)=O)nc2)ccc(C2=CCCC2)cc1 99381,c1(CC)ccc(F)cc1NC1CCN(C(=O)Nc2ccc(OC)nc2)C1 99382,c1(OC)ccc(Cl)c(C(=O)NC2CC3CCC2N3C(=O)C(F)(F)C(F)F)c1 99383,N1(C(CCCCCC)=O)CCC(C)N(C(=O)Cn2nc(C)oc2=O)CC1 99384,c1(C(N(C2CCCN(C(C(CC)F)=O)C2)C)=O)ccc(C(F)F)nc1O 99385,C1(C(=O)NC2C(CNC(CCc3c(C)noc3Cl)=O)C2)CC2OC(C)(C)OC2C1 99386,N1(C(C(C)n2cccn2)=O)CC2CN(Cc3c[nH]nc3-c3ccccc3)C2C1 99387,C1(CC)CN(C(c2cnco2)=O)CCC1CNC(=O)CCCN(C)C(C)=O 99388,c1(-c2nnc(SCC(=O)N(c3cccc(C)c3)CC)o2)cccc(F)c1F 99389,C1(NC(Cn2nc(C)c(Cl)c2)=O)CC(=O)N(CC2CCCCC2)C1C 99390,c1(OC)nc(OC)nc(N2CCCC2(C)CNC(c2cc(CC3CC3)on2)=O)n1 99391,N1(C(C2(CC)CCOC2)=O)C2CCC1CN(C(=O)CNC(c1ccoc1C)=O)C2 99392,C1(C(N)=O)CCCN(C(c2cc(CNC(=O)C=C(C3CC3)C3CC3)[nH]n2)=O)C1 99393,C1(C(=O)OCC)CN(C(=O)NC(C2CS(=O)(=O)C2)C)C1(C)C 99394,Cc1csc2ccc(CC(N3CC(NC(C4CC45CCOC5)=O)C3)=O)cc12 99395,c1(-c2ccc(-c3cc(NC(CC(=O)OC)=O)sc3)cc2)c(F)cccc1[N+](=O)[O-] 99396,CC1CCN(C(C2OCCCO2)=O)CC1NC(=O)C(C1CC1)C1CC1 99397,c1(CC(=O)NCC2N(C(C(C)Cc3ccccn3)=O)CC2)ccc2c(c1)CCC2 99398,CCC(CC(C)C)C(=O)N(CCCNC(=O)COCC(C)C)C1CC1 99399,C1(CC)(CNC(C2CCN(C(=O)C(C)C3CCCC3)CC2)=O)CCOCC1 99400,CC(C)CC(C(=O)N(CCCCCC(=O)NC1CCC(F)CC1)C)C(N)=O 99401,N1(C(c2ccc(C(C)=O)[nH]2)=O)CCC(C(N2CCC(C)(N(C)C)C2)=O)(C(C)C)C1 99402,C(=O)(C(N)CC(F)F)NCC(=O)Nc1[nH]nc(-c2nccc(C)c2)n1 99403,C(=O)(CC(C)c1ccccc1)NC(C1CCCN1C(=O)C=CC(F)F)C 99404,O=C(C1=CCN(C(c2cnns2)=O)C1)NCCOCC(F)F 99405,C(=O)(CC(F)(F)C(C)C)N(CCC)CCNC(=O)C(C)CS(C)=O 99406,C12(C(=O)NC3C(C)(C)CN(C(=O)CSS(C)(=O)=O)C3)CCOC1CC(=O)NC2 99407,CC1(C(=O)NC(c2ccc(Br)cn2)(C)C)CCCN(C(c2ccccc2)=O)C1 99408,N1(C(c2cc(CC)no2)=O)CCC2CC12C(N1CCC(CC(=O)OC)C1)=O 99409,c1(C(N2CC(NC(=O)CC3CC4(CCC4)C3)CC(C)C2)=O)cccc([N+](=O)[O-])c1 99410,N1(C(C2CC(C)OCC2)=O)CC2CC(NC(C3(N(C)C)CCC3)=O)CC1C2 99411,Cc1oc(CNC(=O)C(C)N2CCCC2)nc1C(=O)NC1(C)CCCC1O 99412,c1(C(=O)NCCNC(=O)OC)ccoc1CNC(C1C(C)C1C)=O 99413,C=C(C)CC(C)C(=O)NC1(COC)CCN(C(c2nnn(C)c2C)=O)CC1 99414,Cn1cnc2c1CC(NCCCc1nc(O)c3ccccc3n1)CC2 99415,C1(C(N(CC(CC)NC(CC(=C)Br)=O)C)=O)CN(C(C)C)CCO1 99416,C1(C(=O)NCC(CN(C(C(C)CSc2ccccc2)=O)C)(C)C)CCC(C)(C)O1 99417,c1(NCc2cc(OC)ns2)[nH]c(=NC(C)C2CCCO2)nc2c1cnn2C 99418,Cc1ccnn1CC(=O)NC(CNC(c1cccs1)=O)C1CCC1 99419,N1(C(c2c(C)nc(O)[nH]2)=O)CC(C)CCC1CNC(c1cnco1)=O 99420,CCC(C)(C)CCCC(=O)NCC(C)(C)CN(C(=O)C(C)(F)C(F)(F)F)C 99421,C(c1ccc(F)cc1)=CCC(=O)NC1CCN(C(=O)CCF)C(C2CC2)C1 99422,C(=O)(C(C)(O)C(C)C)NCC1CC(COC)CN1C(C1CCCCCC1)=O 99423,C1(CNC(C(C)O)=O)CC2COCC2N1C(=O)C(F)(F)c1cnn(C)c1 99424,C1(NC(CSC(C)C)=O)CCC(C)N(C(c2cc(C3CC3)[nH]n2)=O)C1 99425,CCCCCCn1cc(C2CCN(C(=O)Cc3nocc3C)C2)nn1 99426,C1(CC(=O)NCC(CNC(CCC(=C)Br)=O)OC)CCCCC12CC2 99427,C1(C(=O)NC(C2(C(=O)NC(C3CCOC3)C#C)CC2)C)CCCCCC1 99428,c1(SC)nc(Cl)c(C)c(=NC2CCN(C(=O)CN3CCCNC3=O)C2)[nH]1 99429,Cc1cc(Br)cc2cc(C(N3CCC(NC(C4CN(C)C4)=O)C3)=O)oc12 99430,CC(CCc1ccccc1)CC(=O)NCC(C)CN(C)C(c1cnoc1)=O 99431,c1(OC)cc(C)c(C(=O)NC2CC(NC(=O)CC(C3CC3)C3CC3)C2)cn1 99432,c1(C(=O)NCCN2CCCN(C(=O)CNC=O)CC2)cc(O)ncc1Br 99433,c1(C(=O)NC2CC(C)N(C(=O)CN(C)S(N)(=O)=O)C2)ccc(O)c(Cl)n1 99434,N1(C(C(=O)NCCSC)c2cnsc2)CCC2NC(=O)CCC2C1 99435,N1(C(C(C)n2cccn2)=O)CCc2ccccc2C1CNC(=O)Cc1cnsc1 99436,C1(C(=O)NCC(CCOC)NC(c2c[nH]c(C(F)(F)F)c2)=O)C(C)(C)C1(F)F 99437,c1(C(N(C)CC2(CNC(=O)COC3CCCC3)CC2)=O)c(F)ccc(Cl)c1F 99438,c1(C(C(=O)NCCOC)N(CC(=O)NC2CC2)C2CC2)cc(C(C)(F)F)ccn1 99439,C1(CNC(c2c(CCC)n(C)nc2)=O)CC(N=c2nc(C)nc3[nH][nH]cc2-3)C1 99440,C1(NC(c2ccc(F)cc2)=O)CC2(CCN(c3ncc4c(n3)CCOC4)CC2)C1 99441,N1(C(CCC2C(=O)NC(=O)N2)=O)CC2(CC(NC(c3cc(F)c[nH]3)=O)CO2)C1 99442,Cc1ccc(C)n1CC(=O)N(CCNCCC1(C)OCCO1)Cc1ccccc1 99443,C(=O)(CC(O)CNC1CCC1NC(C)=O)N1C(C(=O)OC)C=CC1 99444,c1(C(=O)NCC(C)N(C(C(c2scc(C)n2)C)=O)C)ccc2n[nH]cc2c1C 99445,C(=O)(C(CC(C)SC)NCCC1CCC(C(=O)OC)C1)Nc1ccccc1NC 99446,C1(CNC(C2C(=C)C2)=O)(CNC(c2nc(Cl)cs2)=O)CC12CCC2 99447,CN=c1cc(C(N2CCOC(C(=O)NC3CCC(C4CC4)C3)C2)=O)cc[nH]1 99448,C1(C(=O)NOC(c2ccccn2)C)(CC#C)CCN(C(=O)CC2CC=CCC2)C1 99449,C(=O)(C1=NOC(C)(C)C1)N(C(CC)CNC(=O)CC1CCCN1C)C 99450,c1(C(N2CC(C(N)=O)(CNC(CCC(C)(F)F)=O)C2)=O)cc(F)cc2cc[nH]c12 99451,C(=O)(C(O)CC(F)(F)F)N1C(C)(CC)CC(NC(c2cccn2C)=O)C1 99452,C1(C(=O)NCCC(C(=O)N(CCOC)CCO)O)CCCC(C#N)C1 99453,Cc1c(C(=O)NC2CC23CCN(C(C2CSCCS2)=O)C3)cncc1Cl 99454,Cc1sc(=O)n(CC(=O)NCC(O)CCNC(C2CC2CN(C)C)=O)c1C 99455,c1(OC)c(C(=O)NCC(CO)NC(c2noc(C3CC3)c2C)=O)nc(O)nc1O 99456,CON(CCC(=O)NC1CCN(C2CC2)C1)C(=O)C1CCOCC1(C)C 99457,CC(C)(C#N)CC(=O)N1CC(CCN)CCC1C1(CN2CCNC(=O)C2)CCC1 99458,C1(NC(C2(SCC)CC2)=O)CC2(C1)CC2NC(=O)Cc1csc(C2CCCC2)n1 99459,C12CN(CC1C)C(=O)COC2.C1(OC(CC(F)(F)F)C)CCCOC1.C1C(=O)N1 99460,C(CC1CC1)(CC(=O)N(c1ccsc1)C)NC(c1ncn(C(C)C)c1)=O 99461,N1(C(C(CN(CC)CC)F)=O)CCC(C)(CCNC(=O)Cc2cn[nH]c2)C1 99462,C1(NC(CC(c2c(C)cccc2)C)=O)COCCN(C(=O)CN2CSCC2=O)C1 99463,C(C)(CC(C)NC(C1(C(C)(F)F)CCC1)=O)NC(CCOCC#C)=O 99464,C1(CCNC(=O)Cc2cscn2)CCCN(C(C23CCCC2CCC3)=O)CC1 99465,C(=O)(C1CCc2c[nH]nc21)NCc1ccc(C(=O)NCC2(C)N=C(C)SC2)o1 99466,N12CCCC(C1)C2=O.N12CC(CC1=O)C(=O)N1CC2C1.CCCCCOCC.OCC 99467,c12ccc(cc1F)[nH]c2=O.c1(C(C(=O)NC)N(C(CC)C)C)ccn(C2CC2)c1 99468,c1(C(=O)NC2C(NC(=O)CC3CCCOC3)CC2)ccc2c(c1)CCCN2 99469,C1(O)(CCNC(c2c(C)ncs2)=O)CCCN(C(C2CCN2C2CCCC2)=O)C1 99470,N1(C(=O)NC(c2ccco2)C)CCN(c2ccc(Cl)cn2)CC1 99471,CCC(C)CCC(=O)N1CC(O)(CCNC(C2CCC(F)CC2)=O)C1 99472,N1(CCNC(=O)NC2CCS(=O)(=O)C2)CCCCc2ccccc21 99473,C1(NC(CCCC)=O)CN(C(=O)C(=O)Nc2ccc(C)c(C)c2)CC2(CCC2)C1 99474,Cc1cc(C(N2CCCC2CCCNC(=O)C(=Cc2cscn2)F)=O)ccn1 99475,Cc1cnc(C(C)NC(C2(NC(c3sccc3CO)=O)CC2)=O)nc1 99476,C(CCC(N)=O)(C(=O)NCCCN(C)CC1CC1)n1cc(COC)nn1 99477,c1(N(CCCOCC)C)ncc(S(=O)(=O)N2CCC(c3ccco3)C2)cc1Cl 99478,N1(C(C(C(C)C)=O)=O)CC2CN(C(=O)Cc3ccc(F)cc3Cl)CC2C1 99479,c1(OC)ccc(C(O)CC(=O)NC(C2CCC(=O)N2)c2nn[nH]n2)cc1OC 99480,CC1(C)CC(C(N2CC3(CC(F)C3)C2)=O)CN1C(c1ccc(CO)cn1)=O 99481,n1(CC(N2CC3C(N(C(CN(CC)CC)=O)C)C3C2)=O)nc(C)ccc1=O 99482,c1(C(=O)NC2CN(C(CC(=C=C)C)=O)C3C2C3)ccc(O)cc1C 99483,C1(NC(=O)CC2CC3CC3C2)CN(C(=O)CC2CCCC2)CC2(CCC2)C1 99484,CC1(CNC(c2ccc(F)s2)=O)CCCN1C(=O)C(F)CC1CCCC1 99485,N1(C(C(=O)NC(C(C)C)C)=O)CCCC(C(=O)CN2CCCC2)C1 99486,C1(NC(c2nc(CCC)oc2)=O)CN(C(=O)CSC2CC2)CCC1C(F)(F)F 99487,c1(C(=O)NC(C(C(C)C)NC(c2c(C)nncc2)=O)C)cc2ccc(F)cc2o1 99488,C(=O)(C(C)(CC)CO)NC(CCCC)CNC(=O)Cc1cnn(C)c1C(F)F 99489,N1(C(CN(C(=O)CC2CCCOCC2)CC)=O)CCC(C)(C#N)C1 99490,c1(C(N(CCC(=O)NC(COC)COC)C)=O)sc(C)cc1C 99491,C1(CNC(C2N(C)CCC2)=O)CN(C(=O)CCC2CC2(F)F)CC(C)(C)O1 99492,Cc1cn(-c2ccc(F)cc2)nc1C(=O)N(CC(C)(C)O)CCO 99493,CC1CN(C(=O)CSc2cccc[n+]2[O-])CC(C)N(C(=O)CCOCCN(C)C)C1 99494,N1(C(CC2(C)CCN(C(c3cnn(C(F)F)c3)=O)C2)=O)CCCC(O)(C2CC2)C1 99495,C1(C2CCCN(C(=O)C(F)(F)C(C)O)C2)(NC(c2ccc(OC)cc2Cl)=O)CC1 99496,c1(C(N2C(CCCNC(CC=C)=O)CCC2)=O)ccc(-c2cn[nH]c2)cc1 99497,Cc1scc(CNC(=O)CC2(C)CCN2C(=O)COCC2CC2)c1C 99498,CC(N=c1nc2sccc2c(NCc2csc(Br)n2)[nH]1)c1cnccn1 99499,CC(CC(=O)N1CCCC(O)(CC(=O)OC(C)(C)C)C1)CC(C)(C)C 99500,c1(SC)cc(=NC(=O)C2CC23CCN(C(=O)Cn2nccc2C)C3)[nH]n1C 99501,Cc1c(C(N2CCC(C(=O)NCC(C)(O)CO)(CO)C2)=O)ncn1C 99502,C1(C(C)(C)C)CCN(C(=O)CCN(C(=O)CC2CCOC2)CCO)C1 99503,c1(CC(=O)N(CCC(C)NC(=O)C(C2CCOCC2)N(C)C)C)c[nH]ccc1=O 99504,C1(NC(C(C)CC2CCC2)=O)COCCN(C(=O)Cc2cnccn2)C1 99505,c1(C(=O)NCC(C(C)C)(C)NC(C2CCC2(C)C)=O)cc2n(c1)CCOC2 99506,Cc1c(NC(C2(C)CCCN(Cc3ccc(I)o3)C2)=O)cccc1Br 99507,C(=O)(CCCC(=O)N1CCN(C(=O)CCOC2CCOCC2)C(C(F)F)C1)OC 99508,Cc1cnc(NC(C)(C)C2CC2)c(S(=O)(=O)N(C)Cc2ccc3c(c2)OCO3)c1 99509,C1(NC(=O)CN2CCCS2(=O)=O)CN(C(c2ccc(C3CC3)o2)=O)CC2(CC2)C1 99510,Cn1c(C(=O)NCC2(C(N3CC(N4CCOC4=O)C3)=O)CCCO2)cnc1Cl 99511,N1(C(C2C(C=C)CC2)=O)CCOCC1CNC(c1nc(Br)sc1C1CC1)=O 99512,C1(NC(C2N(CC)CC2)=O)C=CC(C(=O)N(CCC(O)CO)C)C1 99513,C(CN=c1cc[nH]cc1S(=O)(=O)N1CCC(C(C)C)C1)c1c(C)cccc1 99514,Cc1ccc(F)c(C(N2CC=CC(NC(=O)CC(C)C3CC3)C2)=O)n1 99515,c1(-n2cc(C(C)(C)NC(c3cnco3)=O)nn2)cccc(F)n1 99516,Cc1[nH]nc2ncc(C(N3CC(C4CN(C(c5cc(Cl)ccn5)=O)C4)C3)=O)cc12 99517,N#CC1CCN(CC(=O)NC2CC(n3cc(C4CCCC(O)C4)nn3)C2)CC1 99518,c1(CC)cscc1C(=O)NCCCN(C(c1ccncc1)=O)CC1CCCC1 99519,N1(C(CCCCC)=O)CC2(C1)CN(C(c1ccc(C3CCCO3)nn1)=O)C2 99520,Cc1ccc2[nH]nc(CNC(=O)NCCCN3CCCC(C)C3)c2c1 99521,C(=O)(C(F)C1=CCCCC1)NC(CNC(Cc1c(C)nc(O)nc1O)=O)C(C)C 99522,Cc1cccn2nc(C(=O)NCC(O)CNC(=O)C(C)Cc3ccncc3)cc12 99523,c1(NCC(N2CC(NC=O)C2)=O)cc(C)cc(C)c1.c12cc([nH]n1)C(=O)N2.C(C)OC 99524,C(=O)(C(C)(C)CS(N)(=O)=O)NCC(CC)NC(=O)Cc1cc2ccccc2s1 99525,n1(C(C)C)ncc(C(=O)NCC(C(C)(C)C)NC(C2(Cl)CC2(F)F)=O)c1C1CC1 99526,c1(C(N2CCC(F)(CNC(c3c(CC)c(C)sc3)=O)C2)=O)ccc2c(c1)CCO2 99527,N1(C(CCc2ccc(C)s2)=O)CCC(CNC(C2CCCC(F)(F)C2)=O)CC1C 99528,N1(C(C2(CC)CCCC2O)=O)CC=C(C(=O)NCC2(CC3CC3)CC2)CC1 99529,C1(C(C(=O)CCc2cncn2C)=O)CCC(CN)C1.C(=O)(CC1(CN)CC1)OC 99530,C(=O)(C(C(C)CCC=C(C)C)N1CCC(C(=O)OC)CC1)NCCCOC 99531,c1(NC)cc(C(N2CC(C)(NC(=O)C(CC3CCC3)NC(C)=O)C2)=O)cc(Cl)n1 99532,C#Cc1cc(F)c(C(=O)N(CC(CC)NC(=O)C(C)Cn2ccnc2)C)cc1F 99533,c1(C(N2C(C(CNC(CC(COC)C)=O)(C)C)CCC2)=O)cc2occc2[nH]1 99534,CCS(=O)(=O)CC(=O)NCC1CCCCN1C(C1CCCN(C(N)=O)C1)=O 99535,C1(NC(c2c(CC)[nH]nc2Cl)=O)COCCN(C(=O)COC2COC2)C1 99536,c1(C(=O)NCC2CCN(C(=O)C=CC3CC3)C2)ccnc(Br)c1F 99537,c1(C(=O)NCCCCCNC(c2c(C)oc(Br)c2)=O)ccc2cc[nH]c2c1 99538,Cc1c(CN2CCN(C(N(C)C(c3ccc(Cl)cc3)=O)=O)CC2)cnn1C 99539,c1(C(N(CC(CNC(C2CC(CC(=O)OC)C2)=O)O)C)=O)c[nH]nc1C(F)(F)F 99540,C1(NC(CCOC(C)C)=O)CCCC(NC(=O)CCN2CCCCC2)C1 99541,c1(SC)ccc([N+](=O)[O-])cc1C(=O)N(CC(C)(C)NC(c1ccncc1F)=O)C 99542,C1(C(=O)NC(CNC(CCc2onc(C(C)C)n2)=O)(C)CO)CCN(C)C1C 99543,C1(NC(C=CC2N(C)CCC2)=O)CCCCCC1C(=O)NC1CCCC1N=[N+]=[N-] 99544,c1(CCC)cc(C(=O)NCCC(C)N(C(=O)C(C)Cc2ccncc2)C)n[nH]1 99545,C#CC1(C(N2CCCC(CCNC(C3COCCN3C)=O)C2)=O)CCCC1 99546,CCC1=NOC(C(=O)NC(C(=O)NCc2cc(CC)no2)C2CC2)C1 99547,C1(CC(=O)N(C2CC2C(=O)Nc2cn(CC(=O)O)nn2)CC)C(=O)N(C)N=C1C 99548,Cc1cc(C(N2CC(NC(c3nc(O)c(C)s3)=O)C3CC23)=O)n2nc(C)cc2n1 99549,N#CCC(=O)NNC(=O)Cc1cc(Cl)ccc1Cl 99550,c1(C(N2CC(OC)C2)=O)ccc(Cn2ccnn2)cc1.C12(CC1)C(=O)NCCS2 99551,C1(NC(C(C(=C)Cl)(C)C)=O)CCC2CCN(C(=O)CCNC(=O)OCC)C1C2 99552,C1(C)(CNC(C2C(c3c(C)ccnc3)C2)=O)CCC(NC(c2cc[nH]n2)=O)CC1 99553,c1(C(=O)NC(CC)(C)CNC(=O)C(C)NC(c2cccs2)=O)sc(CO)nc1C 99554,C1(C(=O)NC(C2(OC)CCC2)C)CC12CCN(C(c1cccc(F)c1O)=O)C2 99555,N1(C(C=CSC)=O)CCC(F)(CNC(c2cn(C3CC3)nn2)=O)CC1 99556,Nc1cccc(C(=O)NCCOC2CCN(C(=O)C(O)CN3CC=CC3)CC2)n1 99557,C(=O)(C1Cc2ccccc21)N1CCC(C(N(CC(C)CO)C)=O)CC1(C)C 99558,c1(C(=O)NC(C2CCN(C(C3CCN3C)=O)C2)C)ccc(CO)cc1 99559,c1(C(=O)NC(C)CCCNC(C2COCCO2)=O)cnc2cc(Br)ccc2c1 99560,CC(C)(C)CC(=O)N1CCCC1CNC(C12CC(c3ccccc3)(C1)C2)=O 99561,N1(C(c2ccc(C(=O)OC)cc2)=O)CC(N(C)C(c2conc2C)=O)C2(CC2)C1 99562,N1(C(Cc2cccc(COC)c2)=O)CCN(C(c2nc(O)sc2C)=O)C2CC12 99563,N1(C(CC(C)C2CC2)=O)CCCCC1CCC1CCCN1C(C12CC(F)(C1)C2)=O 99564,c1(COC(=O)NCC(c2cccnc2)N(C)C)cc(F)ccc1N1CCC(O)CC1 99565,Cc1cccc(C2=CCN(C(=O)NCC3C(CN=[N+]=[N-])C3(C)C)CC2)c1 99566,C(CN=c1nc(O)c(Cl)c[nH]1)c1ccc(-c2c(C)cccc2)cc1 99567,N1(C(CC2C=NN(C)C2=O)=O)CCC(C(=O)NCC2CSC2)CC1(C)C 99568,CC1COc2c(C(=O)NC3(CNC(=O)C=CS(C)=O)CC3)cccc21 99569,c1(C(N2CCCN(C(CC(C)C3CCCO3)=O)CC2)=O)ncccc1N=[N+]=[N-] 99570,C(CC(=O)N1CCCC(CNC(=O)CN(C(=O)C(C)C)C)CC1)(C(C)C)OCC 99571,C(=O)(C1=C(Cl)CCOC1)NCC12CN(C(c3c(OC)cccn3)=O)C(C1)CO2 99572,C1(CNC(C=CCC)=O)CCCC(CNC(=O)C(F)(F)c2cscn2)C1 99573,c1(C(N(C(CNC(c2cc(CC)[nH]n2)=O)C)C)=O)cc(OC)c(OC)cc1O 99574,N(C(=NCC(C(C)C)c1ccnn1C)NC(c1ccccc1[N+](=O)[O-])C)C(C)C 99575,c1(C(N2CCN(C(C3C(C)CCCC3)=O)CC2)=O)cc(P(C)(C)=O)ccn1 99576,CCC(CC(F)F)C(=O)N1CCCC1C(=O)NC1(c2ccc(F)cc2)CC1 99577,CS(=O)(=O)CC(F)(F)CCOC(c1nnn(-c2ccccc2)c1C1CC1)=O 99578,N1(C(C2CC(C#C)(O)C2)=O)CCC(C)(C)C1CNC(c1cc(C)nn1CCC)=O 99579,c1(C(N2CCC(NC(C3CCCS3)=O)C2)=O)cc(F)c2cc[nH]c2c1 99580,N1(C(c2cc(C(CC)C)no2)=O)CC(NC(=O)Cc2cnn(C)c2C)CCC1C 99581,c1(COC)nn(C)cc1C(=O)N(CCNC(c1cc[nH]c1C1CC1)=O)C(C)C 99582,N1(CC(=O)NCCCN2CCN(C(C(CC)(C)O)=O)CC2)C(=O)NC(C)(C)C1=O 99583,C(=O)(C1=CC2(CCOC2)C1)N(CC(C)(C)CNC(=O)CCCn1ccnc1)C 99584,CC(C)(CCCCNC(C1CC(C2CC2)=NO1)=O)NC(C1CC2CCC(C1)S2)=O 99585,CC(C)CC(C)C(=O)NCC1CC2CCC1N2C(C1CC=CCC1)=O 99586,S(=O)(=O)(c1ccc(Br)cc1NCC1CCCCCCC1)N1C2CC(=C)CC1CC2 99587,c1(C(=O)NCCC2(CNC(C(CCOC)C)=O)CC2)cc(C)c(F)cc1F 99588,N1(C(C(CCC#C)O)=O)CCCN(C(c2cccc(C)c2N)=O)C(CO)C1 99589,CC(C)(O)C(F)CNC(C1(C2CCCN2C(=O)CC2CCCO2)CC1)=O 99590,CC1CC(CNC(C2CCC(CNC(C3Cc4nccn4C3)=O)O2)=O)CC(C)C1 99591,CC1C(NC(c2cnccc2Cl)=O)C(C)CCN1C(c1cc(N(C)C)ccn1)=O 99592,c1(OCC)ccc2c(c1)C(NC(=O)NCCNc1nc(C)cs1)CCO2 99593,N1(SCC(=O)NCC(C)NC(=O)C(C)Sc2ccccn2)CCCCS1(=O)=O 99594,c1(C(=O)NCC2CCCN2C(c2cnn(C3CCOC3)n2)=O)cnn2c1CCC2 99595,c1(C(=O)NC2(C)CCN(C(C34COCC3C4)=O)CC2)ccc(Cl)c([N+](=O)[O-])c1 99596,C1(NC(c2cc(C)oc2)=O)CCCCN(C(C2CC(OC(C)(C)C)C2)=O)C1 99597,CCC(C)(O)C(=O)N(CCCNC(C1C(C(F)F)C1(C)C)=O)CCO 99598,CC(C)(F)CC(=O)N1CC(C(=O)NCCNC(c2c[nH]nc2C2CCCO2)=O)C1 99599,N1(C(c2c(OC)cc(Cl)c(Cl)c2)=O)CCCC2(CCC2O)C1 99600,c1(-n2c(C(c3n(CC)ccn3)NCCn3cncn3)nnn2)ccc(Cl)cc1F 99601,Cc1ncc(Br)c(N2CCOC(C(=O)NC(c3ccc(F)cc3)CO)C2)n1 99602,c1(CCCC(=O)OCCSC(C)(C)C)ccc(Oc2cc(F)cc(Br)c2)c(F)c1 99603,Cc1csc(Cl)c1C(=O)N(C)CC1COCCN1C(C1CC(C)(C#N)C1)=O 99604,N1(C(C2(C)CN(C(CC(CC)O)=O)C2)=O)CCOC(C)CC1 99605,c1(COC)cncc(C(=O)N(C(C)CN(C(=O)CCc2cccs2)C)C)c1 99606,c1(CC)cc(C(=O)NCC(C)(C2CC2)NC(c2cc(C)[nH]n2)=O)ccc1O 99607,CC1SCCCC1C(N1CCC2CC12C(=O)NCCNC(=O)CO)=O 99608,Cc1cn2ccc(C(N3CCC(Cc4cn(CCO)nn4)C3)=O)cc2n1 99609,N1(C(C2C(C)(C)C2)=O)CCN(C(c2ccnc(C3CC3)c2)=O)C(c2cccs2)C1 99610,Cc1nc(Cl)ncc1NC(C1CCCN(C(C2CC(C)(C)C2)=O)CC1)=O 99611,N1(C(C(C)S(N)(=O)=O)=O)CC(NC(=O)C(F)(F)C2CC2)CC12CCCCCC2 99612,C(c1ccccn1)=C(C)C(=O)NC1CCC(C)(CNC(c2ccncc2)=O)C1 99613,c1(C(=O)NC(C)C(=O)NC(C)CC2(O)CCC2)sccc1CC(C)(C)C 99614,CC1CCN(C(c2ncsc2C2CC2)=O)CC1NC(=O)CSc1cn[nH]c1 99615,C(=O)(C(C(=O)NCCNC(=O)C(C1(O)CCCCC1)OC)OC)OCC 99616,C=C(C)CC(C(=O)NCC1(C)COCCO1)NC(=O)CC1CCCN1C 99617,N1(C(C)=O)CC(C(=O)NC2CC2C(=O)NCCN(C)C2CC2)(CO)C1 99618,C1(CCNC(c2cnn(C)c2Cl)=O)CCN(C(=O)Cc2cc[nH]c2)CCC1(F)F 99619,c1(C(N(CC)CC2CCN(C(=O)CC3C=CCC3)CC2)=O)cnc(O)cc1C 99620,C1(NC(C=CCN(C(=O)CCOC2CCCC2)C)=O)CCC(F)(F)C1 99621,C1(CNC(C(COC)OC)=O)CCCC2(CN(C(=O)C(CC(C)C)OC)C2)O1 99622,S(=O)(=O)(c1c[nH]ccc1=NC(Cc1cccs1)CO)NCCC(CC)C 99623,C(=O)(C1c2c[nH]nc2CN1C(C1CCC1C)=O)N1CCCC(C)(OC)C1 99624,N1(C(C(C)n2cccn2)=O)CC2CCC(C1)N(C(=O)CCc1cc(F)ccn1)C2 99625,N1(C(C(C)CF)=O)Cc2ccccc2CC1CNC(=O)C(c1ccccn1)O 99626,N1(C(C(CCOC)NC(=O)C=Cc2ccsc2)=O)CCC2(CCC(O)C2)C1 99627,c1(CNC(=O)C(=O)NC(C2C(C(=O)OCC)C2)C)cc(C2CCC2)[nH]n1 99628,C1(C(=O)NCC2(F)CC(NC(c3cnc(Cl)s3)=O)C2)CC2C=CCC(C1)C2 99629,O=C1NC(=O)C2CN(C(=NCCCCl)NCc3ccc4occc4c3)CC12 99630,C1(NC(c2cccnc2N2CCCCC2)C)CCN(C(=O)C(C)(C)CO)CC1C 99631,CCC1=NOC(C(=O)N(C2(C(=O)NC3CCNC(=O)C3)CCC2)C2CC2)C1 99632,C(CC(C(C)(C)C)NC(C1CC1OC(C)(C)C)=O)N(C(C=C(C)C(F)F)=O)C 99633,N1(C(C2(CC#C)CCCOC2)=O)C2CCC1CC(NC(=O)COC)C2 99634,C(=O)(CC(COC)NC(C12CCC(CC1)C2)=O)NC(c1cccnc1)CC 99635,C1(OCCSC)CCN(C(C2(CC(=O)Nc3cncnc3)CC2)=O)CC1 99636,C(=O)(CCC(C(C)O)NCc1ccc(N(C)C)cc1F)OC 99637,C12(CCNC(C(C)=C(CC)C)=O)CCC(C1)N(C(=O)C(C(C)C)NC(N)=O)C2 99638,CC1CN(C(C2CC(C)(F)C2)=O)CCCN1C(c1cnc(C(F)(F)F)nc1)=O 99639,Cc1ccc(S(=O)(=O)NCc2ccco2)cc1C(=O)Nc1cccc2nncn12 99640,N1(C(CCSC)=O)CCC(CNC(=O)C(C(C)C)n2ccc(C3CC3)n2)C12CC2 99641,C(=O)(CCCC(C)(C)C)N1CC(CC)N(C(=O)C(C)N(C)C)CC1 99642,C1(CCCNC(C)=O)CCCN1C(c1cccn1Cc1cccs1)=O 99643,c1(C(=O)NC(CC)CNC(c2nc(=N)cc[nH]2)=O)ccc(NC)c(F)c1 99644,Cc1nc(Cl)nc(N2CC=C(CNC(c3c(Cl)cncc3Cl)=O)CC2)c1[N+](=O)[O-] 99645,Cc1c(C(=O)NCC2CC2NC(=O)Cn2cnc(=N)[nH]2)[nH]c2c1CCCC2 99646,c1(C(N2CC(CC(C)NC(CN3CC(C)C3)=O)C2)=O)nc(C(C)C)ncc1Br 99647,C(C)(C(C)C(=O)NC1CCC(C(C)O)CC1)NC(c1c(C)snn1)=O 99648,c1(C(=O)NCC2C(NC(=O)CC(F)F)CCC2)ccc(-c2nc(=O)o[nH]2)cc1 99649,c1(C(=O)O)c(NC(=O)C=Cc2c(Cl)nc3sccn23)c(C#N)c2n1CCCC2 99650,CC(C)C(C)(Cc1ccccc1)C(=O)NCCc1ccccc1O 99651,c1(CC)cnc(C(=O)NC(c2cccc(C)c2)CNC(=O)C(=O)C(C)C)nc1 99652,n1(CC)nc(C(=O)NC2CCC(NC(=O)C(C)CC(F)F)C2)c2c1CCOC2 99653,Cc1cc(Cc2nc(-c3cncnc3)nn2C(C)C(F)(F)F)ccc1Br